Cc1ccc(C(=O)NCC(F)(F)F)cc1NC(=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147000059 HJ On-Demand Anodyne MAPK11 26 42 Cc1ccc(C(=O)NCC(F)(F)F)cc1NC(=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147000059 HJ On-Demand Anodyne MAPK14 20 42 CCCCOc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c(C)c1 ZINC000147000095 EF On-Demand Anodyne PLA2G4B 54 33 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(Cl)c(F)c1 ZINC000147000154 DG On-Demand Anodyne ENV 48 41 O=C(Nc1ccccc1C(F)(F)F)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147000170 EE On-Demand Anodyne RBP4 53 40 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne OPRM1 18 44 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne OPRD1 24 44 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne KLK3 61 38 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne HLA-A 82 51 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne GRIA1 48 40 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne FURIN 67 47 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne ST14 15 40 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne SIRT1 27 43 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne POLG_WNV 68 32 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne F2RL1 48 36 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne DLG4 57 33 C[C@H](O)[C@H](NC(=O)[C@@H](CC(N)=O)NC(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147000187 HA For-Sale Anodyne NOD1 64 38 CCCCOc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c(C)c1 ZINC000147000250 EF On-Demand Anodyne PLA2G4B 54 33 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(NC(C)=O)c(OC)c1)C2 ZINC000147000279 FF On-Demand Anodyne MTNR1A 24 43 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(NC(C)=O)c(OC)c1)C2 ZINC000147000279 FF On-Demand Anodyne ROCK2 42 58 O=C(Nc1ccccc1C(F)(F)F)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147000305 EE On-Demand Anodyne RBP4 53 40 O=C1c2ccccc2C(=O)c2c(Br)ccc(Br)c21 ZINC000147000334 FH For-Sale Anodyne CDC25B 19 55 Cc1ccc(-n2nnc(CC(=O)NCc3cccc(CN4CCCC4)c3)c2C)cc1 ZINC000147000386 HG On-Demand Anodyne HRH2 31 41 Cc1ccc(-n2nnc(CC(=O)NCc3cccc(CN4CCCC4)c3)c2C)cc1 ZINC000147000386 HG On-Demand Anodyne CHRM3 15 41 Cc1ccc(-n2nnc(CC(=O)NCc3cccc(CN4CCCC4)c3)c2C)cc1 ZINC000147000386 HG On-Demand Anodyne NPFFR1 43 35 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(OCc2cccc(F)c2)c1 ZINC000147000396 GG On-Demand Anodyne F10 16 46 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147000445 GD On-Demand Anodyne PIK3CA 24 41 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147000445 GD On-Demand Anodyne MTOR 39 41 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147000445 GD On-Demand Anodyne EPHX2 34 53 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147000445 GD On-Demand Anodyne PIK3CG 21 41 O=C(Nc1cccc(C(F)(F)F)c1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147000476 EE On-Demand Anodyne CCR2 22 41 O=C(Nc1cccc(C(F)(F)F)c1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147000476 EE On-Demand Anodyne EPHX2 18 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc2c(c1)NC(=O)[C@H](C)O2 ZINC000147000506 ED On-Demand Anodyne HDAC10 43 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc2c(c1)NC(=O)[C@H](C)O2 ZINC000147000506 ED On-Demand Anodyne HDAC11 43 35 CCCc1nc(C)c2c(C)nc3sc(C)nc3n12 ZINC000147000570 CG For-Sale Anodyne PDE10A 15 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(OCc2cccc(F)c2)c1 ZINC000147000592 GG On-Demand Anodyne F10 16 46 O=C(C[C@@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147000643 GD On-Demand Anodyne PIK3CA 24 41 O=C(C[C@@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147000643 GD On-Demand Anodyne MTOR 39 41 O=C(C[C@@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147000643 GD On-Demand Anodyne EPHX2 34 53 O=C(C[C@@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147000643 GD On-Demand Anodyne PIK3CG 21 41 O=C(Nc1cccc(C(F)(F)F)c1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147000668 EE On-Demand Anodyne DHODH 15 47 O=C(Nc1cccc(C(F)(F)F)c1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147000668 EE On-Demand Anodyne CCR2 22 41 O=C(Nc1cccc(C(F)(F)F)c1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147000668 EE On-Demand Anodyne EPHX2 18 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc2c(c1)NC(=O)[C@H](C)O2 ZINC000147000677 ED On-Demand Anodyne HDAC10 43 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc2c(c1)NC(=O)[C@H](C)O2 ZINC000147000677 ED On-Demand Anodyne HDAC11 43 35 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(COc3cccc(F)c3)c2)c1 ZINC000147000686 GJ On-Demand Bother MAOB 28 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(COc3cccc(F)c3)c2)c1 ZINC000147000686 GJ On-Demand Bother TAAR1 39 52 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(COc3cccc(F)c3)c2)c1 ZINC000147000686 GJ On-Demand Bother KCNK3 54 36 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(COc3cccc(F)c3)c2)c1 ZINC000147000686 GJ On-Demand Bother KCNK9 46 36 N#CCc1nc(-c2ccccc2)c(-c2ccccc2)[nH]1 ZINC000147000773 CH For-Sale Mild SOAT1 32 56 CCCc1nc(C)c2c(C)nc3sc(Br)nc3n12 ZINC000147000802 EH For-Sale Anodyne PDE10A 24 51 COC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147000825 FD On-Demand Anodyne PRSS1 18 42 COC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147000825 FD On-Demand Anodyne ADORA2B 39 41 COC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147000825 FD On-Demand Anodyne MTNR1A 18 41 COC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147000825 FD On-Demand Anodyne MTNR1B 18 43 COC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147000825 FD On-Demand Anodyne PLA2G4B 45 36 COC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147000825 FD On-Demand Anodyne ACR 57 38 COC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147000825 FD On-Demand Anodyne HIF1A 24 48 COC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147000825 FD On-Demand Anodyne TAAR1 33 40 COC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147000825 FD On-Demand Anodyne KCNK3 43 37 COC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147000825 FD On-Demand Anodyne KCNK9 40 34 O=C(Nc1cccc(C(F)(F)F)c1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147000862 EE On-Demand Anodyne DHODH 15 47 O=C(Nc1cccc(C(F)(F)F)c1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147000862 EE On-Demand Anodyne CCR2 22 41 O=C(Nc1cccc(C(F)(F)F)c1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147000862 EE On-Demand Anodyne EPHX2 18 41 CCCCCCCCn1nnc2c(C(=O)O)cccc21 ZINC000147000878 CG For-Sale Mild PLA2G4B 70 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc2c(c1)NC(=O)[C@@H](C)O2 ZINC000147000885 ED On-Demand Anodyne HDAC10 43 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc2c(c1)NC(=O)[C@@H](C)O2 ZINC000147000885 ED On-Demand Anodyne HDAC11 43 35 O=C(Nc1cccc(C(F)(F)F)c1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147001048 EE On-Demand Anodyne CCR2 22 41 O=C(Nc1cccc(C(F)(F)F)c1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147001048 EE On-Demand Anodyne EPHX2 18 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(C(=O)NC3CC3)c1)C2 ZINC000147001073 GE On-Demand Anodyne DRD4 44 35 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(C(=O)NC3CC3)c1)C2 ZINC000147001073 GE On-Demand Anodyne MTNR1A 48 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(C(=O)NC3CC3)c1)C2 ZINC000147001073 GE On-Demand Anodyne ROCK2 43 38 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(C(=O)NC3CC3)c1)C2 ZINC000147001073 GE On-Demand Anodyne MCHR1 19 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc2c(c1)NC(=O)[C@@H](C)O2 ZINC000147001084 ED On-Demand Anodyne HDAC10 43 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc2c(c1)NC(=O)[C@@H](C)O2 ZINC000147001084 ED On-Demand Anodyne HDAC11 43 35 CCN(Cc1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1)C(C)=O ZINC000147001155 FG On-Demand Bother ROCK2 18 41 CCN(Cc1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1)C(C)=O ZINC000147001155 FG On-Demand Bother TAAR1 28 47 CCN(Cc1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1)C(C)=O ZINC000147001155 FG On-Demand Bother AKR1C2 26 40 CCN(Cc1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1)C(C)=O ZINC000147001155 FG On-Demand Bother KCNK3 48 36 O=C(Nc1cccc2cnccc12)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147001246 ED On-Demand Anodyne TRPV1 21 42 O=C(Nc1cccc2cnccc12)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147001246 ED On-Demand Anodyne CDK5 28 47 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne TSHR 41 33 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne PPIA 31 43 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne PDGFRB 44 38 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne ADORA2B 38 40 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne SYK 19 42 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne FLT1 22 45 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne ACR 44 34 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne PDGFRA 48 35 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne HIF1A 25 41 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne ENPP1 81 39 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne DRTS_TRYCR 51 44 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1OCc1ccncc1 ZINC000147001263 HF On-Demand Anodyne KLK_PIG 41 32 CC(C)=CCC/C(C)=C/CC/C(C)=C/CSCCO ZINC000147001362 CK Annotated Anodyne GGPS1 43 45 CC(C)=CCC/C(C)=C/CC/C(C)=C/CSCCO ZINC000147001362 CK Annotated Anodyne FDFT1 35 45 CC(C)=CCC/C(C)=C/CC/C(C)=C/CSCCO ZINC000147001362 CK Annotated Anodyne LSS 17 41 CC(C)=CCC/C(C)=C/CC/C(C)=C/CSCCO ZINC000147001362 CK Annotated Anodyne STE14 0 60 CCOC(=O)COc1ccc(/C=C(\C#N)C(=O)OCC)cc1OC ZINC000147001396 EE In-Stock Reactive EGFR 21 43 CCOC(=O)COc1ccc(/C=C(\C#N)C(=O)OCC)cc1OC ZINC000147001396 EE In-Stock Reactive ESRRA 19 41 CCOC(=O)COc1ccc(/C=C(\C#N)C(=O)OCC)cc1OC ZINC000147001396 EE In-Stock Reactive TUBB1 42 34 O=C(Nc1cccc2cnccc12)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147001473 ED On-Demand Anodyne TRPV1 21 42 O=C(Nc1cccc2cnccc12)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147001473 ED On-Demand Anodyne CDK5 28 47 CCCOc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147001532 GG On-Demand Bother TAAR1 40 45 CCCOc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147001532 GG On-Demand Bother KCNK3 71 35 CCCOc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147001532 GG On-Demand Bother KCNK9 48 35 c1ccc(-c2cc(-c3ccc(-n4c5ccccc5c5ccccc54)cc3)cc(-c3ccccn3)n2)nc1 ZINC000147001545 JK For-Sale Anodyne METAP1 45 42 Cc1ccc(S(=O)(=O)n2nc(C)c3c(Cl)c(C)ccc32)cc1 ZINC000147001559 EH In-Stock Anodyne ALDH3A1 35 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(OCc2ccccc2Cl)cc1 ZINC000147001579 HH On-Demand Anodyne ADAMTS4 17 41 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCc3cc(C)ccc32)cc1 ZINC000147001608 GG On-Demand Anodyne KCNA5 36 43 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCc3cc(C)ccc32)cc1 ZINC000147001608 GG On-Demand Anodyne LIMK2 23 40 O=C(Nc1cccc2cnccc12)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147001663 ED On-Demand Anodyne TRPV1 21 42 O=C(Nc1cccc2cnccc12)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147001663 ED On-Demand Anodyne CDK5 28 47 Cc1n[nH]c(C)c1-c1ccccn1 ZINC000147001691 AE On-Demand Anodyne METAP1 17 50 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)[C@H](C)n3cccn3)c2)c1 ZINC000147001719 HG On-Demand Bother TAAR1 34 51 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)[C@H](C)n3cccn3)c2)c1 ZINC000147001719 HG On-Demand Bother KCNK3 53 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)[C@H](C)n3cccn3)c2)c1 ZINC000147001719 HG On-Demand Bother KCNK9 42 38 CCCNC1=N[C@H]2[C@H](O[C@H]([C@@H](O)CC)[C@@H](O)[C@@H]2O)S1 ZINC000147001742 CB Annotated Anodyne MGEA5 28 50 COc1ccc(S)c(C(C)=O)c1 ZINC000147001773 AE For-Sale Anodyne MTR1B_CHICK 61 36 COc1ccc(S)c(C(C)=O)c1 ZINC000147001773 AE For-Sale Anodyne MTNR1A 55 39 COc1ccc(S)c(C(C)=O)c1 ZINC000147001773 AE For-Sale Anodyne MTNR1B 47 39 COc1ccc(S)c(C(C)=O)c1 ZINC000147001773 AE For-Sale Anodyne AKR1C3 30 44 COc1ccc(S)c(C(C)=O)c1 ZINC000147001773 AE For-Sale Anodyne AKR1C2 60 44 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(OCc2ccccc2Cl)cc1 ZINC000147001775 HH On-Demand Anodyne ADAMTS4 17 41 O=C1[C@H](C2=CCCC2)CN1Cc1ccccc1 ZINC000147001795 BF For-Sale Anodyne SAP2 33 40 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCc3cc(C)ccc32)cc1 ZINC000147001805 GG On-Demand Anodyne KCNA5 36 43 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCc3cc(C)ccc32)cc1 ZINC000147001805 GG On-Demand Anodyne LIMK2 23 40 CC[C@H](CNC(=O)c1cccn(Cc2ccccc2)c1=O)N1CCc2ccccc2C1 ZINC000147001817 HG On-Demand Anodyne NOD2 41 36 O=C(Nc1cccc2cnccc12)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147001872 ED On-Demand Anodyne TRPV1 21 42 O=C(Nc1cccc2cnccc12)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147001872 ED On-Demand Anodyne CDK5 28 47 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)[C@@H](C)n3cccn3)c2)c1 ZINC000147001896 HG On-Demand Bother TAAR1 34 51 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)[C@@H](C)n3cccn3)c2)c1 ZINC000147001896 HG On-Demand Bother KCNK3 53 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)[C@@H](C)n3cccn3)c2)c1 ZINC000147001896 HG On-Demand Bother KCNK9 42 38 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1CN1CCOCC1 ZINC000147001958 FD On-Demand Anodyne CASR 40 36 CN1CCC(C)(C(=O)Nc2ccc3[nH]nc(-c4nc5ccccc5[nH]4)c3c2)CC1 ZINC000147001989 GH Annotated Anodyne FGFR1 44 47 CN1CCC(C)(C(=O)Nc2ccc3[nH]nc(-c4nc5ccccc5[nH]4)c3c2)CC1 ZINC000147001989 GH Annotated Anodyne ITK 41 46 CN1CCC(C)(C(=O)Nc2ccc3[nH]nc(-c4nc5ccccc5[nH]4)c3c2)CC1 ZINC000147001989 GH Annotated Anodyne FLT1 25 47 CN1CCC(C)(C(=O)Nc2ccc3[nH]nc(-c4nc5ccccc5[nH]4)c3c2)CC1 ZINC000147001989 GH Annotated Anodyne KDR 0 47 CN1CCC(C)(C(=O)Nc2ccc3[nH]nc(-c4nc5ccccc5[nH]4)c3c2)CC1 ZINC000147001989 GH Annotated Anodyne CDK2 0 47 CN1CCC(C)(C(=O)Nc2ccc3[nH]nc(-c4nc5ccccc5[nH]4)c3c2)CC1 ZINC000147001989 GH Annotated Anodyne CDK1 0 42 CN1CCC(C)(C(=O)Nc2ccc3[nH]nc(-c4nc5ccccc5[nH]4)c3c2)CC1 ZINC000147001989 GH Annotated Anodyne TTK 39 41 CN1CCC(C)(C(=O)Nc2ccc3[nH]nc(-c4nc5ccccc5[nH]4)c3c2)CC1 ZINC000147001989 GH Annotated Anodyne PAK4 17 47 CN1CCC(C)(C(=O)Nc2ccc3[nH]nc(-c4nc5ccccc5[nH]4)c3c2)CC1 ZINC000147001989 GH Annotated Anodyne NR2E3 64 37 O=C1[C@@H](C2=CCCC2)CN1Cc1ccccc1 ZINC000147002004 BF For-Sale Anodyne SAP2 33 40 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147002076 EE On-Demand Anodyne CPT1A 54 34 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147002076 EE On-Demand Anodyne CPT2 44 34 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147002076 EE On-Demand Anodyne RBP4 30 43 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccccc1CN1CCOCC1 ZINC000147002158 FD On-Demand Anodyne CASR 40 36 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147002268 EE On-Demand Anodyne CPT1A 54 34 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147002268 EE On-Demand Anodyne CPT2 44 34 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147002268 EE On-Demand Anodyne RBP4 30 43 Fc1cc(F)c(F)c(-c2ccccn2)c1 ZINC000147002363 BG For-Sale Anodyne GRM5 15 43 CC(C)CNC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147002378 GE On-Demand Anodyne F3 48 31 CC(C)CNC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147002378 GE On-Demand Anodyne SLC6A9 15 40 COc1ccc(S(=O)(=O)Nc2ccc(Cl)cc2C(=O)c2nccn2C)cc1 ZINC000147002425 HG Annotated Anodyne PIK3CA 21 40 COc1ccc(S(=O)(=O)Nc2ccc(Cl)cc2C(=O)c2nccn2C)cc1 ZINC000147002425 HG Annotated Anodyne PRTN3 53 34 COc1ccc(S(=O)(=O)Nc2ccc(Cl)cc2C(=O)c2nccn2C)cc1 ZINC000147002425 HG Annotated Anodyne FFAR4 21 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002431 FF On-Demand Anodyne F2R 56 38 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002431 FF On-Demand Anodyne GRIA1 43 31 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002431 FF On-Demand Anodyne PCSK5 56 35 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002431 FF On-Demand Anodyne FURIN 60 36 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002431 FF On-Demand Anodyne DPP7 40 35 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002431 FF On-Demand Anodyne POLG_WNV 65 31 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002431 FF On-Demand Anodyne NPFFR1 42 35 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147002463 EE On-Demand Anodyne CPT1A 54 34 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147002463 EE On-Demand Anodyne CPT2 44 34 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147002463 EE On-Demand Anodyne RBP4 30 43 CC(C)CNC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147002552 GE On-Demand Anodyne F3 48 31 CC(C)CNC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147002552 GE On-Demand Anodyne SLC6A9 15 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002611 FF On-Demand Anodyne F2R 56 38 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002611 FF On-Demand Anodyne GRIA1 43 31 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002611 FF On-Demand Anodyne PCSK5 56 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002611 FF On-Demand Anodyne FURIN 60 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002611 FF On-Demand Anodyne DPP7 40 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002611 FF On-Demand Anodyne POLG_WNV 65 31 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1CN1CCCCC1 ZINC000147002611 FF On-Demand Anodyne NPFFR1 42 35 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(Cl)cc2C(=O)c2cccc[n+]2[O-])cc1 ZINC000147002624 II Annotated Clean PRTN3 58 37 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(Cl)cc2C(=O)c2cccc[n+]2[O-])cc1 ZINC000147002624 II Annotated Clean CYNT 21 45 NCCc1cccc([N+](=O)[O-])c1Cl ZINC000147002636 BD For-Sale Anodyne COLA 44 35 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147002655 EE On-Demand Anodyne CPT1A 54 34 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147002655 EE On-Demand Anodyne CPT2 44 34 COc1ccc(Cl)cc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147002655 EE On-Demand Anodyne RBP4 30 43 C[C@@H](NS(=O)(=O)c1ccccc1C(F)(F)F)C(=O)N1CCC(C#N)CC1 ZINC000147002704 GE On-Demand Mild ST14 52 34 C[C@@H](NS(=O)(=O)c1ccccc1C(F)(F)F)C(=O)N1CCC(C#N)CC1 ZINC000147002704 GE On-Demand Mild RBP4 67 37 C[C@@H](NS(=O)(=O)c1ccccc1C(F)(F)F)C(=O)N1CCC(C#N)CC1 ZINC000147002704 GE On-Demand Mild SFRP1 128 38 C[C@@H](NS(=O)(=O)c1ccccc1C(F)(F)F)C(=O)N1CCC(C#N)CC1 ZINC000147002704 GE On-Demand Mild WNT3 88 38 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C1CC1 ZINC000147002762 BF On-Demand Anodyne MME 48 37 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C1CC1 ZINC000147002762 BF On-Demand Anodyne CTSS 24 43 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C1CC1 ZINC000147002762 BF On-Demand Anodyne PIN1 41 41 CC(C)(C)OC(=O)N1CCC(C(=O)Nc2ccc3[nH]ccc3c2)CC1 ZINC000147002911 EH On-Demand Anodyne HDAC8 15 41 CC(C)(C)OC(=O)N1CCC(C(=O)Nc2ccc3[nH]ccc3c2)CC1 ZINC000147002911 EH On-Demand Anodyne EPHX2 21 44 CC(C)(C)OC(=O)N1CCC(C(=O)Nc2ccc3[nH]ccc3c2)CC1 ZINC000147002911 EH On-Demand Anodyne GPR119 40 42 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C1CC1 ZINC000147002954 BF On-Demand Anodyne MME 48 37 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C1CC1 ZINC000147002954 BF On-Demand Anodyne CTSS 24 43 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C1CC1 ZINC000147002954 BF On-Demand Anodyne PIN1 41 41 CN1[C@H]2CC[C@H]1CC(NC(=O)c1cc3ncccn3n1)C2 ZINC000147003014 CD On-Demand Anodyne HTR3A 35 43 CN1[C@H]2CC[C@H]1CC(NC(=O)c1cc3ncccn3n1)C2 ZINC000147003014 CD On-Demand Anodyne HTR4 26 40 CN1[C@H]2CC[C@H]1CC(NC(=O)c1cc3ncccn3n1)C2 ZINC000147003014 CD On-Demand Anodyne GLRA1 43 34 COc1cc(C(=O)c2cc(Cl)ccc2NS(=O)(=O)c2ccc(C(C)(C)C)cc2)ccn1 ZINC000147003022 JK Annotated Clean PRTN3 46 33 CN1CCN(c2ccc(Nc3nc4cccc(-c5cccc(NS(C)(=O)=O)c5)n4n3)cc2)CC1 ZINC000147003112 JG Annotated Anodyne LCK 22 40 CN1CCN(c2ccc(Nc3nc4cccc(-c5cccc(NS(C)(=O)=O)c5)n4n3)cc2)CC1 ZINC000147003112 JG Annotated Anodyne JAK3 24 46 CN1CCN(c2ccc(Nc3nc4cccc(-c5cccc(NS(C)(=O)=O)c5)n4n3)cc2)CC1 ZINC000147003112 JG Annotated Anodyne JAK1 15 48 CN1CCN(c2ccc(Nc3nc4cccc(-c5cccc(NS(C)(=O)=O)c5)n4n3)cc2)CC1 ZINC000147003112 JG Annotated Anodyne JAK2 58 79 CN1CCN(c2ccc(Nc3nc4cccc(-c5cccc(NS(C)(=O)=O)c5)n4n3)cc2)CC1 ZINC000147003112 JG Annotated Anodyne AURKA 15 45 CN1CCN(c2ccc(Nc3nc4cccc(-c5cccc(NS(C)(=O)=O)c5)n4n3)cc2)CC1 ZINC000147003112 JG Annotated Anodyne STAT6 48 38 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(C)C)cc2C(C)C)c1 ZINC000147003135 FK On-Demand Bother TAAR1 20 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(C)C)cc2C(C)C)c1 ZINC000147003135 FK On-Demand Bother AKR1C3 16 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(C)C)cc2C(C)C)c1 ZINC000147003135 FK On-Demand Bother AKR1C2 42 43 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C1CC1 ZINC000147003139 BF On-Demand Anodyne MME 48 37 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C1CC1 ZINC000147003139 BF On-Demand Anodyne CTSS 24 43 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C1CC1 ZINC000147003139 BF On-Demand Anodyne PIN1 41 41 O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(CO)o2)CC1 ZINC000147003334 EE On-Demand Anodyne DRD4 22 43 O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(CO)o2)CC1 ZINC000147003334 EE On-Demand Anodyne OPRM1 0 59 O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(CO)o2)CC1 ZINC000147003334 EE On-Demand Anodyne OPRL1 22 66 O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(CO)o2)CC1 ZINC000147003334 EE On-Demand Anodyne AKT2 33 51 O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(CO)o2)CC1 ZINC000147003334 EE On-Demand Anodyne PLD1 116 54 O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(CO)o2)CC1 ZINC000147003334 EE On-Demand Anodyne CTSS 0 42 O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(CO)o2)CC1 ZINC000147003334 EE On-Demand Anodyne PLD2 98 55 O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(CO)o2)CC1 ZINC000147003334 EE On-Demand Anodyne AKT1 17 53 O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(CO)o2)CC1 ZINC000147003334 EE On-Demand Anodyne GRIN3A 0 41 O=c1[nH]c2ccccc2n1C1CCN(Cc2ccc(CO)o2)CC1 ZINC000147003334 EE On-Demand Anodyne CALCRL 54 44 O=C(c1cccnc1)c1cc(Cl)ccc1NS(=O)(=O)c1ccc(-c2cocn2)cc1 ZINC000147003460 II Annotated Clean PIK3CA 23 42 O=C(c1cccnc1)c1cc(Cl)ccc1NS(=O)(=O)c1ccc(-c2cocn2)cc1 ZINC000147003460 II Annotated Clean PIK3C3 51 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1nc(C)c(SCC#N)s1)C2 ZINC000147003471 GG On-Demand Mild ROCK2 34 44 N#CC1CCN(C(=O)Cc2csc(NC(=O)c3ccccc3)n2)CC1 ZINC000147003518 FF On-Demand Mild COLA 24 40 N#CC1CCN(C(=O)Cc2csc(NC(=O)c3ccccc3)n2)CC1 ZINC000147003518 FF On-Demand Mild CPT1A 35 40 N#CC1CCN(C(=O)Cc2csc(NC(=O)c3ccccc3)n2)CC1 ZINC000147003518 FF On-Demand Mild CPT1B 40 40 N#CC1CCN(C(=O)Cc2csc(NC(=O)c3ccccc3)n2)CC1 ZINC000147003518 FF On-Demand Mild GCK 15 40 CN(Cc1ccc(F)cc1Cl)C(=O)c1ccccc1 ZINC000147003570 CH On-Demand Anodyne P2RX7 68 43 CN(Cc1ccc(F)cc1Cl)C(=O)c1ccccc1 ZINC000147003570 CH On-Demand Anodyne LIMK2 38 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(C)(C)C)nn2-c2ccc(F)cc2)c1 ZINC000147003596 HI On-Demand Bother TNF 40 34 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(C)(C)C)nn2-c2ccc(F)cc2)c1 ZINC000147003596 HI On-Demand Bother PTK2B 35 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(C)(C)C)nn2-c2ccc(F)cc2)c1 ZINC000147003596 HI On-Demand Bother DDR2 31 41 COc1cc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@@H]32)cc(OC)c1OC ZINC000147003598 FD On-Demand Anodyne FKBP1A 18 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1nc(C)c(SCC#N)s1)C2 ZINC000147003664 GG On-Demand Mild ROCK2 34 44 N#CC1CCN(C(=O)c2ccc(Nc3ccccc3)c([N+](=O)[O-])c2)CC1 ZINC000147003712 FH On-Demand Mild TAAR1 16 46 N#CC1CCN(C(=O)c2ccc(Nc3ccccc3)c([N+](=O)[O-])c2)CC1 ZINC000147003712 FH On-Demand Mild AKR1C3 17 45 N#CC1CCN(C(=O)c2ccc(Nc3ccccc3)c([N+](=O)[O-])c2)CC1 ZINC000147003712 FH On-Demand Mild L3MBTL3 59 48 CCCCC1(CCCC)CN(c2ccccc2)c2cc(SC)c(OCC(=O)O)cc2S(=O)(=O)C1 ZINC000147003756 KK For-Sale Anodyne SLC10A2 93 43 COc1cc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@@H]32)cc(OC)c1OC ZINC000147003772 FD On-Demand Anodyne FKBP1A 18 41 CCOC(=O)c1sc(Cc2ccccc2)nc1O ZINC000147003845 CF In-Stock Anodyne ALOX5 16 45 CCOC(=O)c1sc(Cc2ccccc2)nc1O ZINC000147003845 CF In-Stock Anodyne DHODH 26 45 CCC(=O)Nc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147003854 EI On-Demand Anodyne MDM2 94 37 CCC(=O)Nc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147003854 EI On-Demand Anodyne NAMPT 25 43 CCC(=O)Nc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147003854 EI On-Demand Anodyne GPR88 0 43 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(Cl)cc2C(=O)c2ncccn2)cc1 ZINC000147003882 II Annotated Anodyne GRM4 20 44 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(Cl)cc2C(=O)c2ncccn2)cc1 ZINC000147003882 II Annotated Anodyne PRTN3 61 39 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(Cl)cc2C(=O)c2ncccn2)cc1 ZINC000147003882 II Annotated Anodyne CCR2 17 41 CCC(C)(C)c1ccc(OC[C@@H](O)CO)cc1 ZINC000147003910 BE For-Sale Anodyne VDR 28 49 COC(=O)[C@H](Cl)Cc1c(Cl)cccc1[N+](=O)[O-] ZINC000147003946 CF For-Sale Reactive COLA 73 35 COC(=O)[C@H](Cl)Cc1c(Cl)cccc1[N+](=O)[O-] ZINC000147003946 CF For-Sale Reactive TAAR1 20 40 COc1cc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@H]32)cc(OC)c1OC ZINC000147003956 FD On-Demand Anodyne FKBP1A 18 41 CCC(=O)Nc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147004073 EI On-Demand Anodyne MDM2 94 37 CCC(=O)Nc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147004073 EI On-Demand Anodyne NAMPT 25 43 CCC(=O)Nc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147004073 EI On-Demand Anodyne GPR88 0 43 CCC(C)(C)c1ccc(OC[C@H](O)CO)cc1 ZINC000147004111 BE For-Sale Anodyne VDR 28 49 COc1cc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@H]32)cc(OC)c1OC ZINC000147004118 FD On-Demand Anodyne FKBP1A 18 41 COC(=O)[C@@H](Cl)Cc1c(Cl)cccc1[N+](=O)[O-] ZINC000147004128 CF For-Sale Reactive COLA 73 35 COC(=O)[C@@H](Cl)Cc1c(Cl)cccc1[N+](=O)[O-] ZINC000147004128 CF For-Sale Reactive TAAR1 20 40 COc1c(Cl)ccc(NS(=O)(=O)c2ccc(C(C)(C)C)cc2)c1C(=O)c1ccncc1 ZINC000147004294 JK Annotated Clean PRTN3 51 31 CCC(=O)Nc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147004298 EI On-Demand Anodyne MDM2 94 37 CCC(=O)Nc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147004298 EI On-Demand Anodyne NAMPT 25 43 CCC(=O)Nc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147004298 EI On-Demand Anodyne GPR88 0 43 Fc1ccc2c(CCNCc3cccc(OCC(F)(F)C(F)(F)F)c3)c[nH]c2c1 ZINC000147004456 HK For-Sale Anodyne MPO 71 46 C[C@@H](CNC(=O)c1cccn(Cc2ccccc2)c1=O)N1CCc2ccccc21 ZINC000147004457 GG On-Demand Anodyne DRTS_PLAFK 19 41 C[C@@H](CNC(=O)c1cccn(Cc2ccccc2)c1=O)N1CCc2ccccc21 ZINC000147004457 GG On-Demand Anodyne AVPR2 41 36 N#CC1CCN(C(=O)COc2ccc3c(c2)CCC(=O)N3)CC1 ZINC000147004466 DD On-Demand Mild HTR1D 15 41 N#CC1CCN(C(=O)COc2ccc3c(c2)CCC(=O)N3)CC1 ZINC000147004466 DD On-Demand Mild HTR1B 17 41 CCC(=O)Nc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147004468 GJ On-Demand Anodyne F2RL1 19 41 CCC(=O)Nc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147004468 GJ On-Demand Anodyne NAMPT 23 43 CCCCCCCC(=O)OC[C@@]1(CCl)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147004516 HD Annotated Mild NPR 25 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne INSR 26 49 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne IGF1R 54 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne DAPK2 20 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne JAK2 18 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne PTK2 26 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne TTK 37 40 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne CAMKK1 23 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne CAMKK2 18 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne ALK 41 49 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne MAPK7 54 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne PTK2B 15 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne DYRK1B 26 40 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne STK32C 0 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne DCLK2 22 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne DCLK1 20 41 COc1cc(N2CCN(C)CC2)ccc1Nc1nc2c(NCc3cccnc3N(C)S(C)(=O)=O)cccn2n1 ZINC000147004544 KF Annotated Anodyne NEK3 0 41 Nc1nc(Cl)cc(CNc2ccc(F)cc2)n1 ZINC000147004612 CE For-Sale Anodyne DHFR 20 43 Nc1nc(Cl)cc(CNc2ccc(F)cc2)n1 ZINC000147004612 CE For-Sale Anodyne DFR1 22 45 Nc1nc(Cl)cc(CNc2ccc(F)cc2)n1 ZINC000147004612 CE For-Sale Anodyne DRTS_TOXGO 30 45 Nc1nc(Cl)cc(CNc2ccc(F)cc2)n1 ZINC000147004612 CE For-Sale Anodyne DYR_PNECA 28 45 CCCN(CCC)[C@@H]1CCC2=C(CC(=O)CC2)C1 ZINC000147004620 BH For-Sale Anodyne HTR1A 36 45 CCCN(CCC)[C@@H]1CCC2=C(CC(=O)CC2)C1 ZINC000147004620 BH For-Sale Anodyne DRD2 28 45 CCCN(CCC)[C@@H]1CCC2=C(CC(=O)CC2)C1 ZINC000147004620 BH For-Sale Anodyne HTR1D 38 43 CCCN(CCC)[C@@H]1CCC2=C(CC(=O)CC2)C1 ZINC000147004620 BH For-Sale Anodyne HTR1B 25 43 CCCN(CCC)[C@@H]1CCC2=C(CC(=O)CC2)C1 ZINC000147004620 BH For-Sale Anodyne DRD3 18 43 C[C@H](CNC(=O)c1cccn(Cc2ccccc2)c1=O)N1CCc2ccccc21 ZINC000147004644 GG On-Demand Anodyne DRTS_PLAFK 19 41 C[C@H](CNC(=O)c1cccn(Cc2ccccc2)c1=O)N1CCc2ccccc21 ZINC000147004644 GG On-Demand Anodyne AVPR2 41 36 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147004656 HH On-Demand Anodyne CCR3 26 43 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147004656 HH On-Demand Anodyne NOS2 84 37 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147004656 HH On-Demand Anodyne EPHX2 17 41 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147004656 HH On-Demand Anodyne PRMT3 46 36 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147004656 HH On-Demand Anodyne NAMPT 44 49 CCC(=O)Nc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147004664 GJ On-Demand Anodyne F2RL1 19 41 CCC(=O)Nc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147004664 GJ On-Demand Anodyne NAMPT 23 43 CCCN(CCC)[C@H]1CCC2=C(CC(=O)CC2)C1 ZINC000147004825 BH For-Sale Anodyne HTR1A 36 45 CCCN(CCC)[C@H]1CCC2=C(CC(=O)CC2)C1 ZINC000147004825 BH For-Sale Anodyne DRD2 28 45 CCCN(CCC)[C@H]1CCC2=C(CC(=O)CC2)C1 ZINC000147004825 BH For-Sale Anodyne HTR1D 38 43 CCCN(CCC)[C@H]1CCC2=C(CC(=O)CC2)C1 ZINC000147004825 BH For-Sale Anodyne HTR1B 25 43 CCCN(CCC)[C@H]1CCC2=C(CC(=O)CC2)C1 ZINC000147004825 BH For-Sale Anodyne DRD3 18 43 CCC(=O)Nc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)cc1 ZINC000147004857 GJ On-Demand Anodyne F2RL1 19 41 CCC(=O)Nc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)cc1 ZINC000147004857 GJ On-Demand Anodyne NAMPT 23 43 CCOc1cccc(CNCCc2c[nH]c3ccc(OC)cc23)c1 ZINC000147004872 DH On-Demand Anodyne HTR1A 20 51 CCOc1cccc(CNCCc2c[nH]c3ccc(OC)cc23)c1 ZINC000147004872 DH On-Demand Anodyne HTR1D 52 51 CCOc1cccc(CNCCc2c[nH]c3ccc(OC)cc23)c1 ZINC000147004872 DH On-Demand Anodyne HTR1B 39 51 CCOc1cccc(CNCCc2c[nH]c3ccc(OC)cc23)c1 ZINC000147004872 DH On-Demand Anodyne NQO2 24 53 CCOc1cccc(CNCCc2c[nH]c3ccc(OC)cc23)c1 ZINC000147004872 DH On-Demand Anodyne MPO 65 44 CCOc1cccc(CNCCc2c[nH]c3ccc(OC)cc23)c1 ZINC000147004872 DH On-Demand Anodyne HTR1E 22 44 CCOc1cccc(CNCCc2c[nH]c3ccc(OC)cc23)c1 ZINC000147004872 DH On-Demand Anodyne MTNR1A 68 54 CCOc1cccc(CNCCc2c[nH]c3ccc(OC)cc23)c1 ZINC000147004872 DH On-Demand Anodyne MTNR1B 48 53 CCOc1cccc(CNCCc2c[nH]c3ccc(OC)cc23)c1 ZINC000147004872 DH On-Demand Anodyne ABCG2 26 43 CCCc1nc(CS(=O)(=O)CC(=O)N2c3ccccc3C[C@@H]2C)no1 ZINC000147004910 FD On-Demand Anodyne DRD4 23 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147004931 EH On-Demand Anodyne INHA 45 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147004931 EH On-Demand Anodyne KLK3 60 38 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147004931 EH On-Demand Anodyne CTSK 38 43 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147004931 EH On-Demand Anodyne HLA-DRB1 29 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147004931 EH On-Demand Anodyne FURIN 63 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147004931 EH On-Demand Anodyne ACE2 44 37 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147004931 EH On-Demand Anodyne POLG_WNV 72 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147004931 EH On-Demand Anodyne NPFFR1 48 33 CCN(CC)C(=O)c1ccc(S(=O)(=O)NCc2ccccc2-n2ccnc2)cc1 ZINC000147004972 HF On-Demand Anodyne LIMK2 41 34 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147004973 HI On-Demand Anodyne CCR3 41 39 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147004973 HI On-Demand Anodyne EPHX2 29 45 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147004973 HI On-Demand Anodyne PRMT3 40 37 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147004973 HI On-Demand Anodyne L3MBTL3 56 38 O=C(N[C@@H]1CCN(c2nccs2)C1)c1ccccc1 ZINC000147005011 CE For-Sale Anodyne DRD4 22 48 C=CCN(CC=C)C(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147005071 GE On-Demand Mild OXTR 25 40 CCCc1nc(CS(=O)(=O)CC(=O)N2c3ccccc3C[C@H]2C)no1 ZINC000147005114 FD On-Demand Anodyne DRD4 23 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147005127 EH On-Demand Anodyne INHA 45 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147005127 EH On-Demand Anodyne KLK3 60 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147005127 EH On-Demand Anodyne CTSK 38 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147005127 EH On-Demand Anodyne HLA-DRB1 29 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147005127 EH On-Demand Anodyne FURIN 63 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147005127 EH On-Demand Anodyne ACE2 44 37 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147005127 EH On-Demand Anodyne POLG_WNV 72 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1Oc1ccccc1 ZINC000147005127 EH On-Demand Anodyne NPFFR1 48 33 CCn1c(=S)[nH]c2cc(C(=O)N3CCC(C#N)CC3)ccc2c1=O ZINC000147005139 EE On-Demand Mild L3MBTL3 46 32 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005152 HI On-Demand Anodyne CCR3 41 39 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005152 HI On-Demand Anodyne EPHX2 29 45 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005152 HI On-Demand Anodyne PRMT3 40 37 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005152 HI On-Demand Anodyne L3MBTL3 56 38 O=C(N[C@H]1CCN(c2nccs2)C1)c1ccccc1 ZINC000147005189 CE For-Sale Anodyne DRD4 22 48 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCc3c(Cl)cccc32)cc1 ZINC000147005222 HH On-Demand Anodyne KCNA5 35 40 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCc3c(Cl)cccc32)cc1 ZINC000147005222 HH On-Demand Anodyne LIMK2 43 37 COc1ccccc1-c1cc(O)ccc1C(=O)O ZINC000147005254 BF In-Stock Anodyne DHODH 16 40 COc1ccccc1-c1cc(O)ccc1C(=O)O ZINC000147005254 BF In-Stock Anodyne CA14 22 44 COc1ccccc1-c1cc(O)ccc1C(=O)O ZINC000147005254 BF In-Stock Anodyne HDAC2 17 40 COc1ccccc1-c1cc(O)ccc1C(=O)O ZINC000147005254 BF In-Stock Anodyne ALS 47 36 COc1ccccc1-c1cc(O)ccc1C(=O)O ZINC000147005254 BF In-Stock Anodyne AKR1C2 56 35 C=CCN(CC=C)C(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147005259 GE On-Demand Mild OXTR 25 40 Nc1cccc(N2CCN(CCCF)CC2)c1 ZINC000147005280 BD For-Sale Anodyne HTR1A 67 55 Nc1cccc(N2CCN(CCCF)CC2)c1 ZINC000147005280 BD For-Sale Anodyne DRD2 36 48 Nc1cccc(N2CCN(CCCF)CC2)c1 ZINC000147005280 BD For-Sale Anodyne DRD4 26 44 Nc1cccc(N2CCN(CCCF)CC2)c1 ZINC000147005280 BD For-Sale Anodyne HTR2A 46 55 Nc1cccc(N2CCN(CCCF)CC2)c1 ZINC000147005280 BD For-Sale Anodyne DRD3 24 41 Nc1cccc(N2CCN(CCCF)CC2)c1 ZINC000147005280 BD For-Sale Anodyne CACNA1G 0 43 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005329 HI On-Demand Anodyne CCR3 41 39 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005329 HI On-Demand Anodyne EPHX2 29 45 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005329 HI On-Demand Anodyne PRMT3 40 37 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005329 HI On-Demand Anodyne L3MBTL3 56 38 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(OC2CCCC2)c(Cl)c1 ZINC000147005470 GG On-Demand Anodyne PDE4A 26 40 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(OCC)cc2)cc1 ZINC000147005493 JI For-Sale Anodyne PTGER2 23 46 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(OCC)cc2)cc1 ZINC000147005493 JI For-Sale Anodyne MMP13 29 52 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(OCC)cc2)cc1 ZINC000147005493 JI For-Sale Anodyne ADAM17 16 52 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(OCC)cc2)cc1 ZINC000147005493 JI For-Sale Anodyne MMP3 16 47 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(OCC)cc2)cc1 ZINC000147005493 JI For-Sale Anodyne MMP8 19 45 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(OCC)cc2)cc1 ZINC000147005493 JI For-Sale Anodyne MMP9 32 52 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(OCC)cc2)cc1 ZINC000147005493 JI For-Sale Anodyne MMP12 15 44 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(OCC)cc2)cc1 ZINC000147005493 JI For-Sale Anodyne CXCR3 26 55 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(OCC)cc2)cc1 ZINC000147005493 JI For-Sale Anodyne MMP1 28 45 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(OCC)cc2)cc1 ZINC000147005493 JI For-Sale Anodyne NAMPT 31 43 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005509 HI On-Demand Anodyne CCR3 41 39 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005509 HI On-Demand Anodyne EPHX2 29 45 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005509 HI On-Demand Anodyne PRMT3 40 37 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147005509 HI On-Demand Anodyne L3MBTL3 56 38 NCc1ccc(Oc2ccccc2)c(C(F)(F)F)c1 ZINC000147005645 CH For-Sale Anodyne TAAR1 25 47 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(OC2CCCC2)c(Cl)c1 ZINC000147005657 GG On-Demand Anodyne PDE4A 26 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCCc1ccc(Cl)s1)C2 ZINC000147005730 FG On-Demand Anodyne NQO2 36 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCCc1ccc(Cl)s1)C2 ZINC000147005730 FG On-Demand Anodyne MTNR1A 80 45 COc1ccc2c(c1)OC[C@@H](C(=O)NCCc1ccc(Cl)s1)C2 ZINC000147005730 FG On-Demand Anodyne MTNR1B 65 39 COc1ccc2c(c1)OC[C@@H](C(=O)NCCc1ccc(Cl)s1)C2 ZINC000147005730 FG On-Demand Anodyne ROCK2 22 40 N#CC1CCN(C(=O)Cc2cccc3cccnc23)CC1 ZINC000147005740 CF On-Demand Mild PTAFR 27 42 CN1[C@@H]2CCC[C@@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005781 DF On-Demand Anodyne HTR3A 53 64 CN1[C@@H]2CCC[C@@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005781 DF On-Demand Anodyne HTR4 47 44 CN1[C@@H]2CCC[C@@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005781 DF On-Demand Anodyne CNR2 25 41 CN1[C@@H]2CCC[C@@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005781 DF On-Demand Anodyne HTR3B 0 64 CN1[C@@H]2CCC[C@@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005781 DF On-Demand Anodyne CASP1 24 45 CN1[C@@H]2CCC[C@@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005781 DF On-Demand Anodyne GLRA1 45 37 COC(=O)N1[C@H](C(=O)O)C[C@@H]2CCCC[C@@H]21 ZINC000147005797 BD For-Sale Anodyne ACE 17 57 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H](C)c2ccc(F)c(Cl)c2)cc1 ZINC000147005843 HI On-Demand Anodyne LEF 57 37 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H](C)c2ccc(F)c(Cl)c2)cc1 ZINC000147005843 HI On-Demand Anodyne LIMK2 23 41 Nc1n[nH]c(-c2ccccn2)c1Br ZINC000147005902 BD For-Sale Anodyne METAP2 42 37 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccnc1OC)C2 ZINC000147005918 DE On-Demand Anodyne ROCK2 40 50 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccnc1OC)C2 ZINC000147005918 DE On-Demand Anodyne CDC42BPA 0 46 CCOC(=O)NCC(=O)Nc1ccc(NS(C)(=O)=O)c(OC)c1 ZINC000147005967 EC On-Demand Anodyne TRPV1 31 43 CCOC(=O)NCC(=O)Nc1ccc(NS(C)(=O)=O)c(OC)c1 ZINC000147005967 EC On-Demand Anodyne ENPP1 59 38 CN1[C@H]2CCC[C@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005983 DF On-Demand Anodyne HTR3A 53 64 CN1[C@H]2CCC[C@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005983 DF On-Demand Anodyne HTR4 47 44 CN1[C@H]2CCC[C@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005983 DF On-Demand Anodyne CNR2 25 41 CN1[C@H]2CCC[C@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005983 DF On-Demand Anodyne HTR3B 0 64 CN1[C@H]2CCC[C@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005983 DF On-Demand Anodyne CASP1 24 45 CN1[C@H]2CCC[C@H]1CC(NC(=O)c1nccc3ccccc13)C2 ZINC000147005983 DF On-Demand Anodyne GLRA1 45 37 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCc3cc(Cl)ccc32)cc1 ZINC000147006038 HH On-Demand Anodyne OPRD1 27 42 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCc3cc(Cl)ccc32)cc1 ZINC000147006038 HH On-Demand Anodyne F10 23 46 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCc3cc(Cl)ccc32)cc1 ZINC000147006038 HH On-Demand Anodyne KCNA5 34 46 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCc3cc(Cl)ccc32)cc1 ZINC000147006038 HH On-Demand Anodyne STS 26 40 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCc3cc(Cl)ccc32)cc1 ZINC000147006038 HH On-Demand Anodyne LIMK2 33 40 O=C(C[C@]1(C(=O)O)CCSC1)Nc1cccc(OCc2cccnc2)c1 ZINC000147006044 FG On-Demand Anodyne PPIA 37 41 O=C(C[C@]1(C(=O)O)CCSC1)Nc1cccc(OCc2cccnc2)c1 ZINC000147006044 FG On-Demand Anodyne NAMPT 26 40 CCCCO[C@@H](C)C(=O)N1CCN(c2cnn(-c3ccccc3)c(=O)c2Cl)CC1 ZINC000147006063 HF On-Demand Anodyne P2RY12 89 33 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCc3cc(Cl)ccc32)cc1 ZINC000147006246 HH On-Demand Anodyne OPRD1 27 42 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCc3cc(Cl)ccc32)cc1 ZINC000147006246 HH On-Demand Anodyne F10 23 46 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCc3cc(Cl)ccc32)cc1 ZINC000147006246 HH On-Demand Anodyne KCNA5 34 46 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCc3cc(Cl)ccc32)cc1 ZINC000147006246 HH On-Demand Anodyne STS 26 40 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCc3cc(Cl)ccc32)cc1 ZINC000147006246 HH On-Demand Anodyne LIMK2 33 40 CC(C)(C)NC(=O)c1cccc(NC(=O)C[C@]2(C(=O)O)CCSC2)c1 ZINC000147006251 FF On-Demand Anodyne KCNK3 93 37 CC(C)(C)NC(=O)c1cccc(NC(=O)C[C@]2(C(=O)O)CCSC2)c1 ZINC000147006251 FF On-Demand Anodyne KCNK9 47 37 CCCCO[C@H](C)C(=O)N1CCN(c2cnn(-c3ccccc3)c(=O)c2Cl)CC1 ZINC000147006263 HF On-Demand Anodyne P2RY12 89 33 COC(=O)N(C1c2ccccc2-c2ccccc21)[C@@H](Cc1ccc(OC)cc1)C(=O)O ZINC000147006308 HJ In-Stock Anodyne PPARG 15 42 COC(=O)N(C1c2ccccc2-c2ccccc21)[C@@H](Cc1ccc(OC)cc1)C(=O)O ZINC000147006308 HJ In-Stock Anodyne PPARA 19 41 COC(=O)N(C1c2ccccc2-c2ccccc21)[C@@H](Cc1ccc(OC)cc1)C(=O)O ZINC000147006308 HJ In-Stock Anodyne MMP2 17 40 COC(=O)N(C1c2ccccc2-c2ccccc21)[C@@H](Cc1ccc(OC)cc1)C(=O)O ZINC000147006308 HJ In-Stock Anodyne MMP3 21 41 COC(=O)N(C1c2ccccc2-c2ccccc21)[C@@H](Cc1ccc(OC)cc1)C(=O)O ZINC000147006308 HJ In-Stock Anodyne MMP1 28 40 COC(=O)N(C1c2ccccc2-c2ccccc21)[C@@H](Cc1ccc(OC)cc1)C(=O)O ZINC000147006308 HJ In-Stock Anodyne PSMB8 43 34 O=C(Nc1cc(C(F)(F)F)c[nH]c1=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147006402 FH On-Demand Anodyne ROCK2 16 47 CC(C)(C)OC(=O)N1CC(C(C)(C)N)C1 ZINC000147006437 BD In-Stock Anodyne GPR119 17 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)c1 ZINC000147006440 GF On-Demand Bother HRH2 17 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)c1 ZINC000147006440 GF On-Demand Bother TAAR1 50 55 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)c1 ZINC000147006440 GF On-Demand Bother AKR1C3 15 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)c1 ZINC000147006440 GF On-Demand Bother AKR1C2 33 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)c1 ZINC000147006440 GF On-Demand Bother KCNK3 49 37 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)c1 ZINC000147006440 GF On-Demand Bother KCNK9 42 37 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(C(N)=O)c1 ZINC000147006459 CC On-Demand Anodyne CCKAR 20 41 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(C(N)=O)c1 ZINC000147006459 CC On-Demand Anodyne CCKBR 17 41 CSc1ccc(C(=O)Nc2ccc(F)c([C@]3(C)CCSC(N)=N3)c2)s1 ZINC000147006554 GJ Annotated Anodyne BACE2 51 67 CSc1ccc(C(=O)Nc2ccc(F)c([C@]3(C)CCSC(N)=N3)c2)s1 ZINC000147006554 GJ Annotated Anodyne BACE1 25 67 O=C(Nc1cc(C(F)(F)F)c[nH]c1=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147006594 FH On-Demand Anodyne ROCK2 16 47 [N-]=[N+]=Nc1ccc(I)cc1Cl ZINC000147006604 CH In-Stock Mild NISCH 20 40 O=C(Nc1ccc(Oc2ccccc2)cc1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147006638 FG On-Demand Anodyne LTA4H 42 38 O=C(Nc1ccc(Oc2ccccc2)cc1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147006638 FG On-Demand Anodyne F13A1 15 40 COc1ccc(OC[C@@H](O)CO)c(C(C)(C)C)c1 ZINC000147006728 CD For-Sale Anodyne ADRB2 0 46 COc1ccc(OC[C@@H](O)CO)c(C(C)(C)C)c1 ZINC000147006728 CD For-Sale Anodyne VDR 26 45 O=C(Nc1cc(C(F)(F)F)c[nH]c1=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147006768 FH On-Demand Anodyne ROCK2 16 47 N#CC1CCN(C(=O)CCCOc2ccc(F)cc2)CC1 ZINC000147006794 CF On-Demand Mild HRH3 19 44 N#CC1CCN(C(=O)CCCOc2ccc(F)cc2)CC1 ZINC000147006794 CF On-Demand Mild MEN1 43 37 O=C(Nc1ccc(Oc2ccccc2)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147006811 FG On-Demand Anodyne LTA4H 42 38 O=C(Nc1ccc(Oc2ccccc2)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147006811 FG On-Demand Anodyne F13A1 15 40 CCOc1ccc(Nc2nc(-c3ccc4c(cnn4C)c3)cn3ccnc23)cc1OC ZINC000147006904 HI For-Sale Anodyne SYK 58 89 COc1ccc(OC[C@H](O)CO)c(C(C)(C)C)c1 ZINC000147006929 CD For-Sale Anodyne ADRB2 0 46 COc1ccc(OC[C@H](O)CO)c(C(C)(C)C)c1 ZINC000147006929 CD For-Sale Anodyne VDR 26 45 O=C(Nc1cc(C(F)(F)F)c[nH]c1=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147006942 FH On-Demand Anodyne ROCK2 16 47 Fc1cc(CN2CCCCC2)cc(C(F)(F)F)c1 ZINC000147006954 CH On-Demand Anodyne TACR1 15 40 O=C(Nc1ccc(Oc2ccccc2)cc1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147007004 FG On-Demand Anodyne LTA4H 42 38 O=C(Nc1ccc(Oc2ccccc2)cc1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147007004 FG On-Demand Anodyne F13A1 15 40 COc1ccc(Nc2nc3c(Nc4ccc(S(C)(=O)=O)cc4)cccn3n2)cc1 ZINC000147007044 HH Annotated Anodyne PTGS2 15 45 COc1ccc(Nc2nc3c(Nc4ccc(S(C)(=O)=O)cc4)cccn3n2)cc1 ZINC000147007044 HH Annotated Anodyne JAK3 15 78 COc1ccc(Nc2nc3c(Nc4ccc(S(C)(=O)=O)cc4)cccn3n2)cc1 ZINC000147007044 HH Annotated Anodyne JAK2 33 78 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cc(C(F)(F)F)c[nH]c1=O)C2 ZINC000147007181 FF On-Demand Anodyne ROCK2 40 49 O=C(Nc1ccc(Oc2ccccc2)cc1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147007191 FG On-Demand Anodyne LTA4H 42 38 O=C(Nc1ccc(Oc2ccccc2)cc1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147007191 FG On-Demand Anodyne F13A1 15 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)NC2CCCCC2)cc1 ZINC000147007372 GE On-Demand Anodyne MAPK14 16 48 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)NC2CCCCC2)cc1 ZINC000147007372 GE On-Demand Anodyne MC5R 18 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)NC2CCCCC2)cc1 ZINC000147007372 GE On-Demand Anodyne EPHX2 19 43 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cc(C(F)(F)F)c[nH]c1=O)C2 ZINC000147007374 FF On-Demand Anodyne ROCK2 40 49 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)NC2CCCCC2)cc1 ZINC000147007558 GE On-Demand Anodyne MAPK14 16 48 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)NC2CCCCC2)cc1 ZINC000147007558 GE On-Demand Anodyne MC5R 18 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)NC2CCCCC2)cc1 ZINC000147007558 GE On-Demand Anodyne EPHX2 19 43 CCC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147007601 KB Annotated Anodyne POLA1 52 55 CCC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147007601 KB Annotated Anodyne P2RY6 121 47 CCC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147007601 KB Annotated Anodyne POLB 57 55 CCC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147007601 KB Annotated Anodyne P2RX4 41 38 CCC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147007601 KB Annotated Anodyne P2RX1 56 38 CCC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147007601 KB Annotated Anodyne P2RY4 130 47 CCC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147007601 KB Annotated Anodyne P2RY1 32 40 CCC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147007601 KB Annotated Anodyne P2RY2 164 49 CCC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147007601 KB Annotated Anodyne P2RY14 54 37 CCC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147007601 KB Annotated Anodyne RNASE1 40 31 CCC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147007601 KB Annotated Anodyne GPR17 45 34 COc1ncccc1NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147007607 DG On-Demand Anodyne NAMPT 24 41 COc1ncccc1NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147007607 DG On-Demand Anodyne G2YM83_BOTF4 61 35 COc1ncccc1NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147007786 DG On-Demand Anodyne NAMPT 24 41 COc1ncccc1NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147007786 DG On-Demand Anodyne G2YM83_BOTF4 61 35 Nc1ccn([C@@H]2O[C@](CF)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147007814 KB Annotated Anodyne POLA1 48 56 Nc1ccn([C@@H]2O[C@](CF)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147007814 KB Annotated Anodyne P2RY6 121 45 Nc1ccn([C@@H]2O[C@](CF)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147007814 KB Annotated Anodyne POLB 57 56 Nc1ccn([C@@H]2O[C@](CF)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147007814 KB Annotated Anodyne P2RX4 42 38 Nc1ccn([C@@H]2O[C@](CF)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147007814 KB Annotated Anodyne P2RX1 57 38 Nc1ccn([C@@H]2O[C@](CF)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147007814 KB Annotated Anodyne P2RY4 130 45 Nc1ccn([C@@H]2O[C@](CF)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147007814 KB Annotated Anodyne P2RY2 163 49 Nc1ccn([C@@H]2O[C@](CF)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147007814 KB Annotated Anodyne P2RY14 53 38 Nc1ccn([C@@H]2O[C@](CF)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147007814 KB Annotated Anodyne RNASE1 42 33 Nc1ccn([C@@H]2O[C@](CF)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147007814 KB Annotated Anodyne GPR17 44 34 CCOC[C@@H](O)COc1ccc(C(C)(C)c2ccccc2)cc1 ZINC000147007886 DH On-Demand Anodyne ADRB2 20 42 COc1ncccc1NC(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147007978 DG On-Demand Anodyne NAMPT 24 41 COc1ncccc1NC(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147007978 DG On-Demand Anodyne G2YM83_BOTF4 61 35 Nc1ccn([C@@H]2O[C@@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(C3CC3)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147008039 KB Annotated Anodyne POLA1 50 59 Nc1ccn([C@@H]2O[C@@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(C3CC3)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147008039 KB Annotated Anodyne P2RY6 118 45 Nc1ccn([C@@H]2O[C@@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(C3CC3)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147008039 KB Annotated Anodyne POLB 59 59 Nc1ccn([C@@H]2O[C@@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(C3CC3)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147008039 KB Annotated Anodyne P2RX4 40 36 Nc1ccn([C@@H]2O[C@@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(C3CC3)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147008039 KB Annotated Anodyne P2RX1 55 36 Nc1ccn([C@@H]2O[C@@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(C3CC3)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147008039 KB Annotated Anodyne P2RY4 125 45 Nc1ccn([C@@H]2O[C@@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(C3CC3)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147008039 KB Annotated Anodyne P2RY2 160 48 Nc1ccn([C@@H]2O[C@@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(C3CC3)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147008039 KB Annotated Anodyne P2RY14 48 37 Nc1ccn([C@@H]2O[C@@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(C3CC3)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147008039 KB Annotated Anodyne GPR17 44 35 CCOC[C@H](O)COc1ccc(C(C)(C)c2ccccc2)cc1 ZINC000147008090 DH On-Demand Anodyne ADRB2 20 42 CC(C)[C@@H](CNC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1)c1ccccc1 ZINC000147008133 GG On-Demand Bother COLA 57 36 COc1ncccc1NC(=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147008171 DG On-Demand Anodyne NAMPT 24 41 COc1ncccc1NC(=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147008171 DG On-Demand Anodyne G2YM83_BOTF4 61 35 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CASP3 15 42 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild BMP1 61 35 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild KLK3 82 46 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CTSB 56 40 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild PAPA1_CARPA 62 42 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CYSP_TRYCR 60 41 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CTSK 31 44 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CTSL 44 47 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CAPNS1 63 39 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild MMP11 43 30 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CTSS 19 44 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CAPN1 81 48 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CASP1 27 43 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CAPN2 110 42 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CASP6 23 40 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild CASP9 30 40 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild TGM2 36 43 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild NPR 62 38 C=CC[C@@H](CO)NC(=O)OCc1ccccc1 ZINC000147008239 BD For-Sale Mild PSMB5 47 41 CC(C)[C@H](CNC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1)c1ccccc1 ZINC000147008327 GG On-Demand Bother COLA 57 36 COc1ncccc1NC(=O)[C@@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147008372 EH On-Demand Anodyne NAMPT 22 40 C=C1C[C@H](C(=O)O)[C@@H]([C@H](N)C(=O)O)C1 ZINC000147008415 AC For-Sale Mild GRM6 22 57 COc1ccc([N+](=O)[O-])c(C(=O)NC[C@@H](c2ccccc2)C(C)C)c1 ZINC000147008541 EH On-Demand Bother COLA 48 37 COc1ccc([N+](=O)[O-])c(C(=O)NC[C@@H](c2ccccc2)C(C)C)c1 ZINC000147008541 EH On-Demand Bother TAAR1 21 41 COc1ccc([N+](=O)[O-])c(C(=O)NC[C@@H](c2ccccc2)C(C)C)c1 ZINC000147008541 EH On-Demand Bother AKR1C3 20 45 COc1ccc([N+](=O)[O-])c(C(=O)NC[C@@H](c2ccccc2)C(C)C)c1 ZINC000147008541 EH On-Demand Bother AKR1C2 47 45 COc1ncccc1NC(=O)[C@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147008563 EH On-Demand Anodyne NAMPT 22 40 C=C1C[C@@H](C(=O)O)[C@H]([C@H](N)C(=O)O)C1 ZINC000147008587 AC For-Sale Mild GRM6 22 57 COc1ccc(C23C[C@H]4C[C@@H](CC(C(=O)N5CCC(C#N)CC5)(C4)C2)C3)cc1 ZINC000147008612 GI On-Demand Mild BOTA 21 48 COc1ccc(C23C[C@H]4C[C@@H](CC(C(=O)N5CCC(C#N)CC5)(C4)C2)C3)cc1 ZINC000147008612 GI On-Demand Mild NPBWR1 51 29 O=C1c2ccc(Cl)cc2C(=O)c2c(Cl)ccc(Cl)c21 ZINC000147008685 DI For-Sale Clean USP7 22 42 CCCOC(=O)[C@@H](CC(C)C)NC(=O)c1ccc2c(c1)OCO2 ZINC000147008694 DF Annotated Anodyne CAPN1 23 40 CCCOC(=O)[C@@H](CC(C)C)NC(=O)c1ccc2c(c1)OCO2 ZINC000147008694 DF Annotated Anodyne CAPN2 33 43 CCCOC(=O)[C@@H](CC(C)C)NC(=O)c1ccc2c(c1)OCO2 ZINC000147008694 DF Annotated Anodyne PLM1_PLAFA 17 46 CCCOC(=O)[C@@H](CC(C)C)NC(=O)c1ccc2c(c1)OCO2 ZINC000147008694 DF Annotated Anodyne NPR 47 32 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(F)c(NC(=O)Cc2ccccc2)c1 ZINC000147008719 HH On-Demand Anodyne CA5B 29 40 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(F)c(NC(=O)Cc2ccccc2)c1 ZINC000147008719 HH On-Demand Anodyne CA5A 33 40 O=C(N[C@H](CCCCO)C(=O)O)OCC1c2ccccc2-c2ccccc21 ZINC000147008732 FG In-Stock Anodyne KLK3 57 36 O=C(N[C@H](CCCCO)C(=O)O)OCC1c2ccccc2-c2ccccc21 ZINC000147008732 FG In-Stock Anodyne C3AR1 56 35 O=C(N[C@H](CCCCO)C(=O)O)OCC1c2ccccc2-c2ccccc21 ZINC000147008732 FG In-Stock Anodyne HDAC2 23 40 CC1(C)CNCCc2ccccc21 ZINC000147008738 AE In-Stock Anodyne PRCP 42 33 COc1ccc([N+](=O)[O-])c(C(=O)NC[C@H](c2ccccc2)C(C)C)c1 ZINC000147008742 EH On-Demand Bother COLA 48 37 COc1ccc([N+](=O)[O-])c(C(=O)NC[C@H](c2ccccc2)C(C)C)c1 ZINC000147008742 EH On-Demand Bother TAAR1 21 41 COc1ccc([N+](=O)[O-])c(C(=O)NC[C@H](c2ccccc2)C(C)C)c1 ZINC000147008742 EH On-Demand Bother AKR1C3 20 45 COc1ccc([N+](=O)[O-])c(C(=O)NC[C@H](c2ccccc2)C(C)C)c1 ZINC000147008742 EH On-Demand Bother AKR1C2 47 45 COc1cccc(Cl)c1CC(=O)NC(C)(C)C#N ZINC000147008747 CE On-Demand Mild CXCL8 41 31 COc1cccc(Cl)c1CC(=O)NC(C)(C)C#N ZINC000147008747 CE On-Demand Mild PLA2G2A 19 41 COc1ccc(C)cc1-n1ccc(C(=O)Nc2ccc3oc(C)nc3c2)n1 ZINC000147008756 FH On-Demand Anodyne AGPAT2 35 41 COc1ccc(C)cc1-n1ccc(C(=O)Nc2ccc3oc(C)nc3c2)n1 ZINC000147008756 FH On-Demand Anodyne ENPP1 56 33 COc1ncccc1NC(=O)[C@H]1C[C@H]1c1cccc(Br)c1 ZINC000147008764 EH On-Demand Anodyne NAMPT 22 40 CCN(CC)C(=O)c1ccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1Cl ZINC000147008768 GI On-Demand Anodyne EPHX2 27 50 CC(C)[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147008837 GF On-Demand Mild ELANE 16 42 CC(C)[C@H](NC(=O)c1ccc([N+](=O)[O-])cc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147008837 GF On-Demand Mild CCR1 72 45 COC(=O)[C@H]1Cc2c([nH]c3ccccc23)[C@H](c2ccc(Cl)nc2)N1 ZINC000147008936 EF For-Sale Anodyne PDE5A 38 40 COC(=O)[C@H]1Cc2c([nH]c3ccccc23)[C@H](c2ccc(Cl)nc2)N1 ZINC000147008936 EF For-Sale Anodyne PDE11A 48 32 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(F)c2)c1 ZINC000147008957 EF On-Demand Bother DRD4 41 32 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(F)c2)c1 ZINC000147008957 EF On-Demand Bother TAAR1 25 44 CCN(CC)C(=O)c1ccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)cc1Cl ZINC000147008980 GI On-Demand Anodyne EPHX2 27 50 O=C(NCCN1CCOCC1)c1cc2ncccn2n1 ZINC000147008991 CB On-Demand Anodyne HTR1A 15 42 O=C(NCCN1CCOCC1)c1cc2ncccn2n1 ZINC000147008991 CB On-Demand Anodyne DRD4 43 33 O=C(NCCN1CCOCC1)c1cc2ncccn2n1 ZINC000147008991 CB On-Demand Anodyne DRD3 21 44 O=C(NCCN1CCOCC1)c1cc2ncccn2n1 ZINC000147008991 CB On-Demand Anodyne EPHX2 16 46 O=C(NCCN1CCOCC1)c1cc2ncccn2n1 ZINC000147008991 CB On-Demand Anodyne PLD2 61 35 O=C(NCCN1CCOCC1)c1cc2ncccn2n1 ZINC000147008991 CB On-Demand Anodyne HPGDS 27 48 ONc1ccccc1CN1CCCC1 ZINC000147009023 AE For-Sale Anodyne KCNQ2 63 37 ONc1ccccc1CN1CCCC1 ZINC000147009023 AE For-Sale Anodyne SIGMAR1 15 43 CC(C)[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147009028 GF On-Demand Mild ELANE 16 42 CC(C)[C@@H](NC(=O)c1ccc([N+](=O)[O-])cc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147009028 GF On-Demand Mild CCR1 72 45 O=C(Nc1nc2ccccc2s1)c1cccc2c1CN(c1ccc(CCCc3ccccc3)c(C(=O)O)n1)CC2 ZINC000147009084 KK Annotated Anodyne BCL2 0 61 O=C(Nc1nc2ccccc2s1)c1cccc2c1CN(c1ccc(CCCc3ccccc3)c(C(=O)O)n1)CC2 ZINC000147009084 KK Annotated Anodyne BCL2L2 30 61 Cn1cc(C(=O)NC2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)cn1 ZINC000147009167 GF On-Demand Anodyne NPBWR1 42 31 CCN(CC)C(=O)c1ccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1Cl ZINC000147009172 GI On-Demand Anodyne EPHX2 27 50 COc1ccc([N+](=O)[O-])c(C(=O)NCC2(N3CCSCC3)CCCC2)c1 ZINC000147009243 GF On-Demand Bother HCN1 88 46 COc1ccc([N+](=O)[O-])c(C(=O)NCC2(N3CCSCC3)CCCC2)c1 ZINC000147009243 GF On-Demand Bother HCN4 64 44 CCCc1nc(CS(=O)(=O)CC(=O)NC23CC4CC(CC(C4)C2)C3)no1 ZINC000147009249 GE On-Demand Anodyne EPHX2 42 41 Cc1[nH]nc(-c2nc3ccccc3[nH]2)c1C(=O)N[C@@H]1CCCNC1 ZINC000147009306 DD Annotated Anodyne CHEK1 31 47 Cn1cc(C(=O)NC2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)cn1 ZINC000147009347 GF On-Demand Anodyne NPBWR1 42 31 CCN(CC)C(=O)c1ccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)cc1Cl ZINC000147009361 GI On-Demand Anodyne EPHX2 27 50 CN1CCC(c2ccc(Nc3nc4c(Nc5ccccc5S(C)(=O)=O)cccn4n3)cc2)CC1 ZINC000147009397 JI Annotated Anodyne HTR1F 46 35 CN1CCC(c2ccc(Nc3nc4c(Nc5ccccc5S(C)(=O)=O)cccn4n3)cc2)CC1 ZINC000147009397 JI Annotated Anodyne JAK2 37 56 Cc1[nH]nc(-c2nc3ccccc3[nH]2)c1C(=O)N[C@H]1CCCNC1 ZINC000147009508 DD Annotated Anodyne CHEK1 31 47 Cn1cc(C(=O)NC2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)cn1 ZINC000147009534 GF On-Demand Anodyne NPBWR1 42 31 CCOC(=O)CN(C1CC1)S(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-] ZINC000147009573 FD On-Demand Bother COLA 40 32 Cn1cc(C(=O)NC2CCN(C(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)CC2)cn1 ZINC000147009746 GF On-Demand Anodyne NPBWR1 42 31 c1ccc2[nH]c(Cc3ccncc3)cc2c1 ZINC000147009787 BG For-Sale Anodyne MAOA 16 43 O=C(Nc1cccc(Cn2cccn2)c1)c1cccn(Cc2ccccc2)c1=O ZINC000147009790 GG On-Demand Anodyne PTGER3 25 46 O=C(Nc1cccc(Cn2cccn2)c1)c1cccn(Cc2ccccc2)c1=O ZINC000147009790 GG On-Demand Anodyne KCNK3 80 39 O=C(Nc1cccc(Cn2cccn2)c1)c1cccn(Cc2ccccc2)c1=O ZINC000147009790 GG On-Demand Anodyne KCNK9 58 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(-n2cnc3ccccc32)cc1 ZINC000147009792 FG On-Demand Anodyne F9 45 49 Cc1cc(N)c(C#N)c(O)n1 ZINC000147009910 AC For-Sale Anodyne RPS27 42 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(-n2cnc3ccccc32)cc1 ZINC000147009987 FG On-Demand Anodyne F9 45 49 CC(C)CNC(=O)c1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1 ZINC000147010007 FF On-Demand Anodyne F3 93 40 CCN(CC)C(=O)Cc1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147010032 HD On-Demand Anodyne CCR5 23 40 CCN(CC)C(=O)Cc1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147010032 HD On-Demand Anodyne EPHX2 44 46 O=C(NCc1ccc(-n2cccn2)cc1)c1ccn(-c2cccc(F)c2)n1 ZINC000147010167 FG On-Demand Anodyne AMP1_PLAFQ 63 44 CCN(CC)C(=O)Cc1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147010214 HD On-Demand Anodyne CCR5 23 40 CCN(CC)C(=O)Cc1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147010214 HD On-Demand Anodyne EPHX2 44 46 O=C(CC1CC1)N[C@H]1CC[C@@H](c2nnc3cnc4[nH]ccc4n23)C1 ZINC000147010398 DE Annotated Anodyne JAK1 18 42 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@H](CCCC)NC(N)=O)c1 ZINC000147010406 GD On-Demand Anodyne CA2 17 50 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@H](CCCC)NC(N)=O)c1 ZINC000147010406 GD On-Demand Anodyne CA4 16 50 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@H](CCCC)NC(N)=O)c1 ZINC000147010406 GD On-Demand Anodyne HDAC11 46 35 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@H](CCCC)NC(N)=O)c1 ZINC000147010406 GD On-Demand Anodyne ST14 43 36 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@H](CCCC)NC(N)=O)c1 ZINC000147010406 GD On-Demand Anodyne LEF 26 41 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@H](CCCC)NC(N)=O)c1 ZINC000147010406 GD On-Demand Anodyne POLG_WNV 40 30 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@@H](CCCC)NC(N)=O)c1 ZINC000147010598 GD On-Demand Anodyne CA2 17 50 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@@H](CCCC)NC(N)=O)c1 ZINC000147010598 GD On-Demand Anodyne CA4 16 50 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@@H](CCCC)NC(N)=O)c1 ZINC000147010598 GD On-Demand Anodyne HDAC11 46 35 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@@H](CCCC)NC(N)=O)c1 ZINC000147010598 GD On-Demand Anodyne ST14 43 36 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@@H](CCCC)NC(N)=O)c1 ZINC000147010598 GD On-Demand Anodyne LEF 26 41 CCCCNS(=O)(=O)c1cccc(NC(=O)[C@@H](CCCC)NC(N)=O)c1 ZINC000147010598 GD On-Demand Anodyne POLG_WNV 40 30 Brc1cccc(Nc2ncnc(Nc3cccc(Br)c3)n2)c1 ZINC000147010775 HJ For-Sale Anodyne EGFR 126 55 Brc1cccc(Nc2ncnc(Nc3cccc(Br)c3)n2)c1 ZINC000147010775 HJ For-Sale Anodyne ERBB2 18 50 Brc1cccc(Nc2ncnc(Nc3cccc(Br)c3)n2)c1 ZINC000147010775 HJ For-Sale Anodyne SYK 28 45 Brc1cccc(Nc2ncnc(Nc3cccc(Br)c3)n2)c1 ZINC000147010775 HJ For-Sale Anodyne FBP1 18 57 Brc1cccc(Nc2ncnc(Nc3cccc(Br)c3)n2)c1 ZINC000147010775 HJ For-Sale Anodyne ERBB4 29 50 Brc1cccc(Nc2ncnc(Nc3cccc(Br)c3)n2)c1 ZINC000147010775 HJ For-Sale Anodyne BMX 21 40 Brc1cccc(Nc2ncnc(Nc3cccc(Br)c3)n2)c1 ZINC000147010775 HJ For-Sale Anodyne ABCG2 16 54 O=C1OCC[C@@H]1CNC1CCCC1 ZINC000147010792 AD For-Sale Anodyne TRAR 51 32 O=C1OCC[C@@H]1CNC1CCCC1 ZINC000147010792 AD For-Sale Anodyne PHZR 50 30 CCOC(=O)N1CCN(c2ncc(I)cn2)CC1 ZINC000147010852 FD On-Demand Anodyne P2RY12 44 36 CCOC(=O)N1CCN(c2ncc(I)cn2)CC1 ZINC000147010852 FD On-Demand Anodyne GPR119 15 44 COc1cccc(F)c1CN1CCC[C@@H](NC(=O)c2ccc3[nH]nc(-c4ccncc4)c3c2)C1 ZINC000147010881 JI Annotated Anodyne DRD2 27 40 COc1cccc(F)c1CN1CCC[C@@H](NC(=O)c2ccc3[nH]nc(-c4ccncc4)c3c2)C1 ZINC000147010881 JI Annotated Anodyne DRD4 36 40 COc1cccc(F)c1CN1CCC[C@@H](NC(=O)c2ccc3[nH]nc(-c4ccncc4)c3c2)C1 ZINC000147010881 JI Annotated Anodyne SSTR5 47 40 COc1cccc(F)c1CN1CCC[C@@H](NC(=O)c2ccc3[nH]nc(-c4ccncc4)c3c2)C1 ZINC000147010881 JI Annotated Anodyne MCHR1 18 46 COc1cccc(F)c1CN1CCC[C@@H](NC(=O)c2ccc3[nH]nc(-c4ccncc4)c3c2)C1 ZINC000147010881 JI Annotated Anodyne TTK 71 40 COc1cccc(F)c1CN1CCC[C@@H](NC(=O)c2ccc3[nH]nc(-c4ccncc4)c3c2)C1 ZINC000147010881 JI Annotated Anodyne ACKR3 44 30 N#Cc1ccccc1Oc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147010900 GF On-Demand Mild ADRB1 43 35 N#Cc1ccccc1Oc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147010900 GF On-Demand Mild PFKFB3 51 35 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H](C)c2oc3ccccc3c2C)cc1 ZINC000147010927 HI On-Demand Anodyne MMP13 25 46 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H](C)c2oc3ccccc3c2C)cc1 ZINC000147010927 HI On-Demand Anodyne MMP12 40 41 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H](C)c2oc3ccccc3c2C)cc1 ZINC000147010927 HI On-Demand Anodyne ADAMTS4 38 46 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H](C)c2oc3ccccc3c2C)cc1 ZINC000147010927 HI On-Demand Anodyne LIMK2 41 35 O=C1OCC[C@H]1CNC1CCCC1 ZINC000147010986 AD For-Sale Anodyne TRAR 51 32 O=C1OCC[C@H]1CNC1CCCC1 ZINC000147010986 AD For-Sale Anodyne PHZR 50 30 CC(C)(C)OC(=O)N1CCN(C(=O)OCc2ccccc2)C[C@H]1CCO ZINC000147010995 FF For-Sale Anodyne PREP 24 40 CC(C)(C)OC(=O)N1CCN(C(=O)OCc2ccccc2)C[C@H]1CCO ZINC000147010995 FF For-Sale Anodyne SLC12A5 49 33 N#Cc1ccccc1Oc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147011076 GF On-Demand Mild ADRB1 43 35 N#Cc1ccccc1Oc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147011076 GF On-Demand Mild PFKFB3 51 35 Fc1ccc(F)c(-c2ccccn2)c1 ZINC000147011100 AG For-Sale Anodyne GRM5 19 51 Nc1nc(NCC(=O)O)cs1 ZINC000147011135 AC For-Sale Anodyne SHV5 41 35 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2ccccc2OC)CC1 ZINC000147011174 GD On-Demand Anodyne F2 28 42 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2ccccc2OC)CC1 ZINC000147011174 GD On-Demand Anodyne P2RY12 186 36 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2ccccc2OC)CC1 ZINC000147011174 GD On-Demand Anodyne CCR1 22 43 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2ccccc2OC)CC1 ZINC000147011174 GD On-Demand Anodyne ST14 51 37 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCC(F)(F)CC1 ZINC000147011247 GJ Annotated Anodyne FGFR1 22 47 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCC(F)(F)CC1 ZINC000147011247 GJ Annotated Anodyne ITK 35 49 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCC(F)(F)CC1 ZINC000147011247 GJ Annotated Anodyne LDLR 0 40 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCC(F)(F)CC1 ZINC000147011247 GJ Annotated Anodyne FLT1 17 47 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCC(F)(F)CC1 ZINC000147011247 GJ Annotated Anodyne HPSE 19 41 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCC(F)(F)CC1 ZINC000147011247 GJ Annotated Anodyne TTK 43 39 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCC(F)(F)CC1 ZINC000147011247 GJ Annotated Anodyne PAK4 16 47 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCC(F)(F)CC1 ZINC000147011247 GJ Annotated Anodyne NR2E3 77 47 COC(=O)C(C)(C)NC(=O)Cc1c(Cl)cccc1OC ZINC000147011259 CD On-Demand Anodyne ECR 23 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(C)s1)C2 ZINC000147011267 DF On-Demand Anodyne MTNR1A 26 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(C)s1)C2 ZINC000147011267 DF On-Demand Anodyne ROCK2 28 42 CCOC[C@@H](O)COc1ccccc1[C@@H](C)CC ZINC000147011347 CF On-Demand Anodyne ADRB2 34 43 CCOC[C@@H](O)COc1ccccc1[C@@H](C)CC ZINC000147011347 CF On-Demand Anodyne ADRB3 0 43 CCOC[C@@H](O)COc1ccccc1[C@@H](C)CC ZINC000147011347 CF On-Demand Anodyne ABCB1 35 42 CCOC[C@@H](O)COc1ccccc1[C@@H](C)CC ZINC000147011347 CF On-Demand Anodyne AO-ACHE 0 47 CC(C)(C)OC(=O)C[C@@H](C#N)c1ccc(F)cc1 ZINC000147011498 BG For-Sale Mild PAPA1_CARPA 36 42 CCOC[C@H](O)COc1ccccc1[C@@H](C)CC ZINC000147011532 CF On-Demand Anodyne ADRB2 0 43 CCOC[C@H](O)COc1ccccc1[C@@H](C)CC ZINC000147011532 CF On-Demand Anodyne ADRB3 0 43 CCOC[C@H](O)COc1ccccc1[C@@H](C)CC ZINC000147011532 CF On-Demand Anodyne ABCB1 22 40 CCOC[C@H](O)COc1ccccc1[C@@H](C)CC ZINC000147011532 CF On-Demand Anodyne AO-ACHE 0 47 COC(=O)C[C@H](NS(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-])c1ccc(F)cc1 ZINC000147011558 HF On-Demand Bother COLA 56 36 CCN(Cc1ccccc1NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1)C(C)=O ZINC000147011633 HF On-Demand Bother COLA 85 36 CC(C)(C)OC(=O)C[C@H](C#N)c1ccc(F)cc1 ZINC000147011684 BG For-Sale Mild PAPA1_CARPA 36 42 CCOC[C@@H](O)COc1ccccc1[C@H](C)CC ZINC000147011721 CF On-Demand Anodyne ADRB2 34 43 CCOC[C@@H](O)COc1ccccc1[C@H](C)CC ZINC000147011721 CF On-Demand Anodyne ADRB3 0 43 CCOC[C@@H](O)COc1ccccc1[C@H](C)CC ZINC000147011721 CF On-Demand Anodyne ABCB1 35 42 CCOC[C@@H](O)COc1ccccc1[C@H](C)CC ZINC000147011721 CF On-Demand Anodyne AO-ACHE 0 47 CCCCNC(=O)C1CCN(C(=O)[C@@H](CCC)NC(N)=O)CC1 ZINC000147011757 EC On-Demand Anodyne P2RY12 92 34 CCCCNC(=O)C1CCN(C(=O)[C@@H](CCC)NC(N)=O)CC1 ZINC000147011757 EC On-Demand Anodyne TPP2 33 41 COC(=O)C[C@@H](NS(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-])c1ccc(F)cc1 ZINC000147011760 HF On-Demand Bother COLA 56 36 CCCc1nc(CS(=O)(=O)CC(=O)NCc2cccc(OC)c2)no1 ZINC000147011832 FD On-Demand Anodyne ROCK1 31 41 CCCc1nc(CS(=O)(=O)CC(=O)NCc2cccc(OC)c2)no1 ZINC000147011832 FD On-Demand Anodyne MTNR1A 52 43 CCCc1nc(CS(=O)(=O)CC(=O)NCc2cccc(OC)c2)no1 ZINC000147011832 FD On-Demand Anodyne MTNR1B 44 39 CCOC[C@H](O)COc1ccccc1[C@H](C)CC ZINC000147011918 CF On-Demand Anodyne ADRB2 34 43 CCOC[C@H](O)COc1ccccc1[C@H](C)CC ZINC000147011918 CF On-Demand Anodyne ADRB3 0 43 CCOC[C@H](O)COc1ccccc1[C@H](C)CC ZINC000147011918 CF On-Demand Anodyne ABCB1 35 42 CCOC[C@H](O)COc1ccccc1[C@H](C)CC ZINC000147011918 CF On-Demand Anodyne AO-ACHE 0 47 CN(C(=O)c1cccc(NC(=O)C[C@]2(C(=O)O)CCSC2)c1)c1ccccc1 ZINC000147011957 GG On-Demand Anodyne KCNK3 48 41 CCCCNC(=O)C1CCN(C(=O)[C@H](CCC)NC(N)=O)CC1 ZINC000147011958 EC On-Demand Anodyne P2RY12 92 34 CCCCNC(=O)C1CCN(C(=O)[C@H](CCC)NC(N)=O)CC1 ZINC000147011958 EC On-Demand Anodyne TPP2 33 41 O=C(CNS(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-])N1CCCc2ccccc21 ZINC000147011976 HF On-Demand Bother AVPR2 40 46 CCN(CC)C(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147012049 HH On-Demand Bother TAAR1 26 47 CCN(CC)C(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147012049 HH On-Demand Bother AKR1C2 44 38 CCN(CC)C(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147012049 HH On-Demand Bother USP7 28 41 CCN(CC)C(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147012049 HH On-Demand Bother USP47 35 41 N#CC1CCN(C(=O)c2cc(-c3ccco3)n(-c3cccc(Cl)c3)n2)CC1 ZINC000147012092 GI On-Demand Mild RPA1 62 34 C=CCCOCC(=O)Nc1ncc(Cc2cccc(F)c2)s1 ZINC000147012211 DG On-Demand Mild SCD1 39 42 C=CCCOCC(=O)Nc1ncc(Cc2cccc(F)c2)s1 ZINC000147012211 DG On-Demand Mild SCD 37 42 CCN(CC)C(=O)COc1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147012248 HG On-Demand Bother MTNR1A 18 40 CCN(CC)C(=O)COc1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147012248 HG On-Demand Bother MTNR1B 22 41 CCN(CC)C(=O)COc1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147012248 HG On-Demand Bother TAAR1 39 52 CCN(CC)C(=O)COc1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147012248 HG On-Demand Bother AKR1C2 23 40 CCN(CC)C(=O)COc1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147012248 HG On-Demand Bother KCNK3 53 43 CCN(CC)C(=O)COc1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147012248 HG On-Demand Bother KCNK9 45 43 CCCc1nc(CS(=O)(=O)c2ccc(S(=O)(=O)N3CCOCC3)cn2)no1 ZINC000147012255 HC On-Demand Anodyne MERTK 25 40 COc1ccc(Nc2nc3c(-c4cnn(S(C)(=O)=O)c4)cccn3n2)cc1 ZINC000147012257 GE Annotated Anodyne JAK2 32 69 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147012293 GH On-Demand Anodyne MTNR1A 42 39 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147012293 GH On-Demand Anodyne ROCK2 43 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc2c(c1)OCCO2 ZINC000147012323 FE On-Demand Anodyne EDNRA 44 39 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc2c(c1)OCCO2 ZINC000147012323 FE On-Demand Anodyne TRHR 49 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc2c(c1)OCCO2 ZINC000147012323 FE On-Demand Anodyne TRY1_BOVIN 51 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc2c(c1)OCCO2 ZINC000147012323 FE On-Demand Anodyne NTSR1 65 32 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc2c(c1)OCCO2 ZINC000147012323 FE On-Demand Anodyne NTSR2 44 32 O=C(Nc1ncc(Cc2cccc(F)c2)s1)c1cccn(Cc2ccccc2)c1=O ZINC000147012426 HI On-Demand Anodyne DRTS_PLAFK 19 42 O=C(Nc1ncc(Cc2cccc(F)c2)s1)c1cccn(Cc2ccccc2)c1=O ZINC000147012426 HI On-Demand Anodyne SCD1 40 42 O=C(Nc1ncc(Cc2cccc(F)c2)s1)c1cccn(Cc2ccccc2)c1=O ZINC000147012426 HI On-Demand Anodyne SCD 37 42 CC[C@H](C)C(=O)Nc1cccc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147012482 GH On-Demand Anodyne MTNR1A 42 39 CC[C@H](C)C(=O)Nc1cccc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147012482 GH On-Demand Anodyne ROCK2 43 42 Cc1ccccc1-c1csc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)n1 ZINC000147012510 HH On-Demand Bother MPL 65 36 Cc1ccccc1-c1csc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)n1 ZINC000147012510 HH On-Demand Bother GCK 32 48 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc2c(c1)OCCO2 ZINC000147012522 FE On-Demand Anodyne EDNRA 44 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc2c(c1)OCCO2 ZINC000147012522 FE On-Demand Anodyne TRHR 49 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc2c(c1)OCCO2 ZINC000147012522 FE On-Demand Anodyne TRY1_BOVIN 51 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc2c(c1)OCCO2 ZINC000147012522 FE On-Demand Anodyne NTSR1 65 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc2c(c1)OCCO2 ZINC000147012522 FE On-Demand Anodyne NTSR2 44 32 CCOC(=O)NCC(=O)Nc1ncc(Cc2cccc(F)c2)s1 ZINC000147012625 EF On-Demand Anodyne SCD1 36 54 CCOC(=O)NCC(=O)Nc1ncc(Cc2cccc(F)c2)s1 ZINC000147012625 EF On-Demand Anodyne SCD 0 54 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147012649 GH On-Demand Anodyne MTNR1A 42 39 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147012649 GH On-Demand Anodyne ROCK2 43 42 CCN(Cc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1)C(C)=O ZINC000147012682 FE On-Demand Anodyne PLA2G4B 43 31 CCN(Cc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1)C(C)=O ZINC000147012682 FE On-Demand Anodyne HIF1A 21 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc2c(c1)OCCO2 ZINC000147012685 FE On-Demand Anodyne EDNRA 44 39 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc2c(c1)OCCO2 ZINC000147012685 FE On-Demand Anodyne TRHR 49 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc2c(c1)OCCO2 ZINC000147012685 FE On-Demand Anodyne TRY1_BOVIN 51 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc2c(c1)OCCO2 ZINC000147012685 FE On-Demand Anodyne NTSR1 65 32 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc2c(c1)OCCO2 ZINC000147012685 FE On-Demand Anodyne NTSR2 44 32 COc1ccc(S(=O)(=O)N2CCC(C(=O)NC3C4CC5CC(C4)CC3C5)CC2)cc1OC ZINC000147012696 JG On-Demand Anodyne HSD11B1 52 34 COc1ccc(S(=O)(=O)N2CCC(C(=O)NC3C4CC5CC(C4)CC3C5)CC2)cc1OC ZINC000147012696 JG On-Demand Anodyne MMP3 18 42 COc1ccc(S(=O)(=O)N2CCC(C(=O)NC3C4CC5CC(C4)CC3C5)CC2)cc1OC ZINC000147012696 JG On-Demand Anodyne EPHX2 46 45 COc1ccc(S(=O)(=O)N2CCC(C(=O)NC3C4CC5CC(C4)CC3C5)CC2)cc1OC ZINC000147012696 JG On-Demand Anodyne TGM2 32 42 COc1ccc(S(=O)(=O)N2CCC(C(=O)NC3C4CC5CC(C4)CC3C5)CC2)cc1OC ZINC000147012696 JG On-Demand Anodyne MMP7 16 42 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147012814 HD On-Demand Anodyne EPHX2 17 41 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147012814 HD On-Demand Anodyne TGM2 62 44 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147012814 HD On-Demand Anodyne F13A1 94 48 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147012814 HD On-Demand Anodyne NAMPT 36 45 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)N2CCOCC2)c(Cl)c1 ZINC000147012816 HE On-Demand Anodyne EPHX2 16 46 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc2c(c1)OCCO2 ZINC000147012840 FE On-Demand Anodyne EDNRA 44 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc2c(c1)OCCO2 ZINC000147012840 FE On-Demand Anodyne TRHR 49 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc2c(c1)OCCO2 ZINC000147012840 FE On-Demand Anodyne TRY1_BOVIN 51 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc2c(c1)OCCO2 ZINC000147012840 FE On-Demand Anodyne NTSR1 65 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc2c(c1)OCCO2 ZINC000147012840 FE On-Demand Anodyne NTSR2 44 32 CC[C@H](C)C(=O)Nc1cccc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147012865 GH On-Demand Anodyne MTNR1A 42 39 CC[C@H](C)C(=O)Nc1cccc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147012865 GH On-Demand Anodyne ROCK2 43 42 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147012997 HD On-Demand Anodyne EPHX2 17 41 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147012997 HD On-Demand Anodyne TGM2 62 44 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147012997 HD On-Demand Anodyne F13A1 94 48 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147012997 HD On-Demand Anodyne AKR1C3 22 41 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147012997 HD On-Demand Anodyne NAMPT 36 45 O=C(C[C@]1(C(=O)O)CCSC1)Nc1cccc(C(=O)N2CCCCC2)c1 ZINC000147013038 GF On-Demand Anodyne EPHX2 18 42 O=C(C[C@]1(C(=O)O)CCSC1)Nc1cccc(C(=O)N2CCCCC2)c1 ZINC000147013038 GF On-Demand Anodyne L3MBTL3 47 40 O=c1cc(N(CCO)CCO)oc2c1ccc1ccccc12 ZINC000147013185 CD For-Sale Bother CYP1A2 15 52 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147013196 HD On-Demand Anodyne EPHX2 17 41 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147013196 HD On-Demand Anodyne TGM2 62 44 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147013196 HD On-Demand Anodyne F13A1 94 48 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147013196 HD On-Demand Anodyne NAMPT 36 45 O=C(c1ccn(-c2cccc(F)c2)n1)N1CCCCc2ccccc21 ZINC000147013240 EH On-Demand Anodyne AVPR2 63 55 O=C(c1ccn(-c2cccc(F)c2)n1)N1CCCCc2ccccc21 ZINC000147013240 EH On-Demand Anodyne AVPR1A 15 43 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)N2CCCCCC2)cc1 ZINC000147013249 GG On-Demand Anodyne L3MBTL3 76 38 CC[C@H](C)NC(=O)c1cccc(CNC(=O)c2ccc3c(c2)COC3)c1 ZINC000147013269 FG On-Demand Anodyne CHRM3 15 42 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147013395 HD On-Demand Anodyne EPHX2 17 41 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147013395 HD On-Demand Anodyne TGM2 62 44 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147013395 HD On-Demand Anodyne F13A1 94 48 O=C(Nc1ccc(S(=O)(=O)N2CCCC2)cc1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147013395 HD On-Demand Anodyne NAMPT 36 45 CC[C@H](C)NC(=O)c1cccc(CNC(=O)c2cnn(-c3ccccc3Cl)c2)c1 ZINC000147013512 HH On-Demand Anodyne MAPK10 17 43 Cc1ccc(Oc2ccc(OCC(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147013751 FH On-Demand Mild CPT1A 58 40 CC[C@H](C)NC(=O)c1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147013919 GI On-Demand Anodyne CTSV 32 40 CC[C@H](C)NC(=O)c1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147013919 GI On-Demand Anodyne MDM2 41 34 CC[C@H](C)NC(=O)c1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147013919 GI On-Demand Anodyne PDS 44 31 CC[C@H](C)NC(=O)c1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147014285 GI On-Demand Anodyne CTSV 32 40 CC[C@H](C)NC(=O)c1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147014285 GI On-Demand Anodyne MDM2 41 34 CC[C@H](C)NC(=O)c1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147014285 GI On-Demand Anodyne PDS 44 31 CC[C@@H](C)NC(=O)c1cccc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147014511 GG On-Demand Anodyne DRD4 42 33 COc1ccc([N+](=O)[O-])c(C(=O)N2CCC(NC(=O)c3ccccc3F)CC2)c1 ZINC000147014547 HF For-Sale Bother DRD4 19 43 COc1ccc([N+](=O)[O-])c(C(=O)N2CCC(NC(=O)c3ccccc3F)CC2)c1 ZINC000147014547 HF For-Sale Bother CCR3 17 42 COc1ccc([N+](=O)[O-])c(C(=O)N2CCC(NC(=O)c3ccccc3F)CC2)c1 ZINC000147014547 HF For-Sale Bother AKR1C2 17 42 CC(C)Oc1ccc(-c2n[nH]c3ccc(C(=O)N[C@@H]4CN(C)CC[C@H]4c4ccccc4)cc23)cn1 ZINC000147014552 JJ Annotated Anodyne TTK 72 48 CC[C@H](C)NC(=O)c1cccc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147014712 GG On-Demand Anodyne DRD4 42 33 COc1cccc(CCOCc2cccc(CCBr)c2)c1 ZINC000147014759 EI For-Sale Reactive ABCB1 15 43 COc1ccc(-c2ccc(Cl)cc2C)cc1C=O ZINC000147014817 CI For-Sale Anodyne PTGS2 18 40 CN(C)C(=O)C[C@H](NS(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-])c1ccccc1 ZINC000147014825 HF On-Demand Bother BDKRB1 22 42 CN(C)C(=O)C[C@H](NS(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-])c1ccccc1 ZINC000147014825 HF On-Demand Bother COLA 107 36 CC[C@@H](C)NC(=O)c1cccc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147014902 GG On-Demand Anodyne DRD4 42 33 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(F)(F)F)c2)cc1 ZINC000147014942 FF On-Demand Anodyne CETP 20 40 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(F)(F)F)c2)cc1 ZINC000147014942 FF On-Demand Anodyne ACR 45 42 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(F)(F)F)c2)cc1 ZINC000147014942 FF On-Demand Anodyne HIF1A 27 45 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(F)(F)F)c2)cc1 ZINC000147014942 FF On-Demand Anodyne TAAR1 34 40 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(F)(F)F)c2)cc1 ZINC000147014942 FF On-Demand Anodyne KCNK3 40 35 CN(C)C(=O)C[C@@H](NS(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-])c1ccccc1 ZINC000147015031 HF On-Demand Bother BDKRB1 22 42 CN(C)C(=O)C[C@@H](NS(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-])c1ccccc1 ZINC000147015031 HF On-Demand Bother COLA 107 36 CC[C@H](C)NC(=O)c1cccc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147015095 GG On-Demand Anodyne DRD4 42 33 CCOC(=O)c1ccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@@H]32)cc1 ZINC000147015170 ED On-Demand Anodyne NOD2 17 41 C[C@@H](C(=O)Nc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1)n1cccn1 ZINC000147015181 HE On-Demand Anodyne ADORA2B 38 43 CC[C@@H](C)[C@@H](C)NS(=O)(=O)c1ccc(C(=O)N(CC)CC)cc1 ZINC000147015243 EF On-Demand Anodyne ADAMTS4 44 36 CC[C@@H](C)[C@@H](C)NS(=O)(=O)c1ccc(C(=O)N(CC)CC)cc1 ZINC000147015243 EF On-Demand Anodyne LIMK2 43 38 CN(C)C(=O)Cc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147015304 FH On-Demand Anodyne MDM2 70 40 CN(C)C(=O)Cc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147015304 FH On-Demand Anodyne NAMPT 23 40 C[C@H](C(=O)Nc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1)n1cccn1 ZINC000147015341 HE On-Demand Anodyne ADORA2B 38 43 CCOC(=O)c1ccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@@H]32)cc1 ZINC000147015395 ED On-Demand Anodyne NOD2 17 41 CC[C@H](C)[C@@H](C)NS(=O)(=O)c1ccc(C(=O)N(CC)CC)cc1 ZINC000147015442 EF On-Demand Anodyne ADAMTS4 44 36 CC[C@H](C)[C@@H](C)NS(=O)(=O)c1ccc(C(=O)N(CC)CC)cc1 ZINC000147015442 EF On-Demand Anodyne LIMK2 43 38 CN(C)C(=O)Cc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147015513 FH On-Demand Anodyne MDM2 70 40 CN(C)C(=O)Cc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147015513 FH On-Demand Anodyne NAMPT 23 40 CCCCc1oc2ccccc2c1CN(C)C(=O)[C@@H](CCC)NC(N)=O ZINC000147015542 FH On-Demand Anodyne THRA 16 43 CCn1cc(Nc2nc3c(-c4ccc(C(F)(F)F)cc4)cccn3n2)cn1 ZINC000147015561 FI Annotated Anodyne JAK2 26 56 CCOC(=O)c1ccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@H]32)cc1 ZINC000147015594 ED On-Demand Anodyne NOD2 17 41 CC[C@@H](C)[C@H](C)NS(=O)(=O)c1ccc(C(=O)N(CC)CC)cc1 ZINC000147015645 EF On-Demand Anodyne ADAMTS4 44 36 CC[C@@H](C)[C@H](C)NS(=O)(=O)c1ccc(C(=O)N(CC)CC)cc1 ZINC000147015645 EF On-Demand Anodyne LIMK2 43 38 CN(C)C(=O)Cc1ccc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147015715 FH On-Demand Anodyne MDM2 70 40 CN(C)C(=O)Cc1ccc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147015715 FH On-Demand Anodyne NAMPT 23 40 CC(C)S(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(N5CCN(C)CC5)cc4)nc23)cc1 ZINC000147015770 JI Annotated Anodyne JAK3 24 83 CC(C)S(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(N5CCN(C)CC5)cc4)nc23)cc1 ZINC000147015770 JI Annotated Anodyne JAK2 49 83 CC(C)S(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(N5CCN(C)CC5)cc4)nc23)cc1 ZINC000147015770 JI Annotated Anodyne HCK 44 36 CC(C)S(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(N5CCN(C)CC5)cc4)nc23)cc1 ZINC000147015770 JI Annotated Anodyne CDK4 17 41 CCOC(=O)c1ccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@H]32)cc1 ZINC000147015783 ED On-Demand Anodyne NOD2 17 41 O=C(C[C@]1(C(=O)O)CCSC1)Nc1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000147015802 HH On-Demand Anodyne TAAR1 37 41 O=C(C[C@]1(C(=O)O)CCSC1)Nc1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000147015802 HH On-Demand Anodyne KCNK3 103 53 O=C(C[C@]1(C(=O)O)CCSC1)Nc1cccc(C(=O)Nc2cccc(F)c2)c1 ZINC000147015802 HH On-Demand Anodyne KCNK9 51 47 CC[C@H](C)[C@H](C)NS(=O)(=O)c1ccc(C(=O)N(CC)CC)cc1 ZINC000147015816 EF On-Demand Anodyne ADAMTS4 44 36 CC[C@H](C)[C@H](C)NS(=O)(=O)c1ccc(C(=O)N(CC)CC)cc1 ZINC000147015816 EF On-Demand Anodyne LIMK2 43 38 CN(C)C(=O)Cc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147015931 FH On-Demand Anodyne MDM2 70 40 CN(C)C(=O)Cc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147015931 FH On-Demand Anodyne NAMPT 23 40 N#Cc1cccc(NC(=O)c2cccc(NC(=O)C[C@]3(C(=O)O)CCSC3)c2)c1 ZINC000147016011 HG On-Demand Anodyne KCNK3 95 38 N#Cc1cccc(NC(=O)c2cccc(NC(=O)C[C@]3(C(=O)O)CCSC3)c2)c1 ZINC000147016011 HG On-Demand Anodyne KCNK9 47 37 CC(C)NC(=O)Cc1ccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147016107 HG On-Demand Anodyne NOS2 97 36 CC(C)NC(=O)Cc1ccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147016107 HG On-Demand Anodyne ROCK2 21 42 CC(C)NC(=O)Cc1ccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147016107 HG On-Demand Anodyne NAMPT 41 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CC(=O)N(C)C)cc1)C2 ZINC000147016201 FF On-Demand Anodyne MTNR1A 30 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CC(=O)N(C)C)cc1)C2 ZINC000147016201 FF On-Demand Anodyne MTNR1B 18 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CC(=O)N(C)C)cc1)C2 ZINC000147016201 FF On-Demand Anodyne ROCK2 35 53 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CC(=O)N(C)C)cc1)C2 ZINC000147016201 FF On-Demand Anodyne CA9 15 40 Clc1cccc(CCNCc2cccc(OCc3ccccn3)c2)c1 ZINC000147016261 FJ On-Demand Anodyne ADRB2 16 41 Clc1cccc(CCNCc2cccc(OCc3ccccn3)c2)c1 ZINC000147016261 FJ On-Demand Anodyne ADRB1 18 41 CC(C)NC(=O)Cc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147016366 HI On-Demand Anodyne NPR1 42 33 CC(C)NC(=O)Cc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147016366 HI On-Demand Anodyne FURIN 53 33 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(CC(=O)N(C)C)cc1)C2 ZINC000147016388 FF On-Demand Anodyne MTNR1A 30 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(CC(=O)N(C)C)cc1)C2 ZINC000147016388 FF On-Demand Anodyne MTNR1B 18 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(CC(=O)N(C)C)cc1)C2 ZINC000147016388 FF On-Demand Anodyne ROCK2 35 53 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(CC(=O)N(C)C)cc1)C2 ZINC000147016388 FF On-Demand Anodyne CA9 15 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCc3cccc(C#N)c3)c2)c1 ZINC000147016484 HI On-Demand Mild MAOB 23 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCc3cccc(C#N)c3)c2)c1 ZINC000147016484 HI On-Demand Mild PTGER3 15 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCc3cccc(C#N)c3)c2)c1 ZINC000147016484 HI On-Demand Mild ADAMTS4 16 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCc3cccc(C#N)c3)c2)c1 ZINC000147016484 HI On-Demand Mild TAAR1 39 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCc3cccc(C#N)c3)c2)c1 ZINC000147016484 HI On-Demand Mild FFAR1 21 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCc3cccc(C#N)c3)c2)c1 ZINC000147016484 HI On-Demand Mild KCNK3 43 36 COc1ccc(-c2ccc(C(C)=O)cc2)cc1C=O ZINC000147016527 CG For-Sale Anodyne RARB 16 43 COc1ccc(-c2ccc(C(C)=O)cc2)cc1C=O ZINC000147016527 CG For-Sale Anodyne TUBB1 43 40 O=C(NCCC1CCCCC1)c1cccn(Cc2ccccc2)c1=O ZINC000147016542 EH On-Demand Anodyne DRD4 16 41 O=C(NCCC1CCCCC1)c1cccn(Cc2ccccc2)c1=O ZINC000147016542 EH On-Demand Anodyne ACHE 32 54 O=C(NCCC1CCCCC1)c1cccn(Cc2ccccc2)c1=O ZINC000147016542 EH On-Demand Anodyne CNR2 23 72 O=C(NCCC1CCCCC1)c1cccn(Cc2ccccc2)c1=O ZINC000147016542 EH On-Demand Anodyne POLR1A 61 37 CC(C)NC(=O)Cc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147016557 HI On-Demand Anodyne NPR1 42 33 CC(C)NC(=O)Cc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147016557 HI On-Demand Anodyne FURIN 53 33 CC(C)NC(=O)Cc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147016713 HI On-Demand Anodyne NPR1 42 33 CC(C)NC(=O)Cc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147016713 HI On-Demand Anodyne FURIN 53 33 CC1CCN(C(=O)c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)CC1 ZINC000147016820 GE On-Demand Anodyne EPHX2 18 40 CC1CCN(C(=O)c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)CC1 ZINC000147016820 GE On-Demand Anodyne L3MBTL3 75 36 Cc1ccccc1C(=O)NC1CCN(C(=O)c2ccn(-c3cccc(F)c3)n2)CC1 ZINC000147016824 HG On-Demand Anodyne MAPK14 15 40 Cc1ccccc1C(=O)NC1CCN(C(=O)c2ccn(-c3cccc(F)c3)n2)CC1 ZINC000147016824 HG On-Demand Anodyne CCR8 64 36 CC(C)NC(=O)Cc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147016870 HI On-Demand Anodyne NPR1 42 33 CC(C)NC(=O)Cc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147016870 HI On-Demand Anodyne FURIN 53 33 CC1CCN(C(=O)c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)CC1 ZINC000147016952 GE On-Demand Anodyne EPHX2 18 40 CC1CCN(C(=O)c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)CC1 ZINC000147016952 GE On-Demand Anodyne L3MBTL3 75 36 Nc1ccnc(-c2ccn3c(-c4cccc(NC(=O)NCC(F)(F)F)c4)cnc3c2)n1 ZINC000147016973 IH Annotated Anodyne BRAF 46 39 CC(C)=CCC/C(C)=C/CC/C(C)=C/CSC(C)(C)C(=O)O ZINC000147016986 DK Annotated Anodyne GGPS1 51 44 CC(C)=CCC/C(C)=C/CC/C(C)=C/CSC(C)(C)C(=O)O ZINC000147016986 DK Annotated Anodyne FDFT1 22 40 CC(C)=CCC/C(C)=C/CC/C(C)=C/CSC(C)(C)C(=O)O ZINC000147016986 DK Annotated Anodyne STE14 0 62 CC(C)=CCC/C(C)=C/CC/C(C)=C/CSC(C)(C)C(=O)O ZINC000147016986 DK Annotated Anodyne TRPA1 22 41 O=C(Nc1cccc2[nH]nc(-c3nc4ccc(N5CCOCC5)cc4[nH]3)c12)[C@H]1CC1(F)F ZINC000147017077 IH Annotated Anodyne PDGFRB 0 57 O=C(Nc1cccc2[nH]nc(-c3nc4ccc(N5CCOCC5)cc4[nH]3)c12)[C@H]1CC1(F)F ZINC000147017077 IH Annotated Anodyne FGFR1 23 49 O=C(Nc1cccc2[nH]nc(-c3nc4ccc(N5CCOCC5)cc4[nH]3)c12)[C@H]1CC1(F)F ZINC000147017077 IH Annotated Anodyne FLT1 17 57 CCNC(=O)COc1cccc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000147017092 HE On-Demand Anodyne ADRB2 24 41 CCNC(=O)COc1cccc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000147017092 HE On-Demand Anodyne ADRB1 57 42 CCNC(=O)COc1cccc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000147017092 HE On-Demand Anodyne ADRB3 21 41 CCNC(=O)COc1cccc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000147017092 HE On-Demand Anodyne ACOX1 48 39 NC(=O)c1ccc(OCC(=O)Nc2ccc(N3CCCS3(=O)=O)cc2)cc1 ZINC000147017095 GD On-Demand Anodyne ADORA2B 37 41 NC(=O)c1ccc(OCC(=O)Nc2ccc(N3CCCS3(=O)=O)cc2)cc1 ZINC000147017095 GD On-Demand Anodyne ACR 53 35 O=C(Nc1cccc2[nH]nc(-c3nc4ccc(N5CCOCC5)cc4[nH]3)c12)[C@@H]1CC1(F)F ZINC000147017174 IH Annotated Anodyne PDGFRB 0 57 O=C(Nc1cccc2[nH]nc(-c3nc4ccc(N5CCOCC5)cc4[nH]3)c12)[C@@H]1CC1(F)F ZINC000147017174 IH Annotated Anodyne FGFR1 23 49 O=C(Nc1cccc2[nH]nc(-c3nc4ccc(N5CCOCC5)cc4[nH]3)c12)[C@@H]1CC1(F)F ZINC000147017174 IH Annotated Anodyne FLT1 17 57 Cc1c(NC(=O)C[C@]2(C(=O)O)CCSC2)cccc1NC(=O)c1ccccc1 ZINC000147017188 GH On-Demand Anodyne KCNK3 80 38 Cc1c(NC(=O)C[C@]2(C(=O)O)CCSC2)cccc1NC(=O)c1ccccc1 ZINC000147017188 GH On-Demand Anodyne KCNK9 40 38 O=C(NCC(F)(F)F)Nc1cccc(-c2cnc3cc(-c4ccncn4)ccn23)c1 ZINC000147017200 HI Annotated Anodyne BRAF 44 43 CCN(Cc1ccccc1)C(=O)CNS(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-] ZINC000147017207 HF On-Demand Bother COLA 103 38 CCN(Cc1ccccc1)C(=O)CNS(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-] ZINC000147017207 HF On-Demand Bother LIMK2 22 42 CCNC(=O)COc1cccc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000147017248 HE On-Demand Anodyne ADRB2 24 41 CCNC(=O)COc1cccc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000147017248 HE On-Demand Anodyne ADRB1 57 42 CCNC(=O)COc1cccc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000147017248 HE On-Demand Anodyne ADRB3 21 41 CCNC(=O)COc1cccc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000147017248 HE On-Demand Anodyne ACOX1 48 39 Cc1ccc(CNC(=O)c2cnn(-c3ccccc3Cl)c2)cn1 ZINC000147017278 EG On-Demand Anodyne NAMPT 51 41 CN1CCC(c2ccc(Nc3nc4c(Nc5cccnc5N(C)S(C)(=O)=O)cccn4n3)cc2)CC1 ZINC000147017339 KH Annotated Anodyne JAK2 34 49 CN1CCC(c2ccc(Nc3nc4c(Nc5cccnc5N(C)S(C)(=O)=O)cccn4n3)cc2)CC1 ZINC000147017339 KH Annotated Anodyne PTK2 22 46 CC(C)CNC(=O)c1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1Cl ZINC000147017447 GG On-Demand Anodyne F3 72 32 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017473 HH On-Demand Anodyne FBP1 21 41 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017473 HH On-Demand Anodyne EPHX2 25 45 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017473 HH On-Demand Anodyne TGM2 56 40 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017473 HH On-Demand Anodyne MDM2 67 36 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017473 HH On-Demand Anodyne F13A1 67 39 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017473 HH On-Demand Anodyne NAMPT 86 47 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017640 HH On-Demand Anodyne FBP1 21 41 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017640 HH On-Demand Anodyne EPHX2 25 45 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017640 HH On-Demand Anodyne TGM2 56 40 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017640 HH On-Demand Anodyne MDM2 67 36 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017640 HH On-Demand Anodyne F13A1 67 39 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017640 HH On-Demand Anodyne NAMPT 86 47 CCCCO[C@@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017682 EE On-Demand Anodyne CA2 48 43 CCCCO[C@@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017682 EE On-Demand Anodyne CA1 38 48 CCCCO[C@@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017682 EE On-Demand Anodyne CA4 38 43 CCCCO[C@@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017682 EE On-Demand Anodyne CA14 28 41 CCCCO[C@@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017682 EE On-Demand Anodyne CA9 25 44 CCCCO[C@@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017682 EE On-Demand Anodyne P96878_MYCTU 23 44 Cc1ccc(CN(C(C)C)S(=O)(=O)c2c(Cl)cccc2[N+](=O)[O-])s1 ZINC000147017750 GI On-Demand Bother COLA 99 38 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017821 HH On-Demand Anodyne FBP1 21 41 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017821 HH On-Demand Anodyne EPHX2 25 45 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017821 HH On-Demand Anodyne TGM2 56 40 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017821 HH On-Demand Anodyne MDM2 67 36 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017821 HH On-Demand Anodyne F13A1 67 39 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147017821 HH On-Demand Anodyne NAMPT 86 47 CC(C)[C@H](NC(=O)NCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147017824 EE On-Demand Mild ACE 24 42 CC(C)[C@H](NC(=O)NCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147017824 EE On-Demand Mild MME 21 42 CC(C)[C@H](NC(=O)NCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147017824 EE On-Demand Mild ANPEP 26 42 CC(C)[C@H](NC(=O)NCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147017824 EE On-Demand Mild PAPA1_CARPA 37 40 CC(C)[C@H](NC(=O)NCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147017824 EE On-Demand Mild CTSL 15 43 CC(C)[C@H](NC(=O)NCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147017824 EE On-Demand Mild CCR1 56 52 CC(C)[C@H](NC(=O)NCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147017824 EE On-Demand Mild DPP4 17 42 CC(C)[C@H](NC(=O)NCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147017824 EE On-Demand Mild CTSS 21 43 CC(C)[C@H](NC(=O)NCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147017824 EE On-Demand Mild XIAP 40 47 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2F)cs1 ZINC000147017831 FF On-Demand Anodyne MPL 53 36 CCCCO[C@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017887 EE On-Demand Anodyne CA2 48 43 CCCCO[C@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017887 EE On-Demand Anodyne CA1 38 48 CCCCO[C@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017887 EE On-Demand Anodyne CA4 38 43 CCCCO[C@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017887 EE On-Demand Anodyne CA14 28 41 CCCCO[C@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017887 EE On-Demand Anodyne CA9 25 44 CCCCO[C@H](C)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147017887 EE On-Demand Anodyne P96878_MYCTU 23 44 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017981 HH On-Demand Anodyne FBP1 21 41 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017981 HH On-Demand Anodyne EPHX2 25 45 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017981 HH On-Demand Anodyne TGM2 56 40 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017981 HH On-Demand Anodyne MDM2 67 36 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017981 HH On-Demand Anodyne F13A1 67 39 O=C(NCc1ccc(S(=O)(=O)N2CCCC2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147017981 HH On-Demand Anodyne NAMPT 86 47 O=C(NC[C@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2F)cs1 ZINC000147017991 FF On-Demand Anodyne MPL 53 36 COc1cc(OCC(=O)N(C)[C@@H](C)c2ccc(-n3cncn3)cc2)ccc1[N+](=O)[O-] ZINC000147018027 HF On-Demand Bother CYP26A1 42 33 CCCCO[C@@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018054 EE On-Demand Anodyne CA2 48 43 CCCCO[C@@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018054 EE On-Demand Anodyne CA1 38 48 CCCCO[C@@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018054 EE On-Demand Anodyne CA4 38 43 CCCCO[C@@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018054 EE On-Demand Anodyne CA14 28 41 CCCCO[C@@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018054 EE On-Demand Anodyne CA9 25 44 CCCCO[C@@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018054 EE On-Demand Anodyne P96878_MYCTU 23 44 CN1CCC(c2cccc(Nc3nc4c(-c5ccccc5N(C)S(C)(=O)=O)cccn4n3)c2)CC1 ZINC000147018112 JI Annotated Anodyne JAK3 15 71 CN1CCC(c2cccc(Nc3nc4c(-c5ccccc5N(C)S(C)(=O)=O)cccn4n3)c2)CC1 ZINC000147018112 JI Annotated Anodyne JAK2 34 71 CN1CCC(c2cccc(Nc3nc4c(-c5ccccc5N(C)S(C)(=O)=O)cccn4n3)c2)CC1 ZINC000147018112 JI Annotated Anodyne PTK2 42 33 COCCOc1ccc([C@H](C)NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1OC ZINC000147018161 HG On-Demand Anodyne ROCK2 26 41 COC(=O)c1ccc(F)c(S(=O)(=O)NC2CCN(C(=O)OC)CC2)c1 ZINC000147018195 FD On-Demand Anodyne ADRA1D 16 41 COC(=O)c1ccc(F)c(S(=O)(=O)NC2CCN(C(=O)OC)CC2)c1 ZINC000147018195 FD On-Demand Anodyne CCR8 91 44 COC(=O)c1ccc(F)c(S(=O)(=O)NC2CCN(C(=O)OC)CC2)c1 ZINC000147018195 FD On-Demand Anodyne SFRP1 111 43 COC(=O)c1ccc(F)c(S(=O)(=O)NC2CCN(C(=O)OC)CC2)c1 ZINC000147018195 FD On-Demand Anodyne WNT3 86 39 CCCCO[C@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018217 EE On-Demand Anodyne CA2 48 43 CCCCO[C@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018217 EE On-Demand Anodyne CA1 38 48 CCCCO[C@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018217 EE On-Demand Anodyne CA4 38 43 CCCCO[C@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018217 EE On-Demand Anodyne CA14 28 41 CCCCO[C@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018217 EE On-Demand Anodyne CA9 25 44 CCCCO[C@H](C)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018217 EE On-Demand Anodyne P96878_MYCTU 23 44 COc1ccc(Nc2ccc(Br)cc2)cc1 ZINC000147018223 CI For-Sale Anodyne EGFR 15 43 COc1ccc(Nc2ccc(Br)cc2)cc1 ZINC000147018223 CI For-Sale Anodyne GALR2 47 35 COc1ccc(Nc2ccc(Br)cc2)cc1 ZINC000147018223 CI For-Sale Anodyne AGPAT2 18 40 COc1ccc(Nc2ccc(Br)cc2)cc1 ZINC000147018223 CI For-Sale Anodyne AKR1C3 17 54 COc1ccc(Nc2ccc(Br)cc2)cc1 ZINC000147018223 CI For-Sale Anodyne AKR1C2 38 54 COCCOc1ccc([C@H](C)NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1OC ZINC000147018352 HG On-Demand Anodyne ROCK2 26 41 N#CC1CCN(C(=O)c2ccccc2C(=O)c2ccc(Cl)cc2)CC1 ZINC000147018402 FH On-Demand Mild L3MBTL3 55 36 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018446 FD On-Demand Anodyne CA2 56 47 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018446 FD On-Demand Anodyne CA1 35 40 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018446 FD On-Demand Anodyne CA7 27 45 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018446 FD On-Demand Anodyne CA4 37 43 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018446 FD On-Demand Anodyne CA14 23 45 COCCOc1ccc([C@@H](C)NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1OC ZINC000147018480 HG On-Demand Anodyne ROCK2 26 41 COC(=O)N1CCC(NS(=O)(=O)c2c(Cl)cccc2[N+](=O)[O-])CC1 ZINC000147018536 GD On-Demand Bother CCR8 82 42 COC(=O)N1CCC(NS(=O)(=O)c2c(Cl)cccc2[N+](=O)[O-])CC1 ZINC000147018536 GD On-Demand Bother SFRP1 108 40 COC(=O)N1CCC(NS(=O)(=O)c2c(Cl)cccc2[N+](=O)[O-])CC1 ZINC000147018536 GD On-Demand Bother WNT3 80 40 O=C(NCCF)NC[C@H]1CCc2ccccc21 ZINC000147018582 BD On-Demand Anodyne NQO2 34 41 O=C(NCCF)NC[C@H]1CCc2ccccc21 ZINC000147018582 BD On-Demand Anodyne MTNR1A 17 48 O=C(NCCF)NC[C@H]1CCc2ccccc21 ZINC000147018582 BD On-Demand Anodyne MTNR1B 20 48 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive PPIA 34 51 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive ANPEP 36 50 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive PAPA1_CARPA 33 40 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive SLC15A1 48 34 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive ROCK2 15 46 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive SLC1A6 54 35 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive SLC6A12 43 35 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive SLC1A7 54 35 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive CPA3 52 32 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive POL 0 44 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive AMP1_PLAFQ 55 44 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive E1 0 40 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive ACAT 0 51 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive NAMPT 37 42 CNNC(=O)NCc1ccccc1 ZINC000147018585 AC For-Sale Reactive PDS 58 41 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018594 FD On-Demand Anodyne CA2 56 47 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018594 FD On-Demand Anodyne CA1 35 40 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018594 FD On-Demand Anodyne CA7 27 45 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018594 FD On-Demand Anodyne CA4 37 43 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018594 FD On-Demand Anodyne CA14 23 45 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(-c3cccc(Cl)c3)cs2)c1 ZINC000147018677 GJ On-Demand Bother CSNK1D 16 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(-c3cccc(Cl)c3)cs2)c1 ZINC000147018677 GJ On-Demand Bother ROCK1 22 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(-c3cccc(Cl)c3)cs2)c1 ZINC000147018677 GJ On-Demand Bother GCK 17 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(-c3cccc(Cl)c3)cs2)c1 ZINC000147018677 GJ On-Demand Bother TAAR1 22 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(-c3cccc(Cl)c3)cs2)c1 ZINC000147018677 GJ On-Demand Bother USP7 26 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(-c3cccc(Cl)c3)cs2)c1 ZINC000147018677 GJ On-Demand Bother USP47 33 40 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne CA2 78 53 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne CA6 22 53 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne CA1 61 53 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne CA7 60 36 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne DPP4 19 46 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne CA13 34 40 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne CA4 63 40 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne CA14 45 39 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne SLC9A1 33 54 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne CA12 53 39 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne CA9 45 40 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne NCE103 27 53 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne P96878_MYCTU 45 39 NS(=O)(=O)c1ccc(C(=O)N2CCC(F)CC2)cc1 ZINC000147018686 CC For-Sale Anodyne L3MBTL3 88 49 O=C(NCCF)NC[C@@H]1CCc2ccccc21 ZINC000147018742 BD On-Demand Anodyne NQO2 34 41 O=C(NCCF)NC[C@@H]1CCc2ccccc21 ZINC000147018742 BD On-Demand Anodyne MTNR1A 17 48 O=C(NCCF)NC[C@@H]1CCc2ccccc21 ZINC000147018742 BD On-Demand Anodyne MTNR1B 20 48 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018744 FD On-Demand Anodyne CA2 56 47 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018744 FD On-Demand Anodyne CA1 35 40 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018744 FD On-Demand Anodyne CA7 27 45 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018744 FD On-Demand Anodyne CA4 37 43 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018744 FD On-Demand Anodyne CA14 23 45 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018876 FD On-Demand Anodyne CA2 56 47 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018876 FD On-Demand Anodyne CA1 35 40 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018876 FD On-Demand Anodyne CA7 27 45 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018876 FD On-Demand Anodyne CA4 37 43 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147018876 FD On-Demand Anodyne CA14 23 45 COc1ccc(N/C=C2\C(=O)NC(=O)c3ccccc32)cc1O ZINC000147018927 DE On-Demand Anodyne HDAC2 18 40 COc1ccc(N/C=C2\C(=O)NC(=O)c3ccccc32)cc1O ZINC000147018927 DE On-Demand Anodyne CDK1 15 53 COc1ccc(N/C=C2\C(=O)NC(=O)c3ccccc32)cc1O ZINC000147018927 DE On-Demand Anodyne CDK4 100 73 Cc1ccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)cn1 ZINC000147018962 EH On-Demand Anodyne NAMPT 20 41 CCOc1ccc([C@H](NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c2ccccc2)cc1 ZINC000147019057 HJ On-Demand Bother AKR1C2 33 44 CCOC(=O)COc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147019075 HG On-Demand Anodyne NOS2 48 37 CCOC(=O)COc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147019075 HG On-Demand Anodyne ROCK2 23 42 CCOC(=O)COc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147019075 HG On-Demand Anodyne NAMPT 31 40 Cc1ccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)cn1 ZINC000147019127 EH On-Demand Anodyne NAMPT 20 41 CCOc1ccc([C@@H](NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c2ccccc2)cc1 ZINC000147019250 HJ On-Demand Bother AKR1C2 33 44 CCCCc1ccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@@H]32)cc1 ZINC000147019323 EF On-Demand Anodyne CFTR 41 37 Cc1ccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)cn1 ZINC000147019350 EH On-Demand Anodyne NAMPT 20 41 CCOC(=O)COc1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147019366 HH On-Demand Anodyne COLA 34 40 CCOC(=O)COc1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147019366 HH On-Demand Anodyne CPT1A 33 40 COCCCCN(Cc1ccccc1)S(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-] ZINC000147019428 HH On-Demand Bother COLA 80 35 COCCCCN(Cc1ccccc1)S(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-] ZINC000147019428 HH On-Demand Bother MMP9 18 42 CC(C)(C)c1ccc(CCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147019450 HG On-Demand Bother CA2 22 58 CC(C)(C)c1ccc(CCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147019450 HG On-Demand Bother CA1 21 47 CC(C)(C)c1ccc(CCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147019450 HG On-Demand Bother TRPV1 24 44 CC(C)(C)c1ccc(CCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147019450 HG On-Demand Bother CA9 15 41 CC(C)(C)c1ccc(CCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147019450 HG On-Demand Bother CYNT 29 58 CCCCc1ccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@@H]32)cc1 ZINC000147019492 EF On-Demand Anodyne CFTR 41 37 Cc1ccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)cn1 ZINC000147019527 EH On-Demand Anodyne NAMPT 20 41 CCOC(=O)COc1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147019592 HH On-Demand Anodyne COLA 34 40 CCOC(=O)COc1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147019592 HH On-Demand Anodyne CPT1A 33 40 CCCCc1ccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@H]32)cc1 ZINC000147019677 EF On-Demand Anodyne CFTR 41 37 CCS(=O)(=O)Nc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1OC ZINC000147019715 HD On-Demand Anodyne ENPP1 58 30 CCOC(=O)COc1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147019803 HH On-Demand Anodyne COLA 34 40 CCOC(=O)COc1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147019803 HH On-Demand Anodyne CPT1A 33 40 CCCCc1ccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@H]32)cc1 ZINC000147019866 EF On-Demand Anodyne CFTR 41 37 COc1ccccc1-c1csc(NC(=O)c2ccn(-c3cccc(F)c3)n2)n1 ZINC000147019894 GI On-Demand Anodyne MPL 57 38 CCOC(=O)COc1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147019971 HH On-Demand Anodyne COLA 34 40 CCOC(=O)COc1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147019971 HH On-Demand Anodyne CPT1A 33 40 CCOC(=O)c1cc2cc(NC(=O)c3ccc(-c4ccccc4)o3)ccc2o1 ZINC000147020180 GK For-Sale Anodyne S1PR4 43 50 CCOC(=O)c1cc2cc(NC(=O)c3ccc(-c4ccccc4)o3)ccc2o1 ZINC000147020180 GK For-Sale Anodyne SCN10A 30 52 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@@H](C)C[C@@H](C)C2)c1 ZINC000147020279 HH On-Demand Bother KCNMA1 25 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@@H](C)C[C@@H](C)C2)c1 ZINC000147020279 HH On-Demand Bother TAAR1 24 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@@H](C)C[C@@H](C)C2)c1 ZINC000147020279 HH On-Demand Bother AKR1C3 17 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@@H](C)C[C@@H](C)C2)c1 ZINC000147020279 HH On-Demand Bother AKR1C2 41 48 CCNC(=O)COc1cccc(NC(=O)N[C@@H](C)COCC)c1 ZINC000147020282 DD On-Demand Anodyne EPHX2 15 42 CCNC(=O)COc1cccc(NC(=O)N[C@@H](C)COCC)c1 ZINC000147020282 DD On-Demand Anodyne PDS 43 33 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc2c(c1)CCC(=O)N2 ZINC000147020326 FI On-Demand Anodyne PKM 29 43 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc2c(c1)CCC(=O)N2 ZINC000147020326 FI On-Demand Anodyne MDM2 64 33 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@@H](C)C[C@H](C)C2)c1 ZINC000147020470 HH On-Demand Bother KCNMA1 25 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@@H](C)C[C@H](C)C2)c1 ZINC000147020470 HH On-Demand Bother TAAR1 24 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@@H](C)C[C@H](C)C2)c1 ZINC000147020470 HH On-Demand Bother AKR1C3 17 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@@H](C)C[C@H](C)C2)c1 ZINC000147020470 HH On-Demand Bother AKR1C2 41 48 COc1cnc(-c2ccn3c(-c4cccc(NC(=O)NCC(F)(F)F)c4)cnc3c2)cn1 ZINC000147020521 II Annotated Anodyne RIPK1 45 33 COC(=O)c1cccc(/C=C(/C)[N+](=O)[O-])c1 ZINC000147020581 BE For-Sale Bother TLR4 32 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@H](C)C[C@@H](C)C2)c1 ZINC000147020653 HH On-Demand Bother KCNMA1 25 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@H](C)C[C@@H](C)C2)c1 ZINC000147020653 HH On-Demand Bother TAAR1 24 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@H](C)C[C@@H](C)C2)c1 ZINC000147020653 HH On-Demand Bother AKR1C3 17 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2C(=O)N2C[C@H](C)C[C@@H](C)C2)c1 ZINC000147020653 HH On-Demand Bother AKR1C2 41 48 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccccc2OCCc2ccccc2)C1 ZINC000147020656 HF On-Demand Anodyne CCR3 37 48 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccccc2OCCc2ccccc2)C1 ZINC000147020656 HF On-Demand Anodyne BIRC2 54 38 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc2c(c1)CCC(=O)N2 ZINC000147020704 FI On-Demand Anodyne PKM 29 43 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc2c(c1)CCC(=O)N2 ZINC000147020704 FI On-Demand Anodyne MDM2 64 33 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147020829 FE On-Demand Anodyne P2RY1 56 40 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147020829 FE On-Demand Anodyne CTSS 24 40 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147020829 FE On-Demand Anodyne EPHX2 62 46 CCN(CC)CC(=O)NCc1ccccc1Cn1cncn1 ZINC000147020838 DD On-Demand Anodyne HIS3 61 38 CCOc1ccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1OC ZINC000147020865 HE On-Demand Bother MAPK9 22 42 CCOc1ccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1OC ZINC000147020865 HE On-Demand Bother MAPK8 19 44 CCOc1ccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1OC ZINC000147020865 HE On-Demand Bother MT-ND1 16 42 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccccc2OCCc2ccccc2)C1 ZINC000147020876 HF On-Demand Anodyne CCR3 37 48 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccccc2OCCc2ccccc2)C1 ZINC000147020876 HF On-Demand Anodyne BIRC2 54 38 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147021010 FE On-Demand Anodyne P2RY1 56 40 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147021010 FE On-Demand Anodyne CTSS 24 40 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147021010 FE On-Demand Anodyne EPHX2 62 46 CCCNC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147021064 GE On-Demand Anodyne SLC6A9 23 46 CCCNC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147021064 GE On-Demand Anodyne ENV 40 32 CC[C@H]1CN(C(=O)COc2ccc(C(N)=O)cc2)CCO1 ZINC000147021181 CC On-Demand Anodyne COLA 87 47 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147021210 FE On-Demand Anodyne P2RY1 56 40 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147021210 FE On-Demand Anodyne CTSS 24 40 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147021210 FE On-Demand Anodyne EPHX2 62 46 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cc(OC)ccc1OC ZINC000147021235 FF On-Demand Anodyne P2RY12 126 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cc(OC)ccc1OC ZINC000147021235 FF On-Demand Anodyne TRHR 46 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cc(OC)ccc1OC ZINC000147021235 FF On-Demand Anodyne TRY1_BOVIN 46 39 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cc(OC)ccc1OC ZINC000147021235 FF On-Demand Anodyne NTSR1 63 32 CCCNC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147021267 GE On-Demand Anodyne SLC6A9 23 46 CCCNC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147021267 GE On-Demand Anodyne ENV 40 32 CCNC(=O)COc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147021389 HF On-Demand Anodyne NOS2 86 35 CCNC(=O)COc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147021389 HF On-Demand Anodyne ROCK2 26 42 CCNC(=O)COc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147021389 HF On-Demand Anodyne NAMPT 33 41 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147021405 FE On-Demand Anodyne P2RY1 56 40 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147021405 FE On-Demand Anodyne CTSS 24 40 O=C(Nc1ccc(OC(F)(F)F)cc1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147021405 FE On-Demand Anodyne EPHX2 62 46 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cc(OC)ccc1OC ZINC000147021460 FF On-Demand Anodyne P2RY12 126 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cc(OC)ccc1OC ZINC000147021460 FF On-Demand Anodyne TRHR 46 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cc(OC)ccc1OC ZINC000147021460 FF On-Demand Anodyne TRY1_BOVIN 46 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cc(OC)ccc1OC ZINC000147021460 FF On-Demand Anodyne NTSR1 63 32 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccnc1N1CCOCC1 ZINC000147021465 EC On-Demand Anodyne PIK3CA 42 36 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccnc1N1CCOCC1 ZINC000147021465 EC On-Demand Anodyne MTOR 50 34 CCn1c2ccccc2c2cc(NC(=O)C(=O)N3CCO[C@H]4CCC[C@@H]43)ccc21 ZINC000147021585 GH On-Demand Anodyne NPY5R 15 52 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cc(OC)ccc1OC ZINC000147021648 FF On-Demand Anodyne P2RY12 126 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cc(OC)ccc1OC ZINC000147021648 FF On-Demand Anodyne TRHR 46 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cc(OC)ccc1OC ZINC000147021648 FF On-Demand Anodyne TRY1_BOVIN 46 39 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cc(OC)ccc1OC ZINC000147021648 FF On-Demand Anodyne NTSR1 63 32 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccnc1N1CCOCC1 ZINC000147021672 EC On-Demand Anodyne PIK3CA 42 36 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccnc1N1CCOCC1 ZINC000147021672 EC On-Demand Anodyne MTOR 50 34 CCCc1nc(C)c2c(C)nc3scnc3n12 ZINC000147021744 BF For-Sale Anodyne PDE10A 15 40 CCn1c2ccccc2c2cc(NC(=O)C(=O)N3CCO[C@@H]4CCC[C@@H]43)ccc21 ZINC000147021757 GH On-Demand Anodyne NPY5R 15 52 CC(C)(C)C[C@H]1N[C@@H](C(=O)NCC[C@H]2CC[C@H](N)C2)[C@H](c2cccc(Cl)c2F)[C@@]12C(=O)Nc1cc(Cl)c(F)cc12 ZINC000147021806 KK Annotated Anodyne MDM2 98 64 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H](C)c1ccc3c(c1)CCC(=O)N3)C2 ZINC000147021819 GG On-Demand Anodyne GRIN2B 15 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cc(OC)ccc1OC ZINC000147021854 FF On-Demand Anodyne P2RY12 126 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cc(OC)ccc1OC ZINC000147021854 FF On-Demand Anodyne TRHR 46 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cc(OC)ccc1OC ZINC000147021854 FF On-Demand Anodyne TRY1_BOVIN 46 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cc(OC)ccc1OC ZINC000147021854 FF On-Demand Anodyne NTSR1 63 32 CCn1c2ccccc2c2cc(NC(=O)C(=O)N3CCO[C@H]4CCC[C@H]43)ccc21 ZINC000147021948 GH On-Demand Anodyne NPY5R 15 52 COc1ccccc1-c1cccn2nc(Nc3cccc(N4CCN(C)CC4)c3)nc12 ZINC000147022028 HH Annotated Anodyne LCK 18 40 COc1ccccc1-c1cccn2nc(Nc3cccc(N4CCN(C)CC4)c3)nc12 ZINC000147022028 HH Annotated Anodyne JAK3 18 72 COc1ccccc1-c1cccn2nc(Nc3cccc(N4CCN(C)CC4)c3)nc12 ZINC000147022028 HH Annotated Anodyne JAK2 54 60 COc1ccccc1-c1cccn2nc(Nc3cccc(N4CCN(C)CC4)c3)nc12 ZINC000147022028 HH Annotated Anodyne PTK2 48 36 COc1ccccc1-c1cccn2nc(Nc3cccc(N4CCN(C)CC4)c3)nc12 ZINC000147022028 HH Annotated Anodyne PAK1 48 35 COc1ccccc1-c1cccn2nc(Nc3cccc(N4CCN(C)CC4)c3)nc12 ZINC000147022028 HH Annotated Anodyne WEE1 15 41 COc1ccccc1-c1cccn2nc(Nc3cccc(N4CCN(C)CC4)c3)nc12 ZINC000147022028 HH Annotated Anodyne ALK 16 45 COc1ccccc1-c1cccn2nc(Nc3cccc(N4CCN(C)CC4)c3)nc12 ZINC000147022028 HH Annotated Anodyne MAPK7 46 39 COc1ccc(C=O)cc1OC1CCC1 ZINC000147022032 BE For-Sale Anodyne PDE4A 51 50 COc1ccc(C=O)cc1OC1CCC1 ZINC000147022032 BE For-Sale Anodyne CYP1B1 22 41 COc1ccc(C=O)cc1OC1CCC1 ZINC000147022032 BE For-Sale Anodyne PDE4B 34 47 COc1ccc(C=O)cc1OC1CCC1 ZINC000147022032 BE For-Sale Anodyne PDE4D 34 42 COc1ccc(C=O)cc1OC1CCC1 ZINC000147022032 BE For-Sale Anodyne CYP1A1 24 41 COc1ccc(C=O)cc1OC1CCC1 ZINC000147022032 BE For-Sale Anodyne PDE4C 29 49 COc1ccc(C=O)cc1OC1CCC1 ZINC000147022032 BE For-Sale Anodyne TUBB1 52 34 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H](C)c1ccc3c(c1)CCC(=O)N3)C2 ZINC000147022035 GG On-Demand Anodyne GRIN2B 15 44 CCOC(=O)N1CCN(S(=O)(=O)NCc2cccc(C#N)c2)CC1 ZINC000147022052 FC On-Demand Mild P2RY12 54 37 CCOC(=O)N1CCN(S(=O)(=O)NCc2cccc(C#N)c2)CC1 ZINC000147022052 FC On-Demand Mild TGM2 29 40 CCOC(=O)N1CCN(S(=O)(=O)NCc2cccc(C#N)c2)CC1 ZINC000147022052 FC On-Demand Mild F13A1 45 40 CCn1c2ccccc2c2cc(NC(=O)C(=O)N3CCO[C@@H]4CCC[C@H]43)ccc21 ZINC000147022167 GH On-Demand Anodyne NPY5R 15 52 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H](C)c1ccc3c(c1)CCC(=O)N3)C2 ZINC000147022241 GG On-Demand Anodyne GRIN2B 15 44 Cc1ccc(/C=C\c2ccccc2/C=C\c2ccc(C)cc2)cc1 ZINC000147022269 DK For-Sale Anodyne CYP1B1 28 45 Cc1ccc(/C=C\c2ccccc2/C=C\c2ccc(C)cc2)cc1 ZINC000147022269 DK For-Sale Anodyne CHAT 51 40 Cc1ccc(/C=C\c2ccccc2/C=C\c2ccc(C)cc2)cc1 ZINC000147022269 DK For-Sale Anodyne CYP1A1 24 45 CC(C)(C)OC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCc1ccc(O)cc1 ZINC000147022315 GG On-Demand Anodyne ACE 23 43 CC(C)(C)OC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCc1ccc(O)cc1 ZINC000147022315 GG On-Demand Anodyne LHCGR 25 41 CC(C)(C)OC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCc1ccc(O)cc1 ZINC000147022315 GG On-Demand Anodyne OPRM1 37 45 CC(C)(C)OC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCc1ccc(O)cc1 ZINC000147022315 GG On-Demand Anodyne OPRD1 36 45 CC(C)(C)OC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCc1ccc(O)cc1 ZINC000147022315 GG On-Demand Anodyne MME 43 43 CC(C)(C)OC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCc1ccc(O)cc1 ZINC000147022315 GG On-Demand Anodyne PAPA1_CARPA 50 50 CC(C)(C)OC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCc1ccc(O)cc1 ZINC000147022315 GG On-Demand Anodyne CTSL 25 50 CC(C)(C)OC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCc1ccc(O)cc1 ZINC000147022315 GG On-Demand Anodyne GRIA1 70 52 CC(C)(C)OC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCc1ccc(O)cc1 ZINC000147022315 GG On-Demand Anodyne YARS 63 34 CC(C)(C)OC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCc1ccc(O)cc1 ZINC000147022315 GG On-Demand Anodyne ACE2 47 40 CC(C)(C)OC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCc1ccc(O)cc1 ZINC000147022315 GG On-Demand Anodyne FPR1 44 36 Cc1cc(CNC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)no1 ZINC000147022389 FE On-Demand Anodyne HRH2 41 42 Cc1cc(CNC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)no1 ZINC000147022389 FE On-Demand Anodyne CPT1A 101 44 Cc1cc(CNC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)no1 ZINC000147022389 FE On-Demand Anodyne CCKBR 25 41 Cc1cc(CNC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)no1 ZINC000147022389 FE On-Demand Anodyne EPHX2 33 43 C[C@H](NC(=O)c1ccc2c(c1)COC2)c1ccc2c(c1)CCC(=O)N2 ZINC000147022455 EG On-Demand Anodyne GRIN2B 15 40 C[C@H](NC(=O)c1ccc2c(c1)COC2)c1ccc2c(c1)CCC(=O)N2 ZINC000147022455 EG On-Demand Anodyne HDAC9 18 43 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cccc(C#N)c3)cc2)cc1 ZINC000147022458 HH On-Demand Mild CA1 17 41 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cccc(C#N)c3)cc2)cc1 ZINC000147022458 HH On-Demand Mild MMP13 24 50 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cccc(C#N)c3)cc2)cc1 ZINC000147022458 HH On-Demand Mild MMP2 19 40 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cccc(C#N)c3)cc2)cc1 ZINC000147022458 HH On-Demand Mild ADAMTS4 19 50 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cccc(C#N)c3)cc2)cc1 ZINC000147022458 HH On-Demand Mild IDO1 38 42 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cccc(C#N)c3)cc2)cc1 ZINC000147022458 HH On-Demand Mild MTCA1 27 41 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cccc(C#N)c3)cc2)cc1 ZINC000147022458 HH On-Demand Mild P96878_MYCTU 36 41 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cccc(C#N)c3)cc2)cc1 ZINC000147022458 HH On-Demand Mild RORC 24 40 Cc1ccc(/C=C\c2ccccc2/C=C/c2ccc(C)cc2)cc1 ZINC000147022469 DK For-Sale Anodyne CYP1B1 28 45 Cc1ccc(/C=C\c2ccccc2/C=C/c2ccc(C)cc2)cc1 ZINC000147022469 DK For-Sale Anodyne CHAT 51 40 Cc1ccc(/C=C\c2ccccc2/C=C/c2ccc(C)cc2)cc1 ZINC000147022469 DK For-Sale Anodyne CYP1A1 24 45 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OCC)cc1 ZINC000147022498 EF On-Demand Anodyne P2RY12 66 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OCC)cc1 ZINC000147022498 EF On-Demand Anodyne TRHR 46 32 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OCC)cc1 ZINC000147022498 EF On-Demand Anodyne TRY1_BOVIN 56 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OCC)cc1 ZINC000147022498 EF On-Demand Anodyne NTSR1 58 32 COC(=O)c1cc2c(CN3CCC[C@H](C(N)=O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147022501 HF For-Sale Anodyne CCR3 61 33 COC(=O)c1cc2c(CN3CCC[C@H](C(N)=O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147022501 HF For-Sale Anodyne F2R 43 37 COC(=O)c1cc2c(CN3CCC[C@H](C(N)=O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147022501 HF For-Sale Anodyne MLNR 44 35 COC(=O)c1cc2c(CN3CCC[C@H](C(N)=O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147022501 HF For-Sale Anodyne MBTPS1 20 40 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147022592 GG On-Demand Anodyne HRH2 46 40 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147022592 GG On-Demand Anodyne CCKAR 40 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147022592 GG On-Demand Anodyne CCR3 27 43 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147022592 GG On-Demand Anodyne CPT1A 108 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147022592 GG On-Demand Anodyne CPT2 47 36 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147022592 GG On-Demand Anodyne CCKBR 54 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147022592 GG On-Demand Anodyne EPHX2 65 48 Cc1ccc(/C=C/c2ccccc2/C=C/c2ccc(C)cc2)cc1 ZINC000147022642 DK For-Sale Anodyne CYP1B1 28 45 Cc1ccc(/C=C/c2ccccc2/C=C/c2ccc(C)cc2)cc1 ZINC000147022642 DK For-Sale Anodyne CHAT 51 40 Cc1ccc(/C=C/c2ccccc2/C=C/c2ccc(C)cc2)cc1 ZINC000147022642 DK For-Sale Anodyne CYP1A1 24 45 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(OC)c(F)c1)C2 ZINC000147022671 EG On-Demand Anodyne MTNR1A 18 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(OC)c(F)c1)C2 ZINC000147022671 EG On-Demand Anodyne ROCK2 40 56 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OCC)cc1 ZINC000147022682 EF On-Demand Anodyne P2RY12 66 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OCC)cc1 ZINC000147022682 EF On-Demand Anodyne TRHR 46 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OCC)cc1 ZINC000147022682 EF On-Demand Anodyne TRY1_BOVIN 56 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OCC)cc1 ZINC000147022682 EF On-Demand Anodyne NTSR1 58 32 COC(=O)c1cc2c(CN3CCC[C@@H](C(N)=O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147022704 HF For-Sale Anodyne CCR3 61 33 COC(=O)c1cc2c(CN3CCC[C@@H](C(N)=O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147022704 HF For-Sale Anodyne F2R 43 37 COC(=O)c1cc2c(CN3CCC[C@@H](C(N)=O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147022704 HF For-Sale Anodyne MLNR 44 35 COC(=O)c1cc2c(CN3CCC[C@@H](C(N)=O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147022704 HF For-Sale Anodyne MBTPS1 20 40 CCOC(=O)NCC(=O)Nc1cccc(-c2ccnc(C)n2)c1 ZINC000147022706 DE On-Demand Anodyne ABL1 18 43 CCN(CC)C(=O)c1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147022726 HF On-Demand Anodyne OPRM1 15 40 CCN(CC)C(=O)c1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147022726 HF On-Demand Anodyne OPRD1 31 43 CCN(CC)C(=O)c1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147022726 HF On-Demand Anodyne LIMK2 53 45 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2cccc(NC(=O)c3ccccc3)c2)c1 ZINC000147022753 HI On-Demand Bother TAAR1 41 52 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2cccc(NC(=O)c3ccccc3)c2)c1 ZINC000147022753 HI On-Demand Bother AKR1C3 32 48 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2cccc(NC(=O)c3ccccc3)c2)c1 ZINC000147022753 HI On-Demand Bother AKR1C2 51 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2cccc(NC(=O)c3ccccc3)c2)c1 ZINC000147022753 HI On-Demand Bother KCNK3 121 51 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2cccc(NC(=O)c3ccccc3)c2)c1 ZINC000147022753 HI On-Demand Bother KCNK9 80 38 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147022787 GG On-Demand Anodyne HRH2 46 40 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147022787 GG On-Demand Anodyne CCKAR 40 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147022787 GG On-Demand Anodyne CCR3 27 43 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147022787 GG On-Demand Anodyne CPT1A 108 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147022787 GG On-Demand Anodyne CPT2 47 36 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147022787 GG On-Demand Anodyne CCKBR 54 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147022787 GG On-Demand Anodyne EPHX2 65 48 C[C@H](Nc1ccc(O)cc1O)C(=O)O ZINC000147022805 AC For-Sale Anodyne KYNU 44 31 Cc1oc(-c2ccccc2)nc1CC(=O)N1CCC(C#N)CC1 ZINC000147022851 DF On-Demand Anodyne PPARG 62 41 Cc1oc(-c2ccccc2)nc1CC(=O)N1CCC(C#N)CC1 ZINC000147022851 DF On-Demand Anodyne PPARA 72 42 Cc1oc(-c2ccccc2)nc1CC(=O)N1CCC(C#N)CC1 ZINC000147022851 DF On-Demand Anodyne PPARD 17 41 Cc1oc(-c2ccccc2)nc1CC(=O)N1CCC(C#N)CC1 ZINC000147022851 DF On-Demand Anodyne PDE8B 68 40 CN1CCN(C2CCN(c3ccc(Nc4nc5c(-c6ccc(S(C)(=O)=O)cc6)cccn5n4)cc3)CC2)CC1 ZINC000147022855 KH Annotated Anodyne JAK3 25 85 CN1CCN(C2CCN(c3ccc(Nc4nc5c(-c6ccc(S(C)(=O)=O)cc6)cccn5n4)cc3)CC2)CC1 ZINC000147022855 KH Annotated Anodyne JAK2 46 85 CN1CCN(C2CCN(c3ccc(Nc4nc5c(-c6ccc(S(C)(=O)=O)cc6)cccn5n4)cc3)CC2)CC1 ZINC000147022855 KH Annotated Anodyne CDK4 17 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OCC)cc1 ZINC000147022867 EF On-Demand Anodyne P2RY12 66 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OCC)cc1 ZINC000147022867 EF On-Demand Anodyne TRHR 46 32 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OCC)cc1 ZINC000147022867 EF On-Demand Anodyne TRY1_BOVIN 56 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OCC)cc1 ZINC000147022867 EF On-Demand Anodyne NTSR1 58 32 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(F)cc1Br)C2 ZINC000147022898 GH On-Demand Anodyne ROCK2 37 52 O=C(C[C@]1(C(=O)O)CCSC1)Nc1cccc(N2CCOCC2)c1 ZINC000147022904 FE On-Demand Anodyne EPHX2 19 43 Cc1nccc(-c2cccc(NC(=O)CCNS(C)(=O)=O)c2)n1 ZINC000147022921 ED On-Demand Anodyne ABL1 16 45 Cc1nccc(-c2cccc(NC(=O)CCNS(C)(=O)=O)c2)n1 ZINC000147022921 ED On-Demand Anodyne MTNN 18 41 Cc1nccc(-c2cccc(NC(=O)CCNS(C)(=O)=O)c2)n1 ZINC000147022921 ED On-Demand Anodyne SMG1 60 34 CCN(CC)C(=O)c1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147022925 HF On-Demand Anodyne OPRM1 15 40 CCN(CC)C(=O)c1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147022925 HF On-Demand Anodyne OPRD1 31 43 CCN(CC)C(=O)c1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147022925 HF On-Demand Anodyne LIMK2 53 45 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2cccc(NC(=O)c3ccccc3)c2)c1 ZINC000147022935 HI On-Demand Bother TAAR1 41 52 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2cccc(NC(=O)c3ccccc3)c2)c1 ZINC000147022935 HI On-Demand Bother AKR1C3 32 48 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2cccc(NC(=O)c3ccccc3)c2)c1 ZINC000147022935 HI On-Demand Bother AKR1C2 51 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2cccc(NC(=O)c3ccccc3)c2)c1 ZINC000147022935 HI On-Demand Bother KCNK3 121 51 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2cccc(NC(=O)c3ccccc3)c2)c1 ZINC000147022935 HI On-Demand Bother KCNK9 80 38 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147022973 GG On-Demand Anodyne HRH2 46 40 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147022973 GG On-Demand Anodyne CCKAR 40 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147022973 GG On-Demand Anodyne CCR3 27 43 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147022973 GG On-Demand Anodyne CPT1A 108 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147022973 GG On-Demand Anodyne CPT2 47 36 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147022973 GG On-Demand Anodyne CCKBR 54 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147022973 GG On-Demand Anodyne EPHX2 65 48 COC(=O)[C@H](NC(=O)OC(C)(C)C)c1ccccc1C ZINC000147023017 CF On-Demand Anodyne PAPA1_CARPA 53 42 COC(=O)[C@H](NC(=O)OC(C)(C)C)c1ccccc1C ZINC000147023017 CF On-Demand Anodyne CTSK 17 47 C[C@@H](Nc1ccc(O)cc1O)C(=O)O ZINC000147023027 AC For-Sale Anodyne KYNU 44 31 NC(=O)c1ccc(OCC(=O)NCc2ccc(N3CCCC3)nc2)cc1 ZINC000147023030 FD On-Demand Anodyne SMO 15 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OCC)cc1 ZINC000147023059 EF On-Demand Anodyne P2RY12 66 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OCC)cc1 ZINC000147023059 EF On-Demand Anodyne TRHR 46 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OCC)cc1 ZINC000147023059 EF On-Demand Anodyne TRY1_BOVIN 56 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OCC)cc1 ZINC000147023059 EF On-Demand Anodyne NTSR1 58 32 COc1cccc(Oc2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2)c1 ZINC000147023120 GI On-Demand Anodyne PDGFRB 29 41 COc1cccc(Oc2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2)c1 ZINC000147023120 GI On-Demand Anodyne LTA4H 36 41 COc1cccc(Oc2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2)c1 ZINC000147023120 GI On-Demand Anodyne RAF1 23 47 COc1cccc(Oc2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2)c1 ZINC000147023120 GI On-Demand Anodyne MTNR1A 36 61 COc1cccc(Oc2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2)c1 ZINC000147023120 GI On-Demand Anodyne MTNR1B 40 61 COc1cccc(Oc2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2)c1 ZINC000147023120 GI On-Demand Anodyne NPY5R 20 40 COc1cccc(Oc2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2)c1 ZINC000147023120 GI On-Demand Anodyne FLT4 21 41 COc1cccc(Oc2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2)c1 ZINC000147023120 GI On-Demand Anodyne MMP10 20 40 COc1cccc(Oc2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2)c1 ZINC000147023120 GI On-Demand Anodyne PFKFB3 44 32 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147023150 GG On-Demand Anodyne HRH2 46 40 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147023150 GG On-Demand Anodyne CCKAR 40 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147023150 GG On-Demand Anodyne CCR3 27 43 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147023150 GG On-Demand Anodyne CPT1A 108 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147023150 GG On-Demand Anodyne CPT2 47 36 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147023150 GG On-Demand Anodyne CCKBR 54 45 O=C(Nc1cccc(OCC(=O)N2CCCC2)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147023150 GG On-Demand Anodyne EPHX2 65 48 C=CCN(C)S(=O)(=O)c1ccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@@H]32)cc1 ZINC000147023152 HD On-Demand Mild F13A1 53 35 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccccc2COCc2ccccc2)c1 ZINC000147023155 HI On-Demand Bother TAAR1 19 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccccc2COCc2ccccc2)c1 ZINC000147023155 HI On-Demand Bother AKR1C2 29 43 COC(=O)c1cc(C(=O)O)ccc1Br ZINC000147023226 CD For-Sale Anodyne CA14 0 50 COC(=O)c1cc(C(=O)O)ccc1Br ZINC000147023226 CD For-Sale Anodyne TPMT 0 41 COC(=O)c1cc(C(=O)O)ccc1Br ZINC000147023226 CD For-Sale Anodyne AKR1C3 49 38 COC(=O)c1cc(C(=O)O)ccc1Br ZINC000147023226 CD For-Sale Anodyne AKR1C2 43 38 COC(=O)c1cc(C(=O)O)ccc1Br ZINC000147023226 CD For-Sale Anodyne KDM3A 0 47 CCO[C@@H]1CCCN(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)C1 ZINC000147023346 GF On-Demand Anodyne CCR3 21 46 CCO[C@@H]1CCCN(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)C1 ZINC000147023346 GF On-Demand Anodyne CPT1A 97 45 CCO[C@@H]1CCCN(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)C1 ZINC000147023346 GF On-Demand Anodyne CPT2 43 39 CCO[C@@H]1CCCN(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)C1 ZINC000147023346 GF On-Demand Anodyne EPHX2 36 41 CCO[C@@H]1CCCN(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)C1 ZINC000147023346 GF On-Demand Anodyne TAAR1 23 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(OC(C)C)cc1)C2 ZINC000147023351 EH On-Demand Anodyne MTNR1A 23 45 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(OC(C)C)cc1)C2 ZINC000147023351 EH On-Demand Anodyne MTNR1B 23 45 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(OC(C)C)cc1)C2 ZINC000147023351 EH On-Demand Anodyne ROCK2 36 56 C=CCN(C)S(=O)(=O)c1ccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@@H]32)cc1 ZINC000147023369 HD On-Demand Mild F13A1 53 35 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(COCc3ccccc3)c2)c1 ZINC000147023380 HI On-Demand Bother MMP13 29 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(COCc3ccccc3)c2)c1 ZINC000147023380 HI On-Demand Bother TAAR1 20 45 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(COCc3ccccc3)c2)c1 ZINC000147023380 HI On-Demand Bother AKR1C3 16 44 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(COCc3ccccc3)c2)c1 ZINC000147023380 HI On-Demand Bother AKR1C2 34 44 CC(=O)c1ccc(S(=O)(=O)N2CCCC[C@@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147023455 HE On-Demand Mild MMP13 27 43 CC(=O)c1ccc(S(=O)(=O)N2CCCC[C@@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147023455 HE On-Demand Mild MMP3 20 43 CC(=O)c1ccc(S(=O)(=O)N2CCCC[C@@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147023455 HE On-Demand Mild MMP9 17 40 CC(=O)c1ccc(S(=O)(=O)N2CCCC[C@@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147023455 HE On-Demand Mild MMP7 39 43 CC(=O)c1ccc(S(=O)(=O)N2CCCC[C@@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147023455 HE On-Demand Mild MMP1 29 43 CC(=O)c1ccc(S(=O)(=O)N2CCCC[C@@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147023455 HE On-Demand Mild SFRP1 43 32 CC(=O)c1ccc(S(=O)(=O)N2CCCC[C@@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147023455 HE On-Demand Mild WNT3 52 33 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(Oc2cccc(F)c2)cc1 ZINC000147023506 GI On-Demand Anodyne LTA4H 34 40 CCO[C@H]1CCCN(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)C1 ZINC000147023509 GF On-Demand Anodyne CCR3 21 46 CCO[C@H]1CCCN(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)C1 ZINC000147023509 GF On-Demand Anodyne CPT1A 97 45 CCO[C@H]1CCCN(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)C1 ZINC000147023509 GF On-Demand Anodyne CPT2 43 39 CCO[C@H]1CCCN(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)C1 ZINC000147023509 GF On-Demand Anodyne EPHX2 36 41 CCO[C@H]1CCCN(C(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)C1 ZINC000147023509 GF On-Demand Anodyne TAAR1 23 40 CN(C)C(=O)c1cccc(CNC(=O)c2cccn(Cc3ccccc3)c2=O)c1 ZINC000147023537 GF On-Demand Anodyne DRTS_PLAFK 22 47 CN(C)C(=O)c1cccc(CNC(=O)c2cccn(Cc3ccccc3)c2=O)c1 ZINC000147023537 GF On-Demand Anodyne PTGER3 25 40 CN(C)C(=O)c1cccc(CNC(=O)c2cccn(Cc3ccccc3)c2=O)c1 ZINC000147023537 GF On-Demand Anodyne MMP13 17 40 CN(C)C(=O)c1cccc(CNC(=O)c2cccn(Cc3ccccc3)c2=O)c1 ZINC000147023537 GF On-Demand Anodyne UL54 67 34 CN(C)C(=O)c1cccc(CNC(=O)c2cccn(Cc3ccccc3)c2=O)c1 ZINC000147023537 GF On-Demand Anodyne POLR1A 47 33 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(NC(=O)c3ccccc3)c1)C2 ZINC000147023571 HI On-Demand Anodyne MTNR1A 24 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(NC(=O)c3ccccc3)c1)C2 ZINC000147023571 HI On-Demand Anodyne MTNR1B 25 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(NC(=O)c3ccccc3)c1)C2 ZINC000147023571 HI On-Demand Anodyne ROCK2 30 50 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(NC(=O)c3ccccc3)c1)C2 ZINC000147023571 HI On-Demand Anodyne TAAR1 48 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(NC(=O)c3ccccc3)c1)C2 ZINC000147023571 HI On-Demand Anodyne SMO 17 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(NC(=O)c3ccccc3)c1)C2 ZINC000147023571 HI On-Demand Anodyne KCNK3 127 56 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(NC(=O)c3ccccc3)c1)C2 ZINC000147023571 HI On-Demand Anodyne KCNK9 78 42 CS(=O)(=O)c1cc(C(=O)NCc2ccsc2)cc([N+](=O)[O-])c1 ZINC000147023583 ED On-Demand Bother MAPK9 33 40 CS(=O)(=O)c1cc(C(=O)NCc2ccsc2)cc([N+](=O)[O-])c1 ZINC000147023583 ED On-Demand Bother MAPK8 26 40 CCOC(=O)[C@H]1CCCC[C@H]1NC(=O)c1ccc(OC)c(Cl)c1 ZINC000147023622 EG Annotated Anodyne HTR4 48 37 CCOC(=O)[C@H]1CCCC[C@H]1NC(=O)c1ccc(OC)c(Cl)c1 ZINC000147023622 EG Annotated Anodyne SSTR3 32 46 CCN(Cc1ccc(OC)c(OC)c1)C(=O)[C@@H](C)OC[C@@H]1CCCO1 ZINC000147023649 FF On-Demand Anodyne OXTR 24 43 CCN(Cc1ccc(OC)c(OC)c1)C(=O)[C@@H](C)OC[C@@H]1CCCO1 ZINC000147023649 FF On-Demand Anodyne AVPR1A 16 41 Cc1ccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cn1 ZINC000147023814 DG On-Demand Anodyne NAMPT 25 46 CCN(Cc1ccc(OC)c(OC)c1)C(=O)[C@H](C)OC[C@@H]1CCCO1 ZINC000147023844 FF On-Demand Anodyne OXTR 24 43 CCN(Cc1ccc(OC)c(OC)c1)C(=O)[C@H](C)OC[C@@H]1CCCO1 ZINC000147023844 FF On-Demand Anodyne AVPR1A 16 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147023845 ED On-Demand Anodyne KCNQ2 78 43 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147023845 ED On-Demand Anodyne HDAC10 42 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147023845 ED On-Demand Anodyne HDAC2 27 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147023845 ED On-Demand Anodyne HDAC3 24 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147023845 ED On-Demand Anodyne HDAC6 24 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147023845 ED On-Demand Anodyne HDAC11 44 37 CCOC(=O)NCC(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147023944 DC On-Demand Anodyne F10 15 40 CCOC(=O)NCC(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147023944 DC On-Demand Anodyne PDS 41 39 Cc1ccc(C(=O)N2CCN(C(=O)c3ccn(-c4cccc(F)c4)n3)CC2)cc1 ZINC000147024004 GF On-Demand Anodyne HPGD 41 38 Cc1ccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cn1 ZINC000147024010 DG On-Demand Anodyne NAMPT 25 46 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147024037 ED On-Demand Anodyne KCNQ2 78 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147024037 ED On-Demand Anodyne HDAC10 42 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147024037 ED On-Demand Anodyne HDAC2 27 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147024037 ED On-Demand Anodyne HDAC3 25 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147024037 ED On-Demand Anodyne HDAC6 24 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147024037 ED On-Demand Anodyne HDAC11 44 37 CCN(Cc1ccc(OC)c(OC)c1)C(=O)[C@@H](C)OC[C@H]1CCCO1 ZINC000147024040 FF On-Demand Anodyne OXTR 24 43 CCN(Cc1ccc(OC)c(OC)c1)C(=O)[C@@H](C)OC[C@H]1CCCO1 ZINC000147024040 FF On-Demand Anodyne AVPR1A 16 41 C[C@@H](CNS(=O)(=O)CCc1ccccc1)N(C)c1ccccc1 ZINC000147024060 EF On-Demand Anodyne MMP12 15 45 COc1ccc(Nc2nc(-c3cccc(-c4ncco4)c3)cn3ccnc23)cc1OC ZINC000147024065 HJ For-Sale Anodyne SYK 67 69 COc1ccc(Nc2nc(-c3cccc(-c4ncco4)c3)cn3ccnc23)cc1OC ZINC000147024065 HJ For-Sale Anodyne EPHB4 43 44 CC[C@H](C)[C@@H]1NC(=O)[C@@H]([C@H](C)CC)NC1=O ZINC000147024090 BD For-Sale Anodyne GALR1 72 63 CC[C@H](C)[C@@H]1NC(=O)[C@@H]([C@H](C)CC)NC1=O ZINC000147024090 BD For-Sale Anodyne GALR2 33 63 Cc1ccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cn1 ZINC000147024202 DG On-Demand Anodyne NAMPT 25 46 CCN(Cc1ccc(OC)c(OC)c1)C(=O)[C@H](C)OC[C@H]1CCCO1 ZINC000147024229 FF On-Demand Anodyne OXTR 24 43 CCN(Cc1ccc(OC)c(OC)c1)C(=O)[C@H](C)OC[C@H]1CCCO1 ZINC000147024229 FF On-Demand Anodyne AVPR1A 16 41 C[C@H](CNS(=O)(=O)CCc1ccccc1)N(C)c1ccccc1 ZINC000147024255 EF On-Demand Anodyne MMP12 15 45 N#CC1CCN(C(=O)CCc2c(-c3ccccc3)[nH]c3ccc(F)cc23)CC1 ZINC000147024298 GJ On-Demand Mild TSPO 28 45 NC(=O)c1cn(C(=O)c2ccccc2)c2ccccc12 ZINC000147024358 CE In-Stock Anodyne ELANE 0 51 Cc1ccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cn1 ZINC000147024403 DG On-Demand Anodyne NAMPT 25 46 CC(=O)Nc1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147024421 FF On-Demand Anodyne CARM1 49 38 O=C(COCCCCCOCC(=O)Nc1ccccc1)Nc1ccccc1 ZINC000147024464 FG For-Sale Anodyne LTA4H 37 40 O=C(COCCCCCOCC(=O)Nc1ccccc1)Nc1ccccc1 ZINC000147024464 FG For-Sale Anodyne HDAC8 29 53 O=C(COCCCCCOCC(=O)Nc1ccccc1)Nc1ccccc1 ZINC000147024464 FG For-Sale Anodyne HDAC10 45 53 O=C(COCCCCCOCC(=O)Nc1ccccc1)Nc1ccccc1 ZINC000147024464 FG For-Sale Anodyne PLA2G4B 44 35 O=C(COCCCCCOCC(=O)Nc1ccccc1)Nc1ccccc1 ZINC000147024464 FG For-Sale Anodyne HDAC1 22 53 O=C(COCCCCCOCC(=O)Nc1ccccc1)Nc1ccccc1 ZINC000147024464 FG For-Sale Anodyne HDAC2 33 53 O=C(COCCCCCOCC(=O)Nc1ccccc1)Nc1ccccc1 ZINC000147024464 FG For-Sale Anodyne HDAC3 34 53 O=C(COCCCCCOCC(=O)Nc1ccccc1)Nc1ccccc1 ZINC000147024464 FG For-Sale Anodyne HDAC6 37 53 O=C(COCCCCCOCC(=O)Nc1ccccc1)Nc1ccccc1 ZINC000147024464 FG For-Sale Anodyne HDAC11 39 53 CCCCOc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147024615 EE On-Demand Anodyne MTNR1B 21 41 CCCCOc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147024615 EE On-Demand Anodyne PLA2G4B 52 39 CCCCOc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147024615 EE On-Demand Anodyne EPHX2 18 44 COC(=O)COc1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147024714 GE On-Demand Anodyne MMP13 44 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147024714 GE On-Demand Anodyne ADAM17 21 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147024714 GE On-Demand Anodyne MMP2 37 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147024714 GE On-Demand Anodyne MMP14 24 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147024714 GE On-Demand Anodyne PRTN3 45 33 COC(=O)COc1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147024714 GE On-Demand Anodyne MMP9 34 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147024714 GE On-Demand Anodyne MMP7 18 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147024714 GE On-Demand Anodyne ADAMTS4 58 38 COC(=O)COc1ccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)cc1 ZINC000147024714 GE On-Demand Anodyne LIMK2 35 40 COc1ccc(S(=O)(=O)N(C)CCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147024754 GD On-Demand Mild CHRM2 45 44 COc1ccc(S(=O)(=O)N(C)CCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147024754 GD On-Demand Mild BMP1 59 39 COc1ccc(S(=O)(=O)N(C)CCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147024754 GD On-Demand Mild MMP13 52 43 COc1ccc(S(=O)(=O)N(C)CCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147024754 GD On-Demand Mild MMP2 28 43 COc1ccc(S(=O)(=O)N(C)CCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147024754 GD On-Demand Mild MMP3 49 43 COc1ccc(S(=O)(=O)N(C)CCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147024754 GD On-Demand Mild MMP8 40 43 COc1ccc(S(=O)(=O)N(C)CCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147024754 GD On-Demand Mild MMP9 47 43 COc1ccc(S(=O)(=O)N(C)CCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147024754 GD On-Demand Mild MMP7 42 40 COc1ccc(S(=O)(=O)N(C)CCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147024754 GD On-Demand Mild MMP1 47 43 CCCCOc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147024795 EE On-Demand Anodyne MTNR1B 21 41 CCCCOc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147024795 EE On-Demand Anodyne PLA2G4B 52 39 CCCCOc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147024795 EE On-Demand Anodyne EPHX2 18 44 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147024823 HG On-Demand Anodyne AVPR2 81 43 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147024823 HG On-Demand Anodyne AVPR1A 43 43 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147024823 HG On-Demand Anodyne PIK3CA 32 42 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147024823 HG On-Demand Anodyne PRNP 57 35 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147024823 HG On-Demand Anodyne MTOR 51 42 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147024823 HG On-Demand Anodyne PIK3CG 23 42 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147024823 HG On-Demand Anodyne BTK 45 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147024890 GE On-Demand Anodyne MMP13 44 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147024890 GE On-Demand Anodyne ADAM17 21 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147024890 GE On-Demand Anodyne MMP2 37 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147024890 GE On-Demand Anodyne MMP14 24 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147024890 GE On-Demand Anodyne PRTN3 45 33 COC(=O)COc1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147024890 GE On-Demand Anodyne MMP9 34 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147024890 GE On-Demand Anodyne MMP7 18 40 COC(=O)COc1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147024890 GE On-Demand Anodyne ADAMTS4 58 38 COC(=O)COc1ccc(S(=O)(=O)NC[C@@H](C)N(C)c2ccccc2)cc1 ZINC000147024890 GE On-Demand Anodyne LIMK2 35 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025023 GE On-Demand Anodyne PIK3CA 21 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025023 GE On-Demand Anodyne MTNR1A 17 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025023 GE On-Demand Anodyne MTNR1B 15 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025023 GE On-Demand Anodyne ROCK2 32 53 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025023 GE On-Demand Anodyne MTOR 38 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025023 GE On-Demand Anodyne EPHX2 19 46 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025023 GE On-Demand Anodyne PIK3CG 17 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025023 GE On-Demand Anodyne LRRK2 26 40 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne HTR1A 35 47 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne DRD2 42 51 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne DRD1 27 63 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne DRD4 27 44 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne HTR2A 38 63 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne SLC6A4 21 40 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne HRH1 16 58 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne DRD3 29 63 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne KCNH2 15 55 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne DRD5 33 42 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne HTR7 35 49 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne HRH3 60 55 Fc1ccc(N2CCN(CCCOc3ccc4c(c3)OCO4)CC2)cc1 ZINC000147025042 FG On-Demand Anodyne SIGMAR1 31 52 N#Cc1ccc(Oc2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2Cl)cc1 ZINC000147025137 HJ On-Demand Anodyne PFKFB3 41 33 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025213 GE On-Demand Anodyne PIK3CA 21 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025213 GE On-Demand Anodyne MTNR1A 17 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025213 GE On-Demand Anodyne MTNR1B 15 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025213 GE On-Demand Anodyne ROCK2 32 53 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025213 GE On-Demand Anodyne MTOR 38 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025213 GE On-Demand Anodyne EPHX2 19 46 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025213 GE On-Demand Anodyne PIK3CG 17 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCOCC3)cc1)C2 ZINC000147025213 GE On-Demand Anodyne LRRK2 26 40 Cc1ccc(CNC(=O)N[C@H](CC(C)C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147025365 FF On-Demand Mild ANPEP 39 57 Cc1ccc(CNC(=O)N[C@H](CC(C)C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147025365 FF On-Demand Mild CCKAR 0 46 Cc1ccc(CNC(=O)N[C@H](CC(C)C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147025365 FF On-Demand Mild CTSK 28 45 Cc1ccc(CNC(=O)N[C@H](CC(C)C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147025365 FF On-Demand Mild CACNA1B 15 40 Cc1ccc(CNC(=O)N[C@H](CC(C)C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147025365 FF On-Demand Mild CCR1 31 43 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147025501 GH On-Demand Anodyne AVPR2 18 40 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147025501 GH On-Demand Anodyne EPHX2 23 56 Cc1cccc(S(=O)(=O)NC[C@H](C)N(C)c2ccccc2)c1 ZINC000147025649 DF On-Demand Anodyne FBP1 18 42 O=C(O)c1ccc(N2C(=O)C=C(c3ccccc3)C2=O)cc1 ZINC000147025680 CE For-Sale Anodyne CA12 15 47 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147025697 GH On-Demand Anodyne AVPR2 18 40 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147025697 GH On-Demand Anodyne EPHX2 23 56 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne CHRM2 35 41 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne CHRM1 19 43 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne DRD2 27 43 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne DRD4 57 42 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne ACHE 41 47 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne DRD3 21 42 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne OPRK1 15 40 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne OPRL1 19 41 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne CHRM3 28 40 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne LTA4H 25 42 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne HRH3 25 45 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne SIGMAR1 75 48 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne CACNA1B 15 42 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne CCR3 46 37 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne CCR5 21 45 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne CXCR3 27 43 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne MCHR1 29 42 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne CACNA1G 31 45 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne GPR119 49 43 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne KDM1A 19 40 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne NPFFR1 43 33 CC(C)(C)OC(=O)N1CCN(C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147025744 FG In-Stock Anodyne L3MBTL3 58 47 CCCc1nc(CS(=O)(=O)CC(=O)N[C@@H]2CCOc3ccccc32)no1 ZINC000147025864 GD On-Demand Anodyne BDKRB1 25 41 CCCc1nc(CS(=O)(=O)CC(=O)N[C@@H]2CCOc3ccccc32)no1 ZINC000147025864 GD On-Demand Anodyne LASR 42 31 NC(=O)c1ccccc1[C@@H]1CCNC1 ZINC000147025867 AC For-Sale Anodyne SLC6A2 22 44 NC(=O)c1ccccc1[C@@H]1CCNC1 ZINC000147025867 AC For-Sale Anodyne PARP2 50 43 NC(=O)c1ccccc1[C@@H]1CCNC1 ZINC000147025867 AC For-Sale Anodyne PARP1 29 54 NC(=O)c1ccccc1[C@@H]1CCNC1 ZINC000147025867 AC For-Sale Anodyne CDK2AP1 42 34 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147025895 GH On-Demand Anodyne AVPR2 18 40 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147025895 GH On-Demand Anodyne EPHX2 23 56 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne CA2 76 50 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne CA6 20 40 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne CA1 62 47 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne CA7 39 40 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne CA4 64 37 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne CA12 39 50 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne ALPL 17 43 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne CA9 49 50 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne CAH_METTE 31 40 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne CYNT 37 40 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne ALPI 15 43 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne CA15 20 40 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne MTCA1 31 40 C[C@@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147025904 GD On-Demand Anodyne A6YCJ1_9METZ 29 40 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne ACE 15 42 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne MME 30 41 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne PAPA1_CARPA 60 60 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne CTSK 27 45 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne CTSL 18 60 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne TACR3 18 47 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne GRIA1 43 38 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne REN 34 41 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne YARS 60 35 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne CTSS 15 60 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne ACE2 39 42 C[C@H](Cc1ccc(O)cc1)NC(=O)OC(C)(C)C ZINC000147026033 CF For-Sale Anodyne FPR1 45 44 CCCc1nc(CS(=O)(=O)CC(=O)N[C@H]2CCOc3ccccc32)no1 ZINC000147026055 GD On-Demand Anodyne BDKRB1 25 41 CCCc1nc(CS(=O)(=O)CC(=O)N[C@H]2CCOc3ccccc32)no1 ZINC000147026055 GD On-Demand Anodyne LASR 42 31 NC(=O)c1ccccc1[C@H]1CCNC1 ZINC000147026075 AC For-Sale Anodyne SLC6A2 22 44 NC(=O)c1ccccc1[C@H]1CCNC1 ZINC000147026075 AC For-Sale Anodyne PARP2 50 43 NC(=O)c1ccccc1[C@H]1CCNC1 ZINC000147026075 AC For-Sale Anodyne PARP1 29 54 NC(=O)c1ccccc1[C@H]1CCNC1 ZINC000147026075 AC For-Sale Anodyne CDK2AP1 42 34 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne CA2 76 50 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne CA6 20 40 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne CA1 62 47 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne CA7 39 40 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne CA4 64 37 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne CA12 39 50 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne ALPL 17 43 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne CA9 49 50 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne CAH_METTE 31 40 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne CYNT 37 40 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne ALPI 15 43 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne CA15 20 40 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne MTCA1 31 40 C[C@H](CNS(=O)(=O)c1ccc(S(N)(=O)=O)cc1)N(C)c1ccccc1 ZINC000147026083 GD On-Demand Anodyne A6YCJ1_9METZ 29 40 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147026108 GH On-Demand Anodyne AVPR2 18 40 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147026108 GH On-Demand Anodyne EPHX2 23 56 CC1CCN(C(=O)c2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2)CC1 ZINC000147026213 GG On-Demand Anodyne L3MBTL3 70 38 COc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1OCC(=O)NC1CC1 ZINC000147026304 HH On-Demand Anodyne ENPP1 50 34 CCCNC(=O)c1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147026347 FG On-Demand Anodyne MAPK10 17 42 CCCNC(=O)c1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147026347 FG On-Demand Anodyne KCNK3 77 42 CCCNC(=O)c1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147026347 FG On-Demand Anodyne KCNK9 42 42 CS(=O)(=O)Nc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147026367 DD On-Demand Mild L3MBTL3 78 40 Cc1c[nH]c2c(Nc3nc(Cl)cc4cn[nH]c(=O)c34)cccc12 ZINC000147026470 EH For-Sale Anodyne ZAP70 15 48 COc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1OCC(=O)NC1CC1 ZINC000147026495 HH On-Demand Anodyne ENPP1 50 34 CCOc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147026544 DD On-Demand Anodyne TAAR1 27 43 NC1=N[C@](c2cccc(NC(=O)c3ccc(O)cn3)c2)(C2CCCCC2)CS1 ZINC000147026659 GH Annotated Anodyne BACE2 46 62 NC1=N[C@](c2cccc(NC(=O)c3ccc(O)cn3)c2)(C2CCCCC2)CS1 ZINC000147026659 GH Annotated Anodyne BACE1 29 74 COc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1OCC(=O)NC1CC1 ZINC000147026704 HH On-Demand Anodyne ENPP1 50 34 CCOc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147026743 DD On-Demand Anodyne TAAR1 27 43 C[C@H](NS(=O)(=O)CCc1ccccc1)c1ccc(OCc2cccnc2)cc1 ZINC000147026775 GH On-Demand Anodyne MMP13 19 40 C[C@H](NS(=O)(=O)CCc1ccccc1)c1ccc(OCc2cccnc2)cc1 ZINC000147026775 GH On-Demand Anodyne ADAMTS4 47 37 NC1=N[C@@](c2cccc(NC(=O)c3ccc(O)cn3)c2)(C2CCCCC2)CS1 ZINC000147026871 GH Annotated Anodyne BACE2 46 62 NC1=N[C@@](c2cccc(NC(=O)c3ccc(O)cn3)c2)(C2CCCCC2)CS1 ZINC000147026871 GH Annotated Anodyne BACE1 29 74 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne ABL1 25 43 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne ESR1 33 40 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne ESR2 24 40 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne FGFR1 19 48 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne SRC 35 50 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne JAK3 25 66 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne JAK2 37 66 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne DAPK1 15 48 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne YES1 24 46 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne TNK2 21 48 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne NEK9 15 48 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne WEE1 23 48 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne EPHB4 15 46 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne PSMB2 44 33 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne RIOK3 15 48 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne ADCK4 15 48 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne PIP5K1A 15 48 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne RIOK1 15 48 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne DCLK3 15 48 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne SNRK 0 48 CS(=O)(=O)c1cccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)c1 ZINC000147026887 JI Annotated Anodyne PKNB 17 48 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne ACE 61 42 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne OPRM1 61 48 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne OPRD1 53 48 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne MME 157 56 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne LTA4H 21 40 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne ANPEP 107 40 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne TACR1 19 45 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne CTRA_BOVIN 18 47 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne FCER2 82 41 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne RNPEP 40 38 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne CTSB 59 45 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne PAPA1_CARPA 79 45 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne CYSP_TRYCR 61 41 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne CTSK 32 45 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne CTSL 59 45 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne CPA1 62 45 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne NPFFR2 56 36 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne TIMP3 80 39 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne NAALAD2 26 42 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne CAPNS1 72 44 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne MMP3 33 47 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne MMP8 21 42 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne GRIA1 48 39 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne HLA-DRB1 61 36 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne CTSS 26 45 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne CAPN1 95 44 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne MMP9 27 42 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne CAPN2 76 45 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne ACE2 82 42 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne LAP3 65 40 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne MMP1 39 48 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne FPR1 73 41 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne CTRB_BOVIN 50 37 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne NPR 67 50 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne AMP1_PLAFQ 54 39 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne BLA1_STEMA 70 37 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne NPFFR1 67 36 COC(=O)CN[C@H](Cc1ccccc1)C(=O)OC ZINC000147026892 CC On-Demand Anodyne GPR142 45 43 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccc2c(c1)COC2 ZINC000147026908 FE On-Demand Anodyne AVPR2 38 45 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccc2c(c1)COC2 ZINC000147026908 FE On-Demand Anodyne AVPR1A 23 45 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccc2c(c1)COC2 ZINC000147026908 FE On-Demand Anodyne PIK3CA 23 44 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccc2c(c1)COC2 ZINC000147026908 FE On-Demand Anodyne PRNP 46 37 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccc2c(c1)COC2 ZINC000147026908 FE On-Demand Anodyne MTOR 33 44 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccc2c(c1)COC2 ZINC000147026908 FE On-Demand Anodyne EPHX2 22 57 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccc2c(c1)COC2 ZINC000147026908 FE On-Demand Anodyne PIK3CG 20 44 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccc2c(c1)COC2 ZINC000147026908 FE On-Demand Anodyne BTK 42 39 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccc2c(c1)COC2 ZINC000147026908 FE On-Demand Anodyne AKR1C3 19 45 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccc2c(c1)COC2 ZINC000147026908 FE On-Demand Anodyne L3MBTL3 48 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCCCC2)cc1 ZINC000147026948 GE On-Demand Anodyne NPY2R 17 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCCCC2)cc1 ZINC000147026948 GE On-Demand Anodyne MTOR 16 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCCCC2)cc1 ZINC000147026948 GE On-Demand Anodyne EPHX2 19 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCCCC2)cc1 ZINC000147026948 GE On-Demand Anodyne L3MBTL3 80 40 CSC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147026962 KB Annotated Anodyne POLA1 48 54 CSC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147026962 KB Annotated Anodyne P2RY6 117 45 CSC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147026962 KB Annotated Anodyne POLB 46 54 CSC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147026962 KB Annotated Anodyne P2RX4 41 40 CSC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147026962 KB Annotated Anodyne P2RX1 56 40 CSC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147026962 KB Annotated Anodyne P2RY4 125 45 CSC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147026962 KB Annotated Anodyne P2RY1 31 40 CSC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147026962 KB Annotated Anodyne P2RY2 158 47 CSC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147026962 KB Annotated Anodyne P2RY14 51 36 CSC[C@]1(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)O[C@@H](n2ccc(N)nc2=O)[C@H](F)[C@@H]1O ZINC000147026962 KB Annotated Anodyne GPR17 54 34 C[C@@H](NS(=O)(=O)CCc1ccccc1)c1ccc(OCc2cccnc2)cc1 ZINC000147026965 GH On-Demand Anodyne MMP13 19 40 C[C@@H](NS(=O)(=O)CCc1ccccc1)c1ccc(OCc2cccnc2)cc1 ZINC000147026965 GH On-Demand Anodyne ADAMTS4 47 37 COc1ccc(/C=C/C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027040 DF On-Demand Anodyne MAOB 0 54 COc1ccc(/C=C/C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027040 DF On-Demand Anodyne MMP2 23 54 COc1ccc(/C=C/C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027040 DF On-Demand Anodyne MMP9 0 46 COc1ccc(/C=C/C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027040 DF On-Demand Anodyne IMPDH2 0 47 COc1ccc(/C=C/C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027040 DF On-Demand Anodyne MMP1 23 46 COc1ccc(/C=C/C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027040 DF On-Demand Anodyne MCHR1 0 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCCCC2)cc1 ZINC000147027119 GE On-Demand Anodyne NPY2R 17 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCCCC2)cc1 ZINC000147027119 GE On-Demand Anodyne MTOR 16 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCCCC2)cc1 ZINC000147027119 GE On-Demand Anodyne EPHX2 19 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCCCC2)cc1 ZINC000147027119 GE On-Demand Anodyne L3MBTL3 80 40 Nc1ccn([C@@H]2O[C@](CBr)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147027166 KB Annotated Reactive POLA1 47 55 Nc1ccn([C@@H]2O[C@](CBr)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147027166 KB Annotated Reactive P2RY6 119 44 Nc1ccn([C@@H]2O[C@](CBr)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147027166 KB Annotated Reactive POLB 56 55 Nc1ccn([C@@H]2O[C@](CBr)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147027166 KB Annotated Reactive P2RX4 41 36 Nc1ccn([C@@H]2O[C@](CBr)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147027166 KB Annotated Reactive P2RX1 56 36 Nc1ccn([C@@H]2O[C@](CBr)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147027166 KB Annotated Reactive P2RY4 128 44 Nc1ccn([C@@H]2O[C@](CBr)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147027166 KB Annotated Reactive P2RY2 160 49 Nc1ccn([C@@H]2O[C@](CBr)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147027166 KB Annotated Reactive P2RY14 52 37 Nc1ccn([C@@H]2O[C@](CBr)(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@@H](O)[C@H]2F)c(=O)n1 ZINC000147027166 KB Annotated Reactive GPR17 44 34 N#CC1CCN(C(=O)CC[C@H]2Cc3ccccc3NC2=O)CC1 ZINC000147027173 DE On-Demand Mild FAP 0 41 COc1ccc(/C=C\C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027229 DF On-Demand Anodyne MAOB 17 54 COc1ccc(/C=C\C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027229 DF On-Demand Anodyne MMP2 23 54 COc1ccc(/C=C\C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027229 DF On-Demand Anodyne ROCK2 18 46 COc1ccc(/C=C\C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027229 DF On-Demand Anodyne MMP9 20 46 COc1ccc(/C=C\C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027229 DF On-Demand Anodyne HPSE 28 40 COc1ccc(/C=C\C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027229 DF On-Demand Anodyne TUBB1 46 44 COc1ccc(/C=C\C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027229 DF On-Demand Anodyne IMPDH2 38 40 COc1ccc(/C=C\C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027229 DF On-Demand Anodyne MMP1 23 46 COc1ccc(/C=C\C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027229 DF On-Demand Anodyne MCHR1 17 40 COc1ccc(/C=C\C(=O)Nc2ccc3[nH]ncc3c2)cc1O ZINC000147027229 DF On-Demand Anodyne ENPP1 51 32 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2)c(F)c1 ZINC000147027329 EE On-Demand Anodyne NPY2R 89 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2)c(F)c1 ZINC000147027329 EE On-Demand Anodyne ENV 43 34 N#CC1CCN(C(=O)CC[C@@H]2Cc3ccccc3NC2=O)CC1 ZINC000147027361 DE On-Demand Mild FAP 0 41 COc1cccc(F)c1CN1C[C@H](NC(=O)c2ccc3[nH]nc(-c4ccnc(C)c4)c3c2)CC[C@H]1C(=O)N1CCNCC1 ZINC000147027409 KG Annotated Anodyne TTK 47 33 C=CCN1C(C)(C)CC(NC(=O)c2ccccc2)CC1(C)C ZINC000147027489 DH In-Stock Mild EZH2 44 35 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2)c(F)c1 ZINC000147027506 EE On-Demand Anodyne NPY2R 89 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2)c(F)c1 ZINC000147027506 EE On-Demand Anodyne ENV 43 34 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCN(c2ccncc2)CC1 ZINC000147027570 II Annotated Anodyne PDGFRB 25 55 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCN(c2ccncc2)CC1 ZINC000147027570 II Annotated Anodyne FGFR1 37 55 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCN(c2ccncc2)CC1 ZINC000147027570 II Annotated Anodyne ITK 29 47 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCN(c2ccncc2)CC1 ZINC000147027570 II Annotated Anodyne FLT1 29 55 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCN(c2ccncc2)CC1 ZINC000147027570 II Annotated Anodyne CDK2 0 42 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCN(c2ccncc2)CC1 ZINC000147027570 II Annotated Anodyne TTK 48 42 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCN(c2ccncc2)CC1 ZINC000147027570 II Annotated Anodyne PAK4 15 42 O=C(Nc1ccc2[nH]nc(-c3nc4ccccc4[nH]3)c2c1)C1CCN(c2ccncc2)CC1 ZINC000147027570 II Annotated Anodyne NR2E3 70 44 C[C@@H](CNC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1)N(C)c1ccccc1 ZINC000147027632 GE On-Demand Bother COLA 71 36 CCCC[C@@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027717 FJ Annotated Anodyne PTGFR 47 38 CCCC[C@@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027717 FJ Annotated Anodyne PTGER2 45 54 CCCC[C@@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027717 FJ Annotated Anodyne TBXA2R 16 44 CCCC[C@@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027717 FJ Annotated Anodyne PTGER1 30 54 CCCC[C@@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027717 FJ Annotated Anodyne PTGER4 26 54 CCCC[C@@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027717 FJ Annotated Anodyne PTGER3 25 54 CCCC[C@@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027717 FJ Annotated Anodyne PTGDR 0 49 CCCC[C@@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027717 FJ Annotated Anodyne SLCO2A1 68 49 C[C@H](CNC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1)N(C)c1ccccc1 ZINC000147027817 GE On-Demand Bother COLA 71 36 NC(=O)c1ccc(OCC(=O)NCc2cccnc2OCC(F)(F)F)cc1 ZINC000147027845 GD On-Demand Anodyne SCN10A 15 49 CCCC[C@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027893 FJ Annotated Anodyne PTGFR 47 38 CCCC[C@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027893 FJ Annotated Anodyne PTGER2 45 54 CCCC[C@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027893 FJ Annotated Anodyne TBXA2R 16 44 CCCC[C@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027893 FJ Annotated Anodyne PTGER1 30 54 CCCC[C@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027893 FJ Annotated Anodyne PTGER4 26 54 CCCC[C@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027893 FJ Annotated Anodyne PTGER3 25 54 CCCC[C@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027893 FJ Annotated Anodyne PTGDR 0 49 CCCC[C@H](C)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147027893 FJ Annotated Anodyne SLCO2A1 68 49 COc1ccccc1Nc1nc2c(-c3cccc(C(F)(F)F)c3)cccn2n1 ZINC000147027998 GK Annotated Anodyne JAK2 21 48 COc1ccc([N+](=O)[O-])c(C(=O)NC2CCN(c3ccccn3)CC2)c1 ZINC000147028109 FE On-Demand Bother GYRB 18 41 COc1ccc([N+](=O)[O-])c(C(=O)NC2CCN(c3ccccn3)CC2)c1 ZINC000147028109 FE On-Demand Bother DRD4 31 46 COc1ccc([N+](=O)[O-])c(C(=O)NC2CCN(c3ccccn3)CC2)c1 ZINC000147028109 FE On-Demand Bother EBP 26 41 COc1ccc([N+](=O)[O-])c(C(=O)NC2CCN(c3ccccn3)CC2)c1 ZINC000147028109 FE On-Demand Bother TAAR1 19 41 CC(C)OCC(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)ccc1Cl ZINC000147028186 FG On-Demand Anodyne F2 27 45 CC(C)OCC(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)ccc1Cl ZINC000147028186 FG On-Demand Anodyne ELANE 43 35 CC(C)OCC(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)ccc1Cl ZINC000147028186 FG On-Demand Anodyne PREP 22 41 CC(C)OCC(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)ccc1Cl ZINC000147028186 FG On-Demand Anodyne LGMN 62 34 CS(=O)(=O)Nc1ccc(/C=C/C(=O)N2CCC(C#N)CC2)cc1 ZINC000147028194 ED On-Demand Mild CCR2 61 41 Cc1cc(N2CCC(N3CCC[C@@H]3C)CC2)ccc1[N+](=O)[O-] ZINC000147028207 DG On-Demand Bother HRH3 56 50 CN(C(=N)Nc1cccc2ccccc12)c1cccc(Br)c1 ZINC000147028476 FK Annotated Anodyne SIGMAR1 19 74 CCN1CC[C@@H](c2ccccc2)[C@H](NC(=O)c2ccc3[nH]nc(-c4ccc(OC(C)C)nc4)c3c2)C1 ZINC000147028494 JK Annotated Anodyne TTK 63 43 CCc1ccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])s1 ZINC000147028513 DG On-Demand Bother AKR1C2 22 40 COc1cc(CNC(=O)c2csc(-c3ccccc3F)n2)ccc1O ZINC000147028591 FH On-Demand Anodyne TRPV1 27 45 COc1ccccc1N1C[C@H](C(=O)N2CCC(C#N)CC2)CC1=O ZINC000147028618 ED On-Demand Mild SSTR2 45 41 COc1ccccc1N1C[C@H](C(=O)N2CCC(C#N)CC2)CC1=O ZINC000147028618 ED On-Demand Mild SSTR1 54 41 CCC[C@@H](c1ccccn1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147028629 KK Annotated Anodyne TP53 42 65 CCC[C@@H](c1ccccn1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147028629 KK Annotated Anodyne MDM2 249 65 Cc1cc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)n(-c2ccc(C(F)(F)F)cn2)n1 ZINC000147028684 HI On-Demand Anodyne EPHX2 23 41 COc1ccc(OC)c2c[n+]3c(cc12)-c1cc2c(cc1CC3)OCO2 ZINC000147028738 EG Annotated Anodyne ACHE 38 73 COc1ccc(OC)c2c[n+]3c(cc12)-c1cc2c(cc1CC3)OCO2 ZINC000147028738 EG Annotated Anodyne BCHE 23 72 COc1ccc(OC)c2c[n+]3c(cc12)-c1cc2c(cc1CC3)OCO2 ZINC000147028738 EG Annotated Anodyne F3 19 40 C[C@@]1(c2cc(NC(=O)c3ccc(-c4ccc[nH]4)cn3)ccc2F)C=CSC(N)=N1 ZINC000147028753 HI Annotated Anodyne BACE2 50 51 C[C@@]1(c2cc(NC(=O)c3ccc(-c4ccc[nH]4)cn3)ccc2F)C=CSC(N)=N1 ZINC000147028753 HI Annotated Anodyne BACE1 25 47 O=C(NC1CC1)C(=O)N1CCN(C(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147028763 GD On-Demand Anodyne NPBWR1 48 34 C=CCCOCC(=O)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147028823 FF On-Demand Mild RBP4 51 38 C=CCCOCC(=O)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147028823 FF On-Demand Mild SCD1 22 44 C=CCCOCC(=O)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147028823 FF On-Demand Mild SCD 24 43 Cc1cc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)n(-c2ccc(C(F)(F)F)cn2)n1 ZINC000147028884 HI On-Demand Anodyne EPHX2 23 41 O=C(NC1CC1)C(=O)N1CCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147028921 GD On-Demand Anodyne NPBWR1 48 34 Cc1cc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)n(-c2ccc(C(F)(F)F)cn2)n1 ZINC000147029090 HI On-Demand Anodyne EPHX2 23 41 O=C(NC1CC1)C(=O)N1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147029111 GD On-Demand Anodyne NPBWR1 57 34 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne MME 56 38 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne LTA4H 21 40 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne MMP13 15 46 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne CTSB 39 41 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne PAPA1_CARPA 51 34 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne CPA1 53 37 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne CAPNS1 61 40 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne CAPN1 75 41 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne CAPN2 95 38 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne ACE2 57 37 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne ADAMTS4 66 40 CN[C@@H](C(=O)O)[C@@H](C)OCc1ccccc1 ZINC000147029115 BD In-Stock Anodyne NPR 59 36 CC(=O)Nc1ccc(Cl)c(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147029209 FD On-Demand Anodyne ENV 42 35 Cc1cc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)n(-c2ccc(C(F)(F)F)cn2)n1 ZINC000147029293 HI On-Demand Anodyne EPHX2 23 41 COc1ccccc1S(=O)(=O)N[C@@H](C)c1ccc(OCc2cccnc2)cc1 ZINC000147029296 GH On-Demand Anodyne ADAMTS4 43 35 O=C(NC1CC1)C(=O)N1CCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147029309 GD On-Demand Anodyne NPBWR1 48 34 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne MME 56 38 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne LTA4H 21 40 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne MMP13 15 46 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne CTSB 39 41 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne PAPA1_CARPA 51 34 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne CPA1 53 37 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne CAPNS1 61 40 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne CAPN1 75 41 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne CAPN2 95 38 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne ACE2 57 37 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne ADAMTS4 66 40 CN[C@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029325 BD In-Stock Anodyne NPR 59 36 CC(C)(C)c1nc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2o1 ZINC000147029385 FG On-Demand Anodyne ADORA2B 37 42 CC(C)(C)c1nc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2o1 ZINC000147029385 FG On-Demand Anodyne MCHR1 16 41 CC(=O)Nc1ccc(Cl)c(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147029393 FD On-Demand Anodyne ENV 42 35 O=C(NCc1cccnc1OCC(F)(F)F)c1cccn(Cc2ccccc2)c1=O ZINC000147029433 HG On-Demand Anodyne SCN10A 29 51 COc1ccccc1S(=O)(=O)N[C@H](C)c1ccc(OCc2cccnc2)cc1 ZINC000147029485 GH On-Demand Anodyne ADAMTS4 43 35 CCCNC(=O)c1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1Cl ZINC000147029498 GG On-Demand Anodyne SLC6A9 40 34 COc1ccc2c(c1)OC[C@H](C(=O)N1CCN(C(=O)C(=O)NC3CC3)CC1)C2 ZINC000147029507 GC On-Demand Anodyne MTNR1A 20 43 COc1ccc2c(c1)OC[C@H](C(=O)N1CCN(C(=O)C(=O)NC3CC3)CC1)C2 ZINC000147029507 GC On-Demand Anodyne MTNR1B 15 45 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne MME 56 38 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne LTA4H 21 40 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne MMP13 15 46 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne CTSB 39 41 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne PAPA1_CARPA 51 34 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne CPA1 53 37 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne CAPNS1 61 40 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne CAPN1 75 41 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne CAPN2 95 38 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne ACE2 57 37 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne ADAMTS4 66 40 CN[C@@H](C(=O)O)[C@H](C)OCc1ccccc1 ZINC000147029517 BD In-Stock Anodyne NPR 59 36 CN1CCN(c2ccc(Nc3nc4ccc(-c5ccc(S(C)(=O)=O)cc5)cn4n3)cc2)CC1 ZINC000147029527 JG Annotated Anodyne JAK3 22 66 CN1CCN(c2ccc(Nc3nc4ccc(-c5ccc(S(C)(=O)=O)cc5)cn4n3)cc2)CC1 ZINC000147029527 JG Annotated Anodyne JAK2 45 70 CN1CCN(c2ccc(Nc3nc4ccc(-c5ccc(S(C)(=O)=O)cc5)cn4n3)cc2)CC1 ZINC000147029527 JG Annotated Anodyne PIK3CG 17 47 CC[C@@H](C)c1ccccc1OCC(=O)N1CCC(C#N)CC1 ZINC000147029555 DG On-Demand Mild AO-ACHE 0 43 CNC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147029576 FD On-Demand Anodyne ENV 41 34 CC(C)c1nc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2o1 ZINC000147029586 FG On-Demand Anodyne ADORA2B 37 42 CC(C)c1nc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2o1 ZINC000147029586 FG On-Demand Anodyne ENPP1 46 32 O=C(O)/C(F)=C(/F)c1ccccc1 ZINC000147029650 AE For-Sale Anodyne PA 15 41 CCOC(=O)N1CCc2ccccc2[C@@H]1c1ccc(F)cc1 ZINC000147029691 CH For-Sale Anodyne CA14 19 42 CCOC(=O)N1CCc2ccccc2[C@@H]1c1ccc(F)cc1 ZINC000147029691 CH For-Sale Anodyne TRPM8 57 55 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCN(C(=O)C(=O)NC3CC3)CC1)C2 ZINC000147029704 GC On-Demand Anodyne MTNR1A 20 43 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCN(C(=O)C(=O)NC3CC3)CC1)C2 ZINC000147029704 GC On-Demand Anodyne MTNR1B 15 45 CNC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147029741 FD On-Demand Anodyne ENV 41 34 CCOC(=O)N1CCc2ccccc2[C@H]1c1ccc(F)cc1 ZINC000147029866 CH For-Sale Anodyne CA14 19 42 CCOC(=O)N1CCc2ccccc2[C@H]1c1ccc(F)cc1 ZINC000147029866 CH For-Sale Anodyne TRPM8 57 55 O=C(Nc1cccc(CNS(=O)(=O)c2cccc3cnccc23)c1)[C@@H]1CCCO1 ZINC000147029894 HF On-Demand Anodyne NPY5R 19 42 CCc1cc(=O)nc(-c2cccc(NC(=O)[C@H]3COc4cc(OC)ccc4C3)c2)[nH]1 ZINC000147029897 HG On-Demand Anodyne ROCK2 33 47 CCOc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1F ZINC000147029935 DD On-Demand Anodyne ENV 43 35 O=C(Nc1cccc(CNS(=O)(=O)c2cccc3cnccc23)c1)[C@H]1CCCO1 ZINC000147030078 HF On-Demand Anodyne NPY5R 19 42 CCOc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1F ZINC000147030123 DD On-Demand Anodyne ENV 43 35 N#Cc1nc(C2CC2)oc1N1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147030250 GD On-Demand Mild CPT1A 36 40 N#CC1CCN(C(=O)CNC(=O)NCc2ccc(F)cc2)CC1 ZINC000147030360 DD On-Demand Mild DPP4 25 42 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)Cc3ccccc3)CC2)c1 ZINC000147030508 GE On-Demand Bother MMP13 26 41 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)Cc3ccccc3)CC2)c1 ZINC000147030508 GE On-Demand Bother MMP9 29 41 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)Cc3ccccc3)CC2)c1 ZINC000147030508 GE On-Demand Bother MMP1 29 41 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)Cc3ccccc3)CC2)c1 ZINC000147030508 GE On-Demand Bother MGLL 0 41 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)Cc3ccccc3)CC2)c1 ZINC000147030508 GE On-Demand Bother AKR1C3 26 45 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)Cc3ccccc3)CC2)c1 ZINC000147030508 GE On-Demand Bother ABHD6 0 41 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)Cc3ccccc3)CC2)c1 ZINC000147030508 GE On-Demand Bother AKR1C2 43 45 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)Cc3ccccc3)CC2)c1 ZINC000147030508 GE On-Demand Bother GPR183 0 53 CCCS(=O)(=O)NC1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147030565 GC On-Demand Anodyne PRSS2 43 32 CCCS(=O)(=O)NC1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147030565 GC On-Demand Anodyne CPT1A 25 43 CCCS(=O)(=O)NC1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147030565 GC On-Demand Anodyne CCR8 72 43 C[C@@]1(c2cc(NC(=O)c3cnc(-n4nccn4)cn3)ccc2F)C=CSC(N)=N1 ZINC000147030571 HE Annotated Anodyne BACE2 49 51 C[C@@]1(c2cc(NC(=O)c3cnc(-n4nccn4)cn3)ccc2F)C=CSC(N)=N1 ZINC000147030571 HE Annotated Anodyne BACE1 25 57 COc1cc(C)c(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1C ZINC000147030642 HF On-Demand Anodyne CCR4 18 41 O=C(Cc1ccccc1)N1CCN(C(=O)c2ccn(-c3cccc(F)c3)n2)CC1 ZINC000147030705 GF On-Demand Anodyne KCNJ1 43 36 O=C(Cc1ccccc1)N1CCN(C(=O)c2ccn(-c3cccc(F)c3)n2)CC1 ZINC000147030705 GF On-Demand Anodyne GPR183 0 43 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030706 ED On-Demand Anodyne KLK3 84 38 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030706 ED On-Demand Anodyne CTSK 48 43 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030706 ED On-Demand Anodyne NPFFR2 40 38 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030706 ED On-Demand Anodyne C3AR1 55 34 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030706 ED On-Demand Anodyne MMP3 21 42 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030706 ED On-Demand Anodyne HLA-DRB1 46 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030706 ED On-Demand Anodyne PCSK5 41 34 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030706 ED On-Demand Anodyne FURIN 54 31 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030706 ED On-Demand Anodyne CAPN2 49 36 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030706 ED On-Demand Anodyne POLG_WNV 83 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030706 ED On-Demand Anodyne NPFFR1 55 38 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne DRD2 15 47 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne DRD4 42 43 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne ACHE 42 45 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne DRD3 18 40 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne LTA4H 20 41 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne SIGMAR1 45 43 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne SSTR5 72 56 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne CCR3 20 47 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne AURKB 15 42 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne ITK 21 42 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne CXCR3 16 50 Nc1ccc2nc(NC3CCN(Cc4ccccc4)CC3)sc2c1 ZINC000147030805 EH On-Demand Anodyne MCHR1 20 44 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030900 ED On-Demand Anodyne KLK3 84 38 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030900 ED On-Demand Anodyne CTSK 48 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030900 ED On-Demand Anodyne NPFFR2 40 38 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030900 ED On-Demand Anodyne C3AR1 55 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030900 ED On-Demand Anodyne MMP3 21 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030900 ED On-Demand Anodyne HLA-DRB1 46 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030900 ED On-Demand Anodyne PCSK5 41 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030900 ED On-Demand Anodyne FURIN 54 31 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030900 ED On-Demand Anodyne CAPN2 49 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030900 ED On-Demand Anodyne POLG_WNV 83 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC(=O)OC)c1ccccc1 ZINC000147030900 ED On-Demand Anodyne NPFFR1 55 38 CS(=O)(=O)c1ccccc1Nc1nc2c(Nc3ccccc3S(C)(=O)=O)cccn2n1 ZINC000147030965 JG Annotated Anodyne JAK2 23 54 Cc1c[nH]c2c(Nc3nc(N[C@@H]4CCCC[C@@H]4N)cc4cn[nH]c(=O)c34)cccc12 ZINC000147030978 HH For-Sale Anodyne SYK 67 79 Cc1c[nH]c2c(Nc3nc(N[C@@H]4CCCC[C@@H]4N)cc4cn[nH]c(=O)c34)cccc12 ZINC000147030978 HH For-Sale Anodyne LYN 18 79 Cc1c[nH]c2c(Nc3nc(N[C@@H]4CCCC[C@@H]4N)cc4cn[nH]c(=O)c34)cccc12 ZINC000147030978 HH For-Sale Anodyne ZAP70 46 79 O=C(Nc1cccc(CNS(=O)(=O)c2cccnc2)c1)[C@@H]1CCCO1 ZINC000147031058 FD On-Demand Anodyne TBXA2R 28 41 O=C(Nc1cccc(CNS(=O)(=O)c2cccnc2)c1)[C@@H]1CCCO1 ZINC000147031058 FD On-Demand Anodyne TBXAS1 52 41 O=C(Nc1cccc(CNS(=O)(=O)c2cccnc2)c1)[C@@H]1CCCO1 ZINC000147031058 FD On-Demand Anodyne NAMPT 71 39 CN(C)/C=C/C(=O)c1cnn2ccccc12 ZINC000147031070 BD For-Sale Mild EPHB3 33 46 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne OPRD1 15 42 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne NPY1R 29 45 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne KLK3 84 38 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne CTSK 48 43 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne CTSL 23 42 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne NPFFR2 40 38 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne C3AR1 55 34 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne MMP3 21 42 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne HLA-DRB1 46 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne PCSK5 41 34 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne FURIN 54 31 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne CAPN2 49 36 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne POLG_WNV 83 35 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031114 ED On-Demand Anodyne NPFFR1 55 38 COc1ccc(C=C2CCN(C(=O)OCc3ccccc3)CC2)cc1[N+](=O)[O-] ZINC000147031246 GI For-Sale Bother TGM2 33 40 COc1ccc(C=C2CCN(C(=O)OCc3ccccc3)CC2)cc1[N+](=O)[O-] ZINC000147031246 GI For-Sale Bother F13A1 52 40 COc1ccc(C=C2CCN(C(=O)OCc3ccccc3)CC2)cc1[N+](=O)[O-] ZINC000147031246 GI For-Sale Bother SLC12A5 51 36 O=C(Nc1cccc(CNS(=O)(=O)c2cccnc2)c1)[C@H]1CCCO1 ZINC000147031252 FD On-Demand Anodyne TBXA2R 28 41 O=C(Nc1cccc(CNS(=O)(=O)c2cccnc2)c1)[C@H]1CCCO1 ZINC000147031252 FD On-Demand Anodyne TBXAS1 52 41 O=C(Nc1cccc(CNS(=O)(=O)c2cccnc2)c1)[C@H]1CCCO1 ZINC000147031252 FD On-Demand Anodyne NAMPT 71 39 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031320 ED On-Demand Anodyne KLK3 84 38 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031320 ED On-Demand Anodyne CTSK 48 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031320 ED On-Demand Anodyne NPFFR2 40 38 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031320 ED On-Demand Anodyne C3AR1 55 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031320 ED On-Demand Anodyne MMP3 21 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031320 ED On-Demand Anodyne HLA-DRB1 46 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031320 ED On-Demand Anodyne PCSK5 41 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031320 ED On-Demand Anodyne FURIN 54 31 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031320 ED On-Demand Anodyne CAPN2 49 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031320 ED On-Demand Anodyne POLG_WNV 83 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC(=O)OC)c1ccccc1 ZINC000147031320 ED On-Demand Anodyne NPFFR1 55 38 O=C(NCCN1CCCCC1)c1cccnc1SC(F)(F)F ZINC000147031338 EF On-Demand Anodyne DRD4 40 31 O=C(NCCN1CCCCC1)c1cccnc1SC(F)(F)F ZINC000147031338 EF On-Demand Anodyne HNMT 44 35 O=C(NCCN1CCCCC1)c1cccnc1SC(F)(F)F ZINC000147031338 EF On-Demand Anodyne PLD2 46 33 O=C(NCCN1CCCCC1)c1cccnc1SC(F)(F)F ZINC000147031338 EF On-Demand Anodyne POLR1A 15 43 c1ccc(CNCCOc2ccccc2Cc2ccccc2)cc1 ZINC000147031406 DI For-Sale Anodyne ADRA1D 17 66 c1ccc(CNCCOc2ccccc2Cc2ccccc2)cc1 ZINC000147031406 DI For-Sale Anodyne ADRA1B 16 66 c1ccc(CNCCOc2ccccc2Cc2ccccc2)cc1 ZINC000147031406 DI For-Sale Anodyne DRD5 19 56 c1ccc(CNCCOc2ccccc2Cc2ccccc2)cc1 ZINC000147031406 DI For-Sale Anodyne SLC5A4 52 38 NC(=O)Nc1cc([N+](=O)[O-])ccc1F ZINC000147031479 AD For-Sale Bother KCNMA1 41 45 NC(=O)Nc1cc([N+](=O)[O-])ccc1F ZINC000147031479 AD For-Sale Bother WDR5 36 42 COC(=O)c1sccc1NC(=O)[C@H](C)Cc1cccc(F)c1 ZINC000147031519 DG On-Demand Anodyne FAS 47 48 CCC[C@@H](NC(=O)NCc1ccc(F)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147031583 FF On-Demand Mild P2RY12 51 33 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)NC2CCCCC2)cc1 ZINC000147031592 GG On-Demand Anodyne EPHX2 22 40 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(C(=O)NC2CCCCC2)cc1 ZINC000147031592 GG On-Demand Anodyne PLAU 17 40 CSc1nc(Nc2ccc3ccccc3c2)nc(SC)n1 ZINC000147031702 DI For-Sale Anodyne TERT 20 49 N#Cc1ccccc1Oc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1 ZINC000147031843 GH On-Demand Anodyne ADRB1 47 38 N#Cc1ccccc1Oc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1 ZINC000147031843 GH On-Demand Anodyne PFKFB3 57 36 C[C@@H]1[C@@H](O)c2cc3c(cc2[C@H](c2ccc4c(c2)OCO4)[C@H]1C)OCO3 ZINC000147031882 EH Annotated Anodyne EDNRB 32 43 C[C@@H]1[C@@H](O)c2cc3c(cc2[C@H](c2ccc4c(c2)OCO4)[C@H]1C)OCO3 ZINC000147031882 EH Annotated Anodyne EDNRA 45 35 N=C(N)c1ccc2c(c1)[C@@H]1c3ccccc3CC[C@H]1[C@@H](c1ccc(O)cc1Cl)N2 ZINC000147032026 HK For-Sale Anodyne F7 15 48 CC(C)Oc1cccc(CC(=O)N(C)[C@@H](C)c2nc3ccccc3s2)c1 ZINC000147032308 FJ On-Demand Anodyne CSNK1D 25 42 N#CC1CCN(C(=O)[C@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032390 FD On-Demand Mild FKBP1A 31 48 N#CC1CCN(C(=O)[C@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032390 FD On-Demand Mild MMP13 16 41 N#CC1CCN(C(=O)[C@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032390 FD On-Demand Mild ITGA4 32 43 N#CC1CCN(C(=O)[C@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032390 FD On-Demand Mild PREP 61 42 N#CC1CCN(C(=O)[C@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032390 FD On-Demand Mild CAPNS1 15 40 N#CC1CCN(C(=O)[C@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032390 FD On-Demand Mild MMP3 15 41 N#CC1CCN(C(=O)[C@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032390 FD On-Demand Mild MMP7 28 41 N#CC1CCN(C(=O)[C@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032390 FD On-Demand Mild SFRP1 78 38 N#CC1CCN(C(=O)[C@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032390 FD On-Demand Mild WNT3 68 38 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(S(C)(=O)=O)nc2)c1 ZINC000147032523 FD On-Demand Bother TAAR1 26 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(S(C)(=O)=O)nc2)c1 ZINC000147032523 FD On-Demand Bother AKR1C2 42 38 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(S(C)(=O)=O)nc2)c1 ZINC000147032523 FD On-Demand Bother USP7 40 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(S(C)(=O)=O)nc2)c1 ZINC000147032523 FD On-Demand Bother USP47 50 44 N#CC1CCN(C(=O)[C@@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032586 FD On-Demand Mild FKBP1A 31 48 N#CC1CCN(C(=O)[C@@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032586 FD On-Demand Mild MMP13 16 41 N#CC1CCN(C(=O)[C@@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032586 FD On-Demand Mild ITGA4 32 43 N#CC1CCN(C(=O)[C@@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032586 FD On-Demand Mild PREP 61 42 N#CC1CCN(C(=O)[C@@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032586 FD On-Demand Mild CAPNS1 15 40 N#CC1CCN(C(=O)[C@@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032586 FD On-Demand Mild MMP3 15 41 N#CC1CCN(C(=O)[C@@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032586 FD On-Demand Mild MMP7 28 41 N#CC1CCN(C(=O)[C@@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032586 FD On-Demand Mild SFRP1 78 38 N#CC1CCN(C(=O)[C@@H]2CCCCN2S(=O)(=O)c2ccccc2)CC1 ZINC000147032586 FD On-Demand Mild WNT3 68 38 O=C(O)[C@@H]1CCCN1C(=O)c1cnc2ccccc2c1 ZINC000147032674 CD For-Sale Anodyne ACE 52 53 O=C(O)[C@@H]1CCCN1C(=O)c1cnc2ccccc2c1 ZINC000147032674 CD For-Sale Anodyne COLA 64 36 O=C(O)[C@@H]1CCCN1C(=O)c1cnc2ccccc2c1 ZINC000147032674 CD For-Sale Anodyne CPT1A 61 36 O=C(O)[C@@H]1CCCN1C(=O)c1cnc2ccccc2c1 ZINC000147032674 CD For-Sale Anodyne PREP 107 47 O=C(O)[C@@H]1CCCN1C(=O)c1cnc2ccccc2c1 ZINC000147032674 CD For-Sale Anodyne SFRP1 43 36 O=C(O)[C@@H]1CCCN1C(=O)c1cnc2ccccc2c1 ZINC000147032674 CD For-Sale Anodyne WNT3 45 36 COc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1F ZINC000147032771 HE On-Demand Anodyne CCR4 20 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne F2 20 46 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne NPY1R 27 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne PCSK2 0 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne GRIA1 41 33 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne PCSK7 0 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne PCSK5 62 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne FURIN 84 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne PCSK1 0 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne F7 22 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne PCSK6 0 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne DPP7 65 36 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne PROC 69 46 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne L3MBTL3 43 34 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147032846 FE On-Demand Anodyne TMPRSS11D 61 34 COc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1F ZINC000147032943 HE On-Demand Anodyne CCR4 20 41 Cc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)[nH]n2)cc1 ZINC000147033017 CF On-Demand Mild TACR3 23 54 CC(C)(C)OC(=O)N/C(=C\c1ccccc1)C(=O)O ZINC000147033049 CF For-Sale Anodyne TLR4 34 47 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne F2 20 46 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne NPY1R 27 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne PCSK2 0 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne GRIA1 41 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne PCSK7 0 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne PCSK5 62 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne FURIN 84 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne PCSK1 0 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne F7 22 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne PCSK6 0 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne DPP7 65 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne PROC 69 46 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne L3MBTL3 43 34 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147033050 FE On-Demand Anodyne TMPRSS11D 61 34 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCCCC3)c2)cc1 ZINC000147033057 FF On-Demand Anodyne ACHE 15 48 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCCCC3)c2)cc1 ZINC000147033057 FF On-Demand Anodyne HRH2 60 50 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCCCC3)c2)cc1 ZINC000147033057 FF On-Demand Anodyne LTA4H 47 43 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCCCC3)c2)cc1 ZINC000147033057 FF On-Demand Anodyne HRH3 22 43 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCCCC3)c2)cc1 ZINC000147033057 FF On-Demand Anodyne CCR3 33 41 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCCCC3)c2)cc1 ZINC000147033057 FF On-Demand Anodyne FAAH 27 41 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCCCC3)c2)cc1 ZINC000147033057 FF On-Demand Anodyne MCHR1 39 42 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCCCC3)c2)cc1 ZINC000147033057 FF On-Demand Anodyne HIF1A 26 45 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCCCC3)c2)cc1 ZINC000147033057 FF On-Demand Anodyne PSMB2 40 34 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCCCC3)c2)cc1 ZINC000147033057 FF On-Demand Anodyne NPFFR1 59 38 Cc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1Cl ZINC000147033131 HG On-Demand Anodyne ST14 45 32 Nc1nc(CC[C@@H]2CCCN2)cc(-c2c[nH]c3ncccc23)n1 ZINC000147033221 DE For-Sale Anodyne CDC7 36 42 Nc1nc(CC[C@@H]2CCCN2)cc(-c2c[nH]c3ncccc23)n1 ZINC000147033221 DE For-Sale Anodyne RET 18 40 CC(C)(C)OC(=O)N/C(=C/c1ccccc1)C(=O)O ZINC000147033244 CF For-Sale Anodyne NS5B 39 45 CC(C)(C)OC(=O)N/C(=C/c1ccccc1)C(=O)O ZINC000147033244 CF For-Sale Anodyne TLR4 34 47 CC1(C)OC(=O)N(c2ccc3c(c2)CCNC3=O)[C@H]1c1ccccc1 ZINC000147033245 EG For-Sale Anodyne TNKS 49 36 O=C(N[C@H](COc1ccccc1F)c1ccccc1)c1ccc2c(c1)COC2 ZINC000147033345 GI On-Demand Anodyne CTSA 43 35 CCNC(=O)c1ccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147033370 HD On-Demand Bother CA2 25 45 CCNC(=O)c1ccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147033370 HD On-Demand Bother MAPK9 38 40 CCNC(=O)c1ccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147033370 HD On-Demand Bother MAPK8 31 43 CCNC(=O)c1ccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147033370 HD On-Demand Bother NAMPT 45 36 COc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)c1 ZINC000147033382 GG On-Demand Anodyne DRD4 40 31 COc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)c1 ZINC000147033382 GG On-Demand Anodyne RAF1 32 45 COc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)c1 ZINC000147033382 GG On-Demand Anodyne MTNR1A 41 54 COc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)c1 ZINC000147033382 GG On-Demand Anodyne MTNR1B 43 54 COc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)c1 ZINC000147033382 GG On-Demand Anodyne PFKFB3 54 33 Nc1nc(CC[C@H]2CCCN2)cc(-c2c[nH]c3ncccc23)n1 ZINC000147033419 DE For-Sale Anodyne CDC7 36 42 Nc1nc(CC[C@H]2CCCN2)cc(-c2c[nH]c3ncccc23)n1 ZINC000147033419 DE For-Sale Anodyne RET 18 40 Cc1cc(N2CCOCC2)ccc1NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147033458 HG On-Demand Anodyne DRTS_PLAFK 18 40 CC[C@@H]1CCCN(C(=O)COc2ccc(C(N)=O)cc2)C1 ZINC000147033522 CD On-Demand Anodyne GRM3 15 50 CC[C@@H]1CCCN(C(=O)COc2ccc(C(N)=O)cc2)C1 ZINC000147033522 CD On-Demand Anodyne CHEK2 44 39 CC[C@@H]1CCCN(C(=O)COc2ccc(C(N)=O)cc2)C1 ZINC000147033522 CD On-Demand Anodyne CPT1A 63 41 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne CNR1 45 69 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne PPARA 23 45 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne FABP4 23 62 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne PLA2G4A 26 53 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne LPAR1 33 41 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne LPAR2 15 51 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne FAAH 52 63 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne PRKCA 28 55 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne EPHX2 34 48 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne LPAR3 57 51 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne FABP3 58 62 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne FABP5 16 53 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne LOX1.1 15 62 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne MGLL 19 61 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne FFAR1 28 62 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne ENPP2 26 50 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne FABP1 17 53 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne OXER1 22 47 CCCCC/C=C/C/C=C/C/C=C/CCCCC(=O)OCC ZINC000147033550 DK In-Stock Anodyne CQSS 54 35 COc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)c1 ZINC000147033581 GG On-Demand Anodyne DRD4 40 31 COc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)c1 ZINC000147033581 GG On-Demand Anodyne RAF1 32 45 COc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)c1 ZINC000147033581 GG On-Demand Anodyne MTNR1A 41 54 COc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)c1 ZINC000147033581 GG On-Demand Anodyne MTNR1B 43 54 COc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)c1 ZINC000147033581 GG On-Demand Anodyne PFKFB3 54 33 C[C@@H]1CCCCN1CCNC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147033629 FD On-Demand Bother HRH3 22 40 CCN(CC)CC(=O)Nc1ccc(N2CCOCC2)cc1C ZINC000147033665 DE On-Demand Anodyne HRH3 15 45 CCN(CC)CC(=O)Nc1ccc(N2CCOCC2)cc1C ZINC000147033665 DE On-Demand Anodyne TTK 17 42 CCN(CC)CC(=O)Nc1ccc(N2CCOCC2)cc1C ZINC000147033665 DE On-Demand Anodyne AKR1C3 22 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne NPY1R 26 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne KLK3 46 38 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne CTSK 44 44 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne NPFFR2 42 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne C3AR1 59 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne PCSK5 54 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne FURIN 58 34 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne CAPN2 51 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne ACE2 41 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne POLG_WNV 75 34 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne QRFPR 42 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033671 DF On-Demand Anodyne NPFFR1 57 40 CC[C@H]1CCCN(C(=O)COc2ccc(C(N)=O)cc2)C1 ZINC000147033693 CD On-Demand Anodyne GRM3 15 50 CC[C@H]1CCCN(C(=O)COc2ccc(C(N)=O)cc2)C1 ZINC000147033693 CD On-Demand Anodyne CHEK2 44 39 CC[C@H]1CCCN(C(=O)COc2ccc(C(N)=O)cc2)C1 ZINC000147033693 CD On-Demand Anodyne CPT1A 63 41 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne PTGER2 26 52 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne TBXA2R 15 45 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne TBXAS1 47 39 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne MMP13 39 54 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne ADAM17 20 54 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne MMP2 20 46 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne MMP3 20 46 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne MMP8 25 46 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne PLA2G4B 40 33 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne PTPN1 18 40 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne MMP9 40 54 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne MMP12 18 45 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne CXCR3 34 59 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne MMP1 33 45 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne DAGLA 36 43 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne TRPM8 54 42 CCOc1ccc(S(=O)(=O)N(Cc2ccc(C(=O)O)cc2)Cc2cccnc2)cc1 ZINC000147033713 IH For-Sale Anodyne NAMPT 45 45 C=CCN(C)S(=O)(=O)c1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147033738 HF On-Demand Mild BMP1 75 37 C=CCN(C)S(=O)(=O)c1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147033738 HF On-Demand Mild MMP3 33 40 C=CCN(C)S(=O)(=O)c1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147033738 HF On-Demand Mild MMP8 31 40 C=CCN(C)S(=O)(=O)c1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147033738 HF On-Demand Mild ROCK2 32 52 O=C(O)N1CCc2ccccc2[C@H]1c1ccc(Cl)cc1 ZINC000147033801 CH For-Sale Anodyne TRPM8 51 50 C[C@H]1CCCCN1CCNC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147033823 FD On-Demand Bother HRH3 22 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne NPY1R 26 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne KLK3 46 38 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne CTSK 44 44 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne NPFFR2 42 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne C3AR1 59 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne PCSK5 54 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne FURIN 58 34 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne CAPN2 51 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne ACE2 41 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne POLG_WNV 75 34 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne QRFPR 42 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](CC)c1ccccc1 ZINC000147033859 DF On-Demand Anodyne NPFFR1 57 40 CCOC(=O)NCC(=O)Nc1ccc(N2CCOCC2)cc1C ZINC000147033878 DD On-Demand Anodyne PRKDC 40 36 O=C(Nc1cccc(-n2ccnc2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147033960 FH On-Demand Anodyne MAPK10 17 41 O=C(Nc1cccc(-n2ccnc2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147033960 FH On-Demand Anodyne CSF1R 21 40 O=C(Nc1cccc(-n2ccnc2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147033960 FH On-Demand Anodyne DDR1 15 47 O=C(Nc1cccc(-n2ccnc2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147033960 FH On-Demand Anodyne KCNK3 50 35 O=C(O)N1CCc2ccccc2[C@@H]1c1ccc(Cl)cc1 ZINC000147033989 CH For-Sale Anodyne TRPM8 51 50 CCCC[C@@H](N)S(=O)(=O)O ZINC000147033993 AC For-Sale Anodyne ANPEP 0 41 CCCC[C@@H](N)S(=O)(=O)O ZINC000147033993 AC For-Sale Anodyne GCLC 49 30 CCCC[C@@H](N)S(=O)(=O)O ZINC000147033993 AC For-Sale Anodyne DPP7 0 45 CCOC(=O)c1[nH]ccc1O ZINC000147034014 AC For-Sale Anodyne CA14 0 53 CCOC(=O)c1[nH]ccc1O ZINC000147034014 AC For-Sale Anodyne HISB 0 43 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne NPY1R 35 43 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne KLK3 46 38 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne CTSK 44 44 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne CTSL 17 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne NPFFR2 42 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne C3AR1 59 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne PCSK5 54 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne FURIN 58 34 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne CAPN2 51 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne ACE2 41 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne POLG_WNV 75 34 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne QRFPR 42 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034050 DF On-Demand Anodyne NPFFR1 57 40 Cc1cc(N2CCOCC2)ccc1NC(=O)CCNS(C)(=O)=O ZINC000147034104 EC On-Demand Anodyne PRKDC 44 34 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne PTGER2 22 43 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne TBXA2R 18 49 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne TBXAS1 52 46 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne MMP13 15 44 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne MMP8 15 40 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne MMP9 22 44 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne CXCR3 23 47 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne MMP1 20 42 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne DAGLA 24 47 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne TRPM8 47 36 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne NAMPT 39 44 CCOC(=O)c1ccc(CN(Cc2cccnc2)S(=O)(=O)c2ccc(Cl)cc2)cc1 ZINC000147034140 II For-Sale Anodyne NR1D1 39 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(-n3ccnc3)c1)C2 ZINC000147034150 EG On-Demand Anodyne ROCK2 34 48 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(N2CCOCC2)c1 ZINC000147034160 ED On-Demand Anodyne TNK2 27 41 CCCC[C@H](N)S(=O)(=O)O ZINC000147034172 AC For-Sale Anodyne ANPEP 0 41 CCCC[C@H](N)S(=O)(=O)O ZINC000147034172 AC For-Sale Anodyne GCLC 49 30 CCCC[C@H](N)S(=O)(=O)O ZINC000147034172 AC For-Sale Anodyne DPP7 0 45 N#CC1CCN(C(=O)C[C@@H](NC(N)=O)c2ccccc2)CC1 ZINC000147034241 DD On-Demand Mild PTAFR 38 45 N#CC1CCN(C(=O)C[C@@H](NC(N)=O)c2ccccc2)CC1 ZINC000147034241 DD On-Demand Mild DPP4 23 42 CCCc1nc(CS(=O)(=O)CC(=O)NCCc2ccccc2OC)no1 ZINC000147034246 GD On-Demand Anodyne MTNR1A 43 39 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne NPY1R 26 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne KLK3 46 38 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne CTSK 44 44 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne NPFFR2 42 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne C3AR1 59 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne PCSK5 54 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne FURIN 58 34 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne CAPN2 51 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne ACE2 41 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne POLG_WNV 75 34 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne QRFPR 42 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](CC)c1ccccc1 ZINC000147034264 DF On-Demand Anodyne NPFFR1 57 40 CCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(SC)cc1 ZINC000147034319 DE On-Demand Anodyne CAPN2 46 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(N2CCOCC2)c1 ZINC000147034366 ED On-Demand Anodyne TNK2 27 41 CCCC(=O)N1CCC(C(C)C)CC1 ZINC000147034398 AF On-Demand Anodyne CPN1 0 40 CCCC(=O)N1CCC(C(C)C)CC1 ZINC000147034398 AF On-Demand Anodyne GNAI1 0 47 CCCC(=O)N1CCC(C(C)C)CC1 ZINC000147034398 AF On-Demand Anodyne GNAI3 0 45 CCCC(=O)N1CCC(C(C)C)CC1 ZINC000147034398 AF On-Demand Anodyne GNAO1 0 45 N#CC1CCN(C(=O)C[C@H](NC(N)=O)c2ccccc2)CC1 ZINC000147034440 DD On-Demand Mild PTAFR 38 45 N#CC1CCN(C(=O)C[C@H](NC(N)=O)c2ccccc2)CC1 ZINC000147034440 DD On-Demand Mild DPP4 23 42 C=C1C[C@@](C)(c2cc(NC(=O)c3ncc(C#N)cc3F)cnc2Cl)N=C(N)S1 ZINC000147034453 HH Annotated Mild BACE2 43 41 C=C1C[C@@](C)(c2cc(NC(=O)c3ncc(C#N)cc3F)cnc2Cl)N=C(N)S1 ZINC000147034453 HH Annotated Mild BACE1 19 43 C[C@@H](Cc1cccc(F)c1)C(=O)N(C)[C@@H](C)c1nc2ccccc2s1 ZINC000147034481 FJ On-Demand Anodyne PIN1 27 41 C=C1C[C@@](C)(c2cncc(NC(=O)c3cnc(OC)cn3)c2)N=C(N)S1 ZINC000147034649 FE Annotated Mild BACE1 0 48 N#CC1CCN(C(=O)c2ccc(NC(N)=O)cc2)CC1 ZINC000147034655 CD On-Demand Mild ACR 41 32 N#CC1CCN(C(=O)c2ccc(NC(N)=O)cc2)CC1 ZINC000147034655 CD On-Demand Mild L3MBTL3 79 42 C[C@@H](c1nc2ccccc2s1)N(C)C(=O)[C@H](C)Cc1cccc(F)c1 ZINC000147034682 FJ On-Demand Anodyne PIN1 27 41 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)CN2CCOCC2)c1 ZINC000147034738 DD On-Demand Bother TAAR1 17 44 O=C(Sc1ccccc1)c1ccc(C(=O)c2ccccc2)cc1 ZINC000147034822 DJ For-Sale Anodyne SRD5A2 18 56 C[C@@H](Cc1cccc(F)c1)C(=O)N(C)[C@H](C)c1nc2ccccc2s1 ZINC000147034860 FJ On-Demand Anodyne PIN1 27 41 CC(C)(C)OC(=O)NCCSc1ccc([N+](=O)[O-])cn1 ZINC000147034917 CF In-Stock Bother PAPA1_CARPA 42 33 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)CN2CCOCC2)c1 ZINC000147034930 DD On-Demand Bother TAAR1 17 44 O=C(CCCc1ccccc1)c1ccccc1C(F)(F)F ZINC000147034957 CJ For-Sale Anodyne PREP 29 40 O=C(CCCc1ccccc1)c1ccccc1C(F)(F)F ZINC000147034957 CJ For-Sale Anodyne FAAH 75 48 O=C(CCCc1ccccc1)c1ccccc1C(F)(F)F ZINC000147034957 CJ For-Sale Anodyne ABCB1 31 41 O=C(CCCc1ccccc1)c1ccccc1C(F)(F)F ZINC000147034957 CJ For-Sale Anodyne CES1 85 50 O=C(CCCc1ccccc1)c1ccccc1C(F)(F)F ZINC000147034957 CJ For-Sale Anodyne MENB 0 44 O=C(CCCc1ccccc1)c1ccccc1C(F)(F)F ZINC000147034957 CJ For-Sale Anodyne EST5_RAT 0 40 O=C(CCCc1ccccc1)c1ccccc1C(F)(F)F ZINC000147034957 CJ For-Sale Anodyne CES1D 45 33 COc1ccc(C=C(C(=O)OC(C)C)C(=O)OC(C)C)cc1 ZINC000147035077 DF For-Sale Anodyne TLR4 38 49 Cc1cc(-n2cccn2)ccc1Br ZINC000147035147 BF For-Sale Anodyne AMP1_PLAFQ 54 39 COCCOc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1F ZINC000147035198 FE On-Demand Anodyne KDR 16 40 COCCOc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1F ZINC000147035198 FE On-Demand Anodyne MET 55 38 C(=C\c1cc(/C=C\c2ccccc2)cc(/C=C\c2ccccc2)c1)\c1ccccc1 ZINC000147035278 GK For-Sale Anodyne CYP1B1 21 48 C(=C\c1cc(/C=C\c2ccccc2)cc(/C=C\c2ccccc2)c1)\c1ccccc1 ZINC000147035278 GK For-Sale Anodyne AHR 61 42 C(=C\c1cc(/C=C\c2ccccc2)cc(/C=C\c2ccccc2)c1)\c1ccccc1 ZINC000147035278 GK For-Sale Anodyne CYP1A1 20 48 CCOC[C@H](C)NC(=O)Nc1cccc(OC2CCCC2)c1 ZINC000147035336 DH On-Demand Anodyne EPHX2 34 42 Cc1cnccc1-c1nc(C)c2c(C)nc3scnc3n12 ZINC000147035382 CG For-Sale Anodyne PDE2A 69 55 Cc1cnccc1-c1nc(C)c2c(C)nc3scnc3n12 ZINC000147035382 CG For-Sale Anodyne PDE7A 24 47 Cc1cnccc1-c1nc(C)c2c(C)nc3scnc3n12 ZINC000147035382 CG For-Sale Anodyne PDE10A 26 55 CC(=O)N[C@@H](CC(=O)N1CCC(C#N)CC1)c1cccs1 ZINC000147035446 DE On-Demand Mild PTAFR 34 45 C(=C\c1cc(/C=C\c2ccccc2)cc(/C=C/c2ccccc2)c1)\c1ccccc1 ZINC000147035464 GK For-Sale Anodyne CYP1B1 21 48 C(=C\c1cc(/C=C\c2ccccc2)cc(/C=C/c2ccccc2)c1)\c1ccccc1 ZINC000147035464 GK For-Sale Anodyne AHR 61 42 C(=C\c1cc(/C=C\c2ccccc2)cc(/C=C/c2ccccc2)c1)\c1ccccc1 ZINC000147035464 GK For-Sale Anodyne CYP1A1 20 48 COc1ccc([N+](=O)[O-])c(C(=O)N(C)CCCc2ccccc2)c1 ZINC000147035489 EG On-Demand Bother AKR1C2 26 43 O=C(NC1CCN(C(=O)Nc2cccc(OC3CCCC3)c2)CC1)c1ccoc1 ZINC000147035531 GI On-Demand Anodyne EPHX2 38 41 COC(=O)c1c(C)ccnc1Br ZINC000147035561 BD For-Sale Anodyne KDM5C 0 40 CCOC(=O)N1CCC(OC(=O)c2cc(C)cc([N+](=O)[O-])c2)CC1 ZINC000147035564 EF On-Demand Bother SLC27A4 45 38 C(=C\c1cc(/C=C/c2ccccc2)cc(/C=C/c2ccccc2)c1)\c1ccccc1 ZINC000147035661 GK For-Sale Anodyne CYP1B1 21 48 C(=C\c1cc(/C=C/c2ccccc2)cc(/C=C/c2ccccc2)c1)\c1ccccc1 ZINC000147035661 GK For-Sale Anodyne AHR 61 42 C(=C\c1cc(/C=C/c2ccccc2)cc(/C=C/c2ccccc2)c1)\c1ccccc1 ZINC000147035661 GK For-Sale Anodyne CYP1A1 20 48 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2cccc(OC(F)F)c2)c1 ZINC000147035741 FH On-Demand Bother TAAR1 24 42 CCCOc1cccc(NC(=O)N[C@@H](C)COCC)c1 ZINC000147035807 CG On-Demand Anodyne ACACA 35 43 CCCOc1cccc(NC(=O)N[C@@H](C)COCC)c1 ZINC000147035807 CG On-Demand Anodyne CCKAR 20 40 CCCOc1cccc(NC(=O)N[C@@H](C)COCC)c1 ZINC000147035807 CG On-Demand Anodyne MTNR1B 24 43 CCCOc1cccc(NC(=O)N[C@@H](C)COCC)c1 ZINC000147035807 CG On-Demand Anodyne EPHX2 19 49 CCCOc1cccc(NC(=O)N[C@@H](C)COCC)c1 ZINC000147035807 CG On-Demand Anodyne PDS 40 35 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2cccc(OC(F)F)c2)c1 ZINC000147035910 FH On-Demand Bother TAAR1 24 42 NC(=O)CNC(=O)OCc1ccc([N+](=O)[O-])cc1 ZINC000147036083 CC For-Sale Bother ACR 17 42 COc1ccc2[nH]cc(CCNCc3cccc(OCC(F)(F)F)c3)c2c1 ZINC000147036143 GI On-Demand Anodyne HTR1A 17 48 COc1ccc2[nH]cc(CCNCc3cccc(OCC(F)(F)F)c3)c2c1 ZINC000147036143 GI On-Demand Anodyne HTR1D 36 47 COc1ccc2[nH]cc(CCNCc3cccc(OCC(F)(F)F)c3)c2c1 ZINC000147036143 GI On-Demand Anodyne HTR1B 34 45 COc1ccc2[nH]cc(CCNCc3cccc(OCC(F)(F)F)c3)c2c1 ZINC000147036143 GI On-Demand Anodyne NQO2 20 49 COc1ccc2[nH]cc(CCNCc3cccc(OCC(F)(F)F)c3)c2c1 ZINC000147036143 GI On-Demand Anodyne MPO 59 44 COc1ccc2[nH]cc(CCNCc3cccc(OCC(F)(F)F)c3)c2c1 ZINC000147036143 GI On-Demand Anodyne HTR1E 15 42 COc1ccc2[nH]cc(CCNCc3cccc(OCC(F)(F)F)c3)c2c1 ZINC000147036143 GI On-Demand Anodyne MTNR1A 43 53 COc1ccc2[nH]cc(CCNCc3cccc(OCC(F)(F)F)c3)c2c1 ZINC000147036143 GI On-Demand Anodyne MTNR1B 32 49 COc1ccc2[nH]cc(CCNCc3cccc(OCC(F)(F)F)c3)c2c1 ZINC000147036143 GI On-Demand Anodyne ABCG2 25 41 CCCOc1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147036196 FJ On-Demand Anodyne HRH2 32 40 CCCOc1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147036196 FJ On-Demand Anodyne EPHX2 28 44 CCCOc1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147036196 FJ On-Demand Anodyne PDS 44 32 COc1cc(OCC(=O)Nc2ncc(Cc3ccc(F)cc3)s2)ccc1[N+](=O)[O-] ZINC000147036236 HH On-Demand Bother SCD1 40 44 COc1cc(OCC(=O)Nc2ncc(Cc3ccc(F)cc3)s2)ccc1[N+](=O)[O-] ZINC000147036236 HH On-Demand Bother SCD 34 44 NC(=O)c1ccc(OCC(=O)Nc2ccc(N3CCNC(=O)C3)nc2)cc1 ZINC000147036314 FC On-Demand Anodyne ADORA2B 40 42 CCCOc1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147036386 FJ On-Demand Anodyne HRH2 32 40 CCCOc1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147036386 FJ On-Demand Anodyne EPHX2 28 44 CCCOc1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147036386 FJ On-Demand Anodyne PDS 44 32 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(OCC(=O)N(C)C)c(OC)c2)c1 ZINC000147036499 HE On-Demand Bother MT-ND1 25 42 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne GYRB 49 33 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne LPL 45 35 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne CA1 23 42 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne FGFR1 16 44 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne CHEK2 17 43 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne P2RY1 17 44 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne KDR 17 44 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne HPSE 30 65 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne NR2E3 67 37 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne SHH 22 46 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne STK33 63 50 O=C(Nc1ccccc1)Nc1ccccc1-c1nc2ccccc2[nH]1 ZINC000147036525 EJ Annotated Anodyne P96878_MYCTU 19 42 CCCOc1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147036556 FJ On-Demand Anodyne HRH2 32 40 CCCOc1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147036556 FJ On-Demand Anodyne EPHX2 28 44 CCCOc1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147036556 FJ On-Demand Anodyne PDS 44 32 O=C(N[C@H](c1ccc(Cl)cc1)c1cccs1)c1ccc2c(c1)COC2 ZINC000147036627 FJ On-Demand Anodyne UTS2 42 31 N#CC1CCN(C(=O)C2CCN(C(=O)c3ccc(C(F)(F)F)cc3)CC2)CC1 ZINC000147036731 GG On-Demand Mild PREP 17 47 N#CC1CCN(C(=O)C2CCN(C(=O)c3ccc(C(F)(F)F)cc3)CC2)CC1 ZINC000147036731 GG On-Demand Mild EPHX2 28 48 N#CC1CCN(C(=O)C2CCN(C(=O)c3ccc(C(F)(F)F)cc3)CC2)CC1 ZINC000147036731 GG On-Demand Mild MLYCD 20 45 N#CC1CCN(C(=O)C2CCN(C(=O)c3ccc(C(F)(F)F)cc3)CC2)CC1 ZINC000147036731 GG On-Demand Mild SFRP1 35 42 N#CC1CCN(C(=O)C2CCN(C(=O)c3ccc(C(F)(F)F)cc3)CC2)CC1 ZINC000147036731 GG On-Demand Mild L3MBTL3 86 42 CCCOc1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147036748 FJ On-Demand Anodyne HRH2 32 40 CCCOc1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147036748 FJ On-Demand Anodyne EPHX2 28 44 CCCOc1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147036748 FJ On-Demand Anodyne PDS 44 32 Cn1cc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1C(N)=O ZINC000147036829 HC On-Demand Anodyne ST14 48 35 CCCCCCCc1ccc(OC(=O)c2ccc(C3CCC(CC)CC3)cc2)cc1 ZINC000147036936 HK Annotated Mild INHA 65 34 CCCCCCCc1ccc(OC(=O)c2ccc(C3CCC(CC)CC3)cc2)cc1 ZINC000147036936 HK Annotated Mild RARB 19 42 CCCCCCCc1ccc(OC(=O)c2ccc(C3CCC(CC)CC3)cc2)cc1 ZINC000147036936 HK Annotated Mild S1PR3 41 35 CCCCCCCc1ccc(OC(=O)c2ccc(C3CCC(CC)CC3)cc2)cc1 ZINC000147036936 HK Annotated Mild PLA2G4B 40 32 CCCCCCCc1ccc(OC(=O)c2ccc(C3CCC(CC)CC3)cc2)cc1 ZINC000147036936 HK Annotated Mild CFTR 40 35 CCCCCCCc1ccc(OC(=O)c2ccc(C3CCC(CC)CC3)cc2)cc1 ZINC000147036936 HK Annotated Mild S1PR2 43 38 CCCCCCCc1ccc(OC(=O)c2ccc(C3CCC(CC)CC3)cc2)cc1 ZINC000147036936 HK Annotated Mild ACR 48 34 CCCOCCOc1ccc(CO)cc1OCC ZINC000147036991 CE For-Sale Anodyne DRTS_PLAFK 20 41 Cn1cc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1C(N)=O ZINC000147037016 HC On-Demand Anodyne ST14 48 35 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne ALOX5 17 43 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne P2RY12 46 34 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne NPR1 46 37 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne NPFFR2 40 36 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne C3AR1 46 33 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne MTNR1A 38 48 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne MTNR1B 27 42 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne GRIA1 56 33 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne PCSK5 56 38 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne FURIN 61 36 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne PLM2_PLAFA 17 43 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne POLG_WNV 85 40 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne QRFPR 41 39 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne F2RL1 46 39 CCCC[C@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037176 EF On-Demand Anodyne NPFFR1 53 36 COc1ccccc1Oc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1F ZINC000147037223 HI On-Demand Anodyne KDR 26 44 COc1ccccc1Oc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1F ZINC000147037223 HI On-Demand Anodyne MST1R 49 37 COc1ccccc1Oc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1F ZINC000147037223 HI On-Demand Anodyne MET 110 43 COc1ccccc1Oc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1F ZINC000147037223 HI On-Demand Anodyne ENPP1 61 31 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147037282 JI For-Sale Bother IGF1R 32 41 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147037282 JI For-Sale Bother SLC2A1 16 41 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147037282 JI For-Sale Bother ZAP70 31 43 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147037282 JI For-Sale Bother CDK4 26 41 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147037282 JI For-Sale Bother MAPK7 61 41 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147037282 JI For-Sale Bother DYRK1B 31 58 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147037282 JI For-Sale Bother DCLK2 20 41 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147037282 JI For-Sale Bother DCLK1 18 41 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne ALOX5 17 43 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne P2RY12 46 34 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne NPR1 46 37 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne NPFFR2 40 36 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne C3AR1 46 33 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne MTNR1A 38 48 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne MTNR1B 27 42 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne GRIA1 56 33 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne PCSK5 56 38 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne FURIN 61 36 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne CAPN2 28 40 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne PLM2_PLAFA 17 43 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne POLG_WNV 85 40 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne QRFPR 41 39 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne F2RL1 46 39 CCCC[C@@H](NC(N)=O)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147037358 EF On-Demand Anodyne NPFFR1 53 36 N#CC1CCN(C(=O)CCn2cnc3sccc3c2=O)CC1 ZINC000147037370 DD On-Demand Mild ETHR 41 32 O=C(NCCC(c1ccccc1)c1ccccc1)c1ccnc(O)c1 ZINC000147037388 EH On-Demand Anodyne EPHX2 22 68 O=C(NCCC(c1ccccc1)c1ccccc1)c1ccnc(O)c1 ZINC000147037388 EH On-Demand Anodyne KDM4E 28 49 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(OC)cc1C(F)(F)F)C2 ZINC000147037417 GH On-Demand Anodyne MTNR1A 18 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(OC)cc1C(F)(F)F)C2 ZINC000147037417 GH On-Demand Anodyne ROCK2 37 51 COc1cc(C)ccc1Oc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1F ZINC000147037425 HI On-Demand Anodyne KDR 21 41 COc1cc(C)ccc1Oc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1F ZINC000147037425 HI On-Demand Anodyne MET 87 41 COc1cc(C)ccc1Oc1ccc(NC(=O)C[C@]2(C(=O)O)CCSC2)cc1F ZINC000147037425 HI On-Demand Anodyne ENPP1 59 30 O=C(Nc1ccc(CN2C(=O)CCC2=O)cc1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147037453 FG On-Demand Anodyne EPHX2 33 44 N#CC1CCN(C(=O)c2cccc(N3CCCS3(=O)=O)c2)CC1 ZINC000147037574 ED On-Demand Mild PREP 18 41 N#CC1CCN(C(=O)c2cccc(N3CCCS3(=O)=O)c2)CC1 ZINC000147037574 ED On-Demand Mild L3MBTL3 50 43 CCCc1nc(CS(=O)(=O)C[C@@H](O)COc2ccc(-c3ccccc3)cc2)no1 ZINC000147037575 HG On-Demand Anodyne ADAMTS4 42 35 COc1ccc([N+](=O)[O-])cc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147037590 ED On-Demand Bother KCNMA1 20 45 O=C(Nc1ccc(CN2C(=O)CCC2=O)cc1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147037620 FG On-Demand Anodyne EPHX2 33 44 Cc1cnccc1-c1cccc(O)c1 ZINC000147037638 AF For-Sale Anodyne CYP11B2 15 45 Cc1cnccc1-c1cccc(O)c1 ZINC000147037638 AF For-Sale Anodyne HSD17B1 58 46 Cc1cnccc1-c1cccc(O)c1 ZINC000147037638 AF For-Sale Anodyne CYP17A1 16 48 Cc1cnccc1-c1cccc(O)c1 ZINC000147037638 AF For-Sale Anodyne HSD17B2 41 43 C[C@H]1CCCN(Cc2ccc(NC(=O)c3ccc4c(c3)COC4)cc2)C1 ZINC000147037658 FI On-Demand Anodyne MLNR 47 33 C[C@H]1CCCN(Cc2ccc(NC(=O)c3ccc4c(c3)COC4)cc2)C1 ZINC000147037658 FI On-Demand Anodyne CCR2 18 40 C[C@H]1CCCN(Cc2ccc(NC(=O)c3ccc4c(c3)COC4)cc2)C1 ZINC000147037658 FI On-Demand Anodyne MCHR1 28 45 C[C@H]1CCCN(Cc2ccc(NC(=O)c3ccc4c(c3)COC4)cc2)C1 ZINC000147037658 FI On-Demand Anodyne NOD1 32 41 C[C@H]1CCCN(Cc2ccc(NC(=O)c3ccc4c(c3)COC4)cc2)C1 ZINC000147037658 FI On-Demand Anodyne NOD2 48 41 COc1ccc([N+](=O)[O-])cc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147037779 ED On-Demand Bother KCNMA1 20 45 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne ALOX5 16 44 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne NPY1R 27 41 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne KLK3 67 38 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne CTSB 22 44 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne PAPA1_CARPA 44 36 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne CTSK 57 39 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne CTSL 36 40 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne SCN2A 22 45 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne NPFFR2 46 42 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne C3AR1 66 38 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne MMP3 33 41 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne GRIA1 83 37 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne PLA2G4B 69 37 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne HLA-DRB1 41 39 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne FAAH 27 42 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne PCSK5 63 44 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne FURIN 85 41 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne CTSS 20 50 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne CAPN2 63 44 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne ACE2 54 37 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne MC1R 44 31 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne ST14 48 34 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne CTRB_BOVIN 46 32 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne AMP1_PLAFQ 25 43 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne KISS1R 46 31 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne POLG_WNV 94 45 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne QRFPR 57 46 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne F2RL1 52 35 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne NPFFR1 63 42 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne NOD1 67 34 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne TMPRSS11D 45 35 CCCC[C@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037798 DD On-Demand Anodyne HPN 57 34 O=C(Nc1ccc(CN2C(=O)CCC2=O)cc1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147037807 FG On-Demand Anodyne EPHX2 33 44 CCC(=O)Nc1ccc(Cl)c(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147037923 GH On-Demand Anodyne MTNR1A 30 41 CCC(=O)Nc1ccc(Cl)c(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147037923 GH On-Demand Anodyne MTNR1B 29 41 CCC(=O)Nc1ccc(Cl)c(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147037923 GH On-Demand Anodyne ROCK2 34 46 Cc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1C(N)=O ZINC000147037963 HD On-Demand Anodyne ST14 45 33 COc1ccc([N+](=O)[O-])cc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147037971 ED On-Demand Bother KCNMA1 20 45 O=C(Nc1ccc(CN2C(=O)CCC2=O)cc1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147037976 FG On-Demand Anodyne EPHX2 33 44 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne ALOX5 16 44 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne NPY1R 27 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne KLK3 67 38 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne CTSB 22 44 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne PAPA1_CARPA 44 36 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne CTSK 57 39 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne CTSL 36 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne SCN2A 22 45 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne NPFFR2 46 42 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne C3AR1 66 38 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne MMP3 33 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne GRIA1 83 37 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne PLA2G4B 69 37 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne HLA-DRB1 41 39 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne FAAH 27 42 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne PCSK5 63 44 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne FURIN 85 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne CTSS 20 50 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne CAPN2 63 44 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne ACE2 54 37 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne MC1R 44 31 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne ST14 48 34 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne CTRB_BOVIN 46 32 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne AMP1_PLAFQ 25 43 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne KISS1R 46 31 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne POLG_WNV 94 45 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne QRFPR 57 46 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne F2RL1 52 35 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne NPFFR1 63 42 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne NOD1 67 34 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne TMPRSS11D 45 35 CCCC[C@@H](NC(N)=O)C(=O)NCCCOc1ccccc1 ZINC000147037998 DD On-Demand Anodyne HPN 57 34 COc1ccc([N+](=O)[O-])cc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147038161 ED On-Demand Bother KCNMA1 20 45 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(CN3C(=O)CCC3=O)cc2)C1 ZINC000147038166 HC On-Demand Anodyne CCR3 26 41 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(CN3C(=O)CCC3=O)cc2)C1 ZINC000147038166 HC On-Demand Anodyne EPHX2 39 46 Cc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1C(N)=O ZINC000147038173 HD On-Demand Anodyne ST14 45 33 Cc1cc(NC(=O)c2ccco2)sc1C(=O)N1CCC(C#N)CC1 ZINC000147038258 EG On-Demand Mild KISS1R 46 32 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccnc(Oc3ccccc3)c2)c1 ZINC000147038328 GH On-Demand Bother TAAR1 19 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccnc(Oc3ccccc3)c2)c1 ZINC000147038328 GH On-Demand Bother AKR1C2 15 42 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccc(CN3C(=O)CCC3=O)cc2)C1 ZINC000147038366 HC On-Demand Anodyne CCR3 26 41 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccc(CN3C(=O)CCC3=O)cc2)C1 ZINC000147038366 HC On-Demand Anodyne EPHX2 39 46 COC(=O)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147038470 HE On-Demand Anodyne KCNA5 19 51 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(CCN2CCOCC2)cc1 ZINC000147038533 GD On-Demand Anodyne CASR 41 35 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(CCN2CCOCC2)cc1 ZINC000147038533 GD On-Demand Anodyne PIK3CA 21 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(CCN2CCOCC2)cc1 ZINC000147038533 GD On-Demand Anodyne MTOR 45 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(CCN2CCOCC2)cc1 ZINC000147038533 GD On-Demand Anodyne EPHX2 24 45 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(CCN2CCOCC2)cc1 ZINC000147038533 GD On-Demand Anodyne L3MBTL3 25 43 CCO[C@@H]1CCCN(C(=O)Nc2ccc(CN3C(=O)CCC3=O)cc2)C1 ZINC000147038576 FE On-Demand Anodyne TIMP3 55 32 CCO[C@@H]1CCCN(C(=O)Nc2ccc(CN3C(=O)CCC3=O)cc2)C1 ZINC000147038576 FE On-Demand Anodyne EPHX2 23 44 COC(=O)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147038672 HE On-Demand Anodyne KCNA5 19 51 N#Cc1cccc(/C=C\C(=O)N2CCC[C@@H]2CN2CCCCC2)c1 ZINC000147038701 DG On-Demand Mild DPP4 15 44 N#Cc1cccc(/C=C\C(=O)N2CCC[C@@H]2CN2CCCCC2)c1 ZINC000147038701 DG On-Demand Mild UTS2R 43 29 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(CCN2CCOCC2)cc1 ZINC000147038702 GD On-Demand Anodyne CASR 41 35 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(CCN2CCOCC2)cc1 ZINC000147038702 GD On-Demand Anodyne PIK3CA 21 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(CCN2CCOCC2)cc1 ZINC000147038702 GD On-Demand Anodyne MTOR 45 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(CCN2CCOCC2)cc1 ZINC000147038702 GD On-Demand Anodyne EPHX2 24 45 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(CCN2CCOCC2)cc1 ZINC000147038702 GD On-Demand Anodyne L3MBTL3 25 43 COc1cc(OCC(=O)Nc2cc(C(C)(C)C)nn2C)ccc1[N+](=O)[O-] ZINC000147038727 FF On-Demand Bother MAPK14 19 45 CCO[C@H]1CCCN(C(=O)Nc2ccc(CN3C(=O)CCC3=O)cc2)C1 ZINC000147038756 FE On-Demand Anodyne TIMP3 55 32 CCO[C@H]1CCCN(C(=O)Nc2ccc(CN3C(=O)CCC3=O)cc2)C1 ZINC000147038756 FE On-Demand Anodyne EPHX2 23 44 O=C(Nc1nc(-c2sccc2Br)cs1)c1ccc2c(c1)COC2 ZINC000147038908 HJ On-Demand Anodyne MPL 53 36 N#Cc1cccc(/C=C\C(=O)N2CCC[C@H]2CN2CCCCC2)c1 ZINC000147038909 DG On-Demand Mild UTS2R 43 29 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne DRD2 17 43 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne HRH2 39 50 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne HTR2A 26 59 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne HTR2C 16 59 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne DRD5 18 41 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne LTA4H 31 48 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne KIT 23 46 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne HTR7 15 42 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne LCK 33 44 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne MAPK14 15 44 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne HRH3 21 51 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne CCR3 19 42 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne CHRNA7 27 41 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne FLT1 15 46 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne KDR 34 49 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne ABCB1 20 44 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne MET 42 41 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne MTTP 56 41 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne CCR2 35 41 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne EPHX2 34 52 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne LYN 22 40 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne GALR3 24 48 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne TEK 36 41 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne MCHR1 23 47 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne BTK 22 42 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne BRAF 38 42 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne TAAR1 28 40 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne PSMB2 46 35 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne PSMB1 40 36 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne HCN1 71 37 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne HCN4 53 36 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne KCNK3 75 51 O=C(Nc1cccc(C(F)(F)F)c1)c1ccccc1OCCN1CCCCC1 ZINC000147038919 GJ Annotated Anodyne KCNK9 66 51 COc1ccc2nc(C(=O)N3CCC(C#N)CC3)ccc2c1 ZINC000147038922 CF On-Demand Mild TRPC6 46 41 COc1ccc2nc(C(=O)N3CCC(C#N)CC3)ccc2c1 ZINC000147038922 CF On-Demand Mild TRPC3 21 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(-c3cc(F)ccc3OC)cs2)c1 ZINC000147038935 HI On-Demand Bother GCK 15 48 CC(C)Cc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147038949 HG On-Demand Anodyne KCNA5 16 46 CC(C)Cc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147038949 HG On-Demand Anodyne ST14 42 31 O=C(Cc1ccc(Cl)cc1)N1CCN(C(=O)c2ccc3c(c2)COC3)CC1 ZINC000147039112 GF On-Demand Anodyne KCNJ1 51 36 COCCNS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147039127 FC On-Demand Mild L3MBTL3 55 36 CCCc1nc(CS(=O)(=O)C[C@@H](O)COc2ccc(C(C)(C)C)cc2C)no1 ZINC000147039139 HF On-Demand Anodyne VDR 52 39 CCN(CC)C(=O)c1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1Cl ZINC000147039150 HF On-Demand Anodyne ADORA2B 39 41 CCN(CC)C(=O)c1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1Cl ZINC000147039150 HF On-Demand Anodyne MCHR1 16 42 CCN(CC)C(=O)c1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1Cl ZINC000147039150 HF On-Demand Anodyne HIF1A 21 41 CC(=O)c1ccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@@H]32)cc1 ZINC000147039156 DD On-Demand Anodyne DHODH 15 42 COCCN(C(=O)c1cnn(-c2ccccc2Cl)c1)C1CC1 ZINC000147039314 DF On-Demand Anodyne MBTPS1 65 33 CC(C)N(C)S(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147039320 EE On-Demand Mild L3MBTL3 64 41 CCCOc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147039380 HG On-Demand Anodyne KCNA5 18 48 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)cc1 ZINC000147039381 GD On-Demand Anodyne HTR1D 17 42 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)cc1 ZINC000147039381 GD On-Demand Anodyne HTR1B 22 42 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)cc1 ZINC000147039381 GD On-Demand Anodyne F10 19 58 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)cc1 ZINC000147039381 GD On-Demand Anodyne CPT1A 100 48 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)cc1 ZINC000147039381 GD On-Demand Anodyne CPT2 45 36 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)cc1 ZINC000147039381 GD On-Demand Anodyne PLAU 20 43 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)cc1 ZINC000147039381 GD On-Demand Anodyne MCHR1 23 41 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)cc1 ZINC000147039381 GD On-Demand Anodyne HIF1A 23 45 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)N3CCCC3)c2)cc1 ZINC000147039381 GD On-Demand Anodyne TAAR1 44 41 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne ACE 107 53 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne TYR 37 44 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne OPRM1 58 46 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne OPRD1 58 46 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne FOLH1 17 45 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne MME 182 54 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne LTA4H 20 53 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne ANPEP 98 53 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne EDNRB 37 44 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne EDNRA 34 49 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne TACR1 29 47 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CTSD 49 41 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne PGC 63 41 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CMA1 22 44 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CTRA_BOVIN 22 42 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne FCER2 105 43 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CASP3 28 49 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne BMP1 20 42 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne RNPEP 30 53 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CASP8 23 41 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne KLK3 108 48 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CTSB 108 66 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne PAPA1_CARPA 106 47 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CYSP_TRYCR 77 54 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CCKAR 37 40 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne NTSR1 116 51 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne NTSR2 72 34 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CTSK 67 53 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CTSL 79 52 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CPA1 41 41 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CACNA1B 52 40 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne PGA 59 41 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne F2R 29 43 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne NPFFR2 72 37 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne TIMP3 87 39 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne C3AR1 42 43 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne HLA-A 98 47 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CAPNS1 103 63 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne MMP2 35 47 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne MMP3 64 48 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne MMP8 38 48 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne ECE1 93 44 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne HLA-DRB1 121 50 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne REN 124 51 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne REN1 71 45 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne LNPEP 28 53 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne SORT1 47 32 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CCKBR 22 42 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CTSS 35 50 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CAPN1 159 67 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne MMP9 44 49 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CASP1 32 49 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CAPN2 205 60 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CTSE 42 33 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne ACE2 123 49 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CASP6 46 36 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne CASP9 52 36 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne BACE1 21 45 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne LAP3 44 53 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne MMP7 40 41 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne MMP1 61 49 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne FPR1 121 62 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne NPR 123 56 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne AMP1_PLAFQ 43 53 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne XIAP 28 46 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne PSMB5 61 52 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne BLA1_STEMA 83 40 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne KISS1R 63 33 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne PSMB8 68 38 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne Q9N6S8_PLAFA 50 35 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne BRCA1 65 37 CC(C)C[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)N[C@@H](Cc1ccccc1)C(=O)O ZINC000147039493 KJ For-Sale Anodyne NPFFR1 71 37 CC(=O)c1ccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@H]32)cc1 ZINC000147039548 DD On-Demand Anodyne DHODH 15 42 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147039556 ED On-Demand Mild CCR8 77 37 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147039556 ED On-Demand Mild SFRP1 96 37 Cc1ccc(S(=O)(=O)NC2CC2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147039556 ED On-Demand Mild WNT3 73 34 CCCOc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147039564 HG On-Demand Anodyne KCNA5 18 48 CCCCC1CCC(NC(=O)Nc2ccc(CN3C(=O)CCC3=O)cc2)CC1 ZINC000147039722 GI On-Demand Anodyne EPHX2 50 44 COC(=O)c1cccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)c1 ZINC000147039756 HE On-Demand Anodyne ST14 45 35 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(OCC(F)(F)F)c2)c1 ZINC000147039793 GG On-Demand Bother ROCK1 23 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(OCC(F)(F)F)c2)c1 ZINC000147039793 GG On-Demand Bother PPARD 18 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(OCC(F)(F)F)c2)c1 ZINC000147039793 GG On-Demand Bother ROCK2 27 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(OCC(F)(F)F)c2)c1 ZINC000147039793 GG On-Demand Bother TAAR1 27 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(OCC(F)(F)F)c2)c1 ZINC000147039793 GG On-Demand Bother PDS 56 37 CO/C=C/c1ccc(Cl)c(C(=O)O)c1 ZINC000147039873 BF For-Sale Anodyne APP 42 43 CO/C=C/c1ccc(Cl)c(C(=O)O)c1 ZINC000147039873 BF For-Sale Anodyne AKR1C2 46 34 CO/C=C/c1ccc(Cl)c(C(=O)O)c1 ZINC000147039873 BF For-Sale Anodyne AKR1C1 47 34 COCCN(C(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1)C1CC1 ZINC000147039881 CG On-Demand Anodyne REN 52 34 COCCN(C(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1)C1CC1 ZINC000147039881 CG On-Demand Anodyne MDM2 62 34 CCNC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147039901 FD On-Demand Anodyne PRSS1 15 41 CCNC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147039901 FD On-Demand Anodyne LTA4H 20 40 CCNC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147039901 FD On-Demand Anodyne ADORA2A 15 44 CCNC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147039901 FD On-Demand Anodyne ADORA2B 43 44 CCNC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147039901 FD On-Demand Anodyne MTNR1A 33 40 CCNC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147039901 FD On-Demand Anodyne MTNR1B 30 42 CCNC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147039901 FD On-Demand Anodyne PLA2G4B 50 38 CCNC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147039901 FD On-Demand Anodyne PLAU 15 48 CCNC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147039901 FD On-Demand Anodyne ACR 57 36 CCNC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147039901 FD On-Demand Anodyne HIF1A 19 44 CCNC(=O)COc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147039901 FD On-Demand Anodyne KCNK3 42 34 Cc1cccc(O[C@@H](C)C(=O)NNC(=O)Nc2cccc(C(=O)N(C)C)c2)c1C ZINC000147039936 GF On-Demand Reactive KCNK3 52 36 Cc1cccc(O[C@@H](C)C(=O)NNC(=O)Nc2cccc(C(=O)N(C)C)c2)c1C ZINC000147039936 GF On-Demand Reactive KCNK9 51 31 COC(=O)c1cccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)c1 ZINC000147039956 HE On-Demand Anodyne ST14 45 35 COCCN(C(=O)[C@H]1C[C@H]1c1cccc(Cl)c1)C1CC1 ZINC000147040080 CG On-Demand Anodyne REN 37 40 Cc1cccc(O[C@H](C)C(=O)NNC(=O)Nc2cccc(C(=O)N(C)C)c2)c1C ZINC000147040136 GF On-Demand Reactive KCNK3 52 36 Cc1cccc(O[C@H](C)C(=O)NNC(=O)Nc2cccc(C(=O)N(C)C)c2)c1C ZINC000147040136 GF On-Demand Reactive KCNK9 51 31 COCCN(C(=O)[C@@H]1C[C@@H]1c1cccc(Br)c1)C1CC1 ZINC000147040264 EG On-Demand Anodyne REN 22 40 CCCCCN1CCN(C(C)=O)CC1 ZINC000147040357 AD On-Demand Anodyne THRB 50 49 CCCCCN1CCN(C(C)=O)CC1 ZINC000147040357 AD On-Demand Anodyne PLA2G2A 36 43 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N(C)C ZINC000147040363 DK For-Sale Anodyne CNR1 23 61 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N(C)C ZINC000147040363 DK For-Sale Anodyne LPAR1 22 43 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N(C)C ZINC000147040363 DK For-Sale Anodyne FAAH 25 53 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N(C)C ZINC000147040363 DK For-Sale Anodyne LPAR3 43 41 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N(C)C ZINC000147040363 DK For-Sale Anodyne FABP3 53 67 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N(C)C ZINC000147040363 DK For-Sale Anodyne FABP5 18 58 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N(C)C ZINC000147040363 DK For-Sale Anodyne LOX1.1 15 67 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N(C)C ZINC000147040363 DK For-Sale Anodyne FABP1 19 58 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N(C)C ZINC000147040363 DK For-Sale Anodyne OXER1 22 47 CCCCC/C=C\C/C=C\CCCCCCCC(=O)N(C)C ZINC000147040363 DK For-Sale Anodyne CQSS 57 35 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OCC(F)(F)F)nc2)c1 ZINC000147040396 FG On-Demand Bother ATF1 43 30 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OCC(F)(F)F)nc2)c1 ZINC000147040396 FG On-Demand Bother BTK 15 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OCC(F)(F)F)nc2)c1 ZINC000147040396 FG On-Demand Bother TAAR1 26 44 N#CC1CCN(C(=O)c2ccc(N3CCNC3=O)cc2)CC1 ZINC000147040399 CD On-Demand Mild L3MBTL3 64 41 COCCN(C(=O)[C@H]1C[C@@H]1c1cccc(Br)c1)C1CC1 ZINC000147040453 EG On-Demand Anodyne REN 22 40 Cc1cccc(NC(=O)N(C)O)c1 ZINC000147040470 AD For-Sale Anodyne CCKAR 22 44 Cc1cccc(NC(=O)N(C)O)c1 ZINC000147040470 AD For-Sale Anodyne KDR 18 43 Cc1cccc(NC(=O)N(C)O)c1 ZINC000147040470 AD For-Sale Anodyne F12 0 43 Cc1cccc(NC(=O)N(C)O)c1 ZINC000147040470 AD For-Sale Anodyne SCN10A 18 40 Cc1cccc(NC(=O)N(C)O)c1 ZINC000147040470 AD For-Sale Anodyne PARP14 42 35 Cc1cccc(NC(=O)N(C)O)c1 ZINC000147040470 AD For-Sale Anodyne PARP15 47 35 Cc1cccc(NC(=O)N(C)O)c1 ZINC000147040470 AD For-Sale Anodyne PSBA 0 77 Cc1cccc(NC(=O)N(C)O)c1 ZINC000147040470 AD For-Sale Anodyne KCNK3 125 53 Cc1cccc(NC(=O)N(C)O)c1 ZINC000147040470 AD For-Sale Anodyne KCNK9 86 53 Cc1cccc(NC(=O)N(C)O)c1 ZINC000147040470 AD For-Sale Anodyne PPX1 0 41 Cc1cccc(NC(=O)N(C)O)c1 ZINC000147040470 AD For-Sale Anodyne PARP10 62 36 CC(C)(C)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147040562 HH On-Demand Anodyne KCNA5 16 45 O=C(Nc1ccc(OCC(F)(F)F)nc1)c1ccn(-c2cccc(F)c2)n1 ZINC000147040605 GH On-Demand Anodyne DGAT1 15 41 COCCN(C(=O)[C@@H]1C[C@H]1c1cccc(Br)c1)C1CC1 ZINC000147040646 EG On-Demand Anodyne REN 22 40 CC(C)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147040808 HG On-Demand Anodyne POL 22 42 COCCc1ccc(Cl)c(C(=O)NC2CC2)c1 ZINC000147040822 CE For-Sale Anodyne DRD2 20 40 COCCc1ccc(Cl)c(C(=O)NC2CC2)c1 ZINC000147040822 CE For-Sale Anodyne DRD4 15 43 COCCc1ccc(Cl)c(C(=O)NC2CC2)c1 ZINC000147040822 CE For-Sale Anodyne HTR4 42 41 COCCc1ccc(Cl)c(C(=O)NC2CC2)c1 ZINC000147040822 CE For-Sale Anodyne MCHR1 22 45 COCCc1ccc(Cl)c(C(=O)NC2CC2)c1 ZINC000147040822 CE For-Sale Anodyne NCE103 19 42 COCCN(C(=O)[C@H]1C[C@H]1c1cccc(Br)c1)C1CC1 ZINC000147040832 EG On-Demand Anodyne REN 22 40 CC(=O)c1cc(Br)c(O)c([N+](=O)[O-])c1 ZINC000147040907 CE In-Stock Bother TPMT 0 40 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2c[nH]c3ccccc23)n1 ZINC000147040985 JI For-Sale Bother HTR1A 19 40 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2c[nH]c3ccccc23)n1 ZINC000147040985 JI For-Sale Bother IGF1R 54 39 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2c[nH]c3ccccc23)n1 ZINC000147040985 JI For-Sale Bother ZAP70 21 41 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2c[nH]c3ccccc23)n1 ZINC000147040985 JI For-Sale Bother TTK 16 53 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2c[nH]c3ccccc23)n1 ZINC000147040985 JI For-Sale Bother MAPK7 63 43 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2c[nH]c3ccccc23)n1 ZINC000147040985 JI For-Sale Bother DYRK1B 38 57 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2c[nH]c3ccccc23)n1 ZINC000147040985 JI For-Sale Bother DCLK2 20 43 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1nccc(-c2c[nH]c3ccccc23)n1 ZINC000147040985 JI For-Sale Bother DCLK1 18 43 CC(C)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147041003 HG On-Demand Anodyne POL 22 42 C[C@@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041026 DH On-Demand Anodyne ACE 36 40 C[C@@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041026 DH On-Demand Anodyne MME 103 40 C[C@@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041026 DH On-Demand Anodyne ANPEP 56 33 C[C@@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041026 DH On-Demand Anodyne FCER2 63 39 C[C@@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041026 DH On-Demand Anodyne PAPA1_CARPA 41 33 C[C@@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041026 DH On-Demand Anodyne CTSL 37 44 C[C@@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041026 DH On-Demand Anodyne CPA1 27 44 C[C@@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041026 DH On-Demand Anodyne CTSS 27 44 C[C@@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041026 DH On-Demand Anodyne ACE2 70 38 C[C@@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041026 DH On-Demand Anodyne FPR1 49 35 C[C@@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041026 DH On-Demand Anodyne AMP1_PLAFQ 54 35 O=C(Nc1cccc(CNS(=O)(=O)c2ccc(Cl)s2)c1)[C@@H]1CCCO1 ZINC000147041207 HF On-Demand Anodyne CCR4 62 50 C/N=C\c1cccc(C(=O)NC)c1 ZINC000147041216 AD For-Sale Mild AMD1 20 40 C/N=C\c1cccc(C(=O)NC)c1 ZINC000147041216 AD For-Sale Mild KCNK3 61 37 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne ACE 36 40 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne OPRM1 23 40 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne MME 103 40 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne ANPEP 56 33 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne FCER2 63 39 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne PAPA1_CARPA 41 33 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne CTSL 37 44 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne CPA1 27 44 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne CTSS 27 44 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne ACE2 70 38 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne FPR1 49 35 C[C@H](Cc1cccc(F)c1)C(=O)NCCSc1ccccc1 ZINC000147041220 DH On-Demand Anodyne AMP1_PLAFQ 54 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1nnc2ccccn12 ZINC000147041231 DD On-Demand Anodyne KLK3 52 36 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1nnc2ccccn12 ZINC000147041231 DD On-Demand Anodyne PCSK5 40 32 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1nnc2ccccn12 ZINC000147041231 DD On-Demand Anodyne POLG_WNV 40 30 N#Cc1ccc(Oc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2Cl)cc1 ZINC000147041245 HH On-Demand Mild PFKFB3 49 33 CCCCCC[C@@H](CC)C(C)C ZINC000147041292 AJ For-Sale Anodyne CQSS 54 33 NC(=O)c1ccc(OCC(=O)NCCc2ccc3ccccc3c2)cc1 ZINC000147041330 EF On-Demand Anodyne MTNR1A 42 39 C[C@@H](C(=O)NCc1ccc(C(F)(F)F)cc1Cl)c1ccc(NS(C)(=O)=O)c(F)c1 ZINC000147041368 JI Annotated Anodyne TRPV1 182 71 CCCc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147041412 HG On-Demand Anodyne KCNA5 21 49 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1nnc2ccccn12 ZINC000147041424 DD On-Demand Anodyne KLK3 52 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1nnc2ccccn12 ZINC000147041424 DD On-Demand Anodyne PCSK5 40 32 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1nnc2ccccn12 ZINC000147041424 DD On-Demand Anodyne POLG_WNV 40 30 COCc1ccccc1NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147041432 FE On-Demand Bother COLA 84 37 N#Cc1ccc(Oc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2Cl)cc1 ZINC000147041439 HH On-Demand Mild PFKFB3 49 33 CCCCCC[C@H](CC)C(C)C ZINC000147041481 AJ For-Sale Anodyne CQSS 54 33 C[C@H](C(=O)NCc1ccc(C(F)(F)F)cc1Cl)c1ccc(NS(C)(=O)=O)c(F)c1 ZINC000147041571 JI Annotated Anodyne TRPV1 182 71 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1nnc2ccccn12 ZINC000147041629 DD On-Demand Anodyne KLK3 52 36 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1nnc2ccccn12 ZINC000147041629 DD On-Demand Anodyne PCSK5 40 32 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1nnc2ccccn12 ZINC000147041629 DD On-Demand Anodyne POLG_WNV 40 30 CCCC[C@H](NC1=NS(=O)(=O)c2ccccc21)C(=O)N1CCC(C#N)CC1 ZINC000147041666 GE On-Demand Mild P2RY12 164 34 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne OPRM1 0 41 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne OPRD1 0 41 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne MME 27 42 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne NPR1 47 38 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne FCER2 40 40 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne TRY2_BOVIN 46 33 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne PAPA1_CARPA 27 41 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne CTSL 30 44 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne BRS3 26 41 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne NPFFR2 46 37 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne MTNR1A 30 40 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne GRIA1 67 36 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne PCSK5 58 38 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne FURIN 62 38 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne CCKBR 0 42 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne CAPN1 32 41 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne CAPN2 59 40 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne ACE2 39 42 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne POLG_WNV 82 38 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne QRFPR 41 39 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne NPFFR1 54 37 CCC[C@@H](NC(N)=O)C(=O)NCCc1ccc2ccccc2c1 ZINC000147041725 DE On-Demand Anodyne IDE 0 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1nnc2ccccn12 ZINC000147041817 DD On-Demand Anodyne KLK3 52 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1nnc2ccccn12 ZINC000147041817 DD On-Demand Anodyne PCSK5 40 32 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1nnc2ccccn12 ZINC000147041817 DD On-Demand Anodyne POLG_WNV 40 30 CCCNc1nccc2[nH]nc(C)c12 ZINC000147041846 AE For-Sale Anodyne UTS2R 26 55 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccccc1[N+](=O)[O-])C2 ZINC000147041850 EE On-Demand Bother COLA 86 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccccc1[N+](=O)[O-])C2 ZINC000147041850 EE On-Demand Bother MTNR1A 30 40 CC(=O)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147041942 HE On-Demand Anodyne KCNA5 15 46 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne ESR1 79 41 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne ACHE 29 52 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne KCNH2 0 51 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne ESR2 47 42 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne LTA4H 55 56 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne HRH3 79 52 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne SIGMAR1 28 43 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne EBP 36 40 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne ABCB1 0 44 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne MCHR1 24 47 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne PSMB2 67 54 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne PSMB5 23 54 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne PSMB1 60 54 COc1ccc(OCCN2CCCCC2)cc1C ZINC000147041946 BF On-Demand Anodyne NORA 0 42 CCCCCCNC(=O)Nc1ccnc(-c2ccncc2)n1 ZINC000147041958 CG For-Sale Anodyne ASAH1 56 34 C[C@@H](O)C(=O)NCCCN ZINC000147041988 AA For-Sale Anodyne GRIA1 52 37 C[C@@H](O)C(=O)NCCCN ZINC000147041988 AA For-Sale Anodyne PCSK6 47 35 C[C@@H](O)C(=O)NCCCN ZINC000147041988 AA For-Sale Anodyne DPP7 0 44 C[C@@H](O)C(=O)NCCCN ZINC000147041988 AA For-Sale Anodyne PAO 42 34 C[C@@H](O)C(=O)NCCCN ZINC000147041988 AA For-Sale Anodyne APHA 41 34 C[C@@H](O)C(=O)NCCCN ZINC000147041988 AA For-Sale Anodyne AGUA 0 40 CN1CCc2ccc(CC(=O)O)cc2C1 ZINC000147042005 BD For-Sale Anodyne DRD5 51 39 OCc1ccc(OC[C@H](O)CO)cc1 ZINC000147042006 AB For-Sale Anodyne ADRB2 28 46 OCc1ccc(OC[C@H](O)CO)cc1 ZINC000147042006 AB For-Sale Anodyne ADRB1 40 46 OCc1ccc(OC[C@H](O)CO)cc1 ZINC000147042006 AB For-Sale Anodyne ADRB3 37 40 COc1cc(N2CC[C@H](N(C)C)C2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147042007 JI For-Sale Bother INSR 28 50 COc1cc(N2CC[C@H](N(C)C)C2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147042007 JI For-Sale Bother IGF1R 24 44 COc1cc(N2CC[C@H](N(C)C)C2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147042007 JI For-Sale Bother MAPK7 54 36 COc1cc(N2CC[C@H](N(C)C)C2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147042007 JI For-Sale Bother DYRK1B 23 47 O=C(NCc1ccccc1[N+](=O)[O-])[C@@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147042059 GH On-Demand Bother COLA 106 35 CC(=O)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147042146 HE On-Demand Anodyne KCNA5 16 46 C[C@H](O)C(=O)NCCCN ZINC000147042179 AA For-Sale Anodyne GRIA1 52 37 C[C@H](O)C(=O)NCCCN ZINC000147042179 AA For-Sale Anodyne PCSK6 47 35 C[C@H](O)C(=O)NCCCN ZINC000147042179 AA For-Sale Anodyne DPP7 0 44 C[C@H](O)C(=O)NCCCN ZINC000147042179 AA For-Sale Anodyne PAO 42 34 C[C@H](O)C(=O)NCCCN ZINC000147042179 AA For-Sale Anodyne APHA 41 34 C[C@H](O)C(=O)NCCCN ZINC000147042179 AA For-Sale Anodyne AGUA 0 40 OCc1ccc(OC[C@@H](O)CO)cc1 ZINC000147042199 AB For-Sale Anodyne ADRB2 28 46 OCc1ccc(OC[C@@H](O)CO)cc1 ZINC000147042199 AB For-Sale Anodyne ADRB1 40 46 OCc1ccc(OC[C@@H](O)CO)cc1 ZINC000147042199 AB For-Sale Anodyne ADRB3 37 40 Cc1cccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@@H]32)c1 ZINC000147042200 CD On-Demand Anodyne KCNK3 41 37 COc1cc(N2CC[C@@H](N(C)C)C2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147042215 JI For-Sale Bother INSR 28 50 COc1cc(N2CC[C@@H](N(C)C)C2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147042215 JI For-Sale Bother IGF1R 24 44 COc1cc(N2CC[C@@H](N(C)C)C2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147042215 JI For-Sale Bother MAPK7 54 36 COc1cc(N2CC[C@@H](N(C)C)C2)c([N+](=O)[O-])cc1Nc1nccc(-c2cn(C)c3ccccc23)n1 ZINC000147042215 JI For-Sale Bother DYRK1B 23 47 COc1ccc(Nc2nc3c(C4=CCN(S(C)(=O)=O)CC4)cccn3n2)cc1 ZINC000147042226 GF Annotated Anodyne JAK2 28 60 N[C@@H]1C[C@@H]1c1ccc(I)cc1 ZINC000147042245 CE For-Sale Anodyne KDM1A 25 44 O=C(NCc1ccccc1[N+](=O)[O-])[C@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147042255 GH On-Demand Bother COLA 106 35 Cc1cccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@@H]32)c1 ZINC000147042394 CD On-Demand Anodyne KCNK3 41 37 N[C@H]1C[C@@H]1c1ccc(I)cc1 ZINC000147042433 CE For-Sale Anodyne KDM1A 25 44 O=C(NCc1ccccc1[N+](=O)[O-])[C@@H]1C[C@H]1c1cccc(Br)c1 ZINC000147042459 GH On-Demand Bother COLA 106 35 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(-c3ccccc3)c(C(C)C)s2)c1 ZINC000147042541 GK On-Demand Bother AKR1C2 22 40 Cc1cccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@H]32)c1 ZINC000147042577 CD On-Demand Anodyne KCNK3 41 37 CC(=O)c1cccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)c1 ZINC000147042612 HE On-Demand Anodyne ST14 44 34 N[C@@H]1C[C@H]1c1ccc(I)cc1 ZINC000147042616 CE For-Sale Anodyne KDM1A 25 44 Cc1cccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@H]32)c1 ZINC000147042767 CD On-Demand Anodyne KCNK3 41 37 NC(N)=NCCC[C@@H](NC(=O)[C@H]1CCCN1)C(=O)NCC(=O)O ZINC000147042791 EA For-Sale Mild MC4R 18 40 NC(N)=NCCC[C@@H](NC(=O)[C@H]1CCCN1)C(=O)NCC(=O)O ZINC000147042791 EA For-Sale Mild NPFFR2 39 60 NC(N)=NCCC[C@@H](NC(=O)[C@H]1CCCN1)C(=O)NCC(=O)O ZINC000147042791 EA For-Sale Mild HDAC11 41 37 N[C@H]1C[C@H]1c1ccc(I)cc1 ZINC000147042794 CE For-Sale Anodyne KDM1A 25 44 CC(=O)c1cccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)c1 ZINC000147042802 HE On-Demand Anodyne ST14 44 34 CCOC(=O)NCC(=O)N1CCC[C@H](c2nc3ccccc3o2)C1 ZINC000147042841 EE On-Demand Anodyne SSTR5 26 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147042862 FD On-Demand Anodyne KLK3 47 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147042862 FD On-Demand Anodyne CTSF 52 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147042862 FD On-Demand Anodyne CTSK 48 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147042862 FD On-Demand Anodyne HLA-DRB1 29 40 NC(N)=NCCC[C@@H](NC(=O)[C@@H]1CCCN1)C(=O)NCC(=O)O ZINC000147042955 EA For-Sale Mild MC4R 18 40 NC(N)=NCCC[C@@H](NC(=O)[C@@H]1CCCN1)C(=O)NCC(=O)O ZINC000147042955 EA For-Sale Mild NPFFR2 39 60 NC(N)=NCCC[C@@H](NC(=O)[C@@H]1CCCN1)C(=O)NCC(=O)O ZINC000147042955 EA For-Sale Mild HDAC11 41 37 COc1cccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@@H]32)c1 ZINC000147042981 DD On-Demand Anodyne CCR3 20 43 COc1cccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@@H]32)c1 ZINC000147042981 DD On-Demand Anodyne MTNR1A 20 42 COc1cccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@@H]32)c1 ZINC000147042981 DD On-Demand Anodyne TAAR1 34 40 CCOC(=O)NCC(=O)N1CCC[C@@H](c2nc3ccccc3o2)C1 ZINC000147043012 EE On-Demand Anodyne SSTR5 26 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043066 FD On-Demand Anodyne KLK3 47 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043066 FD On-Demand Anodyne CTSF 52 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043066 FD On-Demand Anodyne CTSK 48 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043066 FD On-Demand Anodyne HLA-DRB1 29 40 COc1cccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@@H]32)c1 ZINC000147043172 DD On-Demand Anodyne CCR3 20 43 COc1cccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@@H]32)c1 ZINC000147043172 DD On-Demand Anodyne MTNR1A 20 42 COc1cccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@@H]32)c1 ZINC000147043172 DD On-Demand Anodyne TAAR1 34 40 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1 ZINC000147043237 JJ For-Sale Bother INSR 49 41 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1 ZINC000147043237 JJ For-Sale Bother IGF1R 50 52 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1 ZINC000147043237 JJ For-Sale Bother MAPK9 25 52 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1 ZINC000147043237 JJ For-Sale Bother TTK 17 40 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1 ZINC000147043237 JJ For-Sale Bother PAK1 55 42 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1 ZINC000147043237 JJ For-Sale Bother TNIK 30 41 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1 ZINC000147043237 JJ For-Sale Bother ALK 62 42 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1 ZINC000147043237 JJ For-Sale Bother MAPK7 64 43 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1 ZINC000147043237 JJ For-Sale Bother DYRK1B 29 43 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1 ZINC000147043237 JJ For-Sale Bother DCLK2 21 43 COc1cc(N2CCN(C)CC2)c([N+](=O)[O-])cc1Nc1ncc(Cl)c(-c2c[nH]c3ccccc23)n1 ZINC000147043237 JJ For-Sale Bother DCLK1 20 43 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043256 FD On-Demand Anodyne KLK3 47 35 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043256 FD On-Demand Anodyne CTSF 52 35 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043256 FD On-Demand Anodyne CTSK 48 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043256 FD On-Demand Anodyne HLA-DRB1 29 40 COc1cccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@H]32)c1 ZINC000147043364 DD On-Demand Anodyne CCR3 20 43 COc1cccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@H]32)c1 ZINC000147043364 DD On-Demand Anodyne MTNR1A 20 42 COc1cccc(NC(=O)C(=O)N2CCO[C@H]3CCC[C@H]32)c1 ZINC000147043364 DD On-Demand Anodyne TAAR1 34 40 CC(C)(C)OC(=O)N1CC[C@H](NS(=O)(=O)C2(C)CC2)C1 ZINC000147043390 DD On-Demand Anodyne SFRP1 33 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043476 FD On-Demand Anodyne KLK3 47 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043476 FD On-Demand Anodyne CTSF 52 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043476 FD On-Demand Anodyne CTSK 48 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(S(C)(=O)=O)cc1 ZINC000147043476 FD On-Demand Anodyne HLA-DRB1 29 40 N#CC1CCN(C(=O)Cc2ccc3c(c2)CCO3)CC1 ZINC000147043516 CD On-Demand Mild KCNJ1 46 37 COc1cccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@H]32)c1 ZINC000147043552 DD On-Demand Anodyne CCR3 20 43 COc1cccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@H]32)c1 ZINC000147043552 DD On-Demand Anodyne MTNR1A 20 42 COc1cccc(NC(=O)C(=O)N2CCO[C@@H]3CCC[C@H]32)c1 ZINC000147043552 DD On-Demand Anodyne TAAR1 34 40 CC(=O)Nc1ncc(SC(C)=O)s1 ZINC000147043639 BD For-Sale Anodyne CAHX_FLABI 0 40 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne CACNA2D1 27 63 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne MME 39 47 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne ANPEP 74 37 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne RNPEP 35 40 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne CPA1 47 39 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne SLC15A1 0 53 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne CTRB1 28 40 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne SLC1A6 55 35 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne SLC1A1 15 47 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne DNPEP 0 43 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne SLC1A7 55 35 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne LAP3 58 48 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne CTSC 15 45 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne CPA3 65 39 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne CYP2A5 0 52 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne SLC15A2 0 50 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne BLAIMP-1 0 45 N[C@@H](Cc1ccccc1)C(O)=S ZINC000147043642 AD For-Sale Anodyne VM1B1_BOTAS 0 40 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CC(=O)N2CCCCCC2)CC1 ZINC000147043661 GC On-Demand Anodyne P2RY12 84 44 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CC(=O)N2CCCCCC2)CC1 ZINC000147043661 GC On-Demand Anodyne DPP7 41 36 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CC(=O)N2CCCCCC2)CC1 ZINC000147043661 GC On-Demand Anodyne NOD1 40 31 CCNC(=O)N1CCC(NC(=O)[C@@H]2N[C@H](CC(C)(C)C)[C@]3(C(=O)Nc4cc(Cl)ccc43)[C@H]2c2cccc(Cl)c2F)CC1 ZINC000147043760 KK Annotated Anodyne MDM2 103 70 CCCCOc1ccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1OC ZINC000147043779 GH On-Demand Bother CNR2 37 40 CCCCOc1ccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1OC ZINC000147043779 GH On-Demand Bother MTNR1A 18 40 CCCCOc1ccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1OC ZINC000147043779 GH On-Demand Bother MTNR1B 21 40 CCCCOc1ccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1OC ZINC000147043779 GH On-Demand Bother S1PR2 42 33 CCCCOc1ccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1OC ZINC000147043779 GH On-Demand Bother MT-ND1 25 43 O=C(Nc1cccc(CNS(=O)(=O)c2ccc3ccccc3c2)c1)[C@@H]1CCCO1 ZINC000147043851 HG On-Demand Anodyne F2 23 45 O=C(Nc1cccc(CNS(=O)(=O)c2ccc3ccccc3c2)c1)[C@@H]1CCCO1 ZINC000147043851 HG On-Demand Anodyne NPY1R 22 40 O=C(Nc1cccc(CNS(=O)(=O)c2ccc3ccccc3c2)c1)[C@@H]1CCCO1 ZINC000147043851 HG On-Demand Anodyne TRY2_BOVIN 71 45 O=C(Nc1cccc(CNS(=O)(=O)c2ccc3ccccc3c2)c1)[C@@H]1CCCO1 ZINC000147043851 HG On-Demand Anodyne NPY2R 17 49 O=C(Nc1cccc(CNS(=O)(=O)c2ccc3ccccc3c2)c1)[C@@H]1CCCO1 ZINC000147043851 HG On-Demand Anodyne ST14 34 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CC(=O)N2CCCCCC2)CC1 ZINC000147043878 GC On-Demand Anodyne P2RY12 84 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CC(=O)N2CCCCCC2)CC1 ZINC000147043878 GC On-Demand Anodyne DPP7 41 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CC(=O)N2CCCCCC2)CC1 ZINC000147043878 GC On-Demand Anodyne NOD1 40 31 O=C(CF)c1ccccc1OCc1ccccc1 ZINC000147043938 BG For-Sale Anodyne PTGER2 23 43 O=C(CF)c1ccccc1OCc1ccccc1 ZINC000147043938 BG For-Sale Anodyne PPIA 51 47 O=C(CF)c1ccccc1OCc1ccccc1 ZINC000147043938 BG For-Sale Anodyne PTGER1 47 50 O=C(CF)c1ccccc1OCc1ccccc1 ZINC000147043938 BG For-Sale Anodyne PTGER4 25 43 O=C(CF)c1ccccc1OCc1ccccc1 ZINC000147043938 BG For-Sale Anodyne PTGER3 16 41 O=C(CF)c1ccccc1OCc1ccccc1 ZINC000147043938 BG For-Sale Anodyne ABCB1 42 43 CC(C)[C@H]1CC[C@@H](C)C[C@H]1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147043978 EF On-Demand Anodyne TRPM8 21 54 CC(=O)Nc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147044105 HE On-Demand Anodyne KCNA5 19 46 CC(=O)Nc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147044105 HE On-Demand Anodyne IDO1 30 40 CC(C)Oc1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1Cl ZINC000147044138 GF On-Demand Anodyne ADRA1D 16 43 CC(C)Oc1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1Cl ZINC000147044138 GF On-Demand Anodyne ADRA1B 15 40 CC(C)Oc1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1Cl ZINC000147044138 GF On-Demand Anodyne EPHX2 42 49 N#CC1CCN(C(=O)CCc2ccc(Cl)cc2)CC1 ZINC000147044147 CG On-Demand Mild C3AR1 39 42 N#CC1CCN(C(=O)CCc2ccc(Cl)cc2)CC1 ZINC000147044147 CG On-Demand Mild MLNR 17 42 N#CC1CCN(C(=O)CCc2ccc(Cl)cc2)CC1 ZINC000147044147 CG On-Demand Mild FAP 0 45 C[C@@H](CCNC(=O)Cc1cccc(F)c1)c1ccccc1 ZINC000147044262 CH On-Demand Anodyne MME 34 40 C[C@@H](CCNC(=O)Cc1cccc(F)c1)c1ccccc1 ZINC000147044262 CH On-Demand Anodyne ANPEP 24 41 C[C@@H](CCNC(=O)Cc1cccc(F)c1)c1ccccc1 ZINC000147044262 CH On-Demand Anodyne CPA1 20 40 C[C@@H](CCNC(=O)Cc1cccc(F)c1)c1ccccc1 ZINC000147044262 CH On-Demand Anodyne NCE103 17 40 CC(=O)Nc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147044296 HE On-Demand Anodyne KCNA5 19 46 CC(=O)Nc1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147044296 HE On-Demand Anodyne IDO1 30 40 CC(C)Oc1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1Cl ZINC000147044324 GF On-Demand Anodyne ADRA1D 16 43 CC(C)Oc1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1Cl ZINC000147044324 GF On-Demand Anodyne ADRA1B 15 40 CC(C)Oc1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1Cl ZINC000147044324 GF On-Demand Anodyne EPHX2 42 49 N#Cc1ccc(CCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147044336 CE On-Demand Mild MLNR 20 40 N#Cc1ccc(CCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147044336 CE On-Demand Mild FAP 0 41 N#Cc1ccc(CCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147044336 CE On-Demand Mild KCNJ1 15 44 O=C1CSC(=O)N1CCCCNCCc1cccc2ccccc12 ZINC000147044366 EG For-Sale Anodyne HTR4 16 47 CC(C)[C@@H]1CC[C@@H](C)C[C@H]1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147044377 EF On-Demand Anodyne TRPM8 21 54 C[C@H](CCNC(=O)Cc1cccc(F)c1)c1ccccc1 ZINC000147044440 CH On-Demand Anodyne MME 34 40 C[C@H](CCNC(=O)Cc1cccc(F)c1)c1ccccc1 ZINC000147044440 CH On-Demand Anodyne ANPEP 24 41 C[C@H](CCNC(=O)Cc1cccc(F)c1)c1ccccc1 ZINC000147044440 CH On-Demand Anodyne CPA1 20 40 C[C@H](CCNC(=O)Cc1cccc(F)c1)c1ccccc1 ZINC000147044440 CH On-Demand Anodyne NCE103 17 40 COc1ccc2c(c1)OC[C@H](C(=O)NC1CCC3(CC1)OCCO3)C2 ZINC000147044449 EE On-Demand Anodyne ROCK2 21 41 CCCC[C@H](NC(N)=O)C(=O)N1CCCCC[C@@H]1c1ccc(OC)cc1 ZINC000147044483 FG On-Demand Anodyne P2RY12 118 34 CCCC[C@H](NC(N)=O)C(=O)N1CCCCC[C@@H]1c1ccc(OC)cc1 ZINC000147044483 FG On-Demand Anodyne TRHR 47 33 CCCC[C@H](NC(N)=O)C(=O)N1CCCCC[C@@H]1c1ccc(OC)cc1 ZINC000147044483 FG On-Demand Anodyne HLA-DRB3 53 35 CCCC[C@H](NC(N)=O)C(=O)N1CCCCC[C@@H]1c1ccc(OC)cc1 ZINC000147044483 FG On-Demand Anodyne TRY1_BOVIN 52 37 CCCC[C@H](NC(N)=O)C(=O)N1CCCCC[C@@H]1c1ccc(OC)cc1 ZINC000147044483 FG On-Demand Anodyne NTSR1 47 31 C[C@@H](Cc1cccc(F)c1)C(=O)N(C)Cc1ccsc1 ZINC000147044638 CH On-Demand Anodyne HSD17B2 25 46 CCCC[C@@H](NC(N)=O)C(=O)N1CCCCC[C@@H]1c1ccc(OC)cc1 ZINC000147044665 FG On-Demand Anodyne P2RY12 118 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCCCC[C@@H]1c1ccc(OC)cc1 ZINC000147044665 FG On-Demand Anodyne TRHR 47 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCCCC[C@@H]1c1ccc(OC)cc1 ZINC000147044665 FG On-Demand Anodyne HLA-DRB3 53 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCCCC[C@@H]1c1ccc(OC)cc1 ZINC000147044665 FG On-Demand Anodyne TRY1_BOVIN 52 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCCCC[C@@H]1c1ccc(OC)cc1 ZINC000147044665 FG On-Demand Anodyne NTSR1 47 31 COc1ccc2c(c1)OC[C@@H](C(=O)NC1CCC3(CC1)OCCO3)C2 ZINC000147044668 EE On-Demand Anodyne ROCK2 21 41 C[C@@](N)(CO)c1ncc(-c2ccc(OCc3ccc(-c4ccccc4)cc3)c(C(F)(F)F)c2)[nH]1 ZINC000147044790 JK For-Sale Anodyne S1PR4 39 58 C[C@@](N)(CO)c1ncc(-c2ccc(OCc3ccc(-c4ccccc4)cc3)c(C(F)(F)F)c2)[nH]1 ZINC000147044790 JK For-Sale Anodyne S1PR1 16 58 C[C@@](N)(CO)c1ncc(-c2ccc(OCc3ccc(-c4ccccc4)cc3)c(C(F)(F)F)c2)[nH]1 ZINC000147044790 JK For-Sale Anodyne S1PR5 23 58 CCCC[C@H](NC(N)=O)C(=O)N1CCCCC[C@H]1c1ccc(OC)cc1 ZINC000147044851 FG On-Demand Anodyne P2RY12 118 34 CCCC[C@H](NC(N)=O)C(=O)N1CCCCC[C@H]1c1ccc(OC)cc1 ZINC000147044851 FG On-Demand Anodyne TRHR 47 33 CCCC[C@H](NC(N)=O)C(=O)N1CCCCC[C@H]1c1ccc(OC)cc1 ZINC000147044851 FG On-Demand Anodyne HLA-DRB3 53 35 CCCC[C@H](NC(N)=O)C(=O)N1CCCCC[C@H]1c1ccc(OC)cc1 ZINC000147044851 FG On-Demand Anodyne TRY1_BOVIN 52 37 CCCC[C@H](NC(N)=O)C(=O)N1CCCCC[C@H]1c1ccc(OC)cc1 ZINC000147044851 FG On-Demand Anodyne NTSR1 47 31 O=C(NCCNC(=O)c1cccs1)c1cnn(-c2ccccc2Cl)c1 ZINC000147044875 FF On-Demand Anodyne DRD3 22 43 COc1ccc(N(C)C(=O)Nc2nc3c(OC)ccc(N4CCOCC4)c3s2)cc1 ZINC000147044952 IH For-Sale Clean ADORA2B 17 45 COc1ccc(N(C)C(=O)Nc2nc3c(OC)ccc(N4CCOCC4)c3s2)cc1 ZINC000147044952 IH For-Sale Clean CASR 24 47 Cc1cc(C)c2cc(C(=O)N3CCC(C#N)CC3)[nH]c2c1 ZINC000147044981 CG On-Demand Mild HRH4 27 42 Cc1cc(C)c2cc(C(=O)N3CCC(C#N)CC3)[nH]c2c1 ZINC000147044981 CG On-Demand Mild AKR1C3 0 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCCCC[C@H]1c1ccc(OC)cc1 ZINC000147045022 FG On-Demand Anodyne P2RY12 118 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCCCC[C@H]1c1ccc(OC)cc1 ZINC000147045022 FG On-Demand Anodyne TRHR 47 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCCCC[C@H]1c1ccc(OC)cc1 ZINC000147045022 FG On-Demand Anodyne HLA-DRB3 53 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCCCC[C@H]1c1ccc(OC)cc1 ZINC000147045022 FG On-Demand Anodyne TRY1_BOVIN 52 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCCCC[C@H]1c1ccc(OC)cc1 ZINC000147045022 FG On-Demand Anodyne NTSR1 47 31 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147045228 HD On-Demand Anodyne F2 31 40 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147045228 HD On-Demand Anodyne P2RY12 141 34 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147045228 HD On-Demand Anodyne TRY2_BOVIN 81 40 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147045228 HD On-Demand Anodyne TGM2 49 40 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147045228 HD On-Demand Anodyne F13A1 63 40 Cc1cc(C)c(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)c(C)c1 ZINC000147045256 HG On-Demand Anodyne ALB 16 42 CCCCOc1ccccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147045393 EE On-Demand Anodyne AMY2 43 30 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147045429 HD On-Demand Anodyne F2 31 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147045429 HD On-Demand Anodyne P2RY12 141 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147045429 HD On-Demand Anodyne TRY2_BOVIN 81 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147045429 HD On-Demand Anodyne TGM2 49 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147045429 HD On-Demand Anodyne F13A1 63 40 CS(=O)(=O)c1cc(C(=O)NC2CCN(c3ccccn3)CC2)cc([N+](=O)[O-])c1 ZINC000147045436 HD On-Demand Bother MAPK13 43 32 CCCCOc1ccccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147045577 EE On-Demand Anodyne AMY2 43 30 N#Cc1ccc(Oc2ccc(NC(=O)C[C@]3(C(=O)O)CCSC3)cc2)cc1 ZINC000147045750 GH On-Demand Anodyne PFKFB3 76 40 COC(=O)[C@@H]1c2ccccc2C[C@@H]1O ZINC000147045782 AC In-Stock Anodyne POL 0 43 COC(=O)[C@@H]1c2ccccc2C[C@@H]1O ZINC000147045782 AC In-Stock Anodyne PLM1_PLAFA 42 42 COC(=O)[C@@H]1c2ccccc2C[C@@H]1O ZINC000147045782 AC In-Stock Anodyne PLM2_PLAFA 44 42 COC(=O)[C@@H]1c2ccccc2C[C@@H]1O ZINC000147045782 AC In-Stock Anodyne O60989_PLAVI 66 32 N#CC1CCN(C(=O)c2sccc2S(=O)(=O)N2CCCCC2)CC1 ZINC000147045840 FE On-Demand Mild L3MBTL3 42 37 CCCCOc1ccc(OC)cc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147045935 FF On-Demand Anodyne MTNR1B 26 44 CCCCOc1ccc(OC)cc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147045935 FF On-Demand Anodyne SLC9A1 51 32 CCCCOc1ccc(OC)cc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147045935 FF On-Demand Anodyne PLA2G4B 80 46 CCCCO[C@@H](C)C(=O)N1CCN(c2cc(C)nc(C(C)C)n2)CC1 ZINC000147045951 EF On-Demand Anodyne P2RY12 68 38 CC(C)CC[C@H]1N[C@@H](C(=O)NCC[C@H](O)CO)[C@H](c2cccc(Cl)c2)[C@@]12C(=O)Nc1cc(Cl)c(F)cc12 ZINC000147045993 KH Annotated Anodyne MDM2 76 83 Cc1ccccc1NS(=O)(=O)c1ccc(C)c(C(=O)N2CCC(C#N)CC2)c1 ZINC000147046066 GG On-Demand Mild CCR8 75 38 Cc1ccccc1NS(=O)(=O)c1ccc(C)c(C(=O)N2CCC(C#N)CC2)c1 ZINC000147046066 GG On-Demand Mild SFRP1 77 34 Cc1ccccc1NS(=O)(=O)c1ccc(C)c(C(=O)N2CCC(C#N)CC2)c1 ZINC000147046066 GG On-Demand Mild WNT3 61 32 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC(F)F)cc2OC(F)F)c1 ZINC000147046117 HI On-Demand Bother KCNMA1 31 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC(F)F)cc2OC(F)F)c1 ZINC000147046117 HI On-Demand Bother TAAR1 20 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC(F)F)cc2OC(F)F)c1 ZINC000147046117 HI On-Demand Bother AKR1C3 16 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC(F)F)cc2OC(F)F)c1 ZINC000147046117 HI On-Demand Bother AKR1C2 46 43 CCCCO[C@H](C)C(=O)N1CCN(c2cc(C)nc(C(C)C)n2)CC1 ZINC000147046138 EF On-Demand Anodyne P2RY12 68 38 COc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c(C(F)(F)F)c1 ZINC000147046164 FK On-Demand Anodyne RBP4 19 40 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1N1CCCC1=O ZINC000147046254 GD On-Demand Anodyne ADORA2B 39 40 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1N1CCCC1=O ZINC000147046254 GD On-Demand Anodyne MCHR1 22 42 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1N1CCCC1=O ZINC000147046254 GD On-Demand Anodyne ENPP1 74 37 Cc1nc(N)nc(N(C)CCc2ccccc2)n1 ZINC000147046283 BD For-Sale Anodyne DFR1 15 43 Cc1nc(N)nc(N(C)CCc2ccccc2)n1 ZINC000147046283 BD For-Sale Anodyne AOC3 19 46 CCCC[C@H](NC(N)=O)C(=O)N1CCN(c2cc(C)nc(C(C)C)n2)CC1 ZINC000147046334 GD On-Demand Anodyne P2RY12 197 44 CCCC[C@H](NC(N)=O)C(=O)N1CCN(c2cc(C)nc(C(C)C)n2)CC1 ZINC000147046334 GD On-Demand Anodyne TRY2_BOVIN 50 33 CC/C(=C\c1ccc(I)cc1)C(=O)O ZINC000147046338 DG In-Stock Anodyne DPEP1 31 44 COc1ccc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c(C(F)(F)F)c1 ZINC000147046340 FK On-Demand Anodyne RBP4 19 40 COc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c(C(F)(F)F)c1 ZINC000147046545 FK On-Demand Anodyne RBP4 19 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(c2cc(C)nc(C(C)C)n2)CC1 ZINC000147046549 GD On-Demand Anodyne P2RY12 197 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(c2cc(C)nc(C(C)C)n2)CC1 ZINC000147046549 GD On-Demand Anodyne TRY2_BOVIN 50 33 CCOc1cc(CNc2cccc(NC(=O)c3cc(Cl)ccc3O)c2)ccc1OC ZINC000147046557 IK For-Sale Anodyne CPT1A 60 40 CCOc1cc(CNc2cccc(NC(=O)c3cc(Cl)ccc3O)c2)ccc1OC ZINC000147046557 IK For-Sale Anodyne CPT2 40 34 CCOc1cc(CNc2cccc(NC(=O)c3cc(Cl)ccc3O)c2)ccc1OC ZINC000147046557 IK For-Sale Anodyne KCNMA1 38 44 CCOc1cc(CNc2cccc(NC(=O)c3cc(Cl)ccc3O)c2)ccc1OC ZINC000147046557 IK For-Sale Anodyne CPT1B 47 40 CCOc1cc(CNc2cccc(NC(=O)c3cc(Cl)ccc3O)c2)ccc1OC ZINC000147046557 IK For-Sale Anodyne PTGDR2 17 40 CCOc1cc(CNc2cccc(NC(=O)c3cc(Cl)ccc3O)c2)ccc1OC ZINC000147046557 IK For-Sale Anodyne DRTS_TRYCR 53 38 CCOc1cc(CNc2cccc(NC(=O)c3cc(Cl)ccc3O)c2)ccc1OC ZINC000147046557 IK For-Sale Anodyne PSBA 0 43 CCOc1cc(CNc2cccc(NC(=O)c3cc(Cl)ccc3O)c2)ccc1OC ZINC000147046557 IK For-Sale Anodyne KCNK3 69 52 CCOc1cc(CNc2cccc(NC(=O)c3cc(Cl)ccc3O)c2)ccc1OC ZINC000147046557 IK For-Sale Anodyne KCNK9 69 52 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(F)c(NC(=O)c3ccoc3C)c2)c1 ZINC000147046565 HI On-Demand Bother TAAR1 29 47 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(F)c(NC(=O)c3ccoc3C)c2)c1 ZINC000147046565 HI On-Demand Bother AKR1C2 45 37 O=C(Nc1cccc(CNS(=O)(=O)c2ccc3c(c2)CCCC3)c1)[C@@H]1CCCO1 ZINC000147046687 HG On-Demand Anodyne KCNA5 17 42 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1 ZINC000147046767 HF On-Demand Anodyne GHRHR 42 34 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1 ZINC000147046767 HF On-Demand Anodyne P2RY12 165 35 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1 ZINC000147046767 HF On-Demand Anodyne MCHR1 21 41 COC(=O)c1cc(C)ccc1NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147046791 FF On-Demand Anodyne ROCK2 35 50 O=C(Nc1cccc(CNS(=O)(=O)c2ccc3c(c2)CCC3)c1)[C@@H]1CCCO1 ZINC000147046906 HF On-Demand Anodyne KCNA5 16 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1 ZINC000147046970 HF On-Demand Anodyne GHRHR 42 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1 ZINC000147046970 HF On-Demand Anodyne P2RY12 165 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1 ZINC000147046970 HF On-Demand Anodyne MCHR1 21 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)NCc2ccc(F)cc2)cc1 ZINC000147046971 HE On-Demand Anodyne SSTR3 30 49 COC(=O)c1cc(C)ccc1NC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147046987 FF On-Demand Anodyne ROCK2 35 50 Cn1ccnc1COc1cnc(C(=O)Nc2ccc(F)c([C@]3(C)C=CSC(N)=N3)c2)cn1 ZINC000147047028 JF Annotated Anodyne BACE2 44 44 Cn1ccnc1COc1cnc(C(=O)Nc2ccc(F)c([C@]3(C)C=CSC(N)=N3)c2)cn1 ZINC000147047028 JF Annotated Anodyne BACE1 23 46 Cc1nc(N)nc(NCCCc2ccccc2)n1 ZINC000147047131 BD On-Demand Anodyne SIGMAR1 16 40 CC(C)C[C@@H](/C=C/C(=O)N1CCc2ccccc21)NC(=O)C1(N)CCOCC1 ZINC000147047154 GE For-Sale Anodyne PSMB2 41 31 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)NCc2ccc(F)cc2)cc1 ZINC000147047156 HE On-Demand Anodyne SSTR3 30 49 O=C(C[C@]1(C(=O)O)CCSC1)Nc1cccc(COC2CCCCC2)c1 ZINC000147047164 GI On-Demand Anodyne TIMP3 68 33 CN(C(=O)COc1ccc(C(N)=O)cc1)C1CCN(C(=O)OC(C)(C)C)CC1 ZINC000147047257 GE On-Demand Anodyne GPR119 51 55 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(-c2csc(C)n2)cc1 ZINC000147047364 FF On-Demand Anodyne NPY1R 22 40 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(-c2csc(C)n2)cc1 ZINC000147047364 FF On-Demand Anodyne PCSK5 46 38 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(-c2csc(C)n2)cc1 ZINC000147047364 FF On-Demand Anodyne FURIN 56 38 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(-c2csc(C)n2)cc1 ZINC000147047364 FF On-Demand Anodyne VHL 54 29 CCCOc1ccc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147047379 FG On-Demand Anodyne MTNR1A 41 42 CCCOc1ccc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147047379 FG On-Demand Anodyne ROCK2 27 41 CC(C)Oc1cccc(CC(=O)N2CCN(C)C[C@H]2c2ccccc2)c1 ZINC000147047480 FH On-Demand Anodyne P2RX7 15 41 CC(C)Oc1cccc(CC(=O)N2CCN(C)C[C@H]2c2ccccc2)c1 ZINC000147047480 FH On-Demand Anodyne COLA 31 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(-c2csc(C)n2)cc1 ZINC000147047552 FF On-Demand Anodyne NPY1R 22 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(-c2csc(C)n2)cc1 ZINC000147047552 FF On-Demand Anodyne PCSK5 46 38 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(-c2csc(C)n2)cc1 ZINC000147047552 FF On-Demand Anodyne FURIN 56 38 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(-c2csc(C)n2)cc1 ZINC000147047552 FF On-Demand Anodyne VHL 54 29 Cc1nc(N)nc(N(C)Cc2ccccc2)n1 ZINC000147047558 BD On-Demand Anodyne DHFR 17 44 Cc1nc(N)nc(N(C)Cc2ccccc2)n1 ZINC000147047558 BD On-Demand Anodyne DFR1 25 40 Cc1nc(N)nc(N(C)Cc2ccccc2)n1 ZINC000147047558 BD On-Demand Anodyne DRTS_TOXGO 28 46 Cc1nc(N)nc(N(C)Cc2ccccc2)n1 ZINC000147047558 BD On-Demand Anodyne DYR_PNECA 33 46 CCCOCC(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147047797 DD On-Demand Anodyne OPRM1 16 50 CCCOCC(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147047797 DD On-Demand Anodyne OPRL1 38 50 CCCOCC(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147047797 DD On-Demand Anodyne AKT2 28 41 CCCOCC(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147047797 DD On-Demand Anodyne PLD1 104 48 CCCOCC(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147047797 DD On-Demand Anodyne PLD2 87 48 CCCOCC(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147047797 DD On-Demand Anodyne CALCRL 70 46 CN(C)C(=N)NCCCC[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147047824 IG For-Sale Anodyne FOLH1 54 38 CN(C)C(=N)NCCCC[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147047824 IG For-Sale Anodyne KLK3 47 32 CN(C)C(=N)NCCCC[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147047824 IG For-Sale Anodyne C3AR1 90 39 CN(C)C(=N)NCCCC[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147047824 IG For-Sale Anodyne FURIN 45 36 CN(C)C(=N)NCCCC[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147047824 IG For-Sale Anodyne CAPN1 22 48 CN(C)C(=N)NCCCC[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147047824 IG For-Sale Anodyne POLG_WNV 68 37 CN(C)C(=N)NCCCC[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147047824 IG For-Sale Anodyne NPFFR1 51 32 O=[N+]([O-])c1ccc(C[P@](=O)(O)Oc2ccccc2)cc1 ZINC000147047913 CG For-Sale Bother CCR3 15 40 O=[N+]([O-])c1ccc(C[P@](=O)(O)Oc2ccccc2)cc1 ZINC000147047913 CG For-Sale Bother LAP3 17 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048015 FD On-Demand Anodyne SSTR2 17 50 CCCC[C@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048015 FD On-Demand Anodyne OPRL1 17 46 CCCC[C@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048015 FD On-Demand Anodyne GHRHR 41 31 CCCC[C@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048015 FD On-Demand Anodyne P2RY12 175 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048015 FD On-Demand Anodyne AKT2 27 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048015 FD On-Demand Anodyne PLD1 103 48 CCCC[C@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048015 FD On-Demand Anodyne PLD2 85 48 CCCC[C@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048015 FD On-Demand Anodyne CALCRL 79 56 C[C@@]1(c2cc(NC(=O)c3cnc(-n4ccnn4)cn3)ccc2F)C=CSC(N)=N1 ZINC000147048032 HE Annotated Anodyne BACE2 46 49 C[C@@]1(c2cc(NC(=O)c3cnc(-n4ccnn4)cn3)ccc2F)C=CSC(N)=N1 ZINC000147048032 HE Annotated Anodyne BACE1 24 59 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048233 FD On-Demand Anodyne SSTR2 17 50 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048233 FD On-Demand Anodyne OPRM1 17 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048233 FD On-Demand Anodyne OPRL1 35 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048233 FD On-Demand Anodyne GHRHR 41 31 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048233 FD On-Demand Anodyne P2RY12 175 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048233 FD On-Demand Anodyne AKT2 27 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048233 FD On-Demand Anodyne PLD1 103 48 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048233 FD On-Demand Anodyne CTSS 15 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048233 FD On-Demand Anodyne PLD2 85 48 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(n2c(=O)[nH]c3ccccc32)CC1 ZINC000147048233 FD On-Demand Anodyne CALCRL 79 56 CC(=O)O[C@@H]1CN(C(=O)OCc2ccccc2)[C@@H]2CO[C@H](c3ccccc3)O[C@@H]2[C@@H]1OC(C)=O ZINC000147048287 JF For-Sale Anodyne KLK5 45 42 CC(=O)O[C@@H]1CN(C(=O)OCc2ccccc2)[C@@H]2CO[C@H](c3ccccc3)O[C@@H]2[C@@H]1OC(C)=O ZINC000147048287 JF For-Sale Anodyne SLC12A5 41 32 NC(=O)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147048453 HD On-Demand Anodyne KCNA5 15 44 NC(=O)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147048453 HD On-Demand Anodyne ST14 47 33 Cc1c(C(=O)NC[C@@H](C)N2CCCC2)nnn1-c1ccccc1 ZINC000147048535 DD On-Demand Anodyne SLC5A1 22 41 NC(=O)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147048658 HD On-Demand Anodyne KCNA5 15 44 NC(=O)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147048658 HD On-Demand Anodyne ST14 47 33 CNC(=O)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147048859 HD On-Demand Anodyne KCNA5 17 46 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(F)c(C(F)(F)F)c1 ZINC000147048898 FG On-Demand Anodyne SLC1A2 44 39 O=[N+]([O-])c1ccc(CP(=O)(Oc2ccccc2)Oc2ccccc2)cc1 ZINC000147048924 FK For-Sale Bother CCR3 22 42 CNC(=O)c1ccc(S(=O)(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147049035 HD On-Demand Anodyne KCNA5 17 46 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(OCc2ccccn2)c(Cl)c1 ZINC000147049104 HH On-Demand Anodyne EGFR 17 44 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(OCc2ccccn2)c(Cl)c1 ZINC000147049104 HH On-Demand Anodyne ERBB2 37 42 O=C(C[C@]1(C(=O)O)CCSC1)Nc1ccc(OCc2ccccn2)c(Cl)c1 ZINC000147049104 HH On-Demand Anodyne GRM4 51 45 CCOc1cc(N2CCCC2)ccc1C(=O)c1ccccc1C(=O)O ZINC000147049107 EH For-Sale Anodyne ABCC8 22 48 CCOc1cc(N2CCCC2)ccc1C(=O)c1ccccc1C(=O)O ZINC000147049107 EH For-Sale Anodyne KCNQ2 60 38 CCOc1cc(N2CCCC2)ccc1C(=O)c1ccccc1C(=O)O ZINC000147049107 EH For-Sale Anodyne HCN1 57 36 CCOc1cc(N2CCCC2)ccc1C(=O)c1ccccc1C(=O)O ZINC000147049107 EH For-Sale Anodyne HCN4 45 35 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)c3cccc4cnccc34)c2)CCO1 ZINC000147049227 HF On-Demand Anodyne P2RX7 40 51 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)c3cccc4cnccc34)c2)CCO1 ZINC000147049227 HF On-Demand Anodyne NPY2R 40 38 CCO[C@@H]1CCCN(C(=O)Nc2ccc(OC(C)C)c(Cl)c2)C1 ZINC000147049283 EI On-Demand Anodyne EPHX2 21 40 C[C@H]1CN(Cc2cccc(CNS(=O)(=O)c3cccc4cnccc34)c2)CCO1 ZINC000147049413 HF On-Demand Anodyne P2RX7 40 51 C[C@H]1CN(Cc2cccc(CNS(=O)(=O)c3cccc4cnccc34)c2)CCO1 ZINC000147049413 HF On-Demand Anodyne NPY2R 40 38 CC[C@H](Cl)C(=O)c1c(F)cccc1F ZINC000147049414 BG For-Sale Anodyne CES2 29 50 CC[C@H](Cl)C(=O)c1c(F)cccc1F ZINC000147049414 BG For-Sale Anodyne DAC 22 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(F)c(NC(=O)C3CCCCC3)c2)c1 ZINC000147049452 HJ On-Demand Bother TAAR1 32 46 CCO[C@H]1CCCN(C(=O)Nc2ccc(OC(C)C)c(Cl)c2)C1 ZINC000147049473 EI On-Demand Anodyne EPHX2 21 40 CC[C@@H](Cl)C(=O)c1c(F)cccc1F ZINC000147049600 BG For-Sale Anodyne CES2 29 50 CC[C@@H](Cl)C(=O)c1c(F)cccc1F ZINC000147049600 BG For-Sale Anodyne DAC 22 40 C=CCN(Cc1ccccc1)C(N)=O ZINC000147049625 AD On-Demand Mild SLC1A6 51 33 C=CCN(Cc1ccccc1)C(N)=O ZINC000147049625 AD On-Demand Mild SLC1A7 51 33 COc1ccc(S(=O)(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)c(C)c1 ZINC000147049642 HF On-Demand Anodyne DRD4 18 42 COc1ccccc1-c1cc(=O)c2c(OC)cc(OC)c(OC)c2o1 ZINC000147049649 EG Annotated Anodyne AKR1B1 0 60 COc1ccccc1-c1cc(=O)c2c(OC)cc(OC)c(OC)c2o1 ZINC000147049649 EG Annotated Anodyne CYP1B1 91 67 COc1ccccc1-c1cc(=O)c2c(OC)cc(OC)c(OC)c2o1 ZINC000147049649 EG Annotated Anodyne CYP1A1 63 67 COc1ccccc1-c1cc(=O)c2c(OC)cc(OC)c(OC)c2o1 ZINC000147049649 EG Annotated Anodyne CYP1A2 49 67 COc1ccccc1-c1cc(=O)c2c(OC)cc(OC)c(OC)c2o1 ZINC000147049649 EG Annotated Anodyne ABCG2 0 52 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(Cl)ccc2C(=O)N2CCCC2)c1 ZINC000147049657 HH On-Demand Bother F10 17 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(Cl)ccc2C(=O)N2CCCC2)c1 ZINC000147049657 HH On-Demand Bother KCNMA1 36 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(Cl)ccc2C(=O)N2CCCC2)c1 ZINC000147049657 HH On-Demand Bother TAAR1 23 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(Cl)ccc2C(=O)N2CCCC2)c1 ZINC000147049657 HH On-Demand Bother AKR1C3 21 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(Cl)ccc2C(=O)N2CCCC2)c1 ZINC000147049657 HH On-Demand Bother AKR1C2 46 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(Cl)ccc2C(=O)N2CCCC2)c1 ZINC000147049657 HH On-Demand Bother GPR35 37 40 CC(C)(C)CNS(=O)(=O)c1ccccc1[N+](=O)[O-] ZINC000147049834 CD On-Demand Bother COLA 79 35 CCOC[C@H](C)NC(=O)Nc1ccccc1-n1nc(C)cc1C ZINC000147049885 DG On-Demand Anodyne KCNQ2 42 33 CCOC[C@H](C)NC(=O)Nc1ccccc1-n1nc(C)cc1C ZINC000147049885 DG On-Demand Anodyne P2RY1 21 44 COc1ccc(N2C[C@H](C(=O)N3CCC(C#N)CC3)CC2=O)c(OC)c1 ZINC000147049920 FD On-Demand Mild SSTR1 47 35 CN(C)CCNc1cc(N2CCCCCC2)ncn1 ZINC000147050052 CD For-Sale Anodyne HRH4 17 55 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(Cl)cc2C(=O)N2CCCC2)c1 ZINC000147050081 HH On-Demand Bother F10 36 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(Cl)cc2C(=O)N2CCCC2)c1 ZINC000147050081 HH On-Demand Bother KCNMA1 36 45 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(Cl)cc2C(=O)N2CCCC2)c1 ZINC000147050081 HH On-Demand Bother TAAR1 23 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(Cl)cc2C(=O)N2CCCC2)c1 ZINC000147050081 HH On-Demand Bother AKR1C3 21 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(Cl)cc2C(=O)N2CCCC2)c1 ZINC000147050081 HH On-Demand Bother AKR1C2 30 42 N#CC1CCN(C(=O)[C@@H]2CC(=O)N(C3CCCC3)C2)CC1 ZINC000147050145 CD On-Demand Mild INHA 36 42 COc1ccc(C(=O)N2CCOCC2)cc1NC(=O)C[C@]1(C(=O)O)CCSC1 ZINC000147050177 HD On-Demand Anodyne LRRK2 29 41 CNc1nc(N)nc(Nc2ccccc2)n1 ZINC000147050226 BD For-Sale Anodyne CYSP_TRYCR 0 63 CNc1nc(N)nc(Nc2ccccc2)n1 ZINC000147050226 BD For-Sale Anodyne AT1 0 40 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000147050296 DB On-Demand Anodyne F2 18 43 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000147050296 DB On-Demand Anodyne P2RY12 91 35 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000147050296 DB On-Demand Anodyne TRY2_BOVIN 68 43 Cc1cc(C)n(-c2ccccc2NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)n1 ZINC000147050369 HI On-Demand Anodyne NOS2 88 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000147050485 DB On-Demand Anodyne F2 18 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000147050485 DB On-Demand Anodyne P2RY12 91 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(C)(=O)=O)CC1 ZINC000147050485 DB On-Demand Anodyne TRY2_BOVIN 68 43 CC(C)CN(Cc1ccc(Br)cc1F)S(=O)(=O)c1ccccc1Cl ZINC000147050501 IK For-Sale Anodyne RORC 26 40 CC(=O)Nc1nc2cc(Cl)ccc2o1 ZINC000147050537 BE For-Sale Anodyne CETP 0 44 CC(=O)Nc1nc2cc(Cl)ccc2o1 ZINC000147050537 BE For-Sale Anodyne FBP1 34 54 CC(=O)Nc1nc2cc(Cl)ccc2o1 ZINC000147050537 BE For-Sale Anodyne AGPAT2 50 49 CC(=O)Nc1nc2cc(Cl)ccc2o1 ZINC000147050537 BE For-Sale Anodyne IMDH_CRYPV 35 41 COC(=O)COc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147050619 HD On-Demand Bother UREA_CANEN 17 40 COC(=O)COc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147050619 HD On-Demand Bother USP7 44 36 COC(=O)COc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147050619 HD On-Demand Bother USP47 55 36 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne MME 27 41 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne LTA4H 15 41 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne BMP1 59 35 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne KLK3 40 31 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne CTSB 53 43 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne PAPA1_CARPA 58 39 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne CTSK 27 44 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne CAPNS1 57 36 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne CTSS 19 45 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne CAPN1 68 40 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne CAPN2 97 42 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne CTSC 17 41 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne NPR 58 36 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne SLC12A5 64 37 CC[C@H](OC)C(=O)OCc1ccccc1 ZINC000147050625 BE On-Demand Anodyne PDS 46 33 Nc1cnc(-c2ccn3c(-c4cccc(NC(=O)NCC(F)(F)F)c4)cnc3c2)cn1 ZINC000147050689 IH Annotated Anodyne RIPK1 56 34 O=C(Nc1ccc(Cl)c(Cl)c1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147050714 EF On-Demand Anodyne ENV 43 33 N#CC1CCN(C(=O)[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147050770 EF On-Demand Mild CTSG 29 40 N#CC1CCN(C(=O)[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147050770 EF On-Demand Mild CCR1 26 42 N#CC1CCN(C(=O)[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147050770 EF On-Demand Mild CTRB1 33 40 N#CC1CCN(C(=O)[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147050770 EF On-Demand Mild MTTP 53 41 N#CC1CCN(C(=O)[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147050770 EF On-Demand Mild FAP 0 43 Nc1cc(C(=O)O)c(N)cc1O ZINC000147050782 AC For-Sale Anodyne AKR1C2 40 35 Nc1cc(C(=O)O)c(N)cc1O ZINC000147050782 AC For-Sale Anodyne AKR1C1 43 35 CC(C)(NC(=O)CCl)c1cccc(Br)c1 ZINC000147050823 CG For-Sale Reactive GUAB 0 41 CC(C)(NC(=O)CCl)c1cccc(Br)c1 ZINC000147050823 CG For-Sale Reactive IMDH_CRYPV 62 42 O=C(O)c1cc2c(CN3CC[C@@H](O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147050851 FE For-Sale Anodyne CCR3 25 40 Nc1ccc(-c2c(F)cccc2F)nc1C(=O)Nc1cnccc1-c1cccnc1N ZINC000147050904 HH Annotated Anodyne PIM1 38 49 Nc1ccc(-c2c(F)cccc2F)nc1C(=O)Nc1cnccc1-c1cccnc1N ZINC000147050904 HH Annotated Anodyne PIM2 21 49 Nc1ccc(-c2c(F)cccc2F)nc1C(=O)Nc1cnccc1-c1cccnc1N ZINC000147050904 HH Annotated Anodyne PIM3 25 49 O=C(Nc1ccc(Cl)c(Cl)c1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147050911 EF On-Demand Anodyne ENV 43 33 O=C(O)c1cc2c(CN3CC[C@H](O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147051022 FE For-Sale Anodyne CCR3 25 40 CN1[C@@H](C(=O)NCC[C@H](O)CO)[C@H](c2cccc(Cl)c2)[C@@]2(C(=O)Nc3cc(Cl)c(F)cc32)[C@H]1CCC1CCCC1 ZINC000147051070 KJ Annotated Anodyne MDM2 80 65 O=C(Nc1ccc(Cl)c(Cl)c1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147051092 EF On-Demand Anodyne ENV 43 33 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051115 FG On-Demand Anodyne ANPEP 19 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051115 FG On-Demand Anodyne NPY1R 23 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051115 FG On-Demand Anodyne ACACB 16 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051115 FG On-Demand Anodyne GRIA1 57 33 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051115 FG On-Demand Anodyne PCSK5 60 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051115 FG On-Demand Anodyne FURIN 68 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051115 FG On-Demand Anodyne PROC 41 37 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051115 FG On-Demand Anodyne PSMB5 19 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051115 FG On-Demand Anodyne LEF 59 37 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051115 FG On-Demand Anodyne POLG_WNV 60 32 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)CCc3ccccc3)c2)CCO1 ZINC000147051183 GF On-Demand Anodyne DRD4 17 44 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)CCc3ccccc3)c2)CCO1 ZINC000147051183 GF On-Demand Anodyne SIGMAR1 17 40 CSc1nc(N2C[C@H]3[C@@H](C2)[C@@H]3C(=O)O)ccc1C(=O)NC1C2CC3CC(C2)CC1C3 ZINC000147051207 IG Annotated Anodyne HSD11B1 41 70 C[C@@H]1CCC[C@H](OCc2cccc(NC(=O)C[C@]3(C(=O)O)CCSC3)c2)C1 ZINC000147051230 GI On-Demand Anodyne TIMP3 70 33 O=C(Nc1ccc(Cl)c(Cl)c1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147051289 EF On-Demand Anodyne ENV 43 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051323 FG On-Demand Anodyne ANPEP 19 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051323 FG On-Demand Anodyne NPY1R 23 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051323 FG On-Demand Anodyne ACACB 16 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051323 FG On-Demand Anodyne GRIA1 57 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051323 FG On-Demand Anodyne PCSK5 60 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051323 FG On-Demand Anodyne FURIN 68 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051323 FG On-Demand Anodyne PROC 41 37 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051323 FG On-Demand Anodyne PSMB5 19 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051323 FG On-Demand Anodyne LEF 59 37 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147051323 FG On-Demand Anodyne POLG_WNV 60 32 C[C@@H]1CCC[C@@H](OCc2cccc(NC(=O)C[C@]3(C(=O)O)CCSC3)c2)C1 ZINC000147051619 GI On-Demand Anodyne TIMP3 70 33 Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4ccc(F)cc4C(F)(F)F)C[C@H]3C2)n1 ZINC000147051637 HG Annotated Anodyne P2RX7 15 41 COc1ccc(S(=O)(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1F ZINC000147051661 HF On-Demand Anodyne DRD4 22 41 Cc1cc(C)nc(N2C[C@H]3CN(C(=O)c4ccc(F)cc4C(F)(F)F)C[C@@H]3C2)n1 ZINC000147051830 HG Annotated Anodyne P2RX7 15 41 COc1ccc(S(=O)(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1F ZINC000147051862 HF On-Demand Anodyne DRD4 22 41 COc1ccc(CN(C(=O)[C@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147051888 EI On-Demand Anodyne BMP1 52 39 COc1ccc(CN(C(=O)[C@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147051888 EI On-Demand Anodyne CCR5 48 33 COc1ccc(CN(C(=O)[C@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147051888 EI On-Demand Anodyne MMP1 19 40 COc1ccc(CN(C(=O)[C@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147051888 EI On-Demand Anodyne ACAT 47 40 Cc1nc(N)nc(N(C)c2ccccc2)n1 ZINC000147051891 BD For-Sale Anodyne DYR_PNECA 25 49 Cc1nc(N)nc(N(C)c2ccccc2)n1 ZINC000147051891 BD For-Sale Anodyne TUBB3 43 37 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne CHRM2 24 42 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne DRD2 28 45 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne DRD4 54 41 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne ACHE 44 45 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne HRH1 22 42 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne OPRM1 22 42 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne DRD3 25 45 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne OPRK1 17 40 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne SLC6A3 15 41 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne HTR4 28 44 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne LTA4H 19 46 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne HRH3 26 41 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne SIGMAR1 68 49 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne CCR3 46 38 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne CCR5 46 43 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne EPHX2 26 42 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne TRPV4 15 40 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne MCHR1 35 42 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne CACNA1G 54 56 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne BIRC2 33 42 C[C@H](CNC(=O)C1CCN(Cc2ccccc2)CC1)N1CCCC1 ZINC000147051948 EE On-Demand Anodyne NPFFR1 49 35 Cc1cc(C)nc(N2C[C@@H]3CN(C(=O)c4ccc(F)cc4C(F)(F)F)C[C@H]3C2)n1 ZINC000147052010 HG Annotated Anodyne P2RX7 15 41 CN(Cc1ccc2c(c1)OCO2)c1nc(N)nc(N)n1 ZINC000147052291 CC On-Demand Anodyne HSP90AB1 15 40 Cc1ccc(CN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)C2CC2)o1 ZINC000147052328 EJ On-Demand Anodyne MDM2 51 33 CCC1CCC(C2CCC(N)CC2)CC1 ZINC000147052475 BH For-Sale Anodyne SPDS 0 41 COc1ccc(-c2ccc(C(C)=O)cc2N)cc1 ZINC000147052481 BG For-Sale Anodyne HDAC2 17 40 COc1ccc(-c2ccc(C(C)=O)cc2N)cc1 ZINC000147052481 BG For-Sale Anodyne AKR1C3 17 45 COc1ccc(-c2ccc(C(C)=O)cc2N)cc1 ZINC000147052481 BG For-Sale Anodyne AKR1C2 19 45 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne GRIA1 81 36 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne PLA2G4B 68 35 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne FAAH 22 47 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne PCSK5 56 37 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne FURIN 68 34 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne CAPN2 15 40 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne TPSAB1 47 35 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne LEF 56 33 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne POLG_WNV 78 36 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne ASAH1 54 30 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne QRFPR 45 40 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne NPFFR1 40 31 CCCC[C@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052507 EE On-Demand Anodyne HPN 68 33 Cc1cccc(Oc2ncccc2NC(=O)C(=O)NC[C@@H]2CCCCO2)c1C ZINC000147052521 GG On-Demand Anodyne P2RY1 51 35 Cc1ccc(CN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)C2CC2)o1 ZINC000147052527 EJ On-Demand Anodyne MDM2 51 33 Cc1ccc(S(=O)(=O)n2ccc3c(N(C)[C@@H]4CCCCN(C(=O)OC(C)(C)C)C4)ncnc32)cc1 ZINC000147052616 JI For-Sale Anodyne GPR119 38 46 COCc1nc(C(=O)Nc2c(C)n(C)n(-c3ccccc3)c2=O)cs1 ZINC000147052693 FE On-Demand Anodyne FPR2 45 47 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne GRIA1 81 36 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne PLA2G4B 68 35 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne FAAH 22 47 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne PCSK5 56 37 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne FURIN 68 34 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne CAPN2 15 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne TPSAB1 47 35 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne LEF 56 33 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne POLG_WNV 78 36 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne ASAH1 54 30 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne QRFPR 45 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne NPFFR1 40 31 CCCC[C@@H](NC(N)=O)C(=O)NCCCCOc1ccc(F)cc1 ZINC000147052703 EE On-Demand Anodyne HPN 68 33 Cc1cccc(Oc2ncccc2NC(=O)C(=O)NC[C@H]2CCCCO2)c1C ZINC000147052721 GG On-Demand Anodyne P2RY1 51 35 Cc1nn(-c2ccc(C(F)(F)F)cn2)c(C)c1CC(=O)NC[C@H](C)N1CCCC1 ZINC000147052732 HG On-Demand Anodyne P2RX7 35 45 Cc1ccc(CN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)C2CC2)o1 ZINC000147052741 EJ On-Demand Anodyne MDM2 51 33 Cc1ccc(S(=O)(=O)n2ccc3c(N(C)[C@H]4CCCCN(C(=O)OC(C)(C)C)C4)ncnc32)cc1 ZINC000147052825 JI For-Sale Anodyne GPR119 38 46 COc1cc(C)ccc1Oc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cn1 ZINC000147052830 HG On-Demand Anodyne PDGFRB 47 36 COc1cc(C)ccc1Oc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cn1 ZINC000147052830 HG On-Demand Anodyne ADORA2B 24 40 COc1cc(C)ccc1Oc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cn1 ZINC000147052830 HG On-Demand Anodyne PDGFRA 50 39 COc1cc(C)ccc1Oc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cn1 ZINC000147052830 HG On-Demand Anodyne ENPP1 73 36 COC(=O)CNS(=O)(=O)c1c(C(=O)OC)sc2ccccc12 ZINC000147052878 ED On-Demand Anodyne FAS 20 44 Cc1ccc(CN(C(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)C2CC2)o1 ZINC000147052934 EJ On-Demand Anodyne MDM2 51 33 Cc1ccc(S(=O)(=O)N2CCN(CC(=O)NC[C@H](C)N3CCCC3)CC2)cc1 ZINC000147052951 HC On-Demand Anodyne EPHX2 17 41 Cc1ccc(S(=O)(=O)N2CCN(CC(=O)NC[C@H](C)N3CCCC3)CC2)cc1 ZINC000147052951 HC On-Demand Anodyne TGM2 52 38 Cc1ccc(S(=O)(=O)N2CCN(CC(=O)NC[C@H](C)N3CCCC3)CC2)cc1 ZINC000147052951 HC On-Demand Anodyne F13A1 63 38 Cc1c(C(=O)N2CCC(C#N)CC2)cnn1-c1ccccc1 ZINC000147053031 CF On-Demand Mild SLC9A2 0 47 C=CCCOCC(=O)Nc1ccc(Oc2ccc(C)cc2OC)nc1 ZINC000147053232 EH On-Demand Mild ENPP1 64 33 C[C@@]1(c2cc(NC(=O)c3ccc(F)cn3)ccc2F)C=CSC(N)=N1 ZINC000147053270 FG Annotated Anodyne BACE2 60 58 C[C@@]1(c2cc(NC(=O)c3ccc(F)cn3)ccc2F)C=CSC(N)=N1 ZINC000147053270 FG Annotated Anodyne BACE1 29 58 COc1ccc(C(=O)N(C)C)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147053316 FD On-Demand Anodyne OXTR 20 40 Cc1cc(C(=O)Nc2ccc3c(c2)OCCO3)cc([N+](=O)[O-])c1 ZINC000147053348 DF On-Demand Bother PLK1 0 44 Cc1cc(S(C)(=O)=O)ccc1OS(=O)(=O)C(F)(F)F ZINC000147053483 DD For-Sale Unstable PTGS2 46 46 Cc1cc(S(C)(=O)=O)ccc1OS(=O)(=O)C(F)(F)F ZINC000147053483 DD For-Sale Unstable PTGDR2 18 40 Cn1c(=O)n(C)c2cc(NC(=O)C[C@@](C)(C(=O)O)c3ccccc3)ccc21 ZINC000147053488 FE On-Demand Anodyne ECE1 34 42 Cn1c(=O)n(C)c2cc(NC(=O)C[C@@](C)(C(=O)O)c3ccccc3)ccc21 ZINC000147053488 FE On-Demand Anodyne CALCRL 56 38 COc1ccc(C(=O)N(C)C)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147053496 FD On-Demand Anodyne OXTR 20 40 N#CC1CCN(C(=O)c2ccc3n[nH]nc3c2)CC1 ZINC000147053517 CD On-Demand Mild L3MBTL3 73 41 N#CC1CCN(C(=O)c2ccc3n[nH]nc3c2)CC1 ZINC000147053517 CD On-Demand Mild HPGD 42 36 COc1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1C=O ZINC000147053521 CF For-Sale Anodyne PTGS1 28 42 COc1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1C=O ZINC000147053521 CF For-Sale Anodyne PTGS2 75 51 COc1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1C=O ZINC000147053521 CF For-Sale Anodyne LOX1.1 21 40 N#CC1CCN(C(=O)CCn2c(=O)[nH]c(=O)c3ccccc32)CC1 ZINC000147053708 EC On-Demand Mild PARP1 18 49 Cc1cc(C(=O)NC23CC4CC(CC(C4)C2)C3)cc([N+](=O)[O-])c1 ZINC000147053736 DH On-Demand Bother CNR2 27 43 Cc1cc(C(=O)NC23CC4CC(CC(C4)C2)C3)cc([N+](=O)[O-])c1 ZINC000147053736 DH On-Demand Bother EPHX2 64 42 CCNC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147053759 EH On-Demand Anodyne PRNP 16 43 CCNC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147053759 EH On-Demand Anodyne MDM2 45 36 CCNC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147053759 EH On-Demand Anodyne NAMPT 26 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)C(=O)NC(C)C)CC1 ZINC000147053778 FB On-Demand Anodyne P2RY12 160 36 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)C(=O)NC(C)C)CC1 ZINC000147053778 FB On-Demand Anodyne NOD1 58 35 N#CC1CCN(C(=O)[C@H]2CCCN(C(=O)c3ccc(F)cc3)C2)CC1 ZINC000147053907 EE On-Demand Mild L3MBTL1 0 43 N#CC1CCN(C(=O)[C@H]2CCCN(C(=O)c3ccc(F)cc3)C2)CC1 ZINC000147053907 EE On-Demand Mild MBTD1 0 42 CCNC(=O)c1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147053966 EH On-Demand Anodyne PRNP 16 43 CCNC(=O)c1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147053966 EH On-Demand Anodyne MDM2 45 36 CCNC(=O)c1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147053966 EH On-Demand Anodyne NAMPT 26 41 COc1ccc2nc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)sc2c1 ZINC000147053969 EH On-Demand Bother LCK 34 47 COc1ccc2nc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)sc2c1 ZINC000147053969 EH On-Demand Bother CSNK1D 50 53 COc1ccc2nc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)sc2c1 ZINC000147053969 EH On-Demand Bother NMT1 30 41 COc1ccc2nc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)sc2c1 ZINC000147053969 EH On-Demand Bother PIK3CA 18 46 COc1ccc2nc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)sc2c1 ZINC000147053969 EH On-Demand Bother ITK 15 41 COc1ccc2nc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)sc2c1 ZINC000147053969 EH On-Demand Bother HSD17B1 27 40 COc1ccc2nc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)sc2c1 ZINC000147053969 EH On-Demand Bother PIK3CG 18 48 COc1ccc2nc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)sc2c1 ZINC000147053969 EH On-Demand Bother TAAR1 21 46 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)C(=O)NC(C)C)CC1 ZINC000147053987 FB On-Demand Anodyne P2RY12 160 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)C(=O)NC(C)C)CC1 ZINC000147053987 FB On-Demand Anodyne NOD1 58 35 CCCCC[N+](CC)(CC)CCO ZINC000147054042 AE For-Sale Bother SLC22A1 25 60 CCNC(=O)c1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147054163 EH On-Demand Anodyne PRNP 16 43 CCNC(=O)c1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147054163 EH On-Demand Anodyne MDM2 45 36 CCNC(=O)c1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147054163 EH On-Demand Anodyne NAMPT 26 41 COc1ccc2cnn(C[C@@H](C)N)c2c1 ZINC000147054188 BD For-Sale Anodyne NPBWR1 54 33 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccccn2)CC1 ZINC000147054224 EC On-Demand Anodyne GHRHR 41 33 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccccn2)CC1 ZINC000147054224 EC On-Demand Anodyne P2RY12 199 40 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccccn2)CC1 ZINC000147054224 EC On-Demand Anodyne TRY2_BOVIN 45 33 COc1ccc(-c2ccc(C(C)=O)cc2F)cc1 ZINC000147054282 BH For-Sale Anodyne RARB 17 43 COc1ccc(-c2ccc(C(C)=O)cc2F)cc1 ZINC000147054282 BH For-Sale Anodyne GYS1 47 33 COc1ccc(-c2ccc(C(C)=O)cc2F)cc1 ZINC000147054282 BH For-Sale Anodyne HDAC2 17 40 COc1ccc(-c2ccc(C(C)=O)cc2F)cc1 ZINC000147054282 BH For-Sale Anodyne AKR1C3 20 45 COc1ccc(-c2ccc(C(C)=O)cc2F)cc1 ZINC000147054282 BH For-Sale Anodyne AKR1C2 23 45 CCNC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147054334 GH On-Demand Anodyne NAMPT 22 41 C=CCCOCC(=O)Nc1cccc(C(=O)NCC(N)=O)c1 ZINC000147054391 DC On-Demand Mild KCNK3 59 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccccn2)CC1 ZINC000147054409 EC On-Demand Anodyne GHRHR 41 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccccn2)CC1 ZINC000147054409 EC On-Demand Anodyne P2RY12 199 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccccn2)CC1 ZINC000147054409 EC On-Demand Anodyne TRY2_BOVIN 45 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccccn2)CC1 ZINC000147054409 EC On-Demand Anodyne CCKAR 17 40 CCOc1cccc(CC(=O)O)c1O ZINC000147054506 AD For-Sale Anodyne PTGER2 32 42 CCOc1cccc(CC(=O)O)c1O ZINC000147054506 AD For-Sale Anodyne CXCL8 34 41 CCOc1cccc(CC(=O)O)c1O ZINC000147054506 AD For-Sale Anodyne FABP5 29 45 Cn1c(=O)n(C)c2cc(NC(=O)C[C@H](C(=O)O)c3ccccc3)ccc21 ZINC000147054521 FE On-Demand Anodyne SLC1A1 55 39 Cn1c(=O)n(C)c2cc(NC(=O)C[C@H](C(=O)O)c3ccccc3)ccc21 ZINC000147054521 FE On-Demand Anodyne SLC1A3 58 39 Cn1c(=O)n(C)c2cc(NC(=O)C[C@H](C(=O)O)c3ccccc3)ccc21 ZINC000147054521 FE On-Demand Anodyne SLC1A2 80 39 CCNC(=O)c1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147054533 GH On-Demand Anodyne NAMPT 22 41 CCN1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147054603 GD On-Demand Anodyne LTA4H 62 48 CCN1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147054603 GD On-Demand Anodyne ADORA2B 49 46 CCN1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147054603 GD On-Demand Anodyne HRH3 15 44 CCN1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147054603 GD On-Demand Anodyne FAAH 21 46 CCN1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147054603 GD On-Demand Anodyne ACR 50 38 CCN1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147054603 GD On-Demand Anodyne MCHR1 35 47 CCN1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147054603 GD On-Demand Anodyne CACNA1G 15 43 CCN1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147054603 GD On-Demand Anodyne NPFFR1 45 38 CCN1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147054603 GD On-Demand Anodyne NOD1 31 42 CCN1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147054603 GD On-Demand Anodyne NOD2 49 47 CCNC(=O)c1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)cc1 ZINC000147054737 GH On-Demand Anodyne NAMPT 22 41 CCN1CCN(Cc2ccccc2CNC(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147054799 HD On-Demand Anodyne SLC9A1 44 31 CCN1CCN(Cc2ccccc2CNC(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147054799 HD On-Demand Anodyne NPFFR1 41 35 CCCC[C@H](NC(N)=O)C(=O)N1CCN(c2cccc(C)c2)CC1 ZINC000147054865 ED On-Demand Anodyne F2 25 46 CCCC[C@H](NC(N)=O)C(=O)N1CCN(c2cccc(C)c2)CC1 ZINC000147054865 ED On-Demand Anodyne GHRHR 41 32 CCCC[C@H](NC(N)=O)C(=O)N1CCN(c2cccc(C)c2)CC1 ZINC000147054865 ED On-Demand Anodyne P2RY12 205 52 CCCC[C@H](NC(N)=O)C(=O)N1CCN(c2cccc(C)c2)CC1 ZINC000147054865 ED On-Demand Anodyne TRY2_BOVIN 85 35 CCNC(=O)c1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147054919 FF On-Demand Anodyne MTNR1A 37 42 CCNC(=O)c1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147054919 FF On-Demand Anodyne MTNR1B 35 40 CCNC(=O)c1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147054919 FF On-Demand Anodyne ROCK2 33 53 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(c2cccc(C)c2)CC1 ZINC000147055049 ED On-Demand Anodyne F2 25 46 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(c2cccc(C)c2)CC1 ZINC000147055049 ED On-Demand Anodyne GHRHR 41 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(c2cccc(C)c2)CC1 ZINC000147055049 ED On-Demand Anodyne P2RY12 205 52 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(c2cccc(C)c2)CC1 ZINC000147055049 ED On-Demand Anodyne TRY2_BOVIN 85 35 C[C@@H](CNC(=O)c1ccc(N(C)c2ccccc2)nc1)N1CCCC1 ZINC000147055095 EG On-Demand Anodyne RXRA 40 36 CCNC(=O)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147055099 FF On-Demand Anodyne MTNR1A 37 42 CCNC(=O)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147055099 FF On-Demand Anodyne MTNR1B 35 40 CCNC(=O)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147055099 FF On-Demand Anodyne ROCK2 33 53 O=C(O)[C@H]1CC=CC[C@H]1C(=O)Nc1ccccc1NS(=O)(=O)c1ccccc1 ZINC000147055107 HG On-Demand Anodyne PRTN3 55 35 O=C(O)[C@H]1CC=CC[C@@H]1C(=O)Nc1ccccc1NS(=O)(=O)c1ccccc1 ZINC000147055276 HG On-Demand Anodyne PRTN3 55 35 C[C@H](CNC(=O)c1ccc(N(C)c2ccccc2)nc1)N1CCCC1 ZINC000147055298 EG On-Demand Anodyne RXRA 40 36 CCOCCCNC(=O)c1cccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147055334 HG On-Demand Anodyne DRD4 46 36 CCOCCCNC(=O)c1cccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147055334 HG On-Demand Anodyne ROCK2 29 42 O=C1c2ccccc2[C@@](O[C@H]2CC[C@@H](O)C2)(c2ccc(Cl)cc2)N1Cc1ccccc1 ZINC000147055343 IK Annotated Anodyne MDM2 45 80 Nc1nc(N)nc(NCCc2ccc3c(c2)OCO3)n1 ZINC000147055455 CC On-Demand Anodyne HSP90AB1 17 40 Nc1nc(N)nc(NCCc2ccc3c(c2)OCO3)n1 ZINC000147055455 CC On-Demand Anodyne DYRK1A 23 44 Nc1nc(N)nc(NCCc2ccc3c(c2)OCO3)n1 ZINC000147055455 CC On-Demand Anodyne CLK1 33 42 Nc1nc(N)nc(NCCc2ccc3c(c2)OCO3)n1 ZINC000147055455 CC On-Demand Anodyne CLK2 35 42 Nc1nc(N)nc(NCCc2ccc3c(c2)OCO3)n1 ZINC000147055455 CC On-Demand Anodyne CLK4 43 44 Nc1nc(N)nc(NCCc2ccc3c(c2)OCO3)n1 ZINC000147055455 CC On-Demand Anodyne DYRK1B 19 42 O=C(O)[C@@H]1CC=CC[C@H]1C(=O)Nc1ccccc1NS(=O)(=O)c1ccccc1 ZINC000147055478 HG On-Demand Anodyne PRTN3 55 35 O=C1c2ccccc2[C@@](O[C@@H]2CC[C@@H](O)C2)(c2ccc(Cl)cc2)N1Cc1ccccc1 ZINC000147055533 IK Annotated Anodyne MDM2 45 80 CCOC(=O)[C@@H](NC(=O)CN)[C@@H](C)CC ZINC000147055620 BC On-Demand Anodyne ENPEP 49 32 CCOC(=O)[C@@H](NC(=O)CN)[C@@H](C)CC ZINC000147055620 BC On-Demand Anodyne LASB 0 44 O=C(O)[C@H]1[C@H]2C=C[C@@H](C2)[C@H]1C(=O)Nc1ccccc1NS(=O)(=O)c1ccccc1 ZINC000147055744 HF On-Demand Anodyne PRTN3 57 36 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccco2)CC1 ZINC000147055868 DD On-Demand Anodyne GHRHR 41 34 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccco2)CC1 ZINC000147055868 DD On-Demand Anodyne P2RY12 179 37 O=C(O)[C@@H]1[C@@H](C(=O)Nc2ccccc2NS(=O)(=O)c2ccccc2)[C@H]2C=C[C@H]1C2 ZINC000147055932 HF On-Demand Anodyne PRTN3 57 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccco2)CC1 ZINC000147056038 DD On-Demand Anodyne GHRHR 41 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccco2)CC1 ZINC000147056038 DD On-Demand Anodyne P2RY12 179 37 O=C(Nc1ccccc1N1CCCCCC1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147056075 FF On-Demand Anodyne KCNQ2 82 47 O=C(Nc1ccccc1N1CCCCCC1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147056238 FF On-Demand Anodyne KCNQ2 82 47 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)Cc3ccc([N+](=O)[O-])cc3)c2)CCO1 ZINC000147056304 HE On-Demand Bother KCNJ1 25 42 O=C(C[C@@H](C(=O)O)c1ccccc1)Nc1cccc(C(=O)N2CCSCC2)c1 ZINC000147056372 GG On-Demand Anodyne NPY2R 24 42 O=C(C[C@@H](C(=O)O)c1ccccc1)Nc1cccc(C(=O)N2CCSCC2)c1 ZINC000147056372 GG On-Demand Anodyne EPHX2 16 44 O=C(C[C@@H](C(=O)O)c1ccccc1)Nc1cccc(C(=O)N2CCSCC2)c1 ZINC000147056372 GG On-Demand Anodyne SLC1A2 42 34 O=C(C[C@@H](C(=O)O)c1ccccc1)Nc1cccc(C(=O)N2CCSCC2)c1 ZINC000147056372 GG On-Demand Anodyne KCNK3 40 34 O=C(Nc1ccccc1N1CCCCCC1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147056407 FF On-Demand Anodyne KCNQ2 88 47 O=C(Nc1ccccc1N1CCCCCC1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147056407 FF On-Demand Anodyne CSF1R 27 46 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(-n2cccn2)c(F)c1 ZINC000147056411 ED On-Demand Anodyne NPY2R 43 34 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(-n2cccn2)c(F)c1 ZINC000147056411 ED On-Demand Anodyne ENV 41 32 C[C@@H](CNC(=O)Cc1cc2ccccc2[nH]c1=O)N1CCCC1 ZINC000147056518 DD On-Demand Anodyne PLD1 33 41 COc1ccc2c(C)c(CCC(=O)N3CCC(C#N)CC3)c(=O)oc2c1 ZINC000147056536 FF On-Demand Mild NQO1 25 41 CC(C)(C)OC(=O)N1CCC(Oc2cc(CO)ccn2)CC1 ZINC000147056576 DE For-Sale Anodyne GPR119 72 46 O=C(Nc1ccccc1N1CCCCCC1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147056594 FF On-Demand Anodyne KCNQ2 82 47 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(-n2cccn2)c(F)c1 ZINC000147056618 ED On-Demand Anodyne NPY2R 43 34 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(-n2cccn2)c(F)c1 ZINC000147056618 ED On-Demand Anodyne ENV 41 32 C[C@H](CNC(=O)Cc1cc2ccccc2[nH]c1=O)N1CCCC1 ZINC000147056721 DD On-Demand Anodyne PLD1 33 41 CNC(=O)c1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1Cl ZINC000147056806 FD On-Demand Anodyne ENV 44 36 COC(=O)c1cc(Cl)ccc1COc1ccc(C)cc1 ZINC000147056962 CI For-Sale Anodyne MAOB 22 42 COC(=O)c1cc(Cl)ccc1COc1ccc(C)cc1 ZINC000147056962 CI For-Sale Anodyne GYS1 52 31 COC(=O)c1cc(Cl)ccc1COc1ccc(C)cc1 ZINC000147056962 CI For-Sale Anodyne FFAR1 24 53 COC(=O)c1cc(Cl)ccc1COc1ccc(C)cc1 ZINC000147056962 CI For-Sale Anodyne FFAR4 44 53 COC(=O)c1cc(Cl)ccc1COc1ccc(C)cc1 ZINC000147056962 CI For-Sale Anodyne MT-CYB 44 36 CNC(=O)c1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1Cl ZINC000147056990 FD On-Demand Anodyne ENV 44 36 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc(OC3CCCC3)nc1)C2 ZINC000147057044 GG On-Demand Anodyne ROCK2 29 41 C[C@@H]1CNC(=O)c2cccc(N)c21 ZINC000147057111 AD For-Sale Anodyne PARP1 29 48 C[C@@H]1CNC(=O)c2cccc(N)c21 ZINC000147057111 AD For-Sale Anodyne PARP4 41 31 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)c3ccc(Cl)s3)c2)CCO1 ZINC000147057113 HG On-Demand Anodyne CCR4 71 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(OC3CCCC3)nc1)C2 ZINC000147057220 GG On-Demand Anodyne ROCK2 29 41 COc1ccc(-c2cnc3ccc(NCc4ccccn4)nn23)cc1OC ZINC000147057288 FG Annotated Anodyne IKBKB 26 40 C[C@H]1CNC(=O)c2cccc(N)c21 ZINC000147057306 AD For-Sale Anodyne PARP1 29 48 C[C@H]1CNC(=O)c2cccc(N)c21 ZINC000147057306 AD For-Sale Anodyne PARP4 41 31 CCC[C@H](NC(N)=O)C(=O)N(C)CCCOc1ccc(F)cc1 ZINC000147057312 ED On-Demand Anodyne FAAH 15 42 C[C@](CC(=O)Nc1cccc(C(=O)N2CCSCC2)c1)(C(=O)O)c1ccccc1 ZINC000147057362 HG On-Demand Anodyne NPY2R 42 41 C[C@](CC(=O)Nc1cccc(C(=O)N2CCSCC2)c1)(C(=O)O)c1ccccc1 ZINC000147057362 HG On-Demand Anodyne EPHX2 21 45 C[C@](CC(=O)Nc1cccc(C(=O)N2CCSCC2)c1)(C(=O)O)c1ccccc1 ZINC000147057362 HG On-Demand Anodyne KCNK3 51 34 C[C@@H](CNC(=O)c1cccc(Cn2ccnc2)c1)N1CCCC1 ZINC000147057365 DE On-Demand Anodyne AGTR2 40 57 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc(Oc3ccc(F)cc3)nc1)C2 ZINC000147057442 HH On-Demand Anodyne ROCK2 35 42 Nc1ccc(OCCCCCCCCCCCOc2ccc(N)cc2)cc1 ZINC000147057468 FK For-Sale Clean LTA4H 15 40 Nc1ccc(OCCCCCCCCCCCOc2ccc(N)cc2)cc1 ZINC000147057468 FK For-Sale Clean PLA2G4B 74 37 Nc1ccc(OCCCCCCCCCCCOc2ccc(N)cc2)cc1 ZINC000147057468 FK For-Sale Clean ACR 55 56 Nc1ccc(OCCCCCCCCCCCOc2ccc(N)cc2)cc1 ZINC000147057468 FK For-Sale Clean SLC47A1 15 56 COc1cc(F)ccc1NC(=O)NCc1ccc(S(=O)(=O)N(C)C(C)C)cc1 ZINC000147057476 HG On-Demand Anodyne GRIN2B 22 41 COc1cc(F)ccc1NC(=O)NCc1ccc(S(=O)(=O)N(C)C(C)C)cc1 ZINC000147057476 HG On-Demand Anodyne BMP1 51 39 COc1cc(F)ccc1NC(=O)NCc1ccc(S(=O)(=O)N(C)C(C)C)cc1 ZINC000147057476 HG On-Demand Anodyne TRPV1 79 37 CCC[C@@H](NC(N)=O)C(=O)N(C)CCCOc1ccc(F)cc1 ZINC000147057500 ED On-Demand Anodyne FAAH 15 42 C[C@H](CNC(=O)c1cccc(Cn2ccnc2)c1)N1CCCC1 ZINC000147057537 DE On-Demand Anodyne CYP19A1 18 40 C[C@H](CNC(=O)c1cccc(Cn2ccnc2)c1)N1CCCC1 ZINC000147057537 DE On-Demand Anodyne CYP11B1 43 45 C[C@H](CNC(=O)c1cccc(Cn2ccnc2)c1)N1CCCC1 ZINC000147057537 DE On-Demand Anodyne TBXAS1 40 46 C[C@H](CNC(=O)c1cccc(Cn2ccnc2)c1)N1CCCC1 ZINC000147057537 DE On-Demand Anodyne AGTR2 40 57 C[C@H](CNC(=O)c1cccc(Cn2ccnc2)c1)N1CCCC1 ZINC000147057537 DE On-Demand Anodyne CYP11B2 47 45 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(Oc3ccc(F)cc3)nc1)C2 ZINC000147057621 HH On-Demand Anodyne ROCK2 35 42 COc1cc(F)ccc1NC(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147057672 FF On-Demand Anodyne MCHR1 18 43 COc1cc(F)ccc1NC(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147057672 FF On-Demand Anodyne ACKR3 46 32 O=C(O)[C@H]1[C@H]2C=C[C@@H](C2)[C@H]1C(=O)Nc1cccc(C(=O)N2CCSCC2)c1 ZINC000147057693 GE On-Demand Anodyne EPHX2 17 46 Cc1nnnn1-c1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147057707 FD On-Demand Anodyne ADORA2B 39 42 Cc1nnnn1-c1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147057707 FD On-Demand Anodyne HIF1A 25 40 CC(=O)c1ccc(S(=O)(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147057712 HF On-Demand Anodyne CHRM3 15 41 Cc1ccc(-n2cc(C(=O)NC[C@@H](C)N3CCCC3)nn2)cc1 ZINC000147057737 DD On-Demand Anodyne ESRRA 19 40 CCc1c[nH]c2cc(F)c(OC)cc12 ZINC000147057855 AF For-Sale Anodyne HTR1D 15 40 CCc1c[nH]c2cc(F)c(OC)cc12 ZINC000147057855 AF For-Sale Anodyne HTR1B 15 40 CCc1c[nH]c2cc(F)c(OC)cc12 ZINC000147057855 AF For-Sale Anodyne MPO 76 37 CC(=O)c1ccc(S(=O)(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147057878 HF On-Demand Anodyne CHRM3 15 41 O=C(O)[C@@H]1[C@@H](C(=O)Nc2cccc(C(=O)N3CCSCC3)c2)[C@H]2C=C[C@H]1C2 ZINC000147057882 GE On-Demand Anodyne EPHX2 17 46 COc1cc(F)ccc1NC(=O)NC[C@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147057906 HG On-Demand Anodyne ADRB2 23 40 COc1cc(F)ccc1NC(=O)NC[C@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147057906 HG On-Demand Anodyne ADRB1 56 37 COc1cc(F)ccc1NC(=O)NC[C@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147057906 HG On-Demand Anodyne P2RY1 23 45 COc1cc(F)ccc1NC(=O)NC[C@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147057906 HG On-Demand Anodyne CCR2 19 40 COc1cc(F)ccc1NC(=O)NC[C@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147057906 HG On-Demand Anodyne PDS 58 43 Cc1ccc(-n2cc(C(=O)NC[C@H](C)N3CCCC3)nn2)cc1 ZINC000147057922 DD On-Demand Anodyne ESRRA 19 40 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild ACE 20 45 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild SSTR2 82 43 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild OPRM1 20 48 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild OPRD1 22 49 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild GHRHR 36 49 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild MME 24 44 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild EDNRB 40 44 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild EDNRA 66 45 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild TACR1 47 44 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild MC4R 61 38 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild TACR2 36 43 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild CCKAR 88 42 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild CTSL 25 42 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild BRS3 41 42 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild CYP51A1 24 40 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild UTS2R 23 41 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild NMBR 31 41 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild MC3R 60 38 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild MC5R 60 35 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild MMP2 22 50 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild MMP8 63 37 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild MMP14 95 39 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild GRPR 42 31 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild ECE1 57 46 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild SSTR3 47 36 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild MMP11 72 36 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild CCKBR 61 44 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild GHSR 79 45 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild CCR2 49 36 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild MMP9 23 50 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild MC1R 73 41 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild CTSC 18 45 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild C5AR1 51 41 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild ST14 57 33 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild NPR 31 44 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild KISS1R 63 35 N#CC1CCN(C(=O)[C@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147057983 ED On-Demand Mild ERAP2 42 37 COc1cc(F)ccc1NC(=O)NC[C@@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147058079 HG On-Demand Anodyne ADRB2 23 40 COc1cc(F)ccc1NC(=O)NC[C@@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147058079 HG On-Demand Anodyne ADRB1 56 37 COc1cc(F)ccc1NC(=O)NC[C@@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147058079 HG On-Demand Anodyne P2RY1 23 45 COc1cc(F)ccc1NC(=O)NC[C@@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147058079 HG On-Demand Anodyne CCR2 19 40 COc1cc(F)ccc1NC(=O)NC[C@@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147058079 HG On-Demand Anodyne PDS 58 43 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild ACE 20 45 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild SSTR2 82 43 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild OPRM1 20 48 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild OPRD1 22 49 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild GHRHR 36 49 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild MME 24 44 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild EDNRB 40 44 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild EDNRA 66 45 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild TACR1 47 44 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild MC4R 61 38 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild TACR2 36 43 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild CCKAR 88 42 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild CTSL 25 42 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild BRS3 41 42 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild CYP51A1 24 40 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild UTS2R 23 41 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild NMBR 31 41 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild MC3R 60 38 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild MC5R 60 35 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild MMP2 22 50 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild MMP8 63 37 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild MMP14 95 39 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild GRPR 42 31 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild ECE1 57 46 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild SSTR3 47 36 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild MMP11 72 36 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild CCKBR 61 44 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild GHSR 79 45 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild CCR2 49 36 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild MMP9 23 50 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild MC1R 73 41 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild CTSC 18 45 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild C5AR1 51 41 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild ST14 57 33 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild NPR 31 44 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild KISS1R 63 35 N#CC1CCN(C(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(N)=O)CC1 ZINC000147058184 ED On-Demand Mild ERAP2 42 37 CC(=O)c1cccc(S(=O)(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)c1 ZINC000147058193 HF On-Demand Anodyne CHRM3 15 43 Cc1nn(C[C@@H](C)N)c2ccccc12 ZINC000147058217 AD For-Sale Anodyne HTR2C 15 46 Cc1nn(-c2ccc(Cl)c(Cl)c2)c(C)c1CC(=O)NC[C@H](C)N1CCCC1 ZINC000147058228 HH On-Demand Anodyne P2RX7 57 54 Cc1nn(-c2ccc(Cl)c(Cl)c2)c(C)c1CC(=O)NC[C@H](C)N1CCCC1 ZINC000147058228 HH On-Demand Anodyne RPA1 72 35 O=C(C[C@]1(C(=O)O)CCSC1)Nc1cccc(C(=O)N2CCSCC2)c1 ZINC000147058253 GE On-Demand Anodyne EPHX2 26 45 O=C(NC1C2CC3CC(C2)CC1C3)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147058368 HG On-Demand Anodyne HSD11B1 58 38 O=C(NC1C2CC3CC(C2)CC1C3)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147058368 HG On-Demand Anodyne EPHX2 55 66 O=C(NC1C2CC3CC(C2)CC1C3)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147058368 HG On-Demand Anodyne TGM2 77 42 O=C(NC1C2CC3CC(C2)CC1C3)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147058368 HG On-Demand Anodyne F13A1 81 37 O=C(NC1C2CC3CC(C2)CC1C3)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147058368 HG On-Demand Anodyne AKR1C3 40 36 O=C(NC1C2CC3CC(C2)CC1C3)C1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147058368 HG On-Demand Anodyne SFRP1 24 40 CC(=O)c1cccc(S(=O)(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)c1 ZINC000147058377 HF On-Demand Anodyne CHRM3 15 43 COc1cc(CC(=O)N2CCC(C#N)CC2)ccc1C ZINC000147058391 CE On-Demand Mild P2RX7 18 43 Cc1nn(C[C@H](C)N)c2ccccc12 ZINC000147058399 AD For-Sale Anodyne HTR2C 15 46 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1CN1C[C@H](C)O[C@H](C)C1)C2 ZINC000147058421 HG On-Demand Anodyne ROCK2 29 43 CNc1nc(Cl)c(Cl)c(N2CCN(CCC3CCC(NC(=O)N4CCOCC4)CC3)CC2)n1 ZINC000147058539 KF Annotated Anodyne DRD3 20 44 CCn1c(CCC(=O)N2CCC(C#N)CC2)nc2cc(S(=O)(=O)N(C)C)ccc21 ZINC000147058581 HE On-Demand Mild CNR2 18 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1CN1C[C@H](C)O[C@@H](C)C1)C2 ZINC000147058619 HG On-Demand Anodyne ROCK2 29 43 O=C(O)c1cc2cc(NC(=O)c3ccc(-c4ccccc4)o3)ccc2o1 ZINC000147058730 EJ For-Sale Anodyne S1PR4 33 51 O=C(O)c1cc2cc(NC(=O)c3ccc(-c4ccccc4)o3)ccc2o1 ZINC000147058730 EJ For-Sale Anodyne SCN10A 23 47 Cc1ccc(CC2CCNCC2)c(F)c1 ZINC000147058805 BF For-Sale Anodyne SLC6A2 20 41 COc1cc(F)ccc1NC(=O)NC[C@@H]1CCCO[C@@H]1c1ccccc1 ZINC000147058817 FI On-Demand Anodyne GRIN2B 26 40 COc1cc(F)ccc1NC(=O)NC[C@@H]1CCCO[C@@H]1c1ccccc1 ZINC000147058817 FI On-Demand Anodyne PYGL 0 40 COc1cc(F)ccc1NC(=O)NC[C@@H]1CCCO[C@@H]1c1ccccc1 ZINC000147058817 FI On-Demand Anodyne ACKR3 64 33 O=C(NCC[C@H](O)CO)[C@@H]1N[C@H](CCCc2ccccc2)[C@]2(C(=O)Nc3cc(Cl)c(F)cc32)[C@H]1c1cccc(Cl)c1 ZINC000147058963 KI Annotated Anodyne MDM2 64 76 COc1cc(F)ccc1NC(=O)NC[C@H]1CCCO[C@@H]1c1ccccc1 ZINC000147059022 FI On-Demand Anodyne GRIN2B 26 40 COc1cc(F)ccc1NC(=O)NC[C@H]1CCCO[C@@H]1c1ccccc1 ZINC000147059022 FI On-Demand Anodyne PYGL 0 40 COc1cc(F)ccc1NC(=O)NC[C@H]1CCCO[C@@H]1c1ccccc1 ZINC000147059022 FI On-Demand Anodyne ACKR3 64 33 CCCC[C@H](NC(N)=O)C(=O)NCC1(c2ccc3c(c2)OCCO3)CCCC1 ZINC000147059145 GF On-Demand Anodyne PCSK5 40 32 CCCC[C@H](NC(N)=O)C(=O)NCC1(c2ccc3c(c2)OCCO3)CCCC1 ZINC000147059145 GF On-Demand Anodyne POLG_WNV 64 30 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild ADRB1 44 35 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild AR 57 47 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild ATF1 52 34 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild GRM4 23 40 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild MTTP 50 37 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild NFKB1 48 34 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild S1PR1 16 47 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild HCN1 45 34 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild HCN4 45 34 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild BLM 0 44 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild KCNK3 78 68 CCOc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147059177 EI On-Demand Mild KCNK9 77 68 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)c3ccc([N+](=O)[O-])cc3)c2)CCO1 ZINC000147059192 HE On-Demand Bother KCNJ1 20 40 COc1cc(F)ccc1NC(=O)NC[C@@H]1CCCO[C@H]1c1ccccc1 ZINC000147059226 FI On-Demand Anodyne GRIN2B 26 40 COc1cc(F)ccc1NC(=O)NC[C@@H]1CCCO[C@H]1c1ccccc1 ZINC000147059226 FI On-Demand Anodyne PYGL 0 40 COc1cc(F)ccc1NC(=O)NC[C@@H]1CCCO[C@H]1c1ccccc1 ZINC000147059226 FI On-Demand Anodyne ACKR3 64 33 CCCC[C@@H](NC(N)=O)C(=O)NCC1(c2ccc3c(c2)OCCO3)CCCC1 ZINC000147059331 GF On-Demand Anodyne PCSK5 40 32 CCCC[C@@H](NC(N)=O)C(=O)NCC1(c2ccc3c(c2)OCCO3)CCCC1 ZINC000147059331 GF On-Demand Anodyne POLG_WNV 64 30 COc1cc(F)ccc1NC(=O)NC[C@H]1CCCO[C@H]1c1ccccc1 ZINC000147059414 FI On-Demand Anodyne GRIN2B 26 40 COc1cc(F)ccc1NC(=O)NC[C@H]1CCCO[C@H]1c1ccccc1 ZINC000147059414 FI On-Demand Anodyne PYGL 0 40 COc1cc(F)ccc1NC(=O)NC[C@H]1CCCO[C@H]1c1ccccc1 ZINC000147059414 FI On-Demand Anodyne ACKR3 64 33 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)c3ccc4ccccc4c3)c2)CCO1 ZINC000147059435 HH On-Demand Anodyne F2 20 41 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)c3ccc4ccccc4c3)c2)CCO1 ZINC000147059435 HH On-Demand Anodyne GNRHR 15 41 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)c3ccc4ccccc4c3)c2)CCO1 ZINC000147059435 HH On-Demand Anodyne HTR7 18 49 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)c3ccc4ccccc4c3)c2)CCO1 ZINC000147059435 HH On-Demand Anodyne TRY2_BOVIN 76 41 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)c3ccc4ccccc4c3)c2)CCO1 ZINC000147059435 HH On-Demand Anodyne BDKRB1 16 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCCCC2)c1 ZINC000147059447 FD On-Demand Anodyne NPY2R 16 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCCCC2)c1 ZINC000147059447 FD On-Demand Anodyne EPHX2 15 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCCCC2)c1 ZINC000147059447 FD On-Demand Anodyne L3MBTL3 53 40 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(Cl)c2)c1 ZINC000147059515 FG On-Demand Bother DRD4 46 37 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(Cl)c2)c1 ZINC000147059515 FG On-Demand Bother CASR 18 43 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(Cl)c2)c1 ZINC000147059515 FG On-Demand Bother TAAR1 25 46 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(Cl)c2)c1 ZINC000147059515 FG On-Demand Bother AKR1C2 27 40 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(F)cc1 ZINC000147059551 DF On-Demand Anodyne NOD1 45 31 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)Nc3ncccn3)cc2)cc([N+](=O)[O-])c1 ZINC000147059580 HF On-Demand Bother GRM4 33 53 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)Nc3ncccn3)cc2)cc([N+](=O)[O-])c1 ZINC000147059580 HF On-Demand Bother KCNK3 43 35 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCCCC2)c1 ZINC000147059625 FD On-Demand Anodyne NPY2R 16 43 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCCCC2)c1 ZINC000147059625 FD On-Demand Anodyne EPHX2 15 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCCCC2)c1 ZINC000147059625 FD On-Demand Anodyne L3MBTL3 53 40 C=CC(=O)Nc1cc(Nc2nccc(-c3c[nH]c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C ZINC000147059673 JI In-Stock Anodyne INSR 29 57 C=CC(=O)Nc1cc(Nc2nccc(-c3c[nH]c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C ZINC000147059673 JI In-Stock Anodyne IGF1R 54 35 C=CC(=O)Nc1cc(Nc2nccc(-c3c[nH]c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C ZINC000147059673 JI In-Stock Anodyne RET 15 42 C=CC(=O)Nc1cc(Nc2nccc(-c3c[nH]c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C ZINC000147059673 JI In-Stock Anodyne MAPK7 41 37 C=CC(=O)Nc1cc(Nc2nccc(-c3c[nH]c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C ZINC000147059673 JI In-Stock Anodyne DYRK1B 28 46 COC(=O)CCOc1ccc(NC(=O)C[C@@](C)(C(=O)O)c2ccccc2)cc1 ZINC000147059718 GF On-Demand Anodyne LTA4H 61 42 COC(=O)CCOc1ccc(NC(=O)C[C@@](C)(C(=O)O)c2ccccc2)cc1 ZINC000147059718 GF On-Demand Anodyne FAAH 18 40 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@@H](C)c1ccc(F)cc1 ZINC000147059733 DF On-Demand Anodyne NOD1 45 31 O=C(Nc1ccc(-n2cccn2)cc1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147059785 ED On-Demand Anodyne AMP1_PLAFQ 49 33 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(F)cc1 ZINC000147059914 DF On-Demand Anodyne NOD1 45 31 COC(=O)CCOc1ccc(NC(=O)C[C@H](C(=O)O)c2ccccc2)cc1 ZINC000147059922 FF On-Demand Anodyne LTA4H 62 47 COC(=O)CCOc1ccc(NC(=O)C[C@H](C(=O)O)c2ccccc2)cc1 ZINC000147059922 FF On-Demand Anodyne FAAH 19 40 COC(=O)CCOc1ccc(NC(=O)C[C@H](C(=O)O)c2ccccc2)cc1 ZINC000147059922 FF On-Demand Anodyne SLC1A1 34 40 COC(=O)CCOc1ccc(NC(=O)C[C@H](C(=O)O)c2ccccc2)cc1 ZINC000147059922 FF On-Demand Anodyne SLC1A2 54 40 N#Cc1ccc(NC(=S)Nc2ccc([N+](=O)[O-])cc2)cc1 ZINC000147059946 CG For-Sale Mild UREA_CANEN 25 42 O=C(Nc1ccc(-n2cccn2)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147059983 ED On-Demand Anodyne AMP1_PLAFQ 49 33 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@H](C)c1ccc(F)cc1 ZINC000147060077 DF On-Demand Anodyne NOD1 45 31 O=C(Nc1ccc(-n2cccn2)cc1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147060179 ED On-Demand Anodyne AMP1_PLAFQ 49 33 COc1ccc(-n2nc(C(N)=O)c3c2C(=O)N(c2ccc(C(C)(C)N(C)C)cc2)CC3)cc1 ZINC000147060221 IF Annotated Anodyne IKBKB 15 40 C=CCNC(=O)CN1CCN(C(=O)[C@H](CCCC)NC(N)=O)CC1 ZINC000147060325 EB On-Demand Mild P2RY12 134 37 C=CCNC(=O)CN1CCN(C(=O)[C@H](CCCC)NC(N)=O)CC1 ZINC000147060325 EB On-Demand Mild NOD1 60 33 O=C(Nc1ccc(-n2cccn2)cc1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147060360 ED On-Demand Anodyne AMP1_PLAFQ 49 33 CCCCCC1CCC(c2ccc(C(=O)Oc3ccc(OC)cc3)cc2)CC1 ZINC000147060429 GK For-Sale Anodyne ACR 60 43 C=CCNC(=O)CN1CCN(C(=O)[C@@H](CCCC)NC(N)=O)CC1 ZINC000147060516 EB On-Demand Mild P2RY12 134 37 C=CCNC(=O)CN1CCN(C(=O)[C@@H](CCCC)NC(N)=O)CC1 ZINC000147060516 EB On-Demand Mild NOD1 60 33 CCN(c1cc(-c2ccc(CN3CC[C@@H](F)C3)cc2)cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C)C1CCOCC1 ZINC000147060533 KK Annotated Anodyne EZH2 56 87 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc(OCC(=O)NC2CC2)cc1 ZINC000147060538 HH On-Demand Anodyne MDM2 51 35 O=C(Nc1ccc(C(=O)N2CCCC2)cc1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147060558 FD On-Demand Anodyne L3MBTL3 76 40 O=C(Nc1ccc(C(=O)N2CCCC2)cc1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147060745 FD On-Demand Anodyne L3MBTL3 76 40 CS(=O)(=O)NC[C@@H]1CCCN(C(=O)COc2ccc(C(N)=O)cc2)C1 ZINC000147060785 FB On-Demand Anodyne COLA 38 43 CS(=O)(=O)NC[C@@H]1CCCN(C(=O)COc2ccc(C(N)=O)cc2)C1 ZINC000147060785 FB On-Demand Anodyne TMPRSS11D 45 32 N#Cc1cn(-c2ccc(C(=O)O)cc2)nc1OCc1ccccc1 ZINC000147060824 DG Annotated Anodyne SRD5A2 15 46 N#Cc1cn(-c2ccc(C(=O)O)cc2)nc1OCc1ccccc1 ZINC000147060824 DG Annotated Anodyne XDH 18 40 CC(C)C[C@@H](Br)CC(=O)O ZINC000147060902 BE For-Sale Reactive RNPEP 23 41 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc(OCC(=O)NC2CC2)cc1 ZINC000147060920 HH On-Demand Anodyne MDM2 51 35 O=C(Nc1ccc(C(=O)N2CCCC2)cc1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147060938 FD On-Demand Anodyne L3MBTL3 76 40 CS(=O)(=O)NC[C@H]1CCCN(C(=O)COc2ccc(C(N)=O)cc2)C1 ZINC000147060981 FB On-Demand Anodyne TMPRSS11D 45 32 COc1ccc([N+](=O)[O-])c(C(=O)NC2CCN(c3ncccn3)CC2)c1 ZINC000147061071 FD On-Demand Bother AKR1C2 22 40 CC(C)C[C@H](Br)CC(=O)O ZINC000147061076 BE For-Sale Reactive RNPEP 23 41 O=C(Nc1ccc(C(=O)N2CCCC2)cc1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147061129 FD On-Demand Anodyne L3MBTL3 76 40 Cc1ccc(C(=O)N2CCC(C#N)CC2)n1C ZINC000147061139 BD On-Demand Mild L3MBTL3 50 33 C[C@@H](O)CCCOc1ccc([N+](=O)[O-])cc1 ZINC000147061288 BE On-Demand Bother ACR 41 55 C[C@@H]1O[C@@H](CO)[C@H](O)[C@@H]1O ZINC000147061298 AA For-Sale Anodyne CDA 57 34 C[C@@H]1O[C@@H](CO)[C@H](O)[C@@H]1O ZINC000147061298 AA For-Sale Anodyne FIMH 27 40 C[C@@H]1O[C@@H](CO)[C@H](O)[C@@H]1O ZINC000147061298 AA For-Sale Anodyne MGEA5 25 40 C[C@@H](NC(=O)c1ccc2c(c1)COC2)c1ccc(OCC(=O)NC2CC2)cc1 ZINC000147061338 GF On-Demand Anodyne ACACA 45 36 C[C@H](O)CCCOc1ccc([N+](=O)[O-])cc1 ZINC000147061488 BE On-Demand Bother ACR 41 55 CCN(c1cc(-c2ccc(CNC)cc2)cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C)C1CCOCC1 ZINC000147061514 KJ Annotated Anodyne EZH2 55 82 CCN(c1cc(-c2ccc(CNCC3CC3)cc2)cc(C(=O)NCc2c(C)cc(C)[nH]c2=O)c1C)C1CCOCC1 ZINC000147061734 KK Annotated Anodyne EZH2 53 79 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA2 195 71 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA6 39 58 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA1 165 58 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA7 106 61 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA13 61 58 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA5B 70 49 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA4 133 61 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA5A 73 49 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA14 76 49 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA12 125 61 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA9 141 61 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CAH_METTE 57 58 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CYNT 57 55 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne NCE103 53 71 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne CA15 36 48 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne MTCA1 57 45 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne P96878_MYCTU 71 51 CC(=O)CCc1ccc(S(N)(=O)=O)cc1 ZINC000147061885 BC For-Sale Anodyne A6YCJ1_9METZ 41 58 CCN(CC)Cc1ccc(-c2cc(C(=O)NCc3c(C)cc(C)[nH]c3=O)c(C)c(N(CC)C3CCOCC3)c2)cc1 ZINC000147061935 KK Annotated Anodyne EZH2 54 80 O=C(NCC(F)(F)F)Nc1cccc(-c2cnc3cc(-c4ccc(=O)[nH]n4)ccn23)c1 ZINC000147061992 IG Annotated Anodyne RIPK1 44 30 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne ALOX5 18 43 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne THRA 48 41 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne PPARG 19 40 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne PPARA 34 42 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne RARB 27 42 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne THRB 38 41 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne RXRA 35 44 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne GRM3 26 40 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne LTB4R 23 40 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne PLA2G4A 23 40 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne PPARD 41 43 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne GRM2 28 42 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne PLA2G4B 89 42 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne LIPG 21 42 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne PTGES 38 41 CCCCOc1ccc(C(C)(C)C)cc1C(=O)O ZINC000147062012 CH In-Stock Anodyne AKR1C2 35 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccccc2CN2CCC[C@@H](C)C2)c1 ZINC000147062146 GH On-Demand Bother EBP 23 43 CCCN(CCC)CCc1cccc([N+](=O)[O-])c1Cl ZINC000147062277 CH For-Sale Anodyne COLA 68 34 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccccc2CN2CCC[C@H](C)C2)c1 ZINC000147062366 GH On-Demand Bother EBP 23 43 CC(C)(C)c1ccccc1NC(=O)Nc1cccc(C#N)c1 ZINC000147062383 CI For-Sale Mild MAPK14 30 42 CC(C)(C)c1ccccc1NC(=O)Nc1cccc(C#N)c1 ZINC000147062383 CI For-Sale Mild P2RY1 35 45 CC(C)(C)c1ccccc1NC(=O)Nc1cccc(C#N)c1 ZINC000147062383 CI For-Sale Mild CCR3 22 49 CC(C)(C)c1ccccc1NC(=O)Nc1cccc(C#N)c1 ZINC000147062383 CI For-Sale Mild MCHR1 15 43 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062392 HH On-Demand Anodyne DRD4 20 41 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062392 HH On-Demand Anodyne HRH2 18 41 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062392 HH On-Demand Anodyne SIGMAR1 25 49 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062392 HH On-Demand Anodyne FAAH 15 45 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062392 HH On-Demand Anodyne CXCR3 17 40 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062392 HH On-Demand Anodyne MCHR1 41 45 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062589 HH On-Demand Anodyne DRD4 20 41 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062589 HH On-Demand Anodyne HRH2 18 41 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062589 HH On-Demand Anodyne SIGMAR1 25 49 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062589 HH On-Demand Anodyne FAAH 15 45 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062589 HH On-Demand Anodyne CXCR3 17 40 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062589 HH On-Demand Anodyne MCHR1 41 45 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062791 HH On-Demand Anodyne DRD4 20 41 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062791 HH On-Demand Anodyne HRH2 18 41 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062791 HH On-Demand Anodyne SIGMAR1 25 49 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062791 HH On-Demand Anodyne FAAH 15 45 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062791 HH On-Demand Anodyne CXCR3 17 40 NC(=O)C1CCN(Cc2cccc(NC(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)c2)CC1 ZINC000147062791 HH On-Demand Anodyne MCHR1 41 45 CC(C)N(C)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1F ZINC000147062949 FE On-Demand Anodyne ENV 42 34 COCc1nc(C(=O)N2CCN(c3ccccc3)CC2)cs1 ZINC000147062983 DE On-Demand Anodyne CCKAR 42 40 COCCOc1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147063003 FH On-Demand Anodyne PDS 72 42 CC(C)N(C)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1F ZINC000147063139 FE On-Demand Anodyne ENV 42 34 COCCOc1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147063190 FH On-Demand Anodyne PDS 72 42 COCc1nc(C(=O)Nc2nc(-c3ccccc3)cs2)cs1 ZINC000147063226 EH On-Demand Anodyne MPL 47 38 COCc1nc(C(=O)Nc2nc(-c3ccccc3)cs2)cs1 ZINC000147063226 EH On-Demand Anodyne ROCK1 24 49 COCc1nc(C(=O)Nc2nc(-c3ccccc3)cs2)cs1 ZINC000147063226 EH On-Demand Anodyne ROCK2 18 49 COCc1nc(C(=O)Nc2nc(-c3ccccc3)cs2)cs1 ZINC000147063226 EH On-Demand Anodyne HDAC9 15 47 COCc1nc(C(=O)Nc2nc(-c3ccccc3)cs2)cs1 ZINC000147063226 EH On-Demand Anodyne TRPA1 19 42 COCc1nc(C(=O)Nc2nc(-c3ccccc3)cs2)cs1 ZINC000147063226 EH On-Demand Anodyne VCP 19 43 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(OCCC(C)C)c(OC)c2)c1 ZINC000147063352 HH On-Demand Bother MT-ND1 24 42 C[C@@H]1CN(Cc2cccc(CNS(=O)(=O)c3ccc(C(N)=O)cc3)c2)CCO1 ZINC000147063374 HD On-Demand Anodyne TRY2_BOVIN 45 35 O=C(NC1CCC(O)CC1)[C@@H]1N[C@H](C=C2CCCC2)[C@]2(C(=O)Nc3cc(Cl)ccc32)[C@H]1c1cccc(Cl)c1F ZINC000147063382 KK Annotated Anodyne MDM2 80 64 COCCOc1cccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147063398 FH On-Demand Anodyne PDS 72 42 N#CC1CCN(C(=O)CCn2cnc3sc4c(c3c2=O)CCCC4)CC1 ZINC000147063537 FE On-Demand Mild HTR1B 19 43 C[C@H]1CN(Cc2cccc(CNS(=O)(=O)c3ccc(C(N)=O)cc3)c2)CCO1 ZINC000147063562 HD On-Demand Anodyne TRY2_BOVIN 45 35 CC(C)Oc1cccc([C@@H](C)NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147063568 HG On-Demand Bother GCK 16 41 COCCOc1cccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147063575 FH On-Demand Anodyne PDS 72 42 CCCC[C@H](NC(N)=O)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147063694 CE On-Demand Anodyne ACE 24 46 CCCC[C@H](NC(N)=O)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147063694 CE On-Demand Anodyne CTSK 30 46 CCCC[C@H](NC(N)=O)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147063694 CE On-Demand Anodyne GZMB 49 30 CCCC[C@H](NC(N)=O)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147063694 CE On-Demand Anodyne BIRC2 45 35 COCCOc1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147063754 HH On-Demand Anodyne ROCK2 21 42 COCCOc1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147063754 HH On-Demand Anodyne PDS 53 42 CC(C)Oc1cccc([C@H](C)NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147063757 HG On-Demand Bother GCK 16 41 COCCOc1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147063941 HH On-Demand Anodyne ROCK2 21 42 COCCOc1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147063941 HH On-Demand Anodyne PDS 53 42 COc1ccc(OC)c([C@@H]2CCCN2C(=O)Cc2cccc(OC(C)C)c2)c1 ZINC000147064005 GI On-Demand Anodyne FKBP1A 68 40 COc1ccc(OC)c([C@@H]2CCCN2C(=O)Cc2cccc(OC(C)C)c2)c1 ZINC000147064005 GI On-Demand Anodyne OPRK1 19 43 COc1ccc(OC)c([C@@H]2CCCN2C(=O)Cc2cccc(OC(C)C)c2)c1 ZINC000147064005 GI On-Demand Anodyne AGTR2 61 34 COc1ccc(OC)c([C@@H]2CCCN2C(=O)Cc2cccc(OC(C)C)c2)c1 ZINC000147064005 GI On-Demand Anodyne COLA 66 37 COc1ccc(OC)c([C@@H]2CCCN2C(=O)Cc2cccc(OC(C)C)c2)c1 ZINC000147064005 GI On-Demand Anodyne CPT1A 61 37 COc1ccc(OC)c([C@@H]2CCCN2C(=O)Cc2cccc(OC(C)C)c2)c1 ZINC000147064005 GI On-Demand Anodyne MTNR1B 43 38 COCCOc1cccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147064134 HH On-Demand Anodyne ROCK2 21 42 COCCOc1cccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147064134 HH On-Demand Anodyne PDS 53 42 COC(=O)/C(=C\O)c1ccccc1OCc1ccccc1 ZINC000147064235 CG For-Sale Clean PPIA 49 44 COC(=O)/C(=C\O)c1ccccc1OCc1ccccc1 ZINC000147064235 CG For-Sale Clean POBA 0 43 COC(=O)/C(=C\O)c1ccccc1OCc1ccccc1 ZINC000147064235 CG For-Sale Clean TRPM8 0 42 COC(=O)/C(=C\O)c1ccccc1OCc1ccccc1 ZINC000147064235 CG For-Sale Clean HCN1 23 44 COC(=O)/C(=C\O)c1ccccc1OCc1ccccc1 ZINC000147064235 CG For-Sale Clean KCNK3 42 38 COC(=O)/C(=C\O)c1ccccc1OCc1ccccc1 ZINC000147064235 CG For-Sale Clean MT-CYB 69 48 CC(=O)N1CCc2cc(C(=O)N3CCC(C#N)CC3)ccc21 ZINC000147064343 CD On-Demand Mild L3MBTL3 57 39 CON(C)C(=O)c1ccccc1CCc1ccccc1 ZINC000147064402 CG On-Demand Anodyne CAPN1 17 46 CON(C)C(=O)c1ccccc1CCc1ccccc1 ZINC000147064402 CG On-Demand Anodyne NPR 46 33 CC(C)(C)OC(=O)NCCN1CCN(CCO)CC1 ZINC000147064405 CC On-Demand Anodyne DRD4 41 32 CCC[C@H](NC(N)=O)C(=O)NCc1cc(-c2ccccc2)no1 ZINC000147064453 DD On-Demand Anodyne PCSK5 41 32 CCC[C@H](NC(N)=O)C(=O)NCc1cc(-c2ccccc2)no1 ZINC000147064453 DD On-Demand Anodyne FURIN 50 34 CCC[C@H](NC(N)=O)C(=O)NCc1cc(-c2ccccc2)no1 ZINC000147064453 DD On-Demand Anodyne POLG_WNV 49 30 O=C(O)C[C@H](Oc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147064480 CF For-Sale Anodyne PTPN1 15 47 CN1CCCN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)CC1 ZINC000147064525 FD On-Demand Anodyne LCK 16 41 CN1CCCN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)CC1 ZINC000147064525 FD On-Demand Anodyne PRNP 38 43 CN1CCCN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)CC1 ZINC000147064525 FD On-Demand Anodyne MTOR 29 43 CN1CCCN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)CC1 ZINC000147064525 FD On-Demand Anodyne HCK 24 41 CN1CCCN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)CC1 ZINC000147064525 FD On-Demand Anodyne TNK2 27 47 CCCCCCCCNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000147064549 CI For-Sale Mild RARB 20 40 CCCCCCCCNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000147064549 CI For-Sale Mild DRTS_TOXGO 15 42 CCCCCCCCNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000147064549 CI For-Sale Mild PLA2G4B 54 52 CCCCCCCCNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000147064549 CI For-Sale Mild TAAR1 20 52 CCCCCCCCNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000147064549 CI For-Sale Mild AKR1C3 16 45 CCCCCCCCNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000147064549 CI For-Sale Mild KAT2B 0 50 CCCCCCCCNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000147064549 CI For-Sale Mild ASAH1 64 32 CCCCCCCCNc1ccc(C(=O)O)cc1[N+](=O)[O-] ZINC000147064549 CI For-Sale Mild AKR1C4 0 40 COCc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147064634 EF On-Demand Bother CACNA1D 52 38 COCc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147064634 EF On-Demand Bother ROCK1 21 40 COCc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147064634 EF On-Demand Bother MMP1 15 41 COCc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147064634 EF On-Demand Bother AKR1C2 26 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064744 DD On-Demand Anodyne MMP3 17 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064744 DD On-Demand Anodyne PCSK5 41 33 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064744 DD On-Demand Anodyne FURIN 59 44 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064744 DD On-Demand Anodyne POLG_DEN26 0 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064744 DD On-Demand Anodyne POLG_WNV 64 32 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064744 DD On-Demand Anodyne Q9JN24_ECOLX 0 46 C[C@H]1CN(c2ccc(C(=O)NC[C@@H](C)N3CCCC3)cn2)C[C@@H](C)O1 ZINC000147064813 ED On-Demand Anodyne HDAC1 17 40 C[C@H]1CN(c2ccc(C(=O)NC[C@@H](C)N3CCCC3)cn2)C[C@@H](C)O1 ZINC000147064813 ED On-Demand Anodyne HPGDS 15 40 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)Cc2ccc(Br)cc2)c1 ZINC000147064844 GH On-Demand Bother COLA 40 37 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)Cc2ccc(Br)cc2)c1 ZINC000147064844 GH On-Demand Bother AKR1C2 30 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064936 DD On-Demand Anodyne MMP3 17 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064936 DD On-Demand Anodyne PCSK5 41 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064936 DD On-Demand Anodyne FURIN 59 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064936 DD On-Demand Anodyne POLG_DEN26 0 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064936 DD On-Demand Anodyne POLG_WNV 64 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(C(=O)N(C)C)cc1 ZINC000147064936 DD On-Demand Anodyne Q9JN24_ECOLX 0 46 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cc(Br)ccc1C)C2 ZINC000147065008 GH On-Demand Anodyne ROCK2 37 51 N#CC1CCN(C(=O)c2ccc(Oc3ccc(C(F)(F)F)cn3)cc2)CC1 ZINC000147065020 GI On-Demand Mild HRH3 15 48 N#CC1CCN(C(=O)c2ccc(Oc3ccc(C(F)(F)F)cn3)cc2)CC1 ZINC000147065020 GI On-Demand Mild LIPE 32 62 N#CC1CCN(C(=O)c2ccc(Oc3ccc(C(F)(F)F)cn3)cc2)CC1 ZINC000147065020 GI On-Demand Mild SLC6A7 0 40 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)Cc2ccc(Br)cc2)c1 ZINC000147065039 GH On-Demand Bother COLA 40 37 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)Cc2ccc(Br)cc2)c1 ZINC000147065039 GH On-Demand Bother AKR1C2 30 40 C[C@@H]1CN(c2ccc(C(=O)NC[C@@H](C)N3CCCC3)cn2)C[C@@H](C)O1 ZINC000147065195 ED On-Demand Anodyne HPGDS 15 40 COc1ccc(C#N)cc1N[C@H](C(=O)NCc1ccc2c(c1)OCO2)c1ccccc1 ZINC000147065237 HH On-Demand Mild EDNRA 39 41 COc1ccc(C#N)cc1N[C@H](C(=O)NCc1ccc2c(c1)OCO2)c1ccccc1 ZINC000147065237 HH On-Demand Mild BMP1 61 38 COc1ccc(C#N)cc1N[C@H](C(=O)NCc1ccc2c(c1)OCO2)c1ccccc1 ZINC000147065237 HH On-Demand Mild NOS2 62 32 Nc1cc(-c2ccncc2NC(=O)c2nc(-c3c(F)cccc3F)ccc2N)ccn1 ZINC000147065413 HH Annotated Anodyne PIM1 37 46 Nc1cc(-c2ccncc2NC(=O)c2nc(-c3c(F)cccc3F)ccc2N)ccn1 ZINC000147065413 HH Annotated Anodyne PIM2 17 46 Nc1cc(-c2ccncc2NC(=O)c2nc(-c3c(F)cccc3F)ccc2N)ccn1 ZINC000147065413 HH Annotated Anodyne PIM3 25 46 C[C@@H](CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2OC(F)F)C1)N1CCCC1 ZINC000147065419 HF On-Demand Anodyne SLC6A1 46 34 C[C@@H](CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2OC(F)F)C1)N1CCCC1 ZINC000147065419 HF On-Demand Anodyne HCN1 48 36 C[C@@H](CNC(=O)[C@@H]1CCCN(C(=O)c2ccccc2OC(F)F)C1)N1CCCC1 ZINC000147065419 HF On-Demand Anodyne HCN4 42 35 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H](C)c1cc(F)ccc1OC)C2 ZINC000147065425 FG On-Demand Anodyne ROCK2 25 43 CCCCNC(=O)N1CC(NC(=O)[C@@H]2N[C@H](CC(C)(C)C)[C@]3(C(=O)Nc4cc(Cl)ccc43)[C@H]2c2cccc(Cl)c2F)C1 ZINC000147065429 KK Annotated Anodyne MDM2 99 68 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cc(N3CCCC3=O)ccc2Cl)C1 ZINC000147065446 HE On-Demand Anodyne AKR1C3 25 45 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cc(N3CCCC3=O)ccc2Cl)C1 ZINC000147065622 HE On-Demand Anodyne AKR1C3 25 45 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H](C)c1cc(F)ccc1OC)C2 ZINC000147065628 FG On-Demand Anodyne ROCK2 25 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(N3CCNC3=O)c2)c1 ZINC000147065638 FE On-Demand Bother TAAR1 35 49 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(N3CCNC3=O)c2)c1 ZINC000147065638 FE On-Demand Bother AKR1C3 16 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(N3CCNC3=O)c2)c1 ZINC000147065638 FE On-Demand Bother AKR1C2 33 41 C[C@@H](CNC(=O)[C@H]1CCCN(C(=O)c2ccccc2OC(F)F)C1)N1CCCC1 ZINC000147065649 HF On-Demand Anodyne SLC6A1 46 34 C[C@@H](CNC(=O)[C@H]1CCCN(C(=O)c2ccccc2OC(F)F)C1)N1CCCC1 ZINC000147065649 HF On-Demand Anodyne HCN1 48 36 C[C@@H](CNC(=O)[C@H]1CCCN(C(=O)c2ccccc2OC(F)F)C1)N1CCCC1 ZINC000147065649 HF On-Demand Anodyne HCN4 42 35 CC[C@@H](Nc1cc(C#N)ccc1OC)C(=O)NCc1ccccc1 ZINC000147065662 DG On-Demand Mild PAPA1_CARPA 46 39 CC[C@@H](Nc1cc(C#N)ccc1OC)C(=O)NCc1ccccc1 ZINC000147065662 DG On-Demand Mild CTSL 33 41 CC[C@@H](Nc1cc(C#N)ccc1OC)C(=O)NCc1ccccc1 ZINC000147065662 DG On-Demand Mild CTSS 37 41 CC[C@@H](Nc1cc(C#N)ccc1OC)C(=O)NCc1ccccc1 ZINC000147065662 DG On-Demand Mild CAPN2 45 36 CC[C@@H](Nc1cc(C#N)ccc1OC)C(=O)NCc1ccccc1 ZINC000147065662 DG On-Demand Mild CTRB_BOVIN 47 34 CC[C@@H](Nc1cc(C#N)ccc1OC)C(=O)NCc1ccccc1 ZINC000147065662 DG On-Demand Mild PDS 45 38 CCc1ncc(C(=O)Nc2cccc(Br)c2)s1 ZINC000147065665 DH On-Demand Anodyne EGFR 62 45 CCc1ncc(C(=O)Nc2cccc(Br)c2)s1 ZINC000147065665 DH On-Demand Anodyne TEK 19 41 CCc1ncc(C(=O)Nc2cccc(Br)c2)s1 ZINC000147065665 DH On-Demand Anodyne KCNK3 91 36 CCc1ncc(C(=O)Nc2cccc(Br)c2)s1 ZINC000147065665 DH On-Demand Anodyne KCNK9 56 35 C[C@H](CNC(=O)[C@H]1CCCN(C(=O)c2ccccc2OC(F)F)C1)N1CCCC1 ZINC000147065837 HF On-Demand Anodyne SLC6A1 46 34 C[C@H](CNC(=O)[C@H]1CCCN(C(=O)c2ccccc2OC(F)F)C1)N1CCCC1 ZINC000147065837 HF On-Demand Anodyne HCN1 48 36 C[C@H](CNC(=O)[C@H]1CCCN(C(=O)c2ccccc2OC(F)F)C1)N1CCCC1 ZINC000147065837 HF On-Demand Anodyne HCN4 42 35 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H](C)c1cc(F)ccc1OC)C2 ZINC000147065847 FG On-Demand Anodyne ROCK2 25 43 C#CC[C@H](NC(=O)OC(C)(C)C)C(=O)N(C)OC ZINC000147065854 CC In-Stock Mild PAPA1_CARPA 52 44 C#CC[C@H](NC(=O)OC(C)(C)C)C(=O)N(C)OC ZINC000147065854 CC In-Stock Mild CTSK 23 40 COc1ccc(C(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)c2ccccc12 ZINC000147065859 HG On-Demand Mild L3MBTL3 28 46 O=[P@](O)(CCOCc1ccccc1)Oc1ccccc1 ZINC000147066032 CG For-Sale Anodyne IMPA1 20 40 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne F2 28 53 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne CA2 23 47 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne ACE 17 44 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne MME 32 44 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne CA1 15 44 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne MMP13 37 66 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne TRY2_BOVIN 73 53 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne CA4 21 44 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne MMP2 39 66 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne MMP3 18 49 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne MMP8 18 48 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne MMP14 17 48 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne CAPN1 15 44 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne MMP9 24 48 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne ACE2 51 44 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne MMP12 36 48 CC[C@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066035 FD On-Demand Anodyne ADAMTS4 23 45 C#CC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(C)OC ZINC000147066043 CC In-Stock Mild PAPA1_CARPA 52 44 C#CC[C@@H](NC(=O)OC(C)(C)C)C(=O)N(C)OC ZINC000147066043 CC In-Stock Mild CTSK 0 40 N#CC1CCN(C(=O)C2CCN(C(=O)c3cccc4ccccc34)CC2)CC1 ZINC000147066062 GG On-Demand Mild CHRM2 20 42 N#CC1CCN(C(=O)C2CCN(C(=O)c3cccc4ccccc34)CC2)CC1 ZINC000147066062 GG On-Demand Mild DPP4 15 43 N#CC1CCN(C(=O)C2CCN(C(=O)c3cccc4ccccc34)CC2)CC1 ZINC000147066062 GG On-Demand Mild PREP 44 42 N#CC1CCN(C(=O)C2CCN(C(=O)c3cccc4ccccc34)CC2)CC1 ZINC000147066062 GG On-Demand Mild L3MBTL3 45 45 Cc1cc(C(=O)Nc2ccccc2C)cc([N+](=O)[O-])c1 ZINC000147066083 CG On-Demand Bother PYGL 25 42 Cc1cc(C(=O)Nc2ccccc2C)cc([N+](=O)[O-])c1 ZINC000147066083 CG On-Demand Bother KCNMA1 25 40 Cc1cc(C(=O)Nc2ccccc2C)cc([N+](=O)[O-])c1 ZINC000147066083 CG On-Demand Bother KCNK9 42 38 COc1ccc(C#N)cc1N[C@H](C)C(=O)N1CCN(c2ccccc2)CC1 ZINC000147066095 FF On-Demand Mild SLC6A9 18 42 C=CC(C)(C)c1cc(O)c(O)c(CC=C(C)C)c1-c1oc2c(CC=C(C)C)c(O)cc(O)c2c(=O)c1O ZINC000147066138 KK Annotated Mild ABCB1A 20 42 C=CC(C)(C)c1cc(O)c(O)c(CC=C(C)C)c1-c1oc2c(CC=C(C)C)c(O)cc(O)c2c(=O)c1O ZINC000147066138 KK Annotated Mild NANH 26 42 CCCCOc1ccc(NC(=O)O[C@@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066141 FK For-Sale Anodyne HRH2 32 40 CCCCOc1ccc(NC(=O)O[C@@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066141 FK For-Sale Anodyne HRH3 53 44 CCCCOc1ccc(NC(=O)O[C@@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066141 FK For-Sale Anodyne PLA2G4B 74 34 CCCCOc1ccc(NC(=O)O[C@@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066141 FK For-Sale Anodyne FAAH 26 46 CCCCOc1ccc(NC(=O)O[C@@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066141 FK For-Sale Anodyne EPHX2 24 44 CCCCOc1ccc(NC(=O)O[C@@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066141 FK For-Sale Anodyne PSMB2 44 33 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne F2 23 53 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne CA2 30 47 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne ACE 21 44 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne MME 26 44 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne MMP13 32 46 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne NPY1R 22 42 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne TRY2_BOVIN 67 53 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne CA4 21 44 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne MMP2 38 45 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne MMP3 20 49 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne MMP8 15 44 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne MMP14 19 44 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne MMP9 27 44 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne ACE2 55 44 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne MMP12 34 46 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne ITGAV 44 33 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne ADAMTS4 40 45 CC[C@@H](NC(=O)CNS(=O)(=O)c1ccc2ccccc2c1)C(=O)O ZINC000147066224 FD On-Demand Anodyne AKR1C3 15 41 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066332 FK For-Sale Anodyne HRH2 32 40 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066332 FK For-Sale Anodyne HRH3 53 44 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066332 FK For-Sale Anodyne PLA2G4B 74 34 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066332 FK For-Sale Anodyne FAAH 26 46 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066332 FK For-Sale Anodyne EPHX2 24 44 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@@H]2N2CCCCC2)cc1 ZINC000147066332 FK For-Sale Anodyne PSMB2 44 33 C[C@@H](CNC(=O)CCc1nc(-c2ccccn2)no1)N1CCCC1 ZINC000147066514 ED On-Demand Anodyne PRCP 15 41 C[C@@H](CNC(=O)CCc1nc(-c2ccccn2)no1)N1CCCC1 ZINC000147066514 ED On-Demand Anodyne HCAR2 38 46 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@H]2N2CCCCC2)cc1 ZINC000147066528 FK For-Sale Anodyne HRH2 32 40 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@H]2N2CCCCC2)cc1 ZINC000147066528 FK For-Sale Anodyne HRH3 53 44 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@H]2N2CCCCC2)cc1 ZINC000147066528 FK For-Sale Anodyne PLA2G4B 74 34 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@H]2N2CCCCC2)cc1 ZINC000147066528 FK For-Sale Anodyne FAAH 26 46 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@H]2N2CCCCC2)cc1 ZINC000147066528 FK For-Sale Anodyne EPHX2 24 44 CCCCOc1ccc(NC(=O)O[C@H]2CCCC[C@H]2N2CCCCC2)cc1 ZINC000147066528 FK For-Sale Anodyne PSMB2 44 33 C=CCCOCC(=O)Nc1cccc(S(=O)(=O)Nc2ccccc2)c1 ZINC000147066604 FG On-Demand Mild CA4 18 43 C=CCCOCC(=O)Nc1cccc(S(=O)(=O)Nc2ccccc2)c1 ZINC000147066604 FG On-Demand Mild F13A1 23 40 O=C(Nc1nccs1)c1ccc2c(c1)CCNC2 ZINC000147066666 CE For-Sale Anodyne MAP 0 47 O=C(Nc1nccs1)c1ccc2c(c1)CCNC2 ZINC000147066666 CE For-Sale Anodyne MAP1 128 47 O=C(Nc1nccs1)c1ccc2c(c1)CCNC2 ZINC000147066666 CE For-Sale Anodyne MAPKAPK2 15 49 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(N3CCCN(C)CC3)cc1)C2 ZINC000147066692 GG On-Demand Anodyne DRD4 41 32 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(N3CCCN(C)CC3)cc1)C2 ZINC000147066692 GG On-Demand Anodyne ROCK2 32 50 C[C@H](CNC(=O)CCc1nc(-c2ccccn2)no1)N1CCCC1 ZINC000147066709 ED On-Demand Anodyne PRCP 15 41 C[C@H](CNC(=O)CCc1nc(-c2ccccn2)no1)N1CCCC1 ZINC000147066709 ED On-Demand Anodyne HCAR2 38 46 COc1ccc(OC)c([C@@H]2CCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)c1 ZINC000147066760 HG On-Demand Bother FKBP1A 49 38 COc1ccc(OC)c([C@@H]2CCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)c1 ZINC000147066760 HG On-Demand Bother CPT1A 119 42 COc1ccc(OC)c([C@@H]2CCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)c1 ZINC000147066760 HG On-Demand Bother CPT2 44 36 NC(=O)c1ccc(OCC(=O)NCc2cccnc2Oc2cccc(F)c2)cc1 ZINC000147066823 GF On-Demand Anodyne P2RY1 16 42 CC(C)[C@H]1CN(Cc2ccccc2)C[C@H]1C(=O)O ZINC000147066881 BE In-Stock Anodyne DRD3 24 40 CS(=O)(=O)c1cc(C(=O)Nc2cccc(OC(F)F)c2)cc([N+](=O)[O-])c1 ZINC000147066918 GF On-Demand Bother GRM4 15 46 CS(=O)(=O)c1cc(C(=O)Nc2cccc(OC(F)F)c2)cc([N+](=O)[O-])c1 ZINC000147066918 GF On-Demand Bother TAAR1 44 46 CS(=O)(=O)c1cc(C(=O)Nc2cccc(OC(F)F)c2)cc([N+](=O)[O-])c1 ZINC000147066918 GF On-Demand Bother KCNK3 106 37 CS(=O)(=O)c1cc(C(=O)Nc2cccc(OC(F)F)c2)cc([N+](=O)[O-])c1 ZINC000147066918 GF On-Demand Bother KCNK9 74 33 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H]1CCCN(c3ncccn3)C1)C2 ZINC000147067048 FD On-Demand Anodyne MTNR1A 22 40 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H]1CCCN(c3ncccn3)C1)C2 ZINC000147067048 FD On-Demand Anodyne MTNR1B 22 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OC(F)F)c2)c1 ZINC000147067114 EG On-Demand Bother GRM4 16 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OC(F)F)c2)c1 ZINC000147067114 EG On-Demand Bother MTNR1A 20 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OC(F)F)c2)c1 ZINC000147067114 EG On-Demand Bother MTNR1B 21 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OC(F)F)c2)c1 ZINC000147067114 EG On-Demand Bother BTK 17 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OC(F)F)c2)c1 ZINC000147067114 EG On-Demand Bother TAAR1 42 59 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OC(F)F)c2)c1 ZINC000147067114 EG On-Demand Bother AKR1C3 25 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OC(F)F)c2)c1 ZINC000147067114 EG On-Demand Bother AKR1C2 55 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OC(F)F)c2)c1 ZINC000147067114 EG On-Demand Bother KCNK3 62 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OC(F)F)c2)c1 ZINC000147067114 EG On-Demand Bother KCNK9 71 43 COC(=O)CN(c1ccccc1)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000147067206 FD In-Stock Bother OXTR 36 43 COC(=O)CN(c1ccccc1)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000147067206 FD In-Stock Bother AVPR1A 22 40 COC(=O)CN(c1ccccc1)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000147067206 FD In-Stock Bother MMP13 18 43 COC(=O)CN(c1ccccc1)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000147067206 FD In-Stock Bother COLA 67 43 COC(=O)CN(c1ccccc1)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000147067206 FD In-Stock Bother MMP2 32 49 COC(=O)CN(c1ccccc1)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000147067206 FD In-Stock Bother MMP8 56 49 COC(=O)CN(c1ccccc1)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000147067206 FD In-Stock Bother MMP9 38 49 COC(=O)CN(c1ccccc1)S(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000147067206 FD In-Stock Bother MMP1 45 49 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H]1CCCN(c3ncccn3)C1)C2 ZINC000147067241 FD On-Demand Anodyne MTNR1A 22 40 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H]1CCCN(c3ncccn3)C1)C2 ZINC000147067241 FD On-Demand Anodyne MTNR1B 22 40 O=C(Nc1cccc(OC(F)F)c1)c1ccn(-c2cccc(F)c2)n1 ZINC000147067300 EH On-Demand Anodyne GRM4 28 56 O=C(Nc1cccc(OC(F)F)c1)c1ccn(-c2cccc(F)c2)n1 ZINC000147067300 EH On-Demand Anodyne TAAR1 26 41 N#CC1CCN(C(=O)c2ccc(N3CCCS3(=O)=O)cc2)CC1 ZINC000147067348 ED On-Demand Mild L3MBTL3 73 42 Cc1cc(CNS(=O)(=O)c2ccc3c(c2)CCCC(=O)N3)no1 ZINC000147067359 ED On-Demand Anodyne PKM 42 48 COc1ccc2c(c1)OC[C@H](C(=O)N[C@H]1CCCN(c3ncccn3)C1)C2 ZINC000147067434 FD On-Demand Anodyne MTNR1A 22 40 COc1ccc2c(c1)OC[C@H](C(=O)N[C@H]1CCCN(c3ncccn3)C1)C2 ZINC000147067434 FD On-Demand Anodyne MTNR1B 22 40 CC(C)=C/C=C/C(C)=C/C=C/C=C(C)/C=C/C=C(C)/C=C/C1=C(C)C[C@@H](O)CC1(C)C ZINC000147067498 HK Annotated Bother RBP4 37 47 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne ALOX5 16 45 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne PTGER2 24 40 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne PPIA 45 35 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne PTGER1 47 43 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne PTGER4 32 40 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne KCNA2 0 46 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne MAP1 16 46 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne ABCB1 16 44 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne KCNA1 0 46 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne POBA 0 45 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne FFAR1 20 40 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne AKR1C3 26 40 CC(=O)c1sccc1OCc1ccccc1 ZINC000147067508 BH On-Demand Anodyne INPPL1 0 54 O=C(O)NCCCN1CCCCC1 ZINC000147067533 AD On-Demand Anodyne DRD3 20 41 O=C(O)NCCCN1CCCCC1 ZINC000147067533 AD On-Demand Anodyne HRH3 23 54 O=C(O)NCCCN1CCCCC1 ZINC000147067533 AD On-Demand Anodyne CHRNA7 28 51 O=C(O)NCCCN1CCCCC1 ZINC000147067533 AD On-Demand Anodyne HNMT 50 35 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H]1CCCN(c3ncccn3)C1)C2 ZINC000147067617 FD On-Demand Anodyne MTNR1A 22 40 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H]1CCCN(c3ncccn3)C1)C2 ZINC000147067617 FD On-Demand Anodyne MTNR1B 22 40 CC(C)=C/C=C/C(C)=C/C=C/C=C(C)/C=C/C=C(C)/C=C/C1=C(C)C[C@H](O)CC1(C)C ZINC000147067691 HK Annotated Bother RBP4 37 47 CCc1ncc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000147067728 DI On-Demand Anodyne MAOB 19 42 CCc1ncc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000147067728 DI On-Demand Anodyne FLT1 19 42 CCc1ncc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000147067728 DI On-Demand Anodyne GRM4 64 42 CCc1ncc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000147067728 DI On-Demand Anodyne TYK2 58 40 CCc1ncc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000147067728 DI On-Demand Anodyne CSF1R 22 41 CCc1ncc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000147067728 DI On-Demand Anodyne SHH 42 36 CCc1ncc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000147067728 DI On-Demand Anodyne USP7 45 34 CCc1ncc(C(=O)Nc2ccc(Cl)c(Cl)c2)s1 ZINC000147067728 DI On-Demand Anodyne USP47 57 34 N#C[C@H]1CCCN1S(N)(=O)=O ZINC000147067748 AB For-Sale Mild DPP4 23 41 N#C[C@@H]1CCCN1S(N)(=O)=O ZINC000147067956 AB For-Sale Mild DPP4 23 41 COC(=O)COc1ccc(S(=O)(=O)NCc2cc(C)on2)cc1 ZINC000147067995 ED On-Demand Anodyne ADAMTS4 44 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CC(F)(F)F)CC1 ZINC000147068013 DC On-Demand Anodyne P2RY12 84 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CC(F)(F)F)CC1 ZINC000147068013 DC On-Demand Anodyne NOD1 45 32 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147068038 HH On-Demand Bother PDE4A 39 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147068038 HH On-Demand Bother PDE4B 25 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147068038 HH On-Demand Bother PDE4D 25 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147068038 HH On-Demand Bother PDE4C 15 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147068038 HH On-Demand Bother MT-ND1 23 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(OC(F)F)c(F)c1 ZINC000147068093 EE On-Demand Anodyne ENV 41 33 C=C1C(=O)O[C@H]2/C=C(\C)C[C@H](OC(C)=O)/C=C(\C)CC/C=C(\C)CC[C@H]12 ZINC000147068186 FJ Annotated Mild MYB 0 45 CCCC(=O)Nc1ccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147068233 HF On-Demand Bother CA2 15 47 C=CC(=O)Nc1cc(Nc2ncc(Cl)c(-c3c[nH]c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C ZINC000147068258 KK In-Stock Anodyne INSR 33 73 C=CC(=O)Nc1cc(Nc2ncc(Cl)c(-c3c[nH]c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C ZINC000147068258 KK In-Stock Anodyne IGF1R 53 73 C=CC(=O)Nc1cc(Nc2ncc(Cl)c(-c3c[nH]c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C ZINC000147068258 KK In-Stock Anodyne JUN 17 47 C=CC(=O)Nc1cc(Nc2ncc(Cl)c(-c3c[nH]c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C ZINC000147068258 KK In-Stock Anodyne MAPK9 24 48 C=CC(=O)Nc1cc(Nc2ncc(Cl)c(-c3c[nH]c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C ZINC000147068258 KK In-Stock Anodyne MAPK8 21 48 C=CC(=O)Nc1cc(Nc2ncc(Cl)c(-c3c[nH]c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C ZINC000147068258 KK In-Stock Anodyne MAPK7 44 36 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(OC(F)F)c(F)c1 ZINC000147068270 EE On-Demand Anodyne ENV 41 33 N#CC1CCN(C(=O)c2csc(-c3ccc(Cl)cc3)n2)CC1 ZINC000147068321 EH On-Demand Mild TRPC6 57 49 N#CC1CCN(C(=O)c2csc(-c3ccc(Cl)cc3)n2)CC1 ZINC000147068321 EH On-Demand Mild TRPC3 37 49 C=C1C(=O)O[C@H]2/C=C(\C)CC/C=C(\C)[C@H](OC(C)=O)C/C=C(\C)CC[C@H]12 ZINC000147068393 FJ Annotated Mild MYB 0 43 Cc1cc(CNS(=O)(=O)c2ccc(-n3ncc(Cl)c(Cl)c3=O)cc2)no1 ZINC000147068515 HE On-Demand Anodyne NPBWR1 51 37 C=C1C(=O)O[C@H]2/C=C(\C)C[C@H](OC(C)=O)/C=C(\C)CC/C=C(\C)C[C@H](OC(C)=O)[C@H]12 ZINC000147068576 HI Annotated Mild MYB 0 54 Cc1cc(C(=O)Nc2cc(Cl)ccc2Cl)cc([N+](=O)[O-])c1 ZINC000147068592 EI On-Demand Bother KCNMA1 42 42 CC(C)N(Cc1ccccc1)C(=O)C(N)=O ZINC000147068690 BC On-Demand Anodyne SLC15A1 0 40 CC(C)N(Cc1ccccc1)C(=O)C(N)=O ZINC000147068690 BC On-Demand Anodyne NPR 42 35 CC(C)N(Cc1ccccc1)C(=O)C(N)=O ZINC000147068690 BC On-Demand Anodyne BLAIMP-1 0 40 COc1cc(/C=C/C(=O)N2CCC(C#N)CC2)ccc1OCC(N)=O ZINC000147068725 ED On-Demand Mild CCR2 39 51 C[C@@H]1CC[C@@H](C)N(Cc2ccccc2)C1 ZINC000147068839 BG On-Demand Anodyne SIGMAR1 36 45 CC(C)(C)c1ccc(S(=O)(=O)N(Cc2ccc(C#N)cc2)Cc2ccccn2)cc1 ZINC000147068913 HJ For-Sale Mild PTGER2 25 47 CC(C)(C)c1ccc(S(=O)(=O)N(Cc2ccc(C#N)cc2)Cc2ccccn2)cc1 ZINC000147068913 HJ For-Sale Mild CXCR3 18 68 N#CC1CCN(C(=O)/C=C/c2ccc(OCC(N)=O)cc2)CC1 ZINC000147068933 DD On-Demand Mild CCR2 43 37 Cc1cc(N2CCOCC2)ccc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147068980 FD On-Demand Anodyne HRH3 15 43 CCCCCNC(=O)C1CCN(C(=O)[C@@H](CCC)NC(N)=O)CC1 ZINC000147069075 ED On-Demand Anodyne P2RY12 117 35 CCCCCNC(=O)C1CCN(C(=O)[C@@H](CCC)NC(N)=O)CC1 ZINC000147069075 ED On-Demand Anodyne TPP2 33 43 Cc1cc(N2CCOCC2)ccc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147069181 FD On-Demand Anodyne HRH3 15 43 CCCCCNC(=O)C1CCN(C(=O)[C@H](CCC)NC(N)=O)CC1 ZINC000147069251 ED On-Demand Anodyne P2RY12 117 35 CCCCCNC(=O)C1CCN(C(=O)[C@H](CCC)NC(N)=O)CC1 ZINC000147069251 ED On-Demand Anodyne TPP2 33 43 CC(C)CC(C)(C)C[C@H]1N(C)[C@@H](C(=O)NCC[C@H](O)CO)[C@H](c2cccc(Cl)c2F)[C@@]12C(=O)Nc1cc(Cl)c(F)cc12 ZINC000147069323 KK Annotated Anodyne MDM2 76 55 Cc1cc(N2CCOCC2)ccc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147069379 FD On-Demand Anodyne HRH3 15 43 C[C@@H](Cc1cccc(F)c1)C(=O)NCCc1nc2ccccc2s1 ZINC000147069452 EH On-Demand Anodyne ST14 41 35 C[C@@H](Cc1cccc(F)c1)C(=O)NCCc1nc2ccccc2s1 ZINC000147069452 EH On-Demand Anodyne PIN1 32 43 C[C@@H](Cc1cccc(F)c1)C(=O)NCCc1nc2ccccc2s1 ZINC000147069452 EH On-Demand Anodyne TMPRSS6 67 35 Cc1cc(N2CCOCC2)ccc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147069577 FD On-Demand Anodyne HRH3 15 43 C[C@H](Cc1cccc(F)c1)C(=O)NCCc1nc2ccccc2s1 ZINC000147069645 EH On-Demand Anodyne ST14 41 35 C[C@H](Cc1cccc(F)c1)C(=O)NCCc1nc2ccccc2s1 ZINC000147069645 EH On-Demand Anodyne PIN1 32 43 C[C@H](Cc1cccc(F)c1)C(=O)NCCc1nc2ccccc2s1 ZINC000147069645 EH On-Demand Anodyne TMPRSS6 67 35 CC(C)[C@@H](C)[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147069659 FI In-Stock Anodyne CASP3 24 40 CC(C)[C@@H](C)[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147069659 FI In-Stock Anodyne CAPN1 29 53 COc1cccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147069671 EF On-Demand Bother DRD4 44 34 COc1cccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147069671 EF On-Demand Bother CTSL 15 46 COc1cccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147069671 EF On-Demand Bother MTNR1A 81 50 COc1cccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147069671 EF On-Demand Bother MTNR1B 66 48 COc1cccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147069671 EF On-Demand Bother TAAR1 26 43 COc1cccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147069671 EF On-Demand Bother AKR1C3 15 43 COc1cccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147069671 EF On-Demand Bother CRTM 57 35 COc1cccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147069671 EF On-Demand Bother AKR1C2 27 42 O=C(OO)c1cccc(C(F)(F)F)c1 ZINC000147069683 BE For-Sale Reactive CCR2 56 37 O=C(OO)c1cccc(C(F)(F)F)c1 ZINC000147069683 BE For-Sale Reactive BTK 15 40 O=C(OO)c1cccc(C(F)(F)F)c1 ZINC000147069683 BE For-Sale Reactive AKR1C3 16 50 O=C(OO)c1cccc(C(F)(F)F)c1 ZINC000147069683 BE For-Sale Reactive KCNK3 18 50 O=C(OO)c1cccc(C(F)(F)F)c1 ZINC000147069683 BE For-Sale Reactive PDS 45 35 CC(C)[C@H](C)[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147069835 FI In-Stock Anodyne CASP3 24 40 CC(C)[C@H](C)[C@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147069835 FI In-Stock Anodyne CAPN1 29 53 C[C@@H]1OC(=O)[C@H](N)[C@H]1C(=O)O ZINC000147069855 AA For-Sale Anodyne NAAA 46 33 CNC(=O)c1cccc(NC(=O)[C@H](C)Nc2cc(C#N)ccc2OC)c1 ZINC000147069891 FE On-Demand Mild KCNK3 81 38 CNC(=O)c1cccc(NC(=O)[C@H](C)Nc2cc(C#N)ccc2OC)c1 ZINC000147069891 FE On-Demand Mild KCNK9 63 37 COCCOc1ccc(S(=O)(=O)NCc2cc(C)on2)cc1 ZINC000147069979 ED On-Demand Anodyne MMP1 17 42 CC(C)[C@@H](C)[C@@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147070018 FI In-Stock Anodyne CASP3 24 40 CC(C)[C@@H](C)[C@@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147070018 FI In-Stock Anodyne CAPN1 29 53 COC(=O)[C@H]1[C@H](C)OC(=O)[C@@H]1N ZINC000147070040 AB For-Sale Anodyne NAAA 87 37 COc1ccc(C(=O)N2CCC(C#N)CC2)cn1 ZINC000147070049 BD On-Demand Mild L3MBTL3 56 37 CCN(CC)c1ccc(NC(=O)c2csc(COC)n2)cc1 ZINC000147070051 DG On-Demand Anodyne GHSR 16 42 CCc1ccccc1-c1ccccc1C(=O)O ZINC000147070072 BH On-Demand Anodyne AGTR1 32 41 CCc1ccccc1-c1ccccc1C(=O)O ZINC000147070072 BH On-Demand Anodyne FOLH1 17 54 CCc1ccccc1-c1ccccc1C(=O)O ZINC000147070072 BH On-Demand Anodyne AGTR1B 44 36 CCc1ccccc1-c1ccccc1C(=O)O ZINC000147070072 BH On-Demand Anodyne AKR1C2 40 38 O=C(NNC(=O)c1occ(-c2ccccc2)c1-c1ccccc1)c1ccc(O)c(Cl)c1 ZINC000147070108 IK Annotated Reactive ADCYAP1R1 69 38 CC(C)[C@H](C)[C@@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147070219 FI In-Stock Anodyne CASP3 24 40 CC(C)[C@H](C)[C@@H](NC(=O)OCC1c2ccccc2-c2ccccc21)C(=O)O ZINC000147070219 FI In-Stock Anodyne CAPN1 29 53 Cc1cc(C(=O)Nc2ccc(Cl)cc2)cc([N+](=O)[O-])c1 ZINC000147070274 CH On-Demand Bother PPIA 17 40 Cc1cc(C(=O)Nc2ccc(Cl)cc2)cc([N+](=O)[O-])c1 ZINC000147070274 CH On-Demand Bother SCN10A 24 44 Cc1cc(C(=O)Nc2ccc(Cl)cc2)cc([N+](=O)[O-])c1 ZINC000147070274 CH On-Demand Bother CSF1R 15 41 Cc1cc(C(=O)Nc2ccc(Cl)cc2)cc([N+](=O)[O-])c1 ZINC000147070274 CH On-Demand Bother Q25615_ONCVO 36 45 Cc1cc(C(=O)Nc2ccc(Cl)cc2)cc([N+](=O)[O-])c1 ZINC000147070274 CH On-Demand Bother USP47 41 33 Cc1cc(C(=O)Nc2ccc(Cl)cc2)cc([N+](=O)[O-])c1 ZINC000147070274 CH On-Demand Bother KCNK3 62 48 Cc1cc(C(=O)Nc2ccc(Cl)cc2)cc([N+](=O)[O-])c1 ZINC000147070274 CH On-Demand Bother KCNK9 44 43 COC[C@@]1(CN)CCN(Cc2ccccc2)C1 ZINC000147070292 BD For-Sale Anodyne SIGMAR1 61 42 COC[C@@]1(CN)CCN(Cc2ccccc2)C1 ZINC000147070292 BD For-Sale Anodyne NPFFR1 53 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OCC(F)(F)F)cc1 ZINC000147070296 EF On-Demand Anodyne SCN2A 17 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OCC(F)(F)F)cc1 ZINC000147070296 EF On-Demand Anodyne ACR 33 43 C[C@H](CNC(=O)c1cnn(-c2cccc(C(F)(F)F)c2)c1C1CC1)N1CCCC1 ZINC000147070330 HH On-Demand Anodyne CCR2 87 37 CCCCC(C)(C)C[C@H]1N(C)[C@@H](C(=O)NCC[C@H](O)CO)[C@H](c2cccc(Cl)c2)[C@@]12C(=O)Nc1cc(Cl)c(F)cc12 ZINC000147070431 KK Annotated Anodyne MDM2 65 68 C#CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147070443 EC On-Demand Mild ST14 75 35 C#CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147070443 EC On-Demand Mild SFRP1 86 42 C#CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147070443 EC On-Demand Mild WNT3 61 33 C#CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147070443 EC On-Demand Mild L3MBTL3 45 41 C#CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147070443 EC On-Demand Mild TMPRSS6 52 32 C[C@H]1OC(=O)[C@@H](N)[C@@H]1C(=O)O ZINC000147070449 AA For-Sale Anodyne NAAA 46 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OCC(F)(F)F)cc1 ZINC000147070499 EF On-Demand Anodyne SCN2A 17 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OCC(F)(F)F)cc1 ZINC000147070499 EF On-Demand Anodyne ACR 33 43 COC[C@]1(CN)CCN(Cc2ccccc2)C1 ZINC000147070502 BD For-Sale Anodyne SIGMAR1 61 42 COC[C@]1(CN)CCN(Cc2ccccc2)C1 ZINC000147070502 BD For-Sale Anodyne NPFFR1 53 40 CCc1ccc(OC(=O)NCc2ccccc2)cc1 ZINC000147070529 CH For-Sale Anodyne PPARA 23 49 CCc1ccc(OC(=O)NCc2ccccc2)cc1 ZINC000147070529 CH For-Sale Anodyne ANPEP 22 43 CCc1ccc(OC(=O)NCc2ccccc2)cc1 ZINC000147070529 CH For-Sale Anodyne ECR 19 40 CCc1ccc(OC(=O)NCc2ccccc2)cc1 ZINC000147070529 CH For-Sale Anodyne BCHE 22 43 CCc1ccc(OC(=O)NCc2ccccc2)cc1 ZINC000147070529 CH For-Sale Anodyne FAAH 44 59 CCc1ccc(OC(=O)NCc2ccccc2)cc1 ZINC000147070529 CH For-Sale Anodyne AMP1_PLAFQ 52 38 CCc1ccc(OC(=O)NCc2ccccc2)cc1 ZINC000147070529 CH For-Sale Anodyne NAAA 19 40 CCc1ccc(OC(=O)NCc2ccccc2)cc1 ZINC000147070529 CH For-Sale Anodyne E3UJZ5_SPOLI 15 40 CCc1ccc(OC(=O)NCc2ccccc2)cc1 ZINC000147070529 CH For-Sale Anodyne PDS 89 51 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne ACE 44 39 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne FKBP1A 38 40 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne CELA1 19 40 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne ELANE 15 42 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne SIGMAR1 15 64 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne CTSB 30 43 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne PAPA1_CARPA 45 37 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne CTSK 28 43 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne CTSL 29 43 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne CCR5 35 52 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne PREP 36 42 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne AMY2 52 37 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne CAPNS1 57 33 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne CTSS 16 43 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne CAPN1 41 37 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne CAPN2 51 35 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne NPR 59 35 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne NAAA 27 40 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne TRPM8 15 44 CN(C(=O)OCc1ccccc1)C1CCCC1 ZINC000147070836 BG For-Sale Anodyne SLC12A5 74 40 Cc1nn(-c2ccccc2)c(N2CCN(C(=O)OC(C)(C)C)CC2)c1C=O ZINC000147070861 FG For-Sale Anodyne GPR119 41 43 C=CCOC(=O)NCCCCCC ZINC000147070877 AE For-Sale Mild EPHX2 16 40 C=CCOC(=O)NCCCCCC ZINC000147070877 AE For-Sale Mild ASAH1 83 35 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne PPIA 16 42 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne CASP3 15 40 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne KLK3 53 35 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne CTSB 50 44 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne PAPA1_CARPA 57 38 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne CYSP_TRYCR 43 37 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne CTSK 32 44 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne CTSL 37 42 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne CAPNS1 65 39 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne CTSS 16 44 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne CAPN1 71 44 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne CAPN2 112 44 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne PLAU 17 41 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne TPSAB1 41 47 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne NPR 70 38 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne KDM1A 15 45 N=C(NCc1ccccc1)NC(=O)OCc1ccccc1 ZINC000147071096 CF Annotated Anodyne PDS 57 40 C[C@@H](CNC(=O)c1cn(-c2ccccc2)nn1)N1CCCC1 ZINC000147071371 CD On-Demand Anodyne ESRRA 23 43 O=C(O)[C@@H]1CCCN(C2CCN(C(=O)c3c4ccccc4cc4ccccc34)CC2)C1 ZINC000147071482 HI In-Stock Anodyne SLC6A1 138 38 O=C(O)[C@@H]1CCCN(C2CCN(C(=O)c3c4ccccc4cc4ccccc34)CC2)C1 ZINC000147071482 HI In-Stock Anodyne ACACA 39 72 O=C(O)[C@@H]1CCCN(C2CCN(C(=O)c3c4ccccc4cc4ccccc34)CC2)C1 ZINC000147071482 HI In-Stock Anodyne ACACB 33 74 O=C(O)[C@@H]1CCCN(C2CCN(C(=O)c3c4ccccc4cc4ccccc34)CC2)C1 ZINC000147071482 HI In-Stock Anodyne L3MBTL3 112 53 Cc1nc(-c2cccc(Cl)c2)sc1C(=O)N1CCC(C#N)CC1 ZINC000147071505 EI On-Demand Mild GRM5 16 41 C[C@H](CNC(=O)c1cn(-c2ccccc2)nn1)N1CCCC1 ZINC000147071561 CD On-Demand Anodyne ESRRA 23 43 O=C(c1cccc(OCc2ccccc2OC(F)F)c1)N1CCOCC1 ZINC000147071572 FG On-Demand Anodyne ITGAL 42 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC(NS(C)(=O)=O)CC1 ZINC000147071665 EB On-Demand Anodyne P2RY12 61 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC(NS(C)(=O)=O)CC1 ZINC000147071665 EB On-Demand Anodyne CCR8 55 33 C[C@@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071793 GG On-Demand Anodyne F2 52 45 C[C@@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071793 GG On-Demand Anodyne ELANE 57 36 C[C@@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071793 GG On-Demand Anodyne P2RX7 21 42 C[C@@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071793 GG On-Demand Anodyne TRY1_BOVIN 33 45 C[C@@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071793 GG On-Demand Anodyne UL80 19 40 C[C@@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071793 GG On-Demand Anodyne PREP 38 45 C[C@@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071793 GG On-Demand Anodyne TPP2 36 40 C[C@@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071793 GG On-Demand Anodyne TMPRSS11D 49 35 COc1ccc(NC(C)=O)cc1S(=O)(=O)NCc1cc(C)on1 ZINC000147071801 ED On-Demand Anodyne COLA 43 33 COc1ccc(NC(C)=O)cc1S(=O)(=O)NCc1cc(C)on1 ZINC000147071801 ED On-Demand Anodyne CPT1A 40 33 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccnn2Cc2cccc3ccccc23)c1 ZINC000147071840 HI On-Demand Bother NPBWR1 61 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(NS(C)(=O)=O)CC1 ZINC000147071852 EB On-Demand Anodyne P2RY12 61 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(NS(C)(=O)=O)CC1 ZINC000147071852 EB On-Demand Anodyne CCR8 55 33 CC(C)CCO[C@@H](C)C(=O)NCCNc1ccccc1[N+](=O)[O-] ZINC000147071938 DF On-Demand Bother COLA 91 37 C[C@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071957 GG On-Demand Anodyne F2 52 45 C[C@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071957 GG On-Demand Anodyne ELANE 57 36 C[C@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071957 GG On-Demand Anodyne P2RX7 21 42 C[C@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071957 GG On-Demand Anodyne TRY1_BOVIN 33 45 C[C@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071957 GG On-Demand Anodyne UL80 19 40 C[C@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071957 GG On-Demand Anodyne PREP 38 45 C[C@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071957 GG On-Demand Anodyne TPP2 36 40 C[C@H](CNC(=O)[C@@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147071957 GG On-Demand Anodyne TMPRSS11D 49 35 Cn1ccnc1COc1ccc(NC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147071995 HI On-Demand Anodyne PRNP 53 32 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(-c3ncc4n3CCCC4)cc2)c1 ZINC000147072024 GI On-Demand Bother TAAR1 21 41 Cc1cc(CNS(=O)(=O)c2cccc(C(F)(F)F)c2)no1 ZINC000147072063 DE On-Demand Anodyne CACNA1B 40 34 C[C@@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072125 GG On-Demand Anodyne F2 52 45 C[C@@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072125 GG On-Demand Anodyne ELANE 57 36 C[C@@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072125 GG On-Demand Anodyne P2RX7 21 42 C[C@@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072125 GG On-Demand Anodyne TRY1_BOVIN 33 45 C[C@@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072125 GG On-Demand Anodyne UL80 19 40 C[C@@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072125 GG On-Demand Anodyne PREP 38 45 C[C@@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072125 GG On-Demand Anodyne TPP2 36 40 C[C@@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072125 GG On-Demand Anodyne TMPRSS11D 49 35 CC(C)CCO[C@H](C)C(=O)NCCNc1ccccc1[N+](=O)[O-] ZINC000147072138 DF On-Demand Bother COLA 91 37 O=C(C1CCN(Cc2ccsc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147072147 II For-Sale Anodyne SIGMAR1 15 41 Cn1ccnc1COc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147072207 GI On-Demand Anodyne NAMPT 24 41 C[C@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072331 GG On-Demand Anodyne F2 52 45 C[C@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072331 GG On-Demand Anodyne ELANE 57 36 C[C@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072331 GG On-Demand Anodyne P2RX7 21 42 C[C@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072331 GG On-Demand Anodyne TRY1_BOVIN 33 45 C[C@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072331 GG On-Demand Anodyne UL80 19 40 C[C@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072331 GG On-Demand Anodyne PREP 38 45 C[C@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072331 GG On-Demand Anodyne TPP2 36 40 C[C@H](CNC(=O)[C@H]1CCCN1C(=O)c1ccc(Cl)c(Cl)c1)N1CCCC1 ZINC000147072331 GG On-Demand Anodyne TMPRSS11D 49 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne F2 74 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne PLG 61 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne PRSS1 27 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne ACE 75 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne ACHE 18 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne OPRM1 19 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne OPRD1 18 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne GHRHR 75 45 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne SLC18A2 40 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne P2RY12 209 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne GRIN2B 35 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne TRY2_BOVIN 85 36 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne TRY1_BOVIN 58 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne CCKAR 26 46 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne CTSK 50 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne CCR1 30 44 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne NPFFR2 50 32 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne CTRB1 42 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne REN 40 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne PCSK5 23 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne FURIN 21 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne CCKBR 44 46 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne GHSR 19 45 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne CAPN1 30 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne DPP7 46 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne ST14 108 39 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne CTRB_BOVIN 56 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne AMP1_PLAFQ 20 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072352 EG On-Demand Anodyne TMPRSS6 74 36 CCCC(=O)Nc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147072388 EE On-Demand Anodyne F2R 16 47 Cn1ccnc1COc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147072413 GI On-Demand Anodyne NAMPT 24 41 CN1CCC(CNC(=O)[C@@H]2N[C@H](CC(C)(C)C)[C@]3(C(=O)Nc4cc(Cl)ccc43)[C@H]2c2cccc(Cl)c2F)CC1 ZINC000147072481 KK Annotated Anodyne MDM2 107 77 CN1CCC(CNC(=O)[C@@H]2N[C@H](CC(C)(C)C)[C@]3(C(=O)Nc4cc(Cl)ccc43)[C@H]2c2cccc(Cl)c2F)CC1 ZINC000147072481 KK Annotated Anodyne CACNA1I 46 37 CCOC(=O)N1CCN(S(=O)(=O)NCc2cc(C)on2)CC1 ZINC000147072488 EC On-Demand Anodyne TGM2 33 43 CCOC(=O)N1CCN(S(=O)(=O)NCc2cc(C)on2)CC1 ZINC000147072488 EC On-Demand Anodyne F13A1 42 43 COc1ccc(C#N)cc1N[C@H](C)C(=O)NCc1ccc(OC)c(OC)c1 ZINC000147072526 FF On-Demand Mild MT-ND1 24 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne F2 74 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne PLG 61 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne PRSS1 27 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne ACE 75 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne ACHE 18 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne OPRM1 19 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne OPRD1 18 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne GHRHR 75 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne SLC18A2 40 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne P2RY12 209 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne GRIN2B 35 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne TRY2_BOVIN 85 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne TRY1_BOVIN 58 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne CCKAR 26 46 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne CTSK 50 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne CCR1 30 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne NPFFR2 50 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne CTRB1 42 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne REN 40 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne PCSK5 23 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne FURIN 21 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne CCKBR 44 46 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne GHSR 19 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne CAPN1 30 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne DPP7 46 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne ST14 108 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne CTRB_BOVIN 56 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne AMP1_PLAFQ 20 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072535 EG On-Demand Anodyne TMPRSS6 74 36 C[C@H](CNC(=O)c1cnc2ccccn2c1=O)N1CCCC1 ZINC000147072545 DC On-Demand Anodyne HCN1 43 37 C[C@H](CNC(=O)c1cnc2ccccn2c1=O)N1CCCC1 ZINC000147072545 DC On-Demand Anodyne POLR1A 72 40 CCCC(=O)Nc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147072565 EE On-Demand Anodyne F2R 16 47 O=C(Nc1c[nH]c2ncc(Br)cc12)c1cnn(Cc2ccccc2)c1 ZINC000147072611 GH For-Sale Anodyne PIM1 48 40 O=C(Nc1c[nH]c2ncc(Br)cc12)c1cnn(Cc2ccccc2)c1 ZINC000147072611 GH For-Sale Anodyne ITK 15 42 O=C(Nc1c[nH]c2ncc(Br)cc12)c1cnn(Cc2ccccc2)c1 ZINC000147072611 GH For-Sale Anodyne CDC7 18 42 O=C(Nc1c[nH]c2ncc(Br)cc12)c1cnn(Cc2ccccc2)c1 ZINC000147072611 GH For-Sale Anodyne PIM3 57 34 Cn1ccnc1COc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147072615 GI On-Demand Anodyne NAMPT 24 41 CCCCC/C=C/COC(=O)CC ZINC000147072693 AG For-Sale Anodyne CNR1 15 49 CCCCC/C=C/COC(=O)CC ZINC000147072693 AG For-Sale Anodyne FAAH 19 49 CCCCC/C=C/COC(=O)CC ZINC000147072693 AG For-Sale Anodyne LPAR3 40 41 CCCCC/C=C/COC(=O)CC ZINC000147072693 AG For-Sale Anodyne FABP3 37 48 CCCCC/C=C/COC(=O)CC ZINC000147072693 AG For-Sale Anodyne FABP1 16 48 Cc1nn(C(F)F)c(C)c1CC(=O)N1CCC(CCc2ccccc2)CC1 ZINC000147072743 GI On-Demand Anodyne GRIN2B 31 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(OCc3nccn3C)cc1)C2 ZINC000147072799 GG On-Demand Anodyne ROCK2 35 50 CN(C)C(=O)COc1ccccc1C(=O)N1CCC(C#N)CC1 ZINC000147072907 DD On-Demand Mild HCN1 44 33 CN(C)C(=O)COc1ccccc1C(=O)N1CCC(C#N)CC1 ZINC000147072907 DD On-Demand Mild HCN4 43 33 COC(=O)CNC(=O)Cc1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147072928 HD On-Demand Bother CA9 17 42 COC(=O)CNC(=O)Cc1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147072928 HD On-Demand Bother TAAR1 26 40 COC(=O)CNC(=O)Cc1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147072928 HD On-Demand Bother AKR1C3 15 41 COC(=O)CNC(=O)Cc1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147072928 HD On-Demand Bother AKR1C2 46 38 COc1cc2nc(-c3ccccn3)[nH]c2cc1C ZINC000147072934 BF On-Demand Anodyne METAP2 47 56 O=C(Cl)c1nc2ccc(Br)cc2s1 ZINC000147072969 CG For-Sale Reactive CSNK1D 21 41 O=C(Cl)c1nc2ccc(Br)cc2s1 ZINC000147072969 CG For-Sale Reactive HSD17B1 28 41 CCc1sc(NC(=O)c2ccc3c(c2)COC3)nc1-c1ccccc1 ZINC000147073018 FJ On-Demand Anodyne ADORA1 18 49 COc1cc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc(OC)c1OC ZINC000147073312 EG On-Demand Bother SMO 19 42 COc1cc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc(OC)c1OC ZINC000147073312 EG On-Demand Bother KCNK3 46 39 COc1cc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc(OC)c1OC ZINC000147073312 EG On-Demand Bother KCNK9 53 39 COc1ccc(OC(F)F)c(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147073325 HF On-Demand Bother TAAR1 20 42 Cc1nc(-c2ccc(F)cc2)sc1C(=O)N1CCC(C#N)CC1 ZINC000147073343 EH On-Demand Mild THRA 17 46 Cc1nc(-c2ccc(F)cc2)sc1C(=O)N1CCC(C#N)CC1 ZINC000147073343 EH On-Demand Mild PPARA 15 43 COc1ccc(OC(F)F)c(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147073527 FG On-Demand Bother KCNMA1 31 44 COc1ccc(OC(F)F)c(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147073527 FG On-Demand Bother TAAR1 18 40 COc1ccc(OC(F)F)c(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147073527 FG On-Demand Bother AKR1C3 16 42 COc1ccc(OC(F)F)c(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147073527 FG On-Demand Bother AKR1C2 52 44 COCc1nc(C(=O)Nc2ccc(C(C)(C)C)cc2)cs1 ZINC000147073532 DH On-Demand Anodyne TRPV1 23 44 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073556 FD On-Demand Anodyne CA2 16 47 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073556 FD On-Demand Anodyne HDAC10 46 39 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073556 FD On-Demand Anodyne CA4 16 47 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073556 FD On-Demand Anodyne HDAC11 46 39 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073556 FD On-Demand Anodyne ST14 76 38 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073556 FD On-Demand Anodyne CCR8 42 32 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073556 FD On-Demand Anodyne TMPRSS6 61 36 Cc1ccc(C(=O)O)c(C#N)c1O ZINC000147073566 AD For-Sale Anodyne AKR1C2 44 33 Cc1ccc(C(=O)O)c(C#N)c1O ZINC000147073566 AD For-Sale Anodyne AKR1C1 48 33 CC(=O)N[C@@H]1CCN(C(=O)[C@H](OC(C)=O)c2ccccc2)[C@H](Cc2ccc(Cl)cc2)C1 ZINC000147073633 IH For-Sale Anodyne TACR1 16 49 C[C@@H](Nc1cc(Cl)nc(SCc2cccc(F)c2F)n1)[C@@H](O)CO ZINC000147073714 GF For-Sale Anodyne CXCR2 53 59 C[C@@H](Nc1cc(Cl)nc(SCc2cccc(F)c2F)n1)[C@@H](O)CO ZINC000147073714 GF For-Sale Anodyne CX3CR1 35 45 O=C(O)CNC(=O)OC/C=C/c1ccccc1 ZINC000147073719 BD For-Sale Anodyne CACNA1B 58 43 O=C(C1CCN(C2CCCCC2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147073728 HJ For-Sale Anodyne HRH3 35 45 O=C(C1CCN(C2CCCCC2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147073728 HJ For-Sale Anodyne L3MBTL3 71 37 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073739 FD On-Demand Anodyne CA2 16 47 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073739 FD On-Demand Anodyne HDAC10 46 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073739 FD On-Demand Anodyne CA4 16 47 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073739 FD On-Demand Anodyne HDAC11 46 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073739 FD On-Demand Anodyne ST14 76 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073739 FD On-Demand Anodyne CCR8 42 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147073739 FD On-Demand Anodyne TMPRSS6 61 36 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1sc2c(c1C#N)CCCCC2 ZINC000147073765 GI On-Demand Mild MAPK10 20 52 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1sc2c(c1C#N)CCCCC2 ZINC000147073765 GI On-Demand Mild FLT3 15 40 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1sc2c(c1C#N)CCCCC2 ZINC000147073765 GI On-Demand Mild VIPR1 31 49 CCc1ccc(C(F)(F)F)cc1OC ZINC000147073804 BG For-Sale Anodyne PPARD 23 40 CCCC(=O)Nc1ccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147073948 FG On-Demand Bother MTNR1A 36 51 CCCC(=O)Nc1ccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147073948 FG On-Demand Bother MTNR1B 33 51 CCCC(=O)Nc1ccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147073948 FG On-Demand Bother CA9 15 41 CCN(CC)C(=O)c1cccc(OCc2ccccc2OC(F)F)c1 ZINC000147073966 EI On-Demand Anodyne PDS 47 34 COc1ccc(Oc2ncc(Br)s2)c(Cl)c1 ZINC000147074314 DI For-Sale Anodyne ACACB 17 44 CCCC[C@H](NC(N)=O)C(=O)NCc1coc(-c2cccs2)n1 ZINC000147074363 EE On-Demand Anodyne HPN 41 31 CC(CO)(CO)NC(=O)Cc1ccc(-c2ccccc2)cc1 ZINC000147074400 CD On-Demand Anodyne MME 45 40 CC(CO)(CO)NC(=O)Cc1ccc(-c2ccccc2)cc1 ZINC000147074400 CD On-Demand Anodyne SLC15A1 0 40 CC(CO)(CO)NC(=O)Cc1ccc(-c2ccccc2)cc1 ZINC000147074400 CD On-Demand Anodyne ACE2 40 40 CC(CO)(CO)NC(=O)Cc1ccc(-c2ccccc2)cc1 ZINC000147074400 CD On-Demand Anodyne E1 0 40 CC(CO)(CO)NC(=O)Cc1ccc(-c2ccccc2)cc1 ZINC000147074400 CD On-Demand Anodyne FFAR1 18 40 CC(CO)(CO)NC(=O)Cc1ccc(-c2ccccc2)cc1 ZINC000147074400 CD On-Demand Anodyne BLAIMP-1 0 43 C[C@H](NC(=O)c1ccn(-c2cccc(F)c2)n1)c1ccc(NC(=O)NC2CC2)cc1 ZINC000147074411 HH On-Demand Anodyne EPHX2 40 36 COc1cc(CNC(=O)[C@@H](C)Cc2cccc(F)c2)ccc1OC(F)F ZINC000147074415 FH On-Demand Anodyne ANPEP 17 46 COc1cc(CNC(=O)[C@@H](C)Cc2cccc(F)c2)ccc1OC(F)F ZINC000147074415 FH On-Demand Anodyne PPARD 18 41 COc1cc(CNC(=O)[C@@H](C)Cc2cccc(F)c2)ccc1OC(F)F ZINC000147074415 FH On-Demand Anodyne CARM1 44 35 COc1ccc(Nc2nc3c(Nc4ccccc4S(C)(=O)=O)cccn3n2)cc1 ZINC000147074507 HH Annotated Anodyne JAK2 29 64 C[C@@H](NC(=O)c1ccn(-c2cccc(F)c2)n1)c1ccc(NC(=O)NC2CC2)cc1 ZINC000147074608 HH On-Demand Anodyne EPHX2 40 36 COc1cc(CNC(=O)[C@H](C)Cc2cccc(F)c2)ccc1OC(F)F ZINC000147074630 FH On-Demand Anodyne ANPEP 17 46 COc1cc(CNC(=O)[C@H](C)Cc2cccc(F)c2)ccc1OC(F)F ZINC000147074630 FH On-Demand Anodyne PPARD 18 41 COc1cc(CNC(=O)[C@H](C)Cc2cccc(F)c2)ccc1OC(F)F ZINC000147074630 FH On-Demand Anodyne CARM1 44 35 COc1cc(N)c(Cl)cc1CC(=O)O ZINC000147074735 BD In-Stock Anodyne HTR3A 0 43 COc1cc(N)c(Cl)cc1CC(=O)O ZINC000147074735 BD In-Stock Anodyne HTR4 85 49 N#CC1CCN(C(=O)c2cc3ccccc3c(=O)[nH]2)CC1 ZINC000147074745 CD On-Demand Mild GRIN2B 27 41 N#CC1CCN(C(=O)c2cc3ccccc3c(=O)[nH]2)CC1 ZINC000147074745 CD On-Demand Mild HRH4 29 44 N#CC1CCN(C(=O)c2cc3ccccc3c(=O)[nH]2)CC1 ZINC000147074745 CD On-Demand Mild AKR1C3 19 46 CC(C)Oc1ccccc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147074831 EF On-Demand Anodyne ADORA2B 27 40 C[C@@H](Nc1cc(NS(=O)(=O)N2CCC2)nc(SCc2cccc(F)c2F)n1)[C@H](O)CO ZINC000147074900 JD In-Stock Anodyne CXCR2 49 82 C[C@@H](Nc1cc(NS(=O)(=O)N2CCC2)nc(SCc2cccc(F)c2F)n1)[C@H](O)CO ZINC000147074900 JD In-Stock Anodyne CX3CR1 15 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2cc(C)on2)CC1 ZINC000147074929 FD On-Demand Anodyne P2RY12 174 38 C[C@@H](CNC(=O)c1cnn(-c2ccccc2)c1C1CC1)N1CCCC1 ZINC000147074952 EF On-Demand Anodyne HCN1 40 33 C[C@@H](CNC(=O)c1cnn(-c2ccccc2)c1C1CC1)N1CCCC1 ZINC000147074952 EF On-Demand Anodyne HCN4 40 33 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne ACE 82 43 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne OPRM1 50 41 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne OPRD1 52 41 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CELA1 18 42 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne MME 119 46 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne LTA4H 40 47 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne ANPEP 80 41 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne TACR1 28 49 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne FCER2 64 36 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CASP3 34 49 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne BMP1 18 40 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne RNPEP 24 41 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CASP8 21 43 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne KLK3 106 47 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CTSB 86 48 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne PAPA1_CARPA 87 43 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CYSP_TRYCR 68 46 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CTSK 50 46 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CTSL 62 46 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne NPFFR2 60 31 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CTRB1 27 48 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CAPNS1 75 44 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne MMP2 27 48 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne MMP3 55 46 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne HLA-DRB1 57 34 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne LNPEP 17 41 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne MMP11 54 34 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CTSS 35 46 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CAPN1 117 49 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CASP1 38 43 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CAPN2 157 46 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne ACE2 73 39 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CASP6 32 43 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne CASP9 43 43 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne LAP3 46 41 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne ST14 43 34 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne MMP1 35 48 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne FPR1 70 38 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne NPR 99 43 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne AMP1_PLAFQ 33 41 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne PSMB5 70 48 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne POLG_WNV 40 35 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne BIRC2 36 42 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne NPFFR1 65 32 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne Q6PRC7_IXORI 40 31 C[C@@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075043 GE For-Sale Anodyne TMPRSS6 51 34 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild GRIN2B 24 41 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild KLK3 55 36 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild CTSB 44 43 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild PAPA1_CARPA 43 34 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild CYSP_TRYCR 36 42 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild CTSK 31 43 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild CTSL 35 44 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild PREP 20 41 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild CAPNS1 55 34 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild CAPN1 59 46 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild CASP1 23 40 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild CAPN2 91 45 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild TGM2 34 50 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild NPR 63 37 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild F13A1 26 50 O=CC1CCC(CNC(=O)OCc2ccccc2)CC1 ZINC000147075089 CF In-Stock Mild VCP 40 33 C[C@H](CNC(=O)c1cnn(-c2ccccc2)c1C1CC1)N1CCCC1 ZINC000147075125 EF On-Demand Anodyne HCN1 40 33 C[C@H](CNC(=O)c1cnn(-c2ccccc2)c1C1CC1)N1CCCC1 ZINC000147075125 EF On-Demand Anodyne HCN4 40 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2cc(C)on2)CC1 ZINC000147075141 FD On-Demand Anodyne P2RY12 174 38 Oc1ccc(CCBr)c(F)c1 ZINC000147075143 BE For-Sale Reactive TYR 27 50 Oc1ccc(CCBr)c(F)c1 ZINC000147075143 BE For-Sale Reactive PPO2 17 50 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne ACE 82 43 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne OPRM1 50 41 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne OPRD1 52 41 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CELA1 18 42 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne MME 119 46 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne LTA4H 40 47 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne ANPEP 80 41 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne TACR1 28 49 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne FCER2 64 36 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CASP3 34 49 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne BMP1 18 40 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne RNPEP 24 41 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CASP8 21 43 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne KLK3 106 47 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CTSB 86 48 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne PAPA1_CARPA 87 43 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CYSP_TRYCR 68 46 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CTSK 50 46 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CTSL 62 46 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne NPFFR2 60 31 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CTRB1 27 48 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CAPNS1 75 44 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne MMP2 27 48 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne MMP3 55 46 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne HLA-DRB1 57 34 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne LNPEP 17 41 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne MMP11 54 34 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CTSS 35 46 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CAPN1 117 49 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CASP1 38 43 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CAPN2 157 46 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne ACE2 73 39 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CASP6 32 43 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne CASP9 43 43 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne LAP3 46 41 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne ST14 43 34 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne MMP1 35 48 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne FPR1 70 38 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne NPR 99 43 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne AMP1_PLAFQ 33 41 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne PSMB5 70 48 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne POLG_WNV 40 35 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne BIRC2 36 42 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne NPFFR1 65 32 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne Q6PRC7_IXORI 40 31 C[C@H](N)C(=O)N[C@H](CCC(=O)OCc1ccccc1)C(=O)OCc1ccccc1 ZINC000147075247 GE For-Sale Anodyne TMPRSS6 51 34 O=Cc1ccc(-c2ccc(O[C@@H]3CC[C@@H](C(=O)O)CC3)nc2)cc1F ZINC000147075296 EH For-Sale Anodyne DGAT1 72 61 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCOCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147075304 HE On-Demand Bother LPL 46 41 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCOCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147075304 HE On-Demand Bother CPT1A 32 40 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCOCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147075304 HE On-Demand Bother EPHX2 18 48 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCOCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147075304 HE On-Demand Bother TGM2 56 37 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCOCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147075304 HE On-Demand Bother F13A1 81 41 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCOCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147075304 HE On-Demand Bother MERTK 30 43 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCOCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147075304 HE On-Demand Bother LIPG 19 41 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCOCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147075304 HE On-Demand Bother NAMPT 29 49 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cc(C)on3)cc2)cc1 ZINC000147075342 GG On-Demand Anodyne CA2 15 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cc(C)on3)cc2)cc1 ZINC000147075342 GG On-Demand Anodyne PPIA 23 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cc(C)on3)cc2)cc1 ZINC000147075342 GG On-Demand Anodyne MMP13 25 40 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cc(C)on3)cc2)cc1 ZINC000147075342 GG On-Demand Anodyne MMP2 18 40 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cc(C)on3)cc2)cc1 ZINC000147075342 GG On-Demand Anodyne CA9 18 40 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3cc(C)on3)cc2)cc1 ZINC000147075342 GG On-Demand Anodyne IDO1 35 45 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(-c2nc3ccccc3s2)o1 ZINC000147075378 GG On-Demand Anodyne PCSK5 40 30 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(-c2nc3ccccc3s2)o1 ZINC000147075378 GG On-Demand Anodyne FURIN 51 32 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(-c2nc3ccccc3s2)o1 ZINC000147075378 GG On-Demand Anodyne ST14 54 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(-c2nc3ccccc3s2)o1 ZINC000147075378 GG On-Demand Anodyne TMPRSS6 84 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(N)=O)ccc2F)c1 ZINC000147075425 EE On-Demand Bother KCNMA1 40 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(N)=O)ccc2F)c1 ZINC000147075425 EE On-Demand Bother TAAR1 28 53 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(N)=O)ccc2F)c1 ZINC000147075425 EE On-Demand Bother AKR1C3 20 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(N)=O)ccc2F)c1 ZINC000147075425 EE On-Demand Bother AKR1C2 44 40 CC(C)(C)C[C@H]1N[C@@H](C(=O)N[C@H]2CC[C@H](O)C2)[C@H](c2cccc(Cl)c2F)[C@@]12C(=O)Nc1cc(Cl)ccc12 ZINC000147075440 KJ Annotated Anodyne MDM2 66 60 NC(=O)c1ccc(OCC(=O)N2CC[C@H]2c2ccccc2)cc1 ZINC000147075533 DE On-Demand Anodyne CHEK2 43 38 NC(=O)c1ccc(OCC(=O)N2CC[C@H]2c2ccccc2)cc1 ZINC000147075533 DE On-Demand Anodyne COLA 167 57 NC(=O)c1ccc(OCC(=O)N2CC[C@H]2c2ccccc2)cc1 ZINC000147075533 DE On-Demand Anodyne CPT1A 139 57 NC(=O)c1ccc(OCC(=O)N2CC[C@H]2c2ccccc2)cc1 ZINC000147075533 DE On-Demand Anodyne CPT2 51 41 NC(=O)c1ccc(OCC(=O)N2CC[C@H]2c2ccccc2)cc1 ZINC000147075533 DE On-Demand Anodyne PLA2G4B 53 38 N#CC1CCN(C(=O)COc2ccc(N3CCCC3=O)cc2)CC1 ZINC000147075574 ED On-Demand Mild CPT1A 30 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(-c2nc3ccccc3s2)o1 ZINC000147075577 GG On-Demand Anodyne PCSK5 40 30 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(-c2nc3ccccc3s2)o1 ZINC000147075577 GG On-Demand Anodyne FURIN 51 32 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(-c2nc3ccccc3s2)o1 ZINC000147075577 GG On-Demand Anodyne ST14 54 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(-c2nc3ccccc3s2)o1 ZINC000147075577 GG On-Demand Anodyne TMPRSS6 84 41 CC(=O)CC(=O)OCc1ccc(C)cc1 ZINC000147075688 BE For-Sale Anodyne NAAA 38 43 C=C1CC[C@@H](OC(C)=O)[C@]2(C)CC[C@@H](C(C)C)[C@H](OC(C)=O)[C@@H]12 ZINC000147075704 DH Annotated Mild TAS2R31 0 41 NC(=O)c1ccc(OCC(=O)N2CC[C@@H]2c2ccccc2)cc1 ZINC000147075720 DE On-Demand Anodyne CHEK2 43 38 NC(=O)c1ccc(OCC(=O)N2CC[C@@H]2c2ccccc2)cc1 ZINC000147075720 DE On-Demand Anodyne CPT1A 139 57 NC(=O)c1ccc(OCC(=O)N2CC[C@@H]2c2ccccc2)cc1 ZINC000147075720 DE On-Demand Anodyne CPT2 51 41 NC(=O)c1ccc(OCC(=O)N2CC[C@@H]2c2ccccc2)cc1 ZINC000147075720 DE On-Demand Anodyne PLA2G4B 53 38 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075807 EF On-Demand Anodyne ANPEP 20 46 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075807 EF On-Demand Anodyne CTSK 19 40 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075807 EF On-Demand Anodyne MTNR1A 41 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075807 EF On-Demand Anodyne MTNR1B 31 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075807 EF On-Demand Anodyne GRIA1 57 35 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075807 EF On-Demand Anodyne PCSK5 60 40 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075807 EF On-Demand Anodyne FURIN 67 40 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075807 EF On-Demand Anodyne POLG_WNV 74 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075807 EF On-Demand Anodyne PROKR1 43 30 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCC(=O)N(C)C)c1)C2 ZINC000147075838 GE On-Demand Anodyne MTNR1A 28 44 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCC(=O)N(C)C)c1)C2 ZINC000147075838 GE On-Demand Anodyne MTNR1B 28 44 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCC(=O)N(C)C)c1)C2 ZINC000147075838 GE On-Demand Anodyne ROCK2 42 48 C[C@@H](CNC(=O)c1ccc(OCc2ccncc2)cc1)N1CCCC1 ZINC000147075875 EF On-Demand Anodyne ADAM17 29 45 C[C@@H](CNC(=O)c1ccc(OCc2ccncc2)cc1)N1CCCC1 ZINC000147075875 EF On-Demand Anodyne SLC6A5 40 39 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075979 EF On-Demand Anodyne ANPEP 20 46 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075979 EF On-Demand Anodyne CTSK 19 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075979 EF On-Demand Anodyne MTNR1A 41 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075979 EF On-Demand Anodyne MTNR1B 31 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075979 EF On-Demand Anodyne GRIA1 57 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075979 EF On-Demand Anodyne PCSK5 60 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075979 EF On-Demand Anodyne FURIN 67 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075979 EF On-Demand Anodyne POLG_WNV 74 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc2cc(OC)ccc2c1 ZINC000147075979 EF On-Demand Anodyne PROKR1 43 30 C[C@H](CNC(=O)c1ccc(OCc2ccncc2)cc1)N1CCCC1 ZINC000147076070 EF On-Demand Anodyne ADAM17 29 45 C[C@H](CNC(=O)c1ccc(OCc2ccncc2)cc1)N1CCCC1 ZINC000147076070 EF On-Demand Anodyne SLC6A5 40 39 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1OCCC(N)=O)C2 ZINC000147076077 FE On-Demand Anodyne ROCK2 45 51 O=Cc1ccc(-c2cnc3[nH]cc(NC(=O)c4cnn(Cc5ccccc5)c4)c3c2)cc1 ZINC000147076088 HJ For-Sale Anodyne ITK 15 40 O=Cc1ccc(-c2cnc3[nH]cc(NC(=O)c4cnn(Cc5ccccc5)c4)c3c2)cc1 ZINC000147076088 HJ For-Sale Anodyne SGK1 37 44 O=Cc1ccc(-c2cnc3[nH]cc(NC(=O)c4cnn(Cc5ccccc5)c4)c3c2)cc1 ZINC000147076088 HJ For-Sale Anodyne CDC7 18 42 O=Cc1ccc(-c2cnc3[nH]cc(NC(=O)c4cnn(Cc5ccccc5)c4)c3c2)cc1 ZINC000147076088 HJ For-Sale Anodyne ALK 19 52 O=Cc1ccc(-c2cnc3[nH]cc(NC(=O)c4cnn(Cc5ccccc5)c4)c3c2)cc1 ZINC000147076088 HJ For-Sale Anodyne RIPK1 41 38 Cc1cc(C(=O)Nc2ccc(Cl)cc2Cl)cc([N+](=O)[O-])c1 ZINC000147076117 EI On-Demand Bother CNR1 26 41 Cc1cc(C(=O)Nc2ccc(Cl)cc2Cl)cc([N+](=O)[O-])c1 ZINC000147076117 EI On-Demand Bother CNR2 17 41 Cc1cc(C(=O)Nc2ccc(Cl)cc2Cl)cc([N+](=O)[O-])c1 ZINC000147076117 EI On-Demand Bother PYGL 19 40 Cc1cc(C(=O)Nc2ccc(Cl)cc2Cl)cc([N+](=O)[O-])c1 ZINC000147076117 EI On-Demand Bother KCNMA1 42 45 CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)N2CCC(C#N)CC2)C1 ZINC000147076214 DE On-Demand Mild PREP 22 50 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ncc(Cc3ccc(C)c(C)c3)s2)c1 ZINC000147076264 GJ On-Demand Bother SCD1 42 45 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ncc(Cc3ccc(C)c(C)c3)s2)c1 ZINC000147076264 GJ On-Demand Bother SCD 38 47 CCCCCCC[C@H](CCCCCCCCO)OC(=O)/C=C/c1ccc(O)c(O)c1 ZINC000147076318 HK Annotated Mild MMP12 0 48 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCOCC3)c2)cc([N+](=O)[O-])c1 ZINC000147076337 HE On-Demand Bother LPL 38 41 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCOCC3)c2)cc([N+](=O)[O-])c1 ZINC000147076337 HE On-Demand Bother EPHX2 15 50 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCOCC3)c2)cc([N+](=O)[O-])c1 ZINC000147076337 HE On-Demand Bother TAAR1 26 44 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCOCC3)c2)cc([N+](=O)[O-])c1 ZINC000147076337 HE On-Demand Bother AKR1C3 49 39 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCOCC3)c2)cc([N+](=O)[O-])c1 ZINC000147076337 HE On-Demand Bother LIPG 17 41 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCOCC3)c2)cc([N+](=O)[O-])c1 ZINC000147076337 HE On-Demand Bother NAMPT 18 41 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCOCC3)c2)cc([N+](=O)[O-])c1 ZINC000147076337 HE On-Demand Bother KCNK3 75 38 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCOCC3)c2)cc([N+](=O)[O-])c1 ZINC000147076337 HE On-Demand Bother KCNK9 43 38 CCOC[C@H](C)NS(=O)(=O)c1ccc(F)c(C(F)(F)F)c1 ZINC000147076413 EF On-Demand Anodyne LEF 59 41 NC(=O)c1ccc(OCC(=O)N2CCC(c3ccccc3)CC2)cc1 ZINC000147076430 EF On-Demand Anodyne CHEK2 49 41 NC(=O)c1ccc(OCC(=O)N2CCC(c3ccccc3)CC2)cc1 ZINC000147076430 EF On-Demand Anodyne CPT1A 109 47 NC(=O)c1ccc(OCC(=O)N2CCC(c3ccccc3)CC2)cc1 ZINC000147076430 EF On-Demand Anodyne CPT2 48 38 NC(=O)c1ccc(OCC(=O)N2CCC(c3ccccc3)CC2)cc1 ZINC000147076430 EF On-Demand Anodyne SLC18A3 52 35 NC(=O)c1ccc(OCC(=O)N2CCC(c3ccccc3)CC2)cc1 ZINC000147076430 EF On-Demand Anodyne PLA2G4B 40 35 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147076462 HJ On-Demand Anodyne KIT 15 44 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147076462 HJ On-Demand Anodyne MAPK14 46 41 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147076462 HJ On-Demand Anodyne CPT1A 52 30 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147076462 HJ On-Demand Anodyne PRNP 45 36 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147076462 HJ On-Demand Anodyne MAPK10 18 41 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147076462 HJ On-Demand Anodyne TAAR1 26 40 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147076462 HJ On-Demand Anodyne KCNK3 89 44 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147076462 HJ On-Demand Anodyne KCNK9 47 42 CCc1ncc(C(=O)Nc2cccc(S(=O)(=O)N3CCOCC3)c2)s1 ZINC000147076548 GD On-Demand Anodyne AXL 16 44 CCc1ncc(C(=O)Nc2cccc(S(=O)(=O)N3CCOCC3)c2)s1 ZINC000147076548 GD On-Demand Anodyne MERTK 27 44 Brc1ccc(OCCn2ccnn2)cc1 ZINC000147076564 CE On-Demand Anodyne LTA4H 17 45 O=C(Nc1cccc(COc2cccc(F)c2)c1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147076628 GG On-Demand Anodyne F10 15 43 O=C([C@@H]1C[C@H]1c1cccc(Cl)c1)N1CCO[C@H]2CCCC[C@@H]21 ZINC000147076719 DH On-Demand Anodyne MDM2 49 32 COCc1nc(C(=O)N2CCN(c3ccccc3F)CC2)cs1 ZINC000147076783 EE On-Demand Anodyne TRPC6 57 35 CCc1nnc(NC(=O)c2ccccc2C(=O)OC)s1 ZINC000147076825 CE For-Sale Anodyne GLS 0 43 CCc1nnc(NC(=O)c2ccccc2C(=O)OC)s1 ZINC000147076825 CE For-Sale Anodyne KCNK3 40 34 COc1cccc(C(=O)NC2(C)CCCCC2)c1 ZINC000147076829 BG On-Demand Anodyne DRD4 58 44 COc1cccc(C(=O)NC2(C)CCCCC2)c1 ZINC000147076829 BG On-Demand Anodyne ECR 16 45 COc1cccc(C(=O)NC2(C)CCCCC2)c1 ZINC000147076829 BG On-Demand Anodyne MTNR1B 31 41 COc1cccc(C(=O)NC2(C)CCCCC2)c1 ZINC000147076829 BG On-Demand Anodyne CASP1 0 48 COc1cccc(C(=O)NC2(C)CCCCC2)c1 ZINC000147076829 BG On-Demand Anodyne KCNK3 29 51 COc1cccc(C(=O)NC2(C)CCCCC2)c1 ZINC000147076829 BG On-Demand Anodyne BRPF1 0 48 O=C(Nc1cccc(COc2cccc(F)c2)c1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147076833 GG On-Demand Anodyne F10 15 43 COc1ccc(-c2nc(C(=O)N3CCC(C#N)CC3)cs2)cc1 ZINC000147076857 EG On-Demand Mild TRPC6 67 52 COc1ccc(-c2nc(C(=O)N3CCC(C#N)CC3)cs2)cc1 ZINC000147076857 EG On-Demand Mild TRPC3 39 52 O=C([C@@H]1C[C@@H]1c1cccc(Cl)c1)N1CCO[C@H]2CCCC[C@@H]21 ZINC000147076924 DH On-Demand Anodyne MDM2 49 32 CCCC(=O)N1CCN(c2ccc(C(N)=O)cc2)CC1 ZINC000147076932 CD On-Demand Anodyne PRNP 40 39 O=C(Nc1cccc(COc2cccc(F)c2)c1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147077012 GG On-Demand Anodyne F10 15 43 O=C(Nc1cccc(COc2cccc(F)c2)c1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147077170 GG On-Demand Anodyne F10 15 43 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(=O)c2ccc(F)cc2)cc1 ZINC000147077200 GF On-Demand Anodyne CA2 19 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(=O)c2ccc(F)cc2)cc1 ZINC000147077200 GF On-Demand Anodyne CA1 15 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(=O)c2ccc(F)cc2)cc1 ZINC000147077200 GF On-Demand Anodyne MMP13 33 43 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(=O)c2ccc(F)cc2)cc1 ZINC000147077200 GF On-Demand Anodyne CXCR2 15 50 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(=O)c2ccc(F)cc2)cc1 ZINC000147077200 GF On-Demand Anodyne MMP2 25 50 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(=O)c2ccc(F)cc2)cc1 ZINC000147077200 GF On-Demand Anodyne MMP8 17 43 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(=O)c2ccc(F)cc2)cc1 ZINC000147077200 GF On-Demand Anodyne CA9 15 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(=O)c2ccc(F)cc2)cc1 ZINC000147077200 GF On-Demand Anodyne LEF 18 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(=O)c2ccc(F)cc2)cc1 ZINC000147077200 GF On-Demand Anodyne IDO1 31 43 CC(C)(C)OC(=O)N1CCN(c2ccc(N3C[C@@H](CO)OC3=O)cc2F)CC1 ZINC000147077214 GE For-Sale Anodyne GPR119 50 41 C[C@@H]1CN(c2ccc(Nc3ncc4c5ccncc5n(C5CCCC5)c4n3)nn2)CCN1 ZINC000147077344 IG Annotated Anodyne FLT3 26 75 Cc1ccc2[nH]c(C(=O)NC[C@@H](C)N3CCCC3)cc2c1 ZINC000147077441 CF On-Demand Anodyne AKR1C3 36 47 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1c(C)n(C)n(-c2ccccc2)c1=O ZINC000147077448 HF On-Demand Mild FPR2 39 42 C[C@H]1CN(c2ccc(Nc3ncc4c5ccncc5n(C5CCCC5)c4n3)nn2)CCN1 ZINC000147077544 IG Annotated Anodyne FLT3 26 75 NC(=O)C1CCN(Cc2cccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)c2)CC1 ZINC000147077568 HD On-Demand Anodyne MCHR1 20 40 CCOC[C@H](C)NS(=O)(=O)c1cccc2cnccc12 ZINC000147077594 CD On-Demand Anodyne P2RX7 31 44 Cc1ccc2[nH]c(C(=O)NC[C@H](C)N3CCCC3)cc2c1 ZINC000147077597 CF On-Demand Anodyne CCKAR 19 42 Cc1ccc2[nH]c(C(=O)NC[C@H](C)N3CCCC3)cc2c1 ZINC000147077597 CF On-Demand Anodyne AKR1C3 36 47 COc1ccc(C#N)cc1N[C@@H](C)C(=O)Nc1ccc(Cl)cn1 ZINC000147077650 EG On-Demand Mild F10 52 34 COc1ccc(C#N)cc1N[C@@H](C)C(=O)Nc1ccc(Cl)cn1 ZINC000147077650 EG On-Demand Mild CHEK1 15 42 N#CC1CCN(C(=O)COc2cccc(N3CCCC3=O)c2)CC1 ZINC000147077678 ED On-Demand Mild COLA 69 47 N#CC1CCN(C(=O)COc2cccc(N3CCCC3=O)c2)CC1 ZINC000147077678 ED On-Demand Mild CPT1A 63 47 CC(C)c1nc(CN(C)C(=O)N[C@H](C(=O)N[C@H](Cc2ccccc2)C[C@@H](O)[C@@H](N)Cc2ccccc2)C(C)C)cs1 ZINC000147077715 KI For-Sale Anodyne HLA-DRB1 40 33 CC(C)c1nc(CN(C)C(=O)N[C@H](C(=O)N[C@H](Cc2ccccc2)C[C@@H](O)[C@@H](N)Cc2ccccc2)C(C)C)cs1 ZINC000147077715 KI For-Sale Anodyne CYP3A5 21 71 CC(C)c1nc(CN(C)C(=O)N[C@H](C(=O)N[C@H](Cc2ccccc2)C[C@@H](O)[C@@H](N)Cc2ccccc2)C(C)C)cs1 ZINC000147077715 KI For-Sale Anodyne CYP3A4 38 65 CC(C)c1nc(CN(C)C(=O)N[C@H](C(=O)N[C@H](Cc2ccccc2)C[C@@H](O)[C@@H](N)Cc2ccccc2)C(C)C)cs1 ZINC000147077715 KI For-Sale Anodyne PLM1_PLAFA 40 30 CC(C)c1nc(CN(C)C(=O)N[C@H](C(=O)N[C@H](Cc2ccccc2)C[C@@H](O)[C@@H](N)Cc2ccccc2)C(C)C)cs1 ZINC000147077715 KI For-Sale Anodyne SLC47A1 19 71 NC(=O)C1CCN(Cc2cccc(NC(=O)C(=O)NC[C@H]3CCCCO3)c2)CC1 ZINC000147077767 HD On-Demand Anodyne MCHR1 20 40 C[C@@H](CNC(=O)c1cc2cc(Br)ccc2[nH]1)N1CCCC1 ZINC000147077796 FG On-Demand Anodyne PYGL 87 45 C[C@@H](CNC(=O)c1cc2cc(Br)ccc2[nH]1)N1CCCC1 ZINC000147077796 FG On-Demand Anodyne PLD1 29 40 C[C@@H](CNC(=O)c1cc2cc(Br)ccc2[nH]1)N1CCCC1 ZINC000147077796 FG On-Demand Anodyne PYGM 25 43 C[C@@H](CNC(=O)c1cc2cc(Br)ccc2[nH]1)N1CCCC1 ZINC000147077796 FG On-Demand Anodyne PLD2 36 40 C[C@@H](CNC(=O)c1cc2cc(Br)ccc2[nH]1)N1CCCC1 ZINC000147077796 FG On-Demand Anodyne PYK 61 44 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild HDAC8 69 56 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild HDAC10 28 42 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild F3 25 42 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild MMP2 15 47 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild HDAC1 70 50 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild HDAC2 34 64 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild HDAC3 30 43 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild HDAC5 46 41 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild HDAC6 47 64 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild MMP9 15 47 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild HDAC9 43 41 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild HDAC11 32 41 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild HDAC7 48 41 Nc1ccc(/C=C\C(=O)NO)cc1 ZINC000147077800 AC For-Sale Mild BOTA 31 43 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)N(CC)CC)cc1 ZINC000147077809 ED On-Demand Anodyne MMP7 16 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)N(CC)CC)cc1 ZINC000147077809 ED On-Demand Anodyne LIMK2 42 38 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(Cl)cn1 ZINC000147077861 EG On-Demand Mild F10 52 34 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(Cl)cn1 ZINC000147077861 EG On-Demand Mild CHEK1 15 42 N#CC1CCN(C(=O)c2ccccc2COc2ccccc2)CC1 ZINC000147077883 DH On-Demand Mild GRIN2B 41 41 COCCOc1ccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cn1 ZINC000147077893 HD On-Demand Bother MAPK8 28 40 COCCOc1ccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cn1 ZINC000147077893 HD On-Demand Bother NAMPT 44 39 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDAC8 69 56 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDAC10 28 42 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild F3 25 42 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild MMP2 15 47 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDAC1 91 50 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDAC2 44 50 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDAC3 30 43 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDAC4 47 46 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDAC5 46 41 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDAC6 47 64 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild MMP9 15 47 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDAC9 43 41 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDAC11 32 41 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDAC7 48 41 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild MMP1 0 47 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HDA106 0 42 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild HD1B 0 40 Nc1ccc(/C=C/C(=O)NO)cc1 ZINC000147077980 AC For-Sale Mild BOTA 31 43 C[C@H](CNC(=O)c1cc2cc(Br)ccc2[nH]1)N1CCCC1 ZINC000147078002 FG On-Demand Anodyne PYGL 87 45 C[C@H](CNC(=O)c1cc2cc(Br)ccc2[nH]1)N1CCCC1 ZINC000147078002 FG On-Demand Anodyne PLD1 29 40 C[C@H](CNC(=O)c1cc2cc(Br)ccc2[nH]1)N1CCCC1 ZINC000147078002 FG On-Demand Anodyne PYGM 25 43 C[C@H](CNC(=O)c1cc2cc(Br)ccc2[nH]1)N1CCCC1 ZINC000147078002 FG On-Demand Anodyne PLD2 36 40 C[C@H](CNC(=O)c1cc2cc(Br)ccc2[nH]1)N1CCCC1 ZINC000147078002 FG On-Demand Anodyne PYK 61 44 Cc1cc(Nc2cc(C3CNC3)nc(-c3ccccc3Cl)n2)n[nH]1 ZINC000147078413 EG In-Stock Anodyne AURKA 25 40 Cc1cc(Nc2cc(C3CNC3)nc(-c3ccccc3Cl)n2)n[nH]1 ZINC000147078413 EG In-Stock Anodyne PKNB 58 36 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCc1ccc(Cl)cc1 ZINC000147078452 EG On-Demand Mild AMP1_PLAFQ 15 41 Cc1ccc(I)c(S(N)(=O)=O)c1 ZINC000147078458 CD For-Sale Anodyne CA2 17 45 Cc1ccc(I)c(S(N)(=O)=O)c1 ZINC000147078458 CD For-Sale Anodyne CA12 15 45 Cc1ccc(I)c(S(N)(=O)=O)c1 ZINC000147078458 CD For-Sale Anodyne CA9 17 45 Cc1ccc(I)c(S(N)(=O)=O)c1 ZINC000147078458 CD For-Sale Anodyne CYNT 34 45 Cc1ccc(I)c(S(N)(=O)=O)c1 ZINC000147078458 CD For-Sale Anodyne CA 0 45 Cc1ccc(I)c(S(N)(=O)=O)c1 ZINC000147078458 CD For-Sale Anodyne A6YCJ1_9METZ 16 45 COc1ccc(C(=O)c2nccs2)c(OC)c1 ZINC000147078754 BE For-Sale Anodyne LUCI_LUCLA 16 45 CS(=O)(=O)Nc1cnc(C(=O)O)cn1 ZINC000147078800 BB For-Sale Anodyne P4HTM 0 49 O=C(Nc1cnc2ccccc2c1)c1ccc2nc3n(c2c1)CCCNC3=O ZINC000147078846 FF Annotated Anodyne MAPKAPK2 18 53 O=C(Nc1cnc2ccccc2c1)c1ccc2nc3n(c2c1)CCCNC3=O ZINC000147078846 FF Annotated Anodyne RPS6KA3 99 76 CCOC[C@H](C)NS(=O)(=O)c1c(Cl)cccc1[N+](=O)[O-] ZINC000147078866 DD On-Demand Bother COLA 68 32 COc1ccc(NC(=O)[C@H](C)Nc2cc(C#N)ccc2OC)c([N+](=O)[O-])c1 ZINC000147078871 FF On-Demand Mild TAAR1 16 41 C[C@@H]1CC[C@]2(C(=O)O)CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)C[C@@H](O)[C@H](O)[C@](C)(C(=O)O)[C@@H]5CC[C@]43C)[C@@H]2[C@]1(C)O ZINC000147078885 KI Annotated Anodyne PTPN2 41 42 C[C@@H]1CC[C@]2(C(=O)O)CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)C[C@@H](O)[C@H](O)[C@](C)(C(=O)O)[C@@H]5CC[C@]43C)[C@@H]2[C@]1(C)O ZINC000147078885 KI Annotated Anodyne PTPN1 30 42 Nc1cccc(C(=O)O)c1N1CCCCC1 ZINC000147078893 BD For-Sale Anodyne FABP4 46 37 CCCOCC(=O)Nc1ccc2nc(N3CCCC3)sc2c1 ZINC000147079004 DG On-Demand Anodyne LDHA 40 36 N#CCc1ccc(N2CCCCC2)c(Cl)c1 ZINC000147079499 BG For-Sale Anodyne CSF1R 15 42 N#CCc1ccc(N2CCCCC2)c(Cl)c1 ZINC000147079499 BG For-Sale Anodyne PAK1 43 36 O=C(NCc1ccccn1)c1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147079573 HH On-Demand Anodyne GRM4 49 38 O=C(NCc1ccccn1)c1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147079573 HH On-Demand Anodyne KCNK3 53 42 CCOc1ccc2nc(NC(=O)c3csc(COC)n3)sc2c1 ZINC000147079613 EH On-Demand Anodyne CSNK1D 49 54 CCOc1ccc2nc(NC(=O)c3csc(COC)n3)sc2c1 ZINC000147079613 EH On-Demand Anodyne PIK3CA 20 41 CCOc1ccc2nc(NC(=O)c3csc(COC)n3)sc2c1 ZINC000147079613 EH On-Demand Anodyne GHSR 17 43 NC(=O)c1ccc(OCC(=O)NC2CCN(c3ncccn3)CC2)cc1 ZINC000147079640 FC On-Demand Anodyne CPT1A 18 41 NC(=O)c1ccc(OCC(=O)NC2CCN(c3ncccn3)CC2)cc1 ZINC000147079640 FC On-Demand Anodyne MCHR1 19 43 COc1ccc(C#N)cc1N[C@@H](C)C(=O)Nc1cccc(S(N)(=O)=O)c1 ZINC000147079655 FD On-Demand Mild CA2 19 46 COc1ccc(C#N)cc1N[C@@H](C)C(=O)Nc1cccc(S(N)(=O)=O)c1 ZINC000147079655 FD On-Demand Mild CA1 19 41 COc1ccc(C#N)cc1N[C@@H](C)C(=O)Nc1cccc(S(N)(=O)=O)c1 ZINC000147079655 FD On-Demand Mild CA4 21 46 O=C(NCCOc1ccc2c(c1)[C@H](C1(c3ccc(Cl)cc3)CCC1)NCC2)Nc1ccccc1 ZINC000147079689 JK Annotated Anodyne ADRB1 15 40 O=C(NCCOc1ccc2c(c1)[C@H](C1(c3ccc(Cl)cc3)CCC1)NCC2)Nc1ccccc1 ZINC000147079689 JK Annotated Anodyne HRH2 24 43 Cc1cc(C(=O)N2CCC(Cc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147079843 EH On-Demand Bother CHRM2 17 41 Cc1cc(C(=O)N2CCC(Cc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147079843 EH On-Demand Bother ACHE 17 43 Cc1cc(C(=O)N2CCC(Cc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147079843 EH On-Demand Bother GRIN2B 89 52 Cc1cc(C(=O)N2CCC(Cc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147079843 EH On-Demand Bother TACR1 15 44 Cc1cc(C(=O)N2CCC(Cc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147079843 EH On-Demand Bother SIGMAR1 15 45 Cc1cc(C(=O)N2CCC(Cc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147079843 EH On-Demand Bother CCR3 48 39 Cc1cc(C(=O)N2CCC(Cc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147079843 EH On-Demand Bother L3MBTL3 46 37 CCCNC(=O)c1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147079862 FD On-Demand Anodyne DRD4 41 31 CCCNC(=O)c1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147079862 FD On-Demand Anodyne ADORA2B 43 43 CCCNC(=O)c1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147079862 FD On-Demand Anodyne PLA2G4B 51 36 CCCNC(=O)c1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147079862 FD On-Demand Anodyne PLAU 18 43 CCCNC(=O)c1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147079862 FD On-Demand Anodyne ACR 40 36 CCCNC(=O)c1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147079862 FD On-Demand Anodyne HIF1A 22 47 CCCNC(=O)c1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147079862 FD On-Demand Anodyne KCNK3 89 37 CCCNC(=O)c1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147079862 FD On-Demand Anodyne KCNK9 55 36 O=C(NCCOc1ccc2c(c1)[C@@H](C1(c3ccc(Cl)cc3)CCC1)NCC2)Nc1ccccc1 ZINC000147079912 JK Annotated Anodyne ADRB1 15 40 O=C(NCCOc1ccc2c(c1)[C@@H](C1(c3ccc(Cl)cc3)CCC1)NCC2)Nc1ccccc1 ZINC000147079912 JK Annotated Anodyne HRH2 24 43 N#CCCCOc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147079914 ED On-Demand Mild EPHX2 17 42 CC(=O)N[C@H]1CC[C@@H](N(C)c2cc(-c3ccc(CN4CCOCC4)cc3)cc(C(=O)NCc3c(C)cc(C)[nH]c3=O)c2C)CC1 ZINC000147080024 KJ Annotated Anodyne EZH2 47 73 N#CCCCOc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147080112 ED On-Demand Mild EPHX2 17 42 CN1CCN(C(=O)C2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)CC1 ZINC000147080129 GC On-Demand Anodyne HTR1D 15 43 CN1CCN(C(=O)C2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)CC1 ZINC000147080129 GC On-Demand Anodyne HTR1B 19 43 CN1CCN(C(=O)C2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)CC1 ZINC000147080129 GC On-Demand Anodyne HRH3 15 44 CN1CCN(C(=O)C2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)CC1 ZINC000147080129 GC On-Demand Anodyne CPT1A 73 49 CN1CCN(C(=O)C2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)CC1 ZINC000147080129 GC On-Demand Anodyne CPT2 44 37 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147080240 HD On-Demand Mild CA2 74 51 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147080240 HD On-Demand Mild CA1 66 51 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147080240 HD On-Demand Mild CA7 40 51 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147080240 HD On-Demand Mild CA5B 22 40 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147080240 HD On-Demand Mild CA4 45 46 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147080240 HD On-Demand Mild CA5A 24 40 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147080240 HD On-Demand Mild CA14 44 51 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147080240 HD On-Demand Mild CA12 54 47 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147080240 HD On-Demand Mild CA9 56 51 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147080240 HD On-Demand Mild CYNT 18 41 COc1ccc(C#N)cc1N[C@@H](C)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147080240 HD On-Demand Mild A6YCJ1_9METZ 15 42 CC(C)(C)C[C@H]1N[C@@H](C(=O)NC2CC(O)C2)[C@H](c2cccc(Cl)c2F)[C@@]12C(=O)Nc1cc(Cl)ccc12 ZINC000147080243 KJ Annotated Anodyne MDM2 67 59 CC(C)CCO[C@@H](C)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147080259 EG On-Demand Anodyne CCKAR 20 47 CCNC(=O)N[C@H](C(=O)N1CCCC1)C(C)C ZINC000147080281 BC On-Demand Anodyne RIR1_HHV11 56 40 CCNC(=O)N[C@H](C(=O)N1CCCC1)C(C)C ZINC000147080281 BC On-Demand Anodyne CCR1 48 39 Nc1ccc(/N=N/S(=O)(=O)O)cc1 ZINC000147080304 BD For-Sale Clean NT5E 0 46 COCCOc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147080342 ED On-Demand Anodyne EPHX2 18 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC)nc1 ZINC000147080347 CC On-Demand Anodyne ACACA 21 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC)nc1 ZINC000147080347 CC On-Demand Anodyne NPY1R 24 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC)nc1 ZINC000147080347 CC On-Demand Anodyne GRIA1 45 33 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC)nc1 ZINC000147080347 CC On-Demand Anodyne PCSK5 60 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC)nc1 ZINC000147080347 CC On-Demand Anodyne FURIN 66 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC)nc1 ZINC000147080347 CC On-Demand Anodyne POLG_WNV 70 34 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC)nc1 ZINC000147080347 CC On-Demand Anodyne NPFFR1 52 39 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC)nc1 ZINC000147080347 CC On-Demand Anodyne HPN 40 31 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(NS(C)(=O)=O)cc2)c1 ZINC000147080383 GD On-Demand Bother TRPV1 33 45 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(NS(C)(=O)=O)cc2)c1 ZINC000147080383 GD On-Demand Bother CA9 18 42 Cc1cc(C)c(CNC(=O)c2cc(-c3cnn(CCN4CCOCC4)c3)cc(N(C)C3CCNCC3)c2C)c(=O)[nH]1 ZINC000147080396 KF Annotated Anodyne EZH2 45 58 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccccc2)cc1 ZINC000147080430 DG On-Demand Anodyne MMP13 17 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccccc2)cc1 ZINC000147080430 DG On-Demand Anodyne MMP14 33 43 CC(C)CCO[C@H](C)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147080450 EG On-Demand Anodyne P2RY12 51 34 CC(C)CCO[C@H](C)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147080450 EG On-Demand Anodyne CCKAR 20 47 COCCOc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147080549 ED On-Demand Anodyne EPHX2 18 42 CS(=O)(=O)Nc1ccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)cc1 ZINC000147080574 GE On-Demand Anodyne TRPV1 21 43 O=C(Nc1cccc(OCCn2cncn2)c1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147080592 GH On-Demand Anodyne NAMPT 24 42 C=Cc1ccc(/C=N/NC(N)=S)cc1 ZINC000147080599 BD For-Sale Mild UREA_CANEN 51 63 C=Cc1ccc(/C=N/NC(N)=S)cc1 ZINC000147080599 BD For-Sale Mild PPO2 37 41 CC(=O)N[C@H]1CC[C@@H](N(C)c2cc(-c3cnn(CCN4CCOCC4)c3)cc(C(=O)NCc3c(C)cc(C)[nH]c3=O)c2C)CC1 ZINC000147080639 KG Annotated Anodyne EZH2 42 56 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147080646 FE On-Demand Anodyne CCKAR 17 45 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147080646 FE On-Demand Anodyne EPHX2 22 40 CCOc1ccc2nc(NC(=O)c3cnc(CC)s3)sc2c1 ZINC000147080704 EH On-Demand Anodyne CA2 18 46 CCOc1ccc2nc(NC(=O)c3cnc(CC)s3)sc2c1 ZINC000147080704 EH On-Demand Anodyne CSNK1D 49 57 CCOc1ccc2nc(NC(=O)c3cnc(CC)s3)sc2c1 ZINC000147080704 EH On-Demand Anodyne PIK3CA 21 45 CCOc1ccc2nc(NC(=O)c3cnc(CC)s3)sc2c1 ZINC000147080704 EH On-Demand Anodyne HSD17B1 28 40 CCOc1ccc2nc(NC(=O)c3cnc(CC)s3)sc2c1 ZINC000147080704 EH On-Demand Anodyne PIK3CG 18 55 O=C(Nc1cccc(OCCn2cncn2)c1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147080783 GH On-Demand Anodyne NAMPT 24 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(N2CCOCC2)nc1 ZINC000147080790 EC On-Demand Anodyne PCSK5 43 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(N2CCOCC2)nc1 ZINC000147080790 EC On-Demand Anodyne FURIN 47 35 C[C@@H](OC[C@@H]1CCCO1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147080834 FE On-Demand Anodyne CCKAR 17 45 C[C@@H](OC[C@@H]1CCCO1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147080834 FE On-Demand Anodyne EPHX2 22 40 COc1ccc(C#N)cc1N[C@@H](C)C(=O)Nc1ccc(OC)c(OC)c1 ZINC000147080839 FG On-Demand Mild ENPP1 58 33 CC(=O)N[C@H]1CC[C@@H](N(C)c2cc(-c3ccc(CN(C)C)cc3)cc(C(=O)NCc3c(C)cc(C)[nH]c3=O)c2C)CC1 ZINC000147080860 KJ Annotated Anodyne EZH2 41 54 Cc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1-n1cnnn1 ZINC000147080914 HH On-Demand Anodyne ROCK2 16 43 Cc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1-n1cnnn1 ZINC000147080914 HH On-Demand Anodyne MET 30 40 Cc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1-n1cnnn1 ZINC000147080914 HH On-Demand Anodyne NAMPT 40 41 COc1ccc(S(=O)(=O)N2CCOCC2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147080916 GD On-Demand Mild CASP3 17 42 COc1ccc(S(=O)(=O)N2CCOCC2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147080916 GD On-Demand Mild SLC6A9 45 44 O=C(Nc1cccc(OCCn2cncn2)c1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147080954 GH On-Demand Anodyne NAMPT 24 42 C[C@H](OC[C@H]1CCCO1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147081033 FE On-Demand Anodyne CCKAR 17 45 C[C@H](OC[C@H]1CCCO1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147081033 FE On-Demand Anodyne EPHX2 22 40 Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(CN(C)C)nc3)cc(N(C)C3CCNCC3)c2C)c(=O)[nH]1 ZINC000147081081 KH Annotated Anodyne EZH2 44 49 C/C=C/c1cncc2ccccc12 ZINC000147081089 AG For-Sale Anodyne CHAT 65 38 C/C=C/c1cncc2ccccc12 ZINC000147081089 AG For-Sale Anodyne CYP11B2 33 40 CN(CCc1ccccc1)C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147081169 DI On-Demand Anodyne GRM3 20 41 CN(CCc1ccccc1)C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147081169 DI On-Demand Anodyne MDM2 65 33 C[C@@H](OC[C@H]1CCCO1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147081197 FE On-Demand Anodyne CCKAR 17 45 C[C@@H](OC[C@H]1CCCO1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147081197 FE On-Demand Anodyne EPHX2 22 40 CS(=O)(=O)c1cc(C(=O)NCc2ccc(-n3cncn3)cc2)cc([N+](=O)[O-])c1 ZINC000147081254 HD On-Demand Bother NAMPT 51 34 Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(CN4CCOCC4)cc3)cc(N(C)[C@@H]3CC[C@H](N)CC3)c2C)c(=O)[nH]1 ZINC000147081312 KI Annotated Anodyne EZH2 49 76 CN(CCc1ccccc1)C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147081340 DI On-Demand Anodyne GRM3 20 41 CN(CCc1ccccc1)C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147081340 DI On-Demand Anodyne MDM2 65 33 CN(CCc1ccccc1)C(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147081460 DI On-Demand Anodyne GRM3 20 41 CN(CCc1ccccc1)C(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147081460 DI On-Demand Anodyne MDM2 65 33 O=C(COc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1)Nc1ccccc1 ZINC000147081510 HE On-Demand Anodyne CPT1A 66 39 O=C(COc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1)Nc1ccccc1 ZINC000147081510 HE On-Demand Anodyne EPHX2 16 41 CCc1ncc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147081564 GG On-Demand Anodyne LPL 43 36 CCc1ncc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147081564 GG On-Demand Anodyne GRM4 20 40 CCc1ncc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147081564 GG On-Demand Anodyne EPHX2 17 40 CCc1ncc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147081564 GG On-Demand Anodyne TGM2 40 32 CCc1ncc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147081564 GG On-Demand Anodyne F13A1 43 38 CCc1ncc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147081564 GG On-Demand Anodyne NAMPT 33 43 O=C(COc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1)Nc1ccccc1 ZINC000147081645 HE On-Demand Anodyne CPT1A 66 39 O=C(COc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1)Nc1ccccc1 ZINC000147081645 HE On-Demand Anodyne EPHX2 16 41 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)NC[C@@H](C)N1CCCC1 ZINC000147081664 GI On-Demand Anodyne TSPO 28 44 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)NC[C@@H](C)N1CCCC1 ZINC000147081664 GI On-Demand Anodyne TACR3 60 38 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)Nc3ccccc3)ccc2C)c1 ZINC000147081706 HI On-Demand Bother LCK 19 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)Nc3ccccc3)ccc2C)c1 ZINC000147081706 HI On-Demand Bother MAPK14 29 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)Nc3ccccc3)ccc2C)c1 ZINC000147081706 HI On-Demand Bother CPT1A 43 30 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)Nc3ccccc3)ccc2C)c1 ZINC000147081706 HI On-Demand Bother NR1H4 18 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)Nc3ccccc3)ccc2C)c1 ZINC000147081706 HI On-Demand Bother TAAR1 43 57 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)Nc3ccccc3)ccc2C)c1 ZINC000147081706 HI On-Demand Bother SIRT2 15 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)Nc3ccccc3)ccc2C)c1 ZINC000147081706 HI On-Demand Bother AKR1C3 37 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)Nc3ccccc3)ccc2C)c1 ZINC000147081706 HI On-Demand Bother DDR1 31 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)Nc3ccccc3)ccc2C)c1 ZINC000147081706 HI On-Demand Bother AKR1C2 66 45 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)Nc3ccccc3)ccc2C)c1 ZINC000147081706 HI On-Demand Bother KCNK3 96 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)Nc3ccccc3)ccc2C)c1 ZINC000147081706 HI On-Demand Bother KCNK9 57 39 COc1cc(OC)c2c(c1)O[C@H](c1ccc(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c(OC)c1)CC2=O ZINC000147081725 JC Annotated Anodyne IL2 28 43 COc1cc(OC)c2c(c1)O[C@H](c1ccc(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c(OC)c1)CC2=O ZINC000147081725 JC Annotated Anodyne SLC5A1 55 39 COc1cc(OC)c2c(c1)O[C@H](c1ccc(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c(OC)c1)CC2=O ZINC000147081725 JC Annotated Anodyne SLC5A2 44 41 COc1cc(OC)c2c(c1)O[C@H](c1ccc(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c(OC)c1)CC2=O ZINC000147081725 JC Annotated Anodyne FIMH 82 39 COc1cc(OC)c2c(c1)O[C@H](c1ccc(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c(OC)c1)CC2=O ZINC000147081725 JC Annotated Anodyne SLC5A4 19 41 COc1cc(OC)c2c(c1)O[C@H](c1ccc(O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c(OC)c1)CC2=O ZINC000147081725 JC Annotated Anodyne TAS2R31 0 48 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)cc([N+](=O)[O-])c1 ZINC000147081728 HG On-Demand Bother LPL 46 39 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)cc([N+](=O)[O-])c1 ZINC000147081728 HG On-Demand Bother CPT1A 48 36 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)cc([N+](=O)[O-])c1 ZINC000147081728 HG On-Demand Bother EPHX2 22 48 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)cc([N+](=O)[O-])c1 ZINC000147081728 HG On-Demand Bother F13A1 51 38 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)cc([N+](=O)[O-])c1 ZINC000147081728 HG On-Demand Bother TAAR1 46 43 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)cc([N+](=O)[O-])c1 ZINC000147081728 HG On-Demand Bother AKR1C3 59 41 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)cc([N+](=O)[O-])c1 ZINC000147081728 HG On-Demand Bother KCNK3 88 40 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)cc([N+](=O)[O-])c1 ZINC000147081728 HG On-Demand Bother KCNK9 45 40 O=C(Nc1ccc(OC[C@H]2CCCO2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147081792 GI On-Demand Anodyne TNK2 40 36 O=C(Nc1ccc(OC[C@H]2CCCO2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147081792 GI On-Demand Anodyne PANC 41 32 COc1ccc(C#N)cc1N[C@@H](C)C(=O)Nc1ccc([N+](=O)[O-])cc1C(F)(F)F ZINC000147081806 HH On-Demand Mild KCNMA1 19 42 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)NC[C@H](C)N1CCCC1 ZINC000147081851 GI On-Demand Anodyne TSPO 28 44 Cc1nc2ccccc2c(-c2ccccc2)c1CC(=O)NC[C@H](C)N1CCCC1 ZINC000147081851 GI On-Demand Anodyne TACR3 60 38 COc1cc(/C=C/C(O)=C/C(=O)C[C@H](O)c2ccc(O)c(OC)c2)ccc1O ZINC000147081863 GG Annotated Mild NA 0 63 COc1cc(/C=C/C(O)=C/C(=O)C[C@H](O)c2ccc(O)c(OC)c2)ccc1O ZINC000147081863 GG Annotated Mild PNLIP 0 45 COc1cc(/C=C/C(O)=C/C(=O)C[C@H](O)c2ccc(O)c(OC)c2)ccc1O ZINC000147081863 GG Annotated Mild FOLH1 24 40 COc1cc(/C=C/C(O)=C/C(=O)C[C@H](O)c2ccc(O)c(OC)c2)ccc1O ZINC000147081863 GG Annotated Mild APP 47 52 COc1cc(/C=C/C(O)=C/C(=O)C[C@H](O)c2ccc(O)c(OC)c2)ccc1O ZINC000147081863 GG Annotated Mild CAMK2A 15 41 COc1cc(/C=C/C(O)=C/C(=O)C[C@H](O)c2ccc(O)c(OC)c2)ccc1O ZINC000147081863 GG Annotated Mild PRKCQ 0 51 COc1cc(/C=C/C(O)=C/C(=O)C[C@H](O)c2ccc(O)c(OC)c2)ccc1O ZINC000147081863 GG Annotated Mild SLC22A3 0 45 COCc1nc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)cs1 ZINC000147081882 GF On-Demand Anodyne LPL 45 37 COCc1nc(C(=O)Nc2cccc(S(=O)(=O)N3CCCCC3)c2)cs1 ZINC000147081882 GF On-Demand Anodyne F13A1 46 41 CCNC(=O)COc1ccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1OC ZINC000147081910 HE On-Demand Bother MT-ND1 24 41 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1C ZINC000147081936 CD On-Demand Anodyne FFAR4 17 40 CCOc1cc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)ccc1OC ZINC000147082017 FG On-Demand Anodyne SSTR5 15 43 CCOc1cc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)ccc1OC ZINC000147082017 FG On-Demand Anodyne ROCK2 36 56 CCOc1cc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)ccc1OC ZINC000147082017 FG On-Demand Anodyne ENPP1 68 34 COCCOc1ccc(C(=O)Nc2ccc(F)c([C@]3(C)C=CSC(N)=N3)c2)nc1 ZINC000147082080 HG Annotated Anodyne BACE2 54 54 COCCOc1ccc(C(=O)Nc2ccc(F)c([C@]3(C)C=CSC(N)=N3)c2)nc1 ZINC000147082080 HG Annotated Anodyne BACE1 26 54 COc1ccc(C)cc1-n1ccc(C(=O)NCCCc2nc3ccccc3[nH]2)n1 ZINC000147082137 GG On-Demand Anodyne F9 33 44 COc1ccc(C)cc1-n1ccc(C(=O)NCCCc2nc3ccccc3[nH]2)n1 ZINC000147082137 GG On-Demand Anodyne CYSP_TRYCR 17 43 COc1ccc(C)cc1-n1ccc(C(=O)NCCCc2nc3ccccc3[nH]2)n1 ZINC000147082137 GG On-Demand Anodyne CACNA1G 29 40 COC(=O)c1ccnc(C(C)C)c1 ZINC000147082155 AD For-Sale Anodyne KDM4C 0 58 COC(=O)c1ccnc(C(C)C)c1 ZINC000147082155 AD For-Sale Anodyne KDM3A 0 58 COC(=O)c1ccnc(C(C)C)c1 ZINC000147082155 AD For-Sale Anodyne KDM5C 0 58 C[C@@]1(c2cc(NC(=O)c3cnc(-c4ncco4)cn3)ccc2F)C=CSC(N)=N1 ZINC000147082251 HG Annotated Anodyne BACE2 54 49 C[C@@]1(c2cc(NC(=O)c3cnc(-c4ncco4)cn3)ccc2F)C=CSC(N)=N1 ZINC000147082251 HG Annotated Anodyne BACE1 26 46 Cc1cc(NC(=O)c2ccc3cc4n(c3n2)CC(C)(C)CNC4=O)no1 ZINC000147082259 FE Annotated Anodyne RPS6KA3 43 39 Cc1cc(C)c(CNC(=O)c2cc(-c3cnn(C)c3)cc(N(C)[C@@H]3CC[C@H](N)CC3)c2C)c(=O)[nH]1 ZINC000147082316 JG Annotated Anodyne EZH2 42 49 CCCCO[C@@H](C)C(=O)NCCCc1nc2ccccc2[nH]1 ZINC000147082375 DF On-Demand Anodyne MTNR1A 26 40 CCCCO[C@@H](C)C(=O)NCCCc1nc2ccccc2[nH]1 ZINC000147082375 DF On-Demand Anodyne MTNR1B 39 40 CCCCO[C@@H](C)C(=O)NCCCc1nc2ccccc2[nH]1 ZINC000147082375 DF On-Demand Anodyne CACNA1G 24 43 COc1cnc(C(=O)Nc2cccc([C@]3(C(F)(F)F)CCSC(N)=N3)c2)cn1 ZINC000147082452 HF Annotated Anodyne BACE2 46 49 COc1cnc(C(=O)Nc2cccc([C@]3(C(F)(F)F)CCSC(N)=N3)c2)cn1 ZINC000147082452 HF Annotated Anodyne BACE1 31 63 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne F2 35 42 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne PLG 42 42 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne TACR1 16 42 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne TRY2_BOVIN 97 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne CCKAR 15 55 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne CCR1 27 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne CCR3 53 39 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne DPP4 15 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne MLNR 25 45 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne F11 36 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne CCKBR 15 55 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne EPHX2 28 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne ST14 117 42 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne CACNA1G 35 43 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne TMPRSS6 63 34 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082468 FH On-Demand Anodyne KCNK3 19 40 Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(CN(C)C)cc3)cc(N(C)[C@@H]3CC[C@H](N)CC3)c2C)c(=O)[nH]1 ZINC000147082479 KJ Annotated Anodyne EZH2 43 56 NC(=O)c1ccc(OCC(=O)N2CCCCC[C@@H]2c2ccncc2)cc1 ZINC000147082483 FF On-Demand Anodyne COLA 170 59 NC(=O)c1ccc(OCC(=O)N2CCCCC[C@@H]2c2ccncc2)cc1 ZINC000147082483 FF On-Demand Anodyne CPT1A 147 59 NC(=O)c1ccc(OCC(=O)N2CCCCC[C@@H]2c2ccncc2)cc1 ZINC000147082483 FF On-Demand Anodyne CPT2 50 40 CCCCO[C@H](C)C(=O)NCCCc1nc2ccccc2[nH]1 ZINC000147082504 DF On-Demand Anodyne CYSP_TRYCR 19 48 CCCCO[C@H](C)C(=O)NCCCc1nc2ccccc2[nH]1 ZINC000147082504 DF On-Demand Anodyne MTNR1A 26 40 CCCCO[C@H](C)C(=O)NCCCc1nc2ccccc2[nH]1 ZINC000147082504 DF On-Demand Anodyne MTNR1B 39 40 CCCCO[C@H](C)C(=O)NCCCc1nc2ccccc2[nH]1 ZINC000147082504 DF On-Demand Anodyne CACNA1G 33 46 CCOC(=O)[C@H](CCC1CCCCC1)N[C@H](C)C(=O)O ZINC000147082506 CE For-Sale Anodyne METAP2 20 55 COc1ccc(C#N)cc1N[C@@H](C)C(=O)Nc1cccc2ncccc12 ZINC000147082513 EH On-Demand Mild P2RX7 23 46 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3cccc(Cn4cccn4)c3)c2)CCO1 ZINC000147082526 HG On-Demand Anodyne CCR3 35 43 CC1(C)CNC(=O)c2cc3ccc(C(=O)Nc4cc(-c5ccccc5)on4)nc3n2C1 ZINC000147082551 HH Annotated Anodyne RPS6KA3 48 41 COc1cnc(C(=O)Nc2cccc([C@@]3(C(F)(F)F)CCSC(N)=N3)c2)cn1 ZINC000147082641 HF Annotated Anodyne BACE2 46 49 COc1cnc(C(=O)Nc2cccc([C@@]3(C(F)(F)F)CCSC(N)=N3)c2)cn1 ZINC000147082641 HF Annotated Anodyne BACE1 31 63 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne F2 35 42 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne PLG 42 42 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne TACR1 16 42 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne TRY2_BOVIN 97 44 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne CCKAR 15 55 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne CCR1 27 44 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne CCR3 53 39 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne DPP4 15 40 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne MLNR 25 45 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne F11 36 40 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne CCKBR 15 55 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne EPHX2 28 44 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne ST14 117 42 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne CACNA1G 35 43 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne TMPRSS6 63 34 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)Nc2ccccc2)CC1 ZINC000147082642 FH On-Demand Anodyne KCNK3 19 40 NC(=O)c1ccc(OCC(=O)N2CCCCC[C@H]2c2ccncc2)cc1 ZINC000147082662 FF On-Demand Anodyne COLA 170 59 Cc1cc(C)c(CNC(=O)c2cc(-c3cnn(CCN4CCOCC4)c3)cc(N(C)[C@@H]3CC[C@H](N)CC3)c2C)c(=O)[nH]1 ZINC000147082682 KG Annotated Anodyne EZH2 44 58 N#CC1CCN(C(=O)c2ccc(NC(=O)Nc3ccccc3)cc2)CC1 ZINC000147082685 EH On-Demand Mild AVPR2 46 47 N#CC1CCN(C(=O)c2ccc(NC(=O)Nc3ccccc3)cc2)CC1 ZINC000147082685 EH On-Demand Mild AVPR1A 44 47 N#CC1CCN(C(=O)c2ccc(NC(=O)Nc3ccccc3)cc2)CC1 ZINC000147082685 EH On-Demand Mild DHODH 60 40 N#CC1CCN(C(=O)c2ccc(NC(=O)Nc3ccccc3)cc2)CC1 ZINC000147082685 EH On-Demand Mild PIK3CA 21 44 N#CC1CCN(C(=O)c2ccc(NC(=O)Nc3ccccc3)cc2)CC1 ZINC000147082685 EH On-Demand Mild MTOR 43 44 N#CC1CCN(C(=O)c2ccc(NC(=O)Nc3ccccc3)cc2)CC1 ZINC000147082685 EH On-Demand Mild EPHX2 55 62 N#CC1CCN(C(=O)c2ccc(NC(=O)Nc3ccccc3)cc2)CC1 ZINC000147082685 EH On-Demand Mild PIK3CG 18 44 N#CC1CCN(C(=O)c2ccc(NC(=O)Nc3ccccc3)cc2)CC1 ZINC000147082685 EH On-Demand Mild DGAT1 17 46 N#CC1CCN(C(=O)c2ccc(NC(=O)Nc3ccccc3)cc2)CC1 ZINC000147082685 EH On-Demand Mild L3MBTL3 90 41 CCCC(=O)Nc1cccc(C(=O)O)c1O ZINC000147082689 BD On-Demand Anodyne CXCR2 43 34 CCCC(=O)Nc1cccc(C(=O)O)c1O ZINC000147082689 BD On-Demand Anodyne CXCR1 45 35 CCCC(=O)Nc1cccc(C(=O)O)c1O ZINC000147082689 BD On-Demand Anodyne HCAR2 44 48 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCCn3cncn3)c1)C2 ZINC000147082691 GF On-Demand Anodyne ROCK2 36 44 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCCn3cncn3)c1)C2 ZINC000147082691 GF On-Demand Anodyne EPHX2 15 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCCn3cncn3)c1)C2 ZINC000147082691 GF On-Demand Anodyne LIMK2 18 40 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3cccc(Cn4cccn4)c3)c2)CCO1 ZINC000147082697 HG On-Demand Anodyne CCR3 35 43 CN1[C@@H](C(=O)NCC[C@H](O)CO)[C@H](c2cccc(Cl)c2)[C@@]2(C(=O)Nc3cc(Cl)c(F)cc32)[C@H]1CCc1cccs1 ZINC000147082724 KI Annotated Anodyne MDM2 45 61 Cc1nn(C(F)F)c(C)c1CC(=O)NCCCc1nc2ccccc2[nH]1 ZINC000147082741 FG On-Demand Anodyne CYSP_TRYCR 19 49 COC(=O)[C@@H](C)C[C@@H](C(=O)c1ccc(Cl)cc1)c1cccc(Cl)c1 ZINC000147082749 FK For-Sale Anodyne UTS2 42 32 COc1ccc(C#N)cc1N[C@H](C)C(=O)NC(=O)NCc1ccccc1 ZINC000147082801 FE On-Demand Mild ANPEP 28 40 COc1ccc(C#N)cc1N[C@H](C)C(=O)NC(=O)NCc1ccccc1 ZINC000147082801 FE On-Demand Mild PDS 39 41 Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(CN4CCOCC4)nc3)cc(N(C)[C@@H]3CC[C@H](N)CC3)c2C)c(=O)[nH]1 ZINC000147082884 KH Annotated Anodyne EZH2 47 62 N#CC1CCN(C(=O)c2ccc(-n3cncn3)cc2)CC1 ZINC000147082888 CD On-Demand Mild L3MBTL3 60 40 COC(=O)[C@H](C)C[C@@H](C(=O)c1ccc(Cl)cc1)c1cccc(Cl)c1 ZINC000147082922 FK For-Sale Anodyne UTS2 42 32 COC(=O)[C@@H](C)C[C@H](C(=O)c1ccc(Cl)cc1)c1cccc(Cl)c1 ZINC000147083023 FK For-Sale Anodyne UTS2 42 32 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083095 GF On-Demand Bother LPL 48 38 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083095 GF On-Demand Bother CPT1A 37 42 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083095 GF On-Demand Bother EPHX2 26 50 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083095 GF On-Demand Bother TGM2 64 42 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083095 GF On-Demand Bother F13A1 92 49 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083095 GF On-Demand Bother NAMPT 33 43 Cc1cc(C)c(CNC(=O)c2cc(-c3ccc(CN(C)C)nc3)cc(N(C)[C@@H]3CC[C@H](N)CC3)c2C)c(=O)[nH]1 ZINC000147083099 KI Annotated Anodyne EZH2 43 48 O=C(c1csc(-c2ccccc2F)n1)N1CCCCC[C@H]1c1ccncc1 ZINC000147083132 GK On-Demand Anodyne CPT1A 46 44 COC(=O)[C@H](C)C[C@H](C(=O)c1ccc(Cl)cc1)c1cccc(Cl)c1 ZINC000147083149 FK For-Sale Anodyne UTS2 42 32 COC[C@H](C)N(C)C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147083164 CF On-Demand Anodyne GPR88 0 52 C=C1C[C@@](C)(c2cc(NC(=O)c3cnc(C)cn3)ccc2F)N=C(N)S1 ZINC000147083197 FG Annotated Mild BACE2 58 62 C=C1C[C@@](C)(c2cc(NC(=O)c3cnc(C)cn3)ccc2F)N=C(N)S1 ZINC000147083197 FG Annotated Mild BACE1 29 56 CC(C)C(NC(=O)c1c(O)cccc1O)C(C)C ZINC000147083374 CF Annotated Anodyne DAC 31 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC)c(OCC(N)=O)c2)c1 ZINC000147083376 GD On-Demand Bother TAAR1 28 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC)c(OCC(N)=O)c2)c1 ZINC000147083376 GD On-Demand Bother AKR1C3 16 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC)c(OCC(N)=O)c2)c1 ZINC000147083376 GD On-Demand Bother AKR1C2 42 39 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC)c(OCC(N)=O)c2)c1 ZINC000147083376 GD On-Demand Bother ENPP1 71 34 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC)c(OCC(N)=O)c2)c1 ZINC000147083376 GD On-Demand Bother KCNK3 42 37 COc1ccc([C@]2(c3cccc(NC(=O)c4ncc(Cl)cc4Cl)c3)CSC(N)=N2)cc1O ZINC000147083388 JJ Annotated Anodyne BACE2 48 46 COc1ccc([C@]2(c3cccc(NC(=O)c4ncc(Cl)cc4Cl)c3)CSC(N)=N2)cc1O ZINC000147083388 JJ Annotated Anodyne BACE1 22 47 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083408 HG On-Demand Bother LPL 49 40 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083408 HG On-Demand Bother CPT1A 34 42 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083408 HG On-Demand Bother EPHX2 26 49 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083408 HG On-Demand Bother TGM2 62 43 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083408 HG On-Demand Bother F13A1 88 48 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083408 HG On-Demand Bother LIPG 20 40 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147083408 HG On-Demand Bother NAMPT 32 45 COC[C@H](C)N(C)C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147083435 CF On-Demand Anodyne GPR88 0 52 Fc1ncccc1OC[C@H]1C=CCN1 ZINC000147083486 AD For-Sale Anodyne CHRNA2 20 60 COc1ccc([C@@]2(c3cccc(NC(=O)c4ncc(Cl)cc4Cl)c3)CSC(N)=N2)cc1O ZINC000147083537 JJ Annotated Anodyne BACE2 48 46 COc1ccc([C@@]2(c3cccc(NC(=O)c4ncc(Cl)cc4Cl)c3)CSC(N)=N2)cc1O ZINC000147083537 JJ Annotated Anodyne BACE1 22 47 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083545 EF On-Demand Anodyne F2 40 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083545 EF On-Demand Anodyne P2RY12 125 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083545 EF On-Demand Anodyne TRHR 49 36 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083545 EF On-Demand Anodyne TRY1_BOVIN 69 39 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083545 EF On-Demand Anodyne NTSR1 57 31 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083545 EF On-Demand Anodyne ADAM17 45 49 CCc1ncc(C(=O)Nc2ccc(C(=O)Nc3ccc(OC)cc3)cc2)s1 ZINC000147083596 GI On-Demand Anodyne PRSS1 15 41 CCc1ncc(C(=O)Nc2ccc(C(=O)Nc3ccc(OC)cc3)cc2)s1 ZINC000147083596 GI On-Demand Anodyne TRPV1 22 42 CCc1ncc(C(=O)Nc2ccc(C(=O)Nc3ccc(OC)cc3)cc2)s1 ZINC000147083596 GI On-Demand Anodyne PRNP 53 40 CCc1ncc(C(=O)Nc2ccc(C(=O)Nc3ccc(OC)cc3)cc2)s1 ZINC000147083596 GI On-Demand Anodyne ACR 42 41 CCc1ncc(C(=O)Nc2ccc(C(=O)Nc3ccc(OC)cc3)cc2)s1 ZINC000147083596 GI On-Demand Anodyne LUCI_LUCLA 16 41 CCc1ncc(C(=O)Nc2ccc(C(=O)Nc3ccc(OC)cc3)cc2)s1 ZINC000147083596 GI On-Demand Anodyne SHH 53 37 CCc1ncc(C(=O)Nc2ccc(C(=O)Nc3ccc(OC)cc3)cc2)s1 ZINC000147083596 GI On-Demand Anodyne DGAT1 18 40 CCc1ncc(C(=O)Nc2ccc(C(=O)Nc3ccc(OC)cc3)cc2)s1 ZINC000147083596 GI On-Demand Anodyne NOD1 16 42 CCc1ncc(C(=O)Nc2ccc(C(=O)Nc3ccc(OC)cc3)cc2)s1 ZINC000147083596 GI On-Demand Anodyne NOD2 34 42 CCc1ncc(C(=O)Nc2ccc(C(=O)Nc3ccc(OC)cc3)cc2)s1 ZINC000147083596 GI On-Demand Anodyne USP7 36 40 CCc1ncc(C(=O)Nc2ccc(C(=O)Nc3ccc(OC)cc3)cc2)s1 ZINC000147083596 GI On-Demand Anodyne USP47 45 40 N#CC1CCN(C(=O)Cc2csc(-c3ccccn3)n2)CC1 ZINC000147083619 DF On-Demand Mild COLA 21 46 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083671 EF On-Demand Anodyne F2 40 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083671 EF On-Demand Anodyne P2RY12 125 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083671 EF On-Demand Anodyne TRHR 49 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083671 EF On-Demand Anodyne TRY1_BOVIN 69 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083671 EF On-Demand Anodyne NTSR1 57 31 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1cccc(OC)c1 ZINC000147083671 EF On-Demand Anodyne ADAM17 45 49 COc1c(C(=O)O)oc2ccccc2c1=O ZINC000147083706 BD For-Sale Anodyne CYP2C9 19 46 COc1c(C(=O)O)oc2ccccc2c1=O ZINC000147083706 BD For-Sale Anodyne NQO1 43 40 CC(=O)N[C@H]1CC[C@@H](N(C)c2cc(-c3ccc(CN4CCOCC4)nc3)cc(C(=O)NCc3c(C)cc(C)[nH]c3=O)c2C)CC1 ZINC000147083761 KI Annotated Anodyne EZH2 45 60 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother GYRB 40 32 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother PLAU 17 40 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother TAAR1 35 54 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother AKR1C3 22 43 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother AKR1C2 48 43 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother NOD1 15 40 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother NOD2 31 40 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother GPR35 20 41 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother USP7 18 40 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother USP47 23 40 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother KCNK3 70 43 COc1ccc(NC(=O)c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)cc2)cc1 ZINC000147083787 HI On-Demand Bother KCNK9 46 37 COc1ccc(S(=O)(=O)[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147083835 CG For-Sale Anodyne MMP13 52 48 COc1ccc(S(=O)(=O)[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147083835 CG For-Sale Anodyne MMP3 59 40 COc1ccc(S(=O)(=O)[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147083835 CG For-Sale Anodyne MMP8 35 46 COc1ccc(S(=O)(=O)[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147083835 CG For-Sale Anodyne MMP9 46 40 COc1ccc(S(=O)(=O)[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147083835 CG For-Sale Anodyne MMP7 46 40 COc1ccc(S(=O)(=O)[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147083835 CG For-Sale Anodyne MMP1 51 46 COC[C@H](C)N(C)C(=O)[C@@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147083851 EG On-Demand Anodyne GPR88 0 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147083858 EF On-Demand Anodyne F2 40 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147083858 EF On-Demand Anodyne P2RY12 125 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147083858 EF On-Demand Anodyne TRHR 49 36 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147083858 EF On-Demand Anodyne TRY1_BOVIN 69 39 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147083858 EF On-Demand Anodyne NTSR1 57 31 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147083858 EF On-Demand Anodyne ADAM17 17 49 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(COc2ccc3c(c2)OCO3)c1 ZINC000147083877 HF On-Demand Anodyne MAOB 17 41 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1cccc(Cn2cccn2)c1 ZINC000147084006 HJ On-Demand Anodyne ROCK2 21 42 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1cccc(Cn2cccn2)c1 ZINC000147084006 HJ On-Demand Anodyne MET 34 43 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1cccc(Cn2cccn2)c1 ZINC000147084006 HJ On-Demand Anodyne NAMPT 43 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147084052 EF On-Demand Anodyne F2 40 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147084052 EF On-Demand Anodyne P2RY12 125 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147084052 EF On-Demand Anodyne TRHR 49 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147084052 EF On-Demand Anodyne TRY1_BOVIN 69 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147084052 EF On-Demand Anodyne NTSR1 57 31 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1cccc(OC)c1 ZINC000147084052 EF On-Demand Anodyne ADAM17 45 49 CC1(C)CNC(=O)c2cc3ccc(C(=O)Nc4cc(Cc5ccccc5)on4)nc3n2C1 ZINC000147084067 IH Annotated Anodyne RPS6KA3 38 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(COc2ccc3c(c2)OCO3)c1 ZINC000147084076 HF On-Demand Anodyne MAOB 17 41 Nc1nc(N)c2ncn([C@@H]3O[C@H](CO)C[C@@H]3O)c2n1 ZINC000147084137 CA For-Sale Anodyne ADA 40 31 Nc1nc(N)c2ncn([C@@H]3O[C@H](CO)C[C@@H]3O)c2n1 ZINC000147084137 CA For-Sale Anodyne ADORA1 97 55 Nc1nc(N)c2ncn([C@@H]3O[C@H](CO)C[C@@H]3O)c2n1 ZINC000147084137 CA For-Sale Anodyne SLC29A1 67 46 Nc1nc(N)c2ncn([C@@H]3O[C@H](CO)C[C@@H]3O)c2n1 ZINC000147084137 CA For-Sale Anodyne ADORA2A 58 52 Nc1nc(N)c2ncn([C@@H]3O[C@H](CO)C[C@@H]3O)c2n1 ZINC000147084137 CA For-Sale Anodyne AHCY 90 41 Nc1nc(N)c2ncn([C@@H]3O[C@H](CO)C[C@@H]3O)c2n1 ZINC000147084137 CA For-Sale Anodyne ADCY5 43 47 Nc1nc(N)c2ncn([C@@H]3O[C@H](CO)C[C@@H]3O)c2n1 ZINC000147084137 CA For-Sale Anodyne ADORA3 33 46 Nc1nc(N)c2ncn([C@@H]3O[C@H](CO)C[C@@H]3O)c2n1 ZINC000147084137 CA For-Sale Anodyne OXGR1 116 38 Nc1nc(N)c2ncn([C@@H]3O[C@H](CO)C[C@@H]3O)c2n1 ZINC000147084137 CA For-Sale Anodyne Q4VQ11_PIG 61 38 Nc1nc(N)c2ncn([C@@H]3O[C@H](CO)C[C@@H]3O)c2n1 ZINC000147084137 CA For-Sale Anodyne DOT1L 50 33 COc1ccc([N+](=O)[O-])cc1NC(=O)[C@@H](C)Nc1cc(C#N)ccc1OC ZINC000147084234 FF On-Demand Mild PYGL 16 44 COc1ccc([N+](=O)[O-])cc1NC(=O)[C@@H](C)Nc1cc(C#N)ccc1OC ZINC000147084234 FF On-Demand Mild KCNMA1 22 53 NC(=O)c1ccc(OCC(=O)NC2CCN(c3ccccn3)CC2)cc1 ZINC000147084245 FD On-Demand Anodyne AVPR1A 15 42 NC(=O)c1ccc(OCC(=O)NC2CCN(c3ccccn3)CC2)cc1 ZINC000147084245 FD On-Demand Anodyne COLA 31 44 NC(=O)c1ccc(OCC(=O)NC2CCN(c3ccccn3)CC2)cc1 ZINC000147084245 FD On-Demand Anodyne CPT1A 26 44 NC(=O)c1ccc(OCC(=O)NC2CCN(c3ccccn3)CC2)cc1 ZINC000147084245 FD On-Demand Anodyne MCHR1 18 46 NC(=O)c1ccc(OCC(=O)NC2CCN(c3ccccn3)CC2)cc1 ZINC000147084245 FD On-Demand Anodyne SIRT2 43 30 COC[C@H](C)N(C)C(=O)[C@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147084246 EG On-Demand Anodyne GPR88 0 43 N#CC1CCN(C(=O)Cc2csc(-c3ccccc3Cl)n2)CC1 ZINC000147084443 EH On-Demand Mild ETHR 43 37 COc1ccc(Nc2nc(-c3ccc4c(cnn4C)c3)cn3ccnc23)cc1OC ZINC000147084556 HI For-Sale Anodyne EPHB4 37 40 CN1CCN(CCCNC(=O)[C@@H]2N[C@H](CC(C)(C)C)[C@]3(C(=O)Nc4cc(Cl)ccc43)[C@H]2c2cccc(Cl)c2F)CC1 ZINC000147084596 KJ Annotated Anodyne ADRA1D 40 34 CN1CCN(CCCNC(=O)[C@@H]2N[C@H](CC(C)(C)C)[C@]3(C(=O)Nc4cc(Cl)ccc43)[C@H]2c2cccc(Cl)c2F)CC1 ZINC000147084596 KJ Annotated Anodyne MDM2 105 84 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000147084652 EF On-Demand Mild CACNA1D 55 36 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000147084652 EF On-Demand Mild KCNMA1 20 46 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000147084652 EF On-Demand Mild AKR1C2 15 40 CCOC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147084671 EG On-Demand Bother CACNA1C 43 38 CCOC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147084671 EG On-Demand Bother CACNA1D 61 38 CCOC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147084671 EG On-Demand Bother ACR 58 38 CCOC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147084671 EG On-Demand Bother NOD2 18 43 CCOC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147084671 EG On-Demand Bother KCNK3 40 35 CCOC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147084671 EG On-Demand Bother KCNK9 41 35 Cc1cc2nc(C)c(CCC(=O)N3CCC(C#N)CC3)c(C)n2n1 ZINC000147084731 EE On-Demand Mild DPP8 17 45 Cc1cc2nc(C)c(CCC(=O)N3CCC(C#N)CC3)c(C)n2n1 ZINC000147084731 EE On-Demand Mild DPP9 28 45 C[C@@]1(c2cc(NC(=O)c3cc4n(n3)CCN4)ccc2F)C=CSC(N)=N1 ZINC000147084771 FE Annotated Anodyne BACE2 44 44 C[C@@]1(c2cc(NC(=O)c3cc4n(n3)CCN4)ccc2F)C=CSC(N)=N1 ZINC000147084771 FE Annotated Anodyne BACE1 22 44 CCCC(=O)Nc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147084816 FG On-Demand Bother ROCK1 20 40 CCCC(=O)Nc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147084816 FG On-Demand Bother MTNR1A 49 50 CCCC(=O)Nc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147084816 FG On-Demand Bother MTNR1B 45 50 CCCC(=O)Nc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147084816 FG On-Demand Bother TAAR1 27 45 CCCC(=O)Nc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147084816 FG On-Demand Bother AKR1C2 23 40 C[C@@H](CNC(=O)Cn1c(=O)[nH]c(=O)c2ccccc21)N1CCCC1 ZINC000147084906 EC On-Demand Anodyne PARP1 17 46 N#CC1CCN(C(=O)Cc2csc(-c3cccs3)n2)CC1 ZINC000147084935 DG On-Demand Mild FAP 0 40 N#CC1CCN(C(=O)Cc2csc(-c3cccs3)n2)CC1 ZINC000147084935 DG On-Demand Mild ETHR 67 51 Cc1cc([N+](=O)[O-])ccc1NC(=O)N1Cc2ccccc2C1 ZINC000147085009 CG On-Demand Bother KCNMA1 24 40 Cc1cc([N+](=O)[O-])ccc1NC(=O)N1Cc2ccccc2C1 ZINC000147085009 CG On-Demand Bother TRPM8 0 42 Cc1cc([N+](=O)[O-])ccc1NC(=O)N1Cc2ccccc2C1 ZINC000147085009 CG On-Demand Bother WDR5 34 41 C[C@H](CNC(=O)Cn1c(=O)[nH]c(=O)c2ccccc21)N1CCCC1 ZINC000147085119 EC On-Demand Anodyne PARP1 17 46 O=C(CCc1ccccc1)NCC1CCN(C2CCOCC2)CC1 ZINC000147085338 EF In-Stock Anodyne HTR4 37 40 O=C(CCc1ccccc1)NCC1CCN(C2CCOCC2)CC1 ZINC000147085338 EF In-Stock Anodyne GRIN2B 46 39 O=C(CCc1ccccc1)NCC1CCN(C2CCOCC2)CC1 ZINC000147085338 EF In-Stock Anodyne SIGMAR1 31 40 O=C(CCc1ccccc1)NCC1CCN(C2CCOCC2)CC1 ZINC000147085338 EF In-Stock Anodyne CCR3 43 37 O=C(CCc1ccccc1)NCC1CCN(C2CCOCC2)CC1 ZINC000147085338 EF In-Stock Anodyne CACNA1I 53 38 CCOc1ccccc1C(=O)N1CCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147085363 HH On-Demand Anodyne HCN1 53 35 CCOc1ccccc1C(=O)N1CCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147085363 HH On-Demand Anodyne HCN4 45 34 Cc1ncnn1-c1cnc(C(=O)Nc2ccc(F)c([C@]3(C)C=CSC(N)=N3)c2)cn1 ZINC000147085424 HF Annotated Anodyne BACE2 51 50 Cc1ncnn1-c1cnc(C(=O)Nc2ccc(F)c([C@]3(C)C=CSC(N)=N3)c2)cn1 ZINC000147085424 HF Annotated Anodyne BACE1 25 54 CCc1nc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])sc1C ZINC000147085465 DG On-Demand Bother CSNK1D 21 40 CCc1nc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])sc1C ZINC000147085465 DG On-Demand Bother USP7 19 40 CCc1nc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])sc1C ZINC000147085465 DG On-Demand Bother USP47 23 40 CCOc1ccccc1C(=O)N1CCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147085538 HH On-Demand Anodyne HCN1 53 35 CCOc1ccccc1C(=O)N1CCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147085538 HH On-Demand Anodyne HCN4 45 34 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc([N+](=O)[O-])cc1Cl ZINC000147085703 FH On-Demand Mild KCNMA1 21 44 CCOc1ccccc1C(=O)N1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147085723 HH On-Demand Anodyne HCN1 53 35 CCOc1ccccc1C(=O)N1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147085723 HH On-Demand Anodyne HCN4 45 34 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147085772 GG On-Demand Anodyne MAPK11 50 51 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147085772 GG On-Demand Anodyne MAPK14 84 55 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147085772 GG On-Demand Anodyne MAPK13 98 39 CC(C)(C)NC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147085865 FD On-Demand Anodyne KCNK3 61 35 CCCOc1ccc([C@@H](C)NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1OC ZINC000147085991 GH On-Demand Bother ACACA 41 38 COc1ccc(Br)cc1S(=O)(=O)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000147085998 IF On-Demand Anodyne EDNRB 48 34 COc1ccc(Br)cc1S(=O)(=O)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000147085998 IF On-Demand Anodyne TACR1 23 42 COc1ccc(Br)cc1S(=O)(=O)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000147085998 IF On-Demand Anodyne CTSL 29 43 COc1ccc(Br)cc1S(=O)(=O)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000147085998 IF On-Demand Anodyne MMP2 23 45 COc1ccc(Br)cc1S(=O)(=O)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000147085998 IF On-Demand Anodyne ECE1 47 40 COc1ccc(Br)cc1S(=O)(=O)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000147085998 IF On-Demand Anodyne CCKBR 43 38 COc1ccc(Br)cc1S(=O)(=O)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000147085998 IF On-Demand Anodyne GHSR 53 35 COc1ccc(Br)cc1S(=O)(=O)N[C@@H](CO)Cc1c[nH]c2ccccc12 ZINC000147085998 IF On-Demand Anodyne MMP9 21 45 CC(C)(C)NC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147086068 FD On-Demand Anodyne KCNK3 61 35 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147086124 GH On-Demand Mild P2RY1 54 41 O=S(=O)(N[C@@H](CO)Cc1c[nH]c2ccccc12)c1ccccc1Br ZINC000147086168 HF On-Demand Anodyne ACE 16 42 O=S(=O)(N[C@@H](CO)Cc1c[nH]c2ccccc12)c1ccccc1Br ZINC000147086168 HF On-Demand Anodyne MME 24 43 O=S(=O)(N[C@@H](CO)Cc1c[nH]c2ccccc12)c1ccccc1Br ZINC000147086168 HF On-Demand Anodyne CTSL 29 48 O=S(=O)(N[C@@H](CO)Cc1c[nH]c2ccccc12)c1ccccc1Br ZINC000147086168 HF On-Demand Anodyne MMP2 25 48 O=S(=O)(N[C@@H](CO)Cc1c[nH]c2ccccc12)c1ccccc1Br ZINC000147086168 HF On-Demand Anodyne ECE1 55 43 O=S(=O)(N[C@@H](CO)Cc1c[nH]c2ccccc12)c1ccccc1Br ZINC000147086168 HF On-Demand Anodyne MMP11 57 32 O=S(=O)(N[C@@H](CO)Cc1c[nH]c2ccccc12)c1ccccc1Br ZINC000147086168 HF On-Demand Anodyne GHSR 49 37 O=S(=O)(N[C@@H](CO)Cc1c[nH]c2ccccc12)c1ccccc1Br ZINC000147086168 HF On-Demand Anodyne MMP9 23 48 O=S(=O)(N[C@@H](CO)Cc1c[nH]c2ccccc12)c1ccccc1Br ZINC000147086168 HF On-Demand Anodyne MMP1 19 41 O=S(=O)(N[C@@H](CO)Cc1c[nH]c2ccccc12)c1ccccc1Br ZINC000147086168 HF On-Demand Anodyne NPR 31 43 CCCOc1ccc([C@H](C)NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1OC ZINC000147086180 GH On-Demand Bother ACACA 41 38 COc1ccc(-c2nn(-c3ccccc3)cc2CC(=O)NC[C@H](C)N2CCCC2)cc1 ZINC000147086354 HH On-Demand Anodyne CDK2 16 47 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1cccc(F)c1 ZINC000147086500 HI On-Demand Anodyne KCNK3 28 41 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1cccc(F)c1 ZINC000147086500 HI On-Demand Anodyne KCNK9 35 41 CC(C)(C)c1cc(NC(=O)c2ccc3cc4n(c3n2)CCCNC4=O)no1 ZINC000147086600 FF Annotated Anodyne FLT3 50 41 CC(C)(C)c1cc(NC(=O)c2ccc3cc4n(c3n2)CCCNC4=O)no1 ZINC000147086600 FF Annotated Anodyne RPS6KA3 83 51 CC(C)(C)c1cc(NC(=O)c2ccc3cc4n(c3n2)CCCNC4=O)no1 ZINC000147086600 FF Annotated Anodyne CSF1R 17 41 CC(C)(C)c1cc(NC(=O)c2ccc3cc4n(c3n2)CCCNC4=O)no1 ZINC000147086600 FF Annotated Anodyne Q8MMZ8_EIMTE 19 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(OC[C@@H]3CCCO3)cc1)C2 ZINC000147086639 GG On-Demand Anodyne MTNR1A 23 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(OC[C@@H]3CCCO3)cc1)C2 ZINC000147086639 GG On-Demand Anodyne MTNR1B 22 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(OC[C@@H]3CCCO3)cc1)C2 ZINC000147086639 GG On-Demand Anodyne ROCK2 28 49 O=C(CCCN1CCC(COC(=O)c2c[nH]c3ccccc23)CC1)OCC(Cl)(Cl)Cl ZINC000147086678 JJ For-Sale Anodyne HTR4 76 75 O=C(CCCN1CCC(COC(=O)c2c[nH]c3ccccc23)CC1)OCC(Cl)(Cl)Cl ZINC000147086678 JJ For-Sale Anodyne CYP2J2 43 31 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1cccc(F)c1 ZINC000147086684 HI On-Demand Anodyne KCNK3 28 41 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1cccc(F)c1 ZINC000147086684 HI On-Demand Anodyne KCNK9 35 41 C[C@@H](CN)C[C@@H](C)C(=O)O ZINC000147086827 AC For-Sale Anodyne GRIK3 23 56 CCCCC(=O)NC1CCN(C(=O)c2cc(OC)ccc2[N+](=O)[O-])CC1 ZINC000147086838 FF For-Sale Bother MTNR1A 16 45 CCCCC(=O)NC1CCN(C(=O)c2cc(OC)ccc2[N+](=O)[O-])CC1 ZINC000147086838 FF For-Sale Bother MTNR1B 19 45 CCCCC(=O)NC1CCN(C(=O)c2cc(OC)ccc2[N+](=O)[O-])CC1 ZINC000147086838 FF For-Sale Bother EPHX2 15 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(OC[C@@H]3CCCO3)cc1)C2 ZINC000147086841 GG On-Demand Anodyne MTNR1A 23 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(OC[C@@H]3CCCO3)cc1)C2 ZINC000147086841 GG On-Demand Anodyne MTNR1B 22 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(OC[C@@H]3CCCO3)cc1)C2 ZINC000147086841 GG On-Demand Anodyne ROCK2 28 49 CNCC1=CC[C@H]2C[C@@H]1C2(C)C ZINC000147086869 AE For-Sale Anodyne CXCR3 60 45 C[C@H](CN)C[C@@H](C)C(=O)O ZINC000147087002 AC For-Sale Anodyne GRIK3 23 56 CCCn1c(CCC(=O)N2CCC(C#N)CC2)nc2cc(S(N)(=O)=O)ccc21 ZINC000147087037 HD On-Demand Mild CNR2 16 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(OC[C@H]3CCCO3)cc1)C2 ZINC000147087043 GG On-Demand Anodyne MTNR1A 23 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(OC[C@H]3CCCO3)cc1)C2 ZINC000147087043 GG On-Demand Anodyne MTNR1B 22 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(OC[C@H]3CCCO3)cc1)C2 ZINC000147087043 GG On-Demand Anodyne ROCK2 28 49 CNCC1=CC[C@H]2C[C@H]1C2(C)C ZINC000147087064 AE For-Sale Anodyne CXCR3 60 45 CC(C)(C)OC(=O)N[C@H](C=O)Cc1ccc([N+](=O)[O-])cc1 ZINC000147087085 CE For-Sale Anodyne CCR3 25 42 CC1=CC(C)(C)Nc2ccc(Oc3cccc(Cl)c3)nc21 ZINC000147087145 DK For-Sale Anodyne PGA 57 37 CNC(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000147087177 BE For-Sale Anodyne SLC6A4 15 47 CNC(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000147087177 BE For-Sale Anodyne P2RX7 28 50 CNC(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000147087177 BE For-Sale Anodyne DNAE 83 35 CNC(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000147087177 BE For-Sale Anodyne NCE103 15 41 CNC(=O)NCc1ccc(Cl)c(Cl)c1 ZINC000147087177 BE For-Sale Anodyne RPA1 62 34 Cc1ccc(NC(=O)CS(=O)(=O)[C@H](C)c2ccc(OC(F)(F)F)cc2)cc1C ZINC000147087180 HI On-Demand Anodyne MCHR1 16 44 Cc1ccc(NC(=O)CS(=O)(=O)[C@H](C)c2ccc(OC(F)(F)F)cc2)cc1C ZINC000147087180 HI On-Demand Anodyne SHH 40 35 COc1cc(Cl)c(C(=O)NN)cc1Cl ZINC000147087183 BD For-Sale Reactive HTR4 70 43 C[C@@H](C[C@@H](C)CN)C(=O)O ZINC000147087191 AC For-Sale Anodyne GRIK3 23 56 CNc1nc(Cl)c(Cl)c(N2CCN(CCC3CCC(NC(=O)N(C)C)CC3)CC2)n1 ZINC000147087340 JG Annotated Anodyne DRD3 23 64 C[C@H](CN)C[C@H](C)C(=O)O ZINC000147087380 AC For-Sale Anodyne GRIK3 23 56 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087464 FD On-Demand Anodyne CCR3 55 42 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087464 FD On-Demand Anodyne HDAC10 50 41 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087464 FD On-Demand Anodyne HDAC2 30 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087464 FD On-Demand Anodyne HDAC3 32 41 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087464 FD On-Demand Anodyne HDAC6 25 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087464 FD On-Demand Anodyne HDAC11 44 41 CCC(=O)Nc1ccc(Cl)c(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147087470 FE On-Demand Anodyne ENV 41 33 CC(=O)c1ccc(OC(=O)c2c3ccccc3nc3ccccc23)cc1 ZINC000147087483 EJ For-Sale Bother ACR 49 35 NC(=O)c1ccc(OCC(=O)N2CCN(C(=O)Cc3ccccc3)CC2)cc1 ZINC000147087493 GD On-Demand Anodyne HTR1D 17 44 NC(=O)c1ccc(OCC(=O)N2CCN(C(=O)Cc3ccccc3)CC2)cc1 ZINC000147087493 GD On-Demand Anodyne HTR1B 19 44 NC(=O)c1ccc(OCC(=O)N2CCN(C(=O)Cc3ccccc3)CC2)cc1 ZINC000147087493 GD On-Demand Anodyne LTA4H 40 38 NC(=O)c1ccc(OCC(=O)N2CCN(C(=O)Cc3ccccc3)CC2)cc1 ZINC000147087493 GD On-Demand Anodyne CPT1A 87 51 NC(=O)c1ccc(OCC(=O)N2CCN(C(=O)Cc3ccccc3)CC2)cc1 ZINC000147087493 GD On-Demand Anodyne CPT2 42 35 NC(=O)c1ccc(OCC(=O)N2CCN(C(=O)Cc3ccccc3)CC2)cc1 ZINC000147087493 GD On-Demand Anodyne PLA2G4B 59 42 N#CC1CCN(C(=O)Cc2csc(-c3cccc(F)c3)n2)CC1 ZINC000147087643 EG On-Demand Mild ETHR 57 44 CCC(=O)Nc1ccc(Cl)c(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147087655 FE On-Demand Anodyne ENV 41 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087667 FD On-Demand Anodyne CCR3 55 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087667 FD On-Demand Anodyne HDAC10 50 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087667 FD On-Demand Anodyne HDAC2 30 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087667 FD On-Demand Anodyne HDAC3 32 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087667 FD On-Demand Anodyne HDAC6 25 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147087667 FD On-Demand Anodyne HDAC11 44 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(OCc3ccccn3)c2)c1 ZINC000147087861 GH On-Demand Bother MMP13 27 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(OCc3ccccn3)c2)c1 ZINC000147087861 GH On-Demand Bother ROCK1 26 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(OCc3ccccn3)c2)c1 ZINC000147087861 GH On-Demand Bother MTNR1B 15 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(OCc3ccccn3)c2)c1 ZINC000147087861 GH On-Demand Bother ROCK2 28 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(OCc3ccccn3)c2)c1 ZINC000147087861 GH On-Demand Bother TAAR1 19 41 CCOP(=O)(CCN1CCC(CNC(=O)c2cc(Cl)c(N)cc2OC)CC1)OCC ZINC000147087885 JH For-Sale Anodyne DRD2 38 42 CCOP(=O)(CCN1CCC(CNC(=O)c2cc(Cl)c(N)cc2OC)CC1)OCC ZINC000147087885 JH For-Sale Anodyne DRD3 18 63 CCOP(=O)(CCN1CCC(CNC(=O)c2cc(Cl)c(N)cc2OC)CC1)OCC ZINC000147087885 JH For-Sale Anodyne HTR4 171 75 CCOP(=O)(CCN1CCC(CNC(=O)c2cc(Cl)c(N)cc2OC)CC1)OCC ZINC000147087885 JH For-Sale Anodyne CACNA1I 77 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne F2 63 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne PLG 33 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne ACE 62 44 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne OPRM1 25 45 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne GHRHR 41 32 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne P2RY12 180 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne TRHR 59 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne HLA-DRB3 56 39 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne CTRA_BOVIN 41 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne PRCP 28 45 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne TRY1_BOVIN 92 38 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne NTSR1 76 36 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne NTSR2 43 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne CTSK 42 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne ADAM17 19 48 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne DPP4 19 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne ACE2 38 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne C5AR1 15 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne TPP2 47 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne XIAP 49 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne BRCA1 44 31 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147087914 DF On-Demand Anodyne TMPRSS11D 54 35 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)N[C@H]1CCCC[C@H]1C ZINC000147087966 HH On-Demand Anodyne CASR 16 40 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc([N+](=O)[O-])cc1 ZINC000147088024 EF On-Demand Mild KCNMA1 20 44 N#CC1CCN(C(=O)Cc2csc(-c3ccc(Cl)cc3)n2)CC1 ZINC000147088055 EH On-Demand Mild ETHR 41 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne F2 63 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne PLG 33 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne ACE 62 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne OPRM1 25 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne GHRHR 41 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne P2RY12 180 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne TRHR 59 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne BDKRB2 44 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne HLA-DRB3 56 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne CTRA_BOVIN 41 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne PRCP 28 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne TRY1_BOVIN 92 38 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne CCKAR 15 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne NTSR1 76 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne NTSR2 43 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne CTSK 42 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne ADAM17 53 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne DPP4 19 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne ACE2 38 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne C5AR1 27 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne TPP2 47 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne XIAP 49 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne BRCA1 44 31 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccccc1 ZINC000147088114 DF On-Demand Anodyne TMPRSS11D 54 35 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne PTGFR 24 44 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne PTGER2 41 48 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne PTGER4 19 49 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne FABP4 15 69 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne FAAH 21 54 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne S1PR2 15 40 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne LPAR3 27 40 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne FABP3 54 69 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne FABP5 23 69 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne FABP1 23 69 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne NOD1 71 42 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne OXER1 35 53 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne CQSS 66 42 CCCCCCCC[C@H](O)/C=C\CCCCCCC(=O)O ZINC000147088129 CK For-Sale Anodyne SLCO2A1 74 51 C[C@H](OC[C@@H]1CCCO1)C(=O)NCCNc1ccccc1[N+](=O)[O-] ZINC000147088135 ED On-Demand Bother COLA 83 33 COc1ccc(C#N)cc1N[C@@H](C)C(=O)Nc1ccccc1[N+](=O)[O-] ZINC000147088188 EF On-Demand Mild COLA 71 33 COc1ccc(C#N)cc1N[C@@H](C)C(=O)Nc1ccccc1[N+](=O)[O-] ZINC000147088188 EF On-Demand Mild KCNMA1 24 44 NC(=O)c1ccc(OCC(=O)NCCN2CCCCC2)cc1 ZINC000147088246 DC On-Demand Anodyne DRD4 43 33 NC(=O)c1ccc(OCC(=O)NCCN2CCCCC2)cc1 ZINC000147088246 DC On-Demand Anodyne LTA4H 40 38 NC(=O)c1ccc(OCC(=O)NCCN2CCCCC2)cc1 ZINC000147088246 DC On-Demand Anodyne HRH3 52 46 NC(=O)c1ccc(OCC(=O)NCCN2CCCCC2)cc1 ZINC000147088246 DC On-Demand Anodyne CHRNA7 23 40 NC(=O)c1ccc(OCC(=O)NCCN2CCCCC2)cc1 ZINC000147088246 DC On-Demand Anodyne HNMT 55 34 NC(=O)c1ccc(OCC(=O)NCCN2CCCCC2)cc1 ZINC000147088246 DC On-Demand Anodyne PSMB2 56 45 NC(=O)c1ccc(OCC(=O)NCCN2CCCCC2)cc1 ZINC000147088246 DC On-Demand Anodyne PSMB1 49 45 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne F2 63 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne PLG 33 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne ACE 62 44 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne OPRM1 25 45 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne GHRHR 41 32 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne P2RY12 180 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne TRHR 59 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne BDKRB2 44 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne HLA-DRB3 56 39 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne CTRA_BOVIN 41 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne PRCP 28 45 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne TRY1_BOVIN 92 38 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne CCKAR 15 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne NTSR1 76 36 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne NTSR2 43 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne CTSK 42 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne ADAM17 53 45 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne DPP4 19 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne ACE2 38 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne C5AR1 27 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne TPP2 47 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne XIAP 49 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne BRCA1 44 31 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088314 DF On-Demand Anodyne TMPRSS11D 54 35 C[C@@H](OC[C@@H]1CCCO1)C(=O)NCCNc1ccccc1[N+](=O)[O-] ZINC000147088342 ED On-Demand Bother COLA 83 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne F2 63 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne PLG 33 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne ACE 62 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne OPRM1 25 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne GHRHR 41 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne P2RY12 180 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne TRHR 59 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne HLA-DRB3 56 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne CTRA_BOVIN 41 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne PRCP 28 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne TRY1_BOVIN 92 38 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne NTSR1 76 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne NTSR2 43 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne CTSK 42 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne ADAM17 19 48 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne DPP4 19 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne ACE2 38 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne C5AR1 15 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne TPP2 47 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne XIAP 49 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne BRCA1 44 31 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccccc1 ZINC000147088517 DF On-Demand Anodyne TMPRSS11D 54 35 Cc1cc(C)cc(NC(=O)CS(=O)(=O)[C@H](C)c2ccc(OC(F)(F)F)cc2)c1 ZINC000147088528 HI On-Demand Anodyne SCN10A 35 47 C[C@H](OC[C@H]1CCCO1)C(=O)NCCNc1ccccc1[N+](=O)[O-] ZINC000147088531 ED On-Demand Bother COLA 83 33 C[C@@H](CNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1)N1CCCC1 ZINC000147088553 HF On-Demand Anodyne ADRB2 17 40 C[C@@H](CNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1)N1CCCC1 ZINC000147088553 HF On-Demand Anodyne ADRB1 24 40 C[C@@H](CNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1)N1CCCC1 ZINC000147088553 HF On-Demand Anodyne ADRB3 50 40 C[C@@H](CNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1)N1CCCC1 ZINC000147088553 HF On-Demand Anodyne HTR6 17 41 C[C@@H](CNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1)N1CCCC1 ZINC000147088553 HF On-Demand Anodyne CACNA1G 20 41 C[C@@H](CNC(=O)Cc1ccc(NS(=O)(=O)c2ccc(F)cc2)cc1)N1CCCC1 ZINC000147088553 HF On-Demand Anodyne LIMK2 41 45 C[C@@H](OC[C@H]1CCCO1)C(=O)NCCNc1ccccc1[N+](=O)[O-] ZINC000147088706 ED On-Demand Bother COLA 83 33 Cc1cscc1CNc1nc(N)nc(N(C)C)n1 ZINC000147088765 CD For-Sale Anodyne AT1 0 48 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000147088828 DE On-Demand Anodyne MMP13 21 49 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000147088828 DE On-Demand Anodyne MMP2 17 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000147088828 DE On-Demand Anodyne MMP14 15 49 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000147088828 DE On-Demand Anodyne MMP9 15 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000147088828 DE On-Demand Anodyne MMP7 16 49 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000147088828 DE On-Demand Anodyne ADAMTS4 55 37 COc1ccc(-c2nc(C(=O)N3CCC(C#N)CC3)cs2)cc1OC ZINC000147088876 FG On-Demand Mild TRPC6 72 44 COc1ccc(-c2nc(C(=O)N3CCC(C#N)CC3)cs2)cc1OC ZINC000147088876 FG On-Demand Mild TRPC3 48 44 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1ccccc1 ZINC000147088913 HI On-Demand Anodyne LTA4H 33 40 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1ccccc1 ZINC000147088913 HI On-Demand Anodyne P2RY1 58 38 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1ccccc1 ZINC000147088913 HI On-Demand Anodyne EPHX2 42 39 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1ccccc1 ZINC000147088913 HI On-Demand Anodyne KCNK3 15 40 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1ccccc1 ZINC000147088913 HI On-Demand Anodyne KCNK9 21 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147088933 GH On-Demand Anodyne CHRNA7 21 44 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147088933 GH On-Demand Anodyne MTNR1A 18 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147088933 GH On-Demand Anodyne MTNR1B 21 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147088933 GH On-Demand Anodyne ROCK2 57 47 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147088933 GH On-Demand Anodyne FAAH 21 52 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147088933 GH On-Demand Anodyne FFAR1 35 43 C[C@H](Nc1nccc(Nc2cc(C3CC3)[nH]n2)n1)c1nc2cc[nH]c2cc1Cl ZINC000147088946 GJ Annotated Anodyne NTRK1 26 59 C[C@H](Nc1nccc(Nc2cc(C3CC3)[nH]n2)n1)c1nc2cc[nH]c2cc1Cl ZINC000147088946 GJ Annotated Anodyne PAK3 28 63 C[C@H](Nc1nccc(Nc2cc(C3CC3)[nH]n2)n1)c1nc2cc[nH]c2cc1Cl ZINC000147088946 GJ Annotated Anodyne PAK1 50 63 C[C@H](Nc1nccc(Nc2cc(C3CC3)[nH]n2)n1)c1nc2cc[nH]c2cc1Cl ZINC000147088946 GJ Annotated Anodyne PAK2 39 63 C[C@H](Nc1nccc(Nc2cc(C3CC3)[nH]n2)n1)c1nc2cc[nH]c2cc1Cl ZINC000147088946 GJ Annotated Anodyne PKNB 88 52 CCNC(=O)c1ccc(C)c(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147089013 FG On-Demand Anodyne MAPK14 46 50 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne HTR1A 16 49 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne DRD2 17 52 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne HTR2A 22 79 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne SLC6A4 37 53 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne HRH1 17 54 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne SLC6A3 58 53 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne GRIN2B 15 43 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne SIGMAR1 27 53 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne CCR3 28 40 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne CCR5 19 79 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne SLC18A3 18 51 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne GRIN2C 17 43 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne CACNA1G 27 46 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne CYP2J2 71 50 O[C@@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089109 IK Annotated Anodyne MEN1 52 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147089120 GH On-Demand Anodyne CHRNA7 21 44 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147089120 GH On-Demand Anodyne MTNR1A 18 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147089120 GH On-Demand Anodyne MTNR1B 21 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147089120 GH On-Demand Anodyne ROCK2 57 47 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147089120 GH On-Demand Anodyne FAAH 21 52 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(OCc3cccnc3)c1)C2 ZINC000147089120 GH On-Demand Anodyne FFAR1 35 43 C[C@H](Nc1nccc(Nc2cc([C@@H]3C[C@@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147089142 GH Annotated Anodyne NTRK1 21 52 C[C@H](Nc1nccc(Nc2cc([C@@H]3C[C@@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147089142 GH Annotated Anodyne PAK3 27 56 C[C@H](Nc1nccc(Nc2cc([C@@H]3C[C@@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147089142 GH Annotated Anodyne PAK1 49 56 C[C@H](Nc1nccc(Nc2cc([C@@H]3C[C@@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147089142 GH Annotated Anodyne PAK2 37 56 C[C@H](Nc1nccc(Nc2cc([C@@H]3C[C@@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147089142 GH Annotated Anodyne PKNB 47 43 CCCC[C@@H](SCCCO)C(=O)O ZINC000147089145 BD For-Sale Anodyne SLC22A20 0 44 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccccc1C ZINC000147089196 DG On-Demand Mild P2RX7 27 42 CCNC(=O)c1ccc(C)c(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147089243 HE On-Demand Bother MAPK14 23 46 C[C@@H](CN1CCOCC1)NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147089286 DC On-Demand Anodyne PTGDS 19 40 O=C1c2ccccc2C(=O)N1Nc1ncnc2scc(-c3cccs3)c12 ZINC000147089298 GI Annotated Anodyne FLT3 17 47 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne HTR1A 16 49 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne DRD2 17 52 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne HTR2A 22 79 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne SLC6A4 37 53 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne HRH1 17 54 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne SLC6A3 58 53 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne GRIN2B 15 43 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne SIGMAR1 27 53 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne CCR3 28 40 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne CCR5 19 79 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne SLC18A3 18 51 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne GRIN2C 17 43 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne CACNA1G 27 46 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne CYP2J2 71 50 O[C@H](CCCN1CCC(C(O)(c2ccccc2)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147089306 IK Annotated Anodyne MEN1 52 40 CCCC[C@H](SCCCO)C(=O)O ZINC000147089329 BD For-Sale Anodyne SLC22A20 0 44 N#CC1CCN(C(=O)Cc2csc(NC(=O)c3ccco3)n2)CC1 ZINC000147089473 EE On-Demand Mild KISS1R 44 33 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147089478 HI On-Demand Bother PDE4A 33 43 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147089478 HI On-Demand Bother PDE4B 15 43 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147089478 HI On-Demand Bother PDE4D 15 43 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147089478 HI On-Demand Bother PDE4C 15 43 C[C@H](CN1CCOCC1)NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147089492 DC On-Demand Anodyne PTGDS 19 40 C[C@H](Nc1nccc(Nc2cc([C@@H]3C[C@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147089518 GH Annotated Anodyne NTRK1 21 52 C[C@H](Nc1nccc(Nc2cc([C@@H]3C[C@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147089518 GH Annotated Anodyne PAK3 27 56 C[C@H](Nc1nccc(Nc2cc([C@@H]3C[C@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147089518 GH Annotated Anodyne PAK1 49 56 C[C@H](Nc1nccc(Nc2cc([C@@H]3C[C@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147089518 GH Annotated Anodyne PAK2 37 56 C[C@H](Nc1nccc(Nc2cc([C@@H]3C[C@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147089518 GH Annotated Anodyne PKNB 47 43 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147089602 FD On-Demand Mild CA2 43 51 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147089602 FD On-Demand Mild CA1 52 51 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147089602 FD On-Demand Mild CA7 23 48 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147089602 FD On-Demand Mild CA4 37 40 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147089602 FD On-Demand Mild CA14 36 47 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147089602 FD On-Demand Mild CA12 51 48 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147089602 FD On-Demand Mild CA9 51 46 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147089602 FD On-Demand Mild UREA_CANEN 27 42 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147089602 FD On-Demand Mild MTCA1 41 51 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147089602 FD On-Demand Mild P96878_MYCTU 51 51 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)c(F)c1 ZINC000147089630 CD On-Demand Anodyne LEF 58 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147089666 HI On-Demand Bother PDE4A 33 43 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147089666 HI On-Demand Bother PDE4B 15 43 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147089666 HI On-Demand Bother PDE4D 15 43 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccc(OC3CCCC3)c(OC)c2)c1 ZINC000147089666 HI On-Demand Bother PDE4C 15 43 CCOC(=O)[C@@H](CCc1ccccc1)[C@@]1(C(=O)O)CCCN1C(=O)[C@H](C)N ZINC000147089746 GD For-Sale Anodyne ACE 47 44 CCOC(=O)[C@@H](CCc1ccccc1)[C@@]1(C(=O)O)CCCN1C(=O)[C@H](C)N ZINC000147089746 GD For-Sale Anodyne GHRHR 49 34 CCOC(=O)[C@@H](CCc1ccccc1)[C@@]1(C(=O)O)CCCN1C(=O)[C@H](C)N ZINC000147089746 GD For-Sale Anodyne SLC12A5 75 38 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1cccc(OC(F)F)c1 ZINC000147089831 FF On-Demand Anodyne ACACA 45 38 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1cccc(OC(F)F)c1 ZINC000147089831 FF On-Demand Anodyne F7 28 47 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1cccc(OC(F)F)c1 ZINC000147089831 FF On-Demand Anodyne AOC3 19 48 COc1ccc([N+](=O)[O-])c(C(=O)NCC2(c3ccc(F)cc3)CCCC2)c1 ZINC000147089864 FH On-Demand Bother KCNA3 42 41 COc1ccc([N+](=O)[O-])c(C(=O)NCC2(c3ccc(F)cc3)CCCC2)c1 ZINC000147089864 FH On-Demand Bother NMBR 61 41 COc1ccc([N+](=O)[O-])c(C(=O)NCC2(c3ccc(F)cc3)CCCC2)c1 ZINC000147089864 FH On-Demand Bother TAAR1 21 40 CC(=O)N[C@@H]1CCN(c2ccc(C(F)(F)F)cn2)C1 ZINC000147089950 CD On-Demand Anodyne EPHX2 15 40 CC(=O)N[C@@H]1CCN(c2ccc(C(F)(F)F)cn2)C1 ZINC000147089950 CD On-Demand Anodyne CXCR3 17 42 CC(=O)N[C@@H]1CCN(c2ccc(C(F)(F)F)cn2)C1 ZINC000147089950 CD On-Demand Anodyne LIPG 51 41 CC(=O)N[C@@H]1CCN(c2ccc(C(F)(F)F)cn2)C1 ZINC000147089950 CD On-Demand Anodyne HPGDS 28 41 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1ccccc1F ZINC000147089991 HI On-Demand Anodyne P2RY1 55 36 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1cccc(OC(F)F)c1 ZINC000147090008 FF On-Demand Anodyne ACACA 45 38 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1cccc(OC(F)F)c1 ZINC000147090008 FF On-Demand Anodyne F7 28 47 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1cccc(OC(F)F)c1 ZINC000147090008 FF On-Demand Anodyne AOC3 19 48 COC(=O)c1ccc(CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147090035 EF On-Demand Bother U38 0 44 C[C@@H](CNC(=O)c1ccc(CN2CCCCC2)cc1)N1CCCC1 ZINC000147090105 EF On-Demand Anodyne ACHE 15 46 C[C@@H](CNC(=O)c1ccc(CN2CCCCC2)cc1)N1CCCC1 ZINC000147090105 EF On-Demand Anodyne HRH3 22 46 C[C@@H](CNC(=O)c1ccc(CN2CCCCC2)cc1)N1CCCC1 ZINC000147090105 EF On-Demand Anodyne SIGMAR1 15 43 C[C@@H](CNC(=O)c1ccc(CN2CCCCC2)cc1)N1CCCC1 ZINC000147090105 EF On-Demand Anodyne CACNA1G 31 40 C[C@@H](CNC(=O)c1ccc(CN2CCCCC2)cc1)N1CCCC1 ZINC000147090105 EF On-Demand Anodyne NOD2 42 36 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1ccccc1F ZINC000147090168 HI On-Demand Anodyne P2RY1 55 36 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1cccc(C)c1 ZINC000147090172 DG On-Demand Mild SCN10A 20 48 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1cccc(C)c1 ZINC000147090172 DG On-Demand Mild KCNK3 55 39 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1cccc(C)c1 ZINC000147090172 DG On-Demand Mild KCNK9 65 39 COCc1nc(C(=O)Nc2ccc(OC(F)(F)F)cc2)cs1 ZINC000147090240 EG On-Demand Anodyne P2RY1 40 34 COCc1nc(C(=O)Nc2ccc(OC(F)(F)F)cc2)cs1 ZINC000147090240 EG On-Demand Anodyne EPHX2 51 44 COCc1nc(C(=O)Nc2ccc(OC(F)(F)F)cc2)cs1 ZINC000147090240 EG On-Demand Anodyne SCN10A 38 55 COCc1nc(C(=O)Nc2ccc(OC(F)(F)F)cc2)cs1 ZINC000147090240 EG On-Demand Anodyne Q8MMZ8_EIMTE 23 44 COCc1nc(C(=O)Nc2ccc(OC(F)(F)F)cc2)cs1 ZINC000147090240 EG On-Demand Anodyne SHH 43 35 N#Cc1cn(-c2ccc(C(=O)O)cc2)cc1OCc1ccccc1 ZINC000147090253 DH Annotated Anodyne SRD5A2 20 47 N#Cc1cn(-c2ccc(C(=O)O)cc2)cc1OCc1ccccc1 ZINC000147090253 DH Annotated Anodyne PTGER2 17 49 N#Cc1cn(-c2ccc(C(=O)O)cc2)cc1OCc1ccccc1 ZINC000147090253 DH Annotated Anodyne XDH 19 47 N#Cc1cn(-c2ccc(C(=O)O)cc2)cc1OCc1ccccc1 ZINC000147090253 DH Annotated Anodyne PPIA 32 41 N#Cc1cn(-c2ccc(C(=O)O)cc2)cc1OCc1ccccc1 ZINC000147090253 DH Annotated Anodyne PTGER1 54 49 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)NCc3ccccn3)c2)c1 ZINC000147090254 HG On-Demand Bother DRD4 40 31 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)NCc3ccccn3)c2)c1 ZINC000147090254 HG On-Demand Bother TAAR1 36 49 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)NCc3ccccn3)c2)c1 ZINC000147090254 HG On-Demand Bother AKR1C3 18 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)NCc3ccccn3)c2)c1 ZINC000147090254 HG On-Demand Bother KCNK3 94 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)NCc3ccccn3)c2)c1 ZINC000147090254 HG On-Demand Bother KCNK9 69 37 CC(C)(C)C(=O)N1CCC(NC(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147090272 FD On-Demand Anodyne SLC6A5 33 42 CC(C)(C)C(=O)N1CCC(NC(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147090272 FD On-Demand Anodyne PLAU 23 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090284 FC On-Demand Anodyne KLK3 48 35 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090284 FC On-Demand Anodyne GRIA1 52 32 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090284 FC On-Demand Anodyne PCSK5 57 36 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090284 FC On-Demand Anodyne FURIN 63 38 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090284 FC On-Demand Anodyne POLG_WNV 77 35 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090284 FC On-Demand Anodyne NPFFR1 54 37 C[C@H](CNC(=O)c1ccc(CN2CCCCC2)cc1)N1CCCC1 ZINC000147090295 EF On-Demand Anodyne ACHE 15 46 C[C@H](CNC(=O)c1ccc(CN2CCCCC2)cc1)N1CCCC1 ZINC000147090295 EF On-Demand Anodyne HRH3 22 46 C[C@H](CNC(=O)c1ccc(CN2CCCCC2)cc1)N1CCCC1 ZINC000147090295 EF On-Demand Anodyne SIGMAR1 15 43 C[C@H](CNC(=O)c1ccc(CN2CCCCC2)cc1)N1CCCC1 ZINC000147090295 EF On-Demand Anodyne CACNA1G 31 40 C[C@H](CNC(=O)c1ccc(CN2CCCCC2)cc1)N1CCCC1 ZINC000147090295 EF On-Demand Anodyne NOD2 42 36 COC(=O)c1cc(N)c(N)c([N+](=O)[O-])c1 ZINC000147090303 BC In-Stock Bother TPMT 0 44 CC(=O)N1C[C@@H](N2CCN(c3cc(C)nn3-c3ccccc3)CC2)C[C@H]1C(=O)N1CCSC1 ZINC000147090344 JD For-Sale Anodyne DPP4 36 68 CC(=O)N1C[C@@H](N2CCN(c3cc(C)nn3-c3ccccc3)CC2)C[C@H]1C(=O)N1CCSC1 ZINC000147090344 JD For-Sale Anodyne DPP9 15 68 CCOC[C@H](C)NS(=O)(=O)c1ccc2c(c1)CCCC(=O)N2 ZINC000147090400 ED On-Demand Anodyne PKM 45 47 CCOC[C@H](C)NS(=O)(=O)c1ccc2c(c1)CCCC(=O)N2 ZINC000147090400 ED On-Demand Anodyne MGAT1 44 32 CCOc1ccc(N2C(=O)c3ccc(C(=O)N4CCC(C#N)CC4)cc3C2=O)cc1 ZINC000147090411 HG On-Demand Mild AVPR1A 19 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090462 FC On-Demand Anodyne KLK3 48 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090462 FC On-Demand Anodyne GRIA1 52 32 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090462 FC On-Demand Anodyne PCSK5 57 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090462 FC On-Demand Anodyne FURIN 63 38 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090462 FC On-Demand Anodyne POLG_WNV 77 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N(C)C ZINC000147090462 FC On-Demand Anodyne NPFFR1 54 37 COC(=O)c1cc2cc(NC(=O)c3cc(OC)ccc3[N+](=O)[O-])ccc2o1 ZINC000147090471 FG On-Demand Bother TAAR1 25 41 Cc1ccccc1CNC(=O)CS(=O)(=O)[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147090543 HH On-Demand Anodyne TRPV1 53 34 Cc1ccccc1CNC(=O)CS(=O)(=O)[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147090543 HH On-Demand Anodyne SCN10A 36 48 N#CC1CCN(C(=O)c2ccc3c(c2)C(=O)N(Cc2ccncc2)C3=O)CC1 ZINC000147090612 FE On-Demand Mild L3MBTL3 42 35 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccccc2OC(C)C)c1 ZINC000147090706 FH On-Demand Bother TAAR1 22 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccccc2OC(C)C)c1 ZINC000147090706 FH On-Demand Bother AKR1C2 19 42 O=C1C[C@H](c2ccccc2)N(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CCN1 ZINC000147090747 FH On-Demand Anodyne MDM2 63 31 O=C(O)[C@@]1(O)CCN(Cc2ccccc2)C1=O ZINC000147090765 BC For-Sale Anodyne NPFFR1 49 37 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)N1CCc2ccccc21 ZINC000147090772 HH On-Demand Anodyne P2RY1 45 42 Cc1nc2cc(C(=O)N3CCC(C#N)CC3)ccc2n1-c1ccccc1 ZINC000147090832 EH On-Demand Mild HPD 40 35 Cc1nc2cc(C(=O)N3CCC(C#N)CC3)ccc2n1-c1ccccc1 ZINC000147090832 EH On-Demand Mild L3MBTL3 49 36 Cc1nc2cc(C(=O)N3CCC(C#N)CC3)ccc2n1-c1ccccc1 ZINC000147090832 EH On-Demand Mild HPGD 52 44 O=C1[C@H]2[C@@H]3C=C[C@H](CC3)[C@H]2C(=O)N1c1ccc(I)cc1 ZINC000147090833 GF In-Stock Anodyne WNT3 17 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccccc2OC(C)C)c1 ZINC000147090892 FH On-Demand Bother TAAR1 22 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccccc2OC(C)C)c1 ZINC000147090892 FH On-Demand Bother AKR1C2 19 42 CCOC(=O)c1ccccc1NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147090933 EG On-Demand Bother CCR3 17 40 CN(C)CCCn1c(NC(=O)c2ccc3cc4n(c3n2)CC(C)(C)CNC4=O)nc2ccccc21 ZINC000147090971 JG Annotated Anodyne RPS6KA3 42 78 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(=O)(=O)NC(C)C)cc1 ZINC000147090991 HF On-Demand Mild MMP13 32 44 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(=O)(=O)NC(C)C)cc1 ZINC000147090991 HF On-Demand Mild MMP2 19 44 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1ccc(S(=O)(=O)NC(C)C)cc1 ZINC000147090991 HF On-Demand Mild MMP7 17 44 Clc1ccc(N2CCCCC2)cc1Cl ZINC000147091029 BH For-Sale Anodyne SIGMAR1 18 43 Clc1ccc(N2CCCCC2)cc1Cl ZINC000147091029 BH For-Sale Anodyne CHRNA4 32 40 Clc1ccc(N2CCCCC2)cc1Cl ZINC000147091029 BH For-Sale Anodyne BCL2A1 57 40 CCCOCC(=O)N1CCc2[nH]c3ccccc3c2C1 ZINC000147091083 CE On-Demand Anodyne DRD5 19 41 CCCOCC(=O)N1CCc2[nH]c3ccccc3c2C1 ZINC000147091083 CE On-Demand Anodyne SSTR4 40 33 O=C1C[C@H](c2ccccc2)N(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CCN1 ZINC000147091117 FH On-Demand Anodyne MDM2 63 31 CN(C)Cc1cccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)c1 ZINC000147091216 GG On-Demand Anodyne ROCK2 21 51 N#CC1CCN(C(=O)c2ccc(NCc3ccccc3Cl)c([N+](=O)[O-])c2)CC1 ZINC000147091256 GI On-Demand Mild PRKCQ 25 41 N#CC1CCN(C(=O)c2ccc(NCc3ccccc3Cl)c([N+](=O)[O-])c2)CC1 ZINC000147091256 GI On-Demand Mild L3MBTL3 40 43 CCCCO[C@@H](C)C(=O)N1CCc2[nH]c3ccccc3c2C1 ZINC000147091292 DG On-Demand Anodyne SSTR4 45 34 CCCCO[C@@H](C)C(=O)N1CCc2[nH]c3ccccc3c2C1 ZINC000147091292 DG On-Demand Anodyne NR1H4 21 44 CC(C)(C)[C@H](NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1)c1ccc(F)cc1 ZINC000147091293 HH On-Demand Bother CTSF 47 32 Cc1cccc(NS(=O)(=O)c2ccc(C)c(C(=O)NC[C@@H](C)N3CCCC3)c2)c1 ZINC000147091331 HG On-Demand Anodyne PKM 18 40 Cc1cccc(NS(=O)(=O)c2ccc(C)c(C(=O)NC[C@@H](C)N3CCCC3)c2)c1 ZINC000147091331 HG On-Demand Anodyne LIMK2 26 43 CN(C)CCCn1c(NC(=O)c2ccc3cc4n(c3n2)CCCNC4=O)nc2ccccc21 ZINC000147091378 IF Annotated Anodyne ITK 40 35 CN(C)CCCn1c(NC(=O)c2ccc3cc4n(c3n2)CCCNC4=O)nc2ccccc21 ZINC000147091378 IF Annotated Anodyne RPS6KA3 96 61 CN(C)Cc1cccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)c1 ZINC000147091415 GG On-Demand Anodyne ROCK2 21 51 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)Nc1ccc(F)cc1 ZINC000147091419 HH On-Demand Anodyne P2RY1 53 38 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)Nc1ccc(F)cc1 ZINC000147091419 HH On-Demand Anodyne CTSS 15 40 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)Nc1ccc(F)cc1 ZINC000147091419 HH On-Demand Anodyne EPHX2 53 43 O=C(NCCc1cccs1)[C@@H]1CCN(c2cccc(Cl)c2)C1=O ZINC000147091442 EG On-Demand Anodyne ADAM17 37 53 CCCCO[C@H](C)C(=O)N1CCc2[nH]c3ccccc3c2C1 ZINC000147091487 DG On-Demand Anodyne SSTR4 45 34 CCCCO[C@H](C)C(=O)N1CCc2[nH]c3ccccc3c2C1 ZINC000147091487 DG On-Demand Anodyne NR1H4 21 44 CC(C)(C)[C@@H](NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1)c1ccc(F)cc1 ZINC000147091497 HH On-Demand Bother CTSF 47 32 CCOC[C@H](C)NS(=O)(=O)c1ccc(C)c(F)c1 ZINC000147091559 CD On-Demand Anodyne LEF 67 45 O=C(NCCc1cccs1)[C@H]1CCN(c2cccc(Cl)c2)C1=O ZINC000147091623 EG On-Demand Anodyne ADAM17 37 53 CCc1ccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)cc1 ZINC000147091647 HI On-Demand Anodyne GCGR 15 41 CCc1ccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)cc1 ZINC000147091647 HI On-Demand Anodyne P2RY1 46 35 CCc1ccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)cc1 ZINC000147091647 HI On-Demand Anodyne EPHX2 45 43 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)c1cccnc1SC(F)(F)F ZINC000147091694 GI On-Demand Anodyne MAPK11 44 59 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)c1cccnc1SC(F)(F)F ZINC000147091694 GI On-Demand Anodyne MAPK14 77 59 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)c1cccnc1SC(F)(F)F ZINC000147091694 GI On-Demand Anodyne MAPK13 74 38 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)c1cccnc1SC(F)(F)F ZINC000147091694 GI On-Demand Anodyne G2YM83_BOTF4 53 35 Cc1nn(C(F)F)c(C)c1CC(=O)N1CCc2[nH]c3ccccc3c2C1 ZINC000147091716 FH On-Demand Anodyne SSTR4 45 34 CCc1ccc(NC(=O)CS(=O)(=O)[C@H](C)c2ccc(OC(F)(F)F)cc2)cc1 ZINC000147091836 HI On-Demand Anodyne GCGR 15 41 CCc1ccc(NC(=O)CS(=O)(=O)[C@H](C)c2ccc(OC(F)(F)F)cc2)cc1 ZINC000147091836 HI On-Demand Anodyne P2RY1 46 35 CCc1ccc(NC(=O)CS(=O)(=O)[C@H](C)c2ccc(OC(F)(F)F)cc2)cc1 ZINC000147091836 HI On-Demand Anodyne EPHX2 45 43 Nc1ccn2c(-c3cccc(NC(=O)NCC(F)(F)F)c3)cnc2c1 ZINC000147091837 EG Annotated Anodyne BRAF 40 39 Nc1ccn2c(-c3cccc(NC(=O)NCC(F)(F)F)c3)cnc2c1 ZINC000147091837 EG Annotated Anodyne RIPK1 51 37 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147091909 HE On-Demand Bother MAPK11 39 45 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147091909 HE On-Demand Bother MAPK14 50 45 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147091909 HE On-Demand Bother MAPK13 69 35 c1ccc(COCc2ccc(COCc3ccccc3)cc2)cc1 ZINC000147092013 DK For-Sale Anodyne TAAR1 22 45 COc1ccccc1NC(=O)CS(=O)(=O)[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147092014 HH On-Demand Anodyne P2RY1 55 40 COc1ccc(Cl)cc1NC(=O)[C@@H](C)Nc1cc(C#N)ccc1OC ZINC000147092018 FH On-Demand Mild RBP4 23 40 COCc1nc(C(=O)N2CCN(C(=O)c3ccco3)CC2)cs1 ZINC000147092175 ED On-Demand Anodyne ALDH1A1 18 42 COCc1nc(C(=O)N2CCN(C(=O)c3ccco3)CC2)cs1 ZINC000147092175 ED On-Demand Anodyne TRPC6 65 38 CC(C)(C)OC(=O)N1CCC=C(C=O)C1 ZINC000147092199 BD For-Sale Reactive GPR119 35 40 Cc1ccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)cc1F ZINC000147092209 HI On-Demand Anodyne MCHR1 15 43 CN(C)S(=O)(=O)c1ccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)cc1 ZINC000147092318 HE On-Demand Anodyne NAMPT 62 40 Cc1ccc(NC(=O)CS(=O)(=O)[C@H](C)c2ccc(OC(F)(F)F)cc2)cc1F ZINC000147092404 HI On-Demand Anodyne MCHR1 15 43 COc1ccc(C#N)cc1N[C@@H](C)C(=O)Nc1ccc2c(c1)OCO2 ZINC000147092412 EF On-Demand Mild EDNRB 19 42 O=C(Nc1ccc(F)cc1)C1CCN(c2ccnc3ccc(Br)cc23)CC1 ZINC000147092511 IJ On-Demand Anodyne MAPK10 16 43 O=C(Nc1ccc(F)cc1)C1CCN(c2ccnc3ccc(Br)cc23)CC1 ZINC000147092511 IJ On-Demand Anodyne LIMK2 21 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147092535 GD On-Demand Bother BMP1 86 44 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147092535 GD On-Demand Bother MMP13 46 44 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147092535 GD On-Demand Bother COLA 48 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147092535 GD On-Demand Bother MMP2 19 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147092535 GD On-Demand Bother MMP8 33 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147092535 GD On-Demand Bother MMP9 45 44 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147092535 GD On-Demand Bother CA9 19 45 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147092535 GD On-Demand Bother MMP1 44 44 CCc1cccc(NC(=O)CS(=O)(=O)[C@H](C)c2ccc(OC(F)(F)F)cc2)c1 ZINC000147092623 HI On-Demand Anodyne SCN10A 23 40 CCc1cccc(NC(=O)CS(=O)(=O)[C@H](C)c2ccc(OC(F)(F)F)cc2)c1 ZINC000147092623 HI On-Demand Anodyne KCNK9 25 40 COc1ccc(C#N)cc1N[C@H](C)C(=O)Nc1cccc(C#N)c1 ZINC000147092633 DF On-Demand Mild CCR3 15 41 Cc1cccc(C)c1OC[C@H](O)CNC(=O)Nc1cccc(CN(C)C)c1 ZINC000147092657 FF On-Demand Anodyne ADRB1 45 36 CCCCO[C@@H](C)C(=O)Nc1cc(C(N)=O)ccc1N1CCCC1 ZINC000147092721 EF On-Demand Anodyne KCNQ2 83 42 CCCCO[C@@H](C)C(=O)Nc1cc(C(N)=O)ccc1N1CCCC1 ZINC000147092721 EF On-Demand Anodyne KCNQ4 0 41 CCOC[C@H](C)NS(=O)(=O)c1cc(C)ccc1F ZINC000147092766 CD On-Demand Anodyne LEF 48 40 O=C(Nc1cccnc1N1CCCC1)c1csc(-c2ccccc2F)n1 ZINC000147092823 FI On-Demand Anodyne KCNQ2 40 34 O=C(Nc1cccnc1N1CCCC1)c1csc(-c2ccccc2F)n1 ZINC000147092823 FI On-Demand Anodyne PIM1 26 43 O=C(Nc1cccnc1N1CCCC1)c1csc(-c2ccccc2F)n1 ZINC000147092823 FI On-Demand Anodyne GRM4 49 39 O=C(Nc1cccnc1N1CCCC1)c1csc(-c2ccccc2F)n1 ZINC000147092823 FI On-Demand Anodyne CHEK1 19 54 O=C(Nc1cccnc1N1CCCC1)c1csc(-c2ccccc2F)n1 ZINC000147092823 FI On-Demand Anodyne PIM3 19 41 Cc1cccc(C)c1OC[C@@H](O)CNC(=O)Nc1cccc(CN(C)C)c1 ZINC000147092825 FF On-Demand Anodyne ADRB1 45 36 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)NCc1ccc(F)cc1 ZINC000147092855 HH On-Demand Anodyne GRIN2B 18 40 O=C(Nc1cccc(NC(=O)c2cccs2)c1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147092869 GF On-Demand Anodyne KCNK3 22 48 O=C(Nc1cccc(NC(=O)c2cccs2)c1)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147092869 GF On-Demand Anodyne KCNK9 17 48 CCCCO[C@H](C)C(=O)Nc1cc(C(N)=O)ccc1N1CCCC1 ZINC000147092934 EF On-Demand Anodyne KCNQ2 83 42 CCCCO[C@H](C)C(=O)Nc1cc(C(N)=O)ccc1N1CCCC1 ZINC000147092934 EF On-Demand Anodyne KCNQ4 0 41 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild NPR1 40 34 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild MC4R 19 43 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild NTSR1 23 41 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild F2R 24 52 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild HLA-A 36 46 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild FURIN 35 70 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild MC1R 41 36 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild SIRT1 31 46 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild POLG_WNV 17 48 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild NOD1 45 32 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild Q9NAW4_PLAFA 18 55 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild HPN 16 55 CSCC[C@H](NC(=O)[C@H](N)CO)C(=O)N[C@H](CCCN=C(N)N)C(=O)O ZINC000147092975 GA For-Sale Mild H9B8T9_CAPHI 53 55 N#CC1CCN(C(=O)c2cc(-c3ccccc3)n[nH]2)CC1 ZINC000147092990 CE On-Demand Mild TACR3 25 55 COc1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093004 IK Annotated Anodyne HTR1A 15 49 COc1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093004 IK Annotated Anodyne HTR2A 15 78 COc1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093004 IK Annotated Anodyne SLC6A4 20 49 COc1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093004 IK Annotated Anodyne SLC6A3 25 78 COc1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093004 IK Annotated Anodyne SIGMAR1 31 50 COc1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093004 IK Annotated Anodyne NPY2R 31 44 COc1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093004 IK Annotated Anodyne CCR5 23 78 COc1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093004 IK Annotated Anodyne EBP 41 36 COc1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093004 IK Annotated Anodyne CACNA1G 18 40 COc1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093004 IK Annotated Anodyne CYP2J2 70 50 COc1ccc([C@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093004 IK Annotated Anodyne MEN1 56 43 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)NCc1ccc(F)cc1 ZINC000147093035 HH On-Demand Anodyne GRIN2B 18 40 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)Nc2cccc(CN(C)C)c2)cc1 ZINC000147093043 HG On-Demand Anodyne BMP1 33 41 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)Nc2cccc(CN(C)C)c2)cc1 ZINC000147093043 HG On-Demand Anodyne ROCK2 19 51 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)Nc2cccc(CN(C)C)c2)cc1 ZINC000147093043 HG On-Demand Anodyne NCE103 19 40 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)Nc2cccc(CN(C)C)c2)cc1 ZINC000147093043 HG On-Demand Anodyne PRMT3 18 41 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)Nc2cccc(CN(C)C)c2)cc1 ZINC000147093043 HG On-Demand Anodyne NAMPT 68 44 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne CACNA2D1 34 43 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne GRIA3 38 46 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne NOS2 0 41 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne GRM6 20 41 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne GRM8 38 46 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne GRIA1 27 46 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne GRIA2 27 46 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne GRIK3 51 46 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne GRIA4 26 46 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne GRIK5 49 29 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne GRIK2 57 46 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne GRIK1 64 46 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne KIF11 27 42 NSC[C@@H](N)C(=O)O ZINC000147093051 AB For-Sale Anodyne BHMT 62 40 O=C(Nc1cccc(NC(=O)c2cccs2)c1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147093053 GF On-Demand Anodyne KCNK3 22 48 O=C(Nc1cccc(NC(=O)c2cccs2)c1)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147093053 GF On-Demand Anodyne KCNK9 17 48 Cc1nn(C(F)F)c(C)c1CC(=O)Nc1cc(C(N)=O)ccc1N1CCCC1 ZINC000147093129 GF On-Demand Anodyne KCNQ2 72 39 COc1ccc([C@@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093181 IK Annotated Anodyne HTR1A 15 49 COc1ccc([C@@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093181 IK Annotated Anodyne HTR2A 15 78 COc1ccc([C@@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093181 IK Annotated Anodyne SLC6A4 20 49 COc1ccc([C@@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093181 IK Annotated Anodyne SLC6A3 25 78 COc1ccc([C@@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093181 IK Annotated Anodyne SIGMAR1 31 50 COc1ccc([C@@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093181 IK Annotated Anodyne NPY2R 31 44 COc1ccc([C@@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093181 IK Annotated Anodyne CCR5 23 78 COc1ccc([C@@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093181 IK Annotated Anodyne EBP 41 36 COc1ccc([C@@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093181 IK Annotated Anodyne CACNA1G 18 40 COc1ccc([C@@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093181 IK Annotated Anodyne CYP2J2 70 50 COc1ccc([C@@H](O)CCCN2CCC(C(O)(c3ccccc3)c3ccccc3)CC2)cc1 ZINC000147093181 IK Annotated Anodyne MEN1 56 43 O=C(Nc1cccc(NC(=O)c2cccs2)c1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147093235 GF On-Demand Anodyne KCNK3 22 48 O=C(Nc1cccc(NC(=O)c2cccs2)c1)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147093235 GF On-Demand Anodyne KCNK9 17 48 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne CACNA2D1 34 43 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne GRIA3 38 46 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne NOS2 0 41 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne GRM6 20 41 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne GRM8 38 46 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne GRIA1 27 46 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne GRIA2 27 46 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne GRIK3 51 46 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne GRIA4 26 46 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne GRIK5 49 29 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne GRIK2 57 46 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne GRIK1 64 46 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne KIF11 27 42 NSC[C@H](N)C(=O)O ZINC000147093244 AB For-Sale Anodyne BHMT 62 40 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)Nc1cccc(F)c1 ZINC000147093246 HH On-Demand Anodyne P2RY1 40 34 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)Nc1cccc(F)c1 ZINC000147093246 HH On-Demand Anodyne KCNK3 25 40 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)Nc1cccc(F)c1 ZINC000147093246 HH On-Demand Anodyne KCNK9 30 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(C(=O)NC2CC2)c1 ZINC000147093364 GD On-Demand Anodyne ENV 47 38 O=C(Nc1cccc(NC(=O)c2cccs2)c1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147093431 GF On-Demand Anodyne KCNK3 22 48 O=C(Nc1cccc(NC(=O)c2cccs2)c1)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147093431 GF On-Demand Anodyne KCNK9 17 48 CN(C)Cc1cccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c1 ZINC000147093473 DG On-Demand Anodyne CCKBR 44 37 CN(C)Cc1cccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c1 ZINC000147093473 DG On-Demand Anodyne NAMPT 18 49 N#CC1CCN(C(=O)c2ccc(SC(F)(F)F)cc2)CC1 ZINC000147093509 DH On-Demand Mild L3MBTL3 77 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(C(=O)NC2CC2)c1 ZINC000147093543 GD On-Demand Anodyne ENV 47 38 C[C@@]1(c2cccc(NC(=O)COc3ccc(C(N)=O)cc3)c2)NC(=O)NC1=O ZINC000147093617 GC On-Demand Anodyne ADORA2B 42 43 C[C@@]1(c2cccc(NC(=O)COc3ccc(C(N)=O)cc3)c2)NC(=O)NC1=O ZINC000147093617 GC On-Demand Anodyne HIF1A 30 43 CN(C)Cc1cccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147093653 DG On-Demand Anodyne CCKAR 41 36 CN(C)Cc1cccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147093653 DG On-Demand Anodyne CCKBR 44 37 CN(C)Cc1cccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147093653 DG On-Demand Anodyne EPHX2 35 48 CN(C)Cc1cccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147093653 DG On-Demand Anodyne KDM1A 43 33 CN(C)Cc1cccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147093653 DG On-Demand Anodyne NAMPT 18 49 O=C1CN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cn2)CCN1 ZINC000147093746 FB On-Demand Anodyne HPGDS 15 47 C[C@]1(c2cccc(NC(=O)COc3ccc(C(N)=O)cc3)c2)NC(=O)NC1=O ZINC000147093783 GC On-Demand Anodyne ADORA2B 42 43 C[C@]1(c2cccc(NC(=O)COc3ccc(C(N)=O)cc3)c2)NC(=O)NC1=O ZINC000147093783 GC On-Demand Anodyne HIF1A 30 43 COc1ccc(C)cc1-n1ccc(C(=O)NC2CCN(C3CC3)CC2)n1 ZINC000147093801 FF On-Demand Anodyne ADRA1D 20 41 COc1ccc(C)cc1-n1ccc(C(=O)NC2CCN(C3CC3)CC2)n1 ZINC000147093801 FF On-Demand Anodyne ADRA1B 23 41 CN(C)Cc1cccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000147093852 DG On-Demand Anodyne CCKAR 41 36 CN(C)Cc1cccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000147093852 DG On-Demand Anodyne CCKBR 44 37 CN(C)Cc1cccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000147093852 DG On-Demand Anodyne EPHX2 35 48 CN(C)Cc1cccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000147093852 DG On-Demand Anodyne KDM1A 43 33 CN(C)Cc1cccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000147093852 DG On-Demand Anodyne NAMPT 18 49 CN(C)c1ccc(/C=C/c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000147093909 DG For-Sale Clean PTGS2 33 54 O=C1CN(c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cn2)CCN1 ZINC000147093939 FB On-Demand Anodyne HPGDS 15 47 O=C(NC1CC1)c1cccc(OCc2ccccc2OC(F)F)c1 ZINC000147094013 EH On-Demand Anodyne PLG 17 45 O=C(NC1CC1)c1cccc(OCc2ccccc2OC(F)F)c1 ZINC000147094013 EH On-Demand Anodyne ST14 16 45 O=C(NC1CC1)c1cccc(OCc2ccccc2OC(F)F)c1 ZINC000147094013 EH On-Demand Anodyne EZH2 40 34 CN(C)Cc1cccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c1 ZINC000147094033 DG On-Demand Anodyne CCKBR 44 37 CN(C)Cc1cccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c1 ZINC000147094033 DG On-Demand Anodyne NAMPT 18 49 CC[C@@H](C)[C@H](NC(=O)c1ccc2c(c1)COC2)c1nc2ccccc2[nH]1 ZINC000147094074 EI On-Demand Anodyne PIN1 33 44 CN(C)Cc1cccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094224 HG On-Demand Anodyne ADRB2 18 40 CN(C)Cc1cccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094224 HG On-Demand Anodyne ADRB1 48 40 CN(C)Cc1cccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094224 HG On-Demand Anodyne HRH2 16 45 CN(C)Cc1cccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094224 HG On-Demand Anodyne ADRB3 19 41 CN(C)Cc1cccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094224 HG On-Demand Anodyne RAF1 28 42 CN(C)Cc1cccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094224 HG On-Demand Anodyne PDS 88 47 CC[C@@H](C)[C@@H](NC(=O)c1ccc2c(c1)COC2)c1nc2ccccc2[nH]1 ZINC000147094269 EI On-Demand Anodyne PIN1 33 44 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCCc2cccc3ccccc23)cc(N2CCCC2=O)c1 ZINC000147094350 KJ Annotated Anodyne CTSD 63 74 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCCc2cccc3ccccc23)cc(N2CCCC2=O)c1 ZINC000147094350 KJ Annotated Anodyne BACE2 71 66 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCCc2cccc3ccccc23)cc(N2CCCC2=O)c1 ZINC000147094350 KJ Annotated Anodyne BACE1 86 84 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCCc2cccc3ccccc23)cc(N2CCCC2=O)c1 ZINC000147094350 KJ Annotated Anodyne PLM1_PLAFA 50 42 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCCc2cccc3ccccc23)cc(N2CCCC2=O)c1 ZINC000147094350 KJ Annotated Anodyne PLM2_PLAFA 34 42 Cc1cc(Oc2ccc(C=O)cc2C#N)ccc1Cl ZINC000147094367 CI For-Sale Mild ESRRA 34 46 CN(C)Cc1cccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094398 HG On-Demand Anodyne ADRB2 18 40 CN(C)Cc1cccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094398 HG On-Demand Anodyne ADRB1 48 40 CN(C)Cc1cccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094398 HG On-Demand Anodyne HRH2 16 45 CN(C)Cc1cccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094398 HG On-Demand Anodyne ADRB3 19 41 CN(C)Cc1cccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094398 HG On-Demand Anodyne RAF1 28 42 CN(C)Cc1cccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)c1 ZINC000147094398 HG On-Demand Anodyne PDS 88 47 CC[C@H](C)[C@@H](NC(=O)c1ccc2c(c1)COC2)c1nc2ccccc2[nH]1 ZINC000147094458 EI On-Demand Anodyne PIN1 33 44 Cc1cc(NC(=O)CCS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)no1 ZINC000147094485 HG On-Demand Anodyne SCN10A 24 42 Cc1cc(NC(=O)c2ccc3nc4n(c3c2)CCCNC4=O)no1 ZINC000147094486 ED Annotated Anodyne RPS6KA3 98 56 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CELA1 18 44 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CASP3 16 43 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild BMP1 61 37 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild KLK3 69 36 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CTSB 62 54 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild PAPA1_CARPA 64 39 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CYSP_TRYCR 52 38 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CTSK 40 54 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CTSL 44 40 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CAPNS1 67 40 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CTSS 21 54 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CAPN1 81 43 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CASP1 23 40 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CAPN2 129 43 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CASP6 22 40 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild CASP9 29 40 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild NPR 84 44 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild NAAA 60 40 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild PSMB5 44 41 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild SLC12A5 57 35 C=C(CC)CNC(=O)OCc1ccccc1 ZINC000147094553 BF For-Sale Mild PDS 45 35 CN(C)Cc1cccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147094593 FD On-Demand Anodyne CCR3 47 41 CN(C)Cc1cccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147094593 FD On-Demand Anodyne EPHX2 42 39 CCC(C)(C)C[C@H]1N(C)[C@@H](C(=O)NCC[C@H](O)CO)[C@H](c2cccc(Cl)c2F)[C@@]12C(=O)Nc1cc(F)c(F)cc12 ZINC000147094661 KI Annotated Anodyne MDM2 78 58 COc1cccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)c1 ZINC000147094700 HH On-Demand Anodyne P2RY1 40 34 COc1cccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)c1 ZINC000147094700 HH On-Demand Anodyne MTNR1A 30 42 COc1cccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)c1 ZINC000147094700 HH On-Demand Anodyne MTNR1B 30 44 COc1cccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)c1 ZINC000147094700 HH On-Demand Anodyne SCN10A 23 42 COc1cccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)c1 ZINC000147094700 HH On-Demand Anodyne TAAR1 35 46 COc1cccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)c1 ZINC000147094700 HH On-Demand Anodyne KCNK3 39 43 COc1cccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)c1 ZINC000147094700 HH On-Demand Anodyne KCNK9 41 43 COCCOc1cccc(C(=O)O)c1[N+](=O)[O-] ZINC000147094718 BD For-Sale Bother KCNK3 40 34 CCOc1ccc([C@H]2CCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)cc1 ZINC000147094729 HH On-Demand Bother CPT1A 123 44 CCOc1ccc([C@H]2CCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)cc1 ZINC000147094729 HH On-Demand Bother CPT2 47 44 N#CC1CCN(C(=O)[C@H]2COc3ccc(Cl)cc3C2)CC1 ZINC000147094778 DF On-Demand Mild ROCK2 18 43 CN(C)Cc1cccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147094785 FD On-Demand Anodyne CCR3 47 41 CN(C)Cc1cccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147094785 FD On-Demand Anodyne EPHX2 42 39 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(OCC(=O)N(C)C)c1)C2 ZINC000147094821 GE On-Demand Anodyne ROCK2 61 39 Cc1ccccc1NC(=O)CS(=O)(=O)[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147094904 HI On-Demand Anodyne P2RY1 54 37 Cc1ccccc1NC(=O)CS(=O)(=O)[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147094904 HI On-Demand Anodyne SHH 34 40 OC[C@@H]1OC(O)=C[C@@H](O)[C@@H]1O ZINC000147094914 AA For-Sale Anodyne PYGB 40 30 Cc1ccc(NC(=O)c2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147094938 HJ On-Demand Anodyne MAPK14 41 44 Cc1ccc(NC(=O)c2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147094938 HJ On-Demand Anodyne PRNP 51 38 Cc1ccc(NC(=O)c2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147094938 HJ On-Demand Anodyne GRM4 39 41 Cc1ccc(NC(=O)c2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147094938 HJ On-Demand Anodyne MAPK10 20 43 Cc1ccc(NC(=O)c2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147094938 HJ On-Demand Anodyne LYN 42 37 Cc1ccc(NC(=O)c2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147094938 HJ On-Demand Anodyne KCNK3 96 46 Cc1ccc(NC(=O)c2ccccc2)cc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147094938 HJ On-Demand Anodyne KCNK9 47 42 CC(C)CNC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147094958 FD On-Demand Anodyne F3 76 35 Cc1cc(Oc2ccc(C=O)cc2C#N)ccc1F ZINC000147094977 CH For-Sale Mild ESRRA 33 46 CCCC[C@@H](NC(N)=O)C(=O)N(C)CCOc1ccccc1C ZINC000147095043 DE On-Demand Anodyne PTGES 17 44 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild MMP13 44 57 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild CPA1 21 42 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild MMP2 52 59 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild MMP3 21 56 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild MMP8 27 40 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild MMP14 28 41 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild CAPN1 20 48 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild MMP9 31 59 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild MMP12 35 43 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild ITGAV 72 39 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild ADAMTS4 62 38 C=CC[C@@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095058 CC On-Demand Mild E1 0 43 OC[C@@H]1OC(O)=C[C@H](O)[C@@H]1O ZINC000147095101 AA For-Sale Anodyne PYGB 40 30 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne CA2 120 48 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne CA1 100 48 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne CA7 64 45 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne CA5B 52 43 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne CA4 85 45 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne CA5A 54 43 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne CA14 50 41 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne CA12 65 43 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne CA9 75 48 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne CYNT 35 40 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne NCE103 21 47 C[C@@H](CNC(=O)CCc1ccc(S(N)(=O)=O)cc1)N1CCCC1 ZINC000147095108 EC On-Demand Anodyne A6YCJ1_9METZ 25 42 CC(C)CNC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147095121 FD On-Demand Anodyne F3 76 35 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2ccc3c(c2)OCO3)c1 ZINC000147095159 FE On-Demand Bother EDNRB 67 39 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2ccc3c(c2)OCO3)c1 ZINC000147095159 FE On-Demand Bother EDNRA 68 40 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2ccc3c(c2)OCO3)c1 ZINC000147095159 FE On-Demand Bother CASR 41 44 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2ccc3c(c2)OCO3)c1 ZINC000147095159 FE On-Demand Bother BMP1 66 40 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2ccc3c(c2)OCO3)c1 ZINC000147095159 FE On-Demand Bother MTNR1A 28 41 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2ccc3c(c2)OCO3)c1 ZINC000147095159 FE On-Demand Bother MTNR1B 21 41 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild MMP13 44 57 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild CPA1 21 42 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild MMP2 52 59 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild MMP3 21 56 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild MMP8 27 40 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild MMP14 28 41 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild CAPN1 20 48 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild MMP9 31 59 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild MMP12 35 43 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild ITGAV 72 39 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild ADAMTS4 62 38 C=CC[C@H](NS(=O)(=O)c1ccccc1)C(=O)O ZINC000147095244 CC On-Demand Mild E1 0 43 Cc1cccc(C)c1NC(=O)CS(=O)(=O)[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147095333 HI On-Demand Anodyne SHH 40 43 NC(=O)c1ccc(OCC(=O)Nc2ccc(OCC(F)(F)F)nc2)cc1 ZINC000147095350 FE On-Demand Anodyne ADORA2B 30 41 NC(=O)c1ccc(OCC(=O)Nc2ccc(OCC(F)(F)F)nc2)cc1 ZINC000147095350 FE On-Demand Anodyne ACR 50 39 NC(=O)c1ccc(OCC(=O)Nc2ccc(OCC(F)(F)F)nc2)cc1 ZINC000147095350 FE On-Demand Anodyne HIF1A 30 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(C(=O)NCC(F)(F)F)ccc2C)c1 ZINC000147095362 HG On-Demand Bother TAAR1 29 44 Cc1nccn1-c1ccc(CNC(=O)Nc2cccc(CN(C)C)c2)cc1F ZINC000147095374 GH On-Demand Anodyne ROCK2 21 47 COc1cc(C(=O)CC(=O)C(C)(C)C)cc(OC)c1OC ZINC000147095401 CF For-Sale Anodyne TUBB1 52 40 COc1cc(C(=O)CC(=O)C(C)(C)C)cc(OC)c1OC ZINC000147095401 CF For-Sale Anodyne ACKR3 40 35 CCOC[C@H](C)NS(=O)(=O)c1c(C)cccc1[N+](=O)[O-] ZINC000147095430 DD On-Demand Bother COLA 58 34 CC(C)n1ncc2c(C(=O)NC[C@@H](C)N3CCCC3)cc(C3CC3)nc21 ZINC000147095435 FG On-Demand Anodyne EZH2 22 60 Cc1cc2c(c(C)c1[C@@H](O)CO)C(=O)[C@@H](C)[C@@H]2O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O ZINC000147095498 HB Annotated Anodyne FIMH 70 32 CCC(=O)Nc1ccc(C)c(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147095538 FE On-Demand Anodyne ADORA2B 42 45 CCC(=O)Nc1ccc(C)c(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147095538 FE On-Demand Anodyne MAPK14 16 45 CCC(=O)Nc1ccc(C)c(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147095538 FE On-Demand Anodyne ACR 54 34 CCC(=O)Nc1ccc(C)c(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147095538 FE On-Demand Anodyne MCHR1 17 40 CCC(=O)Nc1ccc(C)c(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147095538 FE On-Demand Anodyne HIF1A 18 40 Cc1cccc(Oc2ccc(C=O)cc2C#N)c1 ZINC000147095551 BG For-Sale Mild ESRRA 31 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(NC(=O)c3ccccc3)ccc2C)c1 ZINC000147095590 HI On-Demand Bother LCK 17 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(NC(=O)c3ccccc3)ccc2C)c1 ZINC000147095590 HI On-Demand Bother MAPK14 29 55 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(NC(=O)c3ccccc3)ccc2C)c1 ZINC000147095590 HI On-Demand Bother PYGL 30 49 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(NC(=O)c3ccccc3)ccc2C)c1 ZINC000147095590 HI On-Demand Bother NR1H4 24 51 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(NC(=O)c3ccccc3)ccc2C)c1 ZINC000147095590 HI On-Demand Bother BTK 18 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(NC(=O)c3ccccc3)ccc2C)c1 ZINC000147095590 HI On-Demand Bother TAAR1 36 52 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(NC(=O)c3ccccc3)ccc2C)c1 ZINC000147095590 HI On-Demand Bother AKR1C3 35 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(NC(=O)c3ccccc3)ccc2C)c1 ZINC000147095590 HI On-Demand Bother AKR1C2 64 45 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(NC(=O)c3ccccc3)ccc2C)c1 ZINC000147095590 HI On-Demand Bother SMO 37 45 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(NC(=O)c3ccccc3)ccc2C)c1 ZINC000147095590 HI On-Demand Bother KCNK3 107 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cc(NC(=O)c3ccccc3)ccc2C)c1 ZINC000147095590 HI On-Demand Bother KCNK9 62 39 CC(C)n1ncc2c(C(=O)NC[C@H](C)N3CCCC3)cc(C3CC3)nc21 ZINC000147095632 FG On-Demand Anodyne EZH2 22 60 N#Cc1cc(CC(=O)O)ccc1O ZINC000147095711 AC For-Sale Mild CAN2 0 56 Cc1ccc(CN(c2ccc(C(=O)NC(C)C)cc2)S(C)(=O)=O)cc1 ZINC000147095739 FG In-Stock Anodyne MMP9 16 47 C[C@@]1(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)NC(=O)NC1=O ZINC000147095782 GC On-Demand Anodyne ADORA2B 45 47 C[C@@]1(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)NC(=O)NC1=O ZINC000147095782 GC On-Demand Anodyne ACR 49 35 C[C@@]1(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)NC(=O)NC1=O ZINC000147095782 GC On-Demand Anodyne HIF1A 27 45 NC(N)=N/N=C/c1c(F)cccc1Br ZINC000147095784 CD For-Sale Mild AMD1 20 40 NC(N)=N/N=C/c1c(F)cccc1Br ZINC000147095784 CD For-Sale Mild UREA_CANEN 16 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(=O)OC)cc1 ZINC000147095800 EC On-Demand Anodyne MMP13 38 41 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(=O)OC)cc1 ZINC000147095800 EC On-Demand Anodyne MMP2 31 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(=O)OC)cc1 ZINC000147095800 EC On-Demand Anodyne MMP3 17 47 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(=O)OC)cc1 ZINC000147095800 EC On-Demand Anodyne MMP14 20 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(=O)OC)cc1 ZINC000147095800 EC On-Demand Anodyne MMP9 27 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(=O)OC)cc1 ZINC000147095800 EC On-Demand Anodyne MMP12 17 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(=O)OC)cc1 ZINC000147095800 EC On-Demand Anodyne MMP7 25 47 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(=O)OC)cc1 ZINC000147095800 EC On-Demand Anodyne ADAMTS4 66 38 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCC(=O)OC)cc1 ZINC000147095800 EC On-Demand Anodyne MMP1 18 47 COCc1nc(C(=O)Nc2ccc(OC)c(OC)c2)cs1 ZINC000147095803 DF On-Demand Anodyne GRM4 30 46 COCc1nc(C(=O)Nc2ccc(OC)c(OC)c2)cs1 ZINC000147095803 DF On-Demand Anodyne ENPP1 72 42 COCc1nc(C(=O)Nc2ccc(OC)c(OC)c2)cs1 ZINC000147095803 DF On-Demand Anodyne DRTS_TRYCR 47 33 COC(=O)c1ccc2c(Br)nsc2c1 ZINC000147095969 CF For-Sale Anodyne TRPA1 15 41 C[C@]1(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)NC(=O)NC1=O ZINC000147095982 GC On-Demand Anodyne ADORA2B 45 47 C[C@]1(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)NC(=O)NC1=O ZINC000147095982 GC On-Demand Anodyne ACR 49 35 C[C@]1(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)NC(=O)NC1=O ZINC000147095982 GC On-Demand Anodyne HIF1A 27 45 Cc1cccc(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)c1C ZINC000147096032 HI On-Demand Anodyne P2RY1 46 35 Cc1cc(=O)c(C(=O)N2CCC(C#N)CC2)nn1-c1cccc(C(F)(F)F)c1 ZINC000147096040 GF On-Demand Mild NPY5R 16 43 COC(=O)c1cc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc(C(=O)OC)c1 ZINC000147096089 FF On-Demand Bother CACNA1D 45 37 COC(=O)c1cc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc(C(=O)OC)c1 ZINC000147096089 FF On-Demand Bother KCNK3 41 33 COC(=O)c1cc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc(C(=O)OC)c1 ZINC000147096089 FF On-Demand Bother KCNK9 40 35 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(OCc2cccnc2)c1 ZINC000147096112 FE On-Demand Anodyne VCP 42 33 CC(C)(C)OC(=O)NC1CCC(N[C@@H](C(=O)O)c2ccccc2)CC1 ZINC000147096139 EG On-Demand Anodyne SCN9A 18 40 CC(C)(C)OC(=O)NC1CCC(N[C@@H](C(=O)O)c2ccccc2)CC1 ZINC000147096139 EG On-Demand Anodyne FPR1 46 37 COc1ccc(Cl)cc1CNC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147096162 GF On-Demand Bother CPT1A 61 35 COc1ccc(Cl)cc1CNC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147096162 GF On-Demand Bother KCNMA1 28 40 COc1ccc(Cl)cc1CNC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147096162 GF On-Demand Bother CPT1B 60 34 CCc1ccccc1NC(=O)CS(=O)(=O)[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147096215 HI On-Demand Anodyne P2RY1 62 39 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(OCc2cccnc2)c1 ZINC000147096297 FE On-Demand Anodyne VCP 42 33 CC(C)(C)OC(=O)NC1CCC(N[C@H](C(=O)O)c2ccccc2)CC1 ZINC000147096328 EG On-Demand Anodyne SCN9A 18 40 CC(C)(C)OC(=O)NC1CCC(N[C@H](C(=O)O)c2ccccc2)CC1 ZINC000147096328 EG On-Demand Anodyne FPR1 46 37 CCc1cccc(Cc2cnc(NC(=O)c3cc(OC)ccc3[N+](=O)[O-])s2)c1 ZINC000147096337 GI On-Demand Bother SCD1 41 45 CCc1cccc(Cc2cnc(NC(=O)c3cc(OC)ccc3[N+](=O)[O-])s2)c1 ZINC000147096337 GI On-Demand Bother SCD 40 55 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)NC1CCCCCC1 ZINC000147096433 HH On-Demand Anodyne EPHX2 36 52 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne ALDH2 69 37 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne ALOX5 15 47 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne INHA 79 40 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne CNR2 16 48 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne RARB 18 49 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne GGPS1 17 42 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne GRM2 19 46 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne MTNR1A 25 45 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne MTNR1B 19 41 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne PLA2G4B 115 49 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne LSS 27 43 CCCCCCOc1ccc(C(C)=O)c(O)c1 ZINC000147096454 BH In-Stock Anodyne FAAH 25 45 COCCOCc1cccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147096463 FG On-Demand Anodyne ROCK2 31 46 COCCOCc1cccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147096463 FG On-Demand Anodyne FFAR1 21 40 COC(=O)c1cc(F)ccc1NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147096532 GE On-Demand Bother PYGL 28 40 CCn1c(=O)c(=O)[nH]c2cc(C(=O)NC[C@@H](C)N3CCCC3)ccc21 ZINC000147096534 EC On-Demand Anodyne PLD1 54 44 CCn1c(=O)c(=O)[nH]c2cc(C(=O)NC[C@@H](C)N3CCCC3)ccc21 ZINC000147096534 EC On-Demand Anodyne PLD2 42 33 CCn1c(=O)c(=O)[nH]c2cc(C(=O)NC[C@H](C)N3CCCC3)ccc21 ZINC000147096724 EC On-Demand Anodyne PLD1 54 44 CCn1c(=O)c(=O)[nH]c2cc(C(=O)NC[C@H](C)N3CCCC3)ccc21 ZINC000147096724 EC On-Demand Anodyne PLD2 42 33 COC(=O)c1cc(F)ccc1NC(=O)c1cc(OC)ccc1[N+](=O)[O-] ZINC000147096725 EF On-Demand Bother TAAR1 25 44 COC(=O)c1cc(F)ccc1NC(=O)c1cc(OC)ccc1[N+](=O)[O-] ZINC000147096725 EF On-Demand Bother AKR1C3 19 42 COC(=O)c1cc(F)ccc1NC(=O)c1cc(OC)ccc1[N+](=O)[O-] ZINC000147096725 EF On-Demand Bother AKR1C2 46 44 Cc1cccc(Oc2ccc(CO)cc2C(F)(F)F)c1 ZINC000147096755 CI For-Sale Anodyne NR1H3 22 44 Cc1cccc(Oc2ccc(CO)cc2C(F)(F)F)c1 ZINC000147096755 CI For-Sale Anodyne NR1H2 15 44 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147096865 FE On-Demand Anodyne CCKAR 0 40 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147096865 FE On-Demand Anodyne EPHX2 25 44 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147096865 FE On-Demand Anodyne TMPRSS11D 55 35 CC1CCC(NC(=O)CS(=O)(=O)[C@@H](C)c2ccc(OC(F)(F)F)cc2)CC1 ZINC000147096871 HH On-Demand Anodyne EPHX2 28 44 N#CC1CCN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147096920 HH On-Demand Mild CCR1 19 51 N#CC1CCN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147096920 HH On-Demand Mild APP 41 36 N#CC1CCN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147096920 HH On-Demand Mild PRTN3 55 36 N#CC1CCN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147096920 HH On-Demand Mild SFRP1 40 39 CC[C@@H](COc1ccc(Cl)cc1)OC ZINC000147096991 BG On-Demand Anodyne EBP 19 43 CC[C@@H](COc1ccc(Cl)cc1)OC ZINC000147096991 BG On-Demand Anodyne PDS 59 38 C[C@@H](OC[C@@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147097055 FE On-Demand Anodyne CCKAR 0 40 C[C@@H](OC[C@@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147097055 FE On-Demand Anodyne EPHX2 25 44 C[C@@H](OC[C@@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147097055 FE On-Demand Anodyne TMPRSS11D 55 35 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CA2 106 57 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CA6 21 40 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CA1 82 57 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CA7 56 57 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CA13 34 40 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CA5B 44 52 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CA4 79 55 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CA5A 44 52 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CA14 47 47 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CA12 60 50 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CA9 67 50 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne CYNT 34 54 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne NCE103 41 49 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne ALPI 17 54 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne MTCA1 22 40 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne P96878_MYCTU 31 42 CCc1ncc(C(=O)NCCc2ccc(S(N)(=O)=O)cc2)s1 ZINC000147097108 ED On-Demand Anodyne A6YCJ1_9METZ 27 57 CN(CCCCc1ccccc1)C(=O)c1ccc2c(c1)COC2 ZINC000147097134 DH On-Demand Anodyne SIGMAR1 16 46 CN(CCCCc1ccccc1)C(=O)c1ccc2c(c1)COC2 ZINC000147097134 DH On-Demand Anodyne FAAH 40 37 CN(CCCCc1ccccc1)C(=O)c1ccc2c(c1)COC2 ZINC000147097134 DH On-Demand Anodyne CES1 42 33 C[C@@H](CCc1c[nH]c2ccc(F)cc12)N(CC1CC1)[C@@H]1COc2c(F)ccc(C(N)=O)c2C1 ZINC000147097184 JJ Annotated Anodyne MPO 85 40 CC[C@H](COc1ccc(Cl)cc1)OC ZINC000147097201 BG On-Demand Anodyne EBP 19 43 CC[C@H](COc1ccc(Cl)cc1)OC ZINC000147097201 BG On-Demand Anodyne PDS 59 38 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CA2 22 44 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne ACE 49 40 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne OPRM1 89 68 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne OPRD1 96 68 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne OPRK1 15 43 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne MME 136 52 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne LTA4H 15 44 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne ANPEP 92 39 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne TACR1 18 49 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CTSD 28 43 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne FCER2 85 38 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne GRB2 57 41 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne TACR2 21 52 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne RNPEP 43 44 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne KLK3 52 38 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CTSB 61 41 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne PAPA1_CARPA 75 37 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CYSP_TRYCR 55 35 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CTSK 23 40 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CTSL 50 41 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CPA1 41 38 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne PGA 45 45 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne NPFFR2 57 31 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne C3AR1 51 54 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne HLA-A 106 53 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne TPH1 56 34 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne TACR3 24 44 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CAPNS1 64 38 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne MMP3 19 46 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne GRIA1 62 41 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne GRPR 50 31 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne HLA-DRB1 77 44 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne REN 37 43 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne REN1 57 36 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne LNPEP 19 44 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne FURIN 66 39 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne YARS 64 40 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CCKBR 20 40 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CTSS 23 40 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CAPN1 88 46 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CAPN2 113 41 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne ACE2 74 38 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne BACE1 29 47 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne LAP3 44 44 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne CTSC 25 45 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne MMP1 25 41 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne FPR1 77 42 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne NPR 70 42 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne AMP1_PLAFQ 30 44 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne XIAP 23 40 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne PSMB2 35 42 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne PSMB5 27 47 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne BLA1_STEMA 57 37 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne KISS1R 53 32 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne POLG_WNV 41 30 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne QRFPR 51 38 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne F2RL1 57 37 C[C@H](O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)C(=O)NCC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147097233 IA For-Sale Anodyne NPFFR1 61 31 C[C@H](OC[C@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147097236 FE On-Demand Anodyne CCKAR 0 40 C[C@H](OC[C@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147097236 FE On-Demand Anodyne EPHX2 25 44 C[C@H](OC[C@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147097236 FE On-Demand Anodyne TMPRSS11D 55 35 C[C@H](CCc1c[nH]c2ccc(F)cc12)N(CC1CC1)[C@@H]1COc2c(F)ccc(C(N)=O)c2C1 ZINC000147097369 JJ Annotated Anodyne MPO 85 40 CCCCCCNC(=O)OCCCC ZINC000147097408 BG For-Sale Anodyne S1PR3 20 45 CCCCCCNC(=O)OCCCC ZINC000147097408 BG For-Sale Anodyne FAAH 23 44 CCCCCCNC(=O)OCCCC ZINC000147097408 BG For-Sale Anodyne S1PR2 25 45 CCCCCCNC(=O)OCCCC ZINC000147097408 BG For-Sale Anodyne EPHX2 21 43 CCCCCCNC(=O)OCCCC ZINC000147097408 BG For-Sale Anodyne CES2C 40 38 CCCCCCNC(=O)OCCCC ZINC000147097408 BG For-Sale Anodyne ASAH1 95 37 CCCCCCNC(=O)OCCCC ZINC000147097408 BG For-Sale Anodyne NOD1 40 35 CCCCCCNC(=O)OCCCC ZINC000147097408 BG For-Sale Anodyne CQSS 52 33 C[C@@H](OC[C@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147097427 FE On-Demand Anodyne CCKAR 0 40 C[C@@H](OC[C@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147097427 FE On-Demand Anodyne EPHX2 25 44 C[C@@H](OC[C@H]1CCCO1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147097427 FE On-Demand Anodyne TMPRSS11D 55 35 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097471 GD On-Demand Anodyne GHRHR 41 33 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097471 GD On-Demand Anodyne P2RY12 190 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097471 GD On-Demand Anodyne HRH3 22 43 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097471 GD On-Demand Anodyne TRY2_BOVIN 57 33 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097471 GD On-Demand Anodyne CACNA1B 15 45 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097471 GD On-Demand Anodyne NOD2 33 43 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne SLC29A1 118 50 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne ADORA2B 15 57 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne DNMT1 20 51 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne TK1 22 40 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne ADK 33 57 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne AHCY 86 44 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne P2RX4 35 40 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne P2RX1 46 40 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne P2RY1 44 55 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne ADCY5 18 42 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne AMD1 16 41 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne GAPDH 20 40 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne ITPR1 34 40 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne ADORA3 70 57 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne OXGR1 121 40 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne DNMT3B 37 41 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne PANC 30 44 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne Q4VQ11_PIG 87 57 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne GPR17 47 41 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne HSPA5 42 38 Nc1nc(Cl)nc2c1ncn2[C@H]1O[C@H](CO)[C@H](O)[C@@H]1F ZINC000147097473 DB For-Sale Anodyne DOT1L 65 37 CCN(CC)CCOc1ccccc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@@H]21 ZINC000147097476 GE On-Demand Anodyne AMY2 58 37 COCc1nc(C(=O)N2CCN(c3cccc(Cl)c3)CC2)cs1 ZINC000147097585 FF On-Demand Anodyne HTR1A 19 42 COCc1nc(C(=O)N2CCN(c3cccc(Cl)c3)CC2)cs1 ZINC000147097585 FF On-Demand Anodyne HTR2A 18 42 COCc1nc(C(=O)N2CCN(c3cccc(Cl)c3)CC2)cs1 ZINC000147097585 FF On-Demand Anodyne CCKAR 42 51 COCc1nc(C(=O)N2CCN(c3cccc(Cl)c3)CC2)cs1 ZINC000147097585 FF On-Demand Anodyne TRPC6 51 39 OC[C@H]1O[C@@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000147097623 AB For-Sale Anodyne ADORA1 45 40 OC[C@H]1O[C@@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000147097623 AB For-Sale Anodyne SLC29A1 73 36 OC[C@H]1O[C@@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000147097623 AB For-Sale Anodyne ADORA2A 35 40 OC[C@H]1O[C@@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000147097623 AB For-Sale Anodyne ADK 47 40 OC[C@H]1O[C@@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000147097623 AB For-Sale Anodyne CDA 73 44 OC[C@H]1O[C@@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000147097623 AB For-Sale Anodyne PNP 19 40 OC[C@H]1O[C@@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000147097623 AB For-Sale Anodyne ADORA3 17 40 OC[C@H]1O[C@@H](n2cccc2)[C@H](O)[C@@H]1O ZINC000147097623 AB For-Sale Anodyne FIMH 77 42 N#CC1CCN(C(=O)c2ccccc2Nc2ccccc2)CC1 ZINC000147097628 DH On-Demand Mild AKR1C3 25 43 N#CC1CCN(C(=O)c2ccccc2Nc2ccccc2)CC1 ZINC000147097628 DH On-Demand Mild AKR1C2 52 51 N#CC1CCN(C(=O)c2ccccc2Nc2ccccc2)CC1 ZINC000147097628 DH On-Demand Mild L3MBTL3 66 52 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097655 GD On-Demand Anodyne GHRHR 41 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097655 GD On-Demand Anodyne P2RY12 190 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097655 GD On-Demand Anodyne HRH3 22 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097655 GD On-Demand Anodyne TRY2_BOVIN 57 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097655 GD On-Demand Anodyne CACNA1B 15 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2ccc(OCC)cc2)CC1 ZINC000147097655 GD On-Demand Anodyne NOD2 33 43 CCN(CC)CCOc1ccccc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@@H]21 ZINC000147097658 GE On-Demand Anodyne AMY2 58 37 CCCc1c(OCc2ccc(Sc3cccc(C(=O)OC)c3)cn2)ccc(C(C)=O)c1O ZINC000147097675 JK For-Sale Anodyne CYSLTR1 32 42 O=C(c1c[nH]c2ccccc12)N1CCCN(C[C@H](O)CN2CCOCC2)CC1 ZINC000147097716 GD On-Demand Anodyne PARP1 15 41 CS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cn1 ZINC000147097747 EC On-Demand Anodyne ADORA2B 40 44 CS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cn1 ZINC000147097747 EC On-Demand Anodyne ACR 42 33 CS(=O)(=O)c1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cn1 ZINC000147097747 EC On-Demand Anodyne HIF1A 25 43 CCN(CC)CCOc1ccccc1NC(=O)C(=O)N1CCO[C@H]2CCC[C@H]21 ZINC000147097852 GE On-Demand Anodyne AMY2 58 37 O=C(c1c[nH]c2ccccc12)N1CCCN(C[C@@H](O)CN2CCOCC2)CC1 ZINC000147097915 GD On-Demand Anodyne PARP1 15 41 Cc1cc(C(=O)N2CCN(c3cccc(Cl)c3)CC2)cc([N+](=O)[O-])c1 ZINC000147098022 FH On-Demand Bother HTR1A 16 47 Cc1cc(C(=O)N2CCN(c3cccc(Cl)c3)CC2)cc([N+](=O)[O-])c1 ZINC000147098022 FH On-Demand Bother SSTR1 40 37 N#CC1CCN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)CC1 ZINC000147098024 HG On-Demand Mild PRTN3 47 34 N#CC1CCN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)CC1 ZINC000147098024 HG On-Demand Mild SFRP1 88 37 N#CC1CCN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)CC1 ZINC000147098024 HG On-Demand Mild WNT3 74 35 CCN(CC)CCOc1ccccc1NC(=O)C(=O)N1CCO[C@@H]2CCC[C@H]21 ZINC000147098034 GE On-Demand Anodyne AMY2 58 37 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1 ZINC000147098091 HF On-Demand Anodyne F2 18 40 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1 ZINC000147098091 HF On-Demand Anodyne LPL 45 42 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1 ZINC000147098091 HF On-Demand Anodyne ADORA2B 21 40 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1 ZINC000147098091 HF On-Demand Anodyne TACR2 21 40 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1 ZINC000147098091 HF On-Demand Anodyne TRY2_BOVIN 93 40 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1 ZINC000147098091 HF On-Demand Anodyne ITGA4 63 31 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1 ZINC000147098091 HF On-Demand Anodyne EPHX2 16 45 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1 ZINC000147098091 HF On-Demand Anodyne TGM2 67 44 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1 ZINC000147098091 HF On-Demand Anodyne ST14 91 37 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1 ZINC000147098091 HF On-Demand Anodyne F13A1 101 44 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccc(S(=O)(=O)N2CCN(C)CC2)cc1 ZINC000147098091 HF On-Demand Anodyne NAMPT 37 58 O=C(Nc1ccc(Cn2cccn2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147098103 GI On-Demand Anodyne NOD2 42 35 COCc1cccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)c1 ZINC000147098142 HG On-Demand Anodyne BMP1 36 44 COCc1cccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)c1 ZINC000147098142 HG On-Demand Anodyne ROCK2 24 41 COCc1cccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)c1 ZINC000147098142 HG On-Demand Anodyne NCE103 19 42 COCc1cccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)c1 ZINC000147098142 HG On-Demand Anodyne PRMT3 19 42 COCc1cccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)c1 ZINC000147098142 HG On-Demand Anodyne NAMPT 60 43 CCOC[C@H](C)NS(=O)(=O)c1cc2c(cc1F)NC(=O)CC2 ZINC000147098144 ED On-Demand Anodyne PKM 49 53 O=C(Nc1ccc(Cn2cccn2)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147098280 FI On-Demand Anodyne NAMPT 27 44 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(N2CCCC2=O)c1 ZINC000147098323 EH On-Demand Anodyne KCNQ2 25 40 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1ccc(F)cc1 ZINC000147098331 HI On-Demand Anodyne P2RY1 50 37 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1ccc(F)cc1 ZINC000147098331 HI On-Demand Anodyne EPHX2 47 41 COCc1cccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147098352 FF On-Demand Anodyne DRD4 19 40 COCc1cccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147098352 FF On-Demand Anodyne MCHR1 15 41 CCOc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147098417 EE On-Demand Anodyne ENV 41 33 N#CC1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000147098440 FJ On-Demand Mild CACNA1B 57 41 N#CC1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000147098440 FJ On-Demand Mild RBP4 42 35 N#CC1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000147098440 FJ On-Demand Mild AKR1C3 27 60 N#CC1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000147098440 FJ On-Demand Mild AKR1C2 41 60 N#CC1CCN(C(=O)c2ccccc2Nc2cccc(C(F)(F)F)c2)CC1 ZINC000147098440 FJ On-Demand Mild L3MBTL3 17 42 O=C(CCSc1ccc(Cl)cc1)Nc1ccc2ccccc2c1 ZINC000147098450 EK In-Stock Anodyne IMDH_CRYPV 48 40 O=C(NC1CC1)c1cccc(CNC(=O)c2cccnc2SC(F)(F)F)c1 ZINC000147098455 GH On-Demand Anodyne MAPK14 18 41 O=C(NC1CC1)c1cccc(CNC(=O)c2cccnc2SC(F)(F)F)c1 ZINC000147098455 GH On-Demand Anodyne CCR2 48 38 O=C(Nc1ccc(Cn2cccn2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147098469 FI On-Demand Anodyne NAMPT 27 44 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(N2CCCC2=O)c1 ZINC000147098505 EH On-Demand Anodyne KCNQ2 25 40 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1ccc(F)cc1 ZINC000147098527 HI On-Demand Anodyne P2RY1 50 37 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CCC(=O)Nc1ccc(F)cc1 ZINC000147098527 HI On-Demand Anodyne EPHX2 47 41 COc1ccc(C)c2ncccc12 ZINC000147098561 AF For-Sale Anodyne CCR1 20 44 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne F2 37 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne CHRM1 17 42 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne ACE 55 38 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne HTR2A 15 44 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne OPRM1 19 45 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne OPRD1 15 42 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne GHRHR 70 44 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne P2RY12 207 42 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne SIGMAR1 26 45 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne TRY2_BOVIN 94 38 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne CCKAR 33 42 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne CTSK 40 40 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne NPFFR2 48 32 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne MMP3 41 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne CCKBR 52 42 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne GHSR 18 45 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne CAPN1 20 40 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne CAPN2 42 35 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne ACE2 40 37 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne TGM2 25 44 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne DPP7 42 42 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne ST14 43 35 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne CTRB_BOVIN 45 32 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne AMP1_PLAFQ 28 42 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098572 ED On-Demand Anodyne POLG_WNV 45 32 CCOc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147098600 EE On-Demand Anodyne ENV 41 33 CS(=O)(=O)c1cc(C(=O)NCc2cccc(C(=O)NC3CC3)c2)cc([N+](=O)[O-])c1 ZINC000147098650 HD On-Demand Bother CCR2 17 40 O=C(Nc1ccc(Cn2cccn2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147098673 FI On-Demand Anodyne NAMPT 27 44 Cc1ccc(C)c(N2C(=O)c3ccc(C(=O)NC[C@@H](C)N4CCCC4)cc3C2=O)c1 ZINC000147098684 HG On-Demand Anodyne ADRA1D 15 46 Cc1ccc(C)c(N2C(=O)c3ccc(C(=O)NC[C@@H](C)N4CCCC4)cc3C2=O)c1 ZINC000147098684 HG On-Demand Anodyne ADRA1A 15 46 Cc1ccc(C)c(N2C(=O)c3ccc(C(=O)NC[C@@H](C)N4CCCC4)cc3C2=O)c1 ZINC000147098684 HG On-Demand Anodyne F3 47 30 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne F2 37 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne CHRM1 17 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne ACE 55 38 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne HTR2A 15 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne OPRM1 19 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne OPRD1 15 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne GHRHR 70 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne P2RY12 207 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne SIGMAR1 26 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne TRY2_BOVIN 94 38 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne CCKAR 33 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne CTSK 40 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne NPFFR2 48 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne MMP3 41 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne CCKBR 52 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne GHSR 18 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne CAPN1 20 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne CAPN2 42 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne ACE2 40 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne TGM2 25 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne DPP7 42 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne ST14 43 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne CTRB_BOVIN 45 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne AMP1_PLAFQ 28 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCc2ccccc2)CC1 ZINC000147098757 ED On-Demand Anodyne POLG_WNV 45 32 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)NCC1CCCCC1 ZINC000147098779 HH On-Demand Anodyne CTSL 18 42 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)NCC1CCCCC1 ZINC000147098779 HH On-Demand Anodyne CTSS 27 42 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)NCC1CCCCC1 ZINC000147098779 HH On-Demand Anodyne EPHX2 20 41 O=[N+]([O-])c1cc(Br)cnc1Nc1cccc(CN2CCOCC2)c1 ZINC000147098806 GG On-Demand Bother EGFR 23 41 O=C(NC1CC1)c1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147098835 GF On-Demand Anodyne MAPK14 31 43 O=C(NC1CC1)c1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147098835 GF On-Demand Anodyne MAPK13 77 33 COC(=O)CNS(=O)(=O)c1cccc(NC(=O)COC(C)C)c1 ZINC000147098839 EC On-Demand Anodyne CA4 15 44 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(Cn3cccn3)cc1)C2 ZINC000147098859 FG On-Demand Anodyne MTNR1A 20 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(Cn3cccn3)cc1)C2 ZINC000147098859 FG On-Demand Anodyne MTNR1B 24 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(Cn3cccn3)cc1)C2 ZINC000147098859 FG On-Demand Anodyne ROCK2 40 51 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(Cn3cccn3)cc1)C2 ZINC000147098859 FG On-Demand Anodyne CFTR 46 32 COCc1nc(C(=O)Nc2ccc(C(F)(F)F)cc2)cs1 ZINC000147098882 DH On-Demand Anodyne TRPV1 23 46 COCc1nc(C(=O)Nc2ccc(C(F)(F)F)cc2)cs1 ZINC000147098882 DH On-Demand Anodyne ATF1 40 43 COCc1nc(C(=O)Nc2ccc(C(F)(F)F)cc2)cs1 ZINC000147098882 DH On-Demand Anodyne FLT1 21 40 COCc1nc(C(=O)Nc2ccc(C(F)(F)F)cc2)cs1 ZINC000147098882 DH On-Demand Anodyne NFKB1 37 43 COCc1nc(C(=O)Nc2ccc(C(F)(F)F)cc2)cs1 ZINC000147098882 DH On-Demand Anodyne EPHX2 18 42 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)NCC1CCCCC1 ZINC000147098954 HH On-Demand Anodyne CTSL 18 42 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)NCC1CCCCC1 ZINC000147098954 HH On-Demand Anodyne CTSS 27 42 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)NCC1CCCCC1 ZINC000147098954 HH On-Demand Anodyne EPHX2 20 41 COCc1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147099114 FI On-Demand Anodyne NPY1R 43 37 COCc1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147099114 FI On-Demand Anodyne KCNK3 41 34 Cc1cccc(C(=O)O)c1OC1CCCCC1 ZINC000147099158 BG For-Sale Anodyne SLC6A1 40 34 Cc1cccc(C(=O)O)c1OC1CCCCC1 ZINC000147099158 BG For-Sale Anodyne FABP4 41 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC(c2nc3cc(Cl)ccc3s2)CC1 ZINC000147099228 HH On-Demand Anodyne P2RY12 192 36 CCCC[C@H](NC(N)=O)C(=O)N1CCC(c2nc3cc(Cl)ccc3s2)CC1 ZINC000147099228 HH On-Demand Anodyne TRY1_BOVIN 42 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC(c2nc3cc(Cl)ccc3s2)CC1 ZINC000147099228 HH On-Demand Anodyne CCR1 41 40 CCOC(=O)NCC(=O)N1CCN(c2nc(C)cs2)CC1 ZINC000147099243 DC On-Demand Anodyne P2RY12 27 40 COCc1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147099334 FI On-Demand Anodyne NPY1R 43 37 COCc1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147099334 FI On-Demand Anodyne KCNK3 41 34 CCOC[C@H](C)NS(=O)(=O)c1ccc(-n2ncc(Cl)c(Cl)c2=O)cc1 ZINC000147099347 HE On-Demand Anodyne NPBWR1 47 41 CCc1cccc2c1[C@@H](N)CC2 ZINC000147099348 AE For-Sale Anodyne HTR1A 17 43 CCc1cccc2c1[C@@H](N)CC2 ZINC000147099348 AE For-Sale Anodyne ANPEP 35 43 CCc1cccc2c1[C@@H](N)CC2 ZINC000147099348 AE For-Sale Anodyne CYP27A1 46 35 CCCCCCCCCCC[C@@H](OC(C)=O)[C@H](C)NC(C)=O ZINC000147099463 DI Annotated Mild PLA2G2C 0 40 CCCCCCCCCCC[C@@H](OC(C)=O)[C@H](C)NC(C)=O ZINC000147099463 DI Annotated Mild PLA2G2A 0 46 CCCCCCCCCCC[C@@H](OC(C)=O)[C@H](C)NC(C)=O ZINC000147099463 DI Annotated Mild NOD1 85 39 CCCCCCCCCCC[C@@H](OC(C)=O)[C@H](C)NC(C)=O ZINC000147099463 DI Annotated Mild CQSS 51 33 COCc1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147099517 FI On-Demand Anodyne NPY1R 43 37 COCc1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147099517 FI On-Demand Anodyne KCNK3 41 34 CCc1cccc2c1[C@H](N)CC2 ZINC000147099542 AE For-Sale Anodyne HTR1A 17 43 CCc1cccc2c1[C@H](N)CC2 ZINC000147099542 AE For-Sale Anodyne ANPEP 35 43 CCc1cccc2c1[C@H](N)CC2 ZINC000147099542 AE For-Sale Anodyne CYP27A1 46 35 N#CCC[C@@H](C#N)CN1CCCN(C(=O)c2c[nH]c3ccccc23)CC1 ZINC000147099565 EF On-Demand Mild AVPR1A 16 40 COc1ccc(Cl)cc1CS(=O)(=O)[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147099588 HJ On-Demand Anodyne GRIN2B 17 40 COCc1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147099678 FI On-Demand Anodyne NPY1R 43 37 COCc1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147099678 FI On-Demand Anodyne KCNK3 41 34 CCC[C@@H](C(=O)O)S(=O)(=O)O ZINC000147099790 AC For-Sale Anodyne GCLC 53 32 N#CCC[C@H](C#N)CN1CCCN(C(=O)c2c[nH]c3ccccc23)CC1 ZINC000147099799 EF On-Demand Mild AVPR1A 16 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)C23CC4CC(CC(C4)C2)C3)CC1 ZINC000147099862 HE On-Demand Anodyne GHRHR 42 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)C23CC4CC(CC(C4)C2)C3)CC1 ZINC000147099862 HE On-Demand Anodyne P2RY12 78 33 CCOc1ccc(O[C@@H](C)C(=O)NNC(=O)Nc2nc(C)cs2)cc1 ZINC000147099934 FE On-Demand Reactive GCK 19 40 CCC[C@H](C(=O)O)S(=O)(=O)O ZINC000147099960 AC For-Sale Anodyne GCLC 53 32 CCOc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1OC ZINC000147099997 ED On-Demand Anodyne SSTR5 34 42 CCOc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1OC ZINC000147099997 ED On-Demand Anodyne QRFPR 41 34 CCOc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1OC ZINC000147099997 ED On-Demand Anodyne ENPP1 49 30 O=C(Nc1ccc2oc(C3CC3)nc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147100054 GI On-Demand Anodyne NR2E3 65 36 COc1ccc(OC)c(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147100085 DG On-Demand Bother EPHX1 0 43 COc1ccc(OC)c(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147100085 DG On-Demand Bother PYGL 34 48 COc1ccc(OC)c(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147100085 DG On-Demand Bother KCNMA1 28 51 COc1ccc(OC)c(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147100085 DG On-Demand Bother TAAR1 24 41 COc1ccc(OC)c(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147100085 DG On-Demand Bother AKR1C2 45 44 CCOc1ccc(O[C@H](C)C(=O)NNC(=O)Nc2nc(C)cs2)cc1 ZINC000147100123 FE On-Demand Reactive GCK 16 40 c1cncc(NC2=NCCN2)c1 ZINC000147100182 AC For-Sale Anodyne NISCH 29 44 CCOc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1OC ZINC000147100208 ED On-Demand Anodyne SSTR5 34 42 CCOc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1OC ZINC000147100208 ED On-Demand Anodyne QRFPR 41 34 CCOc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1OC ZINC000147100208 ED On-Demand Anodyne ENPP1 49 30 C[C@H](Cn1ccnc1)NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147100253 DC On-Demand Anodyne CYP11B1 16 41 C[C@H](Cn1ccnc1)NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147100253 DC On-Demand Anodyne TBXAS1 44 52 C[C@H](Cn1ccnc1)NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147100253 DC On-Demand Anodyne CYP11B2 15 41 C[C@H](Cn1ccnc1)NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147100253 DC On-Demand Anodyne CYP26A1 63 37 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(Cl)s2)c1 ZINC000147100370 EG In-Stock Bother MTNR1A 45 36 Cc1ccc(Oc2ccc(CCO)cc2)nc1 ZINC000147100395 BF For-Sale Anodyne ACACA 36 44 Cc1ccc(Oc2ccc(CCO)cc2)nc1 ZINC000147100395 BF For-Sale Anodyne ACACB 23 44 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne GRIN2B 0 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne NPY1R 23 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne CTSK 19 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne PCSK2 0 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne SCN9A 0 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne GRIA1 40 33 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne PCSK7 0 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne PCSK5 60 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne FURIN 67 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne PCSK1 0 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne PCSK6 0 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100483 EE On-Demand Anodyne POLG_WNV 60 32 O=C1CN[C@H](C(=O)N2CCSC2)C1 ZINC000147100676 BB For-Sale Anodyne DPP9 15 43 CC(C)(C)c1nc2cc(NC(=O)c3cccn(Cc4ccccc4)c3=O)ccc2o1 ZINC000147100681 HJ On-Demand Anodyne DRTS_PLAFK 18 40 CC(C)(C)c1nc2cc(NC(=O)c3cccn(Cc4ccccc4)c3=O)ccc2o1 ZINC000147100681 HJ On-Demand Anodyne PTGER3 25 40 CC(C)(C)c1nc2cc(NC(=O)c3cccn(Cc4ccccc4)c3=O)ccc2o1 ZINC000147100681 HJ On-Demand Anodyne NR2E3 63 34 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne GRIN2B 0 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne NPY1R 23 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne CTSK 19 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne PCSK2 0 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne SCN9A 0 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne GRIA1 40 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne PCSK7 0 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne PCSK5 60 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne FURIN 67 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne PCSK1 0 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne PCSK6 0 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147100691 EE On-Demand Anodyne POLG_WNV 60 32 O=C(Nc1ccc2nccnc2c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147100772 EH On-Demand Anodyne GRM4 71 42 O=C(Nc1ccc2nccnc2c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147100772 EH On-Demand Anodyne MAPK10 21 43 O=C(Nc1ccc2nccnc2c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147100772 EH On-Demand Anodyne TYK2 50 34 O=C(Nc1ccc2nccnc2c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147100772 EH On-Demand Anodyne NR2E3 67 41 O=C(Nc1ccc2nccnc2c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147100772 EH On-Demand Anodyne SHH 41 43 O=C(Nc1ccc2nccnc2c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147100772 EH On-Demand Anodyne SMO 24 40 O=C(Nc1ccc2nccnc2c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147100772 EH On-Demand Anodyne KCNK3 61 40 O=C1CN[C@@H](C(=O)N2CCSC2)C1 ZINC000147100861 BB For-Sale Anodyne DPP9 15 43 CCOCCO[C@@H](C)C(=O)Nc1ccc2oc(C(C)(C)C)nc2c1 ZINC000147100867 EH On-Demand Anodyne IMDH_CRYPV 45 46 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000147100879 GE On-Demand Anodyne GHRHR 40 32 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000147100879 GE On-Demand Anodyne P2RY12 205 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000147100879 GE On-Demand Anodyne THRB 28 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000147100879 GE On-Demand Anodyne TRY2_BOVIN 41 32 COCc1nc(C(=O)Nc2cc(OC)ccc2OC)cs1 ZINC000147100948 DF On-Demand Anodyne PYGL 15 40 COCc1nc(C(=O)Nc2cc(OC)ccc2OC)cs1 ZINC000147100948 DF On-Demand Anodyne PYGM 16 40 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne CHRM2 26 50 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne DRD2 31 48 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne DRD4 60 48 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne ACHE 52 56 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne SLC6A4 16 40 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne OPRM1 27 44 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne DRD3 29 47 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne OPRD1 19 41 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne OPRK1 32 42 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne AVPR1B 42 34 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne SLC6A3 18 48 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne CHRM3 24 50 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne LTA4H 50 48 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne HRH3 28 42 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne SIGMAR1 96 58 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne SSTR5 63 36 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne MMP13 34 48 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne BCHE 20 45 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne CCR3 53 38 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne CCR5 58 72 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne ADAM17 31 48 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne SLC18A3 20 40 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne MMP3 28 44 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne FAAH 18 42 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne SLC6A5 16 42 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne MMP9 37 48 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne PDK1 34 40 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne CXCR3 27 40 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne MMP1 35 48 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne MCHR1 62 58 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne CACNA1G 37 46 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne CCR8 36 46 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne MBTPS1 55 40 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne NOD1 16 41 COc1ccc(CC(=O)N(C)C2CCN(Cc3ccccc3)CC2)cc1 ZINC000147101016 FG On-Demand Anodyne NOD2 33 41 CCOCCO[C@H](C)C(=O)Nc1ccc2oc(C(C)(C)C)nc2c1 ZINC000147101038 EH On-Demand Anodyne IMDH_CRYPV 45 46 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000147101055 GE On-Demand Anodyne GHRHR 40 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000147101055 GE On-Demand Anodyne P2RY12 205 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000147101055 GE On-Demand Anodyne THRB 28 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CCOc2ccccc2Cl)CC1 ZINC000147101055 GE On-Demand Anodyne TRY2_BOVIN 41 32 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild FGFR1 17 67 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild FLT1 16 46 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild PRKAA1 28 60 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild FLT4 28 46 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild PDGFRA 57 75 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild CDK4 22 45 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild TGFBR1 65 75 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild CAMK1G 15 45 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild SRPK3 15 45 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild RIOK3 15 45 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild MAP3K7 15 45 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild PIP5K1A 15 45 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild RIOK1 15 45 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild LTK 19 60 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild PIP4K2B 15 45 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild GRK4 15 45 CCNC(=O)C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1 ZINC000147101163 JJ Annotated Mild AURKB-A 0 60 O=C(Nc1ccc2nccnc2c1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147101168 DI On-Demand Anodyne TYK2 45 40 O=C(Nc1ccc2nccnc2c1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147101168 DI On-Demand Anodyne NAMPT 25 42 CCOC(=O)NCC(=O)Nc1ccc2oc(C(C)(C)C)nc2c1 ZINC000147101283 DF On-Demand Anodyne CETP 40 39 O=C(Nc1ccc2nccnc2c1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147101350 DI On-Demand Anodyne TYK2 45 40 O=C(Nc1ccc2nccnc2c1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147101350 DI On-Demand Anodyne NAMPT 25 42 Cc1cc(C(=O)Nc2ccc(C)c(F)c2)cc([N+](=O)[O-])c1 ZINC000147101362 CH On-Demand Bother TAAR1 26 44 Cc1cc(C(=O)Nc2ccc(C)c(F)c2)cc([N+](=O)[O-])c1 ZINC000147101362 CH On-Demand Bother KCNK3 71 40 Cc1cc(C(=O)Nc2ccc(C)c(F)c2)cc([N+](=O)[O-])c1 ZINC000147101362 CH On-Demand Bother KCNK9 45 40 CC[C@@H](C)NC(=O)c1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147101378 GG On-Demand Anodyne PLD1 24 40 CC[C@@H](C)NC(=O)c1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147101378 GG On-Demand Anodyne PLD2 20 40 CC[C@@H](C)NC(=O)c1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147101378 GG On-Demand Anodyne CARM1 51 37 NC(N)=NNC(=O)c1ccccc1O ZINC000147101396 AB For-Sale Reactive KCNMA1 33 40 NC(N)=NNC(=O)c1ccccc1O ZINC000147101396 AB For-Sale Reactive PYK 92 37 O=C(O)CC[C@H](c1ccccc1)c1ccccc1F ZINC000147101468 CH For-Sale Anodyne FOLH1 26 40 O=C(O)CC[C@H](c1ccccc1)c1ccccc1F ZINC000147101468 CH For-Sale Anodyne NAALAD2 34 41 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne F2 58 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne PLG 43 46 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne ANPEP 19 41 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne TACR1 23 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne MC4R 35 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne TRY2_BOVIN 98 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne TRY1_BOVIN 32 48 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne CCKAR 0 43 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne CCR1 36 46 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne CCR5 52 39 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne DPP4 23 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne MTTP 15 42 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne CCKBR 0 43 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne CAPN1 18 41 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne EPHX2 33 47 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne DPP7 56 38 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne ST14 113 46 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne AMP1_PLAFQ 47 38 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne CACNA1G 53 47 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne TMPRSS11D 64 35 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne TMPRSS6 72 32 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101489 GH On-Demand Anodyne PDS 42 39 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne F2 42 40 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne ACE 26 46 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne OPRM1 27 44 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne OPRD1 15 40 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne TRHR 62 35 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne HLA-DRB3 52 33 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne TRY1_BOVIN 58 35 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne NTSR1 108 36 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne NTSR2 76 34 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne HLA-A 68 39 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne SORT1 48 33 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne SLC5A1 25 56 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne TPP2 31 40 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne XIAP 45 49 N[C@@H](CS)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N[C@@H](CS)C(=O)O ZINC000147101502 GA For-Sale Anodyne BRCA1 44 31 O=C(Nc1ccc2nccnc2c1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147101549 DI On-Demand Anodyne TYK2 45 40 O=C(Nc1ccc2nccnc2c1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147101549 DI On-Demand Anodyne NAMPT 25 42 CC[C@H](C)NC(=O)c1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147101561 GG On-Demand Anodyne PLD1 24 40 CC[C@H](C)NC(=O)c1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147101561 GG On-Demand Anodyne PLD2 20 40 CC[C@H](C)NC(=O)c1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147101561 GG On-Demand Anodyne CARM1 51 37 COc1cc(-c2cc(N3CCCC3)ccn2)nc(-c2cc(N3CCCC3)ccn2)c1 ZINC000147101644 HI For-Sale Anodyne GALR2 41 35 O=C(O)CC[C@@H](c1ccccc1)c1ccccc1F ZINC000147101663 CH For-Sale Anodyne FOLH1 26 40 O=C(O)CC[C@@H](c1ccccc1)c1ccccc1F ZINC000147101663 CH For-Sale Anodyne NAALAD2 34 41 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne F2 58 40 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne PLG 43 46 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne ANPEP 19 41 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne TACR1 23 40 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne MC4R 35 40 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne TRY2_BOVIN 98 44 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne TRY1_BOVIN 32 48 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne CCKAR 0 43 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne CCR1 36 46 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne CCR5 52 39 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne DPP4 23 40 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne MTTP 15 42 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne CCKBR 0 43 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne CAPN1 18 41 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne EPHX2 33 47 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne DPP7 56 38 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne ST14 113 46 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne AMP1_PLAFQ 47 38 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne CACNA1G 53 47 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne TMPRSS11D 64 35 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne TMPRSS6 72 32 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(C(=O)NCc2ccccc2)CC1 ZINC000147101692 GH On-Demand Anodyne PDS 42 39 O=C(Nc1ccc2nccnc2c1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147101722 DI On-Demand Anodyne TYK2 45 40 O=C(Nc1ccc2nccnc2c1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147101722 DI On-Demand Anodyne NAMPT 25 42 CN(C)C(=O)Cc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147101781 HD On-Demand Bother MMP2 15 40 CC(C)c1nc2cc(NC(=O)c3cccn(Cc4ccccc4)c3=O)ccc2o1 ZINC000147101918 GI On-Demand Anodyne DRTS_PLAFK 18 40 CC(C)c1nc2cc(NC(=O)c3cccn(Cc4ccccc4)c3=O)ccc2o1 ZINC000147101918 GI On-Demand Anodyne PTGER3 25 40 CC(C)c1nc2cc(NC(=O)c3cccn(Cc4ccccc4)c3=O)ccc2o1 ZINC000147101918 GI On-Demand Anodyne NR2E3 64 36 CC(C)c1nc2cc(NC(=O)c3cccn(Cc4ccccc4)c3=O)ccc2o1 ZINC000147101918 GI On-Demand Anodyne IMDH_CRYPV 43 38 O=C(Nc1ccc2nccnc2c1)[C@H]1C[C@H]1c1cccc(Br)c1 ZINC000147101926 FI On-Demand Anodyne NAMPT 25 42 NC(=O)c1ccc(OCC(=O)Nc2ccc(-c3ncc4n3CCCC4)cc2)cc1 ZINC000147101956 GG On-Demand Anodyne ADORA2B 44 46 NC(=O)c1ccc(OCC(=O)Nc2ccc(-c3ncc4n3CCCC4)cc2)cc1 ZINC000147101956 GG On-Demand Anodyne HIF1A 20 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc2nc(C)[nH]c2c1 ZINC000147101963 DE On-Demand Anodyne NOD1 41 32 COc1ccc(-c2cnc3ccc(NCC4CC4)nn23)cn1 ZINC000147101973 CF Annotated Anodyne IKBKB 37 59 COc1cccc(-c2nn(Cc3ccccc3)cc2C(=O)N2CCC(C#N)CC2)c1 ZINC000147101990 HH On-Demand Mild SIGMAR1 18 43 COc1cccc(-c2nn(Cc3ccccc3)cc2C(=O)N2CCC(C#N)CC2)c1 ZINC000147101990 HH On-Demand Mild DPP9 18 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccnc1Oc1ccccc1 ZINC000147102001 FE On-Demand Anodyne P2RY1 40 39 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccnc1Oc1ccccc1 ZINC000147102001 FE On-Demand Anodyne CPT1A 45 33 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccnc1Oc1ccccc1 ZINC000147102001 FE On-Demand Anodyne TNK2 42 33 CCOC[C@H](C)NS(=O)(=O)c1ccc(I)cc1 ZINC000147102032 FD On-Demand Anodyne MMP7 15 40 O=C(Nc1ccc2nccnc2c1)[C@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147102119 FI On-Demand Anodyne NAMPT 25 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)c1 ZINC000147102179 HE On-Demand Bother MMP13 64 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)c1 ZINC000147102179 HE On-Demand Bother MMP2 24 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)c1 ZINC000147102179 HE On-Demand Bother MMP3 54 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)c1 ZINC000147102179 HE On-Demand Bother MMP8 23 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)c1 ZINC000147102179 HE On-Demand Bother MMP9 43 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)c1 ZINC000147102179 HE On-Demand Bother CASP7 16 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)c1 ZINC000147102179 HE On-Demand Bother TGM2 31 40 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)c1 ZINC000147102179 HE On-Demand Bother MMP7 55 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)c1 ZINC000147102179 HE On-Demand Bother CA9 15 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)c1 ZINC000147102179 HE On-Demand Bother MMP1 64 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)c1 ZINC000147102179 HE On-Demand Bother NAMPT 73 46 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccnc1Oc1ccccc1 ZINC000147102194 FE On-Demand Anodyne P2RY1 40 39 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccnc1Oc1ccccc1 ZINC000147102194 FE On-Demand Anodyne CPT1A 45 33 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccnc1Oc1ccccc1 ZINC000147102194 FE On-Demand Anodyne TNK2 42 33 Nc1cccc(CC(=O)c2ccccc2)c1 ZINC000147102293 BF For-Sale Anodyne SRD5A2 15 50 Nc1cccc(CC(=O)c2ccccc2)c1 ZINC000147102293 BF For-Sale Anodyne PROTEASE 0 41 O=C(Nc1ccc2nccnc2c1)[C@@H]1C[C@H]1c1cccc(Br)c1 ZINC000147102312 FI On-Demand Anodyne NAMPT 25 42 Cc1cc(Nc2cccc(Cl)c2)nc(Nc2cccc(Cl)c2)n1 ZINC000147102347 EK For-Sale Anodyne CAMK2D 20 45 Cc1cc(Nc2cccc(Cl)c2)nc(Nc2cccc(Cl)c2)n1 ZINC000147102347 EK For-Sale Anodyne AGPAT2 39 42 Cc1cc(Nc2cccc(Cl)c2)nc(Nc2cccc(Cl)c2)n1 ZINC000147102347 EK For-Sale Anodyne EPHB4 17 43 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OC(F)(F)F)cc2)c1 ZINC000147102373 GG On-Demand Bother NQO2 41 36 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OC(F)(F)F)cc2)c1 ZINC000147102373 GG On-Demand Bother MTNR1A 53 37 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OC(F)(F)F)cc2)c1 ZINC000147102373 GG On-Demand Bother MTNR1B 45 37 CCOC(=O)Nc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147102435 DF On-Demand Mild NPY2R 24 41 CCOC(=O)Nc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147102435 DF On-Demand Mild ACR 41 33 CCOC(=O)Nc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147102435 DF On-Demand Mild L3MBTL3 75 39 O=C(CCSc1nc2ccccc2o1)Nc1ccccn1 ZINC000147102449 CG For-Sale Anodyne FAS 21 42 O=C(Nc1ccc2nccnc2c1)[C@@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147102535 FI On-Demand Anodyne NAMPT 25 42 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC)c1ccc(Cl)cc1 ZINC000147102595 EG On-Demand Anodyne NPY1R 15 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC)c1ccc(Cl)cc1 ZINC000147102595 EG On-Demand Anodyne POLG_WNV 69 30 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CC)c1ccc(Cl)cc1 ZINC000147102595 EG On-Demand Anodyne UTS2 46 37 NC(=O)c1ccc(OCC(=O)N2CC=C(c3c[nH]c4cc(F)ccc34)CC2)cc1 ZINC000147102647 GG On-Demand Anodyne HTR1D 22 53 NC(=O)c1ccc(OCC(=O)N2CC=C(c3c[nH]c4cc(F)ccc34)CC2)cc1 ZINC000147102647 GG On-Demand Anodyne SLC6A4 19 53 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc3nccnc3c1)C2 ZINC000147102734 EF On-Demand Anodyne MTNR1A 15 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc3nccnc3c1)C2 ZINC000147102734 EF On-Demand Anodyne ROCK2 41 54 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc3nccnc3c1)C2 ZINC000147102734 EF On-Demand Anodyne CDC42BPA 0 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC)c1ccc(Cl)cc1 ZINC000147102796 EG On-Demand Anodyne NPY1R 15 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC)c1ccc(Cl)cc1 ZINC000147102796 EG On-Demand Anodyne POLG_WNV 69 30 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CC)c1ccc(Cl)cc1 ZINC000147102796 EG On-Demand Anodyne UTS2 46 37 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc3nccnc3c1)C2 ZINC000147102941 EF On-Demand Anodyne MTNR1A 15 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc3nccnc3c1)C2 ZINC000147102941 EF On-Demand Anodyne ROCK2 41 54 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc3nccnc3c1)C2 ZINC000147102941 EF On-Demand Anodyne CDC42BPA 0 43 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother EDNRB 53 39 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother TACR1 0 45 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother TPR 15 44 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother MC4R 27 45 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother NQO2 23 40 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother CCKAR 25 43 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother BRS3 23 42 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother NMBR 72 38 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother GRPR 47 38 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother CCKBR 25 43 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother ALOX15 27 47 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother GABRA2 16 44 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother KISS1R 44 33 Cc1cc(C(=O)NCCc2c[nH]c3ccccc23)cc([N+](=O)[O-])c1 ZINC000147102955 DG On-Demand Bother MAPT 19 45 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC)c1ccc(Cl)cc1 ZINC000147102991 EG On-Demand Anodyne NPY1R 15 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC)c1ccc(Cl)cc1 ZINC000147102991 EG On-Demand Anodyne POLG_WNV 69 30 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CC)c1ccc(Cl)cc1 ZINC000147102991 EG On-Demand Anodyne UTS2 46 37 C[C@@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)NCc1ccccc1F ZINC000147103042 HH On-Demand Anodyne TRPV1 94 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC)c1ccc(Cl)cc1 ZINC000147103177 EG On-Demand Anodyne NPY1R 15 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC)c1ccc(Cl)cc1 ZINC000147103177 EG On-Demand Anodyne POLG_WNV 69 30 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CC)c1ccc(Cl)cc1 ZINC000147103177 EG On-Demand Anodyne UTS2 46 37 C[C@H](c1ccc(OC(F)(F)F)cc1)S(=O)(=O)CC(=O)NCc1ccccc1F ZINC000147103233 HH On-Demand Anodyne TRPV1 94 36 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCCOC)cc1 ZINC000147103234 DD On-Demand Anodyne MMP13 33 47 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCCOC)cc1 ZINC000147103234 DD On-Demand Anodyne MMP2 28 47 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCCOC)cc1 ZINC000147103234 DD On-Demand Anodyne MMP3 22 49 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCCOC)cc1 ZINC000147103234 DD On-Demand Anodyne MMP8 18 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCCOC)cc1 ZINC000147103234 DD On-Demand Anodyne MMP14 18 49 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCCOC)cc1 ZINC000147103234 DD On-Demand Anodyne MMP9 24 41 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCCOC)cc1 ZINC000147103234 DD On-Demand Anodyne MMP7 28 49 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCCOC)cc1 ZINC000147103234 DD On-Demand Anodyne ADAMTS4 62 37 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCCOC)cc1 ZINC000147103234 DD On-Demand Anodyne MMP1 21 49 O=C(Nc1ccc(-n2cccn2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147103239 FG On-Demand Anodyne DRTS_PLAFK 20 42 O=C(Nc1ccc(-n2cccn2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147103239 FG On-Demand Anodyne PTGER3 26 40 O=C(Nc1ccc(-n2cccn2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147103239 FG On-Demand Anodyne FLT1 18 40 O=C(Nc1ccc(-n2cccn2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147103239 FG On-Demand Anodyne PDE7A 23 42 O=C(Nc1ccc(-n2cccn2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147103239 FG On-Demand Anodyne AMP1_PLAFQ 54 39 O=C(Nc1ccc(-n2cccn2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147103239 FG On-Demand Anodyne NR2E3 51 32 Cc1onc(-c2ccccc2)c1C(=O)N1CCC(C#N)CC1 ZINC000147103272 CG On-Demand Mild GPBAR1 25 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103360 GF On-Demand Anodyne NPY1R 30 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103360 GF On-Demand Anodyne KLK3 48 36 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103360 GF On-Demand Anodyne CTSK 23 45 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103360 GF On-Demand Anodyne GRIA1 47 35 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103360 GF On-Demand Anodyne PCSK5 48 39 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103360 GF On-Demand Anodyne FURIN 73 39 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103360 GF On-Demand Anodyne POLG_WNV 67 35 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne F2 33 44 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne SIGMAR1 15 51 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne MMP13 25 42 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne P2RX7 37 43 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne BCHE 0 40 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne CCR5 17 44 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne PREP 24 43 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne MTNR1A 19 43 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne MTNR1B 17 43 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne EPHX2 34 47 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne AMP1_PLAFQ 44 38 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne CACNA1G 43 40 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne SCD 23 41 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne TMPRSS11D 64 35 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne PDS 56 36 CC(C)Oc1cccc(CC(=O)N2CCC(C(=O)NCc3ccccc3)CC2)c1 ZINC000147103376 GH On-Demand Anodyne PANK3 0 46 C[C@H](NC(=O)c1ccn(-c2cccc(F)c2)n1)c1ccc2c(c1)CCC(=O)N2 ZINC000147103459 GG In-Stock Anodyne GRIN2B 17 49 CCCc1ccccc1NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147103499 EI On-Demand Anodyne DRTS_PLAFK 20 44 CCCc1ccccc1NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147103499 EI On-Demand Anodyne PTGER3 34 47 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103533 GF On-Demand Anodyne NPY1R 30 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103533 GF On-Demand Anodyne KLK3 48 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103533 GF On-Demand Anodyne CTSK 23 45 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103533 GF On-Demand Anodyne GRIA1 47 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103533 GF On-Demand Anodyne PCSK5 48 39 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103533 GF On-Demand Anodyne FURIN 73 39 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COCC(F)(F)F)cc1 ZINC000147103533 GF On-Demand Anodyne POLG_WNV 67 35 C[C@@H](NC(=O)c1ccn(-c2cccc(F)c2)n1)c1ccc2c(c1)CCC(=O)N2 ZINC000147103659 GG In-Stock Anodyne GRIN2B 17 49 COc1cnc(C(=O)Nc2ccc(F)c([C@@]3(C)N=C(N)SC=C3C)c2)cn1 ZINC000147103695 GG Annotated Anodyne BACE2 54 50 COc1cnc(C(=O)Nc2ccc(F)c([C@@]3(C)N=C(N)SC=C3C)c2)cn1 ZINC000147103695 GG Annotated Anodyne BACE1 26 59 COCc1nc(C(=O)Nc2nc3ccc(C)cc3s2)cs1 ZINC000147103812 DG On-Demand Anodyne HSD17B1 29 42 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)NCC(F)(F)F)C2 ZINC000147104001 ED On-Demand Anodyne ROCK2 24 41 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother MAOB 21 40 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother LTA4H 17 40 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother NQO2 28 40 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother PTGER3 53 39 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother MTNR1A 65 45 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother MTNR1B 60 45 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother SLC6A5 37 42 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother TAAR1 34 47 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother FFAR1 45 44 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother AKR1C3 15 43 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother FFAR4 45 38 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2ccc(OCc3ccccc3)cc2)c1 ZINC000147104071 HI On-Demand Bother AKR1C2 29 43 CCCN1C(=O)c2ccccc2N[C@H]1c1ccc(OC)c(OCCCC#N)c1 ZINC000147104494 GI On-Demand Mild TSHR 63 51 CCc1cccc(Oc2ccc(NC(=O)c3cc(OC)ccc3[N+](=O)[O-])cn2)c1 ZINC000147104508 GJ On-Demand Bother MTNR1B 21 42 CCc1cccc(Oc2ccc(NC(=O)c3cc(OC)ccc3[N+](=O)[O-])cn2)c1 ZINC000147104508 GJ On-Demand Bother TAAR1 32 49 CC1=CSC(N)=N[C@]1(C)c1cc(NC(=O)c2cnc(C)cn2)ccc1F ZINC000147104554 FG Annotated Anodyne BACE2 60 55 CC1=CSC(N)=N[C@]1(C)c1cc(NC(=O)c2cnc(C)cn2)ccc1F ZINC000147104554 FG Annotated Anodyne BACE1 29 51 Cc1cc(C)n(-c2ccc(NC(=O)c3cccn(Cc4ccccc4)c3=O)cn2)n1 ZINC000147104612 GG On-Demand Anodyne DRTS_PLAFK 18 40 Cc1cc(C)n(-c2ccc(NC(=O)c3cccn(Cc4ccccc4)c3=O)cn2)n1 ZINC000147104612 GG On-Demand Anodyne PTGER3 25 40 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne ABL1 20 42 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne ESR1 28 47 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne LTA4H 38 40 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne SRC 27 48 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne JAK3 25 71 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne JAK2 38 71 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne YES1 24 46 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne TNK2 24 44 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne WEE1 17 44 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne PSMB2 46 35 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne PSMB1 40 35 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1 ZINC000147104635 JI Annotated Anodyne TBK1 15 44 CCCCOc1cccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147104672 HG On-Demand Bother MMP13 21 40 CCCCOc1cccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147104672 HG On-Demand Bother PLA2G4B 58 40 CCCCOc1cccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147104672 HG On-Demand Bother PDS 43 42 CCCN1C(=O)c2ccccc2N[C@@H]1c1ccc(OC)c(OCCCC#N)c1 ZINC000147104677 GI On-Demand Mild TSHR 63 51 NC(=O)COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147104688 EC On-Demand Anodyne PRSS1 17 42 NC(=O)COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147104688 EC On-Demand Anodyne LTA4H 34 44 NC(=O)COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147104688 EC On-Demand Anodyne ADORA2B 45 48 NC(=O)COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147104688 EC On-Demand Anodyne ACR 77 40 NC(=O)COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147104688 EC On-Demand Anodyne HIF1A 23 46 O=C(c1ccc2c(c1)COC2)N1CCN(c2ncc(Cl)cc2Cl)CC1 ZINC000147104766 GG On-Demand Anodyne CXCR3 23 40 N#CC1CCN(C(=O)[C@H]2CCCN(S(=O)(=O)c3ccc(F)cc3)C2)CC1 ZINC000147104775 GD On-Demand Mild TGM2 21 41 N#CC1CCN(C(=O)[C@H]2CCCN(S(=O)(=O)c3ccc(F)cc3)C2)CC1 ZINC000147104775 GD On-Demand Mild F13A1 25 41 N#CC1CCN(C(=O)[C@H]2CCCN(S(=O)(=O)c3ccc(F)cc3)C2)CC1 ZINC000147104775 GD On-Demand Mild NAMPT 18 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(C)c(C(N)=O)c1 ZINC000147104777 DC On-Demand Anodyne LEF 60 40 CCOC(=O)N1CCC[C@H](C(=O)OC(C)(C)C)C1 ZINC000147104823 CE Annotated Anodyne PREP 20 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(Oc3ccc(C)c(C)c3)nc2)c1 ZINC000147104878 GJ On-Demand Bother TAAR1 27 42 COCCOc1cc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)ccc1OC ZINC000147104932 HD On-Demand Anodyne CYSLTR1 22 42 COCCOc1cc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)ccc1OC ZINC000147104932 HD On-Demand Anodyne CCR3 20 43 COCCOc1cc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)ccc1OC ZINC000147104932 HD On-Demand Anodyne EPHX2 41 40 COCCOc1cc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)ccc1OC ZINC000147104932 HD On-Demand Anodyne ENPP1 69 32 COc1cc(C(=O)N2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)ccc1C ZINC000147104955 HH On-Demand Anodyne HRH3 24 40 COc1cc(C(=O)N2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)ccc1C ZINC000147104955 HH On-Demand Anodyne NPBWR1 42 31 N#CC1CCN(C(=O)[C@@H]2CCCN(S(=O)(=O)c3ccc(F)cc3)C2)CC1 ZINC000147104978 GD On-Demand Mild TGM2 21 41 N#CC1CCN(C(=O)[C@@H]2CCCN(S(=O)(=O)c3ccc(F)cc3)C2)CC1 ZINC000147104978 GD On-Demand Mild F13A1 25 41 N#CC1CCN(C(=O)[C@@H]2CCCN(S(=O)(=O)c3ccc(F)cc3)C2)CC1 ZINC000147104978 GD On-Demand Mild NAMPT 18 40 COCCOc1cc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)ccc1OC ZINC000147105115 HD On-Demand Anodyne CCR3 20 43 COCCOc1cc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)ccc1OC ZINC000147105115 HD On-Demand Anodyne EPHX2 41 40 COCCOc1cc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)ccc1OC ZINC000147105115 HD On-Demand Anodyne ENPP1 69 32 COc1cc(C(=O)N2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)ccc1C ZINC000147105131 HH On-Demand Anodyne HRH3 24 40 COc1cc(C(=O)N2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)ccc1C ZINC000147105131 HH On-Demand Anodyne NPBWR1 42 31 Cc1cc(C(=O)Nc2ccccc2N2CCCCC2)cc([N+](=O)[O-])c1 ZINC000147105202 EI On-Demand Bother KCNQ2 94 47 Cc1cc(C(=O)Nc2ccccc2N2CCCCC2)cc([N+](=O)[O-])c1 ZINC000147105202 EI On-Demand Bother CSF1R 22 63 Cc1cc(C(=O)Nc2ccccc2N2CCCCC2)cc([N+](=O)[O-])c1 ZINC000147105202 EI On-Demand Bother TAAR1 31 43 Cc1cc(C(=O)Nc2ccccc2N2CCCCC2)cc([N+](=O)[O-])c1 ZINC000147105202 EI On-Demand Bother WDR5 39 45 O=C(NCc1ccc(Cl)cc1Cl)c1ccnc(O)c1 ZINC000147105231 CG On-Demand Anodyne P2RX7 60 50 O=C(NCc1ccc(Cl)cc1Cl)c1ccnc(O)c1 ZINC000147105231 CG On-Demand Anodyne SCN10A 35 44 O=C(NCc1ccc(Cl)cc1Cl)c1ccnc(O)c1 ZINC000147105231 CG On-Demand Anodyne ALPL 42 34 CC[C@@H](COc1ccccc1OC)OC ZINC000147105302 BE On-Demand Anodyne PDS 41 37 COc1cc(C(=O)N2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)ccc1C ZINC000147105321 HH On-Demand Anodyne HRH3 24 40 COc1cc(C(=O)N2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)ccc1C ZINC000147105321 HH On-Demand Anodyne NPBWR1 42 31 COCCOc1cc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)ccc1OC ZINC000147105365 HG On-Demand Anodyne NOS2 74 34 COCCOc1cc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)ccc1OC ZINC000147105365 HG On-Demand Anodyne ROCK2 24 49 COCCOc1cc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)ccc1OC ZINC000147105365 HG On-Demand Anodyne MET 59 34 COCCOc1cc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)ccc1OC ZINC000147105365 HG On-Demand Anodyne QPCT 25 49 COCCOc1cc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)ccc1OC ZINC000147105365 HG On-Demand Anodyne ENPP1 68 33 COCCOc1cc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)ccc1OC ZINC000147105365 HG On-Demand Anodyne DRTS_TRYCR 50 37 COCCOc1cc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)ccc1OC ZINC000147105365 HG On-Demand Anodyne NAMPT 18 40 CCCOCC(=O)Nc1cc(C(N)=O)ccc1N1CCCC1 ZINC000147105382 DD On-Demand Anodyne KCNQ2 78 39 CC[C@H](COc1ccccc1OC)OC ZINC000147105462 BE On-Demand Anodyne PDS 41 37 NC(=O)c1ccc(OCC(=O)N2CCN(c3ncnc4sccc34)CC2)cc1 ZINC000147105479 GD On-Demand Anodyne PDGFRB 51 37 NC(=O)c1ccc(OCC(=O)N2CCN(c3ncnc4sccc34)CC2)cc1 ZINC000147105479 GD On-Demand Anodyne SIRT3 50 31 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)OC)cc1 ZINC000147105532 DD On-Demand Anodyne MMP2 24 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)OC)cc1 ZINC000147105532 DD On-Demand Anodyne MMP14 15 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)OC)cc1 ZINC000147105532 DD On-Demand Anodyne MMP9 19 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)OC)cc1 ZINC000147105532 DD On-Demand Anodyne MMP7 20 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)OC)cc1 ZINC000147105532 DD On-Demand Anodyne ADAMTS4 49 40 COCCOc1cc(NC(=O)N2C[C@H](c3ccccc3)O[C@H](C)C2)ccc1OC ZINC000147105572 HH On-Demand Anodyne PDGFRB 44 43 COCCOc1cc(NC(=O)N2C[C@H](c3ccccc3)O[C@H](C)C2)ccc1OC ZINC000147105572 HH On-Demand Anodyne ENPP1 67 33 CCCC[C@H](NC(N)=O)C(=O)Nc1cc(C(N)=O)ccc1N1CCCC1 ZINC000147105586 FD On-Demand Anodyne KCNQ2 79 43 N#CC1CCN(C(=O)[C@H]2CCCN(C(=O)Nc3ccccc3)C2)CC1 ZINC000147105607 EF On-Demand Mild DHODH 41 40 N#CC1CCN(C(=O)[C@H]2CCCN(C(=O)Nc3ccccc3)C2)CC1 ZINC000147105607 EF On-Demand Mild DPP4 26 44 N#CC1CCN(C(=O)[C@H]2CCCN(C(=O)Nc3ccccc3)C2)CC1 ZINC000147105607 EF On-Demand Mild PREP 56 38 COc1ccc([C@H]2Nc3ccccc3C(=O)N2C)cc1OCCCC#N ZINC000147105623 FH On-Demand Mild TSHR 58 43 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne INHA 40 38 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne HDAC8 18 45 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne HDAC10 36 44 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne PLA2G4B 50 31 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne HDAC1 24 46 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne HDAC2 27 45 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne HDAC3 45 46 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne HDAC6 37 43 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne HDAC9 15 45 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne ENPP2 37 51 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne NOD1 49 38 CCCCCCCCCCCC(=O)Nc1ccc(C(=O)O)c(O)c1 ZINC000147105649 EJ For-Sale Anodyne CQSS 48 30 Cc1cc(C(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2C)cc([N+](=O)[O-])c1 ZINC000147105708 HE On-Demand Bother CNR2 15 42 Cc1cc(C(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2C)cc([N+](=O)[O-])c1 ZINC000147105708 HE On-Demand Bother NR1H4 15 40 COCCOc1cc(NC(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)ccc1OC ZINC000147105745 HH On-Demand Anodyne PDGFRB 44 43 COCCOc1cc(NC(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)ccc1OC ZINC000147105745 HH On-Demand Anodyne ENPP1 67 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1cc(C(N)=O)ccc1N1CCCC1 ZINC000147105758 FD On-Demand Anodyne KCNQ2 79 43 Cc1cnc(C(=O)Nc2cccc([C@]3(C(F)(F)F)CCSC(N)=N3)c2)cn1 ZINC000147105772 GG Annotated Anodyne BACE2 48 51 Cc1cnc(C(=O)Nc2cccc([C@]3(C(F)(F)F)CCSC(N)=N3)c2)cn1 ZINC000147105772 GG Annotated Anodyne BACE1 22 49 COCCOc1cc(NC(=O)N2C[C@@H](C)O[C@H](c3ccccc3)C2)ccc1OC ZINC000147105826 HH On-Demand Anodyne PDGFRB 44 43 COCCOc1cc(NC(=O)N2C[C@@H](C)O[C@H](c3ccccc3)C2)ccc1OC ZINC000147105826 HH On-Demand Anodyne ENPP1 67 33 N#CC1CCN(C(=O)[C@@H]2CCCN(C(=O)Nc3ccccc3)C2)CC1 ZINC000147105829 EF On-Demand Mild DPP4 26 44 N#CC1CCN(C(=O)[C@@H]2CCCN(C(=O)Nc3ccccc3)C2)CC1 ZINC000147105829 EF On-Demand Mild PREP 56 38 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccc3c(c2)CCC(=O)N3)c1 ZINC000147105854 FF On-Demand Bother GRIN2B 15 45 Cc1cnc(C(=O)Nc2cccc([C@@]3(C(F)(F)F)CCSC(N)=N3)c2)cn1 ZINC000147105961 GG Annotated Anodyne BACE2 48 51 Cc1cnc(C(=O)Nc2cccc([C@@]3(C(F)(F)F)CCSC(N)=N3)c2)cn1 ZINC000147105961 GG Annotated Anodyne BACE1 22 49 CCN(C(=O)CS(=O)(=O)[C@H](C)c1ccc(OC(F)(F)F)cc1)c1ccccc1 ZINC000147105994 HI On-Demand Anodyne HCRTR2 15 40 COCCOc1cc(NC(=O)N2C[C@H](C)O[C@H](c3ccccc3)C2)ccc1OC ZINC000147106021 HH On-Demand Anodyne PDGFRB 44 43 COCCOc1cc(NC(=O)N2C[C@H](C)O[C@H](c3ccccc3)C2)ccc1OC ZINC000147106021 HH On-Demand Anodyne ENPP1 67 33 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccc3c(c2)CCC(=O)N3)c1 ZINC000147106025 FF On-Demand Bother GRIN2B 15 45 N#CC1CCN(C(=O)c2csc(-c3ccsc3)n2)CC1 ZINC000147106047 DG For-Sale Mild TRPC6 52 38 C[C@@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106059 BD For-Sale Anodyne BMP1 67 39 C[C@@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106059 BD For-Sale Anodyne CHRNA4 59 55 C[C@@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106059 BD For-Sale Anodyne MMP14 23 43 C[C@@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106059 BD For-Sale Anodyne CAPN2 39 47 COCCOc1cc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)ccc1OC ZINC000147106214 HI On-Demand Anodyne TSHR 46 30 COCCOc1cc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)ccc1OC ZINC000147106214 HI On-Demand Anodyne MCHR1 15 43 COCCOc1cc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)ccc1OC ZINC000147106214 HI On-Demand Anodyne ENPP1 61 31 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne F2 68 41 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne ACE 47 46 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne FKBP1A 55 46 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne LHCGR 33 44 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne SSTR2 81 37 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne OPRM1 42 52 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne OPRD1 36 48 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne CELA1 27 52 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne ELANE 29 41 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne MME 28 46 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne EDNRA 34 42 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne TACR1 43 48 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne MC4R 37 45 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne CTRA_BOVIN 66 36 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne BMP1 27 40 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne SSTR4 40 37 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne TACR2 44 48 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne TRY1_BOVIN 71 38 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne CCKAR 87 52 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne NTSR1 53 39 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne CTSG 45 36 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne BCHE 18 40 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne BRS3 28 44 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne C3AR1 17 44 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne HLA-A 33 41 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne PREP 73 52 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne NMBR 44 42 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne MC3R 63 47 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne MC5R 48 54 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne MMP8 59 37 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne MMP14 77 37 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne ECE1 45 39 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne CELA2A 54 36 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne LGMN 88 50 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne SSTR3 46 37 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne MMP11 93 37 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne CCKBR 93 47 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne GHSR 63 38 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne MMP9 17 45 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne MC1R 68 47 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne KLK5 27 46 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne C5AR1 43 42 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne XIAP 39 45 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne RHODESAIN 0 40 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne KISS1R 50 30 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne F1PEP1 0 52 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne TMPRSS11D 71 40 O=C(NCCc1c[nH]c2ccccc12)[C@@H]1CCCN1C(=O)OCc1ccccc1 ZINC000147106220 GH On-Demand Anodyne DSBA 0 41 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne MME 53 40 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne ANPEP 41 42 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne HRAS 50 35 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CASP3 22 46 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne BMP1 67 39 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne KLK3 74 41 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CTSB 79 51 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne PAPA1_CARPA 70 48 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CYSP_TRYCR 60 43 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CTSK 40 52 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CTSL 47 48 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne PGA 22 41 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CHRNA4 59 55 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne AMY2 52 29 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CAPNS1 71 46 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne MMP14 23 43 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne LGMN 17 41 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CTSS 22 54 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CAPN1 97 48 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CASP1 27 43 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CAPN2 132 48 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne ACE2 43 35 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CASP6 34 45 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne CASP9 38 45 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne TPSAB1 21 41 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne NPR 87 53 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne NAAA 45 33 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne PSMB5 45 40 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne SLC12A5 48 35 C[C@H](CNC(=O)OCc1ccccc1)N(C)C ZINC000147106233 BD For-Sale Anodyne PDS 47 38 OC[C@H]1O[C@@H](Oc2ccccn2)[C@H](O)[C@@H](O)[C@H]1O ZINC000147106243 CA For-Sale Anodyne TYR 23 44 OC[C@H]1O[C@@H](Oc2ccccn2)[C@H](O)[C@@H](O)[C@H]1O ZINC000147106243 CA For-Sale Anodyne SLC29A1 56 32 OC[C@H]1O[C@@H](Oc2ccccn2)[C@H](O)[C@@H](O)[C@H]1O ZINC000147106243 CA For-Sale Anodyne VEGFA 38 43 OC[C@H]1O[C@@H](Oc2ccccn2)[C@H](O)[C@@H](O)[C@H]1O ZINC000147106243 CA For-Sale Anodyne ADK 53 37 OC[C@H]1O[C@@H](Oc2ccccn2)[C@H](O)[C@@H](O)[C@H]1O ZINC000147106243 CA For-Sale Anodyne SLC5A1 74 44 OC[C@H]1O[C@@H](Oc2ccccn2)[C@H](O)[C@@H](O)[C@H]1O ZINC000147106243 CA For-Sale Anodyne SLC5A2 97 47 OC[C@H]1O[C@@H](Oc2ccccn2)[C@H](O)[C@@H](O)[C@H]1O ZINC000147106243 CA For-Sale Anodyne FIMH 118 63 OC[C@H]1O[C@@H](Oc2ccccn2)[C@H](O)[C@@H](O)[C@H]1O ZINC000147106243 CA For-Sale Anodyne SLC5A4 21 47 COc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1F ZINC000147106250 FE On-Demand Bother COLA 66 38 COc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1F ZINC000147106250 FE On-Demand Bother CPT1A 63 38 COc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1F ZINC000147106250 FE On-Demand Bother CPT2 46 38 COc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1F ZINC000147106250 FE On-Demand Bother CPT1B 43 36 COc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1F ZINC000147106250 FE On-Demand Bother TAAR1 29 45 COc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1F ZINC000147106250 FE On-Demand Bother ENPP1 60 31 COCCOc1cc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)ccc1OC ZINC000147106407 HI On-Demand Anodyne TSHR 46 30 COCCOc1cc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)ccc1OC ZINC000147106407 HI On-Demand Anodyne MCHR1 15 43 COCCOc1cc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)ccc1OC ZINC000147106407 HI On-Demand Anodyne ENPP1 61 31 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106531 FG On-Demand Anodyne PTGER4 15 42 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106531 FG On-Demand Anodyne ACACA 22 42 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106531 FG On-Demand Anodyne ACACB 29 44 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106531 FG On-Demand Anodyne PPARD 41 36 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106531 FG On-Demand Anodyne MTTP 41 33 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106531 FG On-Demand Anodyne F7 30 40 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106531 FG On-Demand Anodyne ACR 24 40 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106531 FG On-Demand Anodyne AOC3 20 47 COCCOc1cc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)ccc1OC ZINC000147106604 HI On-Demand Anodyne TSHR 46 30 COCCOc1cc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)ccc1OC ZINC000147106604 HI On-Demand Anodyne MCHR1 15 43 COCCOc1cc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)ccc1OC ZINC000147106604 HI On-Demand Anodyne ENPP1 61 31 COc1ccc([C@@H]2Nc3ccccc3C(=O)N2Cc2ccco2)cc1OCCCC#N ZINC000147106616 HJ On-Demand Mild TSHR 67 44 CC(C)Oc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147106680 GG On-Demand Bother GCK 32 45 CC(C)Oc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147106680 GG On-Demand Bother USP47 46 39 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106705 FG On-Demand Anodyne PTGER4 15 42 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106705 FG On-Demand Anodyne ACACA 22 42 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106705 FG On-Demand Anodyne ACACB 29 44 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106705 FG On-Demand Anodyne PPARD 41 36 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106705 FG On-Demand Anodyne MTTP 41 33 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106705 FG On-Demand Anodyne F7 30 40 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106705 FG On-Demand Anodyne ACR 24 40 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(C(F)(F)F)cc1 ZINC000147106705 FG On-Demand Anodyne AOC3 20 47 CCOC[C@H](C)NS(=O)(=O)c1ccc(OCCOC)c(C)c1 ZINC000147106730 ED On-Demand Anodyne LEF 57 41 COCCOc1cc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)ccc1OC ZINC000147106732 HI On-Demand Anodyne TSHR 46 30 COCCOc1cc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)ccc1OC ZINC000147106732 HI On-Demand Anodyne MCHR1 15 43 COCCOc1cc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)ccc1OC ZINC000147106732 HI On-Demand Anodyne ENPP1 61 31 CC[C@@H](/C=C/c1ccccc1)C(=O)O ZINC000147106762 AF For-Sale Anodyne ACE2 48 34 CC[C@@H](/C=C/c1ccccc1)C(=O)O ZINC000147106762 AF For-Sale Anodyne GRIK1 21 40 N#CC1CCN(C(=O)CCc2nc(-c3ccsc3)no2)CC1 ZINC000147106873 DE On-Demand Mild ETHR 72 40 CCOC(=O)NCC(=O)Nc1ccc2oc(C(C)C)nc2c1 ZINC000147106907 DF On-Demand Anodyne ENPP1 49 30 CCOC(=O)NCC(=O)Nc1ccc2oc(C(C)C)nc2c1 ZINC000147106907 DF On-Demand Anodyne IMDH_CRYPV 41 38 CCCOc1ccc(S(=O)(=O)N[C@@H](C)COCC)cc1 ZINC000147106947 DE On-Demand Anodyne MMP13 26 48 CCCOc1ccc(S(=O)(=O)N[C@@H](C)COCC)cc1 ZINC000147106947 DE On-Demand Anodyne MMP2 18 48 CCCOc1ccc(S(=O)(=O)N[C@@H](C)COCC)cc1 ZINC000147106947 DE On-Demand Anodyne MMP7 25 48 CCCOc1ccc(S(=O)(=O)N[C@@H](C)COCC)cc1 ZINC000147106947 DE On-Demand Anodyne ADAMTS4 50 36 CCCOc1ccc(S(=O)(=O)N[C@@H](C)COCC)cc1 ZINC000147106947 DE On-Demand Anodyne MMP1 15 48 COCCOc1ccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147106948 HG On-Demand Anodyne ADRB1 19 40 COCCOc1ccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147106948 HG On-Demand Anodyne HRH2 26 40 COCCOc1ccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147106948 HG On-Demand Anodyne ROCK2 27 42 COCCOc1ccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147106948 HG On-Demand Anodyne EPHX2 41 38 COC(=O)c1cc(NC(=O)CCNC(=O)OC(C)(C)C)cn1C ZINC000147107010 ED On-Demand Anodyne HRAS 41 32 N#CC1CCN(C(=O)c2ccc(-c3ccc(F)cc3)o2)CC1 ZINC000147107023 CG On-Demand Mild SCN10A 15 51 COCCN1C(=O)c2ccccc2N[C@H]1c1ccc(OC)c(OCCCC#N)c1 ZINC000147107027 GH On-Demand Mild TSHR 62 48 Cn1cc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cn1 ZINC000147107095 DD On-Demand Anodyne DRTS_PLAFK 20 44 Cn1cc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cn1 ZINC000147107095 DD On-Demand Anodyne PTGER3 29 42 Cn1cc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cn1 ZINC000147107095 DD On-Demand Anodyne ITK 40 44 Cn1cc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cn1 ZINC000147107095 DD On-Demand Anodyne PANC 47 37 COCCOc1ccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147107151 HG On-Demand Anodyne ADRB1 19 40 COCCOc1ccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147107151 HG On-Demand Anodyne HRH2 26 40 COCCOc1ccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147107151 HG On-Demand Anodyne ROCK2 27 42 COCCOc1ccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147107151 HG On-Demand Anodyne EPHX2 41 38 Cc1cc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2[nH]1 ZINC000147107162 DF On-Demand Anodyne ADORA2A 17 48 Cc1cc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2[nH]1 ZINC000147107162 DF On-Demand Anodyne ADORA2B 50 48 Cc1cc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2[nH]1 ZINC000147107162 DF On-Demand Anodyne CETP 28 40 Cc1cc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2[nH]1 ZINC000147107162 DF On-Demand Anodyne CHEK2 73 39 Cc1cc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2[nH]1 ZINC000147107162 DF On-Demand Anodyne ACR 55 35 Cc1cc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2[nH]1 ZINC000147107162 DF On-Demand Anodyne HIF1A 22 41 Cc1cc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2[nH]1 ZINC000147107162 DF On-Demand Anodyne ENPP1 58 33 COCCN1C(=O)c2ccccc2N[C@@H]1c1ccc(OC)c(OCCCC#N)c1 ZINC000147107216 GH On-Demand Mild TSHR 62 48 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne FKBP1A 21 43 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne BMP1 92 38 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne SIGMAR1 17 49 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne MMP13 55 43 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne CSNK1D 19 45 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne ADAM17 35 42 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne MTNR1A 49 34 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne MMP2 38 40 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne MMP3 62 44 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne MMP8 42 42 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne MMP9 59 43 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne MMP12 28 40 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne MMP7 55 44 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne CA9 21 48 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne MMP1 72 46 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne PROKR1 52 33 COc1ccc(CC(=O)NN2CCCC2)cc1 ZINC000147107230 BD On-Demand Anodyne H9B8T9_CAPHI 20 40 CS(=O)(=O)NCCC(=O)Nc1ccc(-n2cccn2)cc1 ZINC000147107276 DC On-Demand Anodyne AMP1_PLAFQ 54 37 CS(=O)(=O)NCCC(=O)Nc1ccc(-n2cccn2)cc1 ZINC000147107276 DC On-Demand Anodyne LAP 0 44 CS(=O)(=O)c1cc(C(=O)Nc2ccc(Cl)c(F)c2)cc([N+](=O)[O-])c1 ZINC000147107331 FG On-Demand Bother MAOB 17 42 CS(=O)(=O)c1cc(C(=O)Nc2ccc(Cl)c(F)c2)cc([N+](=O)[O-])c1 ZINC000147107331 FG On-Demand Bother ENV 49 40 CS(=O)(=O)c1cc(C(=O)Nc2ccc(Cl)c(F)c2)cc([N+](=O)[O-])c1 ZINC000147107331 FG On-Demand Bother SHH 44 45 CS(=O)(=O)c1cc(C(=O)Nc2ccc(Cl)c(F)c2)cc([N+](=O)[O-])c1 ZINC000147107331 FG On-Demand Bother USP7 28 40 CS(=O)(=O)c1cc(C(=O)Nc2ccc(Cl)c(F)c2)cc([N+](=O)[O-])c1 ZINC000147107331 FG On-Demand Bother USP47 35 40 COCCOc1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147107338 HG On-Demand Anodyne TSHR 41 32 COCCOc1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147107338 HG On-Demand Anodyne HRH2 49 49 COCCOc1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147107338 HG On-Demand Anodyne CCR3 23 41 COCCOc1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147107338 HG On-Demand Anodyne ROCK2 23 40 COCCOc1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147107338 HG On-Demand Anodyne EPHX2 37 43 COCCOc1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147107535 HG On-Demand Anodyne TSHR 41 32 COCCOc1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147107535 HG On-Demand Anodyne HRH2 49 49 COCCOc1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147107535 HG On-Demand Anodyne CCR3 23 41 COCCOc1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147107535 HG On-Demand Anodyne ROCK2 23 40 COCCOc1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147107535 HG On-Demand Anodyne EPHX2 37 43 O=C(Nc1ccc(Cl)c(F)c1)c1ccn(-c2cccc(F)c2)n1 ZINC000147107549 EI On-Demand Anodyne MAOB 16 41 O=C(Nc1ccc(Cl)c(F)c1)c1ccn(-c2cccc(F)c2)n1 ZINC000147107549 EI On-Demand Anodyne GRM4 50 39 O=C(Nc1ccc(Cl)c(F)c1)c1ccn(-c2cccc(F)c2)n1 ZINC000147107549 EI On-Demand Anodyne ENV 41 37 CCOC[C@H](C)NS(=O)(=O)c1cccc(C(=O)OC)c1 ZINC000147107558 DD On-Demand Anodyne ADAMTS4 23 44 NC1=N[C@@](c2cccc(F)c2)(c2cccc(NC(=O)c3ncc(Cl)cc3Cl)c2)CS1 ZINC000147107590 JK Annotated Anodyne BACE2 55 51 NC1=N[C@@](c2cccc(F)c2)(c2cccc(NC(=O)c3ncc(Cl)cc3Cl)c2)CS1 ZINC000147107590 JK Annotated Anodyne BACE1 22 51 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1OC1CCCC1)C2 ZINC000147107694 FI On-Demand Anodyne ROCK2 36 51 NC1=N[C@](c2cccc(F)c2)(c2cccc(NC(=O)c3ncc(Cl)cc3Cl)c2)CS1 ZINC000147107771 JK Annotated Anodyne BACE2 55 51 NC1=N[C@](c2cccc(F)c2)(c2cccc(NC(=O)c3ncc(Cl)cc3Cl)c2)CS1 ZINC000147107771 JK Annotated Anodyne BACE1 22 51 CN(C)c1cc2ccccc2[nH]1 ZINC000147107794 AE In-Stock Anodyne DDO 0 42 COCCOc1ccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147107805 GF On-Demand Anodyne PDGFRB 49 41 COCCOc1ccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147107805 GF On-Demand Anodyne EPHX2 54 40 COCc1nc(C(=O)Nc2ccc(C)c(S(=O)(=O)N3CCCCC3)c2)cs1 ZINC000147107909 HG On-Demand Anodyne LPL 35 40 COCc1nc(C(=O)Nc2ccc(C)c(S(=O)(=O)N3CCCCC3)c2)cs1 ZINC000147107909 HG On-Demand Anodyne CNR2 16 50 COCc1nc(C(=O)Nc2ccc(C)c(S(=O)(=O)N3CCCCC3)c2)cs1 ZINC000147107909 HG On-Demand Anodyne NR1H4 19 43 COCc1nc(C(=O)Nc2ccc(C)c(S(=O)(=O)N3CCCCC3)c2)cs1 ZINC000147107909 HG On-Demand Anodyne LIPG 16 40 CCCOCC(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147107926 DF On-Demand Anodyne CHRM2 26 47 CCCOCC(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147107926 DF On-Demand Anodyne SLC18A3 35 48 O=C(Nc1cccc(C(=O)N2CCOCC2)c1)c1ccn(-c2cccc(F)c2)n1 ZINC000147107929 GF On-Demand Anodyne EPHX2 15 52 COCCOc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147108148 HI On-Demand Anodyne RAF1 41 37 COCCOc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147108148 HI On-Demand Anodyne ROCK2 37 51 COCCOc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147108148 HI On-Demand Anodyne FAAH 17 45 COCCOc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147108148 HI On-Demand Anodyne MET 84 48 COCCOc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147108148 HI On-Demand Anodyne PDGFRA 54 38 COCCOc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147108148 HI On-Demand Anodyne NAMPT 65 52 CCN1C(=O)c2ccccc2N[C@@H]1c1ccc(OC)c(OCCCC#N)c1 ZINC000147108247 FH On-Demand Mild TSHR 63 47 C=CCCOCC(=O)Nc1ccccc1NS(=O)(=O)c1ccc(F)cc1 ZINC000147108385 GG On-Demand Mild PRTN3 55 35 COCCOc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147108406 GI On-Demand Anodyne ADRB1 24 43 COCCOc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147108406 GI On-Demand Anodyne EPHX2 23 42 O=C(NCC[C@H](O)CO)[C@@H]1N[C@H](CC2CCCCC2)[C@]2(C(=O)Nc3cc(Cl)c(F)cc32)[C@H]1c1cccc(Cl)c1 ZINC000147108423 KI Annotated Anodyne MDM2 58 77 CCCCO[C@@H](C)C(=O)N1CCN(Cc2nc(-c3ccc(C)cc3)no2)CC1 ZINC000147108492 GF On-Demand Anodyne HRH3 27 43 CCCCO[C@@H](C)C(=O)N1CCN(Cc2nc(-c3ccc(C)cc3)no2)CC1 ZINC000147108492 GF On-Demand Anodyne ACOX1 17 43 CS(=O)(=O)c1cc(C(=O)Nc2ccc(F)cc2Br)cc([N+](=O)[O-])c1 ZINC000147108537 HG On-Demand Bother CA4 15 41 CCc1ncc(C(=O)Nc2cc(S(=O)(=O)N(C)C)ccc2C)s1 ZINC000147108601 FF On-Demand Anodyne MAPK14 18 45 COCCOc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147108612 GI On-Demand Anodyne ADRB1 24 43 COCCOc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147108612 GI On-Demand Anodyne EPHX2 23 42 CCCCO[C@H](C)C(=O)N1CCN(Cc2nc(-c3ccc(C)cc3)no2)CC1 ZINC000147108710 GF On-Demand Anodyne HRH3 27 43 CCCCO[C@H](C)C(=O)N1CCN(Cc2nc(-c3ccc(C)cc3)no2)CC1 ZINC000147108710 GF On-Demand Anodyne ACOX1 17 43 CN(C)S(=O)(=O)c1ccc(N2CCCC2)c(C(=O)N2CCC(C#N)CC2)c1 ZINC000147108741 GD On-Demand Mild SLC6A9 38 52 COc1cc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)ccc1NC(C)=O ZINC000147108792 HE On-Demand Bother KCNMA1 20 44 COc1cc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)ccc1NC(C)=O ZINC000147108792 HE On-Demand Bother TAAR1 23 44 COc1cc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)ccc1NC(C)=O ZINC000147108792 HE On-Demand Bother ENPP1 54 30 COCCOc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147108796 GI On-Demand Anodyne ADRB1 24 43 COCCOc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147108796 GI On-Demand Anodyne EPHX2 23 42 CCc1ncc(C(=O)Nc2ccc(C)c(S(=O)(=O)N(CC)CC)c2)s1 ZINC000147108798 GG On-Demand Anodyne SMG1 31 42 O=C(Cc1ccccc1)NCCOCc1ccccc1 ZINC000147108941 CF In-Stock Anodyne MME 20 40 O=C(Cc1ccccc1)NCCOCc1ccccc1 ZINC000147108941 CF In-Stock Anodyne CA5B 40 47 O=C(Cc1ccccc1)NCCOCc1ccccc1 ZINC000147108941 CF In-Stock Anodyne CA5A 41 47 O=C(Cc1ccccc1)NCCOCc1ccccc1 ZINC000147108941 CF In-Stock Anodyne CAPN2 50 30 O=C(Cc1ccccc1)NCCOCc1ccccc1 ZINC000147108941 CF In-Stock Anodyne POL 0 40 O=C(Cc1ccccc1)NCCOCc1ccccc1 ZINC000147108941 CF In-Stock Anodyne NPR 53 34 O=C(Cc1ccccc1)NCCOCc1ccccc1 ZINC000147108941 CF In-Stock Anodyne NCE103 35 42 O=C(Cc1ccccc1)NCCOCc1ccccc1 ZINC000147108941 CF In-Stock Anodyne CRTM 40 37 O=C(Cc1ccccc1)NCCOCc1ccccc1 ZINC000147108941 CF In-Stock Anodyne P96878_MYCTU 20 42 O=C(Cc1ccccc1)NCCOCc1ccccc1 ZINC000147108941 CF In-Stock Anodyne CAN2 0 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1OC(F)F ZINC000147108950 EE On-Demand Anodyne GRIA1 41 31 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1OC(F)F ZINC000147108950 EE On-Demand Anodyne PCSK5 55 35 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1OC(F)F ZINC000147108950 EE On-Demand Anodyne FURIN 61 36 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1OC(F)F ZINC000147108950 EE On-Demand Anodyne POLG_WNV 66 32 COCCOc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147108990 GI On-Demand Anodyne ADRB1 24 43 COCCOc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147108990 GI On-Demand Anodyne EPHX2 23 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000147109000 FE On-Demand Bother DRD4 44 33 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000147109000 FE On-Demand Bother ROCK2 27 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000147109000 FE On-Demand Bother MCHR1 18 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(C(=O)NC3CC3)c2)c1 ZINC000147109000 FE On-Demand Bother TAAR1 24 42 CCOC[C@H](C)NS(=O)(=O)c1c(C)cc(OC)cc1C ZINC000147109101 DE On-Demand Anodyne NR3C1 15 49 CC[C@@]1(N)C[C@@H]1c1ccc(O)cc1 ZINC000147109126 AD For-Sale Anodyne KDM1A 49 67 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1OC(F)F ZINC000147109135 EE On-Demand Anodyne GRIA1 41 31 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1OC(F)F ZINC000147109135 EE On-Demand Anodyne PCSK5 55 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1OC(F)F ZINC000147109135 EE On-Demand Anodyne FURIN 61 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1OC(F)F ZINC000147109135 EE On-Demand Anodyne POLG_WNV 66 32 CN(C)S(=O)(=O)c1ccc(N2CCOCC2)c(C(=O)N2CCC(C#N)CC2)c1 ZINC000147109176 HD On-Demand Mild SLC6A9 44 49 CCc1ncc(C(=O)Nc2ccc(C)c(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147109209 GG On-Demand Anodyne CNR2 19 52 CCc1ncc(C(=O)Nc2ccc(C)c(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147109209 GG On-Demand Anodyne NR1H4 20 45 CCc1ncc(C(=O)Nc2ccc(C)c(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147109209 GG On-Demand Anodyne EPHX2 27 40 CC[C@@]1(N)C[C@H]1c1ccc(O)cc1 ZINC000147109312 AD For-Sale Anodyne KDM1A 49 67 CC1CCN(c2ccc([N+](=O)[O-])cc2C(=O)N2CCC(C#N)CC2)CC1 ZINC000147109374 FG On-Demand Mild SLC6A9 27 52 CC[C@@H](COc1ccccc1Cl)OC ZINC000147109420 BG On-Demand Anodyne PDS 41 56 CCOC[C@H](C)NS(=O)(=O)c1cccc(Cl)c1 ZINC000147109466 CE On-Demand Anodyne FBP1 24 42 CCOC(=O)CN1CCC(c2ccccn2)CC1 ZINC000147109484 BD On-Demand Anodyne DRD4 25 56 NC(=O)N1CC[C@@]2(C1)OCc1ccccc12 ZINC000147109521 BD On-Demand Anodyne AVPR1A 22 53 NC(=O)N1CC[C@@]2(C1)OCc1ccccc12 ZINC000147109521 BD On-Demand Anodyne SIGMAR1 20 44 CCOCCOCc1cccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147109535 GG On-Demand Anodyne ROCK2 28 45 CNCCCN1CCN(c2ccc(C(F)(F)F)cc2)CC1 ZINC000147109631 DE On-Demand Anodyne CACNA1G 24 49 NC(=O)N1CC[C@]2(C1)OCc1ccccc12 ZINC000147109685 BD On-Demand Anodyne AVPR1A 22 53 NC(=O)N1CC[C@]2(C1)OCc1ccccc12 ZINC000147109685 BD On-Demand Anodyne SIGMAR1 20 44 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne ACE 40 41 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne OPRM1 67 52 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne OPRD1 63 52 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne CACNA2D1 15 61 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne MME 127 55 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne LTA4H 18 42 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne ANPEP 107 41 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne TACR1 15 55 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne FCER2 72 36 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne RNPEP 43 39 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne CTSB 45 39 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne PAPA1_CARPA 49 37 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne CTSL 30 42 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne CPA1 62 40 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne NPFFR2 47 38 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne TPH1 91 40 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne CTRB1 29 43 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne CAPNS1 52 32 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne YARS 68 52 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne SLC1A1 15 44 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne CAPN1 56 44 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne CAPN2 58 40 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne ACE2 53 34 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne LAP3 66 43 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne CTSC 43 52 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne MMP1 17 41 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne AMP1_PLAFQ 70 42 N[C@H](Cc1ccccc1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147109716 EH On-Demand Anodyne NPFFR1 62 38 CCOCCOCc1cccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147109739 GG On-Demand Anodyne ROCK2 28 45 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147109893 GH On-Demand Bother ANPEP 17 41 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147109893 GH On-Demand Bother TAAR1 29 46 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother CPT1A 43 30 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother PRNP 40 36 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother ABCB1B 23 41 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother NR1H4 15 45 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother HDAC1 15 48 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother HDAC2 15 42 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother KCNMA1 28 47 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother TAAR1 32 48 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother ABCG2 42 47 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother SMO 27 41 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother KCNK3 91 43 COc1ccccc1NC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147109954 HI On-Demand Bother KCNK9 64 43 CCCC[C@@H](CC)CNc1ccc(C(=O)O)cc1 ZINC000147109976 BI For-Sale Anodyne RARB 23 40 CSc1ccc([C@H](C)NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147110003 EF On-Demand Anodyne ACACA 23 43 CSc1ccc([C@H](C)NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147110003 EF On-Demand Anodyne ACACB 29 45 CSc1ccc([C@H](C)NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147110003 EF On-Demand Anodyne F7 28 41 CC[C@H](C)C(=O)Nc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147110063 GH On-Demand Bother ANPEP 17 41 CC[C@H](C)C(=O)Nc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147110063 GH On-Demand Bother TAAR1 29 46 N#CC1CCN(C(=O)c2cn(-c3ccccc3)nc2-c2ccc(Cl)cc2)CC1 ZINC000147110097 GJ On-Demand Mild CDK2 17 48 C[C@H](N[C@@H]1C[C@H]1c1ccccc1)C1CCCCC1 ZINC000147110129 BI For-Sale Anodyne EPHX2 17 40 C[C@H](N[C@@H]1C[C@H]1c1ccccc1)C1CCCCC1 ZINC000147110129 BI For-Sale Anodyne KDM1A 26 45 CCCC[C@H](CC)CNc1ccc(C(=O)O)cc1 ZINC000147110163 BI For-Sale Anodyne RARB 23 40 CC/C=C\CCCCCC(=O)OC ZINC000147110179 AG For-Sale Anodyne LPAR2 15 47 CC/C=C\CCCCCC(=O)OC ZINC000147110179 AG For-Sale Anodyne FAAH 17 45 CC/C=C\CCCCCC(=O)OC ZINC000147110179 AG For-Sale Anodyne LPAR3 35 47 CC/C=C\CCCCCC(=O)OC ZINC000147110179 AG For-Sale Anodyne FABP3 45 58 CC/C=C\CCCCCC(=O)OC ZINC000147110179 AG For-Sale Anodyne FABP1 16 48 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2csc(-c3ccccc3)n2)CC1 ZINC000147110320 HF On-Demand Anodyne GHRHR 46 38 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2csc(-c3ccccc3)n2)CC1 ZINC000147110320 HF On-Demand Anodyne P2RY12 224 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2csc(-c3ccccc3)n2)CC1 ZINC000147110320 HF On-Demand Anodyne TRY2_BOVIN 61 34 COc1ccc(-c2nn(-c3ccccc3)cc2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147110321 GH On-Demand Mild CDK2 18 52 N#Cc1ccc(CCC(=O)O)cn1 ZINC000147110368 AC For-Sale Mild FAAH 20 42 N#Cc1ccc(CCC(=O)O)cn1 ZINC000147110368 AC For-Sale Mild CES1 25 42 N#Cc1ccc(CCC(=O)O)cn1 ZINC000147110368 AC For-Sale Mild FFAR1 81 48 N#Cc1ccc(CCC(=O)O)cn1 ZINC000147110368 AC For-Sale Mild FFAR4 55 40 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne HTR1A 22 47 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne DRD2 23 54 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne DRD4 41 33 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne SLC6A1 17 50 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne OPRM1 20 46 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne OPRD1 17 46 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne OPRK1 16 46 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne SLC6A3 18 50 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne SLC18A2 49 39 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne HRH3 46 63 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne SIGMAR1 49 54 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne EBP 50 41 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne CHRNA10 58 44 COc1cccc([C@@H]2CCCN2CCc2ccccc2)c1 ZINC000147110373 CI On-Demand Anodyne LUCI_PHOPY 18 40 Cc1cc(C(=O)Nc2cc(S(=O)(=O)N3CCCCC3)ccc2C)cc([N+](=O)[O-])c1 ZINC000147110475 HH On-Demand Bother EPHX2 26 43 CCCOCC(=O)NCC1(c2ccccc2)CCC1 ZINC000147110510 CF On-Demand Anodyne KCNA3 23 42 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne HTR1A 22 47 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne DRD2 23 54 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne DRD4 41 33 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne SLC6A1 17 50 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne OPRM1 20 46 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne OPRD1 17 46 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne OPRK1 16 46 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne SLC6A3 18 50 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne SLC18A2 49 39 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne HRH3 46 63 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne SIGMAR1 49 54 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne EBP 50 41 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne CHRNA10 58 44 COc1cccc([C@H]2CCCN2CCc2ccccc2)c1 ZINC000147110569 CI On-Demand Anodyne LUCI_PHOPY 18 40 CC[C@H](COc1ccccc1Cl)OC ZINC000147110616 BG On-Demand Anodyne PDS 41 56 Cc1cc(C(=O)Nc2ccccc2-c2ccccc2)cc([N+](=O)[O-])c1 ZINC000147110693 EJ On-Demand Bother ABCG2 17 47 Cc1cc(C(=O)Nc2ccccc2-c2ccccc2)cc([N+](=O)[O-])c1 ZINC000147110693 EJ On-Demand Bother KCNK3 40 37 COc1cccc(-c2nn(-c3ccccc3)cc2C(=O)N2CCC(C#N)CC2)c1 ZINC000147110709 GH On-Demand Mild CDK2 15 43 O=C(C1CCN(C2CCCC2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147110729 HI For-Sale Anodyne HRH3 38 46 O=C(C1CCN(C2CCCC2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147110729 HI For-Sale Anodyne L3MBTL3 72 38 CCCC[C@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110803 HG On-Demand Anodyne OPRD1 15 41 CCCC[C@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110803 HG On-Demand Anodyne KLK3 45 37 CCCC[C@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110803 HG On-Demand Anodyne CTSK 23 43 CCCC[C@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110803 HG On-Demand Anodyne NPFFR2 52 37 CCCC[C@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110803 HG On-Demand Anodyne GRIA1 41 34 CCCC[C@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110803 HG On-Demand Anodyne PCSK5 56 36 CCCC[C@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110803 HG On-Demand Anodyne FURIN 75 38 CCCC[C@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110803 HG On-Demand Anodyne POLG_WNV 64 33 CCCC[C@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110803 HG On-Demand Anodyne QRFPR 40 37 CCCC[C@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110803 HG On-Demand Anodyne NPFFR1 65 37 C[C@@]1(c2cc(NC(=O)c3ncc(Br)cn3)ccc2F)C=CSC(N)=N1 ZINC000147110843 HG Annotated Anodyne BACE2 47 48 C[C@@]1(c2cc(NC(=O)c3ncc(Br)cn3)ccc2F)C=CSC(N)=N1 ZINC000147110843 HG Annotated Anodyne BACE1 23 48 C=CCCOCC(=O)Nc1ccc(CC(=O)N2CCN(c3ncccn3)CC2)cc1 ZINC000147110904 HD On-Demand Mild F13A1 50 34 CCCC[C@@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110982 HG On-Demand Anodyne OPRD1 15 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110982 HG On-Demand Anodyne KLK3 45 37 CCCC[C@@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110982 HG On-Demand Anodyne CTSK 23 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110982 HG On-Demand Anodyne NPFFR2 52 37 CCCC[C@@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110982 HG On-Demand Anodyne GRIA1 41 34 CCCC[C@@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110982 HG On-Demand Anodyne PCSK5 56 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110982 HG On-Demand Anodyne FURIN 75 38 CCCC[C@@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110982 HG On-Demand Anodyne POLG_WNV 64 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110982 HG On-Demand Anodyne QRFPR 40 37 CCCC[C@@H](NC(N)=O)C(=O)NCc1cn(Cc2ccccc2)nc1-c1ccccc1 ZINC000147110982 HG On-Demand Anodyne NPFFR1 65 37 O=C(N[C@@H](c1ccccc1)C1CCCC1)c1ccc2c(c1)COC2 ZINC000147110986 DI On-Demand Anodyne AKT1 22 48 O=C(N[C@@H](c1ccccc1)C1CCCC1)c1ccc2c(c1)COC2 ZINC000147110986 DI On-Demand Anodyne TTK 37 41 CCOC[C@H](C)NC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111056 DG On-Demand Anodyne EPHX2 20 42 CCOC[C@H](C)NC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111056 DG On-Demand Anodyne KCNK3 49 40 CCOC[C@H](C)NC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111056 DG On-Demand Anodyne KCNK9 42 40 CCOC[C@H](C)NC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111056 DG On-Demand Anodyne PDS 56 42 O=C(N[C@H](c1ccccc1)C1CCCC1)c1ccc2c(c1)COC2 ZINC000147111190 DI On-Demand Anodyne TTK 37 41 O=C(O)Cc1ccc(Cl)cc1I ZINC000147111191 CF For-Sale Anodyne CXCL8 36 44 COc1ccc(Cn2cnc3cc4c(cc32)CCCC4)cc1OC ZINC000147111247 DH Annotated Anodyne PDE4D 41 39 COc1ccc(Cn2cnc3cc4c(cc32)CCCC4)cc1OC ZINC000147111247 DH Annotated Anodyne NR1I2 40 35 Cc1cccc(C)c1OC[C@H](O)CNC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111258 HH On-Demand Anodyne ADRB2 23 42 Cc1cccc(C)c1OC[C@H](O)CNC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111258 HH On-Demand Anodyne ADRB1 62 44 Cc1cccc(C)c1OC[C@H](O)CNC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111258 HH On-Demand Anodyne ADRB3 15 41 Cc1cccc(C)c1OC[C@H](O)CNC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111258 HH On-Demand Anodyne ACOX1 40 36 Cc1cccc(C)c1OC[C@H](O)CNC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111258 HH On-Demand Anodyne PDS 43 37 CC[C@@H](C)C(=O)Nc1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147111278 GH On-Demand Anodyne CARM1 63 38 C#CCN1C(=O)c2ccccc2N[C@@H]1c1ccc(OC)c(OCCCC#N)c1 ZINC000147111347 GH On-Demand Mild TSHR 62 44 Cc1cccc(C)c1OC[C@@H](O)CNC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111461 HH On-Demand Anodyne ADRB2 23 42 Cc1cccc(C)c1OC[C@@H](O)CNC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111461 HH On-Demand Anodyne ADRB1 62 44 Cc1cccc(C)c1OC[C@@H](O)CNC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111461 HH On-Demand Anodyne ADRB3 15 41 Cc1cccc(C)c1OC[C@@H](O)CNC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111461 HH On-Demand Anodyne ACOX1 40 36 Cc1cccc(C)c1OC[C@@H](O)CNC(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147111461 HH On-Demand Anodyne PDS 43 37 CC[C@H](C)C(=O)Nc1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147111490 GH On-Demand Anodyne CARM1 63 38 Cc1ccc(-c2nn(-c3ccc(F)cc3)cc2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147111589 GI On-Demand Mild CDK2 15 46 CCOC(=O)NCC(=O)Nc1ccc(-n2cccn2)cc1 ZINC000147111719 CD On-Demand Anodyne AMP1_PLAFQ 56 39 CCOC(=O)NCC(=O)Nc1ccc(-n2cccn2)cc1 ZINC000147111719 CD On-Demand Anodyne LAP 0 45 O=C(Nc1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1)c1ccccc1 ZINC000147111727 HJ On-Demand Anodyne PRNP 46 44 O=C(Nc1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1)c1ccccc1 ZINC000147111727 HJ On-Demand Anodyne MAPK10 18 44 O=C(Nc1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1)c1ccccc1 ZINC000147111727 HJ On-Demand Anodyne KCNK3 135 61 O=C(Nc1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1)c1ccccc1 ZINC000147111727 HJ On-Demand Anodyne KCNK9 85 48 Cc1cccc(-c2nn(-c3ccccc3)cc2C(=O)N2CCC(C#N)CC2)c1 ZINC000147111780 FI On-Demand Mild CDK2 15 40 C[C@@H](OC[C@@H]1CCCO1)C(=O)NCCc1cccc(F)c1 ZINC000147111805 CE On-Demand Anodyne OXTR 25 44 C[C@@H](OC[C@@H]1CCCO1)C(=O)NCCc1cccc(F)c1 ZINC000147111805 CE On-Demand Anodyne AVPR1A 17 44 CCOC[C@H](C)NS(=O)(=O)c1ccccc1OC ZINC000147111828 CD On-Demand Anodyne ITGAV 24 47 O=C(Nc1cccc(OCC(F)(F)F)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147111851 FI On-Demand Anodyne PPIA 23 40 O=C(Nc1cccc(OCC(F)(F)F)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147111851 FI On-Demand Anodyne EPHX2 67 47 COc1cccc(-c2nn(-c3ccc(C)cc3)cc2C(=O)N2CCC(C#N)CC2)c1 ZINC000147112002 HI On-Demand Mild CCKAR 27 41 COCc1nc(C(=O)N2CCN(C/C=C/c3ccccc3)CC2)cs1 ZINC000147112045 FF On-Demand Anodyne TRPC6 53 34 O=C(Nc1cccc(OCC(F)(F)F)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147112058 FI On-Demand Anodyne PPIA 23 40 O=C(Nc1cccc(OCC(F)(F)F)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147112058 FI On-Demand Anodyne EPHX2 67 47 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)c1 ZINC000147112159 GE On-Demand Bother AVPR2 37 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)c1 ZINC000147112159 GE On-Demand Bother EPHX2 22 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)c1 ZINC000147112159 GE On-Demand Bother TAAR1 33 54 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)c1 ZINC000147112159 GE On-Demand Bother AKR1C3 25 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)c1 ZINC000147112159 GE On-Demand Bother AKR1C2 48 38 Cc1ccc(-n2cc(C(=O)N3CCC(C#N)CC3)c(-c3ccccc3)n2)cc1 ZINC000147112208 FI On-Demand Mild CDK2 16 46 O=C(Nc1cccc(OCC(F)(F)F)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147112239 FI On-Demand Anodyne PPIA 23 40 O=C(Nc1cccc(OCC(F)(F)F)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147112239 FI On-Demand Anodyne EPHX2 67 47 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccn(-c2cccc(F)c2)n1 ZINC000147112371 GF On-Demand Anodyne PRNP 43 31 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1ccn(-c2cccc(F)c2)n1 ZINC000147112371 GF On-Demand Anodyne EPHX2 19 53 O=C(Nc1cccc(OCC(F)(F)F)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147112453 FI On-Demand Anodyne PPIA 23 40 O=C(Nc1cccc(OCC(F)(F)F)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147112453 FI On-Demand Anodyne EPHX2 67 47 N[C@H](CC[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 ZINC000147112490 HI In-Stock Anodyne KLK3 43 31 N[C@H](CC[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 ZINC000147112490 HI In-Stock Anodyne PAPA1_CARPA 42 35 N[C@H](CC[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 ZINC000147112490 HI In-Stock Anodyne CYSP_TRYCR 55 36 N[C@H](CC[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 ZINC000147112490 HI In-Stock Anodyne CAPNS1 56 36 N[C@H](CC[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 ZINC000147112490 HI In-Stock Anodyne CAPN1 42 35 N[C@H](CC[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 ZINC000147112490 HI In-Stock Anodyne CAPN2 53 39 N[C@H](CC[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 ZINC000147112490 HI In-Stock Anodyne LAP3 47 34 N[C@H](CC[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 ZINC000147112490 HI In-Stock Anodyne CYP3A4 79 69 N[C@H](CC[C@H](Cc1ccccc1)NC(=O)OCc1cncs1)Cc1ccccc1 ZINC000147112490 HI In-Stock Anodyne GPR142 33 40 COc1ccc(-c2nn(-c3ccccc3)cc2C(=O)N2CCC(C#N)CC2)c(OC)c1 ZINC000147112627 HH On-Demand Mild OXTR 24 41 CN(CCCOc1ccc(F)cc1)C1CCC1 ZINC000147112639 BG On-Demand Anodyne LTA4H 23 49 CN(CCCOc1ccc(F)cc1)C1CCC1 ZINC000147112639 BG On-Demand Anodyne HRH3 27 43 CN(CCCOc1ccc(F)cc1)C1CCC1 ZINC000147112639 BG On-Demand Anodyne SHC 28 43 CN(CCCOc1ccc(F)cc1)C1CCC1 ZINC000147112639 BG On-Demand Anodyne LSS 26 48 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147112699 HI On-Demand Anodyne NOS2 62 33 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147112699 HI On-Demand Anodyne ROCK2 19 42 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147112699 HI On-Demand Anodyne EPHX2 18 42 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147112699 HI On-Demand Anodyne NAMPT 39 42 COc1ccc([C@@H]2CCCN2C(=O)Cc2cccc(OC(C)C)c2)c(OC)c1 ZINC000147112805 GI On-Demand Anodyne FKBP1A 63 38 COc1ccc([C@@H]2CCCN2C(=O)Cc2cccc(OC(C)C)c2)c(OC)c1 ZINC000147112805 GI On-Demand Anodyne OPRK1 19 43 COc1ccc([C@@H]2CCCN2C(=O)Cc2cccc(OC(C)C)c2)c(OC)c1 ZINC000147112805 GI On-Demand Anodyne CPT1A 69 36 COc1ccc([C@@H]2CCCN2C(=O)Cc2cccc(OC(C)C)c2)c(OC)c1 ZINC000147112805 GI On-Demand Anodyne MTNR1B 40 38 COC(=O)c1ccc(O)c(/C=N/N)c1 ZINC000147112864 AC For-Sale Mild CA14 16 44 CCOC[C@H](C)NS(=O)(=O)c1c(Cl)cccc1Cl ZINC000147112969 DF On-Demand Anodyne NR3C1 15 49 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147112971 HJ On-Demand Anodyne EPHX2 29 40 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147112971 HJ On-Demand Anodyne PDS 41 35 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147113157 HJ On-Demand Anodyne EPHX2 29 40 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147113157 HJ On-Demand Anodyne PDS 41 35 CCn1cc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)ccc1=O ZINC000147113212 DG On-Demand Anodyne MDM2 93 33 CCn1cc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)ccc1=O ZINC000147113212 DG On-Demand Anodyne NAMPT 23 41 C=C1C[C@@](C)(c2cc(NC(=O)c3cnc(OC)cn3)cnc2C)N=C(N)S1 ZINC000147113247 GF Annotated Mild BACE2 33 40 C=C1C[C@@](C)(c2cc(NC(=O)c3cnc(OC)cn3)cnc2C)N=C(N)S1 ZINC000147113247 GF Annotated Mild BACE1 15 45 COCc1nc(C(=O)NCCc2ccc(Cl)cc2Cl)cs1 ZINC000147113275 EH On-Demand Anodyne CNR1 20 45 COCc1nc(C(=O)NCCc2ccc(Cl)cc2Cl)cs1 ZINC000147113275 EH On-Demand Anodyne PTGDR 19 40 COCc1nc(C(=O)NCCc2ccc(Cl)cc2Cl)cs1 ZINC000147113275 EH On-Demand Anodyne ALPL 38 40 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147113349 HJ On-Demand Anodyne EPHX2 29 40 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147113349 HJ On-Demand Anodyne PDS 41 35 CCn1cc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)ccc1=O ZINC000147113413 DG On-Demand Anodyne MDM2 93 33 CCn1cc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)ccc1=O ZINC000147113413 DG On-Demand Anodyne NAMPT 23 41 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)C(=O)NC3CC3)CC2)c1 ZINC000147113442 GC On-Demand Bother AKR1C2 25 40 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147113529 HJ On-Demand Anodyne EPHX2 29 40 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(OCC(F)(F)F)c1 ZINC000147113529 HJ On-Demand Anodyne PDS 41 35 COc1cc2c(cc1O)CCN1C[C@@H](CC(C)C)[C@@H](O)C[C@H]21 ZINC000147113552 DF For-Sale Anodyne DRD1 30 54 COc1cc2c(cc1O)CCN1C[C@@H](CC(C)C)[C@@H](O)C[C@H]21 ZINC000147113552 DF For-Sale Anodyne SLC18A2 94 85 COc1cc2c(cc1O)CCN1C[C@@H](CC(C)C)[C@@H](O)C[C@H]21 ZINC000147113552 DF For-Sale Anodyne F3 31 48 COc1cc2c(cc1O)CCN1C[C@@H](CC(C)C)[C@@H](O)C[C@H]21 ZINC000147113552 DF For-Sale Anodyne SLC2A1 17 48 CCC[C@@H](CO)N(Cc1ccccc1)C(=O)OC(C)(C)C ZINC000147113561 CH For-Sale Anodyne CTSB 15 41 CCn1cc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)ccc1=O ZINC000147113604 DG On-Demand Anodyne MDM2 93 33 CCn1cc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)ccc1=O ZINC000147113604 DG On-Demand Anodyne NAMPT 23 41 CCn1c(SCC(=O)Nc2ccc(C(=O)O)cc2)nnc1[C@H](NC(=O)c1ccc(Cl)cc1Cl)C(C)C ZINC000147113658 KK In-Stock Anodyne SLC27A1 28 42 CCn1cc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)ccc1=O ZINC000147113804 DG On-Demand Anodyne MDM2 93 33 CCn1cc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)ccc1=O ZINC000147113804 DG On-Demand Anodyne NAMPT 23 41 CCn1c(SCC(=O)Nc2ccc(C(=O)O)cc2)nnc1[C@@H](NC(=O)c1ccc(Cl)cc1Cl)C(C)C ZINC000147113858 KK In-Stock Anodyne SLC27A1 28 42 CCCCOc1ccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147113899 FH On-Demand Bother CNR2 43 42 CCCCOc1ccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147113899 FH On-Demand Bother CTSL 17 40 CCCCOc1ccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147113899 FH On-Demand Bother MTNR1A 59 42 CCCCOc1ccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147113899 FH On-Demand Bother MTNR1B 43 36 CCCCOc1ccc(CCNC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1 ZINC000147113899 FH On-Demand Bother PLA2G4B 61 40 CCn1cc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)ccc1=O ZINC000147114007 FG On-Demand Anodyne NAMPT 22 41 Cc1cccc(C(=O)NCc2nnc(SCC(=O)N(C3CCCCC3)C3CCCCC3)n2C)c1 ZINC000147114060 JJ In-Stock Anodyne SCARB1 40 34 N#CC1CCN(C(=O)Cc2cn(-c3ccccc3)nc2-c2ccc([N+](=O)[O-])cc2)CC1 ZINC000147114086 HH On-Demand Mild HDAC1 16 47 CCOC(=O)Cc1nc(N2CCOCC2)cc(=O)n1C ZINC000147114092 CB For-Sale Anodyne PIK3CA 21 40 CCOC(=O)Cc1nc(N2CCOCC2)cc(=O)n1C ZINC000147114092 CB For-Sale Anodyne PIK3CD 37 59 CCOC(=O)Cc1nc(N2CCOCC2)cc(=O)n1C ZINC000147114092 CB For-Sale Anodyne PIK3CB 71 59 CCc1ncc(C(=O)N2CCN(c3ccccn3)CC2)s1 ZINC000147114101 DE On-Demand Anodyne SCD1 15 40 CCc1ncc(C(=O)N2CCN(c3ccccn3)CC2)s1 ZINC000147114101 DE On-Demand Anodyne SLC27A1 20 40 Cc1nc2ccccc2n1CCCNC(=O)COc1ccc(C(N)=O)cc1 ZINC000147114114 FE On-Demand Anodyne CYSP_TRYCR 16 48 Cc1nc2ccccc2n1CCCNC(=O)COc1ccc(C(N)=O)cc1 ZINC000147114114 FE On-Demand Anodyne PDE6D 35 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC)c(OCC(=O)NC3CC3)c2)c1 ZINC000147114124 HF On-Demand Bother ENPP1 67 32 CCn1cc(NC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)ccc1=O ZINC000147114177 FG On-Demand Anodyne NAMPT 22 41 NC(=O)c1ccc(OCC(=O)NCc2ccc(-n3cccn3)cc2)cc1 ZINC000147114334 FD On-Demand Anodyne AMP1_PLAFQ 57 39 CCn1cc(NC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)ccc1=O ZINC000147114367 FG On-Demand Anodyne NAMPT 22 41 N#CC1(C#N)CCN(Cc2ccccc2)CC1 ZINC000147114493 BE For-Sale Mild DRD2 26 51 N#CC1(C#N)CCN(Cc2ccccc2)CC1 ZINC000147114493 BE For-Sale Mild DRD3 25 41 N#CC1(C#N)CCN(Cc2ccccc2)CC1 ZINC000147114493 BE For-Sale Mild OPRL1 17 47 N#CC1(C#N)CCN(Cc2ccccc2)CC1 ZINC000147114493 BE For-Sale Mild SIGMAR1 90 59 N#CC1(C#N)CCN(Cc2ccccc2)CC1 ZINC000147114493 BE For-Sale Mild KCNA3 30 48 N#CC1(C#N)CCN(Cc2ccccc2)CC1 ZINC000147114493 BE For-Sale Mild NPFFR2 33 41 N#CC1(C#N)CCN(Cc2ccccc2)CC1 ZINC000147114493 BE For-Sale Mild SLC18A3 24 41 N#CC1(C#N)CCN(Cc2ccccc2)CC1 ZINC000147114493 BE For-Sale Mild EBP 18 41 N#CC1(C#N)CCN(Cc2ccccc2)CC1 ZINC000147114493 BE For-Sale Mild NPFFR1 58 41 CCn1cc(NC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)ccc1=O ZINC000147114562 FG On-Demand Anodyne NAMPT 22 41 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114566 HG On-Demand Anodyne HRAS 48 33 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114566 HG On-Demand Anodyne ACACA 23 43 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114566 HG On-Demand Anodyne ACACB 30 43 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114566 HG On-Demand Anodyne F7 26 48 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114566 HG On-Demand Anodyne CYP26A1 28 42 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114566 HG On-Demand Anodyne VCP 37 43 COCc1nc(C(=O)N2CCN(c3cccc(C(F)(F)F)c3)CC2)cs1 ZINC000147114578 GG On-Demand Anodyne TRPC6 45 33 COc1cc2nccc(Oc3ccc([N+](=O)[O-])c(OC)c3)c2cc1OC ZINC000147114669 FH For-Sale Bother PDGFRB 43 48 COc1cc2nccc(Oc3ccc([N+](=O)[O-])c(OC)c3)c2cc1OC ZINC000147114669 FH For-Sale Bother FGFR2 72 52 COc1cc2nccc(Oc3ccc([N+](=O)[O-])c(OC)c3)c2cc1OC ZINC000147114669 FH For-Sale Bother MAP2K5 17 47 COc1cc2nccc(Oc3ccc([N+](=O)[O-])c(OC)c3)c2cc1OC ZINC000147114669 FH For-Sale Bother FLT1 37 46 COc1cc2nccc(Oc3ccc([N+](=O)[O-])c(OC)c3)c2cc1OC ZINC000147114669 FH For-Sale Bother KDR 102 52 COc1cc2nccc(Oc3ccc([N+](=O)[O-])c(OC)c3)c2cc1OC ZINC000147114669 FH For-Sale Bother PDE3B 50 34 COc1cc2nccc(Oc3ccc([N+](=O)[O-])c(OC)c3)c2cc1OC ZINC000147114669 FH For-Sale Bother MET 36 48 COc1cc2nccc(Oc3ccc([N+](=O)[O-])c(OC)c3)c2cc1OC ZINC000147114669 FH For-Sale Bother FLT4 24 47 COc1cc2nccc(Oc3ccc([N+](=O)[O-])c(OC)c3)c2cc1OC ZINC000147114669 FH For-Sale Bother PDGFRA 80 60 COc1cc2nccc(Oc3ccc([N+](=O)[O-])c(OC)c3)c2cc1OC ZINC000147114669 FH For-Sale Bother CSF1R 26 45 COc1cc2nccc(Oc3ccc([N+](=O)[O-])c(OC)c3)c2cc1OC ZINC000147114669 FH For-Sale Bother EPHB6 16 47 Cc1ccc(-c2csc(NC(=O)CSc3nnc([C@@H](C)NC(=O)c4cccc(C)c4)n3C)n2)cc1 ZINC000147114671 KJ In-Stock Anodyne ROCK1 19 40 Cc1ccc(-c2csc(NC(=O)CSc3nnc([C@@H](C)NC(=O)c4cccc(C)c4)n3C)n2)cc1 ZINC000147114671 KJ In-Stock Anodyne TRPA1 21 40 CC(C)(C)OC(=O)NCCCC(=O)N1CCC(C#N)CC1 ZINC000147114735 CE On-Demand Mild PREP 15 44 CCn1cc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)ccc1=O ZINC000147114743 EE On-Demand Anodyne ROCK2 32 50 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114760 HG On-Demand Anodyne HRAS 48 33 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114760 HG On-Demand Anodyne ACACA 23 43 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114760 HG On-Demand Anodyne ACACB 30 43 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114760 HG On-Demand Anodyne F7 26 48 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114760 HG On-Demand Anodyne CYP26A1 28 42 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc(OCc2cccnc2)cc1 ZINC000147114760 HG On-Demand Anodyne VCP 37 43 Cc1noc(C)c1CNC(=O)NCc1cccnc1 ZINC000147114813 CD On-Demand Anodyne NAMPT 60 50 CC(=O)c1ccc(NCC(=O)N2CCN(c3cccc(Cl)c3)CC2)cc1 ZINC000147114822 FG For-Sale Anodyne HTR1A 24 45 CC(=O)c1ccc(NCC(=O)N2CCN(c3cccc(Cl)c3)CC2)cc1 ZINC000147114822 FG For-Sale Anodyne HTR2A 18 45 CC(=O)c1ccc(NCC(=O)N2CCN(c3cccc(Cl)c3)CC2)cc1 ZINC000147114822 FG For-Sale Anodyne HTR7 15 40 CC(=O)c1ccc(NCC(=O)N2CCN(c3cccc(Cl)c3)CC2)cc1 ZINC000147114822 FG For-Sale Anodyne CCR1 36 40 CC(=O)c1ccc(NCC(=O)N2CCN(c3cccc(Cl)c3)CC2)cc1 ZINC000147114822 FG For-Sale Anodyne PRNP 51 35 CC(=O)c1ccc(NCC(=O)N2CCN(c3cccc(Cl)c3)CC2)cc1 ZINC000147114822 FG For-Sale Anodyne MAPK1 41 48 CC(=O)c1ccc(NCC(=O)N2CCN(c3cccc(Cl)c3)CC2)cc1 ZINC000147114822 FG For-Sale Anodyne SSTR1 18 45 Cc1ccc(-c2csc(NC(=O)CSc3nnc([C@H](C)NC(=O)c4cccc(C)c4)n3C)n2)cc1 ZINC000147114869 KJ In-Stock Anodyne ROCK1 19 40 Cc1ccc(-c2csc(NC(=O)CSc3nnc([C@H](C)NC(=O)c4cccc(C)c4)n3C)n2)cc1 ZINC000147114869 KJ In-Stock Anodyne TRPA1 21 40 Nc1nc(N)c2ncn([C@@H]3S[C@H](CO)[C@H](O)[C@@H]3O)c2n1 ZINC000147114923 CA Annotated Anodyne ADORA1 52 78 Nc1nc(N)c2ncn([C@@H]3S[C@H](CO)[C@H](O)[C@@H]3O)c2n1 ZINC000147114923 CA Annotated Anodyne ADORA2A 54 78 Nc1nc(N)c2ncn([C@@H]3S[C@H](CO)[C@H](O)[C@@H]3O)c2n1 ZINC000147114923 CA Annotated Anodyne ADORA2B 25 41 Nc1nc(N)c2ncn([C@@H]3S[C@H](CO)[C@H](O)[C@@H]3O)c2n1 ZINC000147114923 CA Annotated Anodyne AHCY 95 43 Nc1nc(N)c2ncn([C@@H]3S[C@H](CO)[C@H](O)[C@@H]3O)c2n1 ZINC000147114923 CA Annotated Anodyne P2RY1 67 33 Nc1nc(N)c2ncn([C@@H]3S[C@H](CO)[C@H](O)[C@@H]3O)c2n1 ZINC000147114923 CA Annotated Anodyne ADCY5 40 39 Nc1nc(N)c2ncn([C@@H]3S[C@H](CO)[C@H](O)[C@@H]3O)c2n1 ZINC000147114923 CA Annotated Anodyne NS5B 32 51 Nc1nc(N)c2ncn([C@@H]3S[C@H](CO)[C@H](O)[C@@H]3O)c2n1 ZINC000147114923 CA Annotated Anodyne ADORA3 28 40 Nc1nc(N)c2ncn([C@@H]3S[C@H](CO)[C@H](O)[C@@H]3O)c2n1 ZINC000147114923 CA Annotated Anodyne OXGR1 96 32 CCn1cc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)ccc1=O ZINC000147114944 EE On-Demand Anodyne ROCK2 32 50 CCOC[C@H](C)NS(=O)(=O)c1cccc(C)c1 ZINC000147114969 CD On-Demand Anodyne FBP1 17 42 COc1ccc(-c2ccc(NC(C)=O)cc2)cc1C=O ZINC000147114988 CG For-Sale Anodyne TSHR 54 34 COc1ccc(-c2ccc(NC(C)=O)cc2)cc1C=O ZINC000147114988 CG For-Sale Anodyne MTNR1B 16 41 COc1ccc(-c2ccc(NC(C)=O)cc2)cc1C=O ZINC000147114988 CG For-Sale Anodyne TUBB1 40 41 O=C(O)CCC1=Cc2ccccc21 ZINC000147115007 AE For-Sale Anodyne CPA3 55 37 O=C(O)CCC1=Cc2ccccc21 ZINC000147115007 AE For-Sale Anodyne FFAR1 50 40 O=C(O)CCC1=Cc2ccccc21 ZINC000147115007 AE For-Sale Anodyne FFAR4 48 38 Cc1noc(C)c1CNC(=O)NCCCn1ccnc1 ZINC000147115014 CD On-Demand Anodyne TBXAS1 40 46 Cc1noc(C)c1CNC(=O)NCCCn1ccnc1 ZINC000147115014 CD On-Demand Anodyne QPCT 44 48 CCCCCCCCCCCCCCC[C@H](O)[C@@H](CCCCCCCCCCCCCC)C(=O)NC[C@@H](O)CO ZINC000147115117 KK For-Sale Mild CQSS 54 33 COc1ccccc1Nc1nc2c(-c3ccc(C(F)(F)F)cc3)cccn2n1 ZINC000147115231 GK Annotated Anodyne JAK2 23 55 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne HTR1A 20 41 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne VDR 20 40 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne FKBP1A 15 42 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne SSTR2 18 40 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne LTA4H 23 40 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne KCNQ2 25 42 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne NPY2R 54 39 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne CCR1 20 42 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne PRNP 39 40 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne MAPK1 39 40 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne SSTR1 33 40 CC(C)c1ccc(NCC(=O)N2CCN(c3ccccc3)CC2)cc1 ZINC000147115258 EH For-Sale Anodyne AKR1C3 20 43 CCOC[C@H](C)NS(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000147115412 DE On-Demand Anodyne CACNA1B 40 35 CCOC[C@H](C)NS(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000147115412 DE On-Demand Anodyne PDS 42 34 CCCCCCCCCCCCCCC[C@H](O)[C@H](CCCCCCCCCCCCCC)C(=O)NC[C@@H](O)CO ZINC000147115496 KK For-Sale Mild CQSS 54 33 CCCCCC[C@@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115527 EK For-Sale Reactive CNR1 15 43 CCCCCC[C@@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115527 EK For-Sale Reactive LPAR1 29 43 CCCCCC[C@@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115527 EK For-Sale Reactive FAAH 22 47 CCCCCC[C@@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115527 EK For-Sale Reactive LPAR3 62 43 CCCCCC[C@@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115527 EK For-Sale Reactive FABP3 37 46 CCCCCC[C@@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115527 EK For-Sale Reactive FABP1 15 46 CCCCCC[C@@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115527 EK For-Sale Reactive NOD1 51 34 CCCCCC[C@@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115527 EK For-Sale Reactive CQSS 53 33 CCCCCC[C@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115732 EK For-Sale Reactive CNR1 15 43 CCCCCC[C@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115732 EK For-Sale Reactive LPAR1 29 43 CCCCCC[C@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115732 EK For-Sale Reactive FAAH 22 47 CCCCCC[C@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115732 EK For-Sale Reactive LPAR3 62 43 CCCCCC[C@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115732 EK For-Sale Reactive FABP3 37 46 CCCCCC[C@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115732 EK For-Sale Reactive FABP1 15 46 CCCCCC[C@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115732 EK For-Sale Reactive NOD1 51 34 CCCCCC[C@H](Cl)C/C=C\CCCCCCCC(=O)OC ZINC000147115732 EK For-Sale Reactive CQSS 53 33 CCc1ncc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCOCC2)s1 ZINC000147115956 GH On-Demand Anodyne TEK 24 43 CCc1ncc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCOCC2)s1 ZINC000147115956 GH On-Demand Anodyne SCD1 19 43 CCc1ncc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCOCC2)s1 ZINC000147115956 GH On-Demand Anodyne LIPG 49 36 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(NS(C)(=O)=O)c1 ZINC000147116091 FC On-Demand Anodyne GRIA1 41 32 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(NS(C)(=O)=O)c1 ZINC000147116091 FC On-Demand Anodyne PCSK5 58 37 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(NS(C)(=O)=O)c1 ZINC000147116091 FC On-Demand Anodyne FURIN 65 39 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(NS(C)(=O)=O)c1 ZINC000147116091 FC On-Demand Anodyne POLG_WNV 59 33 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(NS(C)(=O)=O)c1 ZINC000147116091 FC On-Demand Anodyne NPFFR1 47 32 Cc1cc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCOCC2)cc([N+](=O)[O-])c1 ZINC000147116143 HI On-Demand Bother SLC6A9 15 51 Cc1cc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCOCC2)cc([N+](=O)[O-])c1 ZINC000147116143 HI On-Demand Bother TEK 22 44 Cc1cc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCOCC2)cc([N+](=O)[O-])c1 ZINC000147116143 HI On-Demand Bother TAAR1 26 41 Cc1cc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCOCC2)cc([N+](=O)[O-])c1 ZINC000147116143 HI On-Demand Bother WDR5 39 46 CS(=O)(=O)c1cc(C(=O)NCc2ccc(Cn3ccnc3)cc2)cc([N+](=O)[O-])c1 ZINC000147116208 HE On-Demand Bother CYP19A1 17 52 CS(=O)(=O)c1cc(C(=O)NCc2ccc(Cn3ccnc3)cc2)cc([N+](=O)[O-])c1 ZINC000147116208 HE On-Demand Bother MAPK8 29 40 CS(=O)(=O)c1cc(C(=O)NCc2ccc(Cn3ccnc3)cc2)cc([N+](=O)[O-])c1 ZINC000147116208 HE On-Demand Bother CYP17A1 19 52 CS(=O)(=O)c1cc(C(=O)NCc2ccc(Cn3ccnc3)cc2)cc([N+](=O)[O-])c1 ZINC000147116208 HE On-Demand Bother NAMPT 68 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(NS(C)(=O)=O)c1 ZINC000147116258 FC On-Demand Anodyne GRIA1 41 32 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(NS(C)(=O)=O)c1 ZINC000147116258 FC On-Demand Anodyne PCSK5 58 37 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(NS(C)(=O)=O)c1 ZINC000147116258 FC On-Demand Anodyne FURIN 65 39 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(NS(C)(=O)=O)c1 ZINC000147116258 FC On-Demand Anodyne POLG_WNV 59 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(NS(C)(=O)=O)c1 ZINC000147116258 FC On-Demand Anodyne NPFFR1 47 32 Cn1ccc(-c2ccc(N)c(F)c2)n1 ZINC000147116262 AD For-Sale Anodyne SCN4A 30 49 O=C(NCc1cccnc1-n1cccn1)c1cccn(Cc2ccccc2)c1=O ZINC000147116362 GE On-Demand Anodyne DRTS_PLAFK 19 40 O=c1ccn([C@@H]2C[C@H](F)[C@H](COC(c3ccccc3)(c3ccccc3)c3ccccc3)O2)c(=O)[nH]1 ZINC000147116388 JI Annotated Anodyne TK 42 34 O=c1ccn([C@@H]2C[C@H](F)[C@H](COC(c3ccccc3)(c3ccccc3)c3ccccc3)O2)c(=O)[nH]1 ZINC000147116388 JI Annotated Anodyne P2RY4 48 36 O=c1ccn([C@@H]2C[C@H](F)[C@H](COC(c3ccccc3)(c3ccccc3)c3ccccc3)O2)c(=O)[nH]1 ZINC000147116388 JI Annotated Anodyne P2RY2 45 38 O=c1ccn([C@@H]2C[C@H](F)[C@H](COC(c3ccccc3)(c3ccccc3)c3ccccc3)O2)c(=O)[nH]1 ZINC000147116388 JI Annotated Anodyne TK2 43 32 O=c1ccn([C@@H]2C[C@H](F)[C@H](COC(c3ccccc3)(c3ccccc3)c3ccccc3)O2)c(=O)[nH]1 ZINC000147116388 JI Annotated Anodyne DUT 34 45 O=c1ccn([C@@H]2C[C@H](F)[C@H](COC(c3ccccc3)(c3ccccc3)c3ccccc3)O2)c(=O)[nH]1 ZINC000147116388 JI Annotated Anodyne Q8II92_PLAF7 79 58 O=c1ccn([C@@H]2C[C@H](F)[C@H](COC(c3ccccc3)(c3ccccc3)c3ccccc3)O2)c(=O)[nH]1 ZINC000147116388 JI Annotated Anodyne P2RY14 57 37 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(Cn3ccnc3)cc2)c1 ZINC000147116431 FF On-Demand Bother CYP19A1 29 53 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(Cn3ccnc3)cc2)c1 ZINC000147116431 FF On-Demand Bother CYP11B1 43 42 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(Cn3ccnc3)cc2)c1 ZINC000147116431 FF On-Demand Bother CYP11B2 49 39 COc1ccc([N+](=O)[O-])c(C(=O)NCc2ccc(Cn3ccnc3)cc2)c1 ZINC000147116431 FF On-Demand Bother CYP17A1 22 50 CC(C)c1nc(CN(C)C(=O)N[C@@H](CCN2CCOCC2)C(=O)O)cs1 ZINC000147116741 GD In-Stock Anodyne CASR 46 39 CC(C)c1nc(CN(C)C(=O)N[C@@H](CCN2CCOCC2)C(=O)O)cs1 ZINC000147116741 GD In-Stock Anodyne CYP3A4 23 61 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cccc3c1OCCO3)C2 ZINC000147116883 DE On-Demand Anodyne HTR3A 34 41 CN1[C@H]2CC[C@H]1CC(NC(=O)Nc1cccc3c1OCCO3)C2 ZINC000147116883 DE On-Demand Anodyne GLRA1 43 33 COC(=O)[C@H](CCN1CCOCC1)NC(=O)N(C)Cc1csc(C(C)C)n1 ZINC000147116932 GD In-Stock Anodyne CASR 40 37 COC(=O)[C@H](CCN1CCOCC1)NC(=O)N(C)Cc1csc(C(C)C)n1 ZINC000147116932 GD In-Stock Anodyne CYP3A4 28 61 COCc1nc(C(=O)Nc2ccccc2Oc2ccccc2)cs1 ZINC000147117402 EI On-Demand Anodyne PYGL 17 42 COCc1nc(C(=O)Nc2ccccc2Oc2ccccc2)cs1 ZINC000147117402 EI On-Demand Anodyne PYGM 32 45 COCc1nc(C(=O)Nc2ccccc2Oc2ccccc2)cs1 ZINC000147117402 EI On-Demand Anodyne CHEK1 18 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117736 FG On-Demand Anodyne TSHR 52 31 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117736 FG On-Demand Anodyne KLK3 63 38 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117736 FG On-Demand Anodyne TIMP3 41 33 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117736 FG On-Demand Anodyne MMP3 44 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117736 FG On-Demand Anodyne HLA-DRB1 44 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117736 FG On-Demand Anodyne PCSK5 45 38 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117736 FG On-Demand Anodyne FURIN 62 36 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117736 FG On-Demand Anodyne MMP1 15 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117736 FG On-Demand Anodyne POLG_WNV 66 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117736 FG On-Demand Anodyne QRFPR 48 38 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117736 FG On-Demand Anodyne NPFFR1 51 36 O=c1cc(N2CCOCC2)[nH]c2c(Oc3ccccc3F)cccc12 ZINC000147117766 EG Annotated Anodyne PRKDC 75 42 O=c1cc(N2CCOCC2)[nH]c2c(Oc3ccccc3F)cccc12 ZINC000147117766 EG Annotated Anodyne PIK3CD 21 75 O=c1cc(N2CCOCC2)[nH]c2c(Oc3ccccc3F)cccc12 ZINC000147117766 EG Annotated Anodyne PIK3CB 32 75 CCc1ncc(C(=O)N2CCN(c3cccc(C)c3C)CC2)s1 ZINC000147117812 EG On-Demand Anodyne ABCB1 22 41 COc1ccc([C@H]2CCCN2C(=O)[C@H](C)OCCC(C)C)c(OC)c1 ZINC000147117842 EH On-Demand Anodyne FKBP1A 42 36 COc1ccc2c(c1)OC[C@H](C(=O)N(C)Cc1cccc(C(F)(F)F)c1)C2 ZINC000147117884 GH On-Demand Anodyne TACR1 22 40 COc1ccc2c(c1)OC[C@H](C(=O)N(C)Cc1cccc(C(F)(F)F)c1)C2 ZINC000147117884 GH On-Demand Anodyne HSD17B2 22 41 COc1ccc2c(c1)OC[C@H](C(=O)N(C)Cc1cccc(C(F)(F)F)c1)C2 ZINC000147117884 GH On-Demand Anodyne SCD 15 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117927 FG On-Demand Anodyne TSHR 52 31 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117927 FG On-Demand Anodyne KLK3 63 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117927 FG On-Demand Anodyne TIMP3 41 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117927 FG On-Demand Anodyne MMP3 44 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117927 FG On-Demand Anodyne HLA-DRB1 44 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117927 FG On-Demand Anodyne PCSK5 45 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117927 FG On-Demand Anodyne FURIN 62 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117927 FG On-Demand Anodyne MMP1 15 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117927 FG On-Demand Anodyne POLG_WNV 66 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117927 FG On-Demand Anodyne QRFPR 48 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(Cc2ccccc2)c1 ZINC000147117927 FG On-Demand Anodyne NPFFR1 51 36 CC(C)c1nc(CN(C)C(=O)N[C@H]2CCOC2=O)cs1 ZINC000147117994 CD For-Sale Anodyne CYP3A4 22 43 CC(C)c1nc(CN(C)C(=O)N[C@H]2CCOC2=O)cs1 ZINC000147117994 CD For-Sale Anodyne LUXR 69 39 CC(C)c1nc(CN(C)C(=O)N[C@H]2CCOC2=O)cs1 ZINC000147117994 CD For-Sale Anodyne TRAR 83 39 CC(C)c1nc(CN(C)C(=O)N[C@H]2CCOC2=O)cs1 ZINC000147117994 CD For-Sale Anodyne LASR 53 39 COc1cc(Cl)c(C)cc1NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147118004 EI On-Demand Bother KCNMA1 28 45 COc1ccc([C@H]2CCCN2C(=O)[C@@H](C)OCCC(C)C)c(OC)c1 ZINC000147118032 EH On-Demand Anodyne FKBP1A 42 36 c1cc(Nc2cc(C3CC3)[nH]n2)nc(NCc2ccc3[nH]ccc3n2)n1 ZINC000147118044 EG Annotated Anodyne NTRK1 20 48 c1cc(Nc2cc(C3CC3)[nH]n2)nc(NCc2ccc3[nH]ccc3n2)n1 ZINC000147118044 EG Annotated Anodyne PAK3 26 54 c1cc(Nc2cc(C3CC3)[nH]n2)nc(NCc2ccc3[nH]ccc3n2)n1 ZINC000147118044 EG Annotated Anodyne PAK1 45 54 c1cc(Nc2cc(C3CC3)[nH]n2)nc(NCc2ccc3[nH]ccc3n2)n1 ZINC000147118044 EG Annotated Anodyne PAK2 36 54 c1cc(Nc2cc(C3CC3)[nH]n2)nc(NCc2ccc3[nH]ccc3n2)n1 ZINC000147118044 EG Annotated Anodyne PKNB 99 63 COc1ccc2c(c1)OC[C@@H](C(=O)N(C)Cc1cccc(C(F)(F)F)c1)C2 ZINC000147118075 GH On-Demand Anodyne TACR1 22 40 COc1ccc2c(c1)OC[C@@H](C(=O)N(C)Cc1cccc(C(F)(F)F)c1)C2 ZINC000147118075 GH On-Demand Anodyne HSD17B2 22 41 COc1ccc2c(c1)OC[C@@H](C(=O)N(C)Cc1cccc(C(F)(F)F)c1)C2 ZINC000147118075 GH On-Demand Anodyne SCD 15 41 COc1ccc([C@@H]2CCCN2C(=O)[C@H](C)OCCC(C)C)c(OC)c1 ZINC000147118217 EH On-Demand Anodyne FKBP1A 42 36 Cc1cc(C(=O)N2CCN(c3cccc(C)c3C)CC2)cc([N+](=O)[O-])c1 ZINC000147118221 FG On-Demand Bother SLC6A9 17 45 CCCC[C@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118265 GE On-Demand Anodyne F2 35 45 CCCC[C@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118265 GE On-Demand Anodyne CHRM2 23 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118265 GE On-Demand Anodyne HRH2 15 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118265 GE On-Demand Anodyne P2RY12 201 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118265 GE On-Demand Anodyne TRY2_BOVIN 64 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118265 GE On-Demand Anodyne SLC18A3 32 47 CCCC[C@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118265 GE On-Demand Anodyne DPP7 33 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118265 GE On-Demand Anodyne ST14 43 38 CN(Cc1cccc(C(F)(F)F)c1)C(=O)c1ccc2c(c1)COC2 ZINC000147118280 EI On-Demand Anodyne TACR1 28 42 CN(Cc1cccc(C(F)(F)F)c1)C(=O)c1ccc2c(c1)COC2 ZINC000147118280 EI On-Demand Anodyne HSD17B2 25 43 COc1ccc([C@@H]2CCCN2C(=O)[C@@H](C)OCCC(C)C)c(OC)c1 ZINC000147118406 EH On-Demand Anodyne FKBP1A 42 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118440 GE On-Demand Anodyne F2 35 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118440 GE On-Demand Anodyne CHRM2 23 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118440 GE On-Demand Anodyne HRH2 15 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118440 GE On-Demand Anodyne P2RY12 201 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118440 GE On-Demand Anodyne TRY2_BOVIN 64 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118440 GE On-Demand Anodyne SLC18A3 32 47 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118440 GE On-Demand Anodyne DPP7 33 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(OC)cc2)CC1 ZINC000147118440 GE On-Demand Anodyne ST14 43 38 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne ACE 98 39 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne OPRM1 65 52 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne OPRD1 62 47 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne CACNA2D1 23 56 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne MME 101 44 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne LTA4H 16 40 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne ANPEP 79 37 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne RNPEP 36 40 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne CPA1 46 40 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne SLC15A1 0 49 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne NPFFR2 46 34 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne DPP4 27 52 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne YARS 67 38 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne DNPEP 0 43 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne ACE2 51 34 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne DPP7 87 50 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne LAP3 72 41 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne CTSC 25 42 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne AKT1 23 52 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne AMP1_PLAFQ 43 40 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne DPP8 59 51 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne DPP9 39 51 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne FAP 0 52 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne SLC15A2 0 46 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne AKT1S1 0 41 N[C@H](Cc1ccccc1)C(=O)N1C[C@H](O)[C@@H](O)C1 ZINC000147118447 CB For-Sale Anodyne BLAIMP-1 0 43 O=C(NCCOc1ccc2cc(Br)ccc2c1)NCc1cccnc1 ZINC000147118503 HH On-Demand Anodyne HRH2 25 43 O=C(NCCOc1ccc2cc(Br)ccc2c1)NCc1cccnc1 ZINC000147118503 HH On-Demand Anodyne NAMPT 61 49 O=C(NCCOc1ccc2cc(Br)ccc2c1)NCc1cccnc1 ZINC000147118503 HH On-Demand Anodyne PDS 40 37 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)OCC)cc1 ZINC000147118601 DD On-Demand Anodyne MMP2 19 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)OCC)cc1 ZINC000147118601 DD On-Demand Anodyne ADAMTS4 53 35 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)OCC)cc1 ZINC000147118601 DD On-Demand Anodyne LEF 41 36 COc1ccc(C(=O)C2CCN(C(=O)Cc3c(C)nn(C(F)F)c3C)CC2)cc1 ZINC000147118625 HH On-Demand Anodyne SLC18A3 38 43 COc1ccc([C@@H]2CCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)c(OC)c1 ZINC000147118696 HG On-Demand Bother FKBP1A 51 35 COc1ccc([C@@H]2CCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)c(OC)c1 ZINC000147118696 HG On-Demand Bother COLA 131 42 COc1ccc([C@@H]2CCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)c(OC)c1 ZINC000147118696 HG On-Demand Bother CPT1A 122 42 COc1ccc([C@@H]2CCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)c(OC)c1 ZINC000147118696 HG On-Demand Bother CPT2 45 38 CN(C)CCOc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147118776 FI On-Demand Anodyne NAMPT 22 45 C[C@@H](NC(=O)OC(C)(C)C)c1ncc(Br)cc1F ZINC000147118791 DH For-Sale Anodyne PAPA1_CARPA 45 37 C[C@@H](NC(=O)OC(C)(C)C)c1ncc(Br)cc1F ZINC000147118791 DH For-Sale Anodyne BDKRB1 28 41 Cc1nn(C(F)F)c(C)c1CC(=O)N1CCC(C(=O)c2ccccc2)CC1 ZINC000147118866 GH On-Demand Anodyne SLC18A3 42 40 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](COc2ccccc2F)c2ccccc2)c1 ZINC000147118923 HI On-Demand Bother PTGER3 50 38 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](COc2ccccc2F)c2ccccc2)c1 ZINC000147118923 HI On-Demand Bother TAAR1 24 41 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](COc2ccccc2F)c2ccccc2)c1 ZINC000147118923 HI On-Demand Bother AKR1C2 30 41 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](COc2ccccc2F)c2ccccc2)c1 ZINC000147118923 HI On-Demand Bother CTSA 56 37 CN(C)CCOc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147118969 FI On-Demand Anodyne NAMPT 22 45 C[C@H](NC(=O)OC(C)(C)C)c1ncc(Br)cc1F ZINC000147118989 DH For-Sale Anodyne PAPA1_CARPA 45 37 C[C@H](NC(=O)OC(C)(C)C)c1ncc(Br)cc1F ZINC000147118989 DH For-Sale Anodyne BDKRB1 28 41 Cc1ccc(C2=CCC(C)(C)c3cc(C(=O)C(=O)O)ccc32)cc1 ZINC000147118990 DI For-Sale Anodyne RARA 77 63 Cc1ccc(C2=CCC(C)(C)c3cc(C(=O)C(=O)O)ccc32)cc1 ZINC000147118990 DI For-Sale Anodyne RARG 73 59 Cc1ccc(C2=CCC(C)(C)c3cc(C(=O)C(=O)O)ccc32)cc1 ZINC000147118990 DI For-Sale Anodyne RXRG 48 33 Cc1ccc(C2=CCC(C)(C)c3cc(C(=O)C(=O)O)ccc32)cc1 ZINC000147118990 DI For-Sale Anodyne RARB 76 63 Cc1ccc(C2=CCC(C)(C)c3cc(C(=O)C(=O)O)ccc32)cc1 ZINC000147118990 DI For-Sale Anodyne RXRB 48 33 CCOC[C@H](C)NS(=O)(=O)c1ccc(C)cc1C ZINC000147118995 CE On-Demand Anodyne NR3C1 20 56 N#CC1CCN(C(=O)CCc2nc(-c3ccc(Cl)cc3)no2)CC1 ZINC000147118997 EG On-Demand Mild COLA 15 40 N#CC1CCN(C(=O)CCc2nc(-c3ccc(Cl)cc3)no2)CC1 ZINC000147118997 EG On-Demand Mild ETHR 64 43 CCOC(=O)C(Cc1cccc2ccccc12)(Cc1cccc2ccccc12)C(=O)OCC ZINC000147119009 IK For-Sale Anodyne MTNR1A 18 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2nc(-c3ccc(C)cc3)no2)CC1 ZINC000147119071 HD On-Demand Anodyne P2RY12 190 40 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](COc2ccccc2F)c2ccccc2)c1 ZINC000147119083 HI On-Demand Bother PTGER3 50 38 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](COc2ccccc2F)c2ccccc2)c1 ZINC000147119083 HI On-Demand Bother TAAR1 24 41 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](COc2ccccc2F)c2ccccc2)c1 ZINC000147119083 HI On-Demand Bother AKR1C2 30 41 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](COc2ccccc2F)c2ccccc2)c1 ZINC000147119083 HI On-Demand Bother CTSA 56 37 COc1ccc(CNC[C@H](O)c2ccccc2)cc1OCCCC#N ZINC000147119096 EG On-Demand Mild ADRB3 40 38 COc1ccc(CNC[C@H](O)c2ccccc2)cc1OCCCC#N ZINC000147119096 EG On-Demand Mild PHES 0 43 CN(C)CCOc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147119215 FI On-Demand Anodyne NAMPT 22 45 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild ELANE 63 39 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild MME 26 44 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild CTSL 17 45 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild CCR1 61 65 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild DPP4 21 43 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild PREP 15 46 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild PCSK5 36 41 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild FURIN 22 41 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild CAPN2 41 36 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild AMP1_PLAFQ 15 41 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild XIAP 49 40 CC(C)[C@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119230 EE On-Demand Mild BRCA1 59 32 COc1ccc(CNC[C@@H](O)c2ccccc2)cc1OCCCC#N ZINC000147119276 EG On-Demand Mild ADRB3 40 38 COc1ccc(CNC[C@@H](O)c2ccccc2)cc1OCCCC#N ZINC000147119276 EG On-Demand Mild PHES 0 43 NC(=O)c1cccc(NC(=O)C(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000147119295 GC On-Demand Clean CASR 38 41 NC(=O)c1cccc(NC(=O)C(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000147119295 GC On-Demand Clean EPHX2 22 45 NC(=O)c1cccc(NC(=O)C(=O)NCc2ccc(N3CCOCC3)cc2)c1 ZINC000147119295 GC On-Demand Clean STAT6 73 42 Nc1nc2ccc(NS(=O)(=O)c3ccccc3)cc2s1 ZINC000147119392 DF For-Sale Anodyne CA2 28 42 Nc1nc2ccc(NS(=O)(=O)c3ccccc3)cc2s1 ZINC000147119392 DF For-Sale Anodyne CA1 32 48 Nc1nc2ccc(NS(=O)(=O)c3ccccc3)cc2s1 ZINC000147119392 DF For-Sale Anodyne CA7 19 41 Nc1nc2ccc(NS(=O)(=O)c3ccccc3)cc2s1 ZINC000147119392 DF For-Sale Anodyne CA4 44 48 Nc1nc2ccc(NS(=O)(=O)c3ccccc3)cc2s1 ZINC000147119392 DF For-Sale Anodyne NR1I2 43 35 Nc1nc2ccc(NS(=O)(=O)c3ccccc3)cc2s1 ZINC000147119392 DF For-Sale Anodyne CYNT 18 41 Nc1nc2ccc(NS(=O)(=O)c3ccccc3)cc2s1 ZINC000147119392 DF For-Sale Anodyne NCE103 23 41 Nc1nc2ccc(NS(=O)(=O)c3ccccc3)cc2s1 ZINC000147119392 DF For-Sale Anodyne A6YCJ1_9METZ 15 41 CC(C)[C@@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119405 EE On-Demand Mild ELANE 63 39 CC(C)[C@@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119405 EE On-Demand Mild MME 26 44 CC(C)[C@@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119405 EE On-Demand Mild CTSL 17 45 CC(C)[C@@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119405 EE On-Demand Mild CCR1 61 65 CC(C)[C@@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119405 EE On-Demand Mild DPP4 21 43 CC(C)[C@@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119405 EE On-Demand Mild PREP 15 46 CC(C)[C@@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119405 EE On-Demand Mild PCSK5 36 41 CC(C)[C@@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119405 EE On-Demand Mild FURIN 22 41 CC(C)[C@@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119405 EE On-Demand Mild AMP1_PLAFQ 15 41 CC(C)[C@@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119405 EE On-Demand Mild XIAP 49 40 CC(C)[C@@H](NC(=O)Cc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119405 EE On-Demand Mild BRCA1 59 32 O=CCCCC(=O)N1CCCC1 ZINC000147119475 AC For-Sale Mild PREP 26 44 COc1ccc(CNC[C@H]2COc3ccccc3O2)cc1OCCCC#N ZINC000147119496 FG On-Demand Mild ADRA1D 21 61 COc1ccc(CNC[C@H]2COc3ccccc3O2)cc1OCCCC#N ZINC000147119496 FG On-Demand Mild ADRA1A 17 56 COc1ccc(CNC[C@H]2COc3ccccc3O2)cc1OCCCC#N ZINC000147119496 FG On-Demand Mild ADRA1B 22 61 O=C(NCCc1c(F)cccc1F)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147119511 EI On-Demand Anodyne MDM2 46 37 CCCCO[C@@H](C)C(=O)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000147119517 EG On-Demand Anodyne PDGFRB 37 41 CCCCO[C@@H](C)C(=O)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000147119517 EG On-Demand Anodyne CTSK 15 43 CCCCO[C@@H](C)C(=O)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000147119517 EG On-Demand Anodyne TIMP3 62 33 CCCCO[C@@H](C)C(=O)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000147119517 EG On-Demand Anodyne EPHX2 52 43 CCCCO[C@@H](C)C(=O)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000147119517 EG On-Demand Anodyne CCR8 46 33 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild PLA2G4B 60 36 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild FAAH 23 62 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild CES2 58 54 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild CES1 60 54 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild EST1_PIG 84 54 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild CES2C 65 41 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild LPAR3 43 42 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild FABP3 37 50 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild FABP5 21 65 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild Q8WS26_TRYCR 43 38 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild FABP1 16 50 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild LUXR 29 41 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild LASR 55 41 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild NOD1 48 39 CCCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCCC ZINC000147119539 KK For-Sale Mild CQSS 87 54 CC(C)[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119621 ED On-Demand Mild P2RY12 73 35 CC(C)[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119621 ED On-Demand Mild ELANE 44 43 CC(C)[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119621 ED On-Demand Mild CCR1 55 51 CC(C)[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119621 ED On-Demand Mild COLA 48 38 CC(C)[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119621 ED On-Demand Mild CPT1A 47 38 CC(C)[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147119621 ED On-Demand Mild CAPN2 51 41 O=C(NCCc1c(F)cccc1F)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147119692 EI On-Demand Anodyne MDM2 46 37 CCCCO[C@H](C)C(=O)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000147119707 EG On-Demand Anodyne PDGFRB 37 41 CCCCO[C@H](C)C(=O)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000147119707 EG On-Demand Anodyne CTSK 15 43 CCCCO[C@H](C)C(=O)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000147119707 EG On-Demand Anodyne TIMP3 62 33 CCCCO[C@H](C)C(=O)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000147119707 EG On-Demand Anodyne EPHX2 52 43 CCCCO[C@H](C)C(=O)NC1CCN(C(=O)Nc2ccccc2)CC1 ZINC000147119707 EG On-Demand Anodyne CCR8 46 33 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild PLA2G4B 60 36 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild FAAH 23 62 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild CES2 58 54 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild CES1 60 54 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild EST1_PIG 84 54 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild CES2C 65 41 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild LPAR3 43 42 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild FABP3 37 50 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild FABP5 21 65 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild Q8WS26_TRYCR 43 38 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild FABP1 16 50 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild LUXR 29 41 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild LASR 55 41 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild NOD1 48 39 CCCCCCCCCCCCCCCCCCCC(=O)CCCCCCCCCCCCCCCCCCC ZINC000147119728 KK For-Sale Mild CQSS 87 54 CCCOc1ccc(Oc2ncc(Br)s2)c(Cl)c1 ZINC000147119819 EK For-Sale Anodyne ACACB 15 55 CN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147119861 EF For-Sale Anodyne HTR1A 18 42 CN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147119861 EF For-Sale Anodyne HTR2A 15 42 CN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147119861 EF For-Sale Anodyne HRH4 20 41 CN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147119861 EF For-Sale Anodyne PRNP 41 36 CN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147119861 EF For-Sale Anodyne IRAK4 17 46 CN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147119861 EF For-Sale Anodyne WNT3 18 46 CN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147119861 EF For-Sale Anodyne TNKS 15 45 CN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147119861 EF For-Sale Anodyne G2YM83_BOTF4 62 36 O=C(NCCc1c(F)cccc1F)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147119875 EI On-Demand Anodyne MDM2 46 37 CCCOCC(=O)NC1CCN(S(=O)(=O)c2ccc(NC(C)=O)cc2)CC1 ZINC000147119908 GD On-Demand Anodyne TGM1 25 46 CCCOCC(=O)NC1CCN(S(=O)(=O)c2ccc(NC(C)=O)cc2)CC1 ZINC000147119908 GD On-Demand Anodyne EPHX2 49 48 CCCOCC(=O)NC1CCN(S(=O)(=O)c2ccc(NC(C)=O)cc2)CC1 ZINC000147119908 GD On-Demand Anodyne TGM2 96 46 CCCOCC(=O)NC1CCN(S(=O)(=O)c2ccc(NC(C)=O)cc2)CC1 ZINC000147119908 GD On-Demand Anodyne F13A1 110 46 CCOc1ccc(CN2C(=O)c3ccccc3C2=O)cc1C(=O)N1CCC(C#N)CC1 ZINC000147120025 HG On-Demand Mild HCN1 47 31 CCOc1ccc(CN2C(=O)c3ccccc3C2=O)cc1C(=O)N1CCC(C#N)CC1 ZINC000147120025 HG On-Demand Mild HCN4 41 31 CCN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147120058 FG For-Sale Anodyne HTR1A 29 44 CCN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147120058 FG For-Sale Anodyne HTR2A 31 41 CCN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147120058 FG For-Sale Anodyne HTR2C 23 40 CCN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147120058 FG For-Sale Anodyne DRD3 25 43 CCN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147120058 FG For-Sale Anodyne HTR7 22 44 CCN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147120058 FG For-Sale Anodyne PRNP 42 45 CCN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147120058 FG For-Sale Anodyne TNKS 21 43 CCN1CCN(c2ccnc(C(=O)Nc3cccc4cccnc34)c2)CC1 ZINC000147120058 FG For-Sale Anodyne G2YM83_BOTF4 66 34 CCOC[C@H](C)NS(=O)(=O)c1ccc(Cl)cc1 ZINC000147120150 CE On-Demand Anodyne S1PR1 16 47 Nc1ccc(-c2ccccc2F)nc1C(=O)Nc1cnccc1-c1ccncc1 ZINC000147120182 GI Annotated Anodyne PIM1 37 61 Nc1ccc(-c2ccccc2F)nc1C(=O)Nc1cnccc1-c1ccncc1 ZINC000147120182 GI Annotated Anodyne HDAC1 16 40 Nc1ccc(-c2ccccc2F)nc1C(=O)Nc1cnccc1-c1ccncc1 ZINC000147120182 GI Annotated Anodyne ATR 42 45 Nc1ccc(-c2ccccc2F)nc1C(=O)Nc1cnccc1-c1ccncc1 ZINC000147120182 GI Annotated Anodyne PIM2 20 61 Nc1ccc(-c2ccccc2F)nc1C(=O)Nc1cnccc1-c1ccncc1 ZINC000147120182 GI Annotated Anodyne PIM3 26 61 CCCCO[C@H](C)C(=O)N1CCN(Cc2csc(-c3ccccc3)n2)CC1 ZINC000147120351 GH On-Demand Anodyne P2RY12 184 35 C=CCN1C(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2C1=O ZINC000147120439 DD On-Demand Mild L3MBTL3 45 34 CCOC[C@H](C)NS(=O)(=O)c1ccc([N+](=O)[O-])cc1 ZINC000147120585 CD On-Demand Bother MMP2 16 50 CC(/C=C/C=O)=C\C(=O)O ZINC000147120932 AC For-Sale Reactive RARA 24 43 CC(/C=C/C=O)=C\C(=O)O ZINC000147120932 AC For-Sale Reactive RARG 23 43 CC(/C=C/C=O)=C\C(=O)O ZINC000147120932 AC For-Sale Reactive RXRG 41 43 CC(/C=C/C=O)=C\C(=O)O ZINC000147120932 AC For-Sale Reactive RARB 18 43 CC(/C=C/C=O)=C\C(=O)O ZINC000147120932 AC For-Sale Reactive RXRA 54 43 CC(/C=C/C=O)=C\C(=O)O ZINC000147120932 AC For-Sale Reactive RXRB 45 36 COc1ccc(Br)c(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147121077 HG On-Demand Anodyne MTNR1A 49 44 COc1ccc(Br)c(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147121077 HG On-Demand Anodyne ROCK2 24 42 NC1=N[C@@](c2cccc(NC(=O)c3cnc(OCCF)cn3)c2)(C(F)(F)F)CCS1 ZINC000147121091 IG Annotated Anodyne BACE2 43 45 NC1=N[C@@](c2cccc(NC(=O)c3cnc(OCCF)cn3)c2)(C(F)(F)F)CCS1 ZINC000147121091 IG Annotated Anodyne BACE1 27 51 CCCCO[C@@H](C)C(=O)Nc1ccc(NS(C)(=O)=O)cc1 ZINC000147121162 DE On-Demand Anodyne GRIN1 50 38 COc1ccc(Br)c(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147121254 HG On-Demand Anodyne MTNR1A 49 44 COc1ccc(Br)c(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147121254 HG On-Demand Anodyne ROCK2 24 42 NC1=N[C@](c2cccc(NC(=O)c3cnc(OCCF)cn3)c2)(C(F)(F)F)CCS1 ZINC000147121265 IG Annotated Anodyne BACE2 43 45 NC1=N[C@](c2cccc(NC(=O)c3cnc(OCCF)cn3)c2)(C(F)(F)F)CCS1 ZINC000147121265 IG Annotated Anodyne BACE1 27 51 CN1CCCNC(=O)C[C@@H]1c1ccccc1 ZINC000147121281 BD For-Sale Anodyne CHRNA2 44 45 CN1CCCNC(=O)C[C@@H]1c1ccccc1 ZINC000147121281 BD For-Sale Anodyne HSD17B2 48 32 CN1CCCNC(=O)C[C@@H]1c1ccccc1 ZINC000147121281 BD For-Sale Anodyne CRTY 0 45 CO[C@@H](CN)C(=O)N1CCCC1 ZINC000147121312 AB On-Demand Anodyne DPP7 50 43 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne DRD2 24 45 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne ACHE 49 51 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne HRH2 43 43 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne DRD3 22 43 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne HTR4 47 36 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne SIGMAR1 56 42 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne BCHE 24 45 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne CCR3 58 52 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne MCHR1 31 40 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne CACNA1I 57 41 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne TYRO3 27 47 O=C(NCCCN1CCCC1=O)NCC1CCN(Cc2ccccc2)CC1 ZINC000147121348 FE On-Demand Anodyne NPFFR1 41 37 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne CA2 19 43 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne CA1 28 43 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne MMP13 33 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne CA4 21 51 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne CA14 17 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne MMP2 26 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne MMP12 40 38 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne CA12 15 43 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne MMP7 22 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne ADAMTS4 47 38 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne IDO1 37 45 CCOC[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147121376 DD On-Demand Anodyne P96878_MYCTU 40 36 COc1ccc(Br)c(CNC(=O)c2ccc3c(c2)COC3)c1 ZINC000147121451 FG On-Demand Anodyne DRD4 42 32 COc1ccc(Br)c(CNC(=O)c2ccc3c(c2)COC3)c1 ZINC000147121451 FG On-Demand Anodyne MT-ND1 18 47 CN1CCCNC(=O)C[C@H]1c1ccccc1 ZINC000147121458 BD For-Sale Anodyne CHRNA2 44 45 CN1CCCNC(=O)C[C@H]1c1ccccc1 ZINC000147121458 BD For-Sale Anodyne HSD17B2 48 32 CN1CCCNC(=O)C[C@H]1c1ccccc1 ZINC000147121458 BD For-Sale Anodyne CRTY 0 45 CO[C@H](CN)C(=O)N1CCCC1 ZINC000147121474 AB For-Sale Anodyne DPP7 50 43 C[C@@]1(c2cc(NC(=O)c3cnc(OCc4ncc[nH]4)cn3)ccc2F)C=CSC(N)=N1 ZINC000147121526 IF Annotated Anodyne BACE2 44 44 C[C@@]1(c2cc(NC(=O)c3cnc(OCc4ncc[nH]4)cn3)ccc2F)C=CSC(N)=N1 ZINC000147121526 IF Annotated Anodyne BACE1 22 46 CN(C)Cc1ccccc1NC(=O)c1csc(-c2ccccc2F)n1 ZINC000147121548 FI On-Demand Anodyne PIM1 18 41 CN(C)Cc1ccccc1NC(=O)c1csc(-c2ccccc2F)n1 ZINC000147121548 FI On-Demand Anodyne CHEK1 15 41 COc1ccc(Cl)cc1C1(CNC(=O)NC2CCCCC2)CCOCC1 ZINC000147121555 GI On-Demand Anodyne CNR2 15 41 COc1ccc(Cl)cc1C1(CNC(=O)NC2CCCCC2)CCOCC1 ZINC000147121555 GI On-Demand Anodyne EPHX2 17 42 N#CC1CCN(C(=O)c2cc3ccccc3[nH]2)CC1 ZINC000147121608 CF On-Demand Mild GRIN2B 37 47 N#CC1CCN(C(=O)c2cc3ccccc3[nH]2)CC1 ZINC000147121608 CF On-Demand Mild HRH4 38 64 N#CC1CCN(C(=O)c2cc3ccccc3[nH]2)CC1 ZINC000147121608 CF On-Demand Mild CYP51A1 23 44 N#CC1CCN(C(=O)c2cc3ccccc3[nH]2)CC1 ZINC000147121608 CF On-Demand Mild FPR2 29 41 N#CC1CCN(C(=O)c2cc3ccccc3[nH]2)CC1 ZINC000147121608 CF On-Demand Mild AKR1C3 26 65 COc1cccc(NC(=O)c2ccccc2-c2nc(-c3cccc(Cl)c3)no2)c1 ZINC000147121712 HK On-Demand Anodyne AVPR2 27 40 COc1cccc(NC(=O)c2ccccc2-c2nc(-c3cccc(Cl)c3)no2)c1 ZINC000147121712 HK On-Demand Anodyne CPT1A 43 30 COc1cccc(NC(=O)c2ccccc2-c2nc(-c3cccc(Cl)c3)no2)c1 ZINC000147121712 HK On-Demand Anodyne KDR 34 41 COc1cccc(NC(=O)c2ccccc2-c2nc(-c3cccc(Cl)c3)no2)c1 ZINC000147121712 HK On-Demand Anodyne GRM5 21 50 COc1cccc(NC(=O)c2ccccc2-c2nc(-c3cccc(Cl)c3)no2)c1 ZINC000147121712 HK On-Demand Anodyne CSF1R 21 43 COc1cccc(NC(=O)c2ccccc2-c2nc(-c3cccc(Cl)c3)no2)c1 ZINC000147121712 HK On-Demand Anodyne TAAR1 41 48 COc1cccc(NC(=O)c2ccccc2-c2nc(-c3cccc(Cl)c3)no2)c1 ZINC000147121712 HK On-Demand Anodyne NR2E3 52 32 COc1cccc(NC(=O)c2ccccc2-c2nc(-c3cccc(Cl)c3)no2)c1 ZINC000147121712 HK On-Demand Anodyne LUCI_PHOPE 31 40 COc1cccc(NC(=O)c2ccccc2-c2nc(-c3cccc(Cl)c3)no2)c1 ZINC000147121712 HK On-Demand Anodyne AKR1C2 25 40 COc1cccc(NC(=O)c2ccccc2-c2nc(-c3cccc(Cl)c3)no2)c1 ZINC000147121712 HK On-Demand Anodyne KCNK3 96 43 COc1cccc(NC(=O)c2ccccc2-c2nc(-c3cccc(Cl)c3)no2)c1 ZINC000147121712 HK On-Demand Anodyne KCNK9 75 43 C[C@@]1(c2cc(NC(=O)c3cnc(NS(C)(=O)=O)cn3)ccc2F)C=CSC(N)=N1 ZINC000147121723 IE Annotated Anodyne BACE2 52 49 C[C@@]1(c2cc(NC(=O)c3cnc(NS(C)(=O)=O)cn3)ccc2F)C=CSC(N)=N1 ZINC000147121723 IE Annotated Anodyne BACE1 26 47 CCOC[C@H](C)NS(=O)(=O)c1cc([N+](=O)[O-])ccc1C ZINC000147121754 DD On-Demand Bother PIK3CA 17 40 Cc1nn(C(F)F)c(C)c1CC(=O)Nc1ccc(NS(C)(=O)=O)cc1 ZINC000147121802 FE On-Demand Anodyne P2RX7 31 41 COc1c(CBr)cccc1C(=O)O ZINC000147121845 BE For-Sale Anodyne AKR1C2 45 36 O=C(Nc1cccc(O)c1)c1ccccc1-c1nc(-c2cccc(Cl)c2)no1 ZINC000147121911 GK On-Demand Anodyne GRM4 16 40 O=C(Nc1cccc(O)c1)c1ccccc1-c1nc(-c2cccc(Cl)c2)no1 ZINC000147121911 GK On-Demand Anodyne GRM5 20 41 O=C(Nc1cccc(O)c1)c1ccccc1-c1nc(-c2cccc(Cl)c2)no1 ZINC000147121911 GK On-Demand Anodyne NR2E3 61 33 O=C(Nc1cccc(O)c1)c1ccccc1-c1nc(-c2cccc(Cl)c2)no1 ZINC000147121911 GK On-Demand Anodyne KCNK3 87 41 O=C(Nc1cccc(O)c1)c1ccccc1-c1nc(-c2cccc(Cl)c2)no1 ZINC000147121911 GK On-Demand Anodyne KCNK9 66 37 CCCCCCCCCCCCn1c(=O)n(CCCCCCCCCCCC)c(=O)n(CCCCCCCCCCCC)c1=O ZINC000147121997 KK For-Sale Mild EST1_PIG 40 33 CCCCCCCCCCCCn1c(=O)n(CCCCCCCCCCCC)c(=O)n(CCCCCCCCCCCC)c1=O ZINC000147121997 KK For-Sale Mild ASAH1 67 38 CCCCCCCCCCCCn1c(=O)n(CCCCCCCCCCCC)c(=O)n(CCCCCCCCCCCC)c1=O ZINC000147121997 KK For-Sale Mild CQSS 54 33 COc1ccc(Cl)cc1C1(CNC(=O)NCCN2CCOCC2)CCOCC1 ZINC000147122067 HE On-Demand Anodyne DRD4 46 39 COc1ccc(Cl)cc1C1(CNC(=O)NCCN2CCOCC2)CCOCC1 ZINC000147122067 HE On-Demand Anodyne HTR4 27 40 COc1ccc(Cl)cc1C1(CNC(=O)NCCN2CCOCC2)CCOCC1 ZINC000147122067 HE On-Demand Anodyne TACR2 15 40 COc1ccc(Cl)cc1C1(CNC(=O)NCCN2CCOCC2)CCOCC1 ZINC000147122067 HE On-Demand Anodyne EPHX2 22 45 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122081 GC On-Demand Anodyne F2 28 40 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122081 GC On-Demand Anodyne GHRHR 57 37 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122081 GC On-Demand Anodyne P2RY12 219 44 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122081 GC On-Demand Anodyne TRY2_BOVIN 76 35 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122081 GC On-Demand Anodyne ST14 55 38 CCCC[C@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122081 GC On-Demand Anodyne NOD1 57 32 NS(=O)(=O)c1ncccc1OCc1ccccc1 ZINC000147122084 CD For-Sale Anodyne PPIA 55 53 NS(=O)(=O)c1ncccc1OCc1ccccc1 ZINC000147122084 CD For-Sale Anodyne CA7 21 50 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne ALOX5 18 44 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne MAOB 19 48 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne PPARG 21 44 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne PPARA 21 44 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne LTA4H 82 49 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne ANPEP 26 43 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne ADORA2B 17 49 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne HDAC8 21 43 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne CA5B 17 45 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne CA5A 20 45 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne MTNR1A 29 40 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne PLA2G4B 58 42 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne FAAH 23 40 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne FURIN 40 33 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne TPSAB1 28 40 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne ADAMTS5 17 57 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne AMP1_PLAFQ 54 38 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne TAAR1 15 45 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne FFAR1 45 45 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne NCE103 23 44 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne FFAR4 40 38 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne CRTM 40 35 O=C(COc1ccc(Cc2ccccc2)cc1)NCc1ccccc1 ZINC000147122136 EH On-Demand Anodyne PDS 65 45 O=C(NCc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc2c(c1)OCO2 ZINC000147122269 GD On-Demand Clean NOS2 92 38 O=C(NCc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc2c(c1)OCO2 ZINC000147122269 GD On-Demand Clean EPHX2 15 44 O=C(NCc1ccc(N2CCOCC2)cc1)C(=O)Nc1ccc2c(c1)OCO2 ZINC000147122269 GD On-Demand Clean STAT6 56 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122274 GC On-Demand Anodyne F2 28 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122274 GC On-Demand Anodyne GHRHR 57 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122274 GC On-Demand Anodyne P2RY12 219 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122274 GC On-Demand Anodyne TRY2_BOVIN 76 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122274 GC On-Demand Anodyne ST14 55 38 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147122274 GC On-Demand Anodyne NOD1 57 32 COc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c(C(F)(F)F)c1 ZINC000147122283 HG On-Demand Bother TAAR1 26 43 CN1CCN(c2ccc([N+](=O)[O-])cc2O)CC1 ZINC000147122354 BD For-Sale Bother WDR5 47 51 Oc1ccc(OC[C@@H](O)CNCCOc2ccccc2)cc1 ZINC000147122374 DD For-Sale Anodyne ADRB2 84 66 Oc1ccc(OC[C@@H](O)CNCCOc2ccccc2)cc1 ZINC000147122374 DD For-Sale Anodyne ADRB1 94 74 Oc1ccc(OC[C@@H](O)CNCCOc2ccccc2)cc1 ZINC000147122374 DD For-Sale Anodyne DRD4 21 47 Oc1ccc(OC[C@@H](O)CNCCOc2ccccc2)cc1 ZINC000147122374 DD For-Sale Anodyne GRIN1 30 51 Oc1ccc(OC[C@@H](O)CNCCOc2ccccc2)cc1 ZINC000147122374 DD For-Sale Anodyne ADRB3 85 74 Oc1ccc(OC[C@@H](O)CNCCOc2ccccc2)cc1 ZINC000147122374 DD For-Sale Anodyne ESRRG 46 35 Oc1ccc(OC[C@@H](O)CNCCOc2ccccc2)cc1 ZINC000147122374 DD For-Sale Anodyne CYP2D6 0 40 Oc1ccc(OC[C@@H](O)CNCCOc2ccccc2)cc1 ZINC000147122374 DD For-Sale Anodyne ABCB1 19 51 CN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C(=O)Cl ZINC000147122535 DJ For-Sale Reactive TACR1 52 57 CN(C(=O)Oc1ccc(Cl)cc1)c1ccc(O)cc1 ZINC000147122584 CH For-Sale Anodyne LIPE 30 54 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne BMP1 44 38 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne MMP13 53 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne MMP2 40 52 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne MMP3 36 51 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne MMP8 28 50 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne MMP14 19 43 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne MMP9 43 52 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne MMP12 31 49 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne MMP7 35 51 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne ADAMTS4 52 34 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne MMP1 39 51 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147122589 CD On-Demand Anodyne FFAR4 20 43 CC(C)CCO[C@@H](C)C(=O)Nc1ccn(C)n1 ZINC000147122618 BD On-Demand Anodyne GCK 17 41 Oc1ccc(OC[C@H](O)CNCCOc2ccccc2)cc1 ZINC000147122637 DD For-Sale Anodyne ADRB2 84 66 Oc1ccc(OC[C@H](O)CNCCOc2ccccc2)cc1 ZINC000147122637 DD For-Sale Anodyne ADRB1 94 74 Oc1ccc(OC[C@H](O)CNCCOc2ccccc2)cc1 ZINC000147122637 DD For-Sale Anodyne DRD4 21 47 Oc1ccc(OC[C@H](O)CNCCOc2ccccc2)cc1 ZINC000147122637 DD For-Sale Anodyne GRIN1 30 51 Oc1ccc(OC[C@H](O)CNCCOc2ccccc2)cc1 ZINC000147122637 DD For-Sale Anodyne ADRB3 85 74 Oc1ccc(OC[C@H](O)CNCCOc2ccccc2)cc1 ZINC000147122637 DD For-Sale Anodyne ESRRG 46 35 Oc1ccc(OC[C@H](O)CNCCOc2ccccc2)cc1 ZINC000147122637 DD For-Sale Anodyne CYP2D6 0 40 Oc1ccc(OC[C@H](O)CNCCOc2ccccc2)cc1 ZINC000147122637 DD For-Sale Anodyne ABCB1 19 51 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne HTR1A 92 59 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne DRD2 70 59 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne DRD1 25 54 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne DRD4 48 42 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne ADRA1D 45 45 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne HTR2A 75 59 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne HTR2C 52 54 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne SLC6A4 24 47 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne ADRA1A 51 45 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne ADRA1B 33 40 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne DRD3 73 54 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne HTR7 94 43 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne HTR6 15 40 Cc1cccc(N2CCN(CCCNC(=O)COC(C)C)CC2)c1 ZINC000147122638 EE On-Demand Anodyne CACNA1G 25 43 O=C(NCCCn1ccnc1)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147122753 FH On-Demand Anodyne TBXAS1 39 45 O=C(NCCCn1ccnc1)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147122753 FH On-Demand Anodyne QPCT 37 44 O=C(NCCCn1ccnc1)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147122753 FH On-Demand Anodyne NAMPT 22 42 CCO[C@@H]1CCCN(C(=O)Nc2ccccc2N2CCc3ccccc32)C1 ZINC000147122805 FI On-Demand Anodyne KCNQ2 63 37 CC(C)CCO[C@H](C)C(=O)Nc1ccn(C)n1 ZINC000147122818 BD On-Demand Anodyne GCK 17 41 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne CA2 25 48 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne LPL 38 41 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne MME 18 40 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne CA1 29 48 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne MMP13 54 47 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne CA4 26 48 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne CA14 19 41 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne MMP2 53 50 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne MMP3 32 47 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne MMP8 33 48 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne CAPN1 20 40 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne MMP9 33 48 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne MMP12 63 41 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne CA12 20 47 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne MMP7 22 43 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne ADAMTS4 59 35 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne CA9 21 47 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne MMP1 16 43 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne LEF 40 38 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne IDO1 35 47 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne LIPG 15 41 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne LIMK2 45 38 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne MTCA1 24 43 C[C@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147122843 IF On-Demand Anodyne P96878_MYCTU 29 43 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild F2 45 50 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild PLG 24 45 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild MMP13 46 55 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild TRY2_BOVIN 96 48 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild TRY1_BOVIN 18 48 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild CCR1 37 45 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild MMP2 29 55 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild MMP3 15 40 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild MMP12 76 38 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild ST14 88 46 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild ADAMTS4 57 42 CC(C)[C@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147122926 GF On-Demand Mild TMPRSS6 46 32 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne ACE 39 44 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne PPARA 15 40 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne FOLH1 71 59 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne MME 144 62 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne LTA4H 15 46 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne ANPEP 113 45 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne PTGER4 18 40 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne RNPEP 47 49 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne CPA1 119 63 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne NAALAD2 54 55 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne MMP2 18 40 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne MMP3 24 40 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne MMP8 15 49 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne SLC1A1 15 43 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne ACE2 59 38 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne AMPD2 27 41 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne LAP3 76 45 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne FPR1 56 35 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne FFAR1 43 43 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne BLA1_STEMA 64 36 O=C(O)CCC[C@@H](Cc1ccccc1)C(=O)O ZINC000147122935 BE For-Sale Anodyne NPFFR1 57 33 COCCNC(=O)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147122974 DF On-Demand Anodyne KCNA3 39 42 COCCNC(=O)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147122974 DF On-Demand Anodyne SOAT1 16 45 COCCNC(=O)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147122974 DF On-Demand Anodyne ICMT 28 41 COCCNC(=O)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147122974 DF On-Demand Anodyne HCN1 49 30 COCCNC(=O)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147122974 DF On-Demand Anodyne HCN4 47 30 CCOC[C@H](C)NS(=O)(=O)c1ccccc1[N+](=O)[O-] ZINC000147122978 CD On-Demand Bother COLA 92 41 COc1ccc(CN[C@@H](C)c2ccc3c(c2)OCCO3)cc1OCCCC#N ZINC000147122993 GH On-Demand Mild PDE10A 22 42 CCO[C@H]1CCCN(C(=O)Nc2ccccc2N2CCc3ccccc32)C1 ZINC000147123014 FI On-Demand Anodyne KCNQ2 63 37 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne CA2 25 48 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne LPL 38 41 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne MME 18 40 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne CA1 29 48 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne MMP13 54 47 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne CA4 26 48 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne CA14 19 41 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne MMP2 53 50 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne MMP3 32 47 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne MMP8 33 48 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne CAPN1 20 40 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne MMP9 33 48 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne MMP12 63 41 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne CA12 20 47 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne MMP7 22 43 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne ADAMTS4 59 35 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne CA9 21 47 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne MMP1 16 43 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne LEF 40 38 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne IDO1 35 47 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne LIPG 15 41 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne LIMK2 45 38 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne MTCA1 24 43 C[C@@H](NS(=O)(=O)c1ccc(I)cc1)C(=O)Nc1ccccc1 ZINC000147123036 IF On-Demand Anodyne P96878_MYCTU 29 43 CC(C)(C)OC(=O)Nc1ccc(C(=O)O)c(N)c1 ZINC000147123056 CE In-Stock Anodyne AKR1C2 47 37 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne ACE 39 44 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne PPARA 15 40 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne FOLH1 71 59 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne MME 144 62 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne LTA4H 15 46 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne ANPEP 113 45 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne PTGER4 18 40 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne RNPEP 47 49 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne CPA1 119 63 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne NAALAD2 54 55 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne MMP2 18 40 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne MMP3 24 40 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne MMP8 15 49 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne SLC1A1 15 43 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne ACE2 59 38 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne AMPD2 27 41 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne LAP3 76 45 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne FPR1 56 35 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne FFAR1 43 43 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne BLA1_STEMA 64 36 O=C(O)CCC[C@H](Cc1ccccc1)C(=O)O ZINC000147123123 BE For-Sale Anodyne NPFFR1 57 33 COc1cc([N+](=O)[O-])ccc1NC(=S)N(C)C1CCCCC1 ZINC000147123130 DH For-Sale Bother KCNMA1 22 49 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild F2 45 50 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild PLG 24 45 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild MMP13 46 55 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild TRY2_BOVIN 96 48 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild TRY1_BOVIN 18 48 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild CCR1 37 45 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild MMP2 29 55 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild MMP3 15 40 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild MMP12 76 38 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild ST14 88 46 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild ADAMTS4 57 42 CC(C)[C@@H](NS(=O)(=O)c1ccc2ccccc2c1)C(=O)N1CCC(C#N)CC1 ZINC000147123131 GF On-Demand Mild TMPRSS6 46 32 COCc1nc(C(=O)Nc2nc(-c3ccc(NC(C)=O)cc3)cs2)cs1 ZINC000147123326 GH On-Demand Anodyne MPL 50 43 COCc1nc(C(=O)Nc2nc(-c3ccc(NC(C)=O)cc3)cs2)cs1 ZINC000147123326 GH On-Demand Anodyne ROCK1 20 40 COCc1nc(C(=O)Nc2nc(-c3ccc(NC(C)=O)cc3)cs2)cs1 ZINC000147123326 GH On-Demand Anodyne ROCK2 15 42 COCc1nc(C(=O)Nc2nc(-c3ccc(NC(C)=O)cc3)cs2)cs1 ZINC000147123326 GH On-Demand Anodyne VCP 16 40 N#CC1CCN(C(=O)c2cccc(CSc3cc(Cl)ccc3Cl)c2)CC1 ZINC000147123334 HK On-Demand Mild CCR3 15 40 N#CC1CCN(C(=O)c2cccc(CSc3cc(Cl)ccc3Cl)c2)CC1 ZINC000147123334 HK On-Demand Mild ST14 51 36 N#CC1CCN(C(=O)c2cccc(CSc3cc(Cl)ccc3Cl)c2)CC1 ZINC000147123334 HK On-Demand Mild TMPRSS6 44 36 CCCCO[C@@H](C)C(=O)NCc1ccc(NC(N)=O)cc1 ZINC000147123378 CD On-Demand Anodyne SCN2A 22 40 CCCCO[C@@H](C)C(=O)NCc1ccc(NC(N)=O)cc1 ZINC000147123378 CD On-Demand Anodyne S1PR4 17 41 CCCCO[C@@H](C)C(=O)NCc1ccc(NC(N)=O)cc1 ZINC000147123378 CD On-Demand Anodyne FURIN 48 35 CCCCO[C@@H](C)C(=O)NCc1ccc(NC(N)=O)cc1 ZINC000147123378 CD On-Demand Anodyne S1PR5 17 41 CO[C@@H](CCc1ccccc1)CC(C)=O ZINC000147123387 BF For-Sale Anodyne MME 46 39 CO[C@@H](CCc1ccccc1)CC(C)=O ZINC000147123387 BF For-Sale Anodyne ANPEP 51 40 CO[C@@H](CCc1ccccc1)CC(C)=O ZINC000147123387 BF For-Sale Anodyne CTSK 15 40 CO[C@@H](CCc1ccccc1)CC(C)=O ZINC000147123387 BF For-Sale Anodyne MMP2 24 43 CO[C@@H](CCc1ccccc1)CC(C)=O ZINC000147123387 BF For-Sale Anodyne MMP3 41 43 CO[C@@H](CCc1ccccc1)CC(C)=O ZINC000147123387 BF For-Sale Anodyne MMP8 15 40 CO[C@@H](CCc1ccccc1)CC(C)=O ZINC000147123387 BF For-Sale Anodyne LAP3 50 40 COc1ccc(C2(CNC(=O)NCCCN3CCCC3=O)CCCCC2)cc1 ZINC000147123474 GG On-Demand Anodyne NMBR 49 38 COc1ccc(C2(CNC(=O)NCCCN3CCCC3=O)CCCCC2)cc1 ZINC000147123474 GG On-Demand Anodyne MTNR1A 15 45 COc1ccc(C2(CNC(=O)NCCCN3CCCC3=O)CCCCC2)cc1 ZINC000147123474 GG On-Demand Anodyne SOAT1 15 41 COc1ccc(C2(CNC(=O)NCCCN3CCCC3=O)CCCCC2)cc1 ZINC000147123474 GG On-Demand Anodyne TYRO3 25 47 COc1ccc(C2(CNC(=O)NCCCN3CCCC3=O)CCCCC2)cc1 ZINC000147123474 GG On-Demand Anodyne ACAT 0 53 N#CC1CCN(C(=O)c2cccc(NC(N)=O)c2)CC1 ZINC000147123531 CD On-Demand Mild PREP 18 42 N#CC1CCN(C(=O)c2cccc(NC(N)=O)c2)CC1 ZINC000147123531 CD On-Demand Mild ST14 56 37 N#CC1CCN(C(=O)c2cccc(NC(N)=O)c2)CC1 ZINC000147123531 CD On-Demand Mild L3MBTL3 55 44 CCCCO[C@H](C)C(=O)NCc1ccc(NC(N)=O)cc1 ZINC000147123567 CD On-Demand Anodyne SCN2A 22 40 CCCCO[C@H](C)C(=O)NCc1ccc(NC(N)=O)cc1 ZINC000147123567 CD On-Demand Anodyne S1PR4 17 41 CCCCO[C@H](C)C(=O)NCc1ccc(NC(N)=O)cc1 ZINC000147123567 CD On-Demand Anodyne FURIN 48 35 CCCCO[C@H](C)C(=O)NCc1ccc(NC(N)=O)cc1 ZINC000147123567 CD On-Demand Anodyne S1PR5 17 41 CO[C@H](CCc1ccccc1)CC(C)=O ZINC000147123572 BF For-Sale Anodyne MME 46 39 CO[C@H](CCc1ccccc1)CC(C)=O ZINC000147123572 BF For-Sale Anodyne ANPEP 51 40 CO[C@H](CCc1ccccc1)CC(C)=O ZINC000147123572 BF For-Sale Anodyne CTSK 15 40 CO[C@H](CCc1ccccc1)CC(C)=O ZINC000147123572 BF For-Sale Anodyne MMP2 24 43 CO[C@H](CCc1ccccc1)CC(C)=O ZINC000147123572 BF For-Sale Anodyne MMP3 41 43 CO[C@H](CCc1ccccc1)CC(C)=O ZINC000147123572 BF For-Sale Anodyne MMP8 15 40 CO[C@H](CCc1ccccc1)CC(C)=O ZINC000147123572 BF For-Sale Anodyne LAP3 50 40 CC(C)Oc1cccc([C@@H](C)NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147123601 FF On-Demand Anodyne ACACA 69 39 CC(C)Oc1cccc([C@@H](C)NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147123601 FF On-Demand Anodyne F7 31 48 CC(C)Oc1cccc([C@@H](C)NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147123601 FF On-Demand Anodyne AOC3 15 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CN3CCC[C@@H](C)C3)cc2)c1 ZINC000147123702 GI On-Demand Bother AVPR1B 40 32 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CN3CCC[C@@H](C)C3)cc2)c1 ZINC000147123702 GI On-Demand Bother MCHR1 22 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CN3CCC[C@@H](C)C3)cc2)c1 ZINC000147123702 GI On-Demand Bother TAAR1 23 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CN3CCC[C@@H](C)C3)cc2)c1 ZINC000147123702 GI On-Demand Bother NOD1 26 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CN3CCC[C@@H](C)C3)cc2)c1 ZINC000147123702 GI On-Demand Bother NOD2 42 41 CC[C@H]1O[C@H](OC)[C@@H](O)[C@@H](O)[C@@H]1O ZINC000147123713 AA For-Sale Anodyne FIMH 51 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1nnc(-c3ccccn3)s1)C2 ZINC000147123726 FF On-Demand Anodyne ROCK2 39 46 COc1ccc2c(c1)OC[C@H](C(=O)Nc1nnc(-c3ccccn3)s1)C2 ZINC000147123726 FF On-Demand Anodyne FAAH 15 49 CCOC[C@H](C)NS(=O)(=O)c1ccc(C)cc1 ZINC000147123761 CD On-Demand Anodyne MMP13 18 47 CCOC[C@H](C)NS(=O)(=O)c1ccc(C)cc1 ZINC000147123761 CD On-Demand Anodyne MMP7 18 48 CCOC[C@H](C)NS(=O)(=O)c1ccc(C)cc1 ZINC000147123761 CD On-Demand Anodyne ADAMTS4 55 34 CC(C)Oc1cccc([C@H](C)NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147123789 FF On-Demand Anodyne ACACA 69 39 CC(C)Oc1cccc([C@H](C)NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147123789 FF On-Demand Anodyne F7 31 48 CC(C)Oc1cccc([C@H](C)NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147123789 FF On-Demand Anodyne AOC3 15 44 CCOC(=O)c1cnc(Cl)cc1NCc1ccc(OC)cc1 ZINC000147123851 DH For-Sale Anodyne PDE5A 24 46 CCOC(=O)c1cnc(Cl)cc1NCc1ccc(OC)cc1 ZINC000147123851 DH For-Sale Anodyne PROKR1 67 35 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CN3CCC[C@H](C)C3)cc2)c1 ZINC000147123899 GI On-Demand Bother AVPR1B 40 32 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CN3CCC[C@H](C)C3)cc2)c1 ZINC000147123899 GI On-Demand Bother MCHR1 22 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CN3CCC[C@H](C)C3)cc2)c1 ZINC000147123899 GI On-Demand Bother TAAR1 23 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CN3CCC[C@H](C)C3)cc2)c1 ZINC000147123899 GI On-Demand Bother NOD1 26 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CN3CCC[C@H](C)C3)cc2)c1 ZINC000147123899 GI On-Demand Bother NOD2 42 41 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne CHRM2 22 45 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne CHRM1 15 42 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne DRD2 24 55 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne DRD4 61 48 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne ACHE 39 47 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne HRH1 16 40 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne DRD3 21 55 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne CHRM3 28 40 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne LTA4H 25 46 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne SIGMAR1 64 63 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne SSTR5 44 35 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne CCR3 39 48 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne EPHX2 39 46 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne PDK1 26 40 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne MCHR1 50 54 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne CACNA1G 42 49 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne CCR8 25 46 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne BIRC2 45 45 CNC(=O)CN1CCC(NC(=O)C2CCN(Cc3ccccc3)CC2)CC1 ZINC000147123917 FD On-Demand Anodyne NPFFR1 50 36 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1nnc(-c3ccccn3)s1)C2 ZINC000147123939 FF On-Demand Anodyne ROCK2 39 46 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1nnc(-c3ccccn3)s1)C2 ZINC000147123939 FF On-Demand Anodyne FAAH 15 49 O=C(NCc1c(F)cc(F)cc1F)c1ccccc1Cl ZINC000147123941 CH On-Demand Anodyne P2RX7 53 38 O=C(NCc1c(F)cc(F)cc1F)c1ccccc1Cl ZINC000147123941 CH On-Demand Anodyne ECR 61 46 O=C(NCc1c(F)cc(F)cc1F)c1ccccc1Cl ZINC000147123941 CH On-Demand Anodyne E3UJZ5_SPOLI 47 45 NC(=O)c1ccc(OCC(=O)N[C@H](C(=O)Nc2ccccc2)c2ccccc2)cc1 ZINC000147124065 HF On-Demand Anodyne LTA4H 33 46 NC(=O)c1ccc(OCC(=O)N[C@H](C(=O)Nc2ccccc2)c2ccccc2)cc1 ZINC000147124065 HF On-Demand Anodyne HDAC8 15 55 NC(=O)c1ccc(OCC(=O)N[C@H](C(=O)Nc2ccccc2)c2ccccc2)cc1 ZINC000147124065 HF On-Demand Anodyne PLAU 43 37 NC(=O)c1ccc(OCC(=O)N[C@H](C(=O)Nc2ccccc2)c2ccccc2)cc1 ZINC000147124065 HF On-Demand Anodyne F7 23 41 NC(=O)c1ccc(OCC(=O)N[C@H](C(=O)Nc2ccccc2)c2ccccc2)cc1 ZINC000147124065 HF On-Demand Anodyne ACR 57 38 CS(=O)(=O)c1cc(C(=O)Nc2nc(-c3ccccc3)ns2)cc([N+](=O)[O-])c1 ZINC000147124411 HF On-Demand Bother GCK 23 41 COc1cc(-c2nc3cc(C)c(C)cc3[nH]2)ccc1O ZINC000147124444 CH On-Demand Anodyne CHEK2 54 41 COc1cc(-c2nc3cc(C)c(C)cc3[nH]2)ccc1O ZINC000147124444 CH On-Demand Anodyne GUSB 0 46 COc1cc(-c2nc3cc(C)c(C)cc3[nH]2)ccc1O ZINC000147124444 CH On-Demand Anodyne QDPR 0 41 COc1cc(-c2nc3cc(C)c(C)cc3[nH]2)ccc1O ZINC000147124444 CH On-Demand Anodyne HPSE 20 53 CC(C)(C)C(=O)NCC(=O)N1CCC(C#N)CC1 ZINC000147124561 CC On-Demand Mild DPP4 23 40 CC(C)(C)C(=O)NCC(=O)N1CCC(C#N)CC1 ZINC000147124561 CC On-Demand Mild PREP 20 48 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(-c3ccccc3)ns2)c1 ZINC000147124589 FG On-Demand Bother LUCI_LUCLA 23 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(-c3ccccc3)ns2)c1 ZINC000147124589 FG On-Demand Bother TAAR1 20 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(-c3ccccc3)ns2)c1 ZINC000147124589 FG On-Demand Bother AKR1C2 42 43 CCCC[C@@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124633 FJ Annotated Anodyne PTGFR 44 38 CCCC[C@@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124633 FJ Annotated Anodyne PTGER2 46 53 CCCC[C@@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124633 FJ Annotated Anodyne PTGER1 31 53 CCCC[C@@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124633 FJ Annotated Anodyne PTGER4 25 53 CCCC[C@@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124633 FJ Annotated Anodyne PTGER3 26 53 CCCC[C@@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124633 FJ Annotated Anodyne PTGDR 0 49 CCCC[C@@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124633 FJ Annotated Anodyne SLCO2A1 68 49 C[C@H](Nc1nccc(Nc2cc([C@H]3C[C@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147124722 GH Annotated Anodyne NTRK1 21 52 C[C@H](Nc1nccc(Nc2cc([C@H]3C[C@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147124722 GH Annotated Anodyne PAK3 27 56 C[C@H](Nc1nccc(Nc2cc([C@H]3C[C@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147124722 GH Annotated Anodyne PAK1 49 56 C[C@H](Nc1nccc(Nc2cc([C@H]3C[C@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147124722 GH Annotated Anodyne PAK2 37 56 C[C@H](Nc1nccc(Nc2cc([C@H]3C[C@H]3F)[nH]n2)n1)c1ccc2[nH]ccc2n1 ZINC000147124722 GH Annotated Anodyne PKNB 47 43 O=C1CC(Cc2ccccc2)CC(=O)O1 ZINC000147124788 BD For-Sale Reactive LUCI_PHOPY 71 34 CCCC[C@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124802 FJ Annotated Anodyne PTGFR 44 38 CCCC[C@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124802 FJ Annotated Anodyne PTGER2 46 53 CCCC[C@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124802 FJ Annotated Anodyne PTGER1 31 53 CCCC[C@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124802 FJ Annotated Anodyne PTGER4 25 53 CCCC[C@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124802 FJ Annotated Anodyne PTGER3 26 53 CCCC[C@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124802 FJ Annotated Anodyne PTGDR 0 49 CCCC[C@H](CC)[C@@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147124802 FJ Annotated Anodyne SLCO2A1 68 49 CCNC(=O)[C@H](C)NCc1ccc(OC)c(OCCCC#N)c1 ZINC000147124828 DD On-Demand Mild REN 25 40 CC(C)Oc1cccc(CC(=O)Nc2nc(-c3ccc[nH]3)cs2)c1 ZINC000147124892 EI On-Demand Anodyne CSNK1D 24 42 CC(C)Oc1cccc(CC(=O)Nc2nc(-c3ccc[nH]3)cs2)c1 ZINC000147124892 EI On-Demand Anodyne ROCK1 26 45 CC(C)Oc1cccc(CC(=O)Nc2nc(-c3ccc[nH]3)cs2)c1 ZINC000147124892 EI On-Demand Anodyne ROCK2 20 45 CC(C)Oc1cccc(CC(=O)Nc2nc(-c3ccc[nH]3)cs2)c1 ZINC000147124892 EI On-Demand Anodyne TRPA1 20 40 CCOC[C@H](C)NS(=O)(=O)c1ccc2c(c1)OCCO2 ZINC000147124915 DD On-Demand Anodyne PKM 30 42 COC(=O)CNC(=O)Cc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147124923 GC On-Demand Anodyne PRSS1 16 40 COC(=O)CNC(=O)Cc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147124923 GC On-Demand Anodyne ADORA2B 42 43 COC(=O)CNC(=O)Cc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147124923 GC On-Demand Anodyne ACR 64 37 COC(=O)CNC(=O)Cc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147124923 GC On-Demand Anodyne CA9 19 43 CCCC[C@@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125009 FJ Annotated Anodyne PTGER2 41 43 CCCC[C@@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125009 FJ Annotated Anodyne PTGER1 31 53 CCCC[C@@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125009 FJ Annotated Anodyne PTGER4 25 53 CCCC[C@@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125009 FJ Annotated Anodyne PTGER3 26 53 CCCC[C@@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125009 FJ Annotated Anodyne PTGDR 0 49 CCCC[C@@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125009 FJ Annotated Anodyne SLCO2A1 68 49 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@H](C)O[C@H](C)C2)n1 ZINC000147125132 GE On-Demand Anodyne HTR1A 20 44 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@H](C)O[C@H](C)C2)n1 ZINC000147125132 GE On-Demand Anodyne DRD2 25 45 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@H](C)O[C@H](C)C2)n1 ZINC000147125132 GE On-Demand Anodyne DRD4 16 45 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@H](C)O[C@H](C)C2)n1 ZINC000147125132 GE On-Demand Anodyne DRD3 46 44 CCCC[C@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125170 FJ Annotated Anodyne PTGFR 44 38 CCCC[C@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125170 FJ Annotated Anodyne PTGER2 46 53 CCCC[C@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125170 FJ Annotated Anodyne PTGER1 31 53 CCCC[C@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125170 FJ Annotated Anodyne PTGER4 25 53 CCCC[C@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125170 FJ Annotated Anodyne PTGER3 26 53 CCCC[C@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125170 FJ Annotated Anodyne PTGDR 0 49 CCCC[C@H](CC)[C@H](O)/C=C/[C@@H]1CCC(=O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147125170 FJ Annotated Anodyne SLCO2A1 68 49 C[C@@H](Cn1cccn1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147125194 ED On-Demand Anodyne DRTS_PLAFK 20 43 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1nc(-c2ccc[nH]2)cs1 ZINC000147125287 EI On-Demand Anodyne ROCK1 23 48 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1nc(-c2ccc[nH]2)cs1 ZINC000147125287 EI On-Demand Anodyne ROCK2 19 48 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1nc(-c2ccc[nH]2)cs1 ZINC000147125287 EI On-Demand Anodyne TRPA1 15 42 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@@H](C)O[C@H](C)C2)n1 ZINC000147125296 GE On-Demand Anodyne HTR1A 20 44 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@@H](C)O[C@H](C)C2)n1 ZINC000147125296 GE On-Demand Anodyne DRD2 25 45 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@@H](C)O[C@H](C)C2)n1 ZINC000147125296 GE On-Demand Anodyne DRD4 16 45 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@@H](C)O[C@H](C)C2)n1 ZINC000147125296 GE On-Demand Anodyne DRD3 46 44 CCOC[C@H](C)NS(=O)(=O)c1ccc(F)c(F)c1 ZINC000147125330 CD On-Demand Anodyne LEF 64 44 C[C@H](Cn1cccn1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147125379 ED On-Demand Anodyne DRTS_PLAFK 20 43 CC(C)NC(=O)NCc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147125464 EE On-Demand Mild L3MBTL3 71 40 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@H](C)O[C@@H](C)C2)n1 ZINC000147125487 GE On-Demand Anodyne HTR1A 20 44 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@H](C)O[C@@H](C)C2)n1 ZINC000147125487 GE On-Demand Anodyne DRD2 25 45 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@H](C)O[C@@H](C)C2)n1 ZINC000147125487 GE On-Demand Anodyne DRD4 16 45 COc1ccc(C)cc1-n1ccc(C(=O)NCCCN2C[C@H](C)O[C@@H](C)C2)n1 ZINC000147125487 GE On-Demand Anodyne DRD3 46 44 C[C@H](Cc1cccc(F)c1)C(=O)Nc1nc(-c2ccc[nH]2)cs1 ZINC000147125496 EI On-Demand Anodyne ROCK1 23 48 C[C@H](Cc1cccc(F)c1)C(=O)Nc1nc(-c2ccc[nH]2)cs1 ZINC000147125496 EI On-Demand Anodyne ROCK2 19 48 C[C@H](Cc1cccc(F)c1)C(=O)Nc1nc(-c2ccc[nH]2)cs1 ZINC000147125496 EI On-Demand Anodyne TRPA1 15 42 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild CELA1 20 45 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild GRIN2B 40 47 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild CTSB 22 41 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild CTSK 25 46 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild CTSL 22 46 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild DPP4 24 41 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild PREP 74 53 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild LGMN 76 46 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild CTSS 29 41 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild ACE2 24 41 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild TGM2 36 41 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild KLK5 22 40 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild DPP8 22 41 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild F13A1 32 41 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild BIRC2 18 47 N#CC[C@@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125595 CF For-Sale Mild SLC12A5 62 40 CCCNC(=O)CC(=O)c1ccccc1 ZINC000147125663 BD In-Stock Anodyne HAO1 45 37 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild CELA1 20 45 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild GRIN2B 40 47 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild CTSB 22 41 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild CTSK 25 46 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild CTSL 22 46 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild DPP4 24 41 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild PREP 74 53 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild LGMN 76 46 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild CTSS 29 41 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild ACE2 24 41 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild TGM2 36 41 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild KLK5 22 40 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild DPP8 22 41 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild F13A1 32 41 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild BIRC2 18 47 N#CC[C@H]1CCCN(C(=O)OCc2ccccc2)C1 ZINC000147125757 CF For-Sale Mild SLC12A5 62 40 CC(C)(C)OC(=O)Nc1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147125934 EG On-Demand Mild NPY2R 30 42 CC(C)(C)OC(=O)Nc1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147125934 EG On-Demand Mild GPR119 23 40 CCCCN(Cc1ccccc1)S(=O)(=O)c1ccccc1[N+](=O)[O-] ZINC000147125943 EH For-Sale Bother COLA 104 45 CCCCN(Cc1ccccc1)S(=O)(=O)c1ccccc1[N+](=O)[O-] ZINC000147125943 EH For-Sale Bother MMP2 16 55 CCCCN(Cc1ccccc1)S(=O)(=O)c1ccccc1[N+](=O)[O-] ZINC000147125943 EH For-Sale Bother MMP8 33 55 CCCCN(Cc1ccccc1)S(=O)(=O)c1ccccc1[N+](=O)[O-] ZINC000147125943 EH For-Sale Bother MMP9 18 55 CCCCN(Cc1ccccc1)S(=O)(=O)c1ccccc1[N+](=O)[O-] ZINC000147125943 EH For-Sale Bother MMP1 24 55 NC(=O)c1ccc(OCC(=O)N2CCN(c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000147126329 GD On-Demand Bother HTR1D 18 49 NC(=O)c1ccc(OCC(=O)N2CCN(c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000147126329 GD On-Demand Bother HTR1B 19 42 NC(=O)c1ccc(OCC(=O)N2CCN(c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000147126329 GD On-Demand Bother CACNA1D 45 37 NC(=O)c1ccc(OCC(=O)N2CCN(c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000147126329 GD On-Demand Bother CPT1A 20 40 NC(=O)c1ccc(OCC(=O)N2CCN(c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000147126329 GD On-Demand Bother SSTR1 45 42 NC(=O)c1ccc(OCC(=O)N2CCN(c3cccc([N+](=O)[O-])c3)CC2)cc1 ZINC000147126329 GD On-Demand Bother ACR 25 40 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne OPRM1 16 41 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne CACNA2D1 23 45 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne MME 42 43 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne ANPEP 61 52 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne FCER2 52 34 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne RNPEP 40 52 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne CAPNS1 54 32 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne CAPN1 40 38 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne CAPN2 43 34 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne LAP3 62 54 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne FPR1 41 35 CC(C)C[C@](N)(C(=O)O)C(=O)[C@H](O)[C@H](N)Cc1ccccc1 ZINC000147126332 DC For-Sale Anodyne AMP1_PLAFQ 44 52 CCOC[C@H](C)NS(=O)(=O)c1c(C)cc(C)cc1C ZINC000147126506 CE On-Demand Anodyne NR3C1 28 63 CCOC[C@H](C)NS(=O)(=O)c1c(C)cc(C)cc1C ZINC000147126506 CE On-Demand Anodyne PGR 17 50 CCOC[C@H](C)NS(=O)(=O)c1c(C)cc(C)cc1C ZINC000147126506 CE On-Demand Anodyne NR3C2 39 50 O=C(Nc1ccn(Cc2ccccc2)n1)c1cnn(-c2ccccc2Cl)c1 ZINC000147126516 GI On-Demand Anodyne ITK 20 48 CN(C)Cc1ccccc1NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147126600 FG On-Demand Anodyne DRTS_PLAFK 20 44 CN(C)Cc1ccccc1NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147126600 FG On-Demand Anodyne PTGER3 34 46 O=C(c1ccc2c(c1)COC2)N1C[C@@H]2CCCN2Cc2ccccc21 ZINC000147126775 EG On-Demand Anodyne AVPR2 73 45 O=C(c1ccc2c(c1)COC2)N1C[C@@H]2CCCN2Cc2ccccc21 ZINC000147126775 EG On-Demand Anodyne AVPR1A 41 41 O=C(c1ccc2c(c1)COC2)N1C[C@@H]2CCCN2Cc2ccccc21 ZINC000147126775 EG On-Demand Anodyne L3MBTL3 46 34 CNS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147126812 DC On-Demand Mild L3MBTL3 71 40 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne CHRM2 18 40 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne DRD2 17 49 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne DRD4 45 46 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne ACHE 32 42 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne SLC6A1 124 38 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne DRD3 18 48 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne SIGMAR1 47 54 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne CCR3 37 43 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne CCR5 15 42 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne MCHR1 38 47 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne CACNA1G 21 45 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne CCR8 19 41 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne BIRC2 65 41 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne BIRC8 43 38 CNC(=O)CN1CCC(NC(=O)[C@@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126825 FD On-Demand Anodyne NPFFR1 44 33 O=C(Nc1cnn(Cc2ccccc2)c1)c1ccc2nc3n(c2c1)CCCNC3=O ZINC000147126872 HF Annotated Anodyne ITK 20 46 O=C(Nc1cnn(Cc2ccccc2)c1)c1ccc2nc3n(c2c1)CCCNC3=O ZINC000147126872 HF Annotated Anodyne RPS6KA3 99 68 O=C(Nc1cnn(Cc2ccccc2)c1)c1ccc2nc3n(c2c1)CCCNC3=O ZINC000147126872 HF Annotated Anodyne PANC 54 38 COc1cccc(C(=O)Nc2ccc(C#N)cc2)c1[N+](=O)[O-] ZINC000147126969 CF On-Demand Mild GLMU 0 40 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne CHRM2 18 40 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne DRD2 17 49 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne DRD4 45 46 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne ACHE 32 42 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne SLC6A1 124 38 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne DRD3 18 48 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne SIGMAR1 47 54 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne CCR3 37 43 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne CCR5 15 42 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne MCHR1 38 47 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne CACNA1G 21 45 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne CCR8 19 41 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne BIRC2 65 41 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne BIRC8 43 38 CNC(=O)CN1CCC(NC(=O)[C@H]2CCCN(Cc3ccccc3)C2)CC1 ZINC000147126997 FD On-Demand Anodyne NPFFR1 44 33 Cc1nc(-c2cccc(NC(=O)c3ccc4nc5n(c4c3)CCCNC5=O)c2)cs1 ZINC000147127064 HH Annotated Anodyne MAPKAPK2 21 49 Cc1nc(-c2cccc(NC(=O)c3ccc4nc5n(c4c3)CCCNC5=O)c2)cs1 ZINC000147127064 HH Annotated Anodyne RPS6KA3 91 57 Cc1nc(-c2cccc(NC(=O)c3ccc4nc5n(c4c3)CCCNC5=O)c2)cs1 ZINC000147127064 HH Annotated Anodyne KCNK3 63 36 CCNC(=O)c1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147127072 GE On-Demand Bother CA2 27 40 CCNC(=O)c1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147127072 GE On-Demand Bother CYNT 18 40 CC(C)c1nc(N(C)S(C)(=O)=O)nc(-c2ccc(F)cc2)c1/C=C/[C@@H](O)CC(=O)CC(=O)OC(C)(C)C ZINC000147127151 KH For-Sale Anodyne HMGCR 66 68 CN1[C@H](C(=O)O)C[C@H]2CCCC[C@@H]21 ZINC000147127172 AD For-Sale Anodyne ACE 30 55 CNC(=O)CN1CCC(NC(=O)CN2CCc3ccccc32)CC1 ZINC000147127218 EC On-Demand Anodyne CHRM1 15 46 CNC(=O)CN1CCC(NC(=O)CN2CCc3ccccc32)CC1 ZINC000147127218 EC On-Demand Anodyne SIGMAR1 19 43 CNC(=O)CN1CCC(NC(=O)CN2CCc3ccccc32)CC1 ZINC000147127218 EC On-Demand Anodyne MCHR1 15 42 Brc1ccc2ncnc(N3CCC(N4CCCCC4)CC3)c2c1 ZINC000147127329 GH On-Demand Anodyne PDE3A 46 35 Brc1ccc2ncnc(N3CCC(N4CCCCC4)CC3)c2c1 ZINC000147127329 GH On-Demand Anodyne HRH3 32 53 Brc1ccc2ncnc(N3CCC(N4CCCCC4)CC3)c2c1 ZINC000147127329 GH On-Demand Anodyne CCR4 22 41 Brc1ccc2ncnc(N3CCC(N4CCCCC4)CC3)c2c1 ZINC000147127329 GH On-Demand Anodyne PDE3B 68 35 Brc1ccc2ncnc(N3CCC(N4CCCCC4)CC3)c2c1 ZINC000147127329 GH On-Demand Anodyne L3MBTL3 71 41 Cc1ccccc1[C@@H](C)NC(=O)N(C)Cc1cscn1 ZINC000147127334 CG On-Demand Anodyne BMP1 52 34 C[C@H](NC(=O)c1cccn(Cc2ccccc2)c1=O)c1nncn1C ZINC000147127342 ED On-Demand Anodyne DRTS_PLAFK 19 41 Cc1ccnc(NC(=O)c2ccc3nc4n(c3c2)CCCNC4=O)c1 ZINC000147127374 EE Annotated Anodyne MAPKAPK2 56 37 Cc1ccnc(NC(=O)c2ccc3nc4n(c3c2)CCCNC4=O)c1 ZINC000147127374 EE Annotated Anodyne RPS6KA3 96 52 Cc1ccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127384 GI On-Demand Anodyne PRCP 46 36 Cc1ccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127384 GI On-Demand Anodyne TYK2 41 35 Cc1ccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127384 GI On-Demand Anodyne MDM2 48 36 Cc1ccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127384 GI On-Demand Anodyne NPBWR1 54 34 Cc1ccccc1[C@H](C)NC(=O)N(C)Cc1cscn1 ZINC000147127491 CG On-Demand Anodyne BMP1 52 34 C[C@@H](NC(=O)c1cccn(Cc2ccccc2)c1=O)c1nncn1C ZINC000147127503 ED On-Demand Anodyne DRTS_PLAFK 19 41 CC(C)(C)OC(=O)Nc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147127556 EG On-Demand Mild EPHX2 21 49 CC(C)(C)OC(=O)Nc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147127556 EG On-Demand Mild L3MBTL3 65 37 Cc1ccc(NC(=O)C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127559 GI On-Demand Anodyne PRCP 46 36 Cc1ccc(NC(=O)C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127559 GI On-Demand Anodyne TYK2 41 35 Cc1ccc(NC(=O)C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127559 GI On-Demand Anodyne MDM2 48 36 Cc1ccc(NC(=O)C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127559 GI On-Demand Anodyne NPBWR1 54 34 O=C(Nc1cccc(F)c1)c1ccc2nc3n(c2c1)CCCNC3=O ZINC000147127561 EF Annotated Anodyne MAPKAPK2 19 55 O=C(Nc1cccc(F)c1)c1ccc2nc3n(c2c1)CCCNC3=O ZINC000147127561 EF Annotated Anodyne RPS6KA3 97 56 O=C(Nc1cccc(F)c1)c1ccc2nc3n(c2c1)CCCNC3=O ZINC000147127561 EF Annotated Anodyne TAAR1 39 45 O=C(Nc1cccc(F)c1)c1ccc2nc3n(c2c1)CCCNC3=O ZINC000147127561 EF Annotated Anodyne KCNK3 92 44 O=C(Nc1cccc(F)c1)c1ccc2nc3n(c2c1)CCCNC3=O ZINC000147127561 EF Annotated Anodyne KCNK9 47 44 O=C(O)C(NC[C@H](NC(C(=O)O)C(=O)O)C(=O)O)C(=O)O ZINC000147127640 DA For-Sale Anodyne CPA1 20 40 Cc1ccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127766 GI On-Demand Anodyne PRCP 46 36 Cc1ccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127766 GI On-Demand Anodyne TYK2 41 35 Cc1ccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127766 GI On-Demand Anodyne MDM2 48 36 Cc1ccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147127766 GI On-Demand Anodyne NPBWR1 54 34 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000147127769 EE On-Demand Anodyne CASR 16 41 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000147127769 EE On-Demand Anodyne MMP9 23 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000147127769 EE On-Demand Anodyne MMP7 15 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC(F)(F)F)cc1 ZINC000147127769 EE On-Demand Anodyne ADAMTS4 45 34 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC(C(=O)Nc3ccc(C)cn3)CC1)C2 ZINC000147127992 HF On-Demand Anodyne ROCK2 34 43 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC(C(=O)Nc3ccc(C)cn3)CC1)C2 ZINC000147127992 HF On-Demand Anodyne LUCI_LUCLA 17 44 Cc1cc(=O)nc(-c2cccc(NC(=O)COc3ccc(C(N)=O)cc3)c2)[nH]1 ZINC000147128152 GD On-Demand Anodyne ADORA1 22 50 Cc1cc(=O)nc(-c2cccc(NC(=O)COc3ccc(C(N)=O)cc3)c2)[nH]1 ZINC000147128152 GD On-Demand Anodyne ADORA2A 20 50 Cc1cc(=O)nc(-c2cccc(NC(=O)COc3ccc(C(N)=O)cc3)c2)[nH]1 ZINC000147128152 GD On-Demand Anodyne ADORA2B 59 50 Cc1cc(=O)nc(-c2cccc(NC(=O)COc3ccc(C(N)=O)cc3)c2)[nH]1 ZINC000147128152 GD On-Demand Anodyne CHEK2 75 40 O=C(Nc1cccc(N2CCCCC2=O)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147128153 EH On-Demand Anodyne CCKBR 43 36 O=C(Nc1cccc(N2CCCCC2=O)c1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147128153 EH On-Demand Anodyne EPHX2 33 47 Cc1ccc(NC(=O)[C@@H]2CCCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)C2)nc1 ZINC000147128202 GI On-Demand Anodyne MDM2 57 35 O=C(Nc1cccc(N2CCCCC2=O)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147128335 EH On-Demand Anodyne CCKBR 43 36 O=C(Nc1cccc(N2CCCCC2=O)c1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147128335 EH On-Demand Anodyne EPHX2 33 47 O=C(Nc1cccc(N2CCCCC2=O)c1)c1cccn(Cc2ccccc2)c1=O ZINC000147128433 HH On-Demand Anodyne DRTS_PLAFK 19 41 O=C(Nc1cccc(N2CCCCC2=O)c1)c1cccn(Cc2ccccc2)c1=O ZINC000147128433 HH On-Demand Anodyne PTGER3 31 43 O=C(Nc1cccc(N2CCCCC2=O)c1)c1cccn(Cc2ccccc2)c1=O ZINC000147128433 HH On-Demand Anodyne KCNK3 51 38 CCOC(=O)[C@H](CCI)NC(=O)N(C)Cc1csc(C(C)C)n1 ZINC000147128505 JG For-Sale Reactive CYP3A4 23 51 O=C(Nc1cccc(N2CCCCC2=O)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147128524 EH On-Demand Anodyne CCKBR 43 36 O=C(Nc1cccc(N2CCCCC2=O)c1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147128524 EH On-Demand Anodyne EPHX2 33 47 Cc1ccc(NC(=O)[C@@H]2CCCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)C2)nc1 ZINC000147128555 GI On-Demand Anodyne MDM2 57 35 N#CC1CCN(C(=O)C[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147128646 FG On-Demand Mild PTAFR 40 44 N#CC1CCN(C(=O)C[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147128646 FG On-Demand Mild DPP4 18 42 N#CC1CCN(C(=O)C[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147128646 FG On-Demand Mild FAP 0 45 N#CC1CCN(C(=O)C[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147128646 FG On-Demand Mild UTS2 47 36 O=C(Nc1cccc(N2CCCCC2=O)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147128729 EH On-Demand Anodyne CCKBR 43 36 O=C(Nc1cccc(N2CCCCC2=O)c1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147128729 EH On-Demand Anodyne EPHX2 33 47 C[C@@H]1NC(=O)c2cc3ccc(C(=O)Nc4nc5ccccc5n4CCCN(C)C)nc3n2[C@H]1C ZINC000147128789 JG Annotated Anodyne RPS6KA3 26 65 O=C(C1CCN(Cc2ccnnc2)CC1)N1CCC(Oc2ccccn2)CC1 ZINC000147128813 GE For-Sale Anodyne HRH3 17 45 O=C(C1CCN(Cc2ccnnc2)CC1)N1CCC(Oc2ccccn2)CC1 ZINC000147128813 GE For-Sale Anodyne SIGMAR1 19 44 O=C(C1CCN(Cc2ccnnc2)CC1)N1CCC(Oc2ccccn2)CC1 ZINC000147128813 GE For-Sale Anodyne SCN5A 50 33 CCc1cccc(C(=O)N2CCN(C(=O)OC(C)(C)C)CC2)n1 ZINC000147128829 DE On-Demand Anodyne GPR119 40 44 COCc1nc(C(=O)Nc2nc3c(s2)CN(Cc2ccccc2)CC3)cs1 ZINC000147128842 HH On-Demand Anodyne NOD2 42 38 COCc1nc(C(=O)Nc2nc3c(s2)CN(Cc2ccccc2)CC3)cs1 ZINC000147128842 HH On-Demand Anodyne SLC27A1 29 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(C)c([N+](=O)[O-])c1 ZINC000147128866 DD On-Demand Bother LEF 40 36 NC(=O)c1ccc(OCC(=O)Nc2cc(C(N)=O)ccc2F)cc1 ZINC000147128901 ED On-Demand Anodyne HIF1A 22 44 CC(C)Nc1cc(Cl)cnc1C(N)=O ZINC000147128904 BD For-Sale Anodyne SYK 45 33 CCOC(=O)N1CCC(NC(=O)NNC(=O)c2ccc(C)s2)CC1 ZINC000147128907 FD On-Demand Reactive CHRM1 15 46 CCOC(=O)N1CCC(NC(=O)NNC(=O)c2ccc(C)s2)CC1 ZINC000147128907 FD On-Demand Reactive EPHX2 39 40 CCOC(=O)N1CCC(NC(=O)NNC(=O)c2ccc(C)s2)CC1 ZINC000147128907 FD On-Demand Reactive CCR8 34 43 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(N3CCCCC3=O)c2)C1 ZINC000147128910 GD On-Demand Anodyne EPHX2 36 41 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(N3CCCCC3=O)c2)C1 ZINC000147128910 GD On-Demand Anodyne AKR1C3 29 42 C[C@H]1[C@@H](C)NC(=O)c2cc3ccc(C(=O)Nc4nc5ccccc5n4CCCN(C)C)nc3n21 ZINC000147128981 JG Annotated Anodyne RPS6KA3 26 65 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccc(OC)cc1)C(C)C ZINC000147128990 EF On-Demand Anodyne KLK3 41 33 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccc(OC)cc1)C(C)C ZINC000147128990 EF On-Demand Anodyne HLA-DRB1 42 36 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccc(OC)cc1)C(C)C ZINC000147128990 EF On-Demand Anodyne PCSK5 53 34 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccc(OC)cc1)C(C)C ZINC000147128990 EF On-Demand Anodyne FURIN 50 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccc(OC)cc1)C(C)C ZINC000147128990 EF On-Demand Anodyne POLG_WNV 52 41 COCc1nc(C(=O)Nc2ccc(OC(F)F)c(Cl)c2)cs1 ZINC000147129040 EH On-Demand Anodyne GRM4 42 46 Nc1ncc(CN2CCC(C(=O)N3CCC(NCc4c(F)cccc4F)CC3)CC2)cn1 ZINC000147129041 IE For-Sale Anodyne SIGMAR1 20 46 COc1ccc2c(c1)OC[C@H](C(=O)N1CCC[C@H](C(=O)Nc3ccc(C)cn3)C1)C2 ZINC000147129084 HF On-Demand Anodyne ROCK2 26 40 COc1ccc2c(c1)OC[C@H](C(=O)N1CCC[C@H](C(=O)Nc3ccc(C)cn3)C1)C2 ZINC000147129084 HF On-Demand Anodyne LUCI_LUCLA 16 41 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(N3CCCCC3=O)c2)C1 ZINC000147129124 GD On-Demand Anodyne EPHX2 36 41 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(N3CCCCC3=O)c2)C1 ZINC000147129124 GD On-Demand Anodyne AKR1C3 29 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccc(OC)cc1)C(C)C ZINC000147129193 EF On-Demand Anodyne KLK3 41 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccc(OC)cc1)C(C)C ZINC000147129193 EF On-Demand Anodyne HLA-DRB1 42 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccc(OC)cc1)C(C)C ZINC000147129193 EF On-Demand Anodyne PCSK5 53 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccc(OC)cc1)C(C)C ZINC000147129193 EF On-Demand Anodyne FURIN 50 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccc(OC)cc1)C(C)C ZINC000147129193 EF On-Demand Anodyne POLG_WNV 52 41 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC[C@@H](C(=O)Nc3ccc(C)cn3)C1)C2 ZINC000147129203 HF On-Demand Anodyne ROCK2 26 40 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC[C@@H](C(=O)Nc3ccc(C)cn3)C1)C2 ZINC000147129203 HF On-Demand Anodyne LUCI_LUCLA 16 41 NC(=O)c1ccc(F)c(NC(=O)c2cccn(Cc3ccccc3)c2=O)c1 ZINC000147129258 FE On-Demand Anodyne HDAC1 25 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccc(OC)cc1)C(C)C ZINC000147129303 EF On-Demand Anodyne KLK3 41 33 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccc(OC)cc1)C(C)C ZINC000147129303 EF On-Demand Anodyne HLA-DRB1 42 36 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccc(OC)cc1)C(C)C ZINC000147129303 EF On-Demand Anodyne PCSK5 53 34 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccc(OC)cc1)C(C)C ZINC000147129303 EF On-Demand Anodyne FURIN 50 35 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccc(OC)cc1)C(C)C ZINC000147129303 EF On-Demand Anodyne POLG_WNV 52 41 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC[C@H](C(=O)Nc3ccc(C)cn3)C1)C2 ZINC000147129310 HF On-Demand Anodyne ROCK2 26 40 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC[C@H](C(=O)Nc3ccc(C)cn3)C1)C2 ZINC000147129310 HF On-Demand Anodyne LUCI_LUCLA 16 41 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(N2CCCCC2=O)c1 ZINC000147129423 HH On-Demand Anodyne NOS2 68 34 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(N2CCCCC2=O)c1 ZINC000147129423 HH On-Demand Anodyne NAMPT 37 42 Nc1ccc([C@@H](O)CC(=O)O)cc1 ZINC000147129436 AC For-Sale Anodyne KYNU 49 31 Nc1ccc([C@@H](O)CC(=O)O)cc1 ZINC000147129436 AC For-Sale Anodyne CPA3 41 33 Nc1ccc([C@@H](O)CC(=O)O)cc1 ZINC000147129436 AC For-Sale Anodyne CPG2 0 40 Nc1ccc([C@@H](O)CC(=O)O)cc1 ZINC000147129436 AC For-Sale Anodyne H9TVJ1_CHISP 0 47 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccc(OC)cc1)C(C)C ZINC000147129503 EF On-Demand Anodyne KLK3 41 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccc(OC)cc1)C(C)C ZINC000147129503 EF On-Demand Anodyne HLA-DRB1 42 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccc(OC)cc1)C(C)C ZINC000147129503 EF On-Demand Anodyne PCSK5 53 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccc(OC)cc1)C(C)C ZINC000147129503 EF On-Demand Anodyne FURIN 50 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccc(OC)cc1)C(C)C ZINC000147129503 EF On-Demand Anodyne POLG_WNV 52 41 Cc1ccc(NC(=O)[C@H]2CCCN(C(=O)c3ccc4c(c3)COC4)C2)nc1 ZINC000147129515 FF On-Demand Anodyne HPGD 41 37 Nc1ccc([C@H](O)CC(=O)O)cc1 ZINC000147129606 AC For-Sale Anodyne KYNU 49 31 Nc1ccc([C@H](O)CC(=O)O)cc1 ZINC000147129606 AC For-Sale Anodyne CPA3 41 33 Nc1ccc([C@H](O)CC(=O)O)cc1 ZINC000147129606 AC For-Sale Anodyne CPG2 0 40 Nc1ccc([C@H](O)CC(=O)O)cc1 ZINC000147129606 AC For-Sale Anodyne H9TVJ1_CHISP 0 47 O=C(Nc1cc(-c2ccccc2)no1)c1ccc2nc3n(c2c1)CCCNC3=O ZINC000147129687 GG Annotated Anodyne RPS6KA3 103 76 O=C(Nc1ccc(NC(=O)c2cnn(-c3ccccc3Cl)c2)cc1)NC1CC1 ZINC000147129707 GI On-Demand Anodyne MAPK10 18 42 O=C(Nc1ccc(NC(=O)c2cnn(-c3ccccc3Cl)c2)cc1)NC1CC1 ZINC000147129707 GI On-Demand Anodyne EPHX2 44 39 O=C(Nc1ccc(NC(=O)c2cnn(-c3ccccc3Cl)c2)cc1)NC1CC1 ZINC000147129707 GI On-Demand Anodyne NR2E3 45 33 NNC(=O)c1cccnc1Nc1ccccc1 ZINC000147129813 BD For-Sale Reactive DHODH 18 41 NNC(=O)c1cccnc1Nc1ccccc1 ZINC000147129813 BD For-Sale Reactive AKR1C2 36 41 O=C(NNC(=O)c1occ(-c2ccccc2)c1-c1ccccc1)c1ccc(O)c(O)c1 ZINC000147129822 HI Annotated Reactive GCGR 68 80 O=C(Nc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1)NC1CC1 ZINC000147129906 FI On-Demand Anodyne EPHX2 46 42 O=C(Nc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1)NC1CC1 ZINC000147129906 FI On-Demand Anodyne NAMPT 23 40 CCOCCO[C@@H](C)C(=O)NCCc1nc2ccccc2[nH]1 ZINC000147129956 DD On-Demand Anodyne CYSP_TRYCR 22 54 CCOCCO[C@@H](C)C(=O)NCCc1nc2ccccc2[nH]1 ZINC000147129956 DD On-Demand Anodyne CACNA1G 30 43 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne OPRM1 22 45 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne OPRD1 26 45 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne MME 35 43 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne ANPEP 46 32 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne NPY1R 31 46 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne KLK3 86 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne CTSK 50 45 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne CTSL 22 43 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne NPFFR2 43 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne C3AR1 58 36 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne MMP2 19 42 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne MMP3 34 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne HLA-DRB1 62 42 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne PCSK5 59 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne FURIN 78 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne GSTP1 15 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne CAPN1 37 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne CAPN2 67 38 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne ACE2 56 39 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne ST14 46 34 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne POLG_WNV 82 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne QRFPR 46 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne NPFFR1 58 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147129969 DF On-Demand Anodyne NOD1 59 35 COCc1nc(C(=O)Nc2cccc(S(=O)(=O)N(C)c3ccccc3)c2)cs1 ZINC000147129976 HG On-Demand Anodyne CACNA1H 15 41 N#CC1CCN(C(=O)C2CCN(C(=O)c3ccc(Br)cc3)CC2)CC1 ZINC000147130006 HG On-Demand Mild PREP 16 47 N#CC1CCN(C(=O)C2CCN(C(=O)c3ccc(Br)cc3)CC2)CC1 ZINC000147130006 HG On-Demand Mild L3MBTL3 91 44 Nc1cc(C(F)(F)F)c(Br)cc1S(N)(=O)=O ZINC000147130085 DD For-Sale Anodyne CAH_METTE 37 73 Nc1cc(C(F)(F)F)c(Br)cc1S(N)(=O)=O ZINC000147130085 DD For-Sale Anodyne CYNT 24 73 Nc1cc(C(F)(F)F)c(Br)cc1S(N)(=O)=O ZINC000147130085 DD For-Sale Anodyne NCE103 19 73 Nc1cc(C(F)(F)F)c(Br)cc1S(N)(=O)=O ZINC000147130085 DD For-Sale Anodyne CA15 21 73 Nc1cc(C(F)(F)F)c(Br)cc1S(N)(=O)=O ZINC000147130085 DD For-Sale Anodyne A6YCJ1_9METZ 25 73 O=C(Nc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1)NC1CC1 ZINC000147130093 FI On-Demand Anodyne EPHX2 46 42 O=C(Nc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1)NC1CC1 ZINC000147130093 FI On-Demand Anodyne NAMPT 23 40 NC(=O)c1ccc(F)c(NC(=O)c2csc(-c3ccccc3F)n2)c1 ZINC000147130121 FG On-Demand Anodyne CHEK1 15 40 CCOCCO[C@H](C)C(=O)NCCc1nc2ccccc2[nH]1 ZINC000147130147 DD On-Demand Anodyne CACNA1G 22 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne MME 35 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne ANPEP 46 32 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne NPY1R 22 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne KLK3 86 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne CTSK 50 45 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne NPFFR2 43 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne C3AR1 58 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne MMP2 19 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne MMP3 34 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne HLA-DRB1 62 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne PCSK5 59 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne FURIN 78 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne GSTP1 15 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne CAPN1 37 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne CAPN2 67 38 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne ACE2 56 39 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne ST14 46 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne POLG_WNV 82 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne QRFPR 46 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne NPFFR1 58 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)C(C)C ZINC000147130151 DF On-Demand Anodyne NOD1 59 35 CCOC[C@H](C)NS(=O)(=O)c1cc(OC)ccc1OC ZINC000147130157 DD On-Demand Anodyne ALPL 17 41 O=C(Nc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1)NC1CC1 ZINC000147130290 FI On-Demand Anodyne EPHX2 46 42 O=C(Nc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1)NC1CC1 ZINC000147130290 FI On-Demand Anodyne NAMPT 23 40 Cc1ccc(-c2nnco2)cc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147130299 FE On-Demand Anodyne CETP 29 40 Cc1ccc(-c2nnco2)cc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147130299 FE On-Demand Anodyne SMO 24 41 OC[C@H]1O[C@@H](n2cnc3c(=S)nc(-c4ccccc4)[nH]c32)[C@H](O)[C@@H]1O ZINC000147130323 FC For-Sale Anodyne ADA 39 40 OC[C@H]1O[C@@H](n2cnc3c(=S)nc(-c4ccccc4)[nH]c32)[C@H](O)[C@@H]1O ZINC000147130323 FC For-Sale Anodyne ADORA1 98 54 OC[C@H]1O[C@@H](n2cnc3c(=S)nc(-c4ccccc4)[nH]c32)[C@H](O)[C@@H]1O ZINC000147130323 FC For-Sale Anodyne SLC29A1 114 46 OC[C@H]1O[C@@H](n2cnc3c(=S)nc(-c4ccccc4)[nH]c32)[C@H](O)[C@@H]1O ZINC000147130323 FC For-Sale Anodyne ADORA2A 44 51 OC[C@H]1O[C@@H](n2cnc3c(=S)nc(-c4ccccc4)[nH]c32)[C@H](O)[C@@H]1O ZINC000147130323 FC For-Sale Anodyne ADK 39 43 OC[C@H]1O[C@@H](n2cnc3c(=S)nc(-c4ccccc4)[nH]c32)[C@H](O)[C@@H]1O ZINC000147130323 FC For-Sale Anodyne CDA 43 34 OC[C@H]1O[C@@H](n2cnc3c(=S)nc(-c4ccccc4)[nH]c32)[C@H](O)[C@@H]1O ZINC000147130323 FC For-Sale Anodyne ADORA3 34 47 OC[C@H]1O[C@@H](n2cnc3c(=S)nc(-c4ccccc4)[nH]c32)[C@H](O)[C@@H]1O ZINC000147130323 FC For-Sale Anodyne FIMH 38 43 OC[C@H]1O[C@@H](n2cnc3c(=S)nc(-c4ccccc4)[nH]c32)[C@H](O)[C@@H]1O ZINC000147130323 FC For-Sale Anodyne DNMT3B 55 34 OC[C@H]1O[C@@H](n2cnc3c(=S)nc(-c4ccccc4)[nH]c32)[C@H](O)[C@@H]1O ZINC000147130323 FC For-Sale Anodyne Q4VQ11_PIG 54 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne OPRM1 22 45 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne OPRD1 26 45 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne MME 35 43 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne ANPEP 46 32 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne NPY1R 31 46 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne KLK3 86 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne CTSK 50 45 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne CTSL 22 43 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne NPFFR2 43 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne C3AR1 58 36 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne MMP2 19 42 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne MMP3 34 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne HLA-DRB1 62 42 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne PCSK5 59 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne FURIN 78 35 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne GSTP1 15 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne CAPN1 37 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne CAPN2 67 38 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne ACE2 56 39 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne ST14 46 34 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne POLG_WNV 82 35 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne QRFPR 46 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne NPFFR1 58 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130333 DF On-Demand Anodyne NOD1 59 35 CC1(C)CNC(=O)c2cc3ccc(C(=O)Nc4cc(C(C)(C)C)on4)nc3n2C1 ZINC000147130344 GG Annotated Anodyne FLT3 46 43 CC1(C)CNC(=O)c2cc3ccc(C(=O)Nc4cc(C(C)(C)C)on4)nc3n2C1 ZINC000147130344 GG Annotated Anodyne RPS6KA3 40 39 CC1(C)CNC(=O)c2cc3ccc(C(=O)Nc4cc(C(C)(C)C)on4)nc3n2C1 ZINC000147130344 GG Annotated Anodyne CSF1R 17 43 O=C(C1CCN(Cc2ccnnc2)CC1)N1CCC(Oc2cccnc2)CC1 ZINC000147130349 GE For-Sale Anodyne HRH3 18 46 O=C(C1CCN(Cc2ccnnc2)CC1)N1CCC(Oc2cccnc2)CC1 ZINC000147130349 GE For-Sale Anodyne CCR3 15 40 O=C(C1CCN(Cc2ccnnc2)CC1)N1CCC(Oc2cccnc2)CC1 ZINC000147130349 GE For-Sale Anodyne SLC18A3 18 43 CCOC(=O)NCC(=O)NCCc1nc2ccccc2[nH]1 ZINC000147130356 CC On-Demand Anodyne F9 27 42 CCOC(=O)NCC(=O)NCCc1nc2ccccc2[nH]1 ZINC000147130356 CC On-Demand Anodyne CYSP_TRYCR 26 63 CCOC(=O)NCC(=O)NCCc1nc2ccccc2[nH]1 ZINC000147130356 CC On-Demand Anodyne CACNA1G 0 44 CCCCCCNC(=O)c1ccc(C(F)(F)F)nc1C ZINC000147130418 CH Annotated Anodyne SHH 28 46 CCCCCCNC(=O)c1ccc(C(F)(F)F)nc1C ZINC000147130418 CH Annotated Anodyne ASAH1 89 38 COc1ccccc1C(=O)N[C@H](C(=O)N1CCC(C#N)CC1)C(C)C ZINC000147130430 EE On-Demand Mild HCN1 42 39 Cc1cc(C(=O)Nc2nc3c(s2)CN(Cc2ccccc2)CC3)cc([N+](=O)[O-])c1 ZINC000147130475 HI On-Demand Bother NOD2 43 36 O=C(Nc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)cc1)NC1CC1 ZINC000147130493 HI On-Demand Anodyne EPHX2 45 42 O=C(Nc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)cc1)NC1CC1 ZINC000147130493 HI On-Demand Anodyne NAMPT 22 40 CN1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)O ZINC000147130506 AD For-Sale Anodyne ACE 30 55 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne MME 35 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne ANPEP 46 32 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne NPY1R 22 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne KLK3 86 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne CTSK 50 45 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne NPFFR2 43 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne C3AR1 58 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne MMP2 19 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne MMP3 34 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne HLA-DRB1 62 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne PCSK5 59 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne FURIN 78 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne GSTP1 15 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne CAPN1 37 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne CAPN2 67 38 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne ACE2 56 39 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne ST14 46 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne POLG_WNV 82 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne QRFPR 46 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne NPFFR1 58 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)C(C)C ZINC000147130520 DF On-Demand Anodyne NOD1 59 35 O=C(Nc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)cc1)NC1CC1 ZINC000147130694 HI On-Demand Anodyne EPHX2 45 42 O=C(Nc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)cc1)NC1CC1 ZINC000147130694 HI On-Demand Anodyne NAMPT 22 40 CS(=O)(=O)c1ccccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147130810 EC On-Demand Anodyne OXTR 15 44 O=C(Nc1ccc(NC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)cc1)NC1CC1 ZINC000147130854 HI On-Demand Anodyne EPHX2 45 42 O=C(Nc1ccc(NC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)cc1)NC1CC1 ZINC000147130854 HI On-Demand Anodyne NAMPT 22 40 CS(=O)(=O)c1ccccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147130992 EC On-Demand Anodyne OXTR 15 44 C=CCCOCC(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1C ZINC000147131010 EH On-Demand Mild MAPK14 25 42 C=CCCOCC(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1C ZINC000147131010 EH On-Demand Mild CPT1A 43 31 C=CCCOCC(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1C ZINC000147131010 EH On-Demand Mild KCNK3 96 38 C=CCCOCC(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1C ZINC000147131010 EH On-Demand Mild KCNK9 50 38 O=C(Nc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)cc1)NC1CC1 ZINC000147131058 HI On-Demand Anodyne EPHX2 45 42 O=C(Nc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)cc1)NC1CC1 ZINC000147131058 HI On-Demand Anodyne NAMPT 22 40 COc1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1N1CCCC1=O ZINC000147131161 HD On-Demand Anodyne CYSLTR1 17 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131184 EE On-Demand Anodyne MAOB 15 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131184 EE On-Demand Anodyne CPT1A 30 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131184 EE On-Demand Anodyne ROCK1 21 44 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131184 EE On-Demand Anodyne ROCK2 15 44 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131184 EE On-Demand Anodyne HDAC9 17 44 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131184 EE On-Demand Anodyne TNK2 49 37 CCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(=O)Cc2ccccc2F)c1 ZINC000147131220 HG On-Demand Anodyne FURIN 42 32 CCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(=O)Cc2ccccc2F)c1 ZINC000147131220 HG On-Demand Anodyne POLG_WNV 42 32 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(NC(=O)NC3CC3)cc1)C2 ZINC000147131243 GG On-Demand Anodyne MTNR1A 24 46 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(NC(=O)NC3CC3)cc1)C2 ZINC000147131243 GG On-Demand Anodyne MTNR1B 25 46 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(NC(=O)NC3CC3)cc1)C2 ZINC000147131243 GG On-Demand Anodyne ROCK2 36 55 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(NC(=O)NC3CC3)cc1)C2 ZINC000147131243 GG On-Demand Anodyne EPHX2 49 39 Nc1ncc(CN2CCC(C(=O)N3CCC(NCc4c(F)cc(F)cc4F)CC3)CC2)cn1 ZINC000147131274 JE For-Sale Anodyne SIGMAR1 18 43 Nc1ncc(CN2CCC(C(=O)N3CCC(NCc4c(F)cc(F)cc4F)CC3)CC2)cn1 ZINC000147131274 JE For-Sale Anodyne SSTR5 40 36 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild CELA1 20 44 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild CASP3 15 51 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild KLK3 62 36 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild CTSB 40 48 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild PAPA1_CARPA 43 34 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild CYSP_TRYCR 36 42 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild CTSK 38 49 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild CTSL 44 48 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild PREP 34 44 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild CAPNS1 61 32 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild TGM1 23 41 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild CTSS 25 42 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild CAPN1 63 43 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild CASP1 21 42 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild CAPN2 92 44 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild TGM2 37 43 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild NPR 54 32 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild F13A1 31 43 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild NAAA 64 50 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild SLC12A5 62 37 O=C[C@H]1CCCC[C@H]1NC(=O)OCc1ccccc1 ZINC000147131328 CF For-Sale Mild Q9NAW4_PLAFA 27 51 COc1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1N1CCCC1=O ZINC000147131368 HD On-Demand Anodyne CYSLTR1 17 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131372 EE On-Demand Anodyne MAOB 15 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131372 EE On-Demand Anodyne CPT1A 30 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131372 EE On-Demand Anodyne ROCK1 21 44 O=C(NC[C@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131372 EE On-Demand Anodyne ROCK2 15 44 O=C(NC[C@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131372 EE On-Demand Anodyne HDAC9 17 44 O=C(NC[C@H]1CCCCO1)C(=O)Nc1nc(-c2ccccc2)cs1 ZINC000147131372 EE On-Demand Anodyne TNK2 49 37 COc1ccccc1NC(=O)CN(c1cc(C)cc(C)c1)S(=O)(=O)c1ccccc1 ZINC000147131378 HI In-Stock Anodyne CA1 16 41 COc1ccccc1NC(=O)CN(c1cc(C)cc(C)c1)S(=O)(=O)c1ccccc1 ZINC000147131378 HI In-Stock Anodyne MMP13 16 44 COc1ccccc1NC(=O)CN(c1cc(C)cc(C)c1)S(=O)(=O)c1ccccc1 ZINC000147131378 HI In-Stock Anodyne MMP9 19 40 COc1ccccc1NC(=O)CN(c1cc(C)cc(C)c1)S(=O)(=O)c1ccccc1 ZINC000147131378 HI In-Stock Anodyne HCRTR2 18 41 COc1ccccc1NC(=O)CN(c1cc(C)cc(C)c1)S(=O)(=O)c1ccccc1 ZINC000147131378 HI In-Stock Anodyne MMP1 18 40 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild CELA1 20 44 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild CASP3 15 51 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild KLK3 62 36 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild CTSB 40 48 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild PAPA1_CARPA 43 34 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild CYSP_TRYCR 36 42 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild CTSK 38 49 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild CTSL 44 48 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild PREP 34 44 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild CAPNS1 61 32 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild TGM1 23 41 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild CTSS 25 42 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild CAPN1 63 43 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild CASP1 21 42 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild CAPN2 92 44 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild TGM2 37 43 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild NPR 54 32 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild F13A1 31 43 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild NAAA 64 50 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild SLC12A5 62 37 O=C[C@H]1CCCC[C@@H]1NC(=O)OCc1ccccc1 ZINC000147131516 CF For-Sale Mild Q9NAW4_PLAFA 27 51 COc1ccc(NC(=O)N2C[C@H](c3ccccc3)O[C@H](C)C2)cc1N1CCCC1=O ZINC000147131615 HH On-Demand Anodyne HTR1D 16 44 CCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(=O)Cc2ccccc2F)c1 ZINC000147131619 HG On-Demand Anodyne FURIN 42 32 CCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(=O)Cc2ccccc2F)c1 ZINC000147131619 HG On-Demand Anodyne POLG_WNV 42 32 CCc1ncc(C(=O)Nc2ccc(OC(F)F)c(Cl)c2)s1 ZINC000147131630 EI On-Demand Anodyne GRM4 48 44 CCc1ncc(C(=O)Nc2ccc(OC(F)F)c(Cl)c2)s1 ZINC000147131630 EI On-Demand Anodyne USP7 42 33 CCc1ncc(C(=O)Nc2ccc(OC(F)F)c(Cl)c2)s1 ZINC000147131630 EI On-Demand Anodyne USP47 53 33 COCc1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147131650 CE On-Demand Mild PREP 25 41 COCc1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147131650 CE On-Demand Mild ST14 57 34 COCc1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147131650 CE On-Demand Mild L3MBTL1 0 43 COCc1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147131650 CE On-Demand Mild L3MBTL3 51 43 CC(C)(C)OC(=O)N1[C@H]2CC[C@@H]([C@H](O)C2)[C@@H]1C(=O)O ZINC000147131696 CD For-Sale Anodyne PREP 16 49 COc1ccc(NC(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)cc1N1CCCC1=O ZINC000147131802 HH On-Demand Anodyne HTR1D 16 44 O=C(C1CCN(Cc2ccnnc2)CC1)N1CCC(NCc2ccc(F)cc2F)CC1 ZINC000147131889 IF For-Sale Anodyne SIGMAR1 27 55 O=C(C1CCN(Cc2ccnnc2)CC1)N1CCC(NCc2ccc(F)cc2F)CC1 ZINC000147131889 IF For-Sale Anodyne SSTR5 43 37 O=C(C1CCN(Cc2ccnnc2)CC1)N1CCC(NCc2ccc(F)cc2F)CC1 ZINC000147131889 IF For-Sale Anodyne CCR3 36 43 O=C(C1CCN(Cc2ccnnc2)CC1)N1CCC(NCc2ccc(F)cc2F)CC1 ZINC000147131889 IF For-Sale Anodyne MLNR 40 38 CCOC[C@H](C)NS(=O)(=O)c1ccc(CC)cc1 ZINC000147131916 CD On-Demand Anodyne MMP7 15 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(CC)cc1 ZINC000147131916 CD On-Demand Anodyne ADAMTS4 47 36 CCc1nc(CN(C)C(=O)N[C@@H](C)c2ccccc2)cs1 ZINC000147131950 DH On-Demand Anodyne CYP3A4 20 41 COc1ccc(NC(=O)N2C[C@@H](C)O[C@H](c3ccccc3)C2)cc1N1CCCC1=O ZINC000147131962 HH On-Demand Anodyne HTR1D 16 44 O=C(NC[C@@H]1CCN(c2ccccc2)C1)c1cccn(Cc2ccccc2)c1=O ZINC000147131978 GG On-Demand Anodyne DRD4 18 44 O=C(NC[C@@H]1CCN(c2ccccc2)C1)c1cccn(Cc2ccccc2)c1=O ZINC000147131978 GG On-Demand Anodyne ACHE 21 46 O=C(NC[C@@H]1CCN(c2ccccc2)C1)c1cccn(Cc2ccccc2)c1=O ZINC000147131978 GG On-Demand Anodyne HTR4 47 41 Cc1cc(C(=O)N2CCC(C#N)CC2)cc(S(=O)(=O)N2CCC(C)CC2)c1C ZINC000147132133 HG On-Demand Mild CNR2 15 44 CC(C)[C@@H]1CCN(C(N)=O)C1 ZINC000147132144 AD On-Demand Anodyne CPN1 0 42 CCc1nc(CN(C)C(=O)N[C@H](C)c2ccccc2)cs1 ZINC000147132146 DH On-Demand Anodyne CYP3A4 20 41 COc1ccc(NC(=O)N2C[C@H](C)O[C@H](c3ccccc3)C2)cc1N1CCCC1=O ZINC000147132157 HH On-Demand Anodyne HTR1D 16 44 CC(C)(C)C(=O)CC(=O)c1ccc2cc(C(=O)CC(=O)C(C)(C)C)ccc2c1 ZINC000147132158 GK For-Sale Anodyne HAO1 50 33 COc1ccc(C(=O)[C@H](O)c2ccccc2)c(F)c1 ZINC000147132168 CF For-Sale Anodyne CES2 58 45 COc1ccc(C(=O)[C@H](O)c2ccccc2)c(F)c1 ZINC000147132168 CF For-Sale Anodyne CES1 28 45 COc1ccc(C(=O)[C@H](O)c2ccccc2)c(F)c1 ZINC000147132168 CF For-Sale Anodyne TUBB2B 19 40 COc1ccc(C(=O)[C@H](O)c2ccccc2)c(F)c1 ZINC000147132168 CF For-Sale Anodyne AKR1C3 25 42 COc1ccc(C(=O)[C@H](O)c2ccccc2)c(F)c1 ZINC000147132168 CF For-Sale Anodyne AKR1C2 55 38 O=C(NC[C@H]1CCN(c2ccccc2)C1)c1cccn(Cc2ccccc2)c1=O ZINC000147132181 GG On-Demand Anodyne DRD4 18 44 O=C(NC[C@H]1CCN(c2ccccc2)C1)c1cccn(Cc2ccccc2)c1=O ZINC000147132181 GG On-Demand Anodyne ACHE 21 46 O=C(NC[C@H]1CCN(c2ccccc2)C1)c1cccn(Cc2ccccc2)c1=O ZINC000147132181 GG On-Demand Anodyne HTR4 47 41 C[C@@]1(c2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)NC(=O)NC1=O ZINC000147132224 HF On-Demand Anodyne KCNK3 50 37 CC(C)[C@H]1CCN(C(N)=O)C1 ZINC000147132333 AD On-Demand Anodyne CPN1 0 42 CN(Cc1cscn1)C(=O)NCc1ccc(Cl)cc1 ZINC000147132347 CG On-Demand Anodyne UL54 63 33 COc1ccc(C(=O)[C@@H](O)c2ccccc2)c(F)c1 ZINC000147132361 CF For-Sale Anodyne CES2 58 45 COc1ccc(C(=O)[C@@H](O)c2ccccc2)c(F)c1 ZINC000147132361 CF For-Sale Anodyne CES1 28 45 COc1ccc(C(=O)[C@@H](O)c2ccccc2)c(F)c1 ZINC000147132361 CF For-Sale Anodyne TUBB2B 19 40 COc1ccc(C(=O)[C@@H](O)c2ccccc2)c(F)c1 ZINC000147132361 CF For-Sale Anodyne AKR1C3 25 42 COc1ccc(C(=O)[C@@H](O)c2ccccc2)c(F)c1 ZINC000147132361 CF For-Sale Anodyne AKR1C2 55 38 C[C@]1(c2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)NC(=O)NC1=O ZINC000147132420 HF On-Demand Anodyne KCNK3 50 37 CCN1CCC(C(=O)NCCN(C)C)CC1 ZINC000147132437 BC On-Demand Anodyne GNAI1 0 46 CCN1CCC(C(=O)NCCN(C)C)CC1 ZINC000147132437 BC On-Demand Anodyne GNAI3 0 46 CCN1CCC(C(=O)NCCN(C)C)CC1 ZINC000147132437 BC On-Demand Anodyne GNAO1 0 46 C/C=C/CN1CCN/C1=C\[N+](=O)[O-] ZINC000147132464 AC For-Sale Bother Q8WSF8_APLCA 16 49 C/C=C/CN1CCN/C1=C\[N+](=O)[O-] ZINC000147132464 AC For-Sale Bother NACHRBETA2 36 49 O=C(C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1)NCC(F)F ZINC000147132612 KJ Annotated Mild PRKAA1 25 54 O=C(C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1)NCC(F)F ZINC000147132612 KJ Annotated Mild FLT4 24 43 O=C(C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1)NCC(F)F ZINC000147132612 KJ Annotated Mild PDGFRA 48 63 O=C(C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1)NCC(F)F ZINC000147132612 KJ Annotated Mild CDK4 0 42 O=C(C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1)NCC(F)F ZINC000147132612 KJ Annotated Mild TGFBR1 57 64 O=C(C#Cc1ccc2c(c1)NC(=O)/C2=C(\Nc1ccc(CN2CCCC2)cc1)c1ccccc1)NCC(F)F ZINC000147132612 KJ Annotated Mild LTK 18 54 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc([C@]3(C)NC(=O)NC3=O)c1)C2 ZINC000147132664 GD On-Demand Anodyne ROCK2 29 47 COC(=O)c1cn(CC(=O)N2CCC(C#N)CC2)c2ccccc12 ZINC000147132747 EE On-Demand Mild CNR2 25 40 COC(=O)c1cn(CC(=O)N2CCC(C#N)CC2)c2ccccc12 ZINC000147132747 EE On-Demand Mild CCR8 50 34 O=C(O)[C@@H](CCO)NS(=O)(=O)c1cccc2cccnc12 ZINC000147132775 DC On-Demand Anodyne PDE4C 47 34 O=C(O)[C@@H](CCO)NS(=O)(=O)c1cccc2cccnc12 ZINC000147132775 DC On-Demand Anodyne ITGAV 54 40 Cc1cc(-c2n[nH]c(C)c2Cl)ccn1 ZINC000147132815 BF For-Sale Anodyne XDH 32 48 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)c(OC)c3)cs2)s1 ZINC000147132837 GI On-Demand Anodyne MPL 44 41 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)c(OC)c3)cs2)s1 ZINC000147132837 GI On-Demand Anodyne SYK 20 40 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)c(OC)c3)cs2)s1 ZINC000147132837 GI On-Demand Anodyne ROCK2 20 41 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)c(OC)c3)cs2)s1 ZINC000147132837 GI On-Demand Anodyne STK17B 44 44 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)c(OC)c3)cs2)s1 ZINC000147132837 GI On-Demand Anodyne STK17A 16 44 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)c(OC)c3)cs2)s1 ZINC000147132837 GI On-Demand Anodyne ENPP1 49 31 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc([C@@]3(C)NC(=O)NC3=O)c1)C2 ZINC000147132849 GD On-Demand Anodyne ROCK2 29 47 O=C(O)CC[C@H](C(=O)O)[C@@H](CC(=O)O)P(=O)(O)O ZINC000147132907 CB For-Sale Anodyne FOLH1 60 48 O=C(O)CC[C@H](C(=O)O)[C@@H](CC(=O)O)P(=O)(O)O ZINC000147132907 CB For-Sale Anodyne NAALAD2 45 48 O=C(O)[C@H](CCO)NS(=O)(=O)c1cccc2cccnc12 ZINC000147132938 DC On-Demand Anodyne PDE4C 47 34 O=C(O)[C@H](CCO)NS(=O)(=O)c1cccc2cccnc12 ZINC000147132938 DC On-Demand Anodyne ITGAV 54 40 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1ccc2oc(C3CC3)nc2c1 ZINC000147132954 HK On-Demand Anodyne ROCK2 15 40 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1ccc2oc(C3CC3)nc2c1 ZINC000147132954 HK On-Demand Anodyne MET 25 40 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1ccc2oc(C3CC3)nc2c1 ZINC000147132954 HK On-Demand Anodyne NAMPT 50 41 O=C(Nc1nc2cc(Cl)ccc2[nH]1)c1ccc2cc3n(c2n1)CCCNC3=O ZINC000147133027 GF Annotated Anodyne RPS6KA3 82 44 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc([C@]3(C)NC(=O)NC3=O)c1)C2 ZINC000147133037 GD On-Demand Anodyne ROCK2 29 47 O=C(O)CC[C@@H](C(=O)O)[C@@H](CC(=O)O)P(=O)(O)O ZINC000147133067 CB For-Sale Anodyne FOLH1 60 48 O=C(O)CC[C@@H](C(=O)O)[C@@H](CC(=O)O)P(=O)(O)O ZINC000147133067 CB For-Sale Anodyne NAALAD2 45 48 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](c1ccccc1)c1ccco1 ZINC000147133071 EJ On-Demand Anodyne MME 74 38 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](c1ccccc1)c1ccco1 ZINC000147133071 EJ On-Demand Anodyne ANPEP 45 33 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](c1ccccc1)c1ccco1 ZINC000147133071 EJ On-Demand Anodyne CTSB 31 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](c1ccccc1)c1ccco1 ZINC000147133071 EJ On-Demand Anodyne PAPA1_CARPA 29 42 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](c1ccccc1)c1ccco1 ZINC000147133071 EJ On-Demand Anodyne CTSL 19 42 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](c1ccccc1)c1ccco1 ZINC000147133071 EJ On-Demand Anodyne CTSS 15 42 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](c1ccccc1)c1ccco1 ZINC000147133071 EJ On-Demand Anodyne ACE2 70 38 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](c1ccccc1)c1ccco1 ZINC000147133071 EJ On-Demand Anodyne FPR1 42 35 O=C(O)CC[C@H](C(=O)O)[C@H](CC(=O)O)P(=O)(O)O ZINC000147133196 CB For-Sale Anodyne FOLH1 60 48 O=C(O)CC[C@H](C(=O)O)[C@H](CC(=O)O)P(=O)(O)O ZINC000147133196 CB For-Sale Anodyne NAALAD2 45 48 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133277 EJ On-Demand Anodyne MME 74 38 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133277 EJ On-Demand Anodyne ANPEP 45 33 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133277 EJ On-Demand Anodyne CTSB 31 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133277 EJ On-Demand Anodyne PAPA1_CARPA 29 42 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133277 EJ On-Demand Anodyne CTSL 19 42 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133277 EJ On-Demand Anodyne CTSS 15 42 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133277 EJ On-Demand Anodyne ACE2 70 38 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133277 EJ On-Demand Anodyne FPR1 42 35 O=C(O)CC[C@@H](C(=O)O)[C@H](CC(=O)O)P(=O)(O)O ZINC000147133328 CB For-Sale Anodyne FOLH1 60 48 O=C(O)CC[C@@H](C(=O)O)[C@H](CC(=O)O)P(=O)(O)O ZINC000147133328 CB For-Sale Anodyne NAALAD2 45 48 CC(C)OCC(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147133403 CG On-Demand Anodyne KCNA3 23 42 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc2oc(C3CC3)nc2c1 ZINC000147133439 GJ On-Demand Anodyne PRMT3 48 35 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133442 EJ On-Demand Anodyne MME 74 38 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133442 EJ On-Demand Anodyne ANPEP 45 33 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133442 EJ On-Demand Anodyne CTSB 31 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133442 EJ On-Demand Anodyne PAPA1_CARPA 29 42 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133442 EJ On-Demand Anodyne CTSL 19 42 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133442 EJ On-Demand Anodyne CTSS 15 42 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133442 EJ On-Demand Anodyne ACE2 70 38 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147133442 EJ On-Demand Anodyne FPR1 42 35 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2cccs2)c1 ZINC000147133444 FG On-Demand Anodyne HDAC10 41 36 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2cccs2)c1 ZINC000147133444 FG On-Demand Anodyne KCNK3 43 49 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2cccs2)c1 ZINC000147133444 FG On-Demand Anodyne KCNK9 53 50 CCOC[C@H](C)NS(=O)(=O)c1cccc([N+](=O)[O-])c1C ZINC000147133543 DD On-Demand Bother COLA 70 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2cccs2)c1 ZINC000147133598 FG On-Demand Anodyne HDAC10 41 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2cccs2)c1 ZINC000147133598 FG On-Demand Anodyne KCNK3 43 49 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2cccs2)c1 ZINC000147133598 FG On-Demand Anodyne KCNK9 53 50 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc2oc(C3CC3)nc2c1 ZINC000147133628 GJ On-Demand Anodyne PRMT3 48 35 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc2oc(C3CC3)nc2c1 ZINC000147133807 GJ On-Demand Anodyne PRMT3 48 35 O=[N+]([O-])c1ccccc1CNc1cccc2cc[nH]c12 ZINC000147133869 CH On-Demand Bother COLA 67 38 O=[N+]([O-])c1ccccc1CNc1cccc2cc[nH]c12 ZINC000147133869 CH On-Demand Bother PRKCQ 17 42 CC1(C)OC(c2ccc3ncnn3c2)=C(c2cccc(Cl)c2)C1=O ZINC000147133931 EH For-Sale Anodyne TGFBR1 80 39 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc2oc(C3CC3)nc2c1 ZINC000147133935 GJ On-Demand Anodyne PRMT3 48 35 c1ccc(Cc2cccc3c2ccc2ccccc23)cc1 ZINC000147133969 CK Annotated Bother ALOX5 16 43 CCCS(=O)(=O)Nc1ccccc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147133982 HG On-Demand Anodyne CYP19A1 15 45 CCCS(=O)(=O)Nc1ccccc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147133982 HG On-Demand Anodyne CYP11B1 44 42 CCCS(=O)(=O)Nc1ccccc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147133982 HG On-Demand Anodyne TBXAS1 41 42 CCCS(=O)(=O)Nc1ccccc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147133982 HG On-Demand Anodyne AGTR2 19 42 CCCS(=O)(=O)Nc1ccccc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147133982 HG On-Demand Anodyne CYP11B2 38 42 CCCS(=O)(=O)Nc1ccccc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147133982 HG On-Demand Anodyne CYP17A1 18 44 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)c1cccc([N+](=O)[O-])c1 ZINC000147134153 EI On-Demand Bother CACNA1C 52 37 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)c1cccc([N+](=O)[O-])c1 ZINC000147134153 EI On-Demand Bother CACNA1D 82 35 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)c1cccc([N+](=O)[O-])c1 ZINC000147134153 EI On-Demand Bother MDM2 85 35 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3cc(F)ccc3F)CC2)CC1 ZINC000147134247 GE On-Demand Mild EPHX2 28 42 CCc1ncc(C(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2OC)s1 ZINC000147134377 HD On-Demand Anodyne MERTK 30 40 CCc1ncc(C(=O)Nc2cc(S(=O)(=O)N3CCOCC3)ccc2OC)s1 ZINC000147134377 HD On-Demand Anodyne NAMPT 17 41 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)c1cccc([N+](=O)[O-])c1 ZINC000147134440 EI On-Demand Bother CACNA1C 52 37 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)c1cccc([N+](=O)[O-])c1 ZINC000147134440 EI On-Demand Bother CACNA1D 82 35 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)c1cccc([N+](=O)[O-])c1 ZINC000147134440 EI On-Demand Bother MDM2 85 35 COc1cccc(Oc2ccc(CNC(=O)c3cc(OC)ccc3[N+](=O)[O-])cn2)c1 ZINC000147134494 HH On-Demand Bother TAAR1 22 41 CCOC[C@H](C)NS(=O)(=O)c1ccc(OC)c(NC(C)=O)c1 ZINC000147134574 ED On-Demand Anodyne MMP12 41 36 CC(C)Oc1ccc(S(C)(=O)=O)cc1C(=O)N1Cc2ccc(Cl)cc2C1 ZINC000147134695 GH On-Demand Anodyne SLC6A9 57 67 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Br)c1)c1cccc([N+](=O)[O-])c1 ZINC000147134715 GI On-Demand Bother CACNA1C 53 37 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Br)c1)c1cccc([N+](=O)[O-])c1 ZINC000147134715 GI On-Demand Bother CACNA1D 83 35 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne CHRM2 15 45 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne CHRM1 15 50 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne DRD2 15 42 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne DRD4 44 61 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne ACHE 26 43 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne HRH2 48 36 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne KCNH2 35 45 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne CHRM3 22 50 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne LTA4H 28 44 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne SIGMAR1 35 48 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne SSTR5 80 44 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne CHEK2 37 42 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne CCR3 50 46 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne UTS2R 18 43 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne FAAH 36 43 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne CCR2 20 41 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne SLC6A5 37 47 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne MCHR1 66 55 Cc1cccc(CN2CCC(NC(=O)COc3ccc(C(N)=O)cc3)CC2)c1 ZINC000147134766 GE On-Demand Anodyne CCR8 28 51 COc1ccc(CNCc2ccc(NC(C)=O)cc2)cc1OCCCC#N ZINC000147134848 FH On-Demand Mild TSHR 66 32 COc1ccc(CNCc2ccc(NC(C)=O)cc2)cc1OCCCC#N ZINC000147134848 FH On-Demand Mild MT-ND1 16 40 COc1ccc(CNCc2ccc(NC(C)=O)cc2)cc1OCCCC#N ZINC000147134848 FH On-Demand Mild DRTS_TRYCR 52 39 CC(C)c1cc(NC(=O)c2ccc3cc4n(c3n2)CC(C)(C)CNC4=O)no1 ZINC000147134868 GG Annotated Anodyne RPS6KA3 51 43 CCCC[C@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147134872 EE On-Demand Anodyne MTNR1A 34 40 CCCC[C@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147134872 EE On-Demand Anodyne GRIA1 42 31 CCCC[C@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147134872 EE On-Demand Anodyne PCSK5 51 34 CCCC[C@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147134872 EE On-Demand Anodyne FURIN 48 32 CCCC[C@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147134872 EE On-Demand Anodyne POLG_WNV 65 31 CCCC[C@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147134872 EE On-Demand Anodyne HPN 51 32 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Br)c1)c1cccc([N+](=O)[O-])c1 ZINC000147134971 GI On-Demand Bother CACNA1C 53 37 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Br)c1)c1cccc([N+](=O)[O-])c1 ZINC000147134971 GI On-Demand Bother CACNA1D 83 35 CCCC[C@@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147135004 EE On-Demand Anodyne MTNR1A 34 40 CCCC[C@@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147135004 EE On-Demand Anodyne GRIA1 42 31 CCCC[C@@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147135004 EE On-Demand Anodyne PCSK5 51 34 CCCC[C@@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147135004 EE On-Demand Anodyne FURIN 48 32 CCCC[C@@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147135004 EE On-Demand Anodyne POLG_WNV 65 31 CCCC[C@@H](NC(N)=O)C(=O)NCCc1cccc2cccnc12 ZINC000147135004 EE On-Demand Anodyne HPN 51 32 CCN(CC)c1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cn1 ZINC000147135052 EE On-Demand Anodyne ADORA2B 42 45 CCN(CC)c1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cn1 ZINC000147135052 EE On-Demand Anodyne HIF1A 24 42 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)NC3=NCCC3)c2)cc([N+](=O)[O-])c1 ZINC000147135060 HF On-Demand Bother KCNK3 66 37 Cc1cc(C(=O)Nc2cccc(S(=O)(=O)NC3=NCCC3)c2)cc([N+](=O)[O-])c1 ZINC000147135060 HF On-Demand Bother KCNK9 42 37 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne DRD4 24 43 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne P2RY12 77 34 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne CHRM3 25 40 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne NPR1 40 31 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne NPFFR2 42 31 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne HDAC8 17 40 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne HDAC10 38 40 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne HDAC2 23 40 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne HDAC6 28 40 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne HDAC11 55 40 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne POLG_WNV 40 30 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135224 GD On-Demand Anodyne BIRC2 47 36 COc1ccc2c(c1)OC[C@H](C(=O)N[C@H](C)c1cccc([N+](=O)[O-])c1)C2 ZINC000147135269 FG On-Demand Bother ROCK2 24 40 Cc1cc(NC(=O)c2ccc3cc4n(c3n2)[C@@H](C)[C@H](C)NC4=O)no1 ZINC000147135278 EE Annotated Anodyne RPS6KA3 24 44 Cc1ccc(NS(C)(=O)=O)c(C(=O)NCc2ccc(Cn3ccnc3)cc2)c1 ZINC000147135322 GF On-Demand Anodyne CYP11B1 33 48 Cc1ccc(NS(C)(=O)=O)c(C(=O)NCc2ccc(Cn3ccnc3)cc2)c1 ZINC000147135322 GF On-Demand Anodyne TBXAS1 42 48 Cc1ccc(NS(C)(=O)=O)c(C(=O)NCc2ccc(Cn3ccnc3)cc2)c1 ZINC000147135322 GF On-Demand Anodyne TRPV1 36 43 Cc1ccc(NS(C)(=O)=O)c(C(=O)NCc2ccc(Cn3ccnc3)cc2)c1 ZINC000147135322 GF On-Demand Anodyne CYP11B2 15 48 Cc1ccc(NS(C)(=O)=O)c(C(=O)NCc2ccc(Cn3ccnc3)cc2)c1 ZINC000147135322 GF On-Demand Anodyne CYP17A1 16 47 Oc1c(Cl)ccc2c1CCNCC2 ZINC000147135348 AD For-Sale Anodyne PNMT 46 53 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne DRD4 24 43 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne P2RY12 77 34 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne CHRM3 25 40 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne NPR1 40 31 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne NPFFR2 42 31 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne HDAC8 17 40 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne HDAC10 38 40 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne HDAC2 23 40 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne HDAC6 28 40 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne HDAC11 55 40 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne POLG_WNV 40 30 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147135369 GD On-Demand Anodyne BIRC2 47 36 CCOC(=O)CCC/C=C\CC(C(=O)OCC)C(=O)OCC ZINC000147135416 DE For-Sale Anodyne LPAR3 29 41 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H](C)c1cccc([N+](=O)[O-])c1)C2 ZINC000147135430 FG On-Demand Bother ROCK2 24 40 CCCCOc1ccc(Br)nc1C(=O)OC ZINC000147135504 CF In-Stock Anodyne PLA2G4B 44 33 CS(=O)(=O)Nc1ccc(F)cc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147135510 HE On-Demand Anodyne CYP19A1 15 47 CS(=O)(=O)Nc1ccc(F)cc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147135510 HE On-Demand Anodyne CYP11B1 36 47 CS(=O)(=O)Nc1ccc(F)cc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147135510 HE On-Demand Anodyne TBXAS1 37 40 CS(=O)(=O)Nc1ccc(F)cc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147135510 HE On-Demand Anodyne TRPV1 77 39 CS(=O)(=O)Nc1ccc(F)cc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147135510 HE On-Demand Anodyne CYP11B2 30 47 CS(=O)(=O)Nc1ccc(F)cc1C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147135510 HE On-Demand Anodyne CYP17A1 18 46 CC1(C)CNC(=O)c2cc3ccc(C(=O)Nc4cc(C5CC5)on4)nc3n2C1 ZINC000147135555 GF Annotated Anodyne RPS6KA3 44 40 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H](C)c1cccc([N+](=O)[O-])c1)C2 ZINC000147135625 FG On-Demand Bother ROCK2 24 40 CC(=O)N1CCN(c2ccc(C(=O)N3CCC(C#N)CC3)cc2[N+](=O)[O-])CC1 ZINC000147135676 GD On-Demand Mild SLC6A9 25 41 CC(=O)N1CCN(c2ccc(C(=O)N3CCC(C#N)CC3)cc2[N+](=O)[O-])CC1 ZINC000147135676 GD On-Demand Mild L3MBTL3 47 46 CNC(=O)c1csc(NC(=O)c2ccc3cc4n(c3n2)[C@@H](C)CNC4=O)n1 ZINC000147135953 GD Annotated Anodyne MAPKAPK2 29 58 CNC(=O)c1csc(NC(=O)c2ccc3cc4n(c3n2)[C@@H](C)CNC4=O)n1 ZINC000147135953 GD Annotated Anodyne MAP2K1 15 41 CNC(=O)c1csc(NC(=O)c2ccc3cc4n(c3n2)[C@@H](C)CNC4=O)n1 ZINC000147135953 GD Annotated Anodyne RPS6KA3 19 43 N#CC1CCN(C(=O)C2CCN(C(=O)c3ccc(F)cc3F)CC2)CC1 ZINC000147135967 FF On-Demand Mild L3MBTL3 41 35 CCOc1ccccc1OCC(=O)NNC(=O)c1csc(COC)n1 ZINC000147135974 FD On-Demand Reactive HCN1 48 32 CCOc1ccccc1OCC(=O)NNC(=O)c1csc(COC)n1 ZINC000147135974 FD On-Demand Reactive HCN4 40 31 CCc1ncc(C(=O)Nc2cc(S(=O)(=O)N3CCCCC3)ccc2OC)s1 ZINC000147136114 HG On-Demand Anodyne NAMPT 25 43 CNC(=O)c1csc(NC(=O)c2ccc3cc4n(c3n2)[C@H](C)CNC4=O)n1 ZINC000147136131 GD Annotated Anodyne MAPKAPK2 29 58 CNC(=O)c1csc(NC(=O)c2ccc3cc4n(c3n2)[C@H](C)CNC4=O)n1 ZINC000147136131 GD Annotated Anodyne MAP2K1 15 41 CNC(=O)c1csc(NC(=O)c2ccc3cc4n(c3n2)[C@H](C)CNC4=O)n1 ZINC000147136131 GD Annotated Anodyne RPS6KA3 19 43 CC(C)(C)OC(=O)CCNC(=O)NCc1ccccc1 ZINC000147136175 CE On-Demand Anodyne ANPEP 29 41 CC(C)(C)OC(=O)CCNC(=O)NCc1ccccc1 ZINC000147136175 CE On-Demand Anodyne FPR1 41 36 CC(C)(C)OC(=O)CCNC(=O)NCc1ccccc1 ZINC000147136175 CE On-Demand Anodyne POL 0 44 CC(C)(C)OC(=O)CCNC(=O)NCc1ccccc1 ZINC000147136175 CE On-Demand Anodyne AMP1_PLAFQ 41 36 CC(C)(C)OC(=O)CCNC(=O)NCc1ccccc1 ZINC000147136175 CE On-Demand Anodyne PDS 43 37 CCN(CC)CC(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147136242 CD On-Demand Anodyne MTNR1A 23 44 CCN(CC)CC(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147136242 CD On-Demand Anodyne KCNK3 42 38 N#CC1CCN(C(=O)CCCNC(=O)c2ccc(F)cc2F)CC1 ZINC000147136316 EE On-Demand Mild PREP 27 40 C[C@@H]1CNC(=O)c2cc3ccc(C(=O)Nc4nccs4)nc3n21 ZINC000147136347 EE Annotated Anodyne MAP1 115 36 C[C@@H]1CNC(=O)c2cc3ccc(C(=O)Nc4nccs4)nc3n21 ZINC000147136347 EE Annotated Anodyne MAPKAPK2 33 55 C[C@@H]1CNC(=O)c2cc3ccc(C(=O)Nc4nccs4)nc3n21 ZINC000147136347 EE Annotated Anodyne RPS6KA3 25 45 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)cc3)cs2)s1 ZINC000147136386 EI On-Demand Anodyne MPL 48 38 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)cc3)cs2)s1 ZINC000147136386 EI On-Demand Anodyne ROCK1 23 44 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)cc3)cs2)s1 ZINC000147136386 EI On-Demand Anodyne ROCK2 19 41 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)cc3)cs2)s1 ZINC000147136386 EI On-Demand Anodyne HDAC9 15 40 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)cc3)cs2)s1 ZINC000147136386 EI On-Demand Anodyne TBK1 40 37 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild ACE 55 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild OPRD1 16 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild GHRHR 55 35 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild P2RY12 53 35 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CELA1 32 47 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild GRIN2B 26 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild ELANE 37 46 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild MME 26 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CTRA_BOVIN 54 31 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CASP3 18 44 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild BMP1 54 34 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild KLK3 72 37 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CTSB 68 52 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild PAPA1_CARPA 65 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CYSP_TRYCR 62 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CCKAR 0 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CTSG 43 34 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CTSK 42 54 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CTSL 46 47 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild DPP4 27 52 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild PREP 31 68 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CAPNS1 74 38 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CELA2A 58 34 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild LGMN 80 37 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CTSS 38 47 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CAPN1 85 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild CAPN2 113 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild PLAU 16 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild TGM2 36 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild PROTEASE 0 44 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild TPSAB1 24 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild POL 0 42 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild NPR 60 36 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild AMP1_PLAFQ 19 40 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild DPP8 26 45 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild RHODESAIN 0 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild PSMB5 45 38 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild BIRC2 34 43 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild Q6PRC7_IXORI 47 36 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild MCA2 0 41 C[C@H](NC(=O)OCc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147136527 DE On-Demand Mild SLC12A5 53 34 COC(=O)c1cc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2o1 ZINC000147136535 FE On-Demand Anodyne ADORA2B 41 42 COC(=O)c1cc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2o1 ZINC000147136535 FE On-Demand Anodyne CETP 42 45 COC(=O)c1cc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2o1 ZINC000147136535 FE On-Demand Anodyne ACR 59 38 COC(=O)c1cc2cc(NC(=O)COc3ccc(C(N)=O)cc3)ccc2o1 ZINC000147136535 FE On-Demand Anodyne HIF1A 22 44 C[C@H]1CNC(=O)c2cc3ccc(C(=O)Nc4nccs4)nc3n21 ZINC000147136563 EE Annotated Anodyne MAP1 115 36 C[C@H]1CNC(=O)c2cc3ccc(C(=O)Nc4nccs4)nc3n21 ZINC000147136563 EE Annotated Anodyne MAPKAPK2 33 55 C[C@H]1CNC(=O)c2cc3ccc(C(=O)Nc4nccs4)nc3n21 ZINC000147136563 EE Annotated Anodyne RPS6KA3 25 45 COCc1nc(C(=O)Nc2nc(-c3ccc(OC)cc3)cs2)cs1 ZINC000147136566 FH On-Demand Anodyne MPL 30 40 COCc1nc(C(=O)Nc2nc(-c3ccc(OC)cc3)cs2)cs1 ZINC000147136566 FH On-Demand Anodyne ROCK1 22 42 COCc1nc(C(=O)Nc2nc(-c3ccc(OC)cc3)cs2)cs1 ZINC000147136566 FH On-Demand Anodyne ROCK2 18 42 COCc1nc(C(=O)Nc2nc(-c3ccc(OC)cc3)cs2)cs1 ZINC000147136566 FH On-Demand Anodyne HDAC9 15 41 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1nc2c(s1)CCC2 ZINC000147136642 DH On-Demand Anodyne SLC27A1 40 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147136667 EC On-Demand Anodyne MTOR 48 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147136667 EC On-Demand Anodyne TNK2 33 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147136667 EC On-Demand Anodyne DGAT1 53 48 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147136667 EC On-Demand Anodyne HPGDS 20 44 N#CC1CCN(C(=O)c2ccc(-n3cnnn3)cc2)CC1 ZINC000147136743 CD On-Demand Mild L3MBTL3 63 41 N#CC1CCN(C(=O)c2ccc(-n3cnnn3)cc2)CC1 ZINC000147136743 CD On-Demand Mild KCNJ1 50 43 CCc1ncc(C(=O)Nc2nc(-c3ccc(F)cc3)cs2)s1 ZINC000147136779 EI On-Demand Anodyne MAOB 18 44 CCc1ncc(C(=O)Nc2nc(-c3ccc(F)cc3)cs2)s1 ZINC000147136779 EI On-Demand Anodyne MPL 73 40 CCc1ncc(C(=O)Nc2nc(-c3ccc(F)cc3)cs2)s1 ZINC000147136779 EI On-Demand Anodyne MAPK14 17 43 CCc1ncc(C(=O)Nc2nc(-c3ccc(F)cc3)cs2)s1 ZINC000147136779 EI On-Demand Anodyne ROCK1 21 47 CCc1ncc(C(=O)Nc2nc(-c3ccc(F)cc3)cs2)s1 ZINC000147136779 EI On-Demand Anodyne ROCK2 15 47 N#Cc1cccc(Oc2ccc(C=O)cc2C(F)(F)F)c1 ZINC000147136816 CI For-Sale Mild ESRRA 18 42 C[C@H](Cc1cccc(F)c1)C(=O)Nc1nc2c(s1)CCC2 ZINC000147136831 DH On-Demand Anodyne SLC27A1 40 43 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147136858 EC On-Demand Anodyne MTOR 48 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147136858 EC On-Demand Anodyne TNK2 33 43 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147136858 EC On-Demand Anodyne DGAT1 53 48 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147136858 EC On-Demand Anodyne HPGDS 20 44 COC(=O)c1cc2cc(NC(=O)c3cccn(Cc4ccccc4)c3=O)ccc2o1 ZINC000147136944 HH On-Demand Anodyne KCNK3 45 34 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)NCc1ccccc1 ZINC000147136994 GF On-Demand Mild GRIN2B 46 38 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)NCc1ccccc1 ZINC000147136994 GF On-Demand Mild FASN 21 40 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)NCc1ccccc1 ZINC000147136994 GF On-Demand Mild CCR8 54 39 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)NCc1ccccc1 ZINC000147136994 GF On-Demand Mild SFRP1 47 37 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)NCc1ccccc1 ZINC000147136994 GF On-Demand Mild L3MBTL3 50 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2)nc1 ZINC000147137070 ED On-Demand Anodyne TNK2 34 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2)nc1 ZINC000147137070 ED On-Demand Anodyne DGAT1 46 45 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2)nc1 ZINC000147137070 ED On-Demand Anodyne HPGDS 15 41 CC(C)CC(C)(C)C[C@H]1N(C)[C@@H](C(=O)NCC[C@H](O)CO)[C@H](c2cccc(Cl)c2)[C@@]12C(=O)Nc1cc(Cl)c(F)cc12 ZINC000147137113 KK Annotated Anodyne MDM2 70 67 COC(=O)c1cc2cc(NC(=O)COC(C)C)ccc2o1 ZINC000147137140 CF On-Demand Anodyne CETP 40 48 Cn1nc(CC(=O)N2CCC(C#N)CC2)c2ccccc2c1=O ZINC000147137188 DD On-Demand Mild IMDH_CRYPV 31 52 CCCC[C@H](NC(N)=O)C(=O)Nc1cnc2ccccc2c1 ZINC000147137201 DE On-Demand Anodyne BDKRB2 20 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cnc2ccccc2c1 ZINC000147137201 DE On-Demand Anodyne CCKAR 17 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cnc2ccccc2c1 ZINC000147137201 DE On-Demand Anodyne CTSK 27 40 CCN(CC)CC(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147137225 EF On-Demand Anodyne PDE4A 20 41 CCN(CC)CC(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147137225 EF On-Demand Anodyne FLT1 21 48 CCN(CC)CC(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147137225 EF On-Demand Anodyne QPCT 15 41 CCN(CC)CC(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147137225 EF On-Demand Anodyne ENPP1 70 42 CCN(CC)CC(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147137225 EF On-Demand Anodyne DRTS_TRYCR 40 38 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2)nc1 ZINC000147137258 ED On-Demand Anodyne TNK2 34 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2)nc1 ZINC000147137258 ED On-Demand Anodyne DGAT1 46 45 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2)nc1 ZINC000147137258 ED On-Demand Anodyne HPGDS 15 41 CC1(C)CC(=O)C2=C(C1)NC1=C(C(=O)CC(C)(C)C1)C2c1cc(Br)c(O)c(Br)c1 ZINC000147137312 KK In-Stock Mild TGFBR2 37 43 CCOC[C@H](C)NS(=O)(=O)c1ccc(N2CCCC2=O)cc1 ZINC000147137405 ED On-Demand Anodyne AKR1C3 25 46 N#CC1CCN(C(=O)c2ccc(C3SCCCS3)cc2)CC1 ZINC000147137409 EH On-Demand Mild L3MBTL3 89 43 CS(=O)(=O)C[C@H](O)COc1ccccc1 ZINC000147137451 BC On-Demand Anodyne ADRB2 42 55 CS(=O)(=O)C[C@H](O)COc1ccccc1 ZINC000147137451 BC On-Demand Anodyne GRIN1 58 42 CS(=O)(=O)C[C@H](O)COc1ccccc1 ZINC000147137451 BC On-Demand Anodyne ADRB3 43 43 CS(=O)(=O)C[C@H](O)COc1ccccc1 ZINC000147137451 BC On-Demand Anodyne ABCB1 40 47 CS(=O)(=O)C[C@H](O)COc1ccccc1 ZINC000147137451 BC On-Demand Anodyne PDS 48 38 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147137525 EE On-Demand Anodyne KCNQ2 74 37 Cc1cccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137565 GI On-Demand Anodyne PRCP 43 38 Cc1cccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137565 GI On-Demand Anodyne GRM5 23 40 Cc1cccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137565 GI On-Demand Anodyne SORT1 15 40 Cc1cccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137565 GI On-Demand Anodyne NPBWR1 42 31 CS(=O)(=O)C[C@@H](O)COc1ccccc1 ZINC000147137630 BC On-Demand Anodyne ADRB2 42 55 CS(=O)(=O)C[C@@H](O)COc1ccccc1 ZINC000147137630 BC On-Demand Anodyne GRIN1 37 41 CS(=O)(=O)C[C@@H](O)COc1ccccc1 ZINC000147137630 BC On-Demand Anodyne ADRB3 43 43 CS(=O)(=O)C[C@@H](O)COc1ccccc1 ZINC000147137630 BC On-Demand Anodyne ABCB1 28 47 CS(=O)(=O)C[C@@H](O)COc1ccccc1 ZINC000147137630 BC On-Demand Anodyne PDS 48 38 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147137703 EE On-Demand Anodyne KCNQ2 74 37 Cc1cccc(NC(=O)C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137736 GI On-Demand Anodyne PRCP 43 38 Cc1cccc(NC(=O)C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137736 GI On-Demand Anodyne GRM5 23 40 Cc1cccc(NC(=O)C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137736 GI On-Demand Anodyne SORT1 15 40 Cc1cccc(NC(=O)C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137736 GI On-Demand Anodyne NPBWR1 42 31 O=C(CCl)NNC(=O)c1cc(Cl)cc(Cl)c1 ZINC000147137823 CD For-Sale Reactive CACNA1I 63 39 C[C@@H](CCc1ccccc1)NC(=O)N(C)Cc1cscn1 ZINC000147137837 DG On-Demand Anodyne BMP1 68 42 C[C@@H](CCc1ccccc1)NC(=O)N(C)Cc1cscn1 ZINC000147137837 DG On-Demand Anodyne ACACA 21 42 C[C@@H](CCc1ccccc1)NC(=O)N(C)Cc1cscn1 ZINC000147137837 DG On-Demand Anodyne CYP3A4 27 55 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cnc2ccccc2c1 ZINC000147137842 DD On-Demand Anodyne SMO 41 34 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147137904 EE On-Demand Anodyne KCNQ2 74 37 Cc1cccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137908 GI On-Demand Anodyne PRCP 43 38 Cc1cccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137908 GI On-Demand Anodyne GRM5 23 40 Cc1cccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137908 GI On-Demand Anodyne SORT1 15 40 Cc1cccc(NC(=O)C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147137908 GI On-Demand Anodyne NPBWR1 42 31 CC(C)[C@@H](CS(=O)(=O)C(C)C)N1C(=O)[C@](C)(CC(=O)O)C[C@@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147137996 KK For-Sale Anodyne TP53 45 73 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cnc2ccccc2c1 ZINC000147138017 DD On-Demand Anodyne SMO 41 34 C[C@H](CCc1ccccc1)NC(=O)N(C)Cc1cscn1 ZINC000147138033 DG On-Demand Anodyne BMP1 18 40 C[C@H](CCc1ccccc1)NC(=O)N(C)Cc1cscn1 ZINC000147138033 DG On-Demand Anodyne CYP3A4 27 55 Cc1cc(C(=O)Nc2nc3c(s2)CCCC3)cc([N+](=O)[O-])c1 ZINC000147138051 DG On-Demand Bother SLC27A1 24 43 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1ccccc1N1CCCC1=O ZINC000147138091 EE On-Demand Anodyne KCNQ2 74 37 CC(C)(C)OC(=O)N1CCC2(CC1)CCN(C(=O)c1cccnc1)CC2 ZINC000147138237 FG On-Demand Anodyne CCR8 42 42 CC(C)(C)OC(=O)N1CCC2(CC1)CCN(C(=O)c1cccnc1)CC2 ZINC000147138237 FG On-Demand Anodyne GPR119 32 43 C[C@H]1CCCCN1Cc1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147138372 FI On-Demand Anodyne HRH3 30 41 C[C@H]1CCCCN1Cc1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147138372 FI On-Demand Anodyne NOD2 44 37 CC(C)[C@@H](CS(=O)(=O)C(C)C)N1C(=O)[C@](C)(CC(=O)O)C[C@@H](c2cccc(Cl)c2)[C@@H]1c1ccc(Cl)cc1 ZINC000147138385 KK For-Sale Anodyne TP53 45 73 Cc1cccc(C)c1OC[C@H](O)CNC(=O)Nc1cccc(OC[C@@H]2CCCO2)c1 ZINC000147138398 HG On-Demand Anodyne ADRB2 17 45 Cc1cccc(C)c1OC[C@H](O)CNC(=O)Nc1cccc(OC[C@@H]2CCCO2)c1 ZINC000147138398 HG On-Demand Anodyne ADRB1 50 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne CA2 17 48 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne CA1 21 41 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne MMP13 56 45 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne CA4 16 48 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne CA14 18 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne MMP2 45 45 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne MMP3 22 45 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne MMP8 21 45 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne MMP14 19 45 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne MMP9 19 45 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne CA12 15 40 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne MMP7 17 45 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne ADAMTS4 41 44 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne CA9 15 44 CCOC[C@H](C)NS(=O)(=O)c1ccc(-c2ccc(NC(C)=O)cc2)cc1 ZINC000147138534 GG On-Demand Anodyne IDO1 36 45 COC(=O)c1cc(NC(=O)c2ccccc2OCCN(C)C)ccc1Cl ZINC000147138547 GG On-Demand Anodyne DHODH 15 40 COC(=O)c1cc(NC(=O)c2ccccc2OCCN(C)C)ccc1Cl ZINC000147138547 GG On-Demand Anodyne KDR 15 50 COC(=O)c1cc(NC(=O)c2ccccc2OCCN(C)C)ccc1Cl ZINC000147138547 GG On-Demand Anodyne GRM4 43 43 COC(=O)c1cc(NC(=O)c2ccccc2OCCN(C)C)ccc1Cl ZINC000147138547 GG On-Demand Anodyne NR2E3 53 34 COC(=O)c1cc(NC(=O)c2ccccc2OCCN(C)C)ccc1Cl ZINC000147138547 GG On-Demand Anodyne SHH 35 43 COC(=O)c1cc(NC(=O)c2ccccc2OCCN(C)C)ccc1Cl ZINC000147138547 GG On-Demand Anodyne KCNK3 65 48 COC(=O)c1cc(NC(=O)c2ccccc2OCCN(C)C)ccc1Cl ZINC000147138547 GG On-Demand Anodyne KCNK9 63 48 CS(=O)(=O)Nc1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147138579 GC On-Demand Anodyne ADRB2 16 42 CS(=O)(=O)Nc1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147138579 GC On-Demand Anodyne ADRB1 15 42 CS(=O)(=O)Nc1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147138579 GC On-Demand Anodyne GRIN1 39 41 CS(=O)(=O)Nc1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147138579 GC On-Demand Anodyne CA1 15 41 CS(=O)(=O)Nc1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147138579 GC On-Demand Anodyne TRPV1 39 52 CS(=O)(=O)Nc1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147138579 GC On-Demand Anodyne PTPRB 42 34 CS(=O)(=O)Nc1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147138579 GC On-Demand Anodyne CA9 23 41 Cc1cccc(C)c1OC[C@@H](O)CNC(=O)Nc1cccc(OC[C@@H]2CCCO2)c1 ZINC000147138616 HG On-Demand Anodyne ADRB2 17 45 Cc1cccc(C)c1OC[C@@H](O)CNC(=O)Nc1cccc(OC[C@@H]2CCCO2)c1 ZINC000147138616 HG On-Demand Anodyne ADRB1 50 42 CC1=CC(C)(C)Nc2ccc(OCc3ccccc3)nc21 ZINC000147138650 CI For-Sale Anodyne NR3C1 19 42 CC1=CC(C)(C)Nc2ccc(OCc3ccccc3)nc21 ZINC000147138650 CI For-Sale Anodyne PGR 18 40 CC1=CC(C)(C)Nc2ccc(OCc3ccccc3)nc21 ZINC000147138650 CI For-Sale Anodyne PGA 48 40 CC(=O)CCc1ccc(OCCc2ccc(C#N)cc2)cc1 ZINC000147138720 CH On-Demand Mild PPARG 15 41 CC(=O)CCc1ccc(OCCc2ccc(C#N)cc2)cc1 ZINC000147138720 CH On-Demand Mild PLA2G4B 47 39 CC(=O)CCc1ccc(OCCc2ccc(C#N)cc2)cc1 ZINC000147138720 CH On-Demand Mild FFAR1 65 47 CC(=O)CCc1ccc(OCCc2ccc(C#N)cc2)cc1 ZINC000147138720 CH On-Demand Mild PPO2 33 40 CC(=O)CCc1ccc(OCCc2ccc(C#N)cc2)cc1 ZINC000147138720 CH On-Demand Mild FFAR4 49 35 C[C@H](CC(=O)N1CCC(C#N)CC1)NC(=O)c1ccccc1 ZINC000147138729 CD On-Demand Mild CCR1 34 43 C[C@H](CC(=O)N1CCC(C#N)CC1)NC(=O)c1ccccc1 ZINC000147138729 CD On-Demand Mild DPP4 22 42 C[C@H](CC(=O)N1CCC(C#N)CC1)NC(=O)c1ccccc1 ZINC000147138729 CD On-Demand Mild FAP 0 46 CCC[C@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138800 EC On-Demand Anodyne TRPV1 39 49 CCC[C@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138800 EC On-Demand Anodyne NPY1R 21 40 CCC[C@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138800 EC On-Demand Anodyne CA14 15 43 CCC[C@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138800 EC On-Demand Anodyne PCSK5 45 36 CCC[C@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138800 EC On-Demand Anodyne FURIN 61 36 CCC[C@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138800 EC On-Demand Anodyne F7 19 43 CCC[C@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138800 EC On-Demand Anodyne PROC 44 34 Cc1cccc(C)c1OC[C@H](O)CNC(=O)Nc1cccc(OC[C@H]2CCCO2)c1 ZINC000147138818 HG On-Demand Anodyne ADRB2 17 45 Cc1cccc(C)c1OC[C@H](O)CNC(=O)Nc1cccc(OC[C@H]2CCCO2)c1 ZINC000147138818 HG On-Demand Anodyne ADRB1 50 42 O=c1cc(-c2ccccc2)oc2cc(O[C@@H]3O[C@H]([C@H](O)CO)[C@H](O)[C@H]3O)c(O)c(O)c12 ZINC000147138829 IC Annotated Clean AKR1B1 0 46 O=c1cc(-c2ccccc2)oc2cc(O[C@@H]3O[C@H]([C@H](O)CO)[C@H](O)[C@H]3O)c(O)c(O)c12 ZINC000147138829 IC Annotated Clean CYP1B1 24 42 O=c1cc(-c2ccccc2)oc2cc(O[C@@H]3O[C@H]([C@H](O)CO)[C@H](O)[C@H]3O)c(O)c(O)c12 ZINC000147138829 IC Annotated Clean CYP1A1 28 42 O=c1cc(-c2ccccc2)oc2cc(O[C@@H]3O[C@H]([C@H](O)CO)[C@H](O)[C@H]3O)c(O)c(O)c12 ZINC000147138829 IC Annotated Clean CYP1A2 15 42 O=[N+]([O-])c1ccc(OCc2ccccc2)c(C(F)(F)F)c1 ZINC000147138830 CI On-Demand Bother CYP19A1 18 53 O=[N+]([O-])c1ccc(OCc2ccccc2)c(C(F)(F)F)c1 ZINC000147138830 CI On-Demand Bother XDH 16 44 O=[N+]([O-])c1ccc(OCc2ccccc2)c(C(F)(F)F)c1 ZINC000147138830 CI On-Demand Bother PPIA 33 44 O=[N+]([O-])c1ccc(OCc2ccccc2)c(C(F)(F)F)c1 ZINC000147138830 CI On-Demand Bother PTGER1 48 40 O=[N+]([O-])c1ccc(OCc2ccccc2)c(C(F)(F)F)c1 ZINC000147138830 CI On-Demand Bother ACR 25 43 O=[N+]([O-])c1ccc(OCc2ccccc2)c(C(F)(F)F)c1 ZINC000147138830 CI On-Demand Bother F2RL3 48 40 CN(Cc1cscn1)C(=O)NCc1cccc(Cl)c1 ZINC000147138854 CG On-Demand Anodyne BMP1 54 39 CC(=O)N[C@@H](CC(=O)N1CCC(C#N)CC1)c1ccc(Cl)cc1 ZINC000147138919 EF On-Demand Mild PTAFR 21 46 CC(=O)N[C@@H](CC(=O)N1CCC(C#N)CC1)c1ccc(Cl)cc1 ZINC000147138919 EF On-Demand Mild CCR1 41 37 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)NC)cc1 ZINC000147138934 DC On-Demand Anodyne CA2 18 47 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)NC)cc1 ZINC000147138934 DC On-Demand Anodyne MMP7 18 42 CCOC[C@H](C)NS(=O)(=O)c1ccc(C(=O)NC)cc1 ZINC000147138934 DC On-Demand Anodyne ADAMTS4 44 35 CCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138998 EC On-Demand Anodyne TRPV1 39 49 CCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138998 EC On-Demand Anodyne NPY1R 21 40 CCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138998 EC On-Demand Anodyne CA14 15 43 CCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138998 EC On-Demand Anodyne PCSK5 45 36 CCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138998 EC On-Demand Anodyne FURIN 61 36 CCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138998 EC On-Demand Anodyne F7 19 43 CCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NS(C)(=O)=O)cc1 ZINC000147138998 EC On-Demand Anodyne PROC 44 34 Cc1cccc(C)c1OC[C@@H](O)CNC(=O)Nc1cccc(OC[C@H]2CCCO2)c1 ZINC000147139017 HG On-Demand Anodyne ADRB2 17 45 Cc1cccc(C)c1OC[C@@H](O)CNC(=O)Nc1cccc(OC[C@H]2CCCO2)c1 ZINC000147139017 HG On-Demand Anodyne ADRB1 50 42 Cc1c(Cl)cccc1NC(=O)CN1CCC(c2ccccn2)CC1 ZINC000147139031 EH On-Demand Anodyne DRD4 32 75 Cc1c(Cl)cccc1NC(=O)CN1CCC(c2ccccn2)CC1 ZINC000147139031 EH On-Demand Anodyne MCHR1 18 40 CC(=O)N[C@H](CC(=O)N1CCC(C#N)CC1)c1ccc(Cl)cc1 ZINC000147139101 EF On-Demand Mild PTAFR 21 46 CC(=O)N[C@H](CC(=O)N1CCC(C#N)CC1)c1ccc(Cl)cc1 ZINC000147139101 EF On-Demand Mild CCR1 41 37 CCCC[C@H](NC(N)=O)C(=O)Nc1cc(C(N)=O)ccc1N1CCCCC1 ZINC000147139538 GD On-Demand Anodyne KCNQ2 78 42 CC(C)N(C)S(=O)(=O)c1ccc(CNS(=O)(=O)c2cccnc2)cc1 ZINC000147139545 GD On-Demand Anodyne TBXA2R 21 40 CC(C)N(C)S(=O)(=O)c1ccc(CNS(=O)(=O)c2cccnc2)cc1 ZINC000147139545 GD On-Demand Anodyne TBXAS1 42 40 CC(C)N(C)S(=O)(=O)c1ccc(CNS(=O)(=O)c2cccnc2)cc1 ZINC000147139545 GD On-Demand Anodyne NAMPT 58 48 CN(Cc1cscn1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147139661 FD On-Demand Anodyne CA2 78 51 CN(Cc1cscn1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147139661 FD On-Demand Anodyne CA1 61 51 CN(Cc1cscn1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147139661 FD On-Demand Anodyne CA7 46 50 CN(Cc1cscn1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147139661 FD On-Demand Anodyne CA5B 37 46 CN(Cc1cscn1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147139661 FD On-Demand Anodyne CA4 55 48 CN(Cc1cscn1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147139661 FD On-Demand Anodyne CA5A 36 46 CN(Cc1cscn1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147139661 FD On-Demand Anodyne CA12 45 45 CN(Cc1cscn1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147139661 FD On-Demand Anodyne CA9 51 44 CN(Cc1cscn1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147139661 FD On-Demand Anodyne NCE103 26 41 CN(Cc1cscn1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147139661 FD On-Demand Anodyne LIG1 0 40 CN(Cc1cscn1)C(=O)NCCc1ccc(S(N)(=O)=O)cc1 ZINC000147139661 FD On-Demand Anodyne A6YCJ1_9METZ 24 47 CC[C@@H](C)Oc1cccc2cccnc12 ZINC000147139691 BG In-Stock Anodyne CCR1 0 42 CC[C@@H](C)Oc1cccc2cccnc12 ZINC000147139691 BG In-Stock Anodyne MCHR1 23 64 CC[C@@H](C)Oc1cccc2cccnc12 ZINC000147139691 BG In-Stock Anodyne METAP2 0 42 COCc1nc(C(=O)N2CCN(c3ccc(OC)cc3)CC2)cs1 ZINC000147139703 EE On-Demand Clean CCKAR 40 44 COCc1nc(C(=O)N2CCN(c3ccc(OC)cc3)CC2)cs1 ZINC000147139703 EE On-Demand Clean NPBWR1 49 30 COCc1nc(C(=O)N2CCN(c3ccc(OC)cc3)CC2)cs1 ZINC000147139703 EE On-Demand Clean TRPC6 53 46 COCc1nc(C(=O)N2CCN(c3ccc(OC)cc3)CC2)cs1 ZINC000147139703 EE On-Demand Clean TRPC3 24 46 CCCC[C@@H](NC(N)=O)C(=O)Nc1cc(C(N)=O)ccc1N1CCCCC1 ZINC000147139724 GD On-Demand Anodyne KCNQ2 78 42 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(OC[C@@H]2CCCO2)c1 ZINC000147139747 HH On-Demand Anodyne CCR3 27 41 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(OC[C@@H]2CCCO2)c1 ZINC000147139747 HH On-Demand Anodyne NOS2 96 36 CCOP(=O)(CCOc1ccc(Cl)cc1)OCC ZINC000147139752 CH For-Sale Anodyne FDPS 20 45 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(COc3ccc(CC#N)cc3)c2)c1 ZINC000147139886 HJ On-Demand Mild MAOB 23 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(COc3ccc(CC#N)cc3)c2)c1 ZINC000147139886 HJ On-Demand Mild TAAR1 34 45 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(COc3ccc(CC#N)cc3)c2)c1 ZINC000147139886 HJ On-Demand Mild KCNK3 41 35 CC[C@H](C)Oc1cccc2cccnc12 ZINC000147139888 BG In-Stock Anodyne CCR1 0 42 CC[C@H](C)Oc1cccc2cccnc12 ZINC000147139888 BG In-Stock Anodyne MCHR1 23 64 CC[C@H](C)Oc1cccc2cccnc12 ZINC000147139888 BG In-Stock Anodyne METAP2 0 42 CCC[C@H](NC(N)=O)C(=O)NCc1ccc(-n2cncn2)cc1 ZINC000147139907 DC On-Demand Anodyne FURIN 51 34 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(OC[C@H]2CCCO2)c1 ZINC000147139936 HH On-Demand Anodyne CCR3 27 41 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1cccc(OC[C@H]2CCCO2)c1 ZINC000147139936 HH On-Demand Anodyne NOS2 96 36 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc5c(c4)CC[C@@H](N4CCOCC4)CC5)nc23)cc1 ZINC000147139942 KI Annotated Anodyne JAK3 19 74 CS(=O)(=O)c1ccc(-c2cccn3nc(Nc4ccc5c(c4)CC[C@@H](N4CCOCC4)CC5)nc23)cc1 ZINC000147139942 KI Annotated Anodyne JAK2 34 74 CN1CCN(NC(=O)Nc2ccc(N)cc2)CC1 ZINC000147139945 BC For-Sale Clean EPHX2 32 43 CN1CCN(NC(=O)Nc2ccc(N)cc2)CC1 ZINC000147139945 BC For-Sale Clean P96878_MYCTU 48 37 Cc1ccc(S(=O)(=O)N2CC[C@@H](C)[C@H]2CO)cc1 ZINC000147139971 CD On-Demand Anodyne MMP13 41 42 Cc1ccc(S(=O)(=O)N2CC[C@@H](C)[C@H]2CO)cc1 ZINC000147139971 CD On-Demand Anodyne ADAM17 47 46 Cc1ccc(S(=O)(=O)N2CC[C@@H](C)[C@H]2CO)cc1 ZINC000147139971 CD On-Demand Anodyne MMP7 55 36 Cc1ccc(S(=O)(=O)N2CC[C@@H](C)[C@H]2CO)cc1 ZINC000147139971 CD On-Demand Anodyne MMP1 42 42 CCC[C@@H](NC(N)=O)C(=O)NCc1ccc(-n2cncn2)cc1 ZINC000147140091 DC On-Demand Anodyne FURIN 51 34 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147140100 HG On-Demand Anodyne COLA 78 40 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147140100 HG On-Demand Anodyne CPT1A 73 40 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147140100 HG On-Demand Anodyne CPT2 51 40 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147140100 HG On-Demand Anodyne CPT1B 79 39 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCCCC3)c2)s1 ZINC000147140100 HG On-Demand Anodyne ENPP1 61 32 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(OC[C@@H]2CCCO2)c1 ZINC000147140182 HJ On-Demand Anodyne EPHX2 21 40 Cc1cc(CNC(=O)N[C@H](Cc2ccc(O)cc2)c2nc3ccccc3[nH]2)no1 ZINC000147140186 GG On-Demand Anodyne F11 42 37 Cc1cc(CNC(=O)N[C@H](Cc2ccc(O)cc2)c2nc3ccccc3[nH]2)no1 ZINC000147140186 GG On-Demand Anodyne PTPN1 43 50 COCCOc1cccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147140253 HD On-Demand Bother CACNA1D 62 36 COCCOc1cccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147140253 HD On-Demand Bother ROCK2 24 42 COCCOc1cccc(CNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147140253 HD On-Demand Bother PDS 37 41 CC(=O)N[C@H](CC(=O)N1CCC(C#N)CC1)c1ccc(C)cc1 ZINC000147140288 DE On-Demand Mild PTAFR 27 48 CCNC(=O)c1ccc(C)c(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147140297 FD On-Demand Anodyne MAPK14 39 48 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000147140312 DF On-Demand Anodyne TRHR 58 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000147140312 DF On-Demand Anodyne HLA-DRB3 41 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000147140312 DF On-Demand Anodyne TRY1_BOVIN 73 38 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000147140312 DF On-Demand Anodyne NTSR1 65 31 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000147140312 DF On-Demand Anodyne ADAM17 38 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000147140312 DF On-Demand Anodyne C5AR1 20 42 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(OC[C@@H]2CCCO2)c1 ZINC000147140372 HJ On-Demand Anodyne EPHX2 21 40 CN(C)CCOc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147140465 ED On-Demand Anodyne TNK2 35 43 CC(=O)N[C@@H](CC(=O)N1CCC(C#N)CC1)c1ccc(C)cc1 ZINC000147140492 DE On-Demand Mild PTAFR 27 48 COCCOc1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147140496 FF On-Demand Anodyne MMP13 24 41 COCCOc1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147140496 FF On-Demand Anodyne ROCK2 27 42 COCCOc1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147140496 FF On-Demand Anodyne CARM1 40 37 COCCOc1cccc(CNC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147140496 FF On-Demand Anodyne PDS 40 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000147140501 DF On-Demand Anodyne TRHR 58 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000147140501 DF On-Demand Anodyne HLA-DRB3 41 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000147140501 DF On-Demand Anodyne TRY1_BOVIN 73 38 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(F)cc1 ZINC000147140501 DF On-Demand Anodyne NTSR1 65 31 Cc1cc(C(=O)Nc2ccc3nc(C)sc3c2)cc([N+](=O)[O-])c1 ZINC000147140564 EI On-Demand Bother LCK 25 40 Cc1cc(C(=O)Nc2ccc3nc(C)sc3c2)cc([N+](=O)[O-])c1 ZINC000147140564 EI On-Demand Bother LDHA 31 41 Cc1cc(C(=O)Nc2ccc3nc(C)sc3c2)cc([N+](=O)[O-])c1 ZINC000147140564 EI On-Demand Bother KCNK3 57 38 Cc1cc(C(=O)Nc2ccc3nc(C)sc3c2)cc([N+](=O)[O-])c1 ZINC000147140564 EI On-Demand Bother KCNK9 42 38 CN(C)CCOc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147140644 ED On-Demand Anodyne TNK2 35 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(F)cc1 ZINC000147140670 DF On-Demand Anodyne TRHR 58 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(F)cc1 ZINC000147140670 DF On-Demand Anodyne HLA-DRB3 41 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(F)cc1 ZINC000147140670 DF On-Demand Anodyne TRY1_BOVIN 73 38 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(F)cc1 ZINC000147140670 DF On-Demand Anodyne NTSR1 65 31 CC(C)N(C)S(=O)(=O)c1ccc(CNS(=O)(=O)N2CCCC[C@@H]2C)cc1 ZINC000147140712 HD On-Demand Anodyne AKR1C3 18 40 COCc1nc(C(=O)Nc2nc(-c3ccc(C)c(C)c3)cs2)cs1 ZINC000147140771 FI On-Demand Anodyne MPL 33 51 COCc1nc(C(=O)Nc2nc(-c3ccc(C)c(C)c3)cs2)cs1 ZINC000147140771 FI On-Demand Anodyne HDAC9 15 43 COCc1nc(C(=O)Nc2nc(-c3ccc(C)c(C)c3)cs2)cs1 ZINC000147140771 FI On-Demand Anodyne TRPA1 15 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(F)cc1 ZINC000147140855 DF On-Demand Anodyne TRHR 58 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(F)cc1 ZINC000147140855 DF On-Demand Anodyne HLA-DRB3 41 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(F)cc1 ZINC000147140855 DF On-Demand Anodyne TRY1_BOVIN 73 38 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(F)cc1 ZINC000147140855 DF On-Demand Anodyne NTSR1 65 31 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(N3CCCC3)c1)C2 ZINC000147140878 FG On-Demand Anodyne DRD4 40 30 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(N3CCCC3)c1)C2 ZINC000147140878 FG On-Demand Anodyne MTNR1A 27 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(N3CCCC3)c1)C2 ZINC000147140878 FG On-Demand Anodyne MTNR1B 30 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(N3CCCC3)c1)C2 ZINC000147140878 FG On-Demand Anodyne ROCK2 31 49 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(N3CCCC3)c1)C2 ZINC000147140878 FG On-Demand Anodyne TAAR1 40 42 Cc1cc(CNC(=O)NCC(=O)Nc2ccc(Cl)cc2)no1 ZINC000147140970 DE On-Demand Anodyne PPIA 18 42 COc1ccc(CNC[C@@H]2Cc3ccccc3O2)cc1OCCCC#N ZINC000147141034 FG On-Demand Mild ADRA1B 16 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(N3CCCC3)c1)C2 ZINC000147141068 FG On-Demand Anodyne DRD4 40 30 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(N3CCCC3)c1)C2 ZINC000147141068 FG On-Demand Anodyne MTNR1A 27 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(N3CCCC3)c1)C2 ZINC000147141068 FG On-Demand Anodyne MTNR1B 30 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(N3CCCC3)c1)C2 ZINC000147141068 FG On-Demand Anodyne ROCK2 31 49 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(N3CCCC3)c1)C2 ZINC000147141068 FG On-Demand Anodyne TAAR1 40 42 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild FABP2 0 46 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild FABP4 17 46 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild FAAH 0 45 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild CES2 22 40 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild CES1 17 40 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild EST1_PIG 23 40 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild JHE 0 40 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild FABP3 24 42 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild FABP5 16 46 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild SLC22A20 0 48 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild Q9GPG0_MANSE 0 40 CCCCC/C(C)=C/C(C)=O ZINC000147141113 AG For-Sale Mild CQSS 65 40 O=C(NCC(F)(F)F)Nc1cccc(-c2cnc3cc(-c4cncnc4)ccn23)c1 ZINC000147141140 HI Annotated Anodyne BRAF 34 41 COCc1nc(C(=O)Nc2nc(-c3ccc4ccccc4c3)cs2)cs1 ZINC000147141217 GJ On-Demand Anodyne MPL 45 40 COCc1nc(C(=O)Nc2nc(-c3ccc4ccccc4c3)cs2)cs1 ZINC000147141217 GJ On-Demand Anodyne ROCK1 22 42 COCc1nc(C(=O)Nc2nc(-c3ccc4ccccc4c3)cs2)cs1 ZINC000147141217 GJ On-Demand Anodyne ROCK2 17 42 COc1ccc(CNCc2cccc(C(=O)N(C)C)c2)cc1OCCCC#N ZINC000147141268 GG On-Demand Mild REN 29 41 COc1cc(-c2n[nH]c3ccc(N)cc23)ccn1 ZINC000147141278 BE For-Sale Anodyne TTK 30 43 O=C(Nc1cccc(N2CCCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147141283 FI On-Demand Anodyne KCNQ2 48 35 O=C(Nc1cccc(N2CCCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147141283 FI On-Demand Anodyne PRNP 62 36 O=C(Nc1cccc(N2CCCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147141283 FI On-Demand Anodyne MAPK10 23 45 O=C(Nc1cccc(N2CCCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147141283 FI On-Demand Anodyne EPHB3 40 42 O=C(Nc1cccc(N2CCCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147141283 FI On-Demand Anodyne TAAR1 39 43 O=C(Nc1cccc(N2CCCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147141283 FI On-Demand Anodyne KCNK3 69 41 CCCCC/C(C)=C\C(C)=O ZINC000147141294 AG For-Sale Mild FABP4 17 46 CCCCC/C(C)=C\C(C)=O ZINC000147141294 AG For-Sale Mild FAAH 0 45 CCCCC/C(C)=C\C(C)=O ZINC000147141294 AG For-Sale Mild CES2 22 40 CCCCC/C(C)=C\C(C)=O ZINC000147141294 AG For-Sale Mild CES1 17 40 CCCCC/C(C)=C\C(C)=O ZINC000147141294 AG For-Sale Mild EST1_PIG 23 40 CCCCC/C(C)=C\C(C)=O ZINC000147141294 AG For-Sale Mild FABP3 24 42 CCCCC/C(C)=C\C(C)=O ZINC000147141294 AG For-Sale Mild FABP5 16 46 CCCCC/C(C)=C\C(C)=O ZINC000147141294 AG For-Sale Mild CQSS 65 40 CC(C)(C)OC(=O)N1CCC(CNc2ccc(C#N)cc2)CC1 ZINC000147141297 DH For-Sale Mild GRIN2B 20 44 CC(C)(C)OC(=O)N1CCC(CNc2ccc(C#N)cc2)CC1 ZINC000147141297 DH For-Sale Mild CETP 0 54 CC(C)(C)OC(=O)N1CCC(CNc2ccc(C#N)cc2)CC1 ZINC000147141297 DH For-Sale Mild CACNA1I 45 34 CC(C)(C)OC(=O)N1CCC(CNc2ccc(C#N)cc2)CC1 ZINC000147141297 DH For-Sale Mild F13A1 18 40 CC(C)(C)OC(=O)N1CCC(CNc2ccc(C#N)cc2)CC1 ZINC000147141297 DH For-Sale Mild GPR119 59 49 CCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccccc1OC(C)C ZINC000147141304 DE On-Demand Anodyne CAPN2 66 41 Cc1cc(CNC(=O)NCc2ccc(F)cc2Br)no1 ZINC000147141615 EF On-Demand Anodyne P2RX7 62 43 CCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccccc1OC(C)C ZINC000147141671 DE On-Demand Anodyne CAPN2 66 41 CN(Cc1cscn1)C(=O)NCc1ccc(Cl)cc1Cl ZINC000147141722 EH On-Demand Anodyne P2RX7 53 45 COc1ccc(OC)c(CCNC(=O)NCc2cc(C)on2)c1 ZINC000147141816 DE On-Demand Anodyne MTNR1A 75 44 COc1ccc(OC)c(CCNC(=O)NCc2cc(C)on2)c1 ZINC000147141816 DE On-Demand Anodyne MTNR1B 56 40 COc1ccc(OC)c(CCNC(=O)NCc2cc(C)on2)c1 ZINC000147141816 DE On-Demand Anodyne MT-ND1 15 40 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne CA2 32 46 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne INHA 18 40 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne CA1 54 37 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne CA7 25 45 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne SCN2A 21 40 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne S1PR4 15 43 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne CA4 15 43 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne CA14 15 45 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne S1PR5 18 43 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne CA12 34 46 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne CA9 35 46 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne NCE103 34 46 CCCCO[C@@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142002 DD On-Demand Anodyne P96878_MYCTU 37 46 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne CA2 32 46 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne INHA 18 40 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne CA1 54 37 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne CA7 25 45 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne SCN2A 21 40 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne S1PR4 15 43 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne CA4 15 43 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne CA14 15 45 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne S1PR5 18 43 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne CA12 34 46 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne CA9 35 46 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne NCE103 34 46 CCCCO[C@H](C)C(=O)Nc1ccc(CS(N)(=O)=O)cc1 ZINC000147142198 DD On-Demand Anodyne P96878_MYCTU 37 46 Cc1cccc(N2CCOCC2)c1[N+](=O)[O-] ZINC000147142281 BD On-Demand Bother PRKDC 43 36 CCOCCCCNC(=O)CCCc1ccc2c(c1)-c1ccccc1C2 ZINC000147142337 FJ On-Demand Anodyne CRTM 41 39 CCOCCCCNC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147142542 CG On-Demand Anodyne SLC6A1 28 46 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)NCc3cccs3)c2)CC1 ZINC000147142646 GF On-Demand Mild ST14 58 32 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCOCC3)c2)s1 ZINC000147142712 HD On-Demand Anodyne CPT1A 67 42 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCOCC3)c2)s1 ZINC000147142712 HD On-Demand Anodyne CPT2 50 38 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCOCC3)c2)s1 ZINC000147142712 HD On-Demand Anodyne NR1H4 22 46 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCOCC3)c2)s1 ZINC000147142712 HD On-Demand Anodyne CPT1B 72 38 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCOCC3)c2)s1 ZINC000147142712 HD On-Demand Anodyne AXL 16 43 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCOCC3)c2)s1 ZINC000147142712 HD On-Demand Anodyne TYRO3 19 40 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCOCC3)c2)s1 ZINC000147142712 HD On-Demand Anodyne MERTK 39 43 CCc1ncc(C(=O)Nc2ccc(OC)c(S(=O)(=O)N3CCOCC3)c2)s1 ZINC000147142712 HD On-Demand Anodyne ENPP1 63 33 CCOCCCCNC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147142736 CG On-Demand Anodyne SLC6A1 28 46 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147142830 HF On-Demand Anodyne CNR2 20 44 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147142830 HF On-Demand Anodyne MAPK11 36 41 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147142830 HF On-Demand Anodyne MAPK14 46 41 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147142830 HF On-Demand Anodyne MAPK13 42 38 CCOCCCCNC(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147142913 CG On-Demand Anodyne SLC6A1 28 46 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147143021 HF On-Demand Anodyne CNR2 20 44 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147143021 HF On-Demand Anodyne MAPK11 36 41 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147143021 HF On-Demand Anodyne MAPK14 46 41 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147143021 HF On-Demand Anodyne MAPK13 42 38 CCOCCCCNC(=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147143105 CG On-Demand Anodyne SLC6A1 28 46 Cc1nn(-c2ccc(C(=O)N3CCC(C#N)CC3)cc2)c(C)c1Cl ZINC000147143110 EH On-Demand Mild L3MBTL3 57 37 CCc1ncc(C(=O)Nc2nnc(SCc3ccc(F)cc3)s2)s1 ZINC000147143112 GI On-Demand Anodyne ABL1 18 60 CN(Cc1cscn1)C(=O)NCCc1ccc(Cl)cc1Cl ZINC000147143180 EH On-Demand Anodyne AKT3 15 44 Cc1cccn2cc(-c3ccc(NC(=O)C(=O)NC[C@@H]4CCCCO4)cc3)nc12 ZINC000147143223 GF On-Demand Anodyne MTOR 46 33 O=c1ncccn1[C@H]1C[C@@H](O)[C@@H](CO)O1 ZINC000147143280 BA For-Sale Anodyne ADA 45 44 O=c1ncccn1[C@H]1C[C@@H](O)[C@@H](CO)O1 ZINC000147143280 BA For-Sale Anodyne TK 44 49 O=c1ncccn1[C@H]1C[C@@H](O)[C@@H](CO)O1 ZINC000147143280 BA For-Sale Anodyne TK1 51 49 O=c1ncccn1[C@H]1C[C@@H](O)[C@@H](CO)O1 ZINC000147143280 BA For-Sale Anodyne POLB 46 39 O=c1ncccn1[C@H]1C[C@@H](O)[C@@H](CO)O1 ZINC000147143280 BA For-Sale Anodyne CDA 69 39 O=c1ncccn1[C@H]1C[C@@H](O)[C@@H](CO)O1 ZINC000147143280 BA For-Sale Anodyne TK2 46 34 CCCOc1ccc(C(F)(F)F)cc1NC(=O)c1csc(COC)n1 ZINC000147143316 FI On-Demand Anodyne RAF1 23 41 COC(=O)c1ccc([N+](=O)[O-])c(C(N)=O)c1 ZINC000147143325 BC In-Stock Bother GSTM2 40 36 COC(=O)c1ccc([N+](=O)[O-])c(C(N)=O)c1 ZINC000147143325 BC In-Stock Bother CACNA1D 43 33 N#CC1CCN(C(=O)CCc2ccsc2)CC1 ZINC000147143330 BE On-Demand Mild C3AR1 38 42 N#CC1CCN(C(=O)CCc2ccsc2)CC1 ZINC000147143330 BE On-Demand Mild ETHR 40 33 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C\c3ccc(OC)cc3)c2)cc1 ZINC000147143344 JK For-Sale Anodyne CYP1B1 76 83 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C\c3ccc(OC)cc3)c2)cc1 ZINC000147143344 JK For-Sale Anodyne APP 26 50 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C\c3ccc(OC)cc3)c2)cc1 ZINC000147143344 JK For-Sale Anodyne AHR 87 83 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C\c3ccc(OC)cc3)c2)cc1 ZINC000147143344 JK For-Sale Anodyne CYP1A1 73 83 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C\c3ccc(OC)cc3)c2)cc1 ZINC000147143344 JK For-Sale Anodyne TUBB2B 20 40 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C\c3ccc(OC)cc3)c2)cc1 ZINC000147143344 JK For-Sale Anodyne TUBB1 43 73 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C\c3ccc(OC)cc3)c2)cc1 ZINC000147143344 JK For-Sale Anodyne CYP1A2 18 55 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C\c3ccc(OC)cc3)c2)cc1 ZINC000147143344 JK For-Sale Anodyne CYP24A1 16 43 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C\c3ccc(OC)cc3)c2)cc1 ZINC000147143344 JK For-Sale Anodyne CYP27B1 22 43 Cc1cccn2cc(-c3ccc(NC(=O)C(=O)NC[C@H]4CCCCO4)cc3)nc12 ZINC000147143405 GF On-Demand Anodyne MTOR 46 33 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne NPY1R 26 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne F2R 41 33 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne NPFFR2 28 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne PCSK2 0 45 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne MMP3 20 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne GRIA1 47 35 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne PCSK7 0 45 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne PCSK5 63 45 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne FURIN 70 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne PCSK1 0 45 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne PCSK6 0 45 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne PROC 49 39 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne POLG_DEN26 0 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne POLG_WNV 60 36 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143434 DD On-Demand Anodyne NPFFR1 52 42 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143545 JK For-Sale Anodyne CYP1B1 76 83 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143545 JK For-Sale Anodyne APP 26 50 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143545 JK For-Sale Anodyne AHR 87 83 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143545 JK For-Sale Anodyne CYP1A1 73 83 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143545 JK For-Sale Anodyne TUBB2B 20 40 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143545 JK For-Sale Anodyne TUBB1 43 73 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143545 JK For-Sale Anodyne CYP1A2 18 55 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143545 JK For-Sale Anodyne CYP24A1 16 43 COc1ccc(/C=C\c2cc(/C=C\c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143545 JK For-Sale Anodyne CYP27B1 22 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne NPY1R 26 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne F2R 41 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne NPFFR2 28 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne PCSK2 0 45 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne MMP3 20 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne GRIA1 47 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne PCSK7 0 45 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne PCSK5 63 45 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne FURIN 70 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne PCSK1 0 45 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne PCSK6 0 45 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne PROC 49 39 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne POLG_DEN26 0 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne POLG_WNV 60 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(NC(C)=O)cc1 ZINC000147143624 DD On-Demand Anodyne NPFFR1 52 42 Cc1c(NC(=O)C(=O)NC[C@@H]2CCCCO2)c(=O)n(-c2ccccc2)n1C ZINC000147143625 FD On-Demand Anodyne FPR2 42 46 CC(C)N(C)S(=O)(=O)c1ccc(CNS(=O)(=O)c2ccc(C#N)cc2)cc1 ZINC000147143740 HE On-Demand Mild A6YCJ1_9METZ 15 42 COc1ccc(/C=C\c2cc(/C=C/c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143742 JK For-Sale Anodyne CYP1B1 76 83 COc1ccc(/C=C\c2cc(/C=C/c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143742 JK For-Sale Anodyne APP 26 50 COc1ccc(/C=C\c2cc(/C=C/c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143742 JK For-Sale Anodyne AHR 87 83 COc1ccc(/C=C\c2cc(/C=C/c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143742 JK For-Sale Anodyne CYP1A1 73 83 COc1ccc(/C=C\c2cc(/C=C/c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143742 JK For-Sale Anodyne TUBB2B 20 40 COc1ccc(/C=C\c2cc(/C=C/c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143742 JK For-Sale Anodyne TUBB1 43 73 COc1ccc(/C=C\c2cc(/C=C/c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143742 JK For-Sale Anodyne CYP1A2 18 55 COc1ccc(/C=C\c2cc(/C=C/c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143742 JK For-Sale Anodyne CYP24A1 16 43 COc1ccc(/C=C\c2cc(/C=C/c3ccc(OC)cc3)cc(/C=C/c3ccc(OC)cc3)c2)cc1 ZINC000147143742 JK For-Sale Anodyne CYP27B1 22 43 N#CC1CCN(C(=O)c2ccc(-n3cccn3)cc2)CC1 ZINC000147143752 CE On-Demand Mild AMP1_PLAFQ 52 35 N#CC1CCN(C(=O)c2ccc(-n3cccn3)cc2)CC1 ZINC000147143752 CE On-Demand Mild L3MBTL1 0 40 N#CC1CCN(C(=O)c2ccc(-n3cccn3)cc2)CC1 ZINC000147143752 CE On-Demand Mild L3MBTL3 66 41 N#CC1CCN(C(=O)c2ccc(-n3cccn3)cc2)CC1 ZINC000147143752 CE On-Demand Mild L3MBTL4 0 40 N#CC1CCN(C(=O)c2ccc(-n3cccn3)cc2)CC1 ZINC000147143752 CE On-Demand Mild MBTD1 0 41 N#CC1CCN(C(=O)c2ccc(-n3cccn3)cc2)CC1 ZINC000147143752 CE On-Demand Mild TP53BP1 0 40 N#CC1CCN(C(=O)c2ccc(-n3cccn3)cc2)CC1 ZINC000147143752 CE On-Demand Mild SLC6A7 0 41 CN(C)S(=O)(=O)c1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147143807 GC On-Demand Anodyne CA2 28 45 CN(C)S(=O)(=O)c1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147143807 GC On-Demand Anodyne CA1 26 45 CN(C)S(=O)(=O)c1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147143807 GC On-Demand Anodyne CA4 17 45 CN(C)S(=O)(=O)c1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147143807 GC On-Demand Anodyne CA12 19 45 CN(C)S(=O)(=O)c1ccc(CNC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147143807 GC On-Demand Anodyne CA9 32 45 Cc1c(NC(=O)C(=O)NC[C@H]2CCCCO2)c(=O)n(-c2ccccc2)n1C ZINC000147143817 FD On-Demand Anodyne FPR2 42 46 C[C@@]1(F)C[C@H](C(=O)OCc2ccccc2)C1 ZINC000147143825 BF In-Stock Anodyne FKBP1A 36 45 C[C@@]1(F)C[C@H](C(=O)OCc2ccccc2)C1 ZINC000147143825 BF In-Stock Anodyne GRM2 31 40 C[C@@]1(F)C[C@H](C(=O)OCc2ccccc2)C1 ZINC000147143825 BF In-Stock Anodyne CAPNS1 50 32 C[C@@]1(F)C[C@H](C(=O)OCc2ccccc2)C1 ZINC000147143825 BF In-Stock Anodyne CELA2A 15 41 C[C@@]1(F)C[C@H](C(=O)OCc2ccccc2)C1 ZINC000147143825 BF In-Stock Anodyne SLC12A5 72 38 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne CA2 15 54 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne ADRB2 15 43 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne HRH2 18 41 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne PPIA 47 51 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne CA1 26 54 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne CCR3 33 45 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne ROCK2 19 48 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne CCKBR 15 41 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne EPHX2 22 45 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne CA12 18 54 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne CA9 21 54 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne NCE103 16 54 O=C(NCCc1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1 ZINC000147143931 FI For-Sale Anodyne KCNK3 69 37 COC(=O)[C@@H](NC(=O)OC(C)(C)C)c1ccc(O)c(OC)c1 ZINC000147143967 DE For-Sale Anodyne PAPA1_CARPA 44 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(N2CCCC2)c(C)c1 ZINC000147144020 EF On-Demand Anodyne KCNQ2 57 37 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(N2CCCC2)c(C)c1 ZINC000147144020 EF On-Demand Anodyne NPY2R 61 37 CCCCCCCC[C@H](O)CC(=O)C(C)(C)C ZINC000147144098 BI For-Sale Mild CES2 51 38 CCCCCCCC[C@H](O)CC(=O)C(C)(C)C ZINC000147144098 BI For-Sale Mild EST1_PIG 74 38 CCCCCCCC[C@H](O)CC(=O)C(C)(C)C ZINC000147144098 BI For-Sale Mild CES2C 59 34 CCCCCCCC[C@H](O)CC(=O)C(C)(C)C ZINC000147144098 BI For-Sale Mild CQSS 62 40 COC(=O)[C@H](NC(=O)OC(C)(C)C)c1ccc(O)c(OC)c1 ZINC000147144164 DE For-Sale Anodyne PAPA1_CARPA 44 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(N2CCCC2)c(C)c1 ZINC000147144207 EF On-Demand Anodyne KCNQ2 57 37 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(N2CCCC2)c(C)c1 ZINC000147144207 EF On-Demand Anodyne NPY2R 61 37 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive ACE 15 41 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive CASP3 16 53 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive KLK3 57 35 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive CTSB 39 50 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive PAPA1_CARPA 44 35 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive CYSP_TRYCR 38 41 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive CTSK 34 51 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive CTSL 42 50 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive PREP 27 43 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive CAPNS1 59 33 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive SSTR3 28 41 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive CTSS 22 41 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive CAPN1 57 40 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive CASP1 21 41 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive CAPN2 98 40 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive TGM2 23 40 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive POL 0 40 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive NPR 58 33 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive F13A1 25 40 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive NAAA 64 42 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive Q9NBD4_PLAFA 0 53 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive SLC12A5 67 39 O=C(N[C@H]1CCCC[C@H]1Cl)OCc1ccccc1 ZINC000147144236 CG For-Sale Reactive Q9NAW4_PLAFA 28 53 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne CA2 110 74 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne CA6 22 61 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne CA1 95 74 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne CA7 26 53 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne PIK3CA 19 43 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne CA5B 24 61 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne CA4 117 70 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne CA14 20 61 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne CA12 36 61 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne CA9 38 53 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne CYNT 31 61 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne NCE103 19 53 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne PRMT3 51 34 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne CA15 30 61 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne MTCA1 45 45 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne P96878_MYCTU 53 45 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne MTCA2 22 53 CC(=O)Nc1ccc2nc(S(N)(=O)=O)sc2c1 ZINC000147144265 CC For-Sale Anodyne A6YCJ1_9METZ 24 61 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne DRD2 21 49 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne DRD4 42 40 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne ACHE 48 48 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne SLC6A4 15 48 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne HRH1 22 44 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne DRD3 16 41 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne SLC6A3 21 45 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne HTR4 23 40 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne LTA4H 36 43 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne SIGMAR1 61 47 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne BCHE 20 41 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne CCR3 47 44 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne CCR5 25 45 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne SLC6A5 16 42 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne EPHX2 24 42 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne MCHR1 44 40 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne CACNA1I 55 40 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne CYP2J2 45 32 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144413 FH In-Stock Anodyne KDM1A 38 42 N#CC1CCN(C(=O)c2ccc3c(c2)OCC(=O)N3)CC1 ZINC000147144416 CD On-Demand Mild L3MBTL3 49 36 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne DRD2 21 49 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne DRD4 42 40 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne ACHE 48 48 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne SLC6A4 15 48 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne HRH1 22 44 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne DRD3 16 41 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne SLC6A3 21 45 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne HTR4 23 40 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne LTA4H 36 43 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne SIGMAR1 61 47 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne BCHE 20 41 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne CCR3 47 44 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne CCR5 25 45 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne SLC6A5 16 42 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne EPHX2 24 42 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne MCHR1 44 40 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne CACNA1I 55 40 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne CYP2J2 45 32 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@@H]3c3ccccc3)CC2)cc1 ZINC000147144610 FH In-Stock Anodyne KDM1A 38 42 CCCNS(=O)(=O)c1ccc(NC(=O)Cn2cc(C)cn2)cc1 ZINC000147144674 ED On-Demand Anodyne CA2 17 40 CCCNS(=O)(=O)c1ccc(NC(=O)Cn2cc(C)cn2)cc1 ZINC000147144674 ED On-Demand Anodyne NAMPT 25 44 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne DRD2 21 49 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne DRD4 42 40 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne ACHE 48 48 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne SLC6A4 15 48 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne HRH1 22 44 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne DRD3 16 41 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne SLC6A3 21 45 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne HTR4 23 40 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne LTA4H 36 43 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne SIGMAR1 61 47 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne BCHE 20 41 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne CCR3 47 44 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne CCR5 25 45 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne SLC6A5 16 42 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne EPHX2 24 42 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne MCHR1 44 40 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne CACNA1I 55 40 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne CYP2J2 45 32 O=C(O)c1ccc(CN2CCC(CN[C@@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144800 FH In-Stock Anodyne KDM1A 38 42 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc2c(c1)OCO2 ZINC000147144802 DD On-Demand Anodyne KCNQ2 21 45 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc2c(c1)OCO2 ZINC000147144802 DD On-Demand Anodyne PCSK5 53 34 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc2c(c1)OCO2 ZINC000147144802 DD On-Demand Anodyne FURIN 52 33 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc2c(c1)OCO2 ZINC000147144802 DD On-Demand Anodyne POLG_WNV 61 31 Cc1cc(C(=O)Nc2nnc(SCc3ccc(F)cc3)s2)cc([N+](=O)[O-])c1 ZINC000147144933 HI On-Demand Bother ABL1 16 76 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne DRD2 21 49 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne DRD4 42 40 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne ACHE 48 48 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne SLC6A4 15 48 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne HRH1 22 44 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne DRD3 16 41 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne SLC6A3 21 45 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne HTR4 23 40 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne LTA4H 36 43 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne SIGMAR1 61 47 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne BCHE 20 41 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne CCR3 47 44 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne CCR5 25 45 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne SLC6A5 16 42 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne EPHX2 24 42 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne MCHR1 44 40 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne CACNA1I 55 40 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne CYP2J2 45 32 O=C(O)c1ccc(CN2CCC(CN[C@H]3C[C@H]3c3ccccc3)CC2)cc1 ZINC000147144952 FH In-Stock Anodyne KDM1A 38 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc2c(c1)OCO2 ZINC000147144966 DD On-Demand Anodyne KCNQ2 21 45 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc2c(c1)OCO2 ZINC000147144966 DD On-Demand Anodyne PCSK5 53 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc2c(c1)OCO2 ZINC000147144966 DD On-Demand Anodyne FURIN 52 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc2c(c1)OCO2 ZINC000147144966 DD On-Demand Anodyne POLG_WNV 61 31 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne LTA4H 50 47 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne HRH3 34 42 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne SRC 21 49 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne JAK3 18 49 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne JAK2 26 52 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne HNMT 31 42 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne YES1 21 44 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne TNK2 33 44 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne PSMB2 49 37 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne PSMB1 43 37 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne MKNK1 32 49 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne BMP4 22 49 c1cc(-c2ccncc2)c2nc(Nc3ccc(OCCN4CCCC4)cc3)nn2c1 ZINC000147144993 HI Annotated Anodyne BMPR1B 15 49 COCc1nc(C(=O)Nc2nnc(SCc3ccc(F)cc3)s2)cs1 ZINC000147145125 GH On-Demand Anodyne ABL1 15 65 CCCCCC(=O)NC1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000147145126 DG On-Demand Anodyne CNR1 18 44 CCCCCC(=O)NC1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000147145126 DG On-Demand Anodyne SIGMAR1 18 43 CCCCCC(=O)NC1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000147145126 DG On-Demand Anodyne CCR3 18 40 CCCCCC(=O)NC1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000147145126 DG On-Demand Anodyne LSS 15 47 CCCCCC(=O)NC1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000147145126 DG On-Demand Anodyne CCR8 26 40 CCCCCC(=O)NC1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000147145126 DG On-Demand Anodyne LASR 42 32 CCCCCC(=O)NC1CCN(C(=O)c2ccc(F)cc2)CC1 ZINC000147145126 DG On-Demand Anodyne L3MBTL3 69 38 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc2c(c1)OCO2 ZINC000147145147 DD On-Demand Anodyne KCNQ2 21 45 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc2c(c1)OCO2 ZINC000147145147 DD On-Demand Anodyne PCSK5 53 34 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc2c(c1)OCO2 ZINC000147145147 DD On-Demand Anodyne FURIN 52 33 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc2c(c1)OCO2 ZINC000147145147 DD On-Demand Anodyne POLG_WNV 61 31 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc2c(c1)OCO2 ZINC000147145334 DD On-Demand Anodyne KCNQ2 21 45 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc2c(c1)OCO2 ZINC000147145334 DD On-Demand Anodyne PCSK5 53 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc2c(c1)OCO2 ZINC000147145334 DD On-Demand Anodyne FURIN 52 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc2c(c1)OCO2 ZINC000147145334 DD On-Demand Anodyne POLG_WNV 61 31 CCOC(=O)CSc1nnc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)s1 ZINC000147145574 GF On-Demand Bother PPXI 23 41 O=C(NC1CCN(S(=O)(=O)c2ccc([N+](=O)[O-])cc2F)CC1)c1ccoc1 ZINC000147145626 GD On-Demand Bother EPHX2 23 49 CC(C)NC(=O)CN1CCCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147145666 GC On-Demand Anodyne CPT1A 33 40 CCCCCC/C=C\CCCCCCCCCCOS(C)(=O)=O ZINC000147145689 EK For-Sale Mild FAAH 15 44 CCCCCC/C=C\CCCCCCCCCCOS(C)(=O)=O ZINC000147145689 EK For-Sale Mild LPAR3 47 51 CCCCCC/C=C\CCCCCCCCCCOS(C)(=O)=O ZINC000147145689 EK For-Sale Mild FABP3 34 44 CCCCCC/C=C\CCCCCCCCCCOS(C)(=O)=O ZINC000147145689 EK For-Sale Mild LOX1.1 16 71 COCc1nc(C(=O)Nc2nc(-c3cccc4ccccc34)cs2)cs1 ZINC000147145800 GJ On-Demand Anodyne MPL 61 39 O=C(NC1CCN(S(=O)(=O)c2cccc(F)c2[N+](=O)[O-])CC1)c1ccoc1 ZINC000147145842 GD On-Demand Bother EPHX2 18 46 COC(=O)c1cc(OC)c(OC)cc1NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147145999 FF On-Demand Bother PYGL 22 41 COC(=O)c1cc(OC)c(OC)cc1NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147145999 FF On-Demand Bother KCNMA1 27 43 O=C(C1CC2(CCNCC2)C1)N1CCCN(C2CCC2)CC1 ZINC000147146076 DD For-Sale Anodyne HRH3 21 63 O=C(C1CC2(CCNCC2)C1)N1CCCN(C2CCC2)CC1 ZINC000147146076 DD For-Sale Anodyne L3MBTL3 61 46 CC(=O)SCCCCCCCCCCCCCCCC(=O)O ZINC000147146126 EK For-Sale Anodyne FABP3 34 41 CC(=O)SCCCCCCCCCCCCCCCC(=O)O ZINC000147146126 EK For-Sale Anodyne FABP5 17 50 CC(=O)SCCCCCCCCCCCCCCCC(=O)O ZINC000147146126 EK For-Sale Anodyne BHMT 28 43 CCCC[C@@H]1C[C@@H]1O ZINC000147146127 AD For-Sale Anodyne GBA 24 41 CCCC[C@@H]1C[C@@H]1O ZINC000147146127 AD For-Sale Anodyne GBA2 44 33 CCCC[C@@H]1C[C@@H]1O ZINC000147146127 AD For-Sale Anodyne P0504H10.9 91 35 CCCC[C@@H]1C[C@@H]1O ZINC000147146127 AD For-Sale Anodyne SIS 67 35 N#CCCNS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147146175 ED On-Demand Mild L3MBTL3 58 37 O=[N+]([O-])c1ccc(OCCc2ccc(Cl)cc2)nc1 ZINC000147146407 CG For-Sale Bother SNCA 43 33 COc1cccc(CCNC(=O)c2cnn(-c3ccccc3Cl)c2)c1OC ZINC000147146429 GH On-Demand Anodyne HTR1A 17 41 COc1cccc(CCNC(=O)c2cnn(-c3ccccc3Cl)c2)c1OC ZINC000147146429 GH On-Demand Anodyne DRD4 45 40 COc1cccc(CCNC(=O)c2cnn(-c3ccccc3Cl)c2)c1OC ZINC000147146429 GH On-Demand Anodyne DRD3 45 38 COc1cccc(CCNC(=O)c2cnn(-c3ccccc3Cl)c2)c1OC ZINC000147146429 GH On-Demand Anodyne NQO2 29 42 COc1cccc(CCNC(=O)c2cnn(-c3ccccc3Cl)c2)c1OC ZINC000147146429 GH On-Demand Anodyne P2RX7 15 42 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne OPRM1 15 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne NPR1 40 31 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne KLK3 56 39 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne CCKAR 24 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne CTSK 31 42 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne CTSL 19 42 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne NPFFR2 44 34 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne TIMP3 55 33 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne HDAC8 26 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne HDAC10 52 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne MMP2 19 49 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne MMP3 46 48 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne HLA-DRB1 29 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne HDAC1 24 44 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne HDAC2 33 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne HDAC3 35 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne HDAC6 34 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne PCSK5 41 34 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne FURIN 67 39 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne CCKBR 26 42 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne HDAC11 62 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne S1PR5 15 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne POLG_WNV 74 33 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne QRFPR 41 39 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne NPFFR1 63 34 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne KCNK3 65 33 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146664 GG On-Demand Anodyne KCNK9 47 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne OPRM1 15 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne NPR1 40 31 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne KLK3 56 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne CCKAR 24 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne CTSK 31 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne CTSL 19 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne NPFFR2 44 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne TIMP3 55 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne HDAC8 26 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne HDAC10 52 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne MMP2 19 49 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne MMP3 46 48 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne HLA-DRB1 29 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne HDAC1 24 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne HDAC2 33 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne HDAC3 35 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne HDAC6 34 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne PCSK5 41 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne FURIN 67 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne CCKBR 26 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne HDAC11 62 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne S1PR5 15 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne POLG_WNV 74 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne QRFPR 41 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne NPFFR1 63 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne KCNK3 65 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)Nc2ccccc2)c1 ZINC000147146867 GG On-Demand Anodyne KCNK9 47 33 COc1cc(C)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1C ZINC000147146901 GE On-Demand Anodyne EPHX2 34 42 COc1cc(C)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1C ZINC000147146901 GE On-Demand Anodyne TGM2 37 41 Cn1c(NC(=O)c2ccc3nc4n(c3c2)CCCNC4=O)nc2ccccc21 ZINC000147146905 FE Annotated Anodyne PYGM 24 41 Cn1c(NC(=O)c2ccc3nc4n(c3c2)CCCNC4=O)nc2ccccc21 ZINC000147146905 FE Annotated Anodyne LYN 40 35 Cn1c(NC(=O)c2ccc3nc4n(c3c2)CCCNC4=O)nc2ccccc21 ZINC000147146905 FE Annotated Anodyne RPS6KA3 104 53 COc1cccc(CCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1OC ZINC000147147015 FH On-Demand Anodyne NQO2 38 42 COc1cccc(CCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1OC ZINC000147147015 FH On-Demand Anodyne MTNR1A 44 44 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)CCC4)CC2)CC1 ZINC000147147057 HE On-Demand Mild CHRM5 17 49 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)CCC4)CC2)CC1 ZINC000147147057 HE On-Demand Mild TGM2 19 41 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)CCC4)CC2)CC1 ZINC000147147057 HE On-Demand Mild F13A1 25 41 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)CCC4)CC2)CC1 ZINC000147147057 HE On-Demand Mild AKR1C3 44 35 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)CCC4)CC2)CC1 ZINC000147147057 HE On-Demand Mild NAMPT 19 43 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(C)c1 ZINC000147147108 GE On-Demand Anodyne EPHX2 35 51 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(C)c1 ZINC000147147108 GE On-Demand Anodyne TGM2 30 42 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(C)c1 ZINC000147147108 GE On-Demand Anodyne ITGAV 17 40 CC1CCN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)CC1 ZINC000147147197 FF On-Demand Anodyne HRH3 28 42 CC1CCN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)CC1 ZINC000147147197 FF On-Demand Anodyne TNK2 27 43 CCc1ncc(C(=O)Nc2cc(C(F)(F)F)ccc2OCCOC)s1 ZINC000147147311 FI On-Demand Anodyne RAF1 23 41 CCc1ncc(C(=O)Nc2cc(C(F)(F)F)ccc2OCCOC)s1 ZINC000147147311 FI On-Demand Anodyne PPARD 30 40 CCc1ncc(C(=O)Nc2cc(C(F)(F)F)ccc2OCCOC)s1 ZINC000147147311 FI On-Demand Anodyne SCD 32 42 O=C(NC1CCN(S(=O)(=O)c2cccnc2)CC1)c1ccoc1 ZINC000147147342 ED On-Demand Anodyne C3AR1 40 38 O=C(NC1CCN(S(=O)(=O)c2cccnc2)CC1)c1ccoc1 ZINC000147147342 ED On-Demand Anodyne EPHX2 15 42 O=C(NC1CCN(S(=O)(=O)c2cccnc2)CC1)c1ccoc1 ZINC000147147342 ED On-Demand Anodyne TGM2 48 46 O=C(NC1CCN(S(=O)(=O)c2cccnc2)CC1)c1ccoc1 ZINC000147147342 ED On-Demand Anodyne ITGAV 22 48 CC1CCN(c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)CC1 ZINC000147147410 FF On-Demand Anodyne HRH3 28 42 CC1CCN(c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)CC1 ZINC000147147410 FF On-Demand Anodyne TNK2 27 43 COc1cccc(CCNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1OC ZINC000147147436 HH On-Demand Anodyne NQO2 40 42 COc1cccc(CCNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1OC ZINC000147147436 HH On-Demand Anodyne MTNR1A 54 44 COc1cccc(CCNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1OC ZINC000147147618 HH On-Demand Anodyne NQO2 40 42 COc1cccc(CCNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1OC ZINC000147147618 HH On-Demand Anodyne MTNR1A 54 44 N#CC1CCN(C(=O)CCCNC(=O)c2ccccc2)CC1 ZINC000147147709 CD On-Demand Mild DRD2 15 40 N#CC1CCN(C(=O)CCCNC(=O)c2ccccc2)CC1 ZINC000147147709 CD On-Demand Mild DRD4 41 32 N#CC1CCN(C(=O)CCCNC(=O)c2ccccc2)CC1 ZINC000147147709 CD On-Demand Mild DRD3 30 40 N#CC1CCN(C(=O)CCCNC(=O)c2ccccc2)CC1 ZINC000147147709 CD On-Demand Mild DPP4 23 55 COc1cccc(CCNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1OC ZINC000147147803 HH On-Demand Anodyne NQO2 40 42 COc1cccc(CCNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1OC ZINC000147147803 HH On-Demand Anodyne MTNR1A 54 44 COc1ccc(/C=N/CCCc2ccccc2)cc1 ZINC000147147904 CH For-Sale Mild SIGMAR1 21 47 COc1ccc(/C=N/CCCc2ccccc2)cc1 ZINC000147147904 CH For-Sale Mild G6PC 42 55 COc1ccc(/C=N/CCCc2ccccc2)cc1 ZINC000147147904 CH For-Sale Mild TAAR1 15 40 N#CC1CCN(C(=O)CCNC(=O)c2cccs2)CC1 ZINC000147147916 CD On-Demand Mild ETHR 45 37 COc1cccc(CCNC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)c1OC ZINC000147147979 HH On-Demand Anodyne NQO2 40 42 COc1cccc(CCNC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)c1OC ZINC000147147979 HH On-Demand Anodyne MTNR1A 54 44 CCOC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147148036 ED On-Demand Anodyne HIF1A 19 41 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc(F)c(Cl)c3)CC2)CC1 ZINC000147148147 HF On-Demand Mild F13A1 32 40 COc1cccc(CCNC(=O)c2ccc3c(c2)COC3)c1OC ZINC000147148155 EF On-Demand Anodyne DRD4 43 32 COc1cccc(CCNC(=O)c2ccc3c(c2)COC3)c1OC ZINC000147148155 EF On-Demand Anodyne NQO2 56 47 COc1cccc(CCNC(=O)c2ccc3c(c2)COC3)c1OC ZINC000147148155 EF On-Demand Anodyne MTNR1A 55 40 COc1cccc(CCNC(=O)c2ccc3c(c2)COC3)c1OC ZINC000147148155 EF On-Demand Anodyne MTNR1B 44 37 CCc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)s1 ZINC000147148173 FE On-Demand Anodyne EPHX2 17 42 CCOC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147148251 ED On-Demand Anodyne HIF1A 19 41 CCCOCC(=O)N1CCC[C@@H]1c1ccc(OC)c(OC)c1 ZINC000147148275 DF On-Demand Anodyne CPT1A 69 38 NC(=O)c1ccc(OCC(=O)Nc2ccc(CC(=O)N3CCOCC3)cc2)cc1 ZINC000147148298 GD On-Demand Anodyne ADORA2B 35 41 NC(=O)c1ccc(OCC(=O)Nc2ccc(CC(=O)N3CCOCC3)cc2)cc1 ZINC000147148298 GD On-Demand Anodyne EPHX2 25 49 CCOc1ccc(C(=O)N2CCC(C#N)CC2)cc1[N+](=O)[O-] ZINC000147148323 DE On-Demand Mild L3MBTL3 47 34 COC(=O)[C@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148335 DF For-Sale Anodyne DRD1 17 43 COC(=O)[C@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148335 DF For-Sale Anodyne HDAC8 17 40 COC(=O)[C@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148335 DF For-Sale Anodyne CA14 25 42 COC(=O)[C@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148335 DF For-Sale Anodyne MTNR1B 41 46 COC(=O)[C@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148335 DF For-Sale Anodyne GHSR 22 60 COC(=O)[C@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148335 DF For-Sale Anodyne MMP12 19 40 COC(=O)[C@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148335 DF For-Sale Anodyne CA9 15 42 COC(=O)[C@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148335 DF For-Sale Anodyne AKR1C3 18 43 CCOCCCCNC(=O)c1cnn(-c2ccccc2Cl)c1 ZINC000147148354 DG On-Demand Anodyne DRD2 23 41 CCOCCCCNC(=O)c1cnn(-c2ccccc2Cl)c1 ZINC000147148354 DG On-Demand Anodyne DRD3 48 44 CCCCS(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147148384 DD On-Demand Anodyne SLC6A9 40 38 CN(C)CCN(Cc1ccccc1)C(=O)[C@@H]1Cc2ccccc2CN1 ZINC000147148414 EE For-Sale Anodyne MC4R 24 44 CCCOCC(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147148492 DF On-Demand Anodyne CPT1A 69 38 COC(=O)[C@@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148529 DF For-Sale Anodyne DRD1 17 43 COC(=O)[C@@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148529 DF For-Sale Anodyne HDAC8 17 40 COC(=O)[C@@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148529 DF For-Sale Anodyne CA14 25 42 COC(=O)[C@@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148529 DF For-Sale Anodyne MTNR1B 41 46 COC(=O)[C@@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148529 DF For-Sale Anodyne GHSR 22 60 COC(=O)[C@@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148529 DF For-Sale Anodyne MMP12 19 40 COC(=O)[C@@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148529 DF For-Sale Anodyne CA9 15 42 COC(=O)[C@@H]1c2ccc(OC)cc2CCN1C(=O)OC(C)(C)C ZINC000147148529 DF For-Sale Anodyne AKR1C3 18 43 N#CC1CCN(C(=O)CCCNC(=O)c2ccco2)CC1 ZINC000147148541 CD On-Demand Mild KISS1R 43 36 COCCNC(=O)c1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1Cl ZINC000147148545 HF On-Demand Anodyne ROCK2 28 47 Cc1cc([N+](=O)[O-])ccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147148580 GE On-Demand Bother EPHX2 33 56 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne F2 64 41 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne ACE 93 65 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne FKBP1A 70 39 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne OPRM1 24 44 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne CELA1 57 35 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne ELANE 66 40 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne MME 17 43 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne TRHR 46 35 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne HLA-DRB3 53 36 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne TRY1_BOVIN 75 37 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne NTSR1 60 34 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne HLA-A 49 36 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne DPP4 16 41 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne PREP 55 41 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne REN 15 41 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne LGMN 62 34 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne MTOR 24 41 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne ACE2 23 53 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne TPP2 41 38 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne XIAP 57 41 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne BRCA1 63 34 CCOC(=O)[C@@H]1CCCN1C(=O)[C@H](C)N[C@H](CC(=O)c1ccccc1)C(=O)OCC ZINC000147148631 HD For-Sale Anodyne TMPRSS11D 69 38 CCCCO[C@@H](C)C(=O)N1CCC[C@@H]1c1ccc(OC)c(OC)c1 ZINC000147148696 EH On-Demand Anodyne ADAM17 43 40 CCOCCCCNC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147148778 DE On-Demand Anodyne MTNR1A 50 42 CCOCCCCNC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147148778 DE On-Demand Anodyne MTNR1B 48 38 CCOCCCCNC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147148778 DE On-Demand Anodyne ROCK2 26 41 CCOCCCCNC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147148778 DE On-Demand Anodyne CDC42BPA 0 41 CCCCO[C@H](C)C(=O)N1CCC[C@@H]1c1ccc(OC)c(OC)c1 ZINC000147148875 EH On-Demand Anodyne ADAM17 43 40 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(N)(=O)=O)c1 ZINC000147148963 HD On-Demand Anodyne CA2 16 43 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(N)(=O)=O)c1 ZINC000147148963 HD On-Demand Anodyne F2R 19 46 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(N)(=O)=O)c1 ZINC000147148963 HD On-Demand Anodyne CA4 22 40 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(N)(=O)=O)c1 ZINC000147148963 HD On-Demand Anodyne NR1H4 21 42 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(N)(=O)=O)c1 ZINC000147148963 HD On-Demand Anodyne KCNK3 120 43 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(N)(=O)=O)c1 ZINC000147148963 HD On-Demand Anodyne KCNK9 89 43 CCOCCCCNC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147148970 DE On-Demand Anodyne MTNR1A 50 42 CCOCCCCNC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147148970 DE On-Demand Anodyne MTNR1B 48 38 CCOCCCCNC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147148970 DE On-Demand Anodyne ROCK2 26 41 O=C(NC1CCN(S(=O)(=O)c2c(F)cc(F)cc2F)CC1)c1ccoc1 ZINC000147149008 GE On-Demand Anodyne MAPK13 56 31 O=C(NC1CCN(S(=O)(=O)c2c(F)cc(F)cc2F)CC1)c1ccoc1 ZINC000147149008 GE On-Demand Anodyne EPHX2 34 41 CCC(=O)C(CCN1CC2CCC1CC2)(c1ccccc1)c1ccccc1 ZINC000147149037 FK For-Sale Anodyne CHRM2 15 45 CCC(=O)C(CCN1CC2CCC1CC2)(c1ccccc1)c1ccccc1 ZINC000147149037 FK For-Sale Anodyne CHRM3 27 46 CCC(=O)C(CCN1CC2CCC1CC2)(c1ccccc1)c1ccccc1 ZINC000147149037 FK For-Sale Anodyne AOX1 18 43 CCCCO[C@@H](C)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149072 EH On-Demand Anodyne ADAM17 43 40 CC(C)(C)OC(=O)N1CCC[C@@]1(CO)CNCc1ccccc1 ZINC000147149078 DF For-Sale Anodyne SLC12A5 69 41 COc1ccc(CN[C@@H](C)c2nnc3n2CCCCC3)cc1OCCCC#N ZINC000147149236 GH On-Demand Mild EHMT2 57 32 CCCCO[C@H](C)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149243 EH On-Demand Anodyne ADAM17 43 40 CC(C)(C)OC(=O)N1CCC[C@]1(CO)CNCc1ccccc1 ZINC000147149268 DF For-Sale Anodyne SLC12A5 69 41 CCCCCCC(S(=O)(=O)C(F)(F)F)S(=O)(=O)C(F)(F)F ZINC000147149410 FG For-Sale Anodyne FDPS 31 41 CCCCCCC(S(=O)(=O)C(F)(F)F)S(=O)(=O)C(F)(F)F ZINC000147149410 FG For-Sale Anodyne CES2 57 42 CCCCCCC(S(=O)(=O)C(F)(F)F)S(=O)(=O)C(F)(F)F ZINC000147149410 FG For-Sale Anodyne CES1 57 42 CCCCCCC(S(=O)(=O)C(F)(F)F)S(=O)(=O)C(F)(F)F ZINC000147149410 FG For-Sale Anodyne EST1_PIG 69 41 CCCCCCC(S(=O)(=O)C(F)(F)F)S(=O)(=O)C(F)(F)F ZINC000147149410 FG For-Sale Anodyne CES2C 66 42 CCCCCCC(S(=O)(=O)C(F)(F)F)S(=O)(=O)C(F)(F)F ZINC000147149410 FG For-Sale Anodyne CQSS 54 34 COc1ccc(CN[C@H](C)c2nnc3n2CCCCC3)cc1OCCCC#N ZINC000147149425 GH On-Demand Mild EHMT2 57 32 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OC)c(OC)c1 ZINC000147149426 FF On-Demand Anodyne ADAM17 44 40 Nc1cccc(Cc2c[nH]c3ccccc23)c1 ZINC000147149494 BG For-Sale Anodyne HTR1D 16 50 Nc1cccc(Cc2c[nH]c3ccccc23)c1 ZINC000147149494 BG For-Sale Anodyne TACR1 17 40 Nc1cccc(Cc2c[nH]c3ccccc23)c1 ZINC000147149494 BG For-Sale Anodyne AHR 15 50 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OC)c(OC)c1 ZINC000147149608 FF On-Demand Anodyne P2RY12 73 31 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OC)c(OC)c1 ZINC000147149608 FF On-Demand Anodyne TRHR 49 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OC)c(OC)c1 ZINC000147149608 FF On-Demand Anodyne HLA-DRB3 48 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OC)c(OC)c1 ZINC000147149608 FF On-Demand Anodyne TRY1_BOVIN 55 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OC)c(OC)c1 ZINC000147149608 FF On-Demand Anodyne NTSR1 65 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OC)c(OC)c1 ZINC000147149608 FF On-Demand Anodyne NTSR2 61 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1c1ccc(OC)c(OC)c1 ZINC000147149608 FF On-Demand Anodyne ADAM17 44 40 CN(Cc1cscn1)C(=O)NCCc1c[nH]c2ccccc12 ZINC000147149623 DG On-Demand Anodyne TACR1 34 41 CN(Cc1cscn1)C(=O)NCCc1c[nH]c2ccccc12 ZINC000147149623 DG On-Demand Anodyne MC4R 33 43 CN(Cc1cscn1)C(=O)NCCc1c[nH]c2ccccc12 ZINC000147149623 DG On-Demand Anodyne BMP1 40 40 CN(Cc1cscn1)C(=O)NCCc1c[nH]c2ccccc12 ZINC000147149623 DG On-Demand Anodyne CCKAR 22 43 CN(Cc1cscn1)C(=O)NCCc1c[nH]c2ccccc12 ZINC000147149623 DG On-Demand Anodyne BRS3 22 40 C[C@@]12CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CCC(=O)[C@](C)(CO)[C@@H]5CC[C@]43C)[C@@H]1C[C@](C)(C(=O)O)CC2 ZINC000147149648 JK Annotated Anodyne PTPN2 43 42 C[C@@]12CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CCC(=O)[C@](C)(CO)[C@@H]5CC[C@]43C)[C@@H]1C[C@](C)(C(=O)O)CC2 ZINC000147149648 JK Annotated Anodyne HSD11B2 80 51 C[C@@]12CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CCC(=O)[C@](C)(CO)[C@@H]5CC[C@]43C)[C@@H]1C[C@](C)(C(=O)O)CC2 ZINC000147149648 JK Annotated Anodyne PTPN1 31 42 C[C@@]12CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CCC(=O)[C@](C)(CO)[C@@H]5CC[C@]43C)[C@@H]1C[C@](C)(C(=O)O)CC2 ZINC000147149648 JK Annotated Anodyne PA2B1_NAJME 0 41 C[C@@]12CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CCC(=O)[C@](C)(CO)[C@@H]5CC[C@]43C)[C@@H]1C[C@](C)(C(=O)O)CC2 ZINC000147149648 JK Annotated Anodyne PA2BA_PROFL 0 41 C[C@@]12CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CCC(=O)[C@](C)(CO)[C@@H]5CC[C@]43C)[C@@H]1C[C@](C)(C(=O)O)CC2 ZINC000147149648 JK Annotated Anodyne PA2A1_ECHCA 0 41 C[C@@]12CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CCC(=O)[C@](C)(CO)[C@@H]5CC[C@]43C)[C@@H]1C[C@](C)(C(=O)O)CC2 ZINC000147149648 JK Annotated Anodyne CD81 0 42 C[C@@]12CC[C@]3(C)C(=CC[C@@H]4[C@@]5(C)CCC(=O)[C@](C)(CO)[C@@H]5CC[C@]43C)[C@@H]1C[C@](C)(C(=O)O)CC2 ZINC000147149648 JK Annotated Anodyne SLCO1B2 0 41 C[C@@H]1CCCCN1Cc1ccccc1CNC(=O)COc1ccc(C(N)=O)cc1 ZINC000147149778 GF On-Demand Anodyne HRH3 41 39 C[C@@H]1CCCCN1Cc1ccccc1CNC(=O)COc1ccc(C(N)=O)cc1 ZINC000147149778 GF On-Demand Anodyne CPT1A 71 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149824 FF On-Demand Anodyne P2RY12 73 31 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149824 FF On-Demand Anodyne TRHR 49 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149824 FF On-Demand Anodyne HLA-DRB3 48 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149824 FF On-Demand Anodyne TRY1_BOVIN 55 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149824 FF On-Demand Anodyne NTSR1 65 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149824 FF On-Demand Anodyne NTSR2 61 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149824 FF On-Demand Anodyne ADAM17 44 40 O=C(NC1CCN(S(=O)(=O)CCc2ccccc2)CC1)c1ccoc1 ZINC000147149833 FE On-Demand Anodyne DRD4 20 47 O=C(NC1CCN(S(=O)(=O)CCc2ccccc2)CC1)c1ccoc1 ZINC000147149833 FE On-Demand Anodyne SIGMAR1 19 47 O=C(NC1CCN(S(=O)(=O)CCc2ccccc2)CC1)c1ccoc1 ZINC000147149833 FE On-Demand Anodyne TGM2 49 46 COc1ccc(NC(=O)C2CCN(C(=O)c3ccccc3)CC2)c(OC)n1 ZINC000147149846 FF On-Demand Anodyne NPY2R 15 40 COc1ccc(NC(=O)C2CCN(C(=O)c3ccccc3)CC2)c(OC)n1 ZINC000147149846 FF On-Demand Anodyne SLC18A3 18 45 COc1ccc(NC(=O)C2CCN(C(=O)c3ccccc3)CC2)c(OC)n1 ZINC000147149846 FF On-Demand Anodyne EPHX2 15 48 COc1ccc(NC(=O)C2CCN(C(=O)c3ccccc3)CC2)c(OC)n1 ZINC000147149846 FF On-Demand Anodyne SFRP1 40 37 COc1ccc(NC(=O)C2CCN(C(=O)c3ccccc3)CC2)c(OC)n1 ZINC000147149846 FF On-Demand Anodyne PTR1 40 35 COc1ccc(NC(=O)C2CCN(C(=O)c3ccccc3)CC2)c(OC)n1 ZINC000147149846 FF On-Demand Anodyne L3MBTL3 67 35 Cc1cccc(-n2nc(C(C)(C)C)cc2NC(=O)NCc2cc(C)on2)c1 ZINC000147149856 FI On-Demand Anodyne TNF 47 41 Cc1cccc(-n2nc(C(C)(C)C)cc2NC(=O)NCc2cc(C)on2)c1 ZINC000147149856 FI On-Demand Anodyne MAPK14 37 57 Cc1cccc(-n2nc(C(C)(C)C)cc2NC(=O)NCc2cc(C)on2)c1 ZINC000147149856 FI On-Demand Anodyne PTK2B 38 43 Cc1cccc(-n2nc(C(C)(C)C)cc2NC(=O)NCc2cc(C)on2)c1 ZINC000147149856 FI On-Demand Anodyne CARM1 46 37 Cc1cccc(-n2nc(C(C)(C)C)cc2NC(=O)NCc2cc(C)on2)c1 ZINC000147149856 FI On-Demand Anodyne DDR2 43 58 CNS(=O)(=O)c1ccc(CCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147149862 ED On-Demand Mild MLNR 20 42 C[C@H]1CCCCN1Cc1ccccc1CNC(=O)COc1ccc(C(N)=O)cc1 ZINC000147149975 GF On-Demand Anodyne HRH3 41 39 C[C@H]1CCCCN1Cc1ccccc1CNC(=O)COc1ccc(C(N)=O)cc1 ZINC000147149975 GF On-Demand Anodyne CPT1A 71 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149993 FF On-Demand Anodyne P2RY12 73 31 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149993 FF On-Demand Anodyne TRHR 49 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149993 FF On-Demand Anodyne HLA-DRB3 48 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149993 FF On-Demand Anodyne TRY1_BOVIN 55 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149993 FF On-Demand Anodyne NTSR1 65 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1c1ccc(OC)c(OC)c1 ZINC000147149993 FF On-Demand Anodyne NTSR2 61 33 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1Cl ZINC000147150015 GF On-Demand Anodyne HTR4 41 41 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1Cl ZINC000147150015 GF On-Demand Anodyne CPT2 43 32 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1Cl ZINC000147150015 GF On-Demand Anodyne UTS2R 23 49 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1Cl ZINC000147150015 GF On-Demand Anodyne EPHX2 21 52 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1Cl ZINC000147150015 GF On-Demand Anodyne TGM2 44 48 CNS(=O)(=O)c1cc(NC(=O)COc2ccc(OCc3ccccc3)cc2)ccc1C ZINC000147150042 IG On-Demand Anodyne TSHR 41 33 CNS(=O)(=O)c1cc(NC(=O)COc2ccc(OCc3ccccc3)cc2)ccc1C ZINC000147150042 IG On-Demand Anodyne PPIA 31 41 CNS(=O)(=O)c1cc(NC(=O)COc2ccc(OCc3ccccc3)cc2)ccc1C ZINC000147150042 IG On-Demand Anodyne LTA4H 40 51 CNS(=O)(=O)c1cc(NC(=O)COc2ccc(OCc3ccccc3)cc2)ccc1C ZINC000147150042 IG On-Demand Anodyne ADORA2B 30 43 CNS(=O)(=O)c1cc(NC(=O)COc2ccc(OCc3ccccc3)cc2)ccc1C ZINC000147150042 IG On-Demand Anodyne CA1 21 46 CNS(=O)(=O)c1cc(NC(=O)COc2ccc(OCc3ccccc3)cc2)ccc1C ZINC000147150042 IG On-Demand Anodyne ADAM17 27 43 CNS(=O)(=O)c1cc(NC(=O)COc2ccc(OCc3ccccc3)cc2)ccc1C ZINC000147150042 IG On-Demand Anodyne MCHR1 21 42 CNS(=O)(=O)c1cc(NC(=O)COc2ccc(OCc3ccccc3)cc2)ccc1C ZINC000147150042 IG On-Demand Anodyne FFAR1 56 38 CC(C)OCC(=O)N1CCN([C@@H](C)c2nc(-c3ccccc3)no2)CC1 ZINC000147150084 FE On-Demand Anodyne PTAFR 33 41 CC(C)OCC(=O)N1CCN([C@@H](C)c2nc(-c3ccccc3)no2)CC1 ZINC000147150084 FE On-Demand Anodyne COLA 50 36 CC(C)OCC(=O)N1CCN([C@@H](C)c2nc(-c3ccccc3)no2)CC1 ZINC000147150084 FE On-Demand Anodyne CPT1A 44 36 CC(C)OCC(=O)N1CCN([C@@H](C)c2nc(-c3ccccc3)no2)CC1 ZINC000147150084 FE On-Demand Anodyne ETHR 43 42 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1F ZINC000147150216 GE On-Demand Anodyne MAPK13 41 30 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1F ZINC000147150216 GE On-Demand Anodyne EPHX2 18 51 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1F ZINC000147150216 GE On-Demand Anodyne TGM2 43 47 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150263 DD On-Demand Anodyne HDAC10 43 37 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150263 DD On-Demand Anodyne MMP2 17 46 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150263 DD On-Demand Anodyne MMP3 32 45 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150263 DD On-Demand Anodyne FURIN 31 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150263 DD On-Demand Anodyne HDAC11 44 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150263 DD On-Demand Anodyne S1PR5 15 41 CC(C)OCC(=O)N1CCN([C@H](C)c2nc(-c3ccccc3)no2)CC1 ZINC000147150291 FE On-Demand Anodyne PTAFR 41 41 CC(C)OCC(=O)N1CCN([C@H](C)c2nc(-c3ccccc3)no2)CC1 ZINC000147150291 FE On-Demand Anodyne COLA 50 36 CC(C)OCC(=O)N1CCN([C@H](C)c2nc(-c3ccccc3)no2)CC1 ZINC000147150291 FE On-Demand Anodyne CPT1A 44 36 CC(C)OCC(=O)N1CCN([C@H](C)c2nc(-c3ccccc3)no2)CC1 ZINC000147150291 FE On-Demand Anodyne ETHR 43 42 Cc1nc(I)sc1C(=O)NCc1ccccc1 ZINC000147150340 FF For-Sale Anodyne CHRM4 35 53 Cc1nc(I)sc1C(=O)NCc1ccccc1 ZINC000147150340 FF For-Sale Anodyne HDAC1 17 46 Cc1nc(I)sc1C(=O)NCc1ccccc1 ZINC000147150340 FF For-Sale Anodyne SCD1 55 60 Cc1nc(I)sc1C(=O)NCc1ccccc1 ZINC000147150340 FF For-Sale Anodyne SCD 48 59 Cc1nc(I)sc1C(=O)NCc1ccccc1 ZINC000147150340 FF For-Sale Anodyne PDS 40 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150456 DD On-Demand Anodyne HDAC10 43 37 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150456 DD On-Demand Anodyne MMP2 17 46 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150456 DD On-Demand Anodyne MMP3 32 45 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150456 DD On-Demand Anodyne FURIN 31 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150456 DD On-Demand Anodyne HDAC11 44 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(N)=O)cc1 ZINC000147150456 DD On-Demand Anodyne S1PR5 15 41 Cc1nc(-c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)cs1 ZINC000147150479 FF On-Demand Anodyne MTOR 55 35 Cc1nc(-c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)cs1 ZINC000147150479 FF On-Demand Anodyne PDE8B 16 42 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne ACE 25 49 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne HRH2 20 44 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne SSTR2 64 43 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne GNRHR 24 47 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne OPRM1 61 55 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne OPRD1 67 54 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne OPRK1 17 48 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne GRIN2A 15 42 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MME 45 45 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne ANPEP 46 35 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne EDNRB 57 41 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne EDNRA 72 48 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne TACR1 65 63 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne TPR 18 48 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MC4R 97 47 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne BMP1 34 47 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne SSTR4 47 39 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne TACR2 48 63 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne TRPV1 15 45 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne CTSB 22 50 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne PAPA1_CARPA 21 41 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne CCKAR 113 45 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne CTSL 47 52 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne BCHE 16 55 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MPO 39 40 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne BRS3 57 59 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne C3AR1 38 51 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne UTS2R 20 44 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne NMBR 60 32 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MC3R 80 49 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MC5R 85 45 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MTNR1A 28 46 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MTNR1B 46 46 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MMP2 33 48 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MMP3 28 41 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MMP8 81 50 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne GRIA1 86 47 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MMP14 119 53 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne GRPR 77 36 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne ECE1 65 50 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne HDAC2 21 46 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne REN1 15 40 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne LNPEP 31 45 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne SSTR3 72 42 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MMP11 92 44 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne FURIN 45 47 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne CCKBR 91 48 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne GHSR 94 57 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne ALOX15 35 44 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne CAPN1 21 46 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MMP9 27 49 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne CAPN2 41 44 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MC1R 115 56 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne ADAM9 39 40 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne LAP3 43 35 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne CTSC 28 49 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne AKT1 44 35 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne C5AR1 54 39 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MMP7 36 46 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne MMP1 24 47 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne FPR1 18 43 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne NPR 39 46 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne AMP1_PLAFQ 56 47 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne SSSIM 29 43 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne KISS1R 79 43 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne ERAP2 54 49 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne NPFFR1 40 31 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne TMPRSS6 19 43 N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCCc1ccccc1 ZINC000147150520 DF On-Demand Anodyne HPN 19 40 CC(=O)CCC(=O)N1CCc2sccc2[C@@H]1c1ccccc1 ZINC000147150565 DH On-Demand Anodyne TRPM8 28 54 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1Cl ZINC000147150598 GF On-Demand Anodyne MAPK13 41 32 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1Cl ZINC000147150598 GF On-Demand Anodyne EPHX2 38 44 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1Cl ZINC000147150598 GF On-Demand Anodyne TGM2 46 46 Cc1nc(-c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)cs1 ZINC000147150635 FF On-Demand Anodyne MTOR 55 35 Cc1nc(-c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)cs1 ZINC000147150635 FF On-Demand Anodyne PDE8B 16 42 CC(C)c1ccc(C(=O)NCCN2CCOCC2)nn1 ZINC000147150669 CC For-Sale Anodyne DRD4 42 33 CC(C)c1ccc(C(=O)NCCN2CCOCC2)nn1 ZINC000147150669 CC For-Sale Anodyne CASR 43 34 CC(C)c1ccc(C(=O)NCCN2CCOCC2)nn1 ZINC000147150669 CC For-Sale Anodyne HPGDS 25 43 CC(=O)CCC(=O)N1CCc2sccc2[C@H]1c1ccccc1 ZINC000147150759 DH On-Demand Anodyne TRPM8 28 54 CCOC(=O)NCC(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147150899 DC On-Demand Anodyne MTNR1A 24 43 CCOC(=O)NCC(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147150899 DC On-Demand Anodyne MTNR1B 21 43 CCOC(=O)NCC(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147150899 DC On-Demand Anodyne KCNK3 43 39 CCOC(=O)NCC(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147150899 DC On-Demand Anodyne KCNK9 41 39 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1F ZINC000147151007 FE On-Demand Anodyne MAPK13 85 35 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1F ZINC000147151007 FE On-Demand Anodyne EPHX2 36 40 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1F ZINC000147151007 FE On-Demand Anodyne TGM2 44 44 CCN(CC)C(=O)Nc1ccc([C@@H](C)NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147151035 HF On-Demand Anodyne ACACA 22 45 CCN(CC)C(=O)Nc1ccc([C@@H](C)NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147151035 HF On-Demand Anodyne ACACB 22 45 CCN(CC)C(=O)Nc1ccc([C@@H](C)NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147151035 HF On-Demand Anodyne F7 29 48 CCN(CC)C(=O)Nc1ccc([C@@H](C)NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147151035 HF On-Demand Anodyne ACR 42 39 COC(=O)COc1cccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)c1 ZINC000147151101 GF On-Demand Anodyne MET 15 47 COC(=O)COc1cccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)c1 ZINC000147151101 GF On-Demand Anodyne CASP1 17 40 COC(=O)COc1cccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)c1 ZINC000147151101 GF On-Demand Anodyne KCNK3 83 42 COC(=O)COc1cccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)c1 ZINC000147151101 GF On-Demand Anodyne KCNK9 62 42 Cc1cc(Cl)ccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151203 GF On-Demand Anodyne CNR1 19 44 Cc1cc(Cl)ccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151203 GF On-Demand Anodyne CNR2 23 50 Cc1cc(Cl)ccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151203 GF On-Demand Anodyne MAPK13 62 33 Cc1cc(Cl)ccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151203 GF On-Demand Anodyne EPHX2 43 48 N#CC1CCN(C(=O)COC(c2ccccc2)c2ccccc2)CC1 ZINC000147151273 EH On-Demand Mild SLC6A3 40 40 N#CC1CCN(C(=O)COC(c2ccccc2)c2ccccc2)CC1 ZINC000147151273 EH On-Demand Mild PTAFR 37 52 N#CC1CCN(C(=O)COC(c2ccccc2)c2ccccc2)CC1 ZINC000147151273 EH On-Demand Mild DPP4 17 41 COC(=O)COc1cccc(NC(=O)CCNS(C)(=O)=O)c1 ZINC000147151311 EC On-Demand Anodyne MTNR1A 23 43 COC(=O)COc1cccc(NC(=O)CCNS(C)(=O)=O)c1 ZINC000147151311 EC On-Demand Anodyne KCNK3 40 36 Cc1ccc(OCCCCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147151363 HF On-Demand Bother TBXA2R 26 43 Cc1ccc(F)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147151401 FE On-Demand Anodyne MAPK13 88 35 Cc1ccc(F)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147151401 FE On-Demand Anodyne EPHX2 41 46 CCCn1c(NC(=O)c2cnc(CC)s2)nc2ccccc21 ZINC000147151447 DH On-Demand Anodyne ITK 39 44 CC(C)(C)NC[C@H](O)c1ccc(OC(=O)C(C)(C)C)c(OC(=O)C(C)(C)C)c1 ZINC000147151449 GI Annotated Anodyne ADRB2 21 52 CC(C)(C)NC[C@H](O)c1ccc(OC(=O)C(C)(C)C)c(OC(=O)C(C)(C)C)c1 ZINC000147151449 GI Annotated Anodyne ADRB1 0 43 CC(C)(C)NC[C@H](O)c1ccc(OC(=O)C(C)(C)C)c(OC(=O)C(C)(C)C)c1 ZINC000147151449 GI Annotated Anodyne ELANE 0 47 CC(C)n1cc(C(=O)c2ccnc(NC(=O)Nc3ccc(F)cc3F)c2)c2c(N)ncnc21 ZINC000147151495 JI Annotated Anodyne PDPK1 51 43 CC(C)n1cc(C(=O)c2ccnc(NC(=O)Nc3ccc(F)cc3F)c2)c2c(N)ncnc21 ZINC000147151495 JI Annotated Anodyne TEK 17 40 Cc1c(Cl)cccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151589 GF On-Demand Anodyne CNR2 15 50 Cc1c(Cl)cccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151589 GF On-Demand Anodyne EPHX2 40 46 Cc1c(Cl)cccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151589 GF On-Demand Anodyne TGM2 38 40 COc1cc2cncc(Cc3ccc(OC)c(OC)c3)c2cc1O ZINC000147151784 EH Annotated Anodyne FOLA 32 49 COc1cc2cncc(Cc3ccc(OC)c(OC)c3)c2cc1O ZINC000147151784 EH Annotated Anodyne DRTS_PLAFK 40 49 COc1cc2cncc(Cc3ccc(OC)c(OC)c3)c2cc1O ZINC000147151784 EH Annotated Anodyne DRTS_PLABA 42 49 COc1cc2cncc(Cc3ccc(OC)c(OC)c3)c2cc1O ZINC000147151784 EH Annotated Anodyne Q9XSW7_PIG 0 47 COc1cc2cncc(Cc3ccc(OC)c(OC)c3)c2cc1O ZINC000147151784 EH Annotated Anodyne DHFRI 18 43 COc1cc2cncc(Cc3ccc(OC)c(OC)c3)c2cc1O ZINC000147151784 EH Annotated Anodyne TTR 0 41 COc1cc2cncc(Cc3ccc(OC)c(OC)c3)c2cc1O ZINC000147151784 EH Annotated Anodyne DFRA17 0 40 Cc1ccc(F)cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151790 FE On-Demand Anodyne CNR2 22 56 Cc1ccc(F)cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151790 FE On-Demand Anodyne MAPK14 42 38 Cc1ccc(F)cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151790 FE On-Demand Anodyne MAPK13 84 35 Cc1ccc(F)cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151790 FE On-Demand Anodyne EPHX2 39 52 Cc1ccc(F)cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147151790 FE On-Demand Anodyne MCHR1 16 40 O=C(NCc1c(F)cc(F)cc1F)c1ccccc1 ZINC000147151983 CG On-Demand Anodyne ECR 40 42 O=C(NCc1c(F)cc(F)cc1F)c1ccccc1 ZINC000147151983 CG On-Demand Anodyne CTRB1 23 40 O=C(NCc1c(F)cc(F)cc1F)c1ccccc1 ZINC000147151983 CG On-Demand Anodyne KCNK3 46 44 O=C(NC1CCN(S(=O)(=O)c2cccc(Cl)c2F)CC1)c1ccoc1 ZINC000147151993 GF On-Demand Anodyne EPHX2 30 45 CCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)CCN2C(=O)CNC2=O)cc1 ZINC000147152008 HC On-Demand Anodyne HDAC11 41 35 CC(=O)Nc1ccc(C#N)nc1 ZINC000147152046 AC For-Sale Mild IDO1 15 41 COc1ccc2cc(-c3cnc(-c4ccccc4)o3)ccc2c1 ZINC000147152116 DK For-Sale Anodyne CYP11B1 20 56 COc1ccc2cc(-c3cnc(-c4ccccc4)o3)ccc2c1 ZINC000147152116 DK For-Sale Anodyne CYP11B2 32 56 COc1ccc2cc(-c3cnc(-c4ccccc4)o3)ccc2c1 ZINC000147152116 DK For-Sale Anodyne LUCI_PHOPE 47 35 CCCCCCCCS(=O)(=O)[C@@H](CC(=O)O)C(=O)O ZINC000147152215 CD For-Sale Anodyne CES2 44 41 CCCCCCCCS(=O)(=O)[C@@H](CC(=O)O)C(=O)O ZINC000147152215 CD For-Sale Anodyne CES1 35 41 CCCCCCCCS(=O)(=O)[C@@H](CC(=O)O)C(=O)O ZINC000147152215 CD For-Sale Anodyne EST1_PIG 55 41 CCCCCCCCS(=O)(=O)[C@@H](CC(=O)O)C(=O)O ZINC000147152215 CD For-Sale Anodyne CES2C 47 41 CCCCCCCCS(=O)(=O)[C@@H](CC(=O)O)C(=O)O ZINC000147152215 CD For-Sale Anodyne CQSS 53 32 NC(=O)NC[C@H]1CCCN(C(=O)c2cccn(Cc3ccccc3)c2=O)C1 ZINC000147152216 FD On-Demand Anodyne F2 21 41 NC(=O)NC[C@@H]1CCCN(C(=O)c2cccn(Cc3ccccc3)c2=O)C1 ZINC000147152389 FD On-Demand Anodyne F2 21 41 COc1ccc(Cl)cc1C1(CNC(=O)NCCCn2ccnc2)CCOCC1 ZINC000147152401 HF On-Demand Anodyne TBXAS1 32 43 COc1ccc(Cl)cc1C1(CNC(=O)NCCCn2ccnc2)CCOCC1 ZINC000147152401 HF On-Demand Anodyne QPCT 47 54 CCCCCCCCS(=O)(=O)[C@H](CC(=O)O)C(=O)O ZINC000147152411 CD For-Sale Anodyne CES2 44 41 CCCCCCCCS(=O)(=O)[C@H](CC(=O)O)C(=O)O ZINC000147152411 CD For-Sale Anodyne CES1 35 41 CCCCCCCCS(=O)(=O)[C@H](CC(=O)O)C(=O)O ZINC000147152411 CD For-Sale Anodyne EST1_PIG 55 41 CCCCCCCCS(=O)(=O)[C@H](CC(=O)O)C(=O)O ZINC000147152411 CD For-Sale Anodyne CES2C 47 41 CCCCCCCCS(=O)(=O)[C@H](CC(=O)O)C(=O)O ZINC000147152411 CD For-Sale Anodyne CQSS 53 32 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)CCCC4)CC2)CC1 ZINC000147152513 HF On-Demand Mild CHRM5 17 46 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)CCCC4)CC2)CC1 ZINC000147152513 HF On-Demand Mild TGM2 19 41 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)CCCC4)CC2)CC1 ZINC000147152513 HF On-Demand Mild F13A1 25 41 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)CCCC4)CC2)CC1 ZINC000147152513 HF On-Demand Mild AKR1C3 44 35 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)CCCC4)CC2)CC1 ZINC000147152513 HF On-Demand Mild NAMPT 25 45 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](c2ccc(Cl)cc2)c2cccs2)c1 ZINC000147152607 HJ On-Demand Bother TAAR1 22 40 C[C@]12Cc3conc3C[C@@H]1CC[C@@H]1[C@@H]2CC[C@]2(C)[C@H]1CC[C@]2(C)O ZINC000147152646 EI In-Stock Anodyne SHBG 33 53 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147152762 ED On-Demand Anodyne MAPK14 30 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147152762 ED On-Demand Anodyne KCNK3 57 37 CC(=O)CCc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147152778 CI For-Sale Anodyne TACR1 38 47 Cc1cccc([N+](=O)[O-])c1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147152790 GE On-Demand Bother EPHX2 23 43 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](c2ccc(Cl)cc2)c2cccs2)c1 ZINC000147152816 HJ On-Demand Bother TAAR1 22 40 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1Cl ZINC000147152829 GE On-Demand Anodyne CA2 19 54 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1Cl ZINC000147152829 GE On-Demand Anodyne CCR4 0 46 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1Cl ZINC000147152829 GE On-Demand Anodyne CA4 30 56 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1Cl ZINC000147152829 GE On-Demand Anodyne SGK1 16 43 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1Cl ZINC000147152829 GE On-Demand Anodyne NFKBIA 0 41 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1Cl ZINC000147152829 GE On-Demand Anodyne CYNT 36 54 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1Cl ZINC000147152829 GE On-Demand Anodyne CA15 17 45 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1Cl ZINC000147152829 GE On-Demand Anodyne CA 0 51 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1Cl ZINC000147152829 GE On-Demand Anodyne A6YCJ1_9METZ 16 45 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1cccc(Cl)c1Cl ZINC000147152829 GE On-Demand Anodyne Q5TU56_ANOGA 0 45 COc1ccc([C@H](O)C(=O)O)c(O)c1 ZINC000147152910 AC For-Sale Anodyne THRA 44 35 COc1ccc([C@H](O)C(=O)O)c(O)c1 ZINC000147152910 AC For-Sale Anodyne THRB 41 35 COc1ccc([C@H](O)C(=O)O)c(O)c1 ZINC000147152910 AC For-Sale Anodyne AKR1C3 24 45 COc1ccc([C@H](O)C(=O)O)c(O)c1 ZINC000147152910 AC For-Sale Anodyne AKR1C2 50 36 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147152944 ED On-Demand Anodyne MAPK14 30 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147152944 ED On-Demand Anodyne KCNK3 57 37 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC)cc2C(F)(F)F)c1 ZINC000147153031 FH On-Demand Bother KCNMA1 30 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC)cc2C(F)(F)F)c1 ZINC000147153031 FH On-Demand Bother TAAR1 23 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC)cc2C(F)(F)F)c1 ZINC000147153031 FH On-Demand Bother AKR1C3 19 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(OC)cc2C(F)(F)F)c1 ZINC000147153031 FH On-Demand Bother AKR1C2 49 46 COc1ccc([C@@H](O)C(=O)O)c(O)c1 ZINC000147153078 AC For-Sale Anodyne THRA 44 35 COc1ccc([C@@H](O)C(=O)O)c(O)c1 ZINC000147153078 AC For-Sale Anodyne THRB 41 35 COc1ccc([C@@H](O)C(=O)O)c(O)c1 ZINC000147153078 AC For-Sale Anodyne AKR1C3 24 45 COc1ccc([C@@H](O)C(=O)O)c(O)c1 ZINC000147153078 AC For-Sale Anodyne AKR1C2 50 36 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccccc2N2CCc3ccccc32)C1 ZINC000147153122 HF On-Demand Anodyne LPL 43 34 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccccc2N2CCc3ccccc32)C1 ZINC000147153122 HF On-Demand Anodyne KCNQ2 54 38 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccccc2N2CCc3ccccc32)C1 ZINC000147153122 HF On-Demand Anodyne P2RY1 16 47 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccccc2N2CCc3ccccc32)C1 ZINC000147153122 HF On-Demand Anodyne EPHX2 23 40 CCNS(=O)(=O)c1ccc(C(=O)N2CCN(Cc3cccc4cccnc34)CC2)cc1 ZINC000147153210 IE On-Demand Anodyne CCR8 35 41 O=C(NC1[C@H]2CN(CCCc3ccccc3)C[C@H]12)[C@@](O)(c1ccccc1)C1CCCC1 ZINC000147153301 HH Annotated Anodyne CHRM2 28 88 O=C(NC1[C@H]2CN(CCCc3ccccc3)C[C@H]12)[C@@](O)(c1ccccc1)C1CCCC1 ZINC000147153301 HH Annotated Anodyne CHRM1 28 58 O=C(NC1[C@H]2CN(CCCc3ccccc3)C[C@H]12)[C@@](O)(c1ccccc1)C1CCCC1 ZINC000147153301 HH Annotated Anodyne CHRM3 45 76 O=C(NC1[C@H]2CN(CCCc3ccccc3)C[C@H]12)[C@@](O)(c1ccccc1)C1CCCC1 ZINC000147153301 HH Annotated Anodyne SIGMAR1 27 40 O=C(NC1[C@H]2CN(CCCc3ccccc3)C[C@H]12)[C@@](O)(c1ccccc1)C1CCCC1 ZINC000147153301 HH Annotated Anodyne AMY2 45 31 O=C(NC1[C@H]2CN(CCCc3ccccc3)C[C@H]12)[C@@](O)(c1ccccc1)C1CCCC1 ZINC000147153301 HH Annotated Anodyne CYP2J2 53 39 O=C(NC1[C@H]2CN(CCCc3ccccc3)C[C@H]12)[C@@](O)(c1ccccc1)C1CCCC1 ZINC000147153301 HH Annotated Anodyne BIRC2 19 40 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccccc2N2CCc3ccccc32)C1 ZINC000147153329 HF On-Demand Anodyne LPL 43 34 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccccc2N2CCc3ccccc32)C1 ZINC000147153329 HF On-Demand Anodyne KCNQ2 54 38 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccccc2N2CCc3ccccc32)C1 ZINC000147153329 HF On-Demand Anodyne P2RY1 16 47 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccccc2N2CCc3ccccc32)C1 ZINC000147153329 HF On-Demand Anodyne EPHX2 23 40 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cc1ccccc1 ZINC000147153507 GF On-Demand Anodyne TSHR 56 32 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cc1ccccc1 ZINC000147153507 GF On-Demand Anodyne QRFPR 47 44 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)NC[C@@H]2CCCO2)cc1 ZINC000147153542 GE On-Demand Anodyne HDAC11 44 35 CC[C@@H](O)c1ccccc1N(C)C ZINC000147153639 AE For-Sale Anodyne AOC3 23 41 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3C[C@H](C)O[C@H](C)C3)cc2)s1 ZINC000147153647 HF On-Demand Anodyne F13A1 58 35 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3C[C@H](C)O[C@H](C)C3)cc2)s1 ZINC000147153647 HF On-Demand Anodyne MERTK 29 41 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3C[C@H](C)O[C@H](C)C3)cc2)s1 ZINC000147153647 HF On-Demand Anodyne NAMPT 38 51 O=C(NCc1cccnc1)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147153679 EH On-Demand Anodyne CHRNA7 32 43 O=C(NCc1cccnc1)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147153679 EH On-Demand Anodyne SCD 15 40 O=C(NCc1cccnc1)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147153679 EH On-Demand Anodyne NAMPT 75 47 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cc1ccccc1 ZINC000147153682 GF On-Demand Anodyne TSHR 56 32 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cc1ccccc1 ZINC000147153682 GF On-Demand Anodyne QRFPR 47 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)NC[C@@H]2CCCO2)cc1 ZINC000147153720 GE On-Demand Anodyne HDAC11 44 35 NC(=O)NC[C@H]1CCCN(C(=O)c2csc(-c3ccccc3F)n2)C1 ZINC000147153727 FE On-Demand Anodyne TRPC6 64 35 NC(=O)NC[C@H]1CCCN(C(=O)c2csc(-c3ccccc3F)n2)C1 ZINC000147153727 FE On-Demand Anodyne TRPC3 43 35 CCOC[C@H](C)NC(=O)Nc1ccc(S(=O)(=O)C2CCCC2)cc1 ZINC000147153755 FF On-Demand Anodyne P96878_MYCTU 40 36 COC(=O)Nc1cccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147153771 EI On-Demand Anodyne MDM2 66 34 COC(=O)Nc1cccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147153771 EI On-Demand Anodyne KCNK3 42 39 CC[C@H](O)c1ccccc1N(C)C ZINC000147153792 AE For-Sale Anodyne AOC3 23 41 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3C[C@@H](C)O[C@H](C)C3)cc2)s1 ZINC000147153854 HF On-Demand Anodyne F13A1 58 35 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3C[C@@H](C)O[C@H](C)C3)cc2)s1 ZINC000147153854 HF On-Demand Anodyne MERTK 29 41 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3C[C@@H](C)O[C@H](C)C3)cc2)s1 ZINC000147153854 HF On-Demand Anodyne NAMPT 38 51 O=C(NCc1ccccn1)NCC1(c2cccc(F)c2)CCCCC1 ZINC000147153877 EH On-Demand Anodyne NMBR 44 33 CCCCCCCCCCCCNC(=O)[C@@H](N)C(C)C ZINC000147153902 CI For-Sale Mild S1PR3 22 51 CCCCCCCCCCCCNC(=O)[C@@H](N)C(C)C ZINC000147153902 CI For-Sale Mild S1PR2 36 51 CCCCCCCCCCCCNC(=O)[C@@H](N)C(C)C ZINC000147153902 CI For-Sale Mild EPHX2 17 40 CCCCCCCCCCCCNC(=O)[C@@H](N)C(C)C ZINC000147153902 CI For-Sale Mild TPP2 21 51 CCCCCCCCCCCCNC(=O)[C@@H](N)C(C)C ZINC000147153902 CI For-Sale Mild ASAH1 96 36 CCCCCCCCCCCCNC(=O)[C@@H](N)C(C)C ZINC000147153902 CI For-Sale Mild NOD1 89 46 CCCCCCCCCCCCNC(=O)[C@@H](N)C(C)C ZINC000147153902 CI For-Sale Mild CQSS 61 44 NC(=O)NC[C@@H]1CCCN(C(=O)c2csc(-c3ccccc3F)n2)C1 ZINC000147153915 FE On-Demand Anodyne TRPC6 64 35 NC(=O)NC[C@@H]1CCCN(C(=O)c2csc(-c3ccccc3F)n2)C1 ZINC000147153915 FE On-Demand Anodyne TRPC3 43 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)NC[C@H]2CCCO2)cc1 ZINC000147153922 GE On-Demand Anodyne HDAC11 44 35 COC(=O)Nc1cccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147153956 EI On-Demand Anodyne MDM2 66 34 COC(=O)Nc1cccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147153956 EI On-Demand Anodyne KCNK3 42 39 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild PTAFR 0 40 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild PAPA1_CARPA 43 40 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild CTSK 22 50 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild FAAH 26 49 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild CES2 50 42 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild S1PR2 15 41 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild EST1_PIG 66 42 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild EPHX2 41 44 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild CES2C 60 42 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild PGA5 47 42 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild ASAH1 95 36 CCCCCCCNC(=O)OC(C)(C)C ZINC000147154019 BG For-Sale Mild CQSS 51 31 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3C[C@H](C)O[C@@H](C)C3)cc2)s1 ZINC000147154025 HF On-Demand Anodyne F13A1 58 35 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3C[C@H](C)O[C@@H](C)C3)cc2)s1 ZINC000147154025 HF On-Demand Anodyne MERTK 29 41 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3C[C@H](C)O[C@@H](C)C3)cc2)s1 ZINC000147154025 HF On-Demand Anodyne NAMPT 38 51 CC[C@H](C)NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147154113 EE On-Demand Mild L3MBTL1 0 40 CC[C@H](C)NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147154113 EE On-Demand Mild MBTD1 0 40 COc1ccc(C2(CNC(=O)NCCc3ccccn3)CCCCC2)cc1 ZINC000147154117 FH On-Demand Anodyne NMBR 72 41 COc1ccc(C2(CNC(=O)NCCc3ccccn3)CCCCC2)cc1 ZINC000147154117 FH On-Demand Anodyne GRPR 43 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)NC[C@H]2CCCO2)cc1 ZINC000147154122 GE On-Demand Anodyne HDAC11 44 35 CC(C)(C)C[C@H]1N[C@@H](C(=O)NCCN2CC[C@H](O)C2)[C@H](c2cccc(Cl)c2)[C@@]12C(=O)Nc1cc(Cl)c(F)cc12 ZINC000147154131 KI Annotated Anodyne MDM2 108 75 Cc1cc(F)ccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147154143 FE On-Demand Anodyne CNR2 18 50 Cc1cc(F)ccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147154143 FE On-Demand Anodyne MAPK13 81 34 Cc1cc(F)ccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147154143 FE On-Demand Anodyne EPHX2 41 61 COC(=O)Nc1cccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147154161 EI On-Demand Anodyne MDM2 66 34 COC(=O)Nc1cccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147154161 EI On-Demand Anodyne KCNK3 42 39 CCCCO[C@@H](C)C(=O)Nc1ccc(NC(=O)NCc2ccco2)cc1 ZINC000147154320 FH On-Demand Anodyne CA1 15 53 COc1ccc(C2(CNC(=O)NCCN3CCOCC3)CCCCC2)cc1 ZINC000147154326 GF On-Demand Anodyne DRD4 48 38 COc1ccc(C2(CNC(=O)NCCN3CCOCC3)CCCCC2)cc1 ZINC000147154326 GF On-Demand Anodyne F10 24 41 COc1ccc(C2(CNC(=O)NCCN3CCOCC3)CCCCC2)cc1 ZINC000147154326 GF On-Demand Anodyne TACR2 24 41 COc1ccc(C2(CNC(=O)NCCN3CCOCC3)CCCCC2)cc1 ZINC000147154326 GF On-Demand Anodyne MTNR1A 28 40 COc1ccc(C2(CNC(=O)NCCN3CCOCC3)CCCCC2)cc1 ZINC000147154326 GF On-Demand Anodyne MTNR1B 15 40 COc1ccc(C2(CNC(=O)NCCN3CCOCC3)CCCCC2)cc1 ZINC000147154326 GF On-Demand Anodyne SOAT1 17 44 COc1ccc(C2(CNC(=O)NCCN3CCOCC3)CCCCC2)cc1 ZINC000147154326 GF On-Demand Anodyne PTGDS 31 41 COc1ccc(C2(CNC(=O)NCCN3CCOCC3)CCCCC2)cc1 ZINC000147154326 GF On-Demand Anodyne EPHX2 22 41 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)NC[C@H]3CCCO3)cc2)CC1 ZINC000147154332 GD On-Demand Mild L3MBTL3 62 39 Cc1ccc(COc2ccc(/C=c3\sc4nc5ccccc5n4c3=O)cc2Br)cc1 ZINC000147154389 JK In-Stock Anodyne PLK1 15 41 Cc1ccc(COc2ccc(/C=c3\sc4nc5ccccc5n4c3=O)cc2Br)cc1 ZINC000147154389 JK In-Stock Anodyne MAPT 53 35 Clc1cccnc1N1CCc2ncnc(Nc3ccccc3)c2C1 ZINC000147154418 EH Annotated Anodyne TRPV1 22 70 Cc1cc(N2CCOCC2)ccc1NC(=O)NC[C@@H](O)COc1c(C)cccc1C ZINC000147154420 HG On-Demand Anodyne MAPK14 17 41 CCCCO[C@H](C)C(=O)Nc1ccc(NC(=O)NCc2ccco2)cc1 ZINC000147154504 FH On-Demand Anodyne CA1 15 53 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne F2 66 47 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne PLG 32 41 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne ACE 47 48 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne FKBP1A 55 43 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne OPRM1 30 42 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne OPRD1 19 42 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne F10 0 53 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne CELA1 33 52 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne ELANE 41 44 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne CTRA_BOVIN 65 36 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne HRH3 23 44 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne TRY1_BOVIN 75 38 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne CTSG 45 36 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne CTSK 18 59 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne COLA 0 41 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne PRNP 38 45 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne ITGA4 37 40 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne PREP 80 52 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne CELA2A 53 36 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne LGMN 93 52 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne CFTR 57 34 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne HCK 32 40 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne ACE2 24 45 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne KLK5 27 46 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne FLT3 15 47 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne XIAP 51 40 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne F13A1 45 39 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne STAT6 17 41 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne F1PEP1 0 52 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne BRCA1 60 32 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne SLC12A5 74 41 CN1CCN(c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154523 HG On-Demand Anodyne TMPRSS11D 66 37 CCNS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147154532 DD On-Demand Mild SFRP1 45 37 CCNS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147154532 DD On-Demand Mild L3MBTL3 69 38 COC(=O)c1cc(Cl)ccc1NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147154534 HF On-Demand Bother F10 27 41 COC(=O)c1cc(Cl)ccc1NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147154534 HF On-Demand Bother KCNMA1 41 48 Cc1cc(N2CCOCC2)ccc1NC(=O)NC[C@H](O)COc1c(C)cccc1C ZINC000147154613 HG On-Demand Anodyne MAPK14 17 41 CC(C)(C)OC(=O)c1ccc(CN2CCC(C=O)CC2)cc1 ZINC000147154623 DG In-Stock Mild LTA4H 16 41 CC(C)(C)OC(=O)c1ccc(CN2CCC(C=O)CC2)cc1 ZINC000147154623 DG In-Stock Mild SIGMAR1 43 47 CC(C)(C)OC(=O)c1ccc(CN2CCC(C=O)CC2)cc1 ZINC000147154623 DG In-Stock Mild CACNA1I 42 33 CC(C)(C)OC(=O)c1ccc(CN2CCC(C=O)CC2)cc1 ZINC000147154623 DG In-Stock Mild PANC 23 40 CC(C)(C)OC(=O)c1ccc(CN2CCC(C=O)CC2)cc1 ZINC000147154623 DG In-Stock Mild NOD2 41 35 COC(=O)c1c(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)sc(C)c1C ZINC000147154662 EH On-Demand Bother CACNA1D 40 33 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne F2 66 47 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne PLG 32 41 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne ACE 47 48 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne FKBP1A 55 43 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne OPRM1 30 42 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne OPRD1 19 42 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne F10 0 53 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne CELA1 33 52 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne ELANE 41 44 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne CTRA_BOVIN 65 36 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne HRH3 23 44 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne TRY1_BOVIN 75 38 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne CTSG 45 36 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne CTSK 18 59 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne COLA 0 41 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne PRNP 38 45 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne ITGA4 37 40 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne PREP 80 52 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne CELA2A 53 36 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne LGMN 93 52 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne CFTR 57 34 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne HCK 32 40 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne ACE2 24 45 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne KLK5 27 46 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne FLT3 15 47 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne XIAP 51 40 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne F13A1 45 39 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne STAT6 17 41 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne F1PEP1 0 52 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne BRCA1 60 32 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne SLC12A5 74 41 CN1CCN(c2ccc(NC(=O)[C@H]3CCCN3C(=O)OCc3ccccc3)cc2)CC1 ZINC000147154725 HG On-Demand Anodyne TMPRSS11D 66 37 C[C@@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147154730 GF On-Demand Mild PREP 26 43 C[C@@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147154730 GF On-Demand Mild AKR1C3 59 43 C[C@@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147154730 GF On-Demand Mild L3MBTL1 0 43 C[C@@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147154730 GF On-Demand Mild L3MBTL3 66 43 COC(=O)c1cc(Cl)ccc1NC(=O)c1cc(OC)ccc1[N+](=O)[O-] ZINC000147154732 FG On-Demand Bother KCNMA1 51 51 COC(=O)c1cc(Cl)ccc1NC(=O)c1cc(OC)ccc1[N+](=O)[O-] ZINC000147154732 FG On-Demand Bother TAAR1 25 42 COC(=O)c1cc(Cl)ccc1NC(=O)c1cc(OC)ccc1[N+](=O)[O-] ZINC000147154732 FG On-Demand Bother AKR1C3 19 42 COC(=O)c1cc(Cl)ccc1NC(=O)c1cc(OC)ccc1[N+](=O)[O-] ZINC000147154732 FG On-Demand Bother AKR1C2 48 44 CC(C)C[C@@H](CNC(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1)N1CCOCC1 ZINC000147154754 HD On-Demand Anodyne TGM2 37 43 CC(C)C[C@@H](CNC(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1)N1CCOCC1 ZINC000147154754 HD On-Demand Anodyne NAMPT 37 41 O=C(NC1CCN(S(=O)(=O)c2ccc(F)cc2Cl)CC1)c1ccoc1 ZINC000147154897 GF On-Demand Anodyne CNR2 15 49 O=C(NC1CCN(S(=O)(=O)c2ccc(F)cc2Cl)CC1)c1ccoc1 ZINC000147154897 GF On-Demand Anodyne MAPK13 53 33 O=C(NC1CCN(S(=O)(=O)c2ccc(F)cc2Cl)CC1)c1ccoc1 ZINC000147154897 GF On-Demand Anodyne EPHX2 32 60 CC(C)(C)c1nc(CN2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)cs1 ZINC000147154914 HE On-Demand Anodyne CPT1A 34 42 C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147154945 GF On-Demand Mild PREP 26 43 C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147154945 GF On-Demand Mild AKR1C3 59 43 C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147154945 GF On-Demand Mild L3MBTL1 0 43 C[C@H]1CCCCN1S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147154945 GF On-Demand Mild L3MBTL3 66 43 Cc1nn(C(F)F)c(C)c1CC(=O)NCC#Cc1ccccc1 ZINC000147154951 DF On-Demand Mild P2RX7 52 45 CC(C)C[C@H](CNC(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1)N1CCOCC1 ZINC000147154958 HD On-Demand Anodyne TGM2 37 43 CC(C)C[C@H](CNC(=O)c1ccc(S(=O)(=O)N2CCCC2)cc1)N1CCOCC1 ZINC000147154958 HD On-Demand Anodyne NAMPT 37 41 Cc1cc(N2CCOCC2)ccc1NC(=O)NCc1ccc(-n2ccnc2)c(F)c1 ZINC000147155127 HG On-Demand Anodyne NOS2 87 36 Cc1cc(N2CCOCC2)ccc1NC(=O)NCc1ccc(-n2ccnc2)c(F)c1 ZINC000147155127 HG On-Demand Anodyne STAT6 44 32 CCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2csc(C(C)(C)C)n2)CC1 ZINC000147155295 GD On-Demand Anodyne P2RY12 154 36 CCCCO[C@@H](C)C(=O)NCC#Cc1ccccc1 ZINC000147155351 CE On-Demand Mild MMP12 15 41 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne PRSS1 19 41 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne KIT 21 41 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne MAPK14 21 55 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne TRPV1 15 47 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne ROCK1 27 42 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne PRNP 56 40 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne KDR 18 41 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne ROCK2 28 44 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne NR1H4 15 43 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne SCN10A 51 41 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne CSF1R 20 42 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne TAAR1 42 41 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne SHH 52 35 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne SMO 23 41 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne KCNK3 131 47 COC(=O)c1cccc(NC(=O)c2ccc(-c3nnc(-c4ccc(C)cc4)o3)cc2)c1 ZINC000147155368 HJ On-Demand Anodyne KCNK9 82 46 Cc1cc(N2CCOCC2)ccc1NC(=O)NC[C@@H]1CCCO[C@@H]1c1ccccc1 ZINC000147155418 HI On-Demand Anodyne HRH3 17 41 Cc1cc(N2CCOCC2)ccc1NC(=O)NC[C@H]1CCCO[C@@H]1c1ccccc1 ZINC000147155612 HI On-Demand Anodyne HRH3 17 41 O=S(=O)(NC[C@@H]1CN(Cc2ccccc2)CCO1)c1ccc(-c2ccccc2)cc1 ZINC000147155648 HH On-Demand Anodyne DRD4 29 53 CC(C)(C)OC(=O)N1CC[C@H](S(=O)(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000147155783 FD For-Sale Anodyne GPR119 37 41 CC(C)(C)OC(=O)N1CC[C@H](S(=O)(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000147155783 FD For-Sale Anodyne SFRP1 57 38 N#CC1CCN(C(=O)/C=C/c2ccc(F)c(Cl)c2)CC1 ZINC000147155800 CG On-Demand Mild CCR2 88 50 Cc1cc(N2CCOCC2)ccc1NC(=O)NC[C@@H]1CCCO[C@H]1c1ccccc1 ZINC000147155815 HI On-Demand Anodyne HRH3 17 41 O=S(=O)(NC[C@H]1CN(Cc2ccccc2)CCO1)c1ccc(-c2ccccc2)cc1 ZINC000147155819 HH On-Demand Anodyne DRD4 29 53 CC(=O)c1sc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)nc1-c1ccccc1 ZINC000147155839 GI On-Demand Bother DHODH 18 41 CC(C)(C)OC(=O)N1CC[C@@H](S(=O)(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000147155956 FD For-Sale Anodyne GPR119 37 41 CC(C)(C)OC(=O)N1CC[C@@H](S(=O)(=O)c2ccc3c(c2)CC(=O)N3)C1 ZINC000147155956 FD For-Sale Anodyne SFRP1 57 38 Cc1cc(N2CCOCC2)ccc1NC(=O)NC[C@H]1CCCO[C@H]1c1ccccc1 ZINC000147155960 HI On-Demand Anodyne HRH3 17 41 C[C@@H]1CCCCN1S(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147156010 GF On-Demand Mild L3MBTL3 86 49 CS(=O)(=O)c1cc(C(=O)NCCc2cccc(Cl)c2Cl)cc([N+](=O)[O-])c1 ZINC000147156039 HG On-Demand Bother NQO2 31 45 O=C(NC1CCN(S(=O)(=O)N2CCCCC2)CC1)c1ccoc1 ZINC000147156150 ED On-Demand Anodyne EPHX2 28 42 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne MME 74 39 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne ANPEP 65 37 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne FCER2 43 34 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne CTSB 44 37 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne PAPA1_CARPA 60 41 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne CYSP_TRYCR 47 34 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne TIMP3 70 37 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne CAPNS1 59 41 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne MMP3 20 51 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne CAPN1 67 41 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne MMP9 22 42 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne CAPN2 52 38 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne ACE2 80 39 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne MMP1 19 42 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne FPR1 42 36 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne CTRB_BOVIN 50 35 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne NPR 43 48 CCc1ncc(C(=O)N[C@@H](Cc2ccccc2)C(=O)OC)s1 ZINC000147156185 DE On-Demand Anodyne BLA1_STEMA 53 41 C[C@H]1CCCCN1S(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147156193 GF On-Demand Mild L3MBTL3 86 49 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne F10 30 40 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne UGCG 37 46 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne TRPV1 15 41 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne COLA 56 38 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne CPT1A 54 38 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne CPT2 42 32 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne JAK1 15 48 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne KDR 28 41 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne GRM4 69 46 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne MET 17 46 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne TYK2 17 46 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne CSF1R 21 40 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne NR2E3 53 33 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne GPBAR1 15 43 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne SHH 31 42 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne SMO 24 40 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne Q25615_ONCVO 31 40 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne KCNK3 56 35 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne KCNK9 52 33 NC(=O)Nc1ccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)cc1 ZINC000147156243 HJ On-Demand Anodyne G2YM83_BOTF4 51 32 CC(C)c1ccc(C(=O)N2CCCC2)cn1 ZINC000147156246 BE On-Demand Anodyne HRH3 0 45 CC(C)c1ccc(C(=O)N2CCCC2)cn1 ZINC000147156246 BE On-Demand Anodyne MLYCD 18 41 CC(C)c1ccc(C(=O)N2CCCC2)cn1 ZINC000147156246 BE On-Demand Anodyne L3MBTL1 0 48 CC(C)c1ccc(C(=O)N2CCCC2)cn1 ZINC000147156246 BE On-Demand Anodyne L3MBTL3 74 41 CC(C)c1ccc(C(=O)N2CCCC2)cn1 ZINC000147156246 BE On-Demand Anodyne MBTD1 0 40 CC(C)c1ccc(C(=O)N2CCCC2)cn1 ZINC000147156246 BE On-Demand Anodyne HPGD 50 43 Cc1cc(Cl)c2cccc(S(=O)(=O)NC(C)C)c2n1 ZINC000147156342 CF For-Sale Anodyne MTNN 47 31 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother PRSS1 15 41 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother MME 53 35 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother ANPEP 61 35 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother TACR1 18 47 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CTSD 21 40 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CTSB 54 38 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother PAPA1_CARPA 50 44 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CYSP_TRYCR 45 34 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CTSK 15 44 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CTSL 39 46 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CACNA1D 69 38 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CCR3 30 62 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother PYGL 16 45 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CAPNS1 55 39 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother HLA-DRB1 42 33 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CTSS 30 46 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CAPN1 52 38 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother ACE2 51 34 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother BACE1 20 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CTSV 42 46 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother CTRB_BOVIN 51 36 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother PLM1_PLAFA 41 33 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother NPR 37 54 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother BLA1_STEMA 67 42 COC(=O)[C@H](Cc1ccccc1)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147156370 EE On-Demand Bother ERAP2 41 38 COC(=O)c1ccc(C)c(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147156616 EG On-Demand Bother CACNA1D 45 34 COC(=O)c1ccc(C)c(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147156616 EG On-Demand Bother PYGL 0 48 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne DRD4 18 41 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne ACHE 18 47 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne LTA4H 67 51 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne ADORA2B 45 43 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne HRH3 26 43 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne CHEK2 34 42 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne CCR3 41 39 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne MLNR 50 33 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne ACR 45 34 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne MCHR1 50 44 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne HIF1A 21 40 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne NPFFR1 40 37 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne NOD1 29 40 CC1CCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147156697 GG On-Demand Anodyne NOD2 47 45 N#CC1CCN(C(=O)C2CCN(c3ccccc3[N+](=O)[O-])CC2)CC1 ZINC000147156718 EF On-Demand Mild SSTR1 27 41 COC(=O)CCc1nc(-c2ccccc2)c(-c2ccccc2)[nH]1 ZINC000147156767 DH For-Sale Clean FABP4 20 40 COC(=O)CCc1nc(-c2ccccc2)c(-c2ccccc2)[nH]1 ZINC000147156767 DH For-Sale Clean SOAT1 63 43 CN(CC(=O)Nc1ccccc1)C(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147156806 GF On-Demand Anodyne DRTS_PLAFK 19 40 CN(CC(=O)Nc1ccccc1)C(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147156806 GF On-Demand Anodyne PTGER3 32 47 COCCNC(=O)c1ccc(C(C)C)nc1 ZINC000147156807 BD On-Demand Anodyne EPHX2 0 41 CC(C)N(C)S(=O)(=O)c1ccc(Cl)c(C(=O)N2CCC(C#N)CC2)c1 ZINC000147156937 GF On-Demand Mild CCR3 15 40 CCOCCCNC(=O)c1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147156973 HG On-Demand Bother DRD4 44 34 CCOCCCNC(=O)c1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147156973 HG On-Demand Bother TAAR1 39 50 CCOCCCNC(=O)c1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147156973 HG On-Demand Bother AKR1C3 18 46 CCOCCCNC(=O)c1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147156973 HG On-Demand Bother KCNK3 74 44 CCOCCCNC(=O)c1cccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147156973 HG On-Demand Bother KCNK9 60 37 CCOC(=O)NCC(=O)N(C)CC(=O)Nc1ccccc1 ZINC000147157031 CC On-Demand Anodyne CA4 23 40 N#CC1CCN(C(=O)CCc2ccc(-c3ccccc3)o2)CC1 ZINC000147157148 DH On-Demand Mild CYP2E1 16 40 NC(=O)c1ccc(OCC(=O)NCc2ccc(N3CCCCCC3)nc2)cc1 ZINC000147157187 GE On-Demand Anodyne SMO 15 42 CCOCCCNC(=O)c1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147157196 HG On-Demand Anodyne MAPK10 15 40 CCOCCCNC(=O)c1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147157196 HG On-Demand Anodyne KCNK3 49 38 Cc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1C(F)(F)F ZINC000147157305 EF On-Demand Anodyne DHODH 30 42 O=C(NCCCCOCCc1ccccc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147157393 FJ On-Demand Anodyne SLC6A1 19 41 O=C(NCCCCOCCc1ccccc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147157393 FJ On-Demand Anodyne SCN5A 15 42 C[C@@H](c1nc(-c2ccccc2)no1)N1CCN(C(=O)CCNS(C)(=O)=O)CC1 ZINC000147157407 HC On-Demand Anodyne PTAFR 40 43 C[C@@H](c1nc(-c2ccccc2)no1)N1CCN(C(=O)CCNS(C)(=O)=O)CC1 ZINC000147157407 HC On-Demand Anodyne ETHR 43 41 CC(=O)C(C)(C)Cn1cncn1 ZINC000147157408 AC For-Sale Anodyne HIS3 72 40 CC(=O)C(C)(C)Cn1cncn1 ZINC000147157408 AC For-Sale Anodyne CYP51 0 41 CC(=O)C(C)(C)Cn1cncn1 ZINC000147157408 AC For-Sale Anodyne CYP51B 43 39 CC(=O)C(C)(C)Cn1cncn1 ZINC000147157408 AC For-Sale Anodyne CYP74A 57 33 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2C(=O)NC2CC2)cc1 ZINC000147157430 EC On-Demand Anodyne CPT1A 112 46 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2C(=O)NC2CC2)cc1 ZINC000147157430 EC On-Demand Anodyne CPT2 52 41 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2C(=O)NC2CC2)cc1 ZINC000147157430 EC On-Demand Anodyne LGMN 61 34 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2C(=O)NC2CC2)cc1 ZINC000147157430 EC On-Demand Anodyne PLAU 28 41 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2C(=O)NC2CC2)cc1 ZINC000147157430 EC On-Demand Anodyne ST14 32 41 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2C(=O)NC2CC2)cc1 ZINC000147157430 EC On-Demand Anodyne TMPRSS11D 56 35 Cc1nn(C(F)F)c(C)c1CC(=O)Nc1ccc(NC(=O)NCc2ccco2)cc1 ZINC000147157470 HH On-Demand Anodyne P2RX7 40 43 Cc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1C(F)(F)F ZINC000147157474 EF On-Demand Anodyne DHODH 30 42 C[C@H](NC(=O)/C=C/c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147157491 DD On-Demand Mild HDAC6 22 40 C[C@H](c1nc(-c2ccccc2)no1)N1CCN(C(=O)CCNS(C)(=O)=O)CC1 ZINC000147157566 HC On-Demand Anodyne PTAFR 40 43 C[C@H](c1nc(-c2ccccc2)no1)N1CCN(C(=O)CCNS(C)(=O)=O)CC1 ZINC000147157566 HC On-Demand Anodyne ETHR 43 41 O=C(NCCCCOCCc1ccccc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147157567 FJ On-Demand Anodyne SLC6A1 19 41 O=C(NCCCCOCCc1ccccc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147157567 FJ On-Demand Anodyne SCN5A 15 42 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2C(=O)NC2CC2)cc1 ZINC000147157612 EC On-Demand Anodyne COLA 130 51 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2C(=O)NC2CC2)cc1 ZINC000147157612 EC On-Demand Anodyne CPT1A 112 46 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2C(=O)NC2CC2)cc1 ZINC000147157612 EC On-Demand Anodyne CPT2 52 41 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2C(=O)NC2CC2)cc1 ZINC000147157612 EC On-Demand Anodyne LGMN 61 34 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2C(=O)NC2CC2)cc1 ZINC000147157612 EC On-Demand Anodyne PLAU 28 41 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2C(=O)NC2CC2)cc1 ZINC000147157612 EC On-Demand Anodyne ST14 32 41 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2C(=O)NC2CC2)cc1 ZINC000147157612 EC On-Demand Anodyne TMPRSS11D 56 35 C[C@@H](NC(=O)/C=C/c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147157678 DD On-Demand Mild HDAC6 22 40 O=C1NC(=O)c2ccccc2/C1=C/Nc1cc(Cl)c([N+](=O)[O-])cc1O ZINC000147157693 FF On-Demand Anodyne CDK4 57 52 CC1(C)CNC(=O)c2cc3ccc(C(=O)Nc4cnc5ccccc5c4)nc3n2C1 ZINC000147157702 GH Annotated Anodyne RPS6KA3 60 53 O=C(NCCCCOCCc1ccccc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147157708 FJ On-Demand Anodyne SLC6A1 19 41 O=C(NCCCCOCCc1ccccc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147157708 FJ On-Demand Anodyne SCN5A 15 42 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147157738 FI On-Demand Anodyne EPHX2 23 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2c(C)cc(Br)cc2Cl)c1 ZINC000147157745 GJ On-Demand Bother TAAR1 24 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2c(C)cc(Br)cc2Cl)c1 ZINC000147157745 GJ On-Demand Bother GPR35 31 40 CCCOC(=O)c1ccc(NC(=O)c2csc(COC)n2)cc1 ZINC000147157793 EG On-Demand Anodyne ACR 42 31 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](C)NC(=O)CCCCCCCCCCCCCCCCCCCCCCCCC ZINC000147157885 KK Annotated Mild CNR1 21 50 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](C)NC(=O)CCCCCCCCCCCCCCCCCCCCCCCCC ZINC000147157885 KK Annotated Mild FABP4 18 47 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](C)NC(=O)CCCCCCCCCCCCCCCCCCCCCCCCC ZINC000147157885 KK Annotated Mild LPAR1 34 43 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](C)NC(=O)CCCCCCCCCCCCCCCCCCCCCCCCC ZINC000147157885 KK Annotated Mild SELP 35 42 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](C)NC(=O)CCCCCCCCCCCCCCCCCCCCCCCCC ZINC000147157885 KK Annotated Mild FAAH 19 56 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](C)NC(=O)CCCCCCCCCCCCCCCCCCCCCCCCC ZINC000147157885 KK Annotated Mild LPAR3 61 38 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](C)NC(=O)CCCCCCCCCCCCCCCCCCCCCCCCC ZINC000147157885 KK Annotated Mild FABP3 37 47 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](C)NC(=O)CCCCCCCCCCCCCCCCCCCCCCCCC ZINC000147157885 KK Annotated Mild FABP5 15 47 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](C)NC(=O)CCCCCCCCCCCCCCCCCCCCCCCCC ZINC000147157885 KK Annotated Mild FABP1 15 47 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](C)NC(=O)CCCCCCCCCCCCCCCCCCCCCCCCC ZINC000147157885 KK Annotated Mild NOD1 101 50 CCCCCCCCCCCCC/C=C/[C@@H](O)[C@H](C)NC(=O)CCCCCCCCCCCCCCCCCCCCCCCCC ZINC000147157885 KK Annotated Mild CQSS 63 42 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne PPIA 25 41 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne UGCG 36 45 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne CPT1A 43 31 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne KDR 29 40 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne GRM4 63 44 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne MET 15 41 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne TYK2 33 44 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne CSF1R 22 43 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne TAAR1 15 41 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne GPBAR1 18 41 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne SHH 20 41 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne KCNK3 119 44 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne KCNK9 88 42 NC(=O)Nc1cccc(NC(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)c1 ZINC000147157886 HJ On-Demand Anodyne G2YM83_BOTF4 65 33 O=C(NCCCCOCCc1ccccc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147157902 FJ On-Demand Anodyne SLC6A1 19 41 O=C(NCCCCOCCc1ccccc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147157902 FJ On-Demand Anodyne SCN5A 15 42 CN(C)c1ccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147157939 FI On-Demand Anodyne EPHX2 23 42 CC(C)Oc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147157957 EJ On-Demand Mild ADRB1 40 32 CC(C)Oc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147157957 EJ On-Demand Mild AR 63 48 CC(C)Oc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147157957 EJ On-Demand Mild MTTP 55 38 CC(C)Oc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147157957 EJ On-Demand Mild S1PR1 24 50 CC(C)Oc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147157957 EJ On-Demand Mild TAAR1 28 42 CC(C)Oc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147157957 EJ On-Demand Mild IMDH_CRYPV 15 50 CC(C)Oc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147157957 EJ On-Demand Mild KCNK3 82 59 CC(C)Oc1ccccc1C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1 ZINC000147157957 EJ On-Demand Mild KCNK9 77 59 Cn1cc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1C(N)=O ZINC000147157964 GC On-Demand Anodyne EPHX2 15 40 CN(C)c1ccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147158124 FI On-Demand Anodyne EPHX2 23 42 CCCCCCNC(=O)N1[C@@H](C)CC[C@@H]1C ZINC000147158259 BG On-Demand Anodyne EPHX2 50 42 CCCCCCNC(=O)N1[C@@H](C)CC[C@@H]1C ZINC000147158259 BG On-Demand Anodyne GNAI1 0 48 CCCCCCNC(=O)N1[C@@H](C)CC[C@@H]1C ZINC000147158259 BG On-Demand Anodyne GNAI3 0 48 CCCCCCNC(=O)N1[C@@H](C)CC[C@@H]1C ZINC000147158259 BG On-Demand Anodyne GNAO1 0 48 CCCCCCNC(=O)N1[C@@H](C)CC[C@@H]1C ZINC000147158259 BG On-Demand Anodyne ASAH1 95 44 CN(C)c1ccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147158299 FI On-Demand Anodyne EPHX2 23 42 Cc1cc[nH]c1CCC(=O)O ZINC000147158386 AD For-Sale Anodyne FFAR1 41 38 CCCCCCNC(=O)N1[C@@H](C)CC[C@H]1C ZINC000147158454 BG On-Demand Anodyne EPHX2 50 42 CCCCCCNC(=O)N1[C@@H](C)CC[C@H]1C ZINC000147158454 BG On-Demand Anodyne GNAI1 0 48 CCCCCCNC(=O)N1[C@@H](C)CC[C@H]1C ZINC000147158454 BG On-Demand Anodyne GNAI3 0 48 CCCCCCNC(=O)N1[C@@H](C)CC[C@H]1C ZINC000147158454 BG On-Demand Anodyne GNAO1 0 48 CCCCCCNC(=O)N1[C@@H](C)CC[C@H]1C ZINC000147158454 BG On-Demand Anodyne ASAH1 95 44 N#Cc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1Cl ZINC000147158461 DD On-Demand Mild DHODH 17 43 N#Cc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1Cl ZINC000147158461 DD On-Demand Mild ENV 43 35 Cc1cc(CNC(=O)Nc2cc(C(C)(C)C)nn2-c2cccc(Cl)c2)no1 ZINC000147158495 GI On-Demand Anodyne TNF 45 40 Cc1cc(CNC(=O)Nc2cc(C(C)(C)C)nn2-c2cccc(Cl)c2)no1 ZINC000147158495 GI On-Demand Anodyne MAPK14 36 55 Cc1cc(CNC(=O)Nc2cc(C(C)(C)C)nn2-c2cccc(Cl)c2)no1 ZINC000147158495 GI On-Demand Anodyne PTK2B 35 44 Cc1cc(CNC(=O)Nc2cc(C(C)(C)C)nn2-c2cccc(Cl)c2)no1 ZINC000147158495 GI On-Demand Anodyne CARM1 41 36 Cc1cc(CNC(=O)Nc2cc(C(C)(C)C)nn2-c2cccc(Cl)c2)no1 ZINC000147158495 GI On-Demand Anodyne DDR2 42 56 CCCCCCNC(=O)N1[C@H](C)CC[C@H]1C ZINC000147158651 BG On-Demand Anodyne EPHX2 50 42 CCCCCCNC(=O)N1[C@H](C)CC[C@H]1C ZINC000147158651 BG On-Demand Anodyne GNAI1 0 48 CCCCCCNC(=O)N1[C@H](C)CC[C@H]1C ZINC000147158651 BG On-Demand Anodyne GNAI3 0 48 CCCCCCNC(=O)N1[C@H](C)CC[C@H]1C ZINC000147158651 BG On-Demand Anodyne GNAO1 0 48 CCCCCCNC(=O)N1[C@H](C)CC[C@H]1C ZINC000147158651 BG On-Demand Anodyne ASAH1 95 44 N#Cc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1Cl ZINC000147158655 DD On-Demand Mild DHODH 17 43 N#Cc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1Cl ZINC000147158655 DD On-Demand Mild ENV 43 35 Cc1cc(CNC(=O)Nc2cc(C(C)(C)C)nn2-c2ccccc2C)no1 ZINC000147158698 FI On-Demand Anodyne TNF 44 38 Cc1cc(CNC(=O)Nc2cc(C(C)(C)C)nn2-c2ccccc2C)no1 ZINC000147158698 FI On-Demand Anodyne MAPK14 32 55 Cc1cc(CNC(=O)Nc2cc(C(C)(C)C)nn2-c2ccccc2C)no1 ZINC000147158698 FI On-Demand Anodyne PTK2B 33 40 Cc1cc(CNC(=O)Nc2cc(C(C)(C)C)nn2-c2ccccc2C)no1 ZINC000147158698 FI On-Demand Anodyne DDR2 36 44 Cc1ccccc1-n1nc(C(=O)Nc2cccc(NC(N)=O)c2)c2c1CCC2 ZINC000147158778 GG On-Demand Anodyne KCNK3 108 40 Cc1ccccc1-n1nc(C(=O)Nc2cccc(NC(N)=O)c2)c2c1CCC2 ZINC000147158778 GG On-Demand Anodyne KCNK9 69 38 Cc1cccnc1-c1ccn2c(-c3cccc(NC(=O)NCC(F)(F)F)c3)cnc2c1 ZINC000147158789 IK Annotated Anodyne BRAF 52 38 COc1ccc2c(c1)OC[C@H](C(=O)NCCCCOCCc1ccccc1)C2 ZINC000147158817 GG On-Demand Anodyne NQO2 28 40 COc1ccc2c(c1)OC[C@H](C(=O)NCCCCOCCc1ccccc1)C2 ZINC000147158817 GG On-Demand Anodyne MTNR1A 86 42 COc1ccc2c(c1)OC[C@H](C(=O)NCCCCOCCc1ccccc1)C2 ZINC000147158817 GG On-Demand Anodyne MTNR1B 84 42 COc1ccccc1Oc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147158850 GG On-Demand Anodyne PDGFRA 49 38 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147158973 DD On-Demand Anodyne HDAC10 47 39 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147158973 DD On-Demand Anodyne MMP2 17 45 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147158973 DD On-Demand Anodyne MMP3 33 44 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147158973 DD On-Demand Anodyne HDAC1 16 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147158973 DD On-Demand Anodyne FURIN 45 35 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147158973 DD On-Demand Anodyne HDAC11 47 39 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147158973 DD On-Demand Anodyne S1PR5 16 42 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147158973 DD On-Demand Anodyne POLG_WNV 65 32 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147158973 DD On-Demand Anodyne KCNK3 50 33 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147158973 DD On-Demand Anodyne KCNK9 47 33 CC(=O)c1ccc(S(=O)(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)cc1 ZINC000147158988 HE On-Demand Mild EPHX2 20 54 CC(=O)c1ccc(S(=O)(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)cc1 ZINC000147158988 HE On-Demand Mild TGM2 53 44 CC(=O)c1ccc(S(=O)(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)cc1 ZINC000147158988 HE On-Demand Mild F13A1 52 44 CC(=O)c1ccc(S(=O)(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)cc1 ZINC000147158988 HE On-Demand Mild NAMPT 22 47 Cc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147159008 HE On-Demand Bother TGM2 44 37 Cc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147159008 HE On-Demand Bother F13A1 56 37 COc1ccc2c(c1)OC[C@@H](C(=O)NCCCCOCCc1ccccc1)C2 ZINC000147159012 GG On-Demand Anodyne NQO2 28 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCCCCOCCc1ccccc1)C2 ZINC000147159012 GG On-Demand Anodyne MTNR1A 86 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCCCCOCCc1ccccc1)C2 ZINC000147159012 GG On-Demand Anodyne MTNR1B 84 42 COc1ccccc1Oc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147159047 GG On-Demand Anodyne PDGFRA 49 38 CN(C)[C@H]1CCN(Cc2ccc(C(N)=O)cc2)C1 ZINC000147159096 BC On-Demand Anodyne LTA4H 17 47 CN(C)[C@H]1CCN(Cc2ccc(C(N)=O)cc2)C1 ZINC000147159096 BC On-Demand Anodyne SIGMAR1 35 42 CN(C)[C@H]1CCN(Cc2ccc(C(N)=O)cc2)C1 ZINC000147159096 BC On-Demand Anodyne CCR3 23 40 CN(C)[C@H]1CCN(Cc2ccc(C(N)=O)cc2)C1 ZINC000147159096 BC On-Demand Anodyne CCR5 25 40 CN(C)[C@H]1CCN(Cc2ccc(C(N)=O)cc2)C1 ZINC000147159096 BC On-Demand Anodyne UTS2R 15 43 CN(C)[C@H]1CCN(Cc2ccc(C(N)=O)cc2)C1 ZINC000147159096 BC On-Demand Anodyne SLC18A3 17 41 CN(C)[C@H]1CCN(Cc2ccc(C(N)=O)cc2)C1 ZINC000147159096 BC On-Demand Anodyne MLNR 56 40 CN(C)[C@H]1CCN(Cc2ccc(C(N)=O)cc2)C1 ZINC000147159096 BC On-Demand Anodyne LSS 21 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147159168 DD On-Demand Anodyne HDAC10 47 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147159168 DD On-Demand Anodyne MMP2 17 45 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147159168 DD On-Demand Anodyne MMP3 33 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147159168 DD On-Demand Anodyne HDAC1 16 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147159168 DD On-Demand Anodyne FURIN 45 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147159168 DD On-Demand Anodyne HDAC11 47 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147159168 DD On-Demand Anodyne S1PR5 16 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147159168 DD On-Demand Anodyne POLG_WNV 65 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147159168 DD On-Demand Anodyne KCNK3 50 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(N)=O)c1 ZINC000147159168 DD On-Demand Anodyne KCNK9 47 33 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N(C)C ZINC000147159175 FD On-Demand Mild L3MBTL3 56 37 Cc1ccc(Cl)cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147159197 GF On-Demand Anodyne CNR1 20 48 Cc1ccc(Cl)cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147159197 GF On-Demand Anodyne CNR2 26 56 Cc1ccc(Cl)cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147159197 GF On-Demand Anodyne CPT2 41 34 Cc1ccc(Cl)cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147159197 GF On-Demand Anodyne MAPK13 68 33 Cc1ccc(Cl)cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147159197 GF On-Demand Anodyne EPHX2 42 44 Cc1ccc(Cl)cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147159197 GF On-Demand Anodyne TGM2 34 40 O=C(NCCCCOCCc1ccccc1)c1ccc2c(c1)COC2 ZINC000147159230 EG On-Demand Anodyne KDM4E 21 41 C=CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147159394 ED On-Demand Mild ST14 72 33 C=CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147159394 ED On-Demand Mild SFRP1 46 38 C=CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147159394 ED On-Demand Mild TMPRSS6 50 31 CCOC(=O)c1cc(Cl)c(C#N)cc1OC ZINC000147159496 BE For-Sale Mild HTR4 81 47 CCOC(=O)c1cc(Cl)c(C#N)cc1OC ZINC000147159496 BE For-Sale Mild HSP90AB1 66 33 CNS(=O)(=O)c1cc(C(=O)N2CCC(C#N)CC2)ccc1OC ZINC000147159608 EC On-Demand Mild HRH3 29 42 CNS(=O)(=O)c1cc(C(=O)N2CCC(C#N)CC2)ccc1OC ZINC000147159608 EC On-Demand Mild COLA 46 37 CNS(=O)(=O)c1cc(C(=O)N2CCC(C#N)CC2)ccc1OC ZINC000147159608 EC On-Demand Mild CPT1A 45 37 CNS(=O)(=O)c1cc(C(=O)N2CCC(C#N)CC2)ccc1OC ZINC000147159608 EC On-Demand Mild CPT2 44 33 CNS(=O)(=O)c1cc(C(=O)N2CCC(C#N)CC2)ccc1OC ZINC000147159608 EC On-Demand Mild SLC9A1 15 40 CNS(=O)(=O)c1cc(C(=O)N2CCC(C#N)CC2)ccc1OC ZINC000147159608 EC On-Demand Mild L3MBTL3 58 35 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147159634 HE On-Demand Anodyne EPHX2 36 40 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147159634 HE On-Demand Anodyne SFRP1 58 37 CN(C)c1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147159634 HE On-Demand Anodyne WNT3 43 35 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(SCc2cccnc2)cc1 ZINC000147159652 GF On-Demand Anodyne NAMPT 41 39 Cc1ccc(Oc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cn2)cc1C ZINC000147159653 GH On-Demand Anodyne ADORA2B 41 43 Cc1ccc(Oc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cn2)cc1C ZINC000147159653 GH On-Demand Anodyne HIF1A 28 42 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1C(N)=O ZINC000147159783 GD On-Demand Anodyne MAPK13 47 32 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1C(N)=O ZINC000147159783 GD On-Demand Anodyne EPHX2 29 42 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1C(N)=O ZINC000147159783 GD On-Demand Anodyne TGM2 43 43 CNC(=O)Nc1cccc(NC(=O)c2nn(-c3ccccc3C)c3c2CCC3)c1 ZINC000147159816 GH On-Demand Anodyne KCNK3 104 40 CNC(=O)Nc1cccc(NC(=O)c2nn(-c3ccccc3C)c3c2CCC3)c1 ZINC000147159816 GH On-Demand Anodyne KCNK9 64 38 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147159838 HE On-Demand Anodyne EPHX2 36 40 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147159838 HE On-Demand Anodyne SFRP1 58 37 CN(C)c1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147159838 HE On-Demand Anodyne WNT3 43 35 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(SCc2cccnc2)cc1 ZINC000147159842 GF On-Demand Anodyne NAMPT 41 39 CCOC(=O)c1ncn2c1CSc1ccccc1-2 ZINC000147159917 CF For-Sale Anodyne ELANE 16 40 CN(Cc1cscn1)C(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000147159932 ED On-Demand Anodyne CA2 76 49 CN(Cc1cscn1)C(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000147159932 ED On-Demand Anodyne CA1 57 49 CN(Cc1cscn1)C(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000147159932 ED On-Demand Anodyne CA7 42 47 CN(Cc1cscn1)C(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000147159932 ED On-Demand Anodyne CA5B 39 43 CN(Cc1cscn1)C(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000147159932 ED On-Demand Anodyne CA4 56 45 CN(Cc1cscn1)C(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000147159932 ED On-Demand Anodyne CA5A 40 43 CN(Cc1cscn1)C(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000147159932 ED On-Demand Anodyne CA14 38 47 CN(Cc1cscn1)C(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000147159932 ED On-Demand Anodyne CA12 41 42 CN(Cc1cscn1)C(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000147159932 ED On-Demand Anodyne CA9 51 42 CN(Cc1cscn1)C(=O)NCc1ccc(S(N)(=O)=O)cc1 ZINC000147159932 ED On-Demand Anodyne CYNT 29 43 C[C@@H]1CN(C(=O)Nc2ccc(N(C)C)cc2C(F)(F)F)C[C@H](c2ccccc2)O1 ZINC000147159996 HJ On-Demand Anodyne RBP4 83 42 CCOC(=O)C[C@H](NC(=O)c1ccc2c(c1)COC2)c1cccc(OC)c1 ZINC000147160076 FG On-Demand Anodyne DRD4 41 32 C[C@H]1CN(C(=O)Nc2ccc(N(C)C)cc2C(F)(F)F)C[C@H](c2ccccc2)O1 ZINC000147160175 HJ On-Demand Anodyne RBP4 83 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(=O)n(Cc3ccccc3Cl)c2)c1 ZINC000147160192 HH On-Demand Bother PTGER3 29 45 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(=O)n(Cc3ccccc3Cl)c2)c1 ZINC000147160192 HH On-Demand Bother PDE7A 16 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(=O)n(Cc3ccccc3Cl)c2)c1 ZINC000147160192 HH On-Demand Bother TAAR1 24 43 O=C(NC1CCN(S(=O)(=O)c2cc(F)cc(F)c2)CC1)c1ccoc1 ZINC000147160226 FE On-Demand Anodyne CCR3 15 43 O=C(NC1CCN(S(=O)(=O)c2cc(F)cc(F)c2)CC1)c1ccoc1 ZINC000147160226 FE On-Demand Anodyne EPHX2 23 42 O=C(NC1CCN(S(=O)(=O)c2cc(F)cc(F)c2)CC1)c1ccoc1 ZINC000147160226 FE On-Demand Anodyne TGM2 44 44 O=C(NC1CCN(S(=O)(=O)c2cc(F)cc(F)c2)CC1)c1ccoc1 ZINC000147160226 FE On-Demand Anodyne MCHR1 15 44 C[C@@H]1CN(C(=O)Nc2ccc(N(C)C)cc2C(F)(F)F)C[C@@H](c2ccccc2)O1 ZINC000147160354 HJ On-Demand Anodyne RBP4 83 42 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)NC)c1 ZINC000147160391 DD On-Demand Anodyne HDAC10 44 37 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)NC)c1 ZINC000147160391 DD On-Demand Anodyne MMP3 29 41 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)NC)c1 ZINC000147160391 DD On-Demand Anodyne HDAC11 44 37 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)NC)c1 ZINC000147160391 DD On-Demand Anodyne POLG_WNV 40 30 CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147160465 DD On-Demand Mild ST14 81 36 CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147160465 DD On-Demand Mild SFRP1 65 39 CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147160465 DD On-Demand Mild L3MBTL3 41 40 CCNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147160465 DD On-Demand Mild TMPRSS6 63 35 CCCCNNC(=O)c1ccc(F)cc1 ZINC000147160501 BD Annotated Reactive ASAH1 66 36 O=C(NC1CCN(S(=O)(=O)c2cccc(Cl)c2)CC1)c1ccoc1 ZINC000147160503 FF On-Demand Anodyne TGM2 44 50 O=C(NC1CCN(S(=O)(=O)c2cccc(Cl)c2)CC1)c1ccoc1 ZINC000147160503 FF On-Demand Anodyne AKR1C3 58 41 O=C(O)c1ccc2nc(-n3ccnc3)nc(N3CCOCC3)c2n1 ZINC000147160540 EC For-Sale Anodyne NOS2 70 34 C[C@H]1CN(C(=O)Nc2ccc(N(C)C)cc2C(F)(F)F)C[C@@H](c2ccccc2)O1 ZINC000147160544 HJ On-Demand Anodyne RBP4 83 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)NC)c1 ZINC000147160557 DD On-Demand Anodyne HDAC10 44 37 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)NC)c1 ZINC000147160557 DD On-Demand Anodyne MMP3 29 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)NC)c1 ZINC000147160557 DD On-Demand Anodyne HDAC11 44 37 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)NC)c1 ZINC000147160557 DD On-Demand Anodyne POLG_WNV 40 30 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160570 EG On-Demand Anodyne MME 74 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160570 EG On-Demand Anodyne ANPEP 55 34 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160570 EG On-Demand Anodyne PAPA1_CARPA 41 32 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160570 EG On-Demand Anodyne CTSL 24 43 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160570 EG On-Demand Anodyne SLC15A1 0 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160570 EG On-Demand Anodyne SOAT1 27 45 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160570 EG On-Demand Anodyne ACE2 75 39 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160570 EG On-Demand Anodyne BLA1_STEMA 46 34 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160570 EG On-Demand Anodyne UTS2 49 37 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160570 EG On-Demand Anodyne GPR88 0 44 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne ACE 32 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne MME 64 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne ANPEP 50 34 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne FCER2 80 42 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne PAPA1_CARPA 49 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne CAPNS1 47 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne HLA-DRB1 41 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne MMP9 15 42 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne ACE2 69 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne MMP1 22 42 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne FPR1 45 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@@H](C)c1cccs1 ZINC000147160683 EG On-Demand Anodyne GPR142 81 36 CCn1c(NC(=O)c2ccc3cc4n(c3n2)[C@H](C)CNC4=O)nc2ccccc21 ZINC000147160698 GF Annotated Anodyne MAPKAPK2 15 44 CCn1c(NC(=O)c2ccc3cc4n(c3n2)[C@H](C)CNC4=O)nc2ccccc21 ZINC000147160698 GF Annotated Anodyne RPS6KA3 42 50 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)s1 ZINC000147160726 FE On-Demand Anodyne EPHX2 21 44 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)s1 ZINC000147160726 FE On-Demand Anodyne TGM2 36 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147160755 ED On-Demand Anodyne MAPK14 22 41 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160818 EG On-Demand Anodyne MME 74 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160818 EG On-Demand Anodyne ANPEP 55 34 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160818 EG On-Demand Anodyne PAPA1_CARPA 41 32 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160818 EG On-Demand Anodyne CTSL 24 43 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160818 EG On-Demand Anodyne SLC15A1 0 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160818 EG On-Demand Anodyne SOAT1 27 45 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160818 EG On-Demand Anodyne ACE2 75 39 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160818 EG On-Demand Anodyne BLA1_STEMA 46 34 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160818 EG On-Demand Anodyne UTS2 49 37 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN(C)C)c1ccccc1 ZINC000147160818 EG On-Demand Anodyne GPR88 0 44 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne HTR1A 15 41 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne DRD2 23 41 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne DRD4 41 41 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne ACHE 29 40 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne PPARA 15 48 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne LTA4H 36 43 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne HRH3 21 45 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne SIGMAR1 62 50 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne CACNA1B 17 43 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne FAAH 28 49 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne CACNA1G 35 42 CCc1ccc(O[C@@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147160868 FG On-Demand Anodyne NOD2 41 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne ACE 32 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne MME 64 41 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne ANPEP 50 34 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne FCER2 80 42 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne PAPA1_CARPA 49 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne CAPNS1 47 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne HLA-DRB1 41 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne MMP9 15 42 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne ACE2 69 36 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne MMP1 22 42 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne FPR1 45 35 CC(=O)[C@H](Cc1ccccc1)NC(=O)CN(C)[C@H](C)c1cccs1 ZINC000147160877 EG On-Demand Anodyne GPR142 81 36 O=C(NC1CCN(S(=O)(=O)Cc2ccccc2)CC1)c1ccoc1 ZINC000147160914 EE On-Demand Anodyne DRD4 18 45 O=C(NC1CCN(S(=O)(=O)Cc2ccccc2)CC1)c1ccoc1 ZINC000147160914 EE On-Demand Anodyne PTPN2 44 39 O=C(NC1CCN(S(=O)(=O)Cc2ccccc2)CC1)c1ccoc1 ZINC000147160914 EE On-Demand Anodyne SIGMAR1 20 50 O=C(NC1CCN(S(=O)(=O)Cc2ccccc2)CC1)c1ccoc1 ZINC000147160914 EE On-Demand Anodyne TGM2 45 43 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc(C)cc3)CC2)s1 ZINC000147160918 GE On-Demand Anodyne TGM2 72 40 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc(C)cc3)CC2)s1 ZINC000147160918 GE On-Demand Anodyne F13A1 77 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147160949 ED On-Demand Anodyne MAPK14 22 41 CCOc1ccc(-c2nnc(SCC(=O)Nc3nc(C)cc(C)n3)[nH]2)cc1 ZINC000147160961 GG Annotated Anodyne ADORA2B 41 36 CCOc1ccc(-c2nnc(SCC(=O)Nc3nc(C)cc(C)n3)[nH]2)cc1 ZINC000147160961 GG Annotated Anodyne ENPP1 79 41 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161007 EG On-Demand Anodyne MME 74 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161007 EG On-Demand Anodyne ANPEP 55 34 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161007 EG On-Demand Anodyne PAPA1_CARPA 41 32 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161007 EG On-Demand Anodyne CTSL 24 43 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161007 EG On-Demand Anodyne SLC15A1 0 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161007 EG On-Demand Anodyne SOAT1 27 45 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161007 EG On-Demand Anodyne ACE2 75 39 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161007 EG On-Demand Anodyne BLA1_STEMA 46 34 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161007 EG On-Demand Anodyne UTS2 49 37 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161007 EG On-Demand Anodyne GPR88 0 44 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne HTR1A 15 41 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne DRD2 23 41 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne DRD4 41 41 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne ACHE 29 40 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne PPARA 15 48 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne LTA4H 36 43 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne HRH3 21 45 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne SIGMAR1 62 50 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne CACNA1B 17 43 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne FAAH 28 49 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne CACNA1G 35 42 CCc1ccc(O[C@H](C)C(=O)N2CCN(Cc3ccccc3)CC2)cc1 ZINC000147161066 FG On-Demand Anodyne NOD2 41 36 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)s1 ZINC000147161098 HG On-Demand Anodyne F2 19 43 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)s1 ZINC000147161098 HG On-Demand Anodyne F10 15 45 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)s1 ZINC000147161098 HG On-Demand Anodyne TRY2_BOVIN 68 43 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)s1 ZINC000147161098 HG On-Demand Anodyne PKM 19 45 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)s1 ZINC000147161098 HG On-Demand Anodyne TGM2 55 34 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)s1 ZINC000147161098 HG On-Demand Anodyne F13A1 57 39 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc4ccccc4c3)CC2)s1 ZINC000147161098 HG On-Demand Anodyne AKR1C3 20 44 COC(=O)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147161114 GD On-Demand Anodyne UTS2R 15 42 COC(=O)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147161114 GD On-Demand Anodyne EPHX2 23 49 COC(=O)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147161114 GD On-Demand Anodyne TGM2 55 49 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161207 EG On-Demand Anodyne MME 74 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161207 EG On-Demand Anodyne ANPEP 55 34 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161207 EG On-Demand Anodyne PAPA1_CARPA 41 32 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161207 EG On-Demand Anodyne CTSL 24 43 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161207 EG On-Demand Anodyne SLC15A1 0 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161207 EG On-Demand Anodyne SOAT1 27 45 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161207 EG On-Demand Anodyne ACE2 75 39 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161207 EG On-Demand Anodyne BLA1_STEMA 46 34 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161207 EG On-Demand Anodyne UTS2 49 37 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN(C)C)c1ccccc1 ZINC000147161207 EG On-Demand Anodyne GPR88 0 44 CC(C)NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147161308 ED On-Demand Mild L3MBTL3 75 41 CCC[C@@H](O)c1cccc(N(C)C)c1 ZINC000147161366 AF For-Sale Anodyne KYNU 43 30 CCC[C@@H](O)c1cccc(N(C)C)c1 ZINC000147161366 AF For-Sale Anodyne AOC3 22 41 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161457 GI In-Stock Anodyne AR 0 47 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161457 GI In-Stock Anodyne NR1I3 0 44 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161457 GI In-Stock Anodyne SHBG 25 46 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161457 GI In-Stock Anodyne SMT1 0 40 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161457 GI In-Stock Anodyne GPBAR1 0 47 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161457 GI In-Stock Anodyne G6PD 0 47 N#CC1CCN(C(=O)CCS(=O)(=O)c2ccc3c(c2)OCCO3)CC1 ZINC000147161501 FD On-Demand Mild PKM 32 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2cc(F)ccc2OC)c1 ZINC000147161506 EG On-Demand Bother AKR1C2 32 40 CCC[C@H](O)c1cccc(N(C)C)c1 ZINC000147161560 AF For-Sale Anodyne KYNU 43 30 CCC[C@H](O)c1cccc(N(C)C)c1 ZINC000147161560 AF For-Sale Anodyne AOC3 22 41 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161658 GI In-Stock Anodyne AR 23 47 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161658 GI In-Stock Anodyne NR1I3 0 44 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161658 GI In-Stock Anodyne SHBG 25 46 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161658 GI In-Stock Anodyne CYP17A1 15 46 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161658 GI In-Stock Anodyne SMT1 0 40 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161658 GI In-Stock Anodyne GPBAR1 24 47 Cn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)cn1 ZINC000147161658 GI In-Stock Anodyne G6PD 0 47 CN1CCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)nc2)CC1 ZINC000147161706 FC On-Demand Anodyne PRNP 42 43 CN1CCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)nc2)CC1 ZINC000147161706 FC On-Demand Anodyne HIF1A 27 44 CN1CCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)nc2)CC1 ZINC000147161706 FC On-Demand Anodyne STAT6 26 40 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2cc(F)ccc2OC)c1 ZINC000147161714 EG On-Demand Bother AKR1C2 32 40 C[C@@H]1CNC(=O)c2cc3ccc(C(=O)Nc4nc5ccccc5n4CCCN(C)C)nc3n21 ZINC000147161860 IF Annotated Anodyne RPS6KA3 30 67 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147161878 HJ In-Stock Anodyne ESR1 34 53 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147161878 HJ In-Stock Anodyne CYP11A1 0 46 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147161878 HJ In-Stock Anodyne AR 29 53 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147161878 HJ In-Stock Anodyne ESR2 39 53 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147161878 HJ In-Stock Anodyne SHBG 22 50 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147161878 HJ In-Stock Anodyne DHCR7 0 43 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147161878 HJ In-Stock Anodyne CYP17A1 59 52 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147161878 HJ In-Stock Anodyne CYP125 0 43 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147161878 HJ In-Stock Anodyne RORC 0 45 COc1ncccc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147161910 DD On-Demand Anodyne ADORA2B 22 40 COc1ncccc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147161910 DD On-Demand Anodyne HIF1A 21 41 Cc1cc(N2CCCC2)ccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147161933 EE On-Demand Anodyne HRH3 18 44 C=CCNC(=O)Nc1ccc(NC(=O)c2ccn(-c3cc(C)ccc3OC)n2)cc1 ZINC000147161956 HH On-Demand Mild ENPP1 55 30 CC(C)[C@](C)(O)Cn1cncn1 ZINC000147161994 AC For-Sale Anodyne HIS3 41 37 CC(C)[C@](C)(O)Cn1cncn1 ZINC000147161994 AC For-Sale Anodyne CYP51 0 48 CC(C)[C@](C)(O)Cn1cncn1 ZINC000147161994 AC For-Sale Anodyne CYP121 0 42 CC(C)[C@](C)(O)Cn1cncn1 ZINC000147161994 AC For-Sale Anodyne CYP51B 0 42 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147162044 HJ In-Stock Anodyne ESR1 34 53 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147162044 HJ In-Stock Anodyne CYP11A1 0 46 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147162044 HJ In-Stock Anodyne AR 29 53 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147162044 HJ In-Stock Anodyne ESR2 39 53 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147162044 HJ In-Stock Anodyne SHBG 22 50 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147162044 HJ In-Stock Anodyne DHCR7 0 43 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147162044 HJ In-Stock Anodyne CYP17A1 59 52 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147162044 HJ In-Stock Anodyne CYP125 0 43 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@H]1O ZINC000147162044 HJ In-Stock Anodyne RORC 0 45 C[C@@H]1CCNC(=O)c2cc3ccc(C(=O)Nc4nc5ccccc5n4CCCN(C)C)nc3n21 ZINC000147162066 JG Annotated Anodyne ITK 40 38 C[C@@H]1CCNC(=O)c2cc3ccc(C(=O)Nc4nc5ccccc5n4CCCN(C)C)nc3n21 ZINC000147162066 JG Annotated Anodyne RPS6KA3 48 78 O=C(NC1CCN(S(=O)(=O)N2CCCCCC2)CC1)c1ccoc1 ZINC000147162072 FD On-Demand Anodyne EPHX2 28 42 CC(C)CCO[C@@H](C)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147162114 GD On-Demand Mild TGM2 42 36 CC(C)CCO[C@@H](C)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147162114 GD On-Demand Mild F13A1 54 36 CC(C)(C)OC(=O)NC1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147162141 GD On-Demand Anodyne CPT1A 40 42 CC(C)(C)OC(=O)NC1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147162141 GD On-Demand Anodyne PLAU 19 40 CC(C)(C)OC(=O)NC1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147162141 GD On-Demand Anodyne GPR119 17 45 Cc1cc(N2CCCC2)ccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147162154 EE On-Demand Anodyne HRH3 18 44 CC(C)[C@@](C)(O)Cn1cncn1 ZINC000147162175 AC For-Sale Anodyne HIS3 41 37 CC(C)[C@@](C)(O)Cn1cncn1 ZINC000147162175 AC For-Sale Anodyne CYP51 0 48 CC(C)[C@@](C)(O)Cn1cncn1 ZINC000147162175 AC For-Sale Anodyne CYP121 0 42 CC(C)[C@@](C)(O)Cn1cncn1 ZINC000147162175 AC For-Sale Anodyne CYP51B 0 42 Cc1cc(C(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147162203 GE On-Demand Bother TGM2 56 35 Cc1cc(C(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147162203 GE On-Demand Bother F13A1 72 37 Cc1cc(C(=O)N2CCN(S(=O)(=O)c3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147162203 GE On-Demand Bother AKR1C3 58 42 C[C@H]1CCNC(=O)c2cc3ccc(C(=O)Nc4nc5ccccc5n4CCCN(C)C)nc3n21 ZINC000147162277 JG Annotated Anodyne ITK 40 38 C[C@H]1CCNC(=O)c2cc3ccc(C(=O)Nc4nc5ccccc5n4CCCN(C)C)nc3n21 ZINC000147162277 JG Annotated Anodyne RPS6KA3 48 78 Cc1nn(C)cc1/C=C1\C[C@H]2[C@@H]3CC[C@@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147162282 GI In-Stock Anodyne NR1I3 0 43 Cc1nn(C)cc1/C=C1\C[C@H]2[C@@H]3CC[C@@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147162282 GI In-Stock Anodyne SHBG 25 45 Cc1nn(C)cc1/C=C1\C[C@H]2[C@@H]3CC[C@@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147162282 GI In-Stock Anodyne GPBAR1 0 45 Cc1nn(C)cc1/C=C1\C[C@H]2[C@@H]3CC[C@@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147162282 GI In-Stock Anodyne G6PD 0 45 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147162283 HD On-Demand Anodyne F2 21 40 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147162283 HD On-Demand Anodyne PCSK5 56 36 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147162283 HD On-Demand Anodyne FURIN 76 36 CCCC[C@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147162283 HD On-Demand Anodyne POLG_WNV 73 32 CC(C)CCO[C@H](C)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147162310 GD On-Demand Mild TGM2 42 36 CC(C)CCO[C@H](C)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147162310 GD On-Demand Mild F13A1 54 36 COc1cc(NC(N)=S)cc(-c2ccccc2)c1 ZINC000147162317 CG For-Sale Anodyne PPO2 22 43 N#CC1CCN(C(=O)C2CCN(c3ccc(C(F)(F)F)cc3[N+](=O)[O-])CC2)CC1 ZINC000147162333 HH On-Demand Mild SERPINE1 22 48 N#CC1CCN(C(=O)C2CCN(c3ccc(C(F)(F)F)cc3[N+](=O)[O-])CC2)CC1 ZINC000147162333 HH On-Demand Mild LIPG 51 34 CN(C)C(=O)/C=C\c1cccc(Cl)c1 ZINC000147162334 BE On-Demand Anodyne MAOB 0 58 CN(C)C(=O)/C=C\c1cccc(Cl)c1 ZINC000147162334 BE On-Demand Anodyne NR1H4 18 41 CN(C)C(=O)/C=C\c1cccc(Cl)c1 ZINC000147162334 BE On-Demand Anodyne MMP1 0 47 CN(C)C(=O)/C=C\c1cccc(Cl)c1 ZINC000147162334 BE On-Demand Anodyne TUBA4A 0 54 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147162464 HD On-Demand Anodyne F2 21 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147162464 HD On-Demand Anodyne PCSK5 56 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147162464 HD On-Demand Anodyne FURIN 76 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147162464 HD On-Demand Anodyne POLG_WNV 73 32 Cc1nn(C)cc1/C=C1\C[C@H]2[C@@H]3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147162477 GI In-Stock Anodyne NR1I3 0 43 Cc1nn(C)cc1/C=C1\C[C@H]2[C@@H]3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147162477 GI In-Stock Anodyne SHBG 25 45 Cc1nn(C)cc1/C=C1\C[C@H]2[C@@H]3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147162477 GI In-Stock Anodyne GPBAR1 0 45 Cc1nn(C)cc1/C=C1\C[C@H]2[C@@H]3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147162477 GI In-Stock Anodyne G6PD 0 45 CCC[C@@H](NC(N)=O)C(=O)N1CCC(NC(=O)OC(C)(C)C)CC1 ZINC000147162539 ED On-Demand Anodyne CTSK 20 45 CCC[C@@H](NC(N)=O)C(=O)N1CCC(NC(=O)OC(C)(C)C)CC1 ZINC000147162539 ED On-Demand Anodyne EPHX2 15 42 COC(=O)c1cccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147162731 GD On-Demand Anodyne SSTR5 21 43 COC(=O)c1cccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147162731 GD On-Demand Anodyne EPHX2 24 52 COC(=O)c1cccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147162731 GD On-Demand Anodyne TGM2 44 42 COC(=O)c1cccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147162731 GD On-Demand Anodyne AKR1C3 62 41 COC(=O)c1cccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147162731 GD On-Demand Anodyne SFRP1 18 43 COc1ccc(Cl)c(CN2OCC(C)(C)C2=O)c1 ZINC000147162767 CF For-Sale Anodyne NPBWR1 44 32 CC[C@@H](O)c1cccc(N(C)C)c1 ZINC000147162866 AE For-Sale Anodyne KYNU 45 32 CC[C@@H](O)c1cccc(N(C)C)c1 ZINC000147162866 AE For-Sale Anodyne AOC3 32 40 CCc1sc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])nc1-c1ccccc1 ZINC000147162927 GJ On-Demand Bother DHODH 22 40 CCc1sc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])nc1-c1ccccc1 ZINC000147162927 GJ On-Demand Bother PTGDR2 21 48 CCc1sc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])nc1-c1ccccc1 ZINC000147162927 GJ On-Demand Bother AKR1C2 28 40 CC[C@H](O)c1cccc(N(C)C)c1 ZINC000147163018 AE For-Sale Anodyne KYNU 45 32 CC[C@H](O)c1cccc(N(C)C)c1 ZINC000147163018 AE For-Sale Anodyne AOC3 32 40 Cc1cnc2c(S(=O)(=O)N3CCC(NC(=O)c4ccoc4)CC3)cccc2c1 ZINC000147163111 GF On-Demand Anodyne CNR2 18 45 Cc1cnc2c(S(=O)(=O)N3CCC(NC(=O)c4ccoc4)CC3)cccc2c1 ZINC000147163111 GF On-Demand Anodyne EPHX2 29 41 CCCN(CCC)C(=O)Oc1ccc2c(c1)OCO2 ZINC000147163128 CG For-Sale Anodyne EDNRB 92 46 CCCN(CCC)C(=O)Oc1ccc2c(c1)OCO2 ZINC000147163128 CG For-Sale Anodyne EDNRA 101 46 CCCN(CCC)C(=O)Oc1ccc2c(c1)OCO2 ZINC000147163128 CG For-Sale Anodyne BMP1 43 37 O=C(NC1CCN(S(=O)(=O)N2CCOCC2)CC1)c1ccoc1 ZINC000147163369 EC On-Demand Anodyne TGM2 33 42 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc(F)c(F)c3)CC2)CC1 ZINC000147163417 GE On-Demand Mild TGM2 33 40 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc(F)c(F)c3)CC2)CC1 ZINC000147163417 GE On-Demand Mild F13A1 36 41 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc(F)c(F)c3)CC2)CC1 ZINC000147163417 GE On-Demand Mild SFRP1 62 34 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc(F)c(F)c3)CC2)CC1 ZINC000147163417 GE On-Demand Mild WNT3 51 32 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147163487 FE On-Demand Anodyne EPHX2 22 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147163487 FE On-Demand Anodyne TAAR1 29 40 O=C(NC1CCN(S(=O)(=O)Cc2ccc(F)cc2)CC1)c1ccoc1 ZINC000147163561 FE On-Demand Anodyne SIGMAR1 15 40 O=C(NC1CCN(S(=O)(=O)Cc2ccc(F)cc2)CC1)c1ccoc1 ZINC000147163561 FE On-Demand Anodyne CCR3 28 47 O=C(NC1CCN(S(=O)(=O)Cc2ccc(F)cc2)CC1)c1ccoc1 ZINC000147163561 FE On-Demand Anodyne MCHR1 18 44 CC/C=C/[C@@H](O)CCCC ZINC000147163607 AF For-Sale Anodyne CQSS 42 33 CC/C=C/[C@@H](O)CCCC ZINC000147163607 AF For-Sale Anodyne SLCO2A1 44 31 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163625 HJ In-Stock Anodyne ESR1 34 50 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163625 HJ In-Stock Anodyne CYP11A1 0 46 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163625 HJ In-Stock Anodyne AR 29 50 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163625 HJ In-Stock Anodyne ESR2 39 50 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163625 HJ In-Stock Anodyne SHBG 21 46 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163625 HJ In-Stock Anodyne DHCR7 0 45 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163625 HJ In-Stock Anodyne CYP17A1 55 50 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163625 HJ In-Stock Anodyne CYP125 0 43 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163625 HJ In-Stock Anodyne RORC 0 43 CCN(CC)S(=O)(=O)c1cc(C(=O)N2CCC(C#N)CC2)ccc1OC ZINC000147163639 GE On-Demand Mild L3MBTL3 70 35 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147163680 FE On-Demand Anodyne EPHX2 22 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(OCC(F)(F)F)c1 ZINC000147163680 FE On-Demand Anodyne TAAR1 29 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147163747 HE On-Demand Mild F2 20 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147163747 HE On-Demand Mild ADORA2B 23 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147163747 HE On-Demand Mild TRY2_BOVIN 109 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147163747 HE On-Demand Mild PKM 27 41 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147163747 HE On-Demand Mild TGM2 41 38 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147163747 HE On-Demand Mild ST14 99 39 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147163747 HE On-Demand Mild F13A1 53 38 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147163747 HE On-Demand Mild NAMPT 17 46 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(S(=O)(=O)c2ccc(C#N)cc2)CC1 ZINC000147163747 HE On-Demand Mild TMPRSS6 46 31 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(Cl)c1 ZINC000147163750 GF On-Demand Anodyne CNR2 15 49 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(Cl)c1 ZINC000147163750 GF On-Demand Anodyne MAPK13 67 33 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(Cl)c1 ZINC000147163750 GF On-Demand Anodyne EPHX2 42 49 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163752 DD On-Demand Anodyne TIMP3 42 32 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163752 DD On-Demand Anodyne MMP2 16 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163752 DD On-Demand Anodyne MMP3 31 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163752 DD On-Demand Anodyne PCSK5 51 32 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163752 DD On-Demand Anodyne FURIN 57 37 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163752 DD On-Demand Anodyne S1PR5 16 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163752 DD On-Demand Anodyne POLG_WNV 43 32 CCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc2c(c1)CCC(=O)N2 ZINC000147163773 ED On-Demand Anodyne GRIN2B 15 41 CC/C=C/[C@H](O)CCCC ZINC000147163796 AF For-Sale Anodyne CQSS 42 33 CC/C=C/[C@H](O)CCCC ZINC000147163796 AF For-Sale Anodyne SLCO2A1 44 31 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163816 HJ In-Stock Anodyne ESR1 0 50 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163816 HJ In-Stock Anodyne CYP11A1 0 46 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163816 HJ In-Stock Anodyne AR 0 50 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163816 HJ In-Stock Anodyne ESR2 0 50 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163816 HJ In-Stock Anodyne SHBG 21 46 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163816 HJ In-Stock Anodyne DHCR7 0 45 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163816 HJ In-Stock Anodyne CYP17A1 55 50 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163816 HJ In-Stock Anodyne CYP125 0 43 CCn1ncc(/C=C2\C[C@H]3[C@@H]4CC=C5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@H]2O)c1C ZINC000147163816 HJ In-Stock Anodyne RORC 0 43 COc1ccc(Oc2cc(CNC(=O)c3ccn(-c4cccc(F)c4)n3)ccn2)cc1 ZINC000147163884 HI On-Demand Anodyne MMP13 27 40 CCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc2c(c1)CCC(=O)N2 ZINC000147163932 ED On-Demand Anodyne GRIN2B 15 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163941 DD On-Demand Anodyne TIMP3 42 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163941 DD On-Demand Anodyne MMP2 16 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163941 DD On-Demand Anodyne MMP3 31 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163941 DD On-Demand Anodyne PCSK5 51 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163941 DD On-Demand Anodyne FURIN 57 37 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163941 DD On-Demand Anodyne S1PR5 16 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(=O)OC)cc1 ZINC000147163941 DD On-Demand Anodyne POLG_WNV 43 32 CCOC(=O)c1cn[nH]c1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147163962 GC On-Demand Anodyne SSTR5 40 36 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164024 HJ In-Stock Anodyne AR 23 43 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164024 HJ In-Stock Anodyne NR1I3 0 41 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164024 HJ In-Stock Anodyne SHBG 24 43 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164024 HJ In-Stock Anodyne ATP12A 45 32 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164024 HJ In-Stock Anodyne GPBAR1 23 43 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164024 HJ In-Stock Anodyne G6PD 0 41 CCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc2c(c1)CCC(=O)N2 ZINC000147164095 ED On-Demand Anodyne GRIN2B 15 41 Cc1ccc(NC(=O)c2cc(N3CCN(C)CC3)cc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCOCC3)nc12 ZINC000147164112 KI Annotated Mild LCK 39 48 Cc1ccc(NC(=O)c2cc(N3CCN(C)CC3)cc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCOCC3)nc12 ZINC000147164112 KI Annotated Mild MAPK14 28 49 Cc1ccc(NC(=O)c2cc(N3CCN(C)CC3)cc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCOCC3)nc12 ZINC000147164112 KI Annotated Mild SRC 0 48 Cc1ccc(NC(=O)c2cc(N3CCN(C)CC3)cc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCOCC3)nc12 ZINC000147164112 KI Annotated Mild HCK 36 48 Cc1ccc(NC(=O)c2cc(N3CCN(C)CC3)cc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCOCC3)nc12 ZINC000147164112 KI Annotated Mild LYN 55 48 Cc1ccc(NC(=O)c2cc(N3CCN(C)CC3)cc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCOCC3)nc12 ZINC000147164112 KI Annotated Mild STAT6 41 30 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164195 HJ In-Stock Anodyne AR 23 43 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164195 HJ In-Stock Anodyne NR1I3 0 41 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164195 HJ In-Stock Anodyne SHBG 24 43 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164195 HJ In-Stock Anodyne ATP12A 45 32 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164195 HJ In-Stock Anodyne GPBAR1 23 43 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c(C)n1 ZINC000147164195 HJ In-Stock Anodyne G6PD 0 41 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@@H]3CCOC3)nc12 ZINC000147164255 KJ Annotated Mild INSR 30 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@@H]3CCOC3)nc12 ZINC000147164255 KJ Annotated Mild LCK 44 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@@H]3CCOC3)nc12 ZINC000147164255 KJ Annotated Mild MAPK14 31 44 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@@H]3CCOC3)nc12 ZINC000147164255 KJ Annotated Mild SRC 0 44 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@@H]3CCOC3)nc12 ZINC000147164255 KJ Annotated Mild HCK 33 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@@H]3CCOC3)nc12 ZINC000147164255 KJ Annotated Mild LYN 53 43 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)Nc1ccc(Br)cc1)C2 ZINC000147164313 HF On-Demand Anodyne MTNR1A 41 43 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)Nc1ccc(Br)cc1)C2 ZINC000147164313 HF On-Demand Anodyne ROCK2 26 48 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1F ZINC000147164320 DD On-Demand Anodyne TSHR 47 32 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1F ZINC000147164320 DD On-Demand Anodyne ADORA2B 40 42 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1F ZINC000147164320 DD On-Demand Anodyne CETP 25 41 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1F ZINC000147164320 DD On-Demand Anodyne MET 60 42 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1F ZINC000147164320 DD On-Demand Anodyne ACR 55 33 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1F ZINC000147164320 DD On-Demand Anodyne PDGFRA 49 40 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1F ZINC000147164320 DD On-Demand Anodyne CSF1R 45 43 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1F ZINC000147164320 DD On-Demand Anodyne HIF1A 22 42 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1F ZINC000147164320 DD On-Demand Anodyne ENPP1 64 37 COc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1F ZINC000147164320 DD On-Demand Anodyne DRTS_TRYCR 45 34 Cc1c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)cnn1C ZINC000147164415 GI In-Stock Anodyne NR1I3 0 43 Cc1c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)cnn1C ZINC000147164415 GI In-Stock Anodyne SHBG 25 45 Cc1c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)cnn1C ZINC000147164415 GI In-Stock Anodyne GPBAR1 23 45 Cc1c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)cnn1C ZINC000147164415 GI In-Stock Anodyne G6PD 0 45 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@H]3CCOC3)nc12 ZINC000147164419 KJ Annotated Mild INSR 30 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@H]3CCOC3)nc12 ZINC000147164419 KJ Annotated Mild LCK 44 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@H]3CCOC3)nc12 ZINC000147164419 KJ Annotated Mild MAPK14 31 44 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@H]3CCOC3)nc12 ZINC000147164419 KJ Annotated Mild SRC 0 44 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@H]3CCOC3)nc12 ZINC000147164419 KJ Annotated Mild HCK 33 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N[C@H]3CCOC3)nc12 ZINC000147164419 KJ Annotated Mild LYN 53 43 COc1ccc2c(c1)OC[C@@H](C(=O)NCC(=O)Nc1ccc(Br)cc1)C2 ZINC000147164478 HF On-Demand Anodyne MTNR1A 41 43 COc1ccc2c(c1)OC[C@@H](C(=O)NCC(=O)Nc1ccc(Br)cc1)C2 ZINC000147164478 HF On-Demand Anodyne ROCK2 26 48 NC(=O)c1ccc(OCC(=O)Nc2ccc(Cl)c(F)c2)cc1 ZINC000147164533 DF On-Demand Anodyne CETP 19 44 Cc1ccc(S(=O)(=O)N2CCCC[C@@H]2C)cc1C(=O)N1CCC(C#N)CC1 ZINC000147164573 GF On-Demand Mild CASP7 42 32 Cc1ccc(S(=O)(=O)N2CCCC[C@@H]2C)cc1C(=O)N1CCC(C#N)CC1 ZINC000147164573 GF On-Demand Mild AKR1C3 23 45 Cc1ccc(S(=O)(=O)N2CCCC[C@@H]2C)cc1C(=O)N1CCC(C#N)CC1 ZINC000147164573 GF On-Demand Mild L3MBTL3 23 40 Cc1c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)cnn1C ZINC000147164590 GI In-Stock Anodyne NR1I3 0 43 Cc1c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)cnn1C ZINC000147164590 GI In-Stock Anodyne SHBG 25 45 Cc1c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)cnn1C ZINC000147164590 GI In-Stock Anodyne GPBAR1 23 45 Cc1c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)cnn1C ZINC000147164590 GI In-Stock Anodyne G6PD 0 45 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCC(F)(F)C3)nc12 ZINC000147164643 KK Annotated Mild INSR 31 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCC(F)(F)C3)nc12 ZINC000147164643 KK Annotated Mild LCK 48 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCC(F)(F)C3)nc12 ZINC000147164643 KK Annotated Mild MAPK14 32 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCC(F)(F)C3)nc12 ZINC000147164643 KK Annotated Mild SRC 0 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCC(F)(F)C3)nc12 ZINC000147164643 KK Annotated Mild KDR 16 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCC(F)(F)C3)nc12 ZINC000147164643 KK Annotated Mild HCK 37 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCC(F)(F)C3)nc12 ZINC000147164643 KK Annotated Mild LYN 58 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCC(F)(F)C3)nc12 ZINC000147164643 KK Annotated Mild BTK 46 41 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCC(F)(F)C3)nc12 ZINC000147164643 KK Annotated Mild BRAF 25 41 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)s1 ZINC000147164700 GD On-Demand Anodyne TGM2 73 39 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)s1 ZINC000147164700 GD On-Demand Anodyne F13A1 76 39 CCCC(=O)Nc1cccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147164755 FJ On-Demand Anodyne MDM2 83 36 Cc1ccc(S(=O)(=O)N2CCCC[C@H]2C)cc1C(=O)N1CCC(C#N)CC1 ZINC000147164763 GF On-Demand Mild CASP7 42 32 Cc1ccc(S(=O)(=O)N2CCCC[C@H]2C)cc1C(=O)N1CCC(C#N)CC1 ZINC000147164763 GF On-Demand Mild AKR1C3 23 45 Cc1ccc(S(=O)(=O)N2CCCC[C@H]2C)cc1C(=O)N1CCC(C#N)CC1 ZINC000147164763 GF On-Demand Mild L3MBTL3 23 40 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1 ZINC000147164812 FE On-Demand Anodyne CA2 17 49 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1 ZINC000147164812 FE On-Demand Anodyne PPIA 19 40 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1 ZINC000147164812 FE On-Demand Anodyne CA1 18 44 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1 ZINC000147164812 FE On-Demand Anodyne CA4 18 44 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1 ZINC000147164812 FE On-Demand Anodyne ALPL 17 48 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1 ZINC000147164812 FE On-Demand Anodyne CA9 15 48 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1 ZINC000147164812 FE On-Demand Anodyne IDO1 29 45 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1 ZINC000147164812 FE On-Demand Anodyne PFKFB3 82 42 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1 ZINC000147164812 FE On-Demand Anodyne PFKFB1 0 46 Cc1ccc(S(=O)(=O)Nc2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1 ZINC000147164812 FE On-Demand Anodyne PFKFB2 0 42 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CC[C@H](F)C3)nc12 ZINC000147164867 KK Annotated Mild INSR 32 44 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CC[C@H](F)C3)nc12 ZINC000147164867 KK Annotated Mild LCK 45 44 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CC[C@H](F)C3)nc12 ZINC000147164867 KK Annotated Mild MAPK14 36 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CC[C@H](F)C3)nc12 ZINC000147164867 KK Annotated Mild SRC 0 46 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CC[C@H](F)C3)nc12 ZINC000147164867 KK Annotated Mild KDR 16 44 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CC[C@H](F)C3)nc12 ZINC000147164867 KK Annotated Mild HCK 37 44 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CC[C@H](F)C3)nc12 ZINC000147164867 KK Annotated Mild LYN 61 44 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CC[C@H](F)C3)nc12 ZINC000147164867 KK Annotated Mild BTK 47 42 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CC[C@H](F)C3)nc12 ZINC000147164867 KK Annotated Mild BRAF 28 41 Cc1cc(C(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)cc([N+](=O)[O-])c1 ZINC000147164882 HE On-Demand Bother PKM 28 40 Cc1cc(C(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)cc([N+](=O)[O-])c1 ZINC000147164882 HE On-Demand Bother F13A1 48 37 CCN(Cc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1)C(C)=O ZINC000147164945 HH On-Demand Anodyne NPY2R 41 32 CCN(Cc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1)C(C)=O ZINC000147164945 HH On-Demand Anodyne NOS2 63 33 CCN(Cc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1)C(C)=O ZINC000147164945 HH On-Demand Anodyne ROCK2 19 40 CCCC(=O)Nc1cccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147164958 FJ On-Demand Anodyne MDM2 83 36 CC1(C)CNC(=O)c2cc3ccc(C(=O)Nc4cnc5c(cnn5C5CCOCC5)c4)nc3n2C1 ZINC000147164966 JG Annotated Anodyne RPS6KA3 36 41 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCCC[C@@H]1c1nc2ccccc2s1 ZINC000147164968 FH On-Demand Anodyne CPT1A 91 37 Cc1ccc(S(=O)(=O)NC(C)(C)C)cc1C(=O)N1CCC(C#N)CC1 ZINC000147164987 FE On-Demand Mild CCR8 56 31 Cc1ccc(S(=O)(=O)NC(C)(C)C)cc1C(=O)N1CCC(C#N)CC1 ZINC000147164987 FE On-Demand Mild SFRP1 51 35 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147165059 HF On-Demand Anodyne DRTS_PLAFK 19 41 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147165059 HF On-Demand Anodyne AVPR2 85 41 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147165059 HF On-Demand Anodyne AVPR1A 49 43 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147165059 HF On-Demand Anodyne EPHX2 18 56 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147165059 HF On-Demand Anodyne PDE7A 17 47 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147165059 HF On-Demand Anodyne BTK 41 39 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147165059 HF On-Demand Anodyne NOD2 40 33 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild ABL1 56 40 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild INSR 35 46 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild KIT 18 40 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild CSNK2A1 49 35 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild LCK 51 47 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild MAPK14 42 49 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild SRC 22 52 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild KDR 20 47 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild HCK 40 47 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild LYN 62 47 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild EPHA3 20 40 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild BMX 28 40 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild BTK 52 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild BRAF 34 41 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)C3CCN(C)CC3)nc12 ZINC000147165072 KK Annotated Mild DDR1 47 33 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)cs1 ZINC000147165082 GD On-Demand Anodyne PKM 19 40 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)cs1 ZINC000147165082 GD On-Demand Anodyne TGM2 53 41 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)cs1 ZINC000147165082 GD On-Demand Anodyne F13A1 60 41 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(F)cc3)CC2)cs1 ZINC000147165082 GD On-Demand Anodyne TRPC6 46 34 COc1c(Cl)cccc1N1CCN(CCCC#N)CC1 ZINC000147165126 CF For-Sale Anodyne HTR1B 18 43 CCCC(=O)Nc1cccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147165160 FJ On-Demand Anodyne MDM2 83 36 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)NC(C)(C)C ZINC000147165183 GE On-Demand Mild L3MBTL3 67 36 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne F2 117 54 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne PLG 63 49 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne PRSS1 45 50 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne ACE 117 50 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne FKBP1A 91 45 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne OPRM1 72 69 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne OPRD1 58 69 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne OPRK1 15 53 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne F10 16 44 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CELA1 71 50 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne ELANE 85 53 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne MME 101 50 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne ANPEP 44 33 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne TACR1 41 63 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne TRHR 79 53 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CTSD 42 40 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne PGC 76 33 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne HLA-DRB3 51 35 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne MC4R 44 38 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CMA1 65 62 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CTRA_BOVIN 85 45 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne TACR2 26 46 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CTSB 56 47 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne TRY2_BOVIN 25 47 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne PAPA1_CARPA 45 37 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne TRY1_BOVIN 134 49 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CYSP_TRYCR 57 41 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne NTSR1 147 45 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne NTSR2 89 40 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CTSG 56 45 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CTSK 32 43 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CTSL 41 38 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CACNA1B 48 43 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne PGA 37 51 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne NPFFR2 73 48 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne TIMP3 82 39 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne C3AR1 16 45 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne HLA-A 75 46 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne DPP4 26 51 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne ITGA4 71 45 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CTRB1 26 57 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne PREP 94 44 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne MC5R 33 45 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CAPNS1 94 47 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne MMP3 27 41 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne HLA-DRB1 51 33 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CELA2A 75 45 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne REN 92 51 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne REN1 83 44 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne LNPEP 26 45 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne LGMN 104 48 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne PLAT 22 49 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne MTOR 25 41 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne SORT1 56 38 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne TGM1 24 45 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CCKBR 16 47 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CAPN1 126 49 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CTRC 50 57 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CAPN2 83 41 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CTSE 64 38 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne ACE2 81 42 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne PLAU 27 43 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne PGA5 44 32 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne LAP3 28 52 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne KLK5 27 54 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne C5AR1 18 47 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne MARS 55 43 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne SLC5A1 19 42 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne PIN1 19 42 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne TPP2 43 40 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne MMP1 33 44 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne KLK1 29 47 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne FPR1 60 36 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CTRB_BOVIN 44 32 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne NPR 23 43 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne CALCRL 43 43 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne XIAP 107 58 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne DPP8 20 41 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne DPP9 16 41 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne BIRC2 42 39 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne PSMB8 60 35 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne Q9N6S8_PLAFA 16 41 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne BRCA1 86 47 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne NPFFR1 48 43 COC(=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)OC ZINC000147165235 FC For-Sale Anodyne TMPRSS11D 72 44 FC(F)(F)COc1cccc2cccnc12 ZINC000147165311 BG For-Sale Anodyne CCR1 0 45 FC(F)(F)COc1cccc2cccnc12 ZINC000147165311 BG For-Sale Anodyne METAP2 0 44 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCCC[C@H]1c1nc2ccccc2s1 ZINC000147165359 FH On-Demand Anodyne CPT1A 91 37 N#CC1CCN(C(=O)c2cc(S(=O)(=O)N3CCCC3)ccc2Cl)CC1 ZINC000147165437 GF On-Demand Mild L3MBTL3 68 45 CC(C)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147165480 GF On-Demand Anodyne EPHX2 22 59 CC(C)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147165480 GF On-Demand Anodyne TGM2 53 49 COc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147165503 HE On-Demand Bother MMP13 35 42 COc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147165503 HE On-Demand Bother MMP2 16 42 COc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147165503 HE On-Demand Bother MMP3 41 42 COc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147165503 HE On-Demand Bother MMP8 24 42 COc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147165503 HE On-Demand Bother MMP9 29 41 COc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147165503 HE On-Demand Bother PKM 17 52 COc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147165503 HE On-Demand Bother TGM2 42 36 COc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147165503 HE On-Demand Bother MMP7 45 42 COc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147165503 HE On-Demand Bother MMP1 39 42 COc1ccc(S(=O)(=O)N2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)cc1 ZINC000147165503 HE On-Demand Bother F13A1 53 37 CS(=O)(=O)c1ccc2c(c1)OCCC2 ZINC000147165565 BD For-Sale Anodyne PKM 22 40 O=C(NC1CCN(S(=O)(=O)c2ccccc2Cl)CC1)c1ccoc1 ZINC000147165678 FF On-Demand Anodyne EPHX2 35 46 O=C(NC1CCN(S(=O)(=O)c2ccccc2Cl)CC1)c1ccoc1 ZINC000147165678 FF On-Demand Anodyne TGM2 41 44 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne MMP13 49 42 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne MMP2 21 42 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne MMP3 47 42 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne MMP8 31 42 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne MMP9 39 42 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne PKM 16 52 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne TGM2 55 36 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne MMP7 49 42 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne MMP1 49 42 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne F13A1 59 37 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne TRPC6 50 43 COCc1nc(C(=O)N2CCN(S(=O)(=O)c3ccc(OC)cc3)CC2)cs1 ZINC000147165751 HD On-Demand Anodyne TRPC3 23 43 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c1C ZINC000147165788 HK In-Stock Mild AR 22 41 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c1C ZINC000147165788 HK In-Stock Mild SHBG 34 41 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c1C ZINC000147165788 HK In-Stock Mild ATP12A 52 33 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c1C ZINC000147165788 HK In-Stock Mild GPBAR1 28 48 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c1C ZINC000147165788 HK In-Stock Mild G6PD 0 48 CCn1c(NC(=O)c2ccc3cc4n(c3n2)CCCNC4=O)nc2ccccc21 ZINC000147165843 GF Annotated Anodyne RPS6KA3 101 48 N#CC1CCN(C(=O)CCNS(=O)(=O)c2cccc(Br)c2)CC1 ZINC000147165854 HD On-Demand Mild ST14 51 33 Cc1ccc(CSCCNC(=O)c2ccc(=O)n(Cc3ccccc3Cl)c2)cc1 ZINC000147165857 IJ On-Demand Anodyne PTGER3 17 40 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne F2 39 49 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne ACE 29 55 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne OPRM1 30 45 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne TRHR 46 31 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne HLA-DRB3 67 42 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne RIR1_HHV11 74 34 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne NTSR1 178 55 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne NTSR2 124 55 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne NPFFR2 40 42 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne C3AR1 24 46 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne HLA-A 117 47 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne SORT1 66 49 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne SLC5A1 21 43 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne TPP2 43 39 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne XIAP 48 44 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne SIRT1 22 47 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne BRCA1 44 31 CC(C)C[C@H](NC(=O)[C@@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147165960 HB For-Sale Anodyne NPFFR1 18 42 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c1C ZINC000147165983 HK In-Stock Mild AR 22 41 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c1C ZINC000147165983 HK In-Stock Mild SHBG 34 41 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c1C ZINC000147165983 HK In-Stock Mild ATP12A 52 33 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c1C ZINC000147165983 HK In-Stock Mild GPBAR1 28 48 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c1C ZINC000147165983 HK In-Stock Mild G6PD 0 48 COc1ccc(C2=C[C@H](c3ccc(Cl)cc3)[C@H](c3ccc(Cl)cc3)N2C(=O)N2CCNC(=O)C2)c(OC(C)C)c1 ZINC000147166038 KK For-Sale Anodyne TP53 25 75 CCn1c(NC(=O)c2ccc3cc4n(c3n2)CC(C)(C)CNC4=O)nc2ccccc21 ZINC000147166068 HG Annotated Anodyne RPS6KA3 61 60 N[C@@H]1CCN2CCc3c([nH]c4ccccc34)[C@@H]2C1 ZINC000147166081 BE For-Sale Anodyne ADRA2A 15 48 N[C@@H]1CCN2CCc3c([nH]c4ccccc34)[C@@H]2C1 ZINC000147166081 BE For-Sale Anodyne ADRA2B 0 48 N[C@@H]1CCN2CCc3c([nH]c4ccccc34)[C@@H]2C1 ZINC000147166081 BE For-Sale Anodyne ADRA2C 0 52 Cc1cccn2cc(-c3ccc(NC(=O)COc4ccc(C(N)=O)cc4)cc3)nc12 ZINC000147166090 HG On-Demand Anodyne ADORA1 16 49 Cc1cccn2cc(-c3ccc(NC(=O)COc4ccc(C(N)=O)cc4)cc3)nc12 ZINC000147166090 HG On-Demand Anodyne ADORA2A 17 49 Cc1cccn2cc(-c3ccc(NC(=O)COc4ccc(C(N)=O)cc4)cc3)nc12 ZINC000147166090 HG On-Demand Anodyne ADORA2B 51 49 Cc1cccn2cc(-c3ccc(NC(=O)COc4ccc(C(N)=O)cc4)cc3)nc12 ZINC000147166090 HG On-Demand Anodyne CETP 45 42 Cc1cccn2cc(-c3ccc(NC(=O)COc4ccc(C(N)=O)cc4)cc3)nc12 ZINC000147166090 HG On-Demand Anodyne SYK 23 46 Cc1cccn2cc(-c3ccc(NC(=O)COc4ccc(C(N)=O)cc4)cc3)nc12 ZINC000147166090 HG On-Demand Anodyne SHH 44 34 OCC/C=C\c1ccc(F)cc1 ZINC000147166099 AE For-Sale Anodyne AHR 15 45 N[C@H]1CCN2CCc3c([nH]c4ccccc34)[C@@H]2C1 ZINC000147166180 BE For-Sale Anodyne ADRA2A 15 48 N[C@H]1CCN2CCc3c([nH]c4ccccc34)[C@@H]2C1 ZINC000147166180 BE For-Sale Anodyne ADRA2B 0 48 N[C@H]1CCN2CCc3c([nH]c4ccccc34)[C@@H]2C1 ZINC000147166180 BE For-Sale Anodyne ADRA2C 0 52 Cn1c(NC(=O)c2ccc3cc4n(c3n2)CC(C)(C)CNC4=O)nc2ccccc21 ZINC000147166260 HF Annotated Anodyne RPS6KA3 64 57 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne F2 39 49 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne ACE 29 55 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne OPRM1 30 45 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne TRHR 46 31 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne HLA-DRB3 67 42 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne RIR1_HHV11 74 34 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne NTSR1 178 55 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne NTSR2 124 55 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne NPFFR2 40 42 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne C3AR1 24 46 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne HLA-A 117 47 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne SORT1 66 49 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne SLC5A1 21 43 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne TPP2 43 39 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne XIAP 48 44 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne SIRT1 22 47 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne BRCA1 44 31 CC(C)C[C@H](NC(=O)[C@H]1CCCN1C(=O)CNC(=O)[C@H](N)CCCCN)C(=O)O ZINC000147166276 HB For-Sale Anodyne NPFFR1 18 42 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c(C)n1 ZINC000147166294 HK In-Stock Mild AR 43 43 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c(C)n1 ZINC000147166294 HK In-Stock Mild SHBG 52 43 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c(C)n1 ZINC000147166294 HK In-Stock Mild ATP12A 53 33 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c(C)n1 ZINC000147166294 HK In-Stock Mild GPBAR1 28 45 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c(C)n1 ZINC000147166294 HK In-Stock Mild G6PD 0 45 CS(=O)(=O)c1cc(C(=O)Nc2ccccc2OCCC(N)=O)cc([N+](=O)[O-])c1 ZINC000147166316 HD On-Demand Bother PYGL 23 40 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c(C)n1 ZINC000147166448 HK In-Stock Mild AR 43 43 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c(C)n1 ZINC000147166448 HK In-Stock Mild SHBG 52 43 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c(C)n1 ZINC000147166448 HK In-Stock Mild ATP12A 53 33 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c(C)n1 ZINC000147166448 HK In-Stock Mild GPBAR1 28 45 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)c(C)n1 ZINC000147166448 HK In-Stock Mild G6PD 0 45 CCCc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147166465 GF On-Demand Anodyne EPHX2 20 45 CCCc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147166465 GF On-Demand Anodyne TGM2 58 50 Cn1c(NC(=O)c2ccc3cc4n(c3n2)CCCNC4=O)nc2ccccc21 ZINC000147166471 FE Annotated Anodyne RPS6KA3 103 51 O=S(=O)(CCN=C=S)c1ccccc1 ZINC000147166565 BD For-Sale Reactive MIF 15 42 O=C(NC1CCN(S(=O)(=O)c2ccc(Cl)s2)CC1)c1ccoc1 ZINC000147166667 FF On-Demand Anodyne EPHX2 15 46 O=C(NC1CCN(S(=O)(=O)c2ccc(Cl)s2)CC1)c1ccoc1 ZINC000147166667 FF On-Demand Anodyne TGM2 36 40 CC(C)n1c(NC(=O)c2ccc3cc4n(c3n2)CC(C)(C)CNC4=O)nc2ccccc21 ZINC000147166684 IH Annotated Anodyne RPS6KA3 62 55 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC[C@@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147166724 HJ In-Stock Anodyne NR1I3 0 42 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC[C@@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147166724 HJ In-Stock Anodyne SHBG 26 46 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC[C@@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147166724 HJ In-Stock Anodyne SMT1 0 40 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC[C@@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147166724 HJ In-Stock Anodyne GPBAR1 25 47 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC[C@@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147166724 HJ In-Stock Anodyne G6PD 0 47 O=C(C[C@@H]1CCCNC1)c1ccccc1F ZINC000147166772 BE For-Sale Anodyne SLC6A2 19 41 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147166866 HJ In-Stock Anodyne NR1I3 0 42 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147166866 HJ In-Stock Anodyne SHBG 26 46 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147166866 HJ In-Stock Anodyne SMT1 0 40 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147166866 HJ In-Stock Anodyne GPBAR1 25 47 Cc1nn(C)c(C)c1/C=C1\C[C@H]2[C@@H]3CC[C@H]4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]2(C)[C@@H]1O ZINC000147166866 HJ In-Stock Anodyne G6PD 0 47 COc1ccccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147166868 FD On-Demand Anodyne EPHX2 24 43 COc1ccccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147166868 FD On-Demand Anodyne TGM2 40 47 COc1ccccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147166868 FD On-Demand Anodyne ITGAV 25 52 COc1ccccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147166868 FD On-Demand Anodyne MCHR1 15 40 CC(C)n1c(NC(=O)c2ccc3cc4n(c3n2)CCCNC4=O)nc2ccccc21 ZINC000147166907 HG Annotated Anodyne RPS6KA3 102 51 C=C(C(N)=O)c1c[nH]c2ccccc12 ZINC000147166913 AD For-Sale Anodyne GABRA1 15 44 C=C(C(N)=O)c1c[nH]c2ccccc12 ZINC000147166913 AD For-Sale Anodyne CFTR 37 42 O=C(C[C@H]1CCCNC1)c1ccccc1F ZINC000147166938 BE For-Sale Anodyne SLC6A2 19 41 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3cccc(Cl)c3)CC2)s1 ZINC000147166985 GF On-Demand Anodyne HTR6 15 40 NC(=O)[C@H]1CCN(Cc2ccnc3ccccc23)C1 ZINC000147166999 CD On-Demand Anodyne HNMT 50 38 Cc1ccc(C(=O)N2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)cc1F ZINC000147167009 HH On-Demand Anodyne INHA 17 50 Cc1ccc(C(=O)N2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)cc1F ZINC000147167009 HH On-Demand Anodyne PRCP 47 36 Cc1ccc(C(=O)N2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)cc1F ZINC000147167009 HH On-Demand Anodyne MDM2 40 31 O=C(NC1CCN(S(=O)(=O)c2ccc(F)c(F)c2F)CC1)c1ccoc1 ZINC000147167046 GE On-Demand Anodyne EPHX2 29 43 CN(Cc1cscn1)C(=O)NCc1cccc(C(F)(F)F)c1 ZINC000147167106 EH On-Demand Anodyne PDS 42 38 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc2cccnc12 ZINC000147167121 DD On-Demand Anodyne WNT3 19 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc2cccnc12 ZINC000147167121 DD On-Demand Anodyne TNKS 20 40 Cc1ccc(C(=O)N2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)cc1F ZINC000147167141 HH On-Demand Anodyne INHA 17 50 Cc1ccc(C(=O)N2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)cc1F ZINC000147167141 HH On-Demand Anodyne PRCP 47 36 Cc1ccc(C(=O)N2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)cc1F ZINC000147167141 HH On-Demand Anodyne MDM2 40 31 N[C@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167208 BF For-Sale Anodyne CHRNA2 15 50 N[C@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167208 BF For-Sale Anodyne CHRNA3 17 50 N[C@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167208 BF For-Sale Anodyne CHRNA4 24 50 N[C@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167208 BF For-Sale Anodyne CHRND 0 50 N[C@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167208 BF For-Sale Anodyne CHRNB4 0 50 N[C@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167208 BF For-Sale Anodyne ACHP_LYMST 19 50 N[C@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167208 BF For-Sale Anodyne Q8WSF8_APLCA 16 50 N[C@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167208 BF For-Sale Anodyne NACHRBETA2 16 50 O=C(CCSc1ccc(Cl)cc1)Nc1ccc(N2CCCCC2)cc1 ZINC000147167218 FK In-Stock Anodyne KCNQ2 48 43 Cc1ccc(C(=O)N2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)cc1F ZINC000147167242 HH On-Demand Anodyne INHA 17 50 Cc1ccc(C(=O)N2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)cc1F ZINC000147167242 HH On-Demand Anodyne PRCP 47 36 Cc1ccc(C(=O)N2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)cc1F ZINC000147167242 HH On-Demand Anodyne MDM2 40 31 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167267 GJ In-Stock Mild AR 0 41 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167267 GJ In-Stock Mild NR1I3 0 40 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167267 GJ In-Stock Mild SHBG 29 41 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167267 GJ In-Stock Mild HSD17B3 20 46 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167267 GJ In-Stock Mild CYP17A1 22 42 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167267 GJ In-Stock Mild ATP12A 53 34 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167267 GJ In-Stock Mild GPBAR1 29 46 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167267 GJ In-Stock Mild G6PD 0 46 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)CCCN(C)C)nc12 ZINC000147167278 KJ Annotated Mild INSR 32 51 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)CCCN(C)C)nc12 ZINC000147167278 KJ Annotated Mild LCK 43 51 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)CCCN(C)C)nc12 ZINC000147167278 KJ Annotated Mild MAPK14 24 45 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)CCCN(C)C)nc12 ZINC000147167278 KJ Annotated Mild SRC 0 51 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)CCCN(C)C)nc12 ZINC000147167278 KJ Annotated Mild KDR 15 45 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)CCCN(C)C)nc12 ZINC000147167278 KJ Annotated Mild HCK 35 51 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)CCCN(C)C)nc12 ZINC000147167278 KJ Annotated Mild LYN 54 51 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)CCCN(C)C)nc12 ZINC000147167278 KJ Annotated Mild BTK 38 42 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N(C)CCCN(C)C)nc12 ZINC000147167278 KJ Annotated Mild BRAF 22 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc2cccnc12 ZINC000147167314 DD On-Demand Anodyne WNT3 19 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc2cccnc12 ZINC000147167314 DD On-Demand Anodyne TNKS 20 40 N[C@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167322 BF For-Sale Anodyne CHRNA2 15 50 N[C@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167322 BF For-Sale Anodyne CHRNA3 17 50 N[C@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167322 BF For-Sale Anodyne CHRNA4 24 50 N[C@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167322 BF For-Sale Anodyne CHRND 0 50 N[C@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167322 BF For-Sale Anodyne CHRNB4 0 50 N[C@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167322 BF For-Sale Anodyne ACHP_LYMST 19 50 N[C@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167322 BF For-Sale Anodyne Q8WSF8_APLCA 16 50 N[C@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167322 BF For-Sale Anodyne NACHRBETA2 16 50 CCOC(=O)c1cnc(-c2cccnc2)nc1N(C)C ZINC000147167355 CD For-Sale Anodyne JUN 18 45 CCOC(=O)c1cnc(-c2cccnc2)nc1N(C)C ZINC000147167355 CD For-Sale Anodyne ADORA3 15 41 CCCC(C)(C)C[C@H]1N[C@@H](C(=O)NCC[C@H](O)CO)[C@H](c2cccc(Cl)c2)[C@@]12C(=O)Nc1cc(Cl)c(F)cc12 ZINC000147167396 KJ Annotated Anodyne MDM2 80 86 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167420 GJ In-Stock Mild NR1I3 0 40 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167420 GJ In-Stock Mild SHBG 29 41 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167420 GJ In-Stock Mild HSD17B3 20 46 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167420 GJ In-Stock Mild CYP17A1 22 42 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167420 GJ In-Stock Mild ATP12A 53 34 CCn1ccc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)n1 ZINC000147167420 GJ In-Stock Mild G6PD 0 46 N[C@@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167460 BF For-Sale Anodyne CHRNA2 15 50 N[C@@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167460 BF For-Sale Anodyne CHRNA3 17 50 N[C@@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167460 BF For-Sale Anodyne CHRNA4 24 50 N[C@@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167460 BF For-Sale Anodyne CHRND 0 50 N[C@@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167460 BF For-Sale Anodyne CHRNB4 0 50 N[C@@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167460 BF For-Sale Anodyne ACHP_LYMST 19 50 N[C@@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167460 BF For-Sale Anodyne Q8WSF8_APLCA 16 50 N[C@@H]1CCCC[C@H]1c1ccc(Cl)nc1 ZINC000147167460 BF For-Sale Anodyne NACHRBETA2 16 50 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCN(C4CC4)CC3)nc12 ZINC000147167527 KJ Annotated Mild INSR 31 42 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCN(C4CC4)CC3)nc12 ZINC000147167527 KJ Annotated Mild LCK 46 42 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCN(C4CC4)CC3)nc12 ZINC000147167527 KJ Annotated Mild MAPK14 36 43 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCN(C4CC4)CC3)nc12 ZINC000147167527 KJ Annotated Mild SRC 0 44 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCN(C4CC4)CC3)nc12 ZINC000147167527 KJ Annotated Mild KDR 15 44 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCN(C4CC4)CC3)nc12 ZINC000147167527 KJ Annotated Mild HCK 37 42 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCN(C4CC4)CC3)nc12 ZINC000147167527 KJ Annotated Mild LYN 59 42 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCN(C4CC4)CC3)nc12 ZINC000147167527 KJ Annotated Mild BTK 46 40 Cc1ccc(NC(=O)c2cccc(C(C)(C)C#N)c2)cc1Nc1ncnc2cnc(N3CCN(C4CC4)CC3)nc12 ZINC000147167527 KJ Annotated Mild BRAF 18 40 c1nc(N[C@@H]2CCCNC2)c2cn[nH]c2n1 ZINC000147167566 BC On-Demand Anodyne CHEK1 28 43 c1nc(N[C@@H]2CCCNC2)c2cn[nH]c2n1 ZINC000147167566 BC On-Demand Anodyne CD38 37 55 N[C@@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167570 BF For-Sale Anodyne CHRNA2 15 50 N[C@@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167570 BF For-Sale Anodyne CHRNA3 17 50 N[C@@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167570 BF For-Sale Anodyne CHRNA4 24 50 N[C@@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167570 BF For-Sale Anodyne CHRND 0 50 N[C@@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167570 BF For-Sale Anodyne CHRNB4 0 50 N[C@@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167570 BF For-Sale Anodyne ACHP_LYMST 19 50 N[C@@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167570 BF For-Sale Anodyne Q8WSF8_APLCA 16 50 N[C@@H]1CCCC[C@@H]1c1ccc(Cl)nc1 ZINC000147167570 BF For-Sale Anodyne NACHRBETA2 16 50 CCN(Cc1ccccc1NC(=O)NCc1ccc(-n2ccnc2)c(F)c1)C(C)=O ZINC000147167595 HH On-Demand Anodyne NOS2 81 35 CCOc1ccccc1C(=O)N1CCN(C(=O)c2cc(OC)ccc2[N+](=O)[O-])CC1 ZINC000147167665 HF On-Demand Bother AKR1C2 30 49 CCOc1ccccc1C(=O)N1CCN(C(=O)c2cc(OC)ccc2[N+](=O)[O-])CC1 ZINC000147167665 HF On-Demand Bother HCN1 59 37 CCOc1ccccc1C(=O)N1CCN(C(=O)c2cc(OC)ccc2[N+](=O)[O-])CC1 ZINC000147167665 HF On-Demand Bother HCN4 45 35 CCc1ccnc2ccc(OC)cc12 ZINC000147167785 AF For-Sale Anodyne PDGFRB 35 43 CCc1ccnc2ccc(OC)cc12 ZINC000147167785 AF For-Sale Anodyne MTR1B_CHICK 61 31 CCc1ccnc2ccc(OC)cc12 ZINC000147167785 AF For-Sale Anodyne MTNR1A 48 64 CCc1ccnc2ccc(OC)cc12 ZINC000147167785 AF For-Sale Anodyne MTNR1B 32 64 CCc1ccnc2ccc(OC)cc12 ZINC000147167785 AF For-Sale Anodyne PDGFRA 40 36 CCc1ccnc2ccc(OC)cc12 ZINC000147167785 AF For-Sale Anodyne CSF1R 16 43 CCN1CCN(c2cc(C(=O)Nc3ccc(C)c(Nc4ncnc5cnc(N6CCOCC6)nc45)c3)cc(C(C)(C)C#N)c2)CC1 ZINC000147167795 KJ Annotated Mild LCK 30 50 CCN1CCN(c2cc(C(=O)Nc3ccc(C)c(Nc4ncnc5cnc(N6CCOCC6)nc45)c3)cc(C(C)(C)C#N)c2)CC1 ZINC000147167795 KJ Annotated Mild MAPK14 26 50 CCN1CCN(c2cc(C(=O)Nc3ccc(C)c(Nc4ncnc5cnc(N6CCOCC6)nc45)c3)cc(C(C)(C)C#N)c2)CC1 ZINC000147167795 KJ Annotated Mild HCK 34 50 CCN1CCN(c2cc(C(=O)Nc3ccc(C)c(Nc4ncnc5cnc(N6CCOCC6)nc45)c3)cc(C(C)(C)C#N)c2)CC1 ZINC000147167795 KJ Annotated Mild LYN 57 50 CCN1CCN(c2cc(C(=O)Nc3ccc(C)c(Nc4ncnc5cnc(N6CCOCC6)nc45)c3)cc(C(C)(C)C#N)c2)CC1 ZINC000147167795 KJ Annotated Mild STAT6 46 31 C/C=C(/OC)C(=O)NC1CCCCC1 ZINC000147167845 AD For-Sale Anodyne EPHX2 19 43 O=C(NC1CCN(S(=O)(=O)/C=C/c2ccccc2)CC1)c1ccoc1 ZINC000147167896 FE On-Demand Anodyne TGM2 38 40 Oc1ccc(-c2cc(F)c(C(F)(F)F)c(F)c2)c(F)c1 ZINC000147167912 CI In-Stock Anodyne ESR1 18 53 Oc1ccc(-c2cc(F)c(C(F)(F)F)c(F)c2)c(F)c1 ZINC000147167912 CI In-Stock Anodyne ESR2 24 53 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168091 GJ In-Stock Mild NR1I3 0 40 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168091 GJ In-Stock Mild SHBG 29 41 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168091 GJ In-Stock Mild HSD17B3 16 46 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168091 GJ In-Stock Mild CYP17A1 17 42 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168091 GJ In-Stock Mild ATP12A 53 34 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168091 GJ In-Stock Mild G6PD 0 46 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168240 GJ In-Stock Mild NR1I3 0 40 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168240 GJ In-Stock Mild SHBG 29 41 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168240 GJ In-Stock Mild HSD17B3 16 46 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168240 GJ In-Stock Mild CYP17A1 17 42 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168240 GJ In-Stock Mild ATP12A 53 34 CCn1cc(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)C2=O)cn1 ZINC000147168240 GJ In-Stock Mild G6PD 0 46 O=C(NC1CCN(S(=O)(=O)c2ccccc2F)CC1)c1ccoc1 ZINC000147168325 FE On-Demand Anodyne CNR2 18 44 O=C(NC1CCN(S(=O)(=O)c2ccccc2F)CC1)c1ccoc1 ZINC000147168325 FE On-Demand Anodyne EPHX2 27 58 O=C(NC1CCN(S(=O)(=O)c2ccccc2F)CC1)c1ccoc1 ZINC000147168325 FE On-Demand Anodyne TGM2 35 43 C[C@]12OCC[C@H]1CC2=O ZINC000147168481 AC For-Sale Anodyne PPP2R1A 43 30 CC(=O)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147168536 GE On-Demand Anodyne EPHX2 22 60 CC(=O)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147168536 GE On-Demand Anodyne TGM2 60 52 CC(=O)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147168536 GE On-Demand Anodyne F13A1 43 37 COc1cc(/C=N/c2ccccc2C(C)C)ccc1OCc1ccc(C(=O)O)cc1 ZINC000147168583 HK In-Stock Mild ADCYAP1R1 46 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(Cl)c(C(=O)NC3CC3)c1)C2 ZINC000147168623 HG On-Demand Anodyne ROCK2 26 48 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(Cl)c(C(=O)NC3CC3)c1)C2 ZINC000147168623 HG On-Demand Anodyne PDK1 40 33 Cc1ccc(S(=O)(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)c(C)c1 ZINC000147168697 GE On-Demand Mild EPHX2 47 57 Cc1ccc(C)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147168702 FE On-Demand Anodyne CNR2 19 45 Cc1ccc(C)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147168702 FE On-Demand Anodyne MAPK13 65 34 Cc1ccc(C)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147168702 FE On-Demand Anodyne EPHX2 41 51 Cc1ccc(C)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147168702 FE On-Demand Anodyne TGM2 38 40 COc1ccc(S(=O)(=O)N(C)C)cc1NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147168766 GE On-Demand Bother KCNMA1 26 47 CCOc1ccc(-n2c(SCC(=O)NCc3ccc4c(c3)OCO4)nnc2-c2ccco2)cc1 ZINC000147168843 JI On-Demand Anodyne CACNA2D1 41 42 CCOc1ccc(-n2c(SCC(=O)NCc3ccc4c(c3)OCO4)nnc2-c2ccco2)cc1 ZINC000147168843 JI On-Demand Anodyne NOS2 86 36 CCOc1ccc(-n2c(SCC(=O)NCc3ccc4c(c3)OCO4)nnc2-c2ccco2)cc1 ZINC000147168843 JI On-Demand Anodyne HCRTR2 17 40 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1C ZINC000147168874 FE On-Demand Anodyne MAPK13 44 32 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1C ZINC000147168874 FE On-Demand Anodyne EPHX2 36 45 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1C ZINC000147168874 FE On-Demand Anodyne TGM2 49 51 COc1ccc(C(=O)NCCNC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147168883 GF On-Demand Anodyne HTR1A 17 47 COc1ccc(C(=O)NCCNC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147168883 GF On-Demand Anodyne DRD2 27 44 COc1ccc(C(=O)NCCNC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147168883 GF On-Demand Anodyne DRD4 52 47 COc1ccc(C(=O)NCCNC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147168883 GF On-Demand Anodyne DRD3 53 44 COc1ccc(C(=O)NCCNC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147168883 GF On-Demand Anodyne ECR 26 44 COc1ccc(C(=O)NCCNC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147168883 GF On-Demand Anodyne PROKR1 55 34 COc1ccc(C(=O)NCCNC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147168883 GF On-Demand Anodyne NPBWR1 66 38 COc1ccc(C(=O)NCCNC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147168883 GF On-Demand Anodyne E3UJZ5_SPOLI 19 44 O=C(NCCCn1ccnc1)NCCOc1ccc2cc(Br)ccc2c1 ZINC000147168923 HH On-Demand Anodyne CYP19A1 26 42 O=C(NCCCn1ccnc1)NCCOc1ccc2cc(Br)ccc2c1 ZINC000147168923 HH On-Demand Anodyne TBXAS1 60 48 O=C(NCCCn1ccnc1)NCCOc1ccc2cc(Br)ccc2c1 ZINC000147168923 HH On-Demand Anodyne HMOX1 20 47 O=C(NCCCn1ccnc1)NCCOc1ccc2cc(Br)ccc2c1 ZINC000147168923 HH On-Demand Anodyne CYP17A1 15 40 O=C(NCCCn1ccnc1)NCCOc1ccc2cc(Br)ccc2c1 ZINC000147168923 HH On-Demand Anodyne HMOX2 64 56 O=C(NCCCn1ccnc1)NCCOc1ccc2cc(Br)ccc2c1 ZINC000147168923 HH On-Demand Anodyne CYP26A1 60 34 O=C(NCCCn1ccnc1)NCCOc1ccc2cc(Br)ccc2c1 ZINC000147168923 HH On-Demand Anodyne QPCT 47 50 Cc1ccc(S(C)(=O)=O)cc1C(=O)N1CCC(C#N)CC1 ZINC000147168932 DD On-Demand Mild CACNA1B 42 42 Cc1ccc(S(C)(=O)=O)cc1C(=O)N1CCC(C#N)CC1 ZINC000147168932 DD On-Demand Mild SLC6A9 50 44 Cc1ccc(S(C)(=O)=O)cc1C(=O)N1CCC(C#N)CC1 ZINC000147168932 DD On-Demand Mild FASN 37 41 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147168988 FF On-Demand Anodyne SLC6A1 17 45 Cn1ncc(C(=O)[C@@H](C#N)c2nc(-c3ccc(Cl)cc3Cl)cs2)c1C1CC1 ZINC000147169008 HK On-Demand Mild ALPL 40 35 CCOC[C@H](C)NC(=O)Nc1cccc(-n2nnnc2C)c1 ZINC000147169030 DD On-Demand Anodyne CCR3 39 41 CO[C@@]1(CN)CCN(Cc2ccccc2)C1 ZINC000147169067 BD For-Sale Anodyne SIGMAR1 67 44 CO[C@@]1(CN)CCN(Cc2ccccc2)C1 ZINC000147169067 BD For-Sale Anodyne NPFFR1 49 35 COc1ccc(-n2c(SCC(=O)NC[C@@H]3CCCO3)nnc2-c2ccco2)cc1 ZINC000147169070 HF On-Demand Anodyne HCRTR2 17 44 COc1ccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147169149 FF On-Demand Anodyne SLC6A1 17 45 Cn1ncc(C(=O)[C@H](C#N)c2nc(-c3ccc(Cl)cc3Cl)cs2)c1C1CC1 ZINC000147169150 HK On-Demand Mild ALPL 40 35 COCCNC(=O)NCCOc1ccc2cc(Br)ccc2c1 ZINC000147169164 FF On-Demand Anodyne MTNR1A 39 40 COCCNC(=O)NCCOc1ccc2cc(Br)ccc2c1 ZINC000147169164 FF On-Demand Anodyne MTNR1B 31 45 COCCNC(=O)NCCOc1ccc2cc(Br)ccc2c1 ZINC000147169164 FF On-Demand Anodyne NCEH1 19 44 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c(C(F)(F)F)c1 ZINC000147169172 FE On-Demand Anodyne NQO2 29 41 CO[C@]1(CN)CCN(Cc2ccccc2)C1 ZINC000147169233 BD For-Sale Anodyne SIGMAR1 67 44 CO[C@]1(CN)CCN(Cc2ccccc2)C1 ZINC000147169233 BD For-Sale Anodyne NPFFR1 49 35 COc1ccc(-n2c(SCC(=O)NC[C@H]3CCCO3)nnc2-c2ccco2)cc1 ZINC000147169245 HF On-Demand Anodyne HCRTR2 17 44 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147169265 FF On-Demand Anodyne DRD4 49 39 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147169265 FF On-Demand Anodyne SLC6A1 17 45 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147169265 FF On-Demand Anodyne DRD3 22 40 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147169265 FF On-Demand Anodyne NQO2 22 41 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147169265 FF On-Demand Anodyne MCHR1 17 44 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c(C(F)(F)F)c1 ZINC000147169310 FE On-Demand Anodyne NQO2 29 41 CC(C)Oc1ccc(CCNC(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147169332 GH On-Demand Anodyne DRTS_PLAFK 19 41 CC(C)Oc1ccc(CCNC(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147169332 GH On-Demand Anodyne ADRB3 22 41 CC(C)Oc1ccc(CCNC(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147169332 GH On-Demand Anodyne POLR1A 58 32 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c1C ZINC000147169399 IK In-Stock Anodyne SHBG 25 43 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c1C ZINC000147169399 IK In-Stock Anodyne ATP12A 44 32 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c1C ZINC000147169399 IK In-Stock Anodyne G6PD 0 44 CN(C)[C@@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169407 HH On-Demand Anodyne CHRM2 17 45 CN(C)[C@@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169407 HH On-Demand Anodyne DRD2 19 46 CN(C)[C@@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169407 HH On-Demand Anodyne DRD4 41 46 CN(C)[C@@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169407 HH On-Demand Anodyne ACHE 51 47 CN(C)[C@@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169407 HH On-Demand Anodyne HTR4 48 46 CN(C)[C@@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169407 HH On-Demand Anodyne SIGMAR1 54 53 CN(C)[C@@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169407 HH On-Demand Anodyne CACNA1I 64 40 C[C@]12OCCC[C@H]1CC2=O ZINC000147169443 AD For-Sale Anodyne PPP2R1A 40 29 COC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147169504 HD On-Demand Anodyne DRD4 35 49 COC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147169504 HD On-Demand Anodyne SIGMAR1 27 45 COC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147169504 HD On-Demand Anodyne MMP13 17 42 COC(=O)c1ccc(S(=O)(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147169504 HD On-Demand Anodyne MMP9 16 42 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147169512 HG On-Demand Anodyne DRD4 47 36 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147169512 HG On-Demand Anodyne DRD3 27 41 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147169512 HG On-Demand Anodyne NQO2 22 41 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c1C ZINC000147169592 IK In-Stock Anodyne SHBG 25 43 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c1C ZINC000147169592 IK In-Stock Anodyne ATP12A 44 32 CCn1nc(C)c(/C=C2\C[C@H]3[C@@H]4CC[C@H]5C[C@@H](O)CC[C@]5(C)[C@H]4CC[C@]3(C)[C@@H]2O)c1C ZINC000147169592 IK In-Stock Anodyne G6PD 0 44 C[C@@H](SCC(=O)Nc1ccc(F)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147169594 EF On-Demand Mild DPP4 16 44 C[C@@H](SCC(=O)Nc1ccc(F)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147169594 EF On-Demand Mild MLNR 15 41 CN(C)[C@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169616 HH On-Demand Anodyne CHRM2 17 45 CN(C)[C@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169616 HH On-Demand Anodyne DRD2 19 46 CN(C)[C@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169616 HH On-Demand Anodyne DRD4 41 46 CN(C)[C@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169616 HH On-Demand Anodyne ACHE 51 47 CN(C)[C@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169616 HH On-Demand Anodyne HTR4 48 46 CN(C)[C@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169616 HH On-Demand Anodyne SIGMAR1 54 53 CN(C)[C@H](CNC(=O)NCC1CCN(Cc2ccccc2)CC1)c1cccs1 ZINC000147169616 HH On-Demand Anodyne CACNA1I 64 40 Cc1nccn1-c1ccc(CNC(=O)Nc2cccc(-n3nnnc3C)c2)cc1F ZINC000147169682 HF On-Demand Anodyne CCR3 31 46 COC(=O)c1ccc(S(=O)(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147169696 HD On-Demand Anodyne DRD4 35 49 COC(=O)c1ccc(S(=O)(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147169696 HD On-Demand Anodyne SIGMAR1 27 45 COC(=O)c1ccc(S(=O)(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147169696 HD On-Demand Anodyne MMP13 17 42 COC(=O)c1ccc(S(=O)(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147169696 HD On-Demand Anodyne MMP9 16 42 COc1ccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147169717 HG On-Demand Anodyne DRD4 47 36 COc1ccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147169717 HG On-Demand Anodyne DRD3 27 41 COc1ccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)cc1 ZINC000147169717 HG On-Demand Anodyne NQO2 22 41 Cc1ccc(S(=O)(=O)n2ccc3c(NC4CN(C(=O)OC(C)(C)C)C4)ncnc32)cc1 ZINC000147169729 IG For-Sale Anodyne GPR119 34 50 CN(C)S(=O)(=O)c1ccc2cc(Br)ccc2c1 ZINC000147169764 DF On-Demand Anodyne NCEH1 19 44 COC(=O)c1ccccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147169849 GD On-Demand Anodyne CNR2 16 43 COC(=O)c1ccccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147169849 GD On-Demand Anodyne EPHX2 28 42 COC(=O)c1ccccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147169849 GD On-Demand Anodyne TGM2 39 41 COC(=O)c1ccccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147169849 GD On-Demand Anodyne ITGAV 22 40 COC(=O)c1ccccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147169849 GD On-Demand Anodyne CCR8 48 34 Cc1nnnn1-c1cccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)c1 ZINC000147169888 HH On-Demand Anodyne ROCK2 17 40 Cc1nnnn1-c1cccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)c1 ZINC000147169888 HH On-Demand Anodyne NAMPT 37 40 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)cc1 ZINC000147169933 HG On-Demand Anodyne DRD4 47 36 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)cc1 ZINC000147169933 HG On-Demand Anodyne DRD3 27 41 COc1ccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)cc1 ZINC000147169933 HG On-Demand Anodyne NQO2 22 41 CCCCOc1c(Cl)cc(C(=O)N2CCC(C#N)CC2)cc1OC ZINC000147170018 FH On-Demand Mild PTAFR 15 41 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147170074 FD On-Demand Anodyne ACACA 20 40 C[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147170074 FD On-Demand Anodyne ACACB 21 40 COc1ccc(C(=O)NCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147170140 GD On-Demand Anodyne DRD4 46 36 COc1ccc(C(=O)NCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147170140 GD On-Demand Anodyne NQO2 33 40 COc1ccc(C(=O)NCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147170140 GD On-Demand Anodyne MTNR1A 71 46 COc1ccc(C(=O)NCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147170140 GD On-Demand Anodyne MTNR1B 58 40 COc1ccc(C(=O)NCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147170140 GD On-Demand Anodyne ROCK2 34 43 COc1ccc(C(=O)NCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147170140 GD On-Demand Anodyne NAAA 18 42 Cc1nnnn1-c1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147170168 GG On-Demand Anodyne CCR3 43 45 CCN1CCN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)c(C)c2)CC1 ZINC000147170247 GD On-Demand Anodyne HRH3 15 41 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147170267 FD On-Demand Anodyne ACACA 20 40 C[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147170267 FD On-Demand Anodyne ACACB 21 40 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(C)c1 ZINC000147170274 FE On-Demand Anodyne CNR2 16 40 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(C)c1 ZINC000147170274 FE On-Demand Anodyne MAPK13 46 32 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(C)c1 ZINC000147170274 FE On-Demand Anodyne EPHX2 43 63 CC(=O)NCc1ccc(-c2ccncc2)cc1 ZINC000147170349 BE On-Demand Anodyne CYP11B2 15 50 CC(=O)NCc1ccc(-c2ccncc2)cc1 ZINC000147170349 BE On-Demand Anodyne ROCK1 20 44 CC(=O)NCc1ccc(-c2ccncc2)cc1 ZINC000147170349 BE On-Demand Anodyne ROCK2 23 55 CC(=O)NCc1ccc(-c2ccncc2)cc1 ZINC000147170349 BE On-Demand Anodyne CYP17A1 21 50 CC(=O)NCc1ccc(-c2ccncc2)cc1 ZINC000147170349 BE On-Demand Anodyne NAMPT 57 35 Cc1nnnn1-c1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147170355 GG On-Demand Anodyne CCR3 43 45 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(F)c(F)c1 ZINC000147170386 DG On-Demand Anodyne BMP1 44 36 CCN1CCN(c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)c(C)c2)CC1 ZINC000147170485 GD On-Demand Anodyne HRH3 15 41 Cc1nnnn1-c1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147170524 GG On-Demand Anodyne CCR3 43 45 C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(F)c(F)c1 ZINC000147170562 DG On-Demand Anodyne BMP1 44 36 Cc1nnnn1-c1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147170686 GG On-Demand Anodyne CCR3 43 45 NC(=O)c1ccc(OCC(=O)Nc2ccccc2NC(=O)N2CCCC2)cc1 ZINC000147170768 GE On-Demand Anodyne COLA 35 45 NC(=O)c1ccc(OCC(=O)Nc2ccccc2NC(=O)N2CCCC2)cc1 ZINC000147170768 GE On-Demand Anodyne CPT1A 33 45 COc1ccc(OCCNC(=O)c2ccc(C(=O)NC(C)(C)C)cc2)cc1 ZINC000147170948 FG For-Sale Anodyne DRD4 41 31 COc1ccc(OCCNC(=O)c2ccc(C(=O)NC(C)(C)C)cc2)cc1 ZINC000147170948 FG For-Sale Anodyne DRD3 15 41 COc1ccc(OCCNC(=O)c2ccc(C(=O)NC(C)(C)C)cc2)cc1 ZINC000147170948 FG For-Sale Anodyne SCNN1A 21 40 COc1ccc(OCCNC(=O)c2ccc(C(=O)NC(C)(C)C)cc2)cc1 ZINC000147170948 FG For-Sale Anodyne NQO2 19 42 COc1ccc(OCCNC(=O)c2ccc(C(=O)NC(C)(C)C)cc2)cc1 ZINC000147170948 FG For-Sale Anodyne MTNR1A 37 44 COc1ccc(OCCNC(=O)c2ccc(C(=O)NC(C)(C)C)cc2)cc1 ZINC000147170948 FG For-Sale Anodyne MTNR1B 28 44 COc1ccc(OCCNC(=O)c2ccc(C(=O)NC(C)(C)C)cc2)cc1 ZINC000147170948 FG For-Sale Anodyne PLA2G4B 42 35 COc1ccc(OCCNC(=O)c2ccc(C(=O)NC(C)(C)C)cc2)cc1 ZINC000147170948 FG For-Sale Anodyne MT-ND1 25 42 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)CCO3)CC1)c1ccoc1 ZINC000147170950 GD On-Demand Anodyne EPHX2 15 49 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)CCO3)CC1)c1ccoc1 ZINC000147170950 GD On-Demand Anodyne PKM 36 41 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)CCO3)CC1)c1ccoc1 ZINC000147170950 GD On-Demand Anodyne TGM2 41 44 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)CCO3)CC1)c1ccoc1 ZINC000147170950 GD On-Demand Anodyne AKR1C3 42 32 CCOC(=O)N1CC[C@H](C(C)C)C1 ZINC000147171107 AE For-Sale Anodyne CHRNA3 34 44 CCOC(=O)N1CC[C@H](C(C)C)C1 ZINC000147171107 AE For-Sale Anodyne CHRNA4 31 44 O=C(NC1CCN(S(=O)(=O)C2=Cc3ccccc3CC2)CC1)c1ccoc1 ZINC000147171155 GF On-Demand Anodyne TGM2 40 46 N#CCCCOc1cccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147171195 FJ On-Demand Mild NAMPT 20 44 CCOC(=O)N1CC[C@@H](C(C)C)C1 ZINC000147171287 AE For-Sale Anodyne CHRNA3 34 44 CCOC(=O)N1CC[C@@H](C(C)C)C1 ZINC000147171287 AE For-Sale Anodyne CHRNA4 31 44 CC(C)(C)n1cc(-c2ccccn2)nn1 ZINC000147171359 BE On-Demand Anodyne GRM5 15 43 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne SSTR2 84 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne EDNRB 28 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne EDNRA 28 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne MC4R 55 44 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne CCKAR 83 43 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne CTSK 20 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne C3AR1 56 34 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne MC3R 74 44 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne MC5R 74 44 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne MMP2 23 43 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne MMP8 29 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne GRIA1 56 38 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne LNPEP 21 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne MMP11 60 36 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne PCSK5 43 34 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne FURIN 70 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne CCKBR 59 47 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne GHSR 49 39 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne MMP9 17 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne MC1R 104 42 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne KISS1R 79 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne POLG_WNV 60 31 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171373 GH On-Demand Anodyne ERAP2 43 40 N#CCCCOc1cccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147171382 FJ On-Demand Mild NAMPT 20 44 COc1ccc([N+](=O)[O-])c(C(=O)NCCC(=O)N2CCCCC2)c1 ZINC000147171401 ED On-Demand Bother DRD4 43 33 COc1ccc([N+](=O)[O-])c(C(=O)NCCC(=O)N2CCCCC2)c1 ZINC000147171401 ED On-Demand Bother TAAR1 17 42 COc1ccc([N+](=O)[O-])c(C(=O)NCCC(=O)N2CCCCC2)c1 ZINC000147171401 ED On-Demand Bother AKR1C2 25 40 CCNC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147171485 ED On-Demand Anodyne KCNK3 59 37 CCNC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147171485 ED On-Demand Anodyne KCNK9 40 35 O=C(NC1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1)c1ccoc1 ZINC000147171559 GG On-Demand Anodyne TRY2_BOVIN 59 39 O=C(NC1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1)c1ccoc1 ZINC000147171559 GG On-Demand Anodyne EPHX2 22 44 O=C(NC1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1)c1ccoc1 ZINC000147171559 GG On-Demand Anodyne PKM 22 44 O=C(NC1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1)c1ccoc1 ZINC000147171559 GG On-Demand Anodyne TGM2 52 52 O=C(NC1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1)c1ccoc1 ZINC000147171559 GG On-Demand Anodyne AKR1C3 47 47 O=C(NC1CCN(S(=O)(=O)c2ccc3ccccc3c2)CC1)c1ccoc1 ZINC000147171559 GG On-Demand Anodyne SFRP1 19 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne SSTR2 84 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne EDNRB 28 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne EDNRA 28 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne MC4R 55 44 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne CCKAR 83 43 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne CTSK 20 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne C3AR1 56 34 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne MC3R 74 44 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne MC5R 74 44 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne MMP2 23 43 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne MMP8 29 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne GRIA1 56 38 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne LNPEP 21 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne MMP11 60 36 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne PCSK5 43 34 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne FURIN 70 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne CCKBR 59 47 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne GHSR 49 39 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne MMP9 17 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne MC1R 104 42 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne KISS1R 79 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne POLG_WNV 60 31 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171562 GH On-Demand Anodyne ERAP2 43 40 N#CCCCOc1cccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147171577 FJ On-Demand Mild NAMPT 20 44 NC(=O)c1ccc(OCC(=O)N2CCN(C(=O)Cc3ccc(Cl)cc3)CC2)cc1 ZINC000147171604 HD On-Demand Anodyne HTR1D 16 45 NC(=O)c1ccc(OCC(=O)N2CCN(C(=O)Cc3ccc(Cl)cc3)CC2)cc1 ZINC000147171604 HD On-Demand Anodyne HTR1B 18 45 NC(=O)c1ccc(OCC(=O)N2CCN(C(=O)Cc3ccc(Cl)cc3)CC2)cc1 ZINC000147171604 HD On-Demand Anodyne COLA 15 42 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne TYMS 15 45 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne POLA1 21 42 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne SLC29A1 62 36 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne TK 63 40 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne P2RY6 63 48 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne TK1 55 61 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne CDA 71 43 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne P2RY4 58 44 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne P2RY2 56 47 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne FIMH 30 41 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne TK2 45 38 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne P2RY14 65 48 O=c1[nH]c(=O)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)cc1C(F)(F)F ZINC000147171619 DA For-Sale Anodyne RNASE1 23 40 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(C(F)(F)F)c2)c1 ZINC000147171628 GG On-Demand Bother DRD4 40 30 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(C(F)(F)F)c2)c1 ZINC000147171628 GG On-Demand Bother MTNR1A 30 47 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(C(F)(F)F)c2)c1 ZINC000147171628 GG On-Demand Bother MTNR1B 28 47 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(C(F)(F)F)c2)c1 ZINC000147171628 GG On-Demand Bother TAAR1 26 40 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(C(F)(F)F)c2)c1 ZINC000147171628 GG On-Demand Bother AKR1C3 16 43 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(C(F)(F)F)c2)c1 ZINC000147171628 GG On-Demand Bother AKR1C2 26 43 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc(C(F)(F)F)c2)c1 ZINC000147171628 GG On-Demand Bother PDS 49 42 CCNC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147171682 ED On-Demand Anodyne KCNK3 59 37 CCNC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147171682 ED On-Demand Anodyne KCNK9 40 35 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne SSTR2 84 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne EDNRB 28 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne EDNRA 28 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne MC4R 55 44 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne CCKAR 83 43 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne CTSK 20 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne C3AR1 56 34 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne MC3R 74 44 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne MC5R 74 44 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne MMP2 23 43 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne MMP8 29 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne GRIA1 56 38 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne LNPEP 21 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne MMP11 60 36 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne PCSK5 43 34 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne FURIN 70 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne CCKBR 59 47 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne GHSR 49 39 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne MMP9 17 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne MC1R 104 42 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne KISS1R 79 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne POLG_WNV 60 31 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171758 GH On-Demand Anodyne ERAP2 43 40 Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147171761 GE On-Demand Bother EPHX2 33 65 O[C@@H]1CCN(c2ccc(Nc3ncc4c5ccncc5n(C5CCCC5)c4n3)nn2)C1 ZINC000147171970 HG Annotated Anodyne FLT3 25 67 O=C(NC1CCN(S(=O)(=O)c2ccccc2[N+](=O)[O-])CC1)c1ccoc1 ZINC000147171974 GD On-Demand Bother EPHX2 18 61 O=C(NC1CCN(S(=O)(=O)c2ccccc2[N+](=O)[O-])CC1)c1ccoc1 ZINC000147171974 GD On-Demand Bother TGM2 40 43 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne SSTR2 84 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne EDNRB 28 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne EDNRA 28 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne MC4R 55 44 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne CCKAR 83 43 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne CTSK 20 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne C3AR1 56 34 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne MC3R 74 44 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne MC5R 74 44 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne MMP2 23 43 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne MMP8 29 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne GRIA1 56 38 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne LNPEP 21 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne MMP11 60 36 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne PCSK5 43 34 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne FURIN 70 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne CCKBR 59 47 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne GHSR 49 39 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne MMP9 17 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne MC1R 104 42 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne KISS1R 79 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne POLG_WNV 60 31 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](c1ccccc1)c1c[nH]c2ccccc12 ZINC000147171978 GH On-Demand Anodyne ERAP2 43 40 NC(=O)c1ccc(OCC(=O)N2CC[C@H](C(N)=O)C2)cc1 ZINC000147172015 CB On-Demand Anodyne CHEK2 40 37 NC(=O)c1ccc(OCC(=O)N2CC[C@H](C(N)=O)C2)cc1 ZINC000147172015 CB On-Demand Anodyne CPT1A 78 44 NC(=O)c1ccc(OCC(=O)N2CC[C@H](C(N)=O)C2)cc1 ZINC000147172015 CB On-Demand Anodyne CPT2 41 34 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(F)c(C(N)=O)c3)c2)CCO1 ZINC000147172040 HE On-Demand Anodyne CHRM3 15 41 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(F)c(C(N)=O)c3)c2)CCO1 ZINC000147172040 HE On-Demand Anodyne CCR3 43 44 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(F)c(C(N)=O)c3)c2)CCO1 ZINC000147172040 HE On-Demand Anodyne F2R 51 31 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(F)c(C(N)=O)c3)c2)CCO1 ZINC000147172040 HE On-Demand Anodyne EPHX2 15 41 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(F)c(C(N)=O)c3)c2)CCO1 ZINC000147172040 HE On-Demand Anodyne STAT6 43 34 O[C@H]1CCN(c2ccc(Nc3ncc4c5ccncc5n(C5CCCC5)c4n3)nn2)C1 ZINC000147172160 HG Annotated Anodyne FLT3 25 67 NC(=O)c1ccc(OCC(=O)N2CC[C@@H](C(N)=O)C2)cc1 ZINC000147172186 CB On-Demand Anodyne CHEK2 40 37 NC(=O)c1ccc(OCC(=O)N2CC[C@@H](C(N)=O)C2)cc1 ZINC000147172186 CB On-Demand Anodyne COLA 88 51 NC(=O)c1ccc(OCC(=O)N2CC[C@@H](C(N)=O)C2)cc1 ZINC000147172186 CB On-Demand Anodyne CPT1A 78 44 NC(=O)c1ccc(OCC(=O)N2CC[C@@H](C(N)=O)C2)cc1 ZINC000147172186 CB On-Demand Anodyne CPT2 41 34 O=C(NC1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1)c1ccoc1 ZINC000147172188 FF On-Demand Anodyne EPHX2 23 42 O=C(NC1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1)c1ccoc1 ZINC000147172188 FF On-Demand Anodyne TGM2 56 54 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(F)c(C(N)=O)c3)c2)CCO1 ZINC000147172261 HE On-Demand Anodyne CHRM3 15 41 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(F)c(C(N)=O)c3)c2)CCO1 ZINC000147172261 HE On-Demand Anodyne CCR3 43 44 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(F)c(C(N)=O)c3)c2)CCO1 ZINC000147172261 HE On-Demand Anodyne F2R 51 31 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(F)c(C(N)=O)c3)c2)CCO1 ZINC000147172261 HE On-Demand Anodyne EPHX2 15 41 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(F)c(C(N)=O)c3)c2)CCO1 ZINC000147172261 HE On-Demand Anodyne STAT6 43 34 COC(=O)c1cc(O)ccc1N=O ZINC000147172307 AD For-Sale Anodyne CA7 0 63 COC(=O)c1cc(O)ccc1N=O ZINC000147172307 AD For-Sale Anodyne CA14 0 45 N#CC1CCN(C(=O)c2ccc(NC3CC3)c([N+](=O)[O-])c2)CC1 ZINC000147172311 DF On-Demand Mild L3MBTL3 46 47 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc3ccccc3n2-c2ccccc2)c1 ZINC000147172329 GI On-Demand Bother AKR1C2 25 42 COc1ccc(CNCc2ccc(OC3CCCC3)nc2)cc1OCCCC#N ZINC000147172350 GI On-Demand Mild PDE4A 45 36 O=C(NC1CCN(S(=O)(=O)c2ccc([N+](=O)[O-])cc2)CC1)c1ccoc1 ZINC000147172364 GD On-Demand Bother EPHX2 18 47 O=C(NC1CCN(S(=O)(=O)c2ccc([N+](=O)[O-])cc2)CC1)c1ccoc1 ZINC000147172364 GD On-Demand Bother TGM2 48 47 CCCOCC(=O)NC[C@@H](c1cccc(OC)c1OC)c1c[nH]c2ccccc12 ZINC000147172389 GH On-Demand Anodyne GRPR 43 34 CCOC(=O)c1cnc(-c2ccc(Cl)cc2)nc1N1CCCC1 ZINC000147172435 EH For-Sale Anodyne P2RY12 58 45 CCOC(=O)c1cnc(-c2ccc(Cl)cc2)nc1N1CCCC1 ZINC000147172435 EH For-Sale Anodyne JUN 17 42 CCOC(=O)c1cnc(-c2ccc(Cl)cc2)nc1N1CCCC1 ZINC000147172435 EH For-Sale Anodyne SCN10A 28 41 Cc1ccccc1N(CC(=O)Nc1ccc(C23CC4CC(CC(C4)C2)C3)cc1)S(C)(=O)=O ZINC000147172459 JJ In-Stock Anodyne HIF1A 37 41 CC(C)CCSc1ccc(C(=O)N2CCC(C#N)CC2)cc1[N+](=O)[O-] ZINC000147172514 FI On-Demand Mild L3MBTL3 36 43 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccoc1 ZINC000147172555 ED On-Demand Anodyne SIGMAR1 15 40 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccoc1 ZINC000147172555 ED On-Demand Anodyne EPHX2 25 55 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccoc1 ZINC000147172555 ED On-Demand Anodyne TGM2 66 53 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccoc1 ZINC000147172555 ED On-Demand Anodyne F13A1 50 42 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccoc1 ZINC000147172555 ED On-Demand Anodyne AKR1C3 57 40 O=C(NC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccoc1 ZINC000147172555 ED On-Demand Anodyne SFRP1 51 42 COC1CN(C2=N[C@H]3[C@H](O[C@H](CO)[C@@H](O)[C@@H]3O)S2)C1 ZINC000147172558 CA Annotated Anodyne MGEA5 35 54 NC(=O)c1ccc(OCC(=O)Nc2ncc(Cc3ccccc3)s2)cc1 ZINC000147172560 FF On-Demand Anodyne SCD1 32 44 NC(=O)c1ccc(OCC(=O)Nc2ncc(Cc3ccccc3)s2)cc1 ZINC000147172560 FF On-Demand Anodyne SCD 20 43 CCCOCC(=O)NC[C@H](c1cccc(OC)c1OC)c1c[nH]c2ccccc12 ZINC000147172611 GH On-Demand Anodyne GRPR 43 34 O=C(NC1CCN(S(=O)(=O)c2ccc(F)cc2F)CC1)c1ccoc1 ZINC000147172746 FE On-Demand Anodyne CNR2 15 45 O=C(NC1CCN(S(=O)(=O)c2ccc(F)cc2F)CC1)c1ccoc1 ZINC000147172746 FE On-Demand Anodyne MAPK13 52 30 O=C(NC1CCN(S(=O)(=O)c2ccc(F)cc2F)CC1)c1ccoc1 ZINC000147172746 FE On-Demand Anodyne EPHX2 29 48 COCc1nc(C(=O)Nc2cc(Cl)c(OC)cc2OC)cs1 ZINC000147172756 EG On-Demand Anodyne GRM4 17 40 C[C@@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172794 GG On-Demand Anodyne LTA4H 55 46 C[C@@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172794 GG On-Demand Anodyne ADORA2B 37 41 C[C@@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172794 GG On-Demand Anodyne HRH3 27 42 C[C@@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172794 GG On-Demand Anodyne CHEK2 35 44 C[C@@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172794 GG On-Demand Anodyne MLNR 62 33 C[C@@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172794 GG On-Demand Anodyne NOD2 44 41 C[C@H](NC(=O)/C=C\c1ccccc1)c1cccc(O)c1 ZINC000147172885 CG On-Demand Anodyne MMP2 24 57 C[C@H](NC(=O)/C=C\c1ccccc1)c1cccc(O)c1 ZINC000147172885 CG On-Demand Anodyne MMP9 22 53 C[C@H](NC(=O)/C=C\c1ccccc1)c1cccc(O)c1 ZINC000147172885 CG On-Demand Anodyne MMP1 26 57 O=C(NC1CCN(S(=O)(=O)c2ccc(F)cc2)CC1)c1ccoc1 ZINC000147172943 FE On-Demand Anodyne EPHX2 24 47 O=C(NC1CCN(S(=O)(=O)c2ccc(F)cc2)CC1)c1ccoc1 ZINC000147172943 FE On-Demand Anodyne PKM 18 40 O=C(NC1CCN(S(=O)(=O)c2ccc(F)cc2)CC1)c1ccoc1 ZINC000147172943 FE On-Demand Anodyne TGM2 59 49 O=C(NC1CCN(S(=O)(=O)c2ccc(F)cc2)CC1)c1ccoc1 ZINC000147172943 FE On-Demand Anodyne F13A1 44 37 C[C@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172986 GG On-Demand Anodyne LTA4H 55 46 C[C@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172986 GG On-Demand Anodyne ADORA2B 37 41 C[C@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172986 GG On-Demand Anodyne HRH3 27 42 C[C@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172986 GG On-Demand Anodyne CHEK2 35 44 C[C@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172986 GG On-Demand Anodyne MLNR 62 33 C[C@H]1CCCN(Cc2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)C1 ZINC000147172986 GG On-Demand Anodyne NOD2 44 41 COc1ccc(CN[C@@H]2CCCN(c3ncccn3)C2)cc1OCCCC#N ZINC000147173006 GF On-Demand Mild EHMT2 71 34 O=C(NCc1ccc(-c2cc[nH]c(=O)c2)cc1)c1c(Cl)cccc1Cl ZINC000147173151 FI Annotated Anodyne SCN10A 22 40 O=C(NCc1ccc(-c2cc[nH]c(=O)c2)cc1)c1c(Cl)cccc1Cl ZINC000147173151 FI Annotated Anodyne TYK2 16 57 O=C(NC1CCN(S(=O)(=O)c2cccc(F)c2)CC1)c1ccoc1 ZINC000147173170 FE On-Demand Anodyne NPY2R 23 42 O=C(NC1CCN(S(=O)(=O)c2cccc(F)c2)CC1)c1ccoc1 ZINC000147173170 FE On-Demand Anodyne EPHX2 23 49 O=C(NC1CCN(S(=O)(=O)c2cccc(F)c2)CC1)c1ccoc1 ZINC000147173170 FE On-Demand Anodyne PKM 34 45 O=C(NC1CCN(S(=O)(=O)c2cccc(F)c2)CC1)c1ccoc1 ZINC000147173170 FE On-Demand Anodyne TGM2 36 44 O=C(NC1CCN(S(=O)(=O)c2cccc(F)c2)CC1)c1ccoc1 ZINC000147173170 FE On-Demand Anodyne AKR1C3 57 41 O=C(NC1CCN(S(=O)(=O)c2cccc(F)c2)CC1)c1ccoc1 ZINC000147173170 FE On-Demand Anodyne SFRP1 19 43 O=C(NC1CCN(S(=O)(=O)c2cccc(F)c2)CC1)c1ccoc1 ZINC000147173170 FE On-Demand Anodyne HPGDS 32 41 CC(=O)N[C@H](C(=O)N1CCC(C#N)CC1)C(C)C ZINC000147173319 CC On-Demand Mild CCR1 41 39 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)OCCO3)CC1)c1ccoc1 ZINC000147173348 GD On-Demand Anodyne EPHX2 16 62 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)OCCO3)CC1)c1ccoc1 ZINC000147173348 GD On-Demand Anodyne PKM 46 55 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)OCCO3)CC1)c1ccoc1 ZINC000147173348 GD On-Demand Anodyne TGM2 44 43 Clc1c(CBr)ccc2ccccc12 ZINC000147173471 CI For-Sale Reactive CYP2A5 0 56 CC(=O)N[C@@H](C(=O)N1CCC(C#N)CC1)C(C)C ZINC000147173513 CC On-Demand Mild CCR1 41 39 CCCC[C@@H](O)c1cccc(CC)c1 ZINC000147173530 AG For-Sale Anodyne KYNU 44 31 Cc1cc(C)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(C)c1 ZINC000147173555 GF On-Demand Anodyne MAPK13 44 32 Cc1cc(C)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(C)c1 ZINC000147173555 GF On-Demand Anodyne EPHX2 47 59 Cc1cc(C)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(C)c1 ZINC000147173555 GF On-Demand Anodyne TGM2 37 40 Cc1cc(C)c(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(C)c1 ZINC000147173555 GF On-Demand Anodyne ITGAV 25 47 CCCC[C@H](O)c1cccc(CC)c1 ZINC000147173719 AG For-Sale Anodyne KYNU 44 31 NC(=O)c1cc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)ccc1Cl ZINC000147173764 HF On-Demand Anodyne ROCK2 17 40 C[C@@H](NC(=O)CNC(=O)CNC(=O)CN)C(=O)O ZINC000147173793 CA For-Sale Anodyne CA2 20 53 CCCOCC(=O)N1CCN(c2ncnc3c2cnn3C)CC1 ZINC000147173818 DC On-Demand Anodyne PDGFRB 49 35 NC(=O)c1cc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)ccc1Cl ZINC000147173955 HF On-Demand Anodyne ROCK2 17 40 CCCCO[C@@H](C)C(=O)N1CCN(c2ncnc3c2cnn3C)CC1 ZINC000147174087 ED On-Demand Anodyne PDGFRB 58 38 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(Cl)c(C(N)=O)c3)c2)CCO1 ZINC000147174134 HF On-Demand Anodyne CCR3 24 52 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(Cl)c(C(N)=O)c3)c2)CCO1 ZINC000147174134 HF On-Demand Anodyne F2R 49 30 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(Cl)c(C(N)=O)c3)c2)CCO1 ZINC000147174134 HF On-Demand Anodyne ROCK2 15 44 O=C(NC1CCN(S(=O)(=O)c2c(F)cccc2F)CC1)c1ccoc1 ZINC000147174233 FE On-Demand Anodyne EPHX2 26 43 O=C(NC1CCN(S(=O)(=O)c2c(F)cccc2F)CC1)c1ccoc1 ZINC000147174233 FE On-Demand Anodyne PKM 25 49 O=C(NC1CCN(S(=O)(=O)c2c(F)cccc2F)CC1)c1ccoc1 ZINC000147174233 FE On-Demand Anodyne TGM2 40 42 CCCCO[C@H](C)C(=O)N1CCN(c2ncnc3c2cnn3C)CC1 ZINC000147174284 ED On-Demand Anodyne PDGFRB 58 38 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(Cl)c(C(N)=O)c3)c2)CCO1 ZINC000147174398 HF On-Demand Anodyne CCR3 24 52 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(Cl)c(C(N)=O)c3)c2)CCO1 ZINC000147174398 HF On-Demand Anodyne F2R 49 30 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(Cl)c(C(N)=O)c3)c2)CCO1 ZINC000147174398 HF On-Demand Anodyne ROCK2 15 44 CCc1ncc(C(=O)Nc2cc(OC)c(NC(=O)c3ccccc3)cc2OC)s1 ZINC000147174419 HI On-Demand Anodyne KCNK3 60 40 O=C(NC1CCN(S(=O)(=O)c2ccc(Cl)nc2)CC1)c1ccoc1 ZINC000147174420 FD On-Demand Anodyne EPHX2 17 43 O=C(NC1CCN(S(=O)(=O)c2ccc(Cl)nc2)CC1)c1ccoc1 ZINC000147174420 FD On-Demand Anodyne TGM2 47 43 N#Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147174617 FD On-Demand Mild EPHX2 17 44 N#Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147174617 FD On-Demand Mild TGM2 48 47 CC(C)c1cccc(C(=O)O)c1Br ZINC000147174678 BG For-Sale Anodyne SOAT1 46 38 CCCC[C@H](NC(N)=O)C(=O)N1c2ccccc2C[C@@H]1C ZINC000147174750 CE On-Demand Anodyne CCKAR 18 45 NNC(=O)C1Cc2ccccc2C1 ZINC000147174807 AC For-Sale Reactive AMPX_VIBPR 0 40 O=C(NC1CCN(S(=O)(=O)c2ccc(Cl)cc2F)CC1)c1ccoc1 ZINC000147174814 GF On-Demand Anodyne CNR2 18 49 O=C(NC1CCN(S(=O)(=O)c2ccc(Cl)cc2F)CC1)c1ccoc1 ZINC000147174814 GF On-Demand Anodyne MAPK13 47 31 O=C(NC1CCN(S(=O)(=O)c2ccc(Cl)cc2F)CC1)c1ccoc1 ZINC000147174814 GF On-Demand Anodyne EPHX2 34 45 O=C(NC1CCN(S(=O)(=O)c2ccc(Cl)cc2F)CC1)c1ccoc1 ZINC000147174814 GF On-Demand Anodyne TGM2 35 40 CCOC[C@H](C)NC(=O)Nc1ccc(Cl)c(C(N)=O)c1 ZINC000147174825 CD On-Demand Anodyne IMDH_CRYPV 25 43 COCCOc1cccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147174855 EI On-Demand Anodyne EPHX2 21 41 COCCOc1cccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147174855 EI On-Demand Anodyne NAMPT 22 44 COCCOc1cccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147174855 EI On-Demand Anodyne KCNK3 40 35 CCCC[C@@H](NC(N)=O)C(=O)N1c2ccccc2C[C@@H]1C ZINC000147174928 CE On-Demand Anodyne CCKAR 18 45 N#CC1CCN(C(=O)CCC(=O)N2CCC(c3ccccc3)=N2)CC1 ZINC000147175009 EE On-Demand Mild ETHR 55 42 N#Cc1ccccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147175019 FD On-Demand Mild EPHX2 16 41 N#Cc1ccccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147175019 FD On-Demand Mild TGM2 38 42 CN(c1ncccc1CNc1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)S(C)(=O)=O ZINC000147175055 KG Annotated Anodyne JAK2 20 41 CN(c1ncccc1CNc1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)S(C)(=O)=O ZINC000147175055 KG Annotated Anodyne PTK2 54 39 CN(c1ncccc1CNc1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)S(C)(=O)=O ZINC000147175055 KG Annotated Anodyne TNK2 17 41 CN(c1ncccc1CNc1cccn2nc(Nc3ccc(OCCN4CCCC4)cc3)nc12)S(C)(=O)=O ZINC000147175055 KG Annotated Anodyne WEE1 0 41 COCCOc1cccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147175057 EI On-Demand Anodyne EPHX2 21 41 COCCOc1cccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147175057 EI On-Demand Anodyne NAMPT 22 44 COCCOc1cccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147175057 EI On-Demand Anodyne KCNK3 40 35 CCOC(=O)c1cnc(-c2ccco2)nc1N(C)C ZINC000147175131 CD For-Sale Anodyne ADORA1 35 59 CCOC(=O)c1cnc(-c2ccco2)nc1N(C)C ZINC000147175131 CD For-Sale Anodyne ADORA2A 37 59 CCOC(=O)c1cnc(-c2ccco2)nc1N(C)C ZINC000147175131 CD For-Sale Anodyne ADORA3 33 63 CCCC[C@H](NC(N)=O)C(=O)N1c2ccccc2C[C@H]1C ZINC000147175134 CE On-Demand Anodyne CCKAR 18 45 Cc1ccc(C[C@H](NN)c2ccccc2)cc1 ZINC000147175186 BF In-Stock Anodyne SOAT1 24 44 N#CC1CCN(C(=O)CCNS(=O)(=O)c2ccc(OC(F)(F)F)cc2)CC1 ZINC000147175195 HE On-Demand Mild MMP13 25 40 N#CC1CCN(C(=O)CCNS(=O)(=O)c2ccc(OC(F)(F)F)cc2)CC1 ZINC000147175195 HE On-Demand Mild MMP2 33 40 N#CC1CCN(C(=O)CCNS(=O)(=O)c2ccc(OC(F)(F)F)cc2)CC1 ZINC000147175195 HE On-Demand Mild MMP8 15 40 N#CC1CCN(C(=O)CCNS(=O)(=O)c2ccc(OC(F)(F)F)cc2)CC1 ZINC000147175195 HE On-Demand Mild MMP14 26 40 N#CC1CCN(C(=O)CCNS(=O)(=O)c2ccc(OC(F)(F)F)cc2)CC1 ZINC000147175195 HE On-Demand Mild EPHX2 46 42 N#CC1CCN(C(=O)CCNS(=O)(=O)c2ccc(OC(F)(F)F)cc2)CC1 ZINC000147175195 HE On-Demand Mild SFRP1 51 38 COCCOc1cccc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147175250 EI On-Demand Anodyne EPHX2 21 41 COCCOc1cccc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147175250 EI On-Demand Anodyne NAMPT 22 44 COCCOc1cccc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147175250 EI On-Demand Anodyne KCNK3 40 35 CCCC[C@@H](NC(N)=O)C(=O)N1c2ccccc2C[C@H]1C ZINC000147175333 CE On-Demand Anodyne CCKAR 18 45 N[C@@H]1[C@@H]2CN(c3nc4c(cc3F)c(=O)c(C(=O)O)cn4-c3ccc(F)cc3F)C[C@@H]21 ZINC000147175374 HD In-Stock Anodyne ATP6V1B2 0 48 Cc1ccc(C[C@@H](NN)c2ccccc2)cc1 ZINC000147175385 BF In-Stock Anodyne SOAT1 0 44 Cc1nccn1-c1ccc(CNC(=O)Nc2ccc(Cl)c(C(N)=O)c2)cc1F ZINC000147175404 HG On-Demand Anodyne ROCK2 18 42 COCCOc1cccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147175445 EI On-Demand Anodyne EPHX2 21 41 COCCOc1cccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147175445 EI On-Demand Anodyne NAMPT 22 44 COCCOc1cccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147175445 EI On-Demand Anodyne KCNK3 40 35 NC(=O)c1cc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)ccc1Cl ZINC000147175601 HI On-Demand Anodyne ROCK2 27 46 NC(=O)c1cc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)ccc1Cl ZINC000147175601 HI On-Demand Anodyne MET 44 46 NC(=O)c1cc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)ccc1Cl ZINC000147175601 HI On-Demand Anodyne NAMPT 58 46 CCCOc1c(Cl)cc(C(=O)N2CCC(C#N)CC2)cc1OC ZINC000147175643 EH On-Demand Mild PTAFR 16 40 COCCOc1cccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147175675 GI On-Demand Anodyne EPHX2 20 41 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc2c1CCCC2 ZINC000147175784 DF On-Demand Anodyne HDAC10 43 36 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc2c1CCCC2 ZINC000147175784 DF On-Demand Anodyne HDAC11 48 35 CCCCC1CCC(NC(=O)Nc2ccc(Cl)c(C(N)=O)c2)CC1 ZINC000147175849 FI On-Demand Anodyne EPHX2 49 49 CCCCC1CCC(NC(=O)Nc2ccc(Cl)c(C(N)=O)c2)CC1 ZINC000147175849 FI On-Demand Anodyne ENV 41 31 CCCCC1CCC(NC(=O)Nc2ccc(Cl)c(C(N)=O)c2)CC1 ZINC000147175849 FI On-Demand Anodyne IMDH_CRYPV 31 42 COCCOc1cccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147175879 GI On-Demand Anodyne EPHX2 20 41 C#CCNS(=O)(=O)c1cccc2ccccc12 ZINC000147175971 BD On-Demand Mild NPY5R 18 43 C#CCNS(=O)(=O)c1cccc2ccccc12 ZINC000147175971 BD On-Demand Mild Q95J97_RABIT 0 46 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc2c1CCCC2 ZINC000147175976 DF On-Demand Anodyne HDAC10 43 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc2c1CCCC2 ZINC000147175976 DF On-Demand Anodyne HDAC11 48 35 NC(=O)c1cc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)ccc1Cl ZINC000147176045 GH On-Demand Anodyne IMDH_CRYPV 21 42 COCCOc1cccc(NC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147176084 GI On-Demand Anodyne EPHX2 20 41 COc1ccc(CNCc2ccc(OC)c(OCCCC#N)c2)c(OC)c1 ZINC000147176159 FH On-Demand Mild MT-ND1 24 43 NC(=O)c1cc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)ccc1Cl ZINC000147176228 GH On-Demand Anodyne IMDH_CRYPV 21 42 CC(C)[C@H](NC(=O)N(C)Cc1cscn1)c1nc2ccccc2[nH]1 ZINC000147176238 EH On-Demand Anodyne BMP1 47 33 CC(C)[C@H](NC(=O)N(C)Cc1cscn1)c1nc2ccccc2[nH]1 ZINC000147176238 EH On-Demand Anodyne CYP3A4 17 42 O=C(C1CCN(CC2CCOCC2)CC1)N1CCC(S(=O)(=O)c2ccccc2)CC1 ZINC000147176266 IF For-Sale Anodyne TACR2 24 43 O=C(C1CCN(CC2CCOCC2)CC1)N1CCC(S(=O)(=O)c2ccccc2)CC1 ZINC000147176266 IF For-Sale Anodyne CTSS 15 43 O=C(C1CCN(CC2CCOCC2)CC1)N1CCC(S(=O)(=O)c2ccccc2)CC1 ZINC000147176266 IF For-Sale Anodyne SFRP1 92 37 O=C(C1CCN(CC2CCOCC2)CC1)N1CCC(S(=O)(=O)c2ccccc2)CC1 ZINC000147176266 IF For-Sale Anodyne WNT3 74 37 O=C(C1CCN(CC2CCOCC2)CC1)N1CCC(S(=O)(=O)c2ccccc2)CC1 ZINC000147176266 IF For-Sale Anodyne NAMPT 18 41 COCCOc1cccc(NC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147176285 GI On-Demand Anodyne EPHX2 20 41 COc1ccc(-n2c(C)nnc2SCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147176313 FE On-Demand Mild WNT3A 20 41 COc1ccc(-n2c(C)nnc2SCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147176313 FE On-Demand Mild TNKS2 15 41 NC(=O)c1cc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)ccc1Cl ZINC000147176407 GH On-Demand Anodyne IMDH_CRYPV 21 42 CCN(C)C(=O)N1CCC1 ZINC000147176424 AC For-Sale Anodyne CHRNA3 28 49 CCN(C)C(=O)N1CCC1 ZINC000147176424 AC For-Sale Anodyne CHRNA4 31 49 CC(C)[C@@H](NC(=O)N(C)Cc1cscn1)c1nc2ccccc2[nH]1 ZINC000147176447 EH On-Demand Anodyne BMP1 47 33 CC(C)[C@@H](NC(=O)N(C)Cc1cscn1)c1nc2ccccc2[nH]1 ZINC000147176447 EH On-Demand Anodyne CYP3A4 17 42 CC1(C)C(=O)C2=C(Oc3ccccc3[C@@H]2CC(=O)O)C(C)(C)C1=O ZINC000147176461 EG Annotated Mild GRM8 40 34 Cc1cc(C)c(S(=O)(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)c(C)c1 ZINC000147176516 HF On-Demand Mild EPHX2 40 54 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1[N+](=O)[O-] ZINC000147176517 GE On-Demand Bother EPHX2 28 44 Cc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1[N+](=O)[O-] ZINC000147176517 GE On-Demand Bother TGM2 40 43 CCCCCc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147176534 EG On-Demand Anodyne PLM2_PLAFA 61 41 NC(=O)c1cc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)ccc1Cl ZINC000147176614 GH On-Demand Anodyne IMDH_CRYPV 21 42 CCCCCc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147176714 EG On-Demand Anodyne CFTR 42 38 CCCCCc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147176714 EG On-Demand Anodyne SPHK1 42 41 CCCCCc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147176714 EG On-Demand Anodyne S1PR5 16 40 CCCCCc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147176714 EG On-Demand Anodyne PLM2_PLAFA 61 41 O=C(O)CCC(=O)N1CCc2sccc2[C@@H]1c1ccc(Cl)cc1 ZINC000147176788 EH On-Demand Anodyne GRIN2D 56 32 O=C(O)CCC(=O)N1CCc2sccc2[C@@H]1c1ccc(Cl)cc1 ZINC000147176788 EH On-Demand Anodyne TRPM8 19 63 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)CCCC3)CC1)c1ccoc1 ZINC000147176930 GF On-Demand Anodyne EPHX2 17 44 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)CCCC3)CC1)c1ccoc1 ZINC000147176930 GF On-Demand Anodyne TGM2 45 45 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)CCCC3)CC1)c1ccoc1 ZINC000147176930 GF On-Demand Anodyne AKR1C3 58 35 O=C(O)CCC(=O)N1CCc2sccc2[C@H]1c1ccc(Cl)cc1 ZINC000147176975 EH On-Demand Anodyne GRIN2D 56 32 O=C(O)CCC(=O)N1CCc2sccc2[C@H]1c1ccc(Cl)cc1 ZINC000147176975 EH On-Demand Anodyne TRPM8 19 63 CCOc1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1OCC ZINC000147177163 EH On-Demand Bother ENPP1 45 32 CCOc1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1OCC ZINC000147177163 EH On-Demand Bother KCNK3 65 46 CCOc1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1OCC ZINC000147177163 EH On-Demand Bother KCNK9 55 46 N#CC1CCN(C(=O)CS[C@@H](c2ccccc2)c2ccc(Cl)cc2)CC1 ZINC000147177209 GJ On-Demand Mild PTAFR 24 46 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1OC ZINC000147177343 GD On-Demand Anodyne UTS2R 16 47 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1OC ZINC000147177343 GD On-Demand Anodyne EPHX2 19 61 COc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1OC ZINC000147177343 GD On-Demand Anodyne TGM2 46 54 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne EPHX1 0 52 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne LTA4H 26 44 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne HDAC8 15 51 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne HDAC10 19 50 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne CA5B 16 41 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne CA5A 19 41 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne HDAC2 23 49 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne HDAC3 16 50 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne HDAC6 18 50 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne SLC1A2 23 41 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne CYP2B1 0 40 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne HDAH 15 50 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne PFHDAC1 0 50 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne P95276_MYCTO 0 52 O=NCC(=O)Nc1ccccc1 ZINC000147177361 AD For-Sale Anodyne KCNK3 42 33 Cc1cc(C(=O)Nc2ccc(S(C)(=O)=O)cc2)cc([N+](=O)[O-])c1 ZINC000147177368 EF On-Demand Bother UREA_CANEN 22 43 Cc1cc(C(=O)Nc2ccc(S(C)(=O)=O)cc2)cc([N+](=O)[O-])c1 ZINC000147177368 EF On-Demand Bother O49150_SOLTU 46 30 Cc1cc(C(=O)Nc2ccc(S(C)(=O)=O)cc2)cc([N+](=O)[O-])c1 ZINC000147177368 EF On-Demand Bother P96878_MYCTU 26 41 Cc1cc(C(=O)Nc2ccc(S(C)(=O)=O)cc2)cc([N+](=O)[O-])c1 ZINC000147177368 EF On-Demand Bother USP7 29 42 Cc1cc(C(=O)Nc2ccc(S(C)(=O)=O)cc2)cc([N+](=O)[O-])c1 ZINC000147177368 EF On-Demand Bother USP47 37 42 Cc1cc(C(=O)Nc2ccc(S(C)(=O)=O)cc2)cc([N+](=O)[O-])c1 ZINC000147177368 EF On-Demand Bother KCNK3 46 38 Cc1cc(C(=O)Nc2ccc(S(C)(=O)=O)cc2)cc([N+](=O)[O-])c1 ZINC000147177368 EF On-Demand Bother KCNK9 41 38 Cc1ccc2cc(C)c(=O)[nH]c2c1 ZINC000147177523 AE For-Sale Anodyne ITK 25 43 Cc1ccc2cc(C)c(=O)[nH]c2c1 ZINC000147177523 AE For-Sale Anodyne CYP2A5 0 41 Cc1ccc2cc(C)c(=O)[nH]c2c1 ZINC000147177523 AE For-Sale Anodyne DAO 21 41 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)CCC3)CC1)c1ccoc1 ZINC000147177538 FE On-Demand Anodyne EPHX2 17 44 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)CCC3)CC1)c1ccoc1 ZINC000147177538 FE On-Demand Anodyne TGM2 45 45 O=C(NC1CCN(S(=O)(=O)c2ccc3c(c2)CCC3)CC1)c1ccoc1 ZINC000147177538 FE On-Demand Anodyne AKR1C3 58 35 NC(=O)c1ccc(OCC(=O)Nc2cc(Cl)ccc2C(=O)N2CCCC2)cc1 ZINC000147177541 HF On-Demand Anodyne F10 15 48 NC(=O)c1ccc(OCC(=O)Nc2cc(Cl)ccc2C(=O)N2CCCC2)cc1 ZINC000147177541 HF On-Demand Anodyne HNMT 44 32 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(COCC(F)(F)C(F)F)c2)c1 ZINC000147177543 HI On-Demand Bother TAAR1 35 45 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(COCC(F)(F)C(F)F)c2)c1 ZINC000147177543 HI On-Demand Bother KCNK3 43 36 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(COCC(F)(F)C(F)F)c2)c1 ZINC000147177543 HI On-Demand Bother KCNK9 42 36 CCOc1ccc(-c2nnc(SCC(=O)NC3CC(C)(C)NC(C)(C)C3)[nH]2)cc1 ZINC000147177758 HG Annotated Anodyne ENPP1 45 32 CCOc1ccc(-c2nnc(SCC(=O)NC3CC(C)(C)NC(C)(C)C3)[nH]2)cc1 ZINC000147177758 HG Annotated Anodyne EZH2 42 33 CCOC(=O)c1cnc(N2CCOCC2)nc1N(C)C ZINC000147177778 CC For-Sale Anodyne SOAT1 15 40 CCOC(=O)c1cnc(N2CCOCC2)nc1N(C)C ZINC000147177778 CC For-Sale Anodyne STAT6 51 32 CCOC(=O)c1cnc(N2CCOCC2)nc1N(C)C ZINC000147177778 CC For-Sale Anodyne DGAT1 28 40 N#CC1CCN(C(=O)c2cccc(-n3cnnn3)c2)CC1 ZINC000147177811 CD On-Demand Mild PREP 17 40 N#CC1CCN(C(=O)c2cccc(-n3cnnn3)c2)CC1 ZINC000147177811 CD On-Demand Mild L3MBTL3 40 31 N#CC1CCN(C(=O)c2cccc(-n3cnnn3)c2)CC1 ZINC000147177811 CD On-Demand Mild KCNJ1 47 39 CCc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147177943 FE On-Demand Anodyne EPHX2 26 47 CCc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147177943 FE On-Demand Anodyne TGM2 61 48 CCc1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147177943 FE On-Demand Anodyne F13A1 43 39 CCn1c(=O)c(=O)[nH]c2cc(C(=O)N3CCC(C#N)CC3)ccc21 ZINC000147178013 ED On-Demand Mild PARP1 15 47 CCn1c(=O)c(=O)[nH]c2cc(C(=O)N3CCC(C#N)CC3)ccc21 ZINC000147178013 ED On-Demand Mild L3MBTL3 60 36 Cc1cc(C(=O)Nc2ccc(Br)cc2Cl)cc([N+](=O)[O-])c1 ZINC000147178078 FJ On-Demand Bother PYGL 19 40 CNC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147178091 DC On-Demand Anodyne KCNK3 64 37 CNC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147178091 DC On-Demand Anodyne KCNK9 41 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne ACE 16 47 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne OPRM1 0 47 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne OPRD1 0 47 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne MME 23 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne NPY1R 31 49 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne KLK3 71 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne CTSK 50 46 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne CTSL 24 43 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne NPFFR2 43 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne C3AR1 59 36 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne MMP3 24 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne HLA-DRB1 53 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne SOAT1 25 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne PAM 0 44 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne PCSK5 54 37 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne FURIN 61 34 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne CAPN1 34 43 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne CAPN2 67 39 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne ACE2 41 39 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne CTSV 16 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne POLG_DEN26 0 46 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne POLG_WNV 78 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne QRFPR 46 42 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne UTS2 33 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne NPFFR1 59 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne Q9JN24_ECOLX 0 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne ACER2 0 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne GPR88 0 42 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178102 DF On-Demand Anodyne Q91H74_9FLAV 0 40 O=C(NC1CCN(S(=O)(=O)c2cc(F)ccc2F)CC1)c1ccoc1 ZINC000147178144 FE On-Demand Anodyne CNR2 15 45 O=C(NC1CCN(S(=O)(=O)c2cc(F)ccc2F)CC1)c1ccoc1 ZINC000147178144 FE On-Demand Anodyne MAPK13 52 30 O=C(NC1CCN(S(=O)(=O)c2cc(F)ccc2F)CC1)c1ccoc1 ZINC000147178144 FE On-Demand Anodyne EPHX2 30 46 O=C(NC1CCN(S(=O)(=O)c2cc(F)ccc2F)CC1)c1ccoc1 ZINC000147178144 FE On-Demand Anodyne MCHR1 16 40 CC(C)NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147178220 ED On-Demand Mild F2 26 40 CC(C)NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147178220 ED On-Demand Mild TRY2_BOVIN 81 38 CC(C)NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147178220 ED On-Demand Mild PREP 23 41 CC(C)NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147178220 ED On-Demand Mild ST14 107 40 CC(C)NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147178220 ED On-Demand Mild AKR1C3 49 36 CC(C)NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147178220 ED On-Demand Mild SFRP1 46 37 CC(C)NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147178220 ED On-Demand Mild L3MBTL3 54 43 CC(C)NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147178220 ED On-Demand Mild TMPRSS6 68 37 Cc1ccc(C(=O)NNC(=O)NCC2(N(C)C)CCCCC2)s1 ZINC000147178233 EE On-Demand Reactive SLC6A5 15 44 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne ACE 16 47 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne OPRM1 0 47 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne OPRD1 0 47 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne MME 23 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne NPY1R 31 49 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne KLK3 71 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne CTSK 50 46 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne CTSL 24 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne NPFFR2 43 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne C3AR1 59 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne MMP3 24 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne HLA-DRB1 53 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne SOAT1 25 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne PAM 0 44 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne PCSK5 54 37 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne FURIN 61 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne CAPN1 34 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne CAPN2 67 39 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne ACE2 41 39 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne CTSV 16 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne POLG_DEN26 0 46 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne POLG_WNV 78 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne QRFPR 46 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne UTS2 33 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne NPFFR1 59 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne Q9JN24_ECOLX 0 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne ACER2 0 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne GPR88 0 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](CCC)c1ccccc1 ZINC000147178265 DF On-Demand Anodyne Q91H74_9FLAV 0 40 CNC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147178281 DC On-Demand Anodyne KCNK3 64 37 CNC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147178281 DC On-Demand Anodyne KCNK9 41 35 Cc1ccc(S(=O)(=O)N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)cc1 ZINC000147178349 HJ Annotated Anodyne PDE5A 37 42 Cc1ccc(S(=O)(=O)N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)cc1 ZINC000147178349 HJ Annotated Anodyne PTGS2 55 39 Cc1ccc(S(=O)(=O)N2CCc3c([nH]c4ccccc34)[C@@H]2c2ccccc2)cc1 ZINC000147178349 HJ Annotated Anodyne KIF11 23 47 Cc1cc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)c(C)s1 ZINC000147178354 FF On-Demand Anodyne EPHX2 29 40 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne ADA 17 40 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne ADORA1 118 56 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne SLC29A1 88 42 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne ADORA2A 57 54 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne ADORA2B 19 41 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne DNMT1 35 67 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne ADK 33 50 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne AHCY 81 49 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne P2RX4 49 47 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne P2RX1 62 46 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne P2RY1 38 47 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne AMD1 42 46 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne GAPDH 28 44 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne ITPR1 58 42 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne P2RY2 21 49 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne PRKACA 49 39 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne ADORA3 97 50 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne OXGR1 149 51 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne AANAT 64 37 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne RNASE1 46 35 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne DNMT3B 104 67 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne PANC 45 47 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne GPR17 53 35 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne HSPA5 59 35 COC(=O)[C@H](CCSC[C@H]1O[C@@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O)NC(=O)C(F)(F)F ZINC000147178370 JB For-Sale Anodyne DOT1L 140 67 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne ACE 16 47 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne OPRM1 0 47 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne OPRD1 0 47 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne MME 23 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne NPY1R 31 49 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne KLK3 71 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne CTSK 50 46 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne CTSL 24 43 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne NPFFR2 43 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne C3AR1 59 36 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne MMP3 24 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne HLA-DRB1 53 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne SOAT1 25 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne PAM 0 44 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne PCSK5 54 37 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne FURIN 61 34 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne CAPN1 34 43 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne CAPN2 67 39 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne ACE2 41 39 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne CTSV 16 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne POLG_DEN26 0 46 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne POLG_WNV 78 35 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne QRFPR 46 42 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne UTS2 33 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne NPFFR1 59 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne Q9JN24_ECOLX 0 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne ACER2 0 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne GPR88 0 42 CCCC[C@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178482 DF On-Demand Anodyne Q91H74_9FLAV 0 40 Cc1ccc(S(=O)(=O)N2CCc3c([nH]c4ccccc34)[C@H]2c2ccccc2)cc1 ZINC000147178550 HJ Annotated Anodyne PDE5A 37 42 Cc1ccc(S(=O)(=O)N2CCc3c([nH]c4ccccc34)[C@H]2c2ccccc2)cc1 ZINC000147178550 HJ Annotated Anodyne PTGS2 55 39 Cc1ccc(S(=O)(=O)N2CCc3c([nH]c4ccccc34)[C@H]2c2ccccc2)cc1 ZINC000147178550 HJ Annotated Anodyne KIF11 23 47 COC(=O)CN(Cc1ccccc1)C(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147178583 FE On-Demand Anodyne MTNR1A 33 40 CC(C)(C)NC(=S)Nc1nccs1 ZINC000147178595 BE For-Sale Anodyne MAP 0 42 CC(C)(C)NC(=S)Nc1nccs1 ZINC000147178595 BE For-Sale Anodyne MAP1 113 41 CCC[C@H](Nc1cccc2ccccc12)C(=O)O ZINC000147178617 BH For-Sale Anodyne ACE 28 42 CCC[C@H](Nc1cccc2ccccc12)C(=O)O ZINC000147178617 BH For-Sale Anodyne MME 52 43 CCC[C@H](Nc1cccc2ccccc12)C(=O)O ZINC000147178617 BH For-Sale Anodyne CCKAR 36 40 CCC[C@H](Nc1cccc2ccccc12)C(=O)O ZINC000147178617 BH For-Sale Anodyne CPA1 29 44 CCC[C@H](Nc1cccc2ccccc12)C(=O)O ZINC000147178617 BH For-Sale Anodyne ACE2 53 43 CC(C)N(C)S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147178663 EE On-Demand Mild CACNA1B 43 39 CC(C)N(C)S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147178663 EE On-Demand Mild L3MBTL3 34 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne ACE 16 47 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne OPRM1 0 47 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne OPRD1 0 47 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne MME 23 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne NPY1R 31 49 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne KLK3 71 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne CTSK 50 46 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne CTSL 24 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne NPFFR2 43 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne C3AR1 59 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne MMP3 24 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne HLA-DRB1 53 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne SOAT1 25 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne PAM 0 44 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne PCSK5 54 37 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne FURIN 61 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne CAPN1 34 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne CAPN2 67 39 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne ACE2 41 39 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne CTSV 16 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne POLG_DEN26 0 46 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne POLG_WNV 78 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne QRFPR 46 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne UTS2 33 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne NPFFR1 59 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne Q9JN24_ECOLX 0 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne ACER2 0 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne GPR88 0 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](CCC)c1ccccc1 ZINC000147178693 DF On-Demand Anodyne Q91H74_9FLAV 0 40 Cc1c([N+](=O)[O-])cccc1S(=O)(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147178754 GE On-Demand Bother EPHX2 25 52 CCC[C@@H](Nc1cccc2ccccc12)C(=O)O ZINC000147178810 BH For-Sale Anodyne ACE 28 42 CCC[C@@H](Nc1cccc2ccccc12)C(=O)O ZINC000147178810 BH For-Sale Anodyne MME 52 43 CCC[C@@H](Nc1cccc2ccccc12)C(=O)O ZINC000147178810 BH For-Sale Anodyne CCKAR 36 40 CCC[C@@H](Nc1cccc2ccccc12)C(=O)O ZINC000147178810 BH For-Sale Anodyne CPA1 29 44 CCC[C@@H](Nc1cccc2ccccc12)C(=O)O ZINC000147178810 BH For-Sale Anodyne ACE2 53 43 Cc1noc(C)c1COc1ccc(CC(=O)N2CCC(C#N)CC2)cc1 ZINC000147178888 FG On-Demand Mild MLNR 19 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(Sc3nncs3)cc1)C2 ZINC000147179026 GH On-Demand Anodyne ROCK2 32 53 Cc1ccc(S(=O)(=O)N(C)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147179142 GG On-Demand Mild L3MBTL3 57 38 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NC3CCCC3)cc1)C2 ZINC000147179271 GH On-Demand Anodyne MTNR1A 21 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NC3CCCC3)cc1)C2 ZINC000147179271 GH On-Demand Anodyne MTNR1B 21 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NC3CCCC3)cc1)C2 ZINC000147179271 GH On-Demand Anodyne ROCK2 33 51 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NC3CCCC3)cc1)C2 ZINC000147179271 GH On-Demand Anodyne EPHX2 15 48 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NC3CCCC3)cc1)C2 ZINC000147179271 GH On-Demand Anodyne MCHR1 15 41 NC(=O)c1cnc(Cl)cc1NCc1c(F)cccc1Cl ZINC000147179352 DG For-Sale Anodyne CSF1R 33 40 NC(=O)c1cnc(Cl)cc1NCc1c(F)cccc1Cl ZINC000147179352 DG For-Sale Anodyne STAT6 46 40 N#CC1CCN(C(=O)c2ccc3c(c2)C(=O)N(Cc2ccccc2)C3=O)CC1 ZINC000147179357 FF On-Demand Mild L3MBTL3 45 36 CC[C@H](C)NC(=O)c1ccccc1NC(=O)COc1ccc([N+](=O)[O-])c(OC)c1 ZINC000147179518 HG In-Stock Bother AKR1C2 18 41 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1NC ZINC000147179562 CF For-Sale Anodyne ADORA1 39 57 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1NC ZINC000147179562 CF For-Sale Anodyne DHODH 24 44 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1NC ZINC000147179562 CF For-Sale Anodyne CACNA1C 51 36 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1NC ZINC000147179562 CF For-Sale Anodyne ADORA2A 19 49 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1NC ZINC000147179562 CF For-Sale Anodyne TSPO 15 40 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1NC ZINC000147179562 CF For-Sale Anodyne PDE4B 25 50 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1NC ZINC000147179562 CF For-Sale Anodyne PDE4D 17 47 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1NC ZINC000147179562 CF For-Sale Anodyne ADORA3 64 57 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1NC ZINC000147179562 CF For-Sale Anodyne ABCG2 23 40 NC(=O)c1ncccc1C(=O)Nc1ccccc1 ZINC000147179628 BD On-Demand Anodyne PRKDC 25 44 NC(=O)c1ncccc1C(=O)Nc1ccccc1 ZINC000147179628 BD On-Demand Anodyne TRPV1 15 40 NC(=O)c1ncccc1C(=O)Nc1ccccc1 ZINC000147179628 BD On-Demand Anodyne MAP1 48 37 NC(=O)c1ncccc1C(=O)Nc1ccccc1 ZINC000147179628 BD On-Demand Anodyne GRM4 54 42 NC(=O)c1ncccc1C(=O)Nc1ccccc1 ZINC000147179628 BD On-Demand Anodyne ATR 58 44 NC(=O)c1ncccc1C(=O)Nc1ccccc1 ZINC000147179628 BD On-Demand Anodyne SHH 18 40 NC(=O)c1ncccc1C(=O)Nc1ccccc1 ZINC000147179628 BD On-Demand Anodyne SMO 28 43 NC(=O)c1ncccc1C(=O)Nc1ccccc1 ZINC000147179628 BD On-Demand Anodyne NAMPT 21 43 NC(=O)c1ncccc1C(=O)Nc1ccccc1 ZINC000147179628 BD On-Demand Anodyne KCNK3 74 42 NC(=O)c1ncccc1C(=O)Nc1ccccc1 ZINC000147179628 BD On-Demand Anodyne KCNK9 65 38 NC(=O)c1ncccc1C(=O)Nc1ccccc1 ZINC000147179628 BD On-Demand Anodyne G2YM83_BOTF4 52 33 O=S(=O)(NCCS)c1ccc(Cl)cc1 ZINC000147179677 CD For-Sale Mild TBXA2R 54 44 O=S(=O)(NCCS)c1ccc(Cl)cc1 ZINC000147179677 CD For-Sale Mild TBXAS1 29 41 O=S(=O)(NCCS)c1ccc(Cl)cc1 ZINC000147179677 CD For-Sale Mild CCR1 15 46 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2=O)cc1 ZINC000147179755 ED On-Demand Anodyne F10 15 46 CC(=O)Nc1ccc(S(=O)(=O)c2sc3ncccc3c2-c2ccc(Cl)cc2)cc1 ZINC000147179853 IK Annotated Anodyne GRM5 41 78 CC(=O)Nc1ccc(S(=O)(=O)c2sc3ncccc3c2-c2ccc(Cl)cc2)cc1 ZINC000147179853 IK Annotated Anodyne IDO1 27 42 CC(=O)Nc1ccc(S(=O)(=O)c2sc3ncccc3c2-c2ccc(Cl)cc2)cc1 ZINC000147179853 IK Annotated Anodyne NAMPT 35 44 COc1cc2c(cc1OC)CN(C(=O)c1cc(C)cc([N+](=O)[O-])c1)CC2 ZINC000147179874 FG On-Demand Bother ABCB1 0 45 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCCC2=O)cc1 ZINC000147179932 ED On-Demand Anodyne F10 15 46 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild ACE 41 43 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild ELANE 57 42 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild MME 17 43 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild HLA-DRB3 50 32 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild CTRA_BOVIN 55 36 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild CASP2 41 33 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild TRY1_BOVIN 41 36 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild NTSR1 91 36 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild NTSR2 59 33 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild CELA2A 41 35 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild XIAP 55 41 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180124 KH For-Sale Mild BRCA1 64 35 COCCCOc1cc([C@@H](O)[C@@H](C[C@H](N)[C@@H](O)C[C@H](C(=O)NCC(C)(C)C(N)=O)C(C)C)C(C)C)ccc1OC ZINC000147180192 KF For-Sale Anodyne REN 55 77 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne FOLH1 15 43 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CELA1 18 41 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne MME 27 41 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne PTGER1 19 42 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CASP3 18 43 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne KLK3 68 36 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CTSB 59 45 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne PAPA1_CARPA 52 36 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CYSP_TRYCR 50 39 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CTSK 37 45 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CTSL 46 41 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne PREP 15 42 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CAPNS1 66 38 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CTSS 19 45 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CAPN1 82 43 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CASP1 24 41 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CAPN2 119 45 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CASP6 15 40 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne CASP9 23 40 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne TPSAB1 15 41 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne NPR 82 43 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne AMP1_PLAFQ 52 39 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne NAAA 48 38 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne SLC12A5 48 35 O=C(NCc1ccccc1C(=O)O)OCc1ccccc1 ZINC000147180243 CF For-Sale Anodyne PDS 51 36 CN(Cc1cscn1)C(=O)NCC1(N2CCCCC2)CCCCC1 ZINC000147180307 FG On-Demand Anodyne HCN1 59 38 CN(Cc1cscn1)C(=O)NCC1(N2CCCCC2)CCCCC1 ZINC000147180307 FG On-Demand Anodyne HCN4 57 38 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild ACE 41 43 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild ELANE 57 42 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild MME 17 43 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild HLA-DRB3 50 32 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild CTRA_BOVIN 55 36 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild CASP2 41 33 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild TRY1_BOVIN 41 36 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild NTSR1 91 36 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild NTSR2 59 33 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild CELA2A 41 35 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild XIAP 55 41 CCCCC[C@@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180327 KH Annotated Mild BRCA1 64 35 CC(C)(C)OC(=O)N1CCC[C@H]1C(C)(C)C ZINC000147180342 BG For-Sale Anodyne PREP 18 58 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147180360 FD On-Demand Mild TGM2 54 43 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147180360 FD On-Demand Mild F13A1 86 45 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147180360 FD On-Demand Mild AKR1C3 46 36 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147180360 FD On-Demand Mild SFRP1 82 38 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147180360 FD On-Demand Mild WNT3 59 32 C=CCCOCC(=O)Nc1ccc(S(=O)(=O)c2ccc(F)cc2)cc1 ZINC000147180452 FG On-Demand Mild TGM2 33 40 C=CCCOCC(=O)Nc1ccc(S(=O)(=O)c2ccc(F)cc2)cc1 ZINC000147180452 FG On-Demand Mild F13A1 53 40 C=CCCOCC(=O)Nc1ccc(S(=O)(=O)c2ccc(F)cc2)cc1 ZINC000147180452 FG On-Demand Mild IDO1 20 40 C=CCCOCC(=O)Nc1ccc(S(=O)(=O)c2ccc(F)cc2)cc1 ZINC000147180452 FG On-Demand Mild NAMPT 15 41 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild ACE 41 43 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild ELANE 57 42 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild MME 17 43 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild HLA-DRB3 50 32 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild CTRA_BOVIN 55 36 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild CASP2 41 33 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild TRY1_BOVIN 41 36 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild NTSR1 91 36 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild NTSR2 59 33 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild CELA2A 41 35 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild XIAP 55 41 CCCCC[C@H](CC(=O)ON1C(=O)CCC1=O)C(=O)N[C@@H](C(=O)N1CCC[C@@H]1COCc1ccccc1)C(C)C ZINC000147180497 KH For-Sale Mild BRCA1 64 35 CCc1nc(CN(C)C(=O)NCC2(N3CCCCC3)CCCCC2)cs1 ZINC000147180501 GI On-Demand Anodyne HCN1 57 37 CCc1nc(CN(C)C(=O)NCC2(N3CCCCC3)CCCCC2)cs1 ZINC000147180501 GI On-Demand Anodyne HCN4 54 37 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc2nc(N3CCOCC3)sc2c1 ZINC000147180519 HD On-Demand Anodyne CASR 30 40 Cc1sc(-c2n[nH]c3ccccc23)nc1-c1ccc(N2CCN(C)CC2)cc1 ZINC000147180534 GI For-Sale Anodyne PRKCZ 34 42 N[C@@H](Cc1ccc(S(=O)(=O)Cl)cc1)C(=O)O ZINC000147180654 CC For-Sale Unstable CA2 40 43 N[C@@H](Cc1ccc(S(=O)(=O)Cl)cc1)C(=O)O ZINC000147180654 CC For-Sale Unstable MME 16 40 N[C@@H](Cc1ccc(S(=O)(=O)Cl)cc1)C(=O)O ZINC000147180654 CC For-Sale Unstable CA1 30 43 N[C@@H](Cc1ccc(S(=O)(=O)Cl)cc1)C(=O)O ZINC000147180654 CC For-Sale Unstable CPA1 50 38 N[C@@H](Cc1ccc(S(=O)(=O)Cl)cc1)C(=O)O ZINC000147180654 CC For-Sale Unstable TPH1 120 44 N[C@@H](Cc1ccc(S(=O)(=O)Cl)cc1)C(=O)O ZINC000147180654 CC For-Sale Unstable YARS 48 38 N[C@@H](Cc1ccc(S(=O)(=O)Cl)cc1)C(=O)O ZINC000147180654 CC For-Sale Unstable CA12 19 43 N[C@@H](Cc1ccc(S(=O)(=O)Cl)cc1)C(=O)O ZINC000147180654 CC For-Sale Unstable LAP3 40 33 N[C@@H](Cc1ccc(S(=O)(=O)Cl)cc1)C(=O)O ZINC000147180654 CC For-Sale Unstable NCE103 19 41 COCCOc1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)c(C)c1 ZINC000147180690 FG On-Demand Anodyne ROCK2 37 49 O=C(NC1CCN(S(=O)(=O)c2ccc3[nH]c(=O)[nH]c3c2)CC1)c1ccoc1 ZINC000147180699 GD On-Demand Anodyne EPHX2 16 40 O=C(NC1CCN(S(=O)(=O)c2ccc3[nH]c(=O)[nH]c3c2)CC1)c1ccoc1 ZINC000147180699 GD On-Demand Anodyne TGM2 42 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc2nc(N3CCOCC3)sc2c1 ZINC000147180716 HD On-Demand Anodyne CASR 34 40 c1ccc2oc(N3CCOCC3)cc2c1 ZINC000147180720 BE For-Sale Anodyne PRKDC 85 67 c1ccc2oc(N3CCOCC3)cc2c1 ZINC000147180720 BE For-Sale Anodyne PIK3CA 22 43 c1ccc2oc(N3CCOCC3)cc2c1 ZINC000147180720 BE For-Sale Anodyne PIK3CD 21 43 c1ccc2oc(N3CCOCC3)cc2c1 ZINC000147180720 BE For-Sale Anodyne PIK3CG 15 43 c1ccc2oc(N3CCOCC3)cc2c1 ZINC000147180720 BE For-Sale Anodyne PIK3CB 31 43 CC(C)(C)[C@@H]1CCCCN1Cc1ccccc1 ZINC000147180961 BI For-Sale Anodyne ACHE 22 44 CC(C)(C)[C@@H]1CCCCN1Cc1ccccc1 ZINC000147180961 BI For-Sale Anodyne SIGMAR1 49 47 COc1ccc2c(N)c(C(=O)O)sc2c1 ZINC000147181102 BE For-Sale Anodyne AKR1C2 51 37 CC(C)(C)[C@H]1CCCCN1Cc1ccccc1 ZINC000147181158 BI For-Sale Anodyne ACHE 22 44 CC(C)(C)[C@H]1CCCCN1Cc1ccccc1 ZINC000147181158 BI For-Sale Anodyne SIGMAR1 49 47 COc1ccc(CNCCNC(=O)c2ccc(C)cc2)cc1OCCCC#N ZINC000147181176 GG On-Demand Mild PPARA 19 48 COc1ccc(CNCCNC(=O)c2ccc(C)cc2)cc1OCCCC#N ZINC000147181176 GG On-Demand Mild LPAR2 38 43 COc1ccc(CNCCNC(=O)c2ccc(C)cc2)cc1OCCCC#N ZINC000147181176 GG On-Demand Mild PPARD 24 48 COc1ccc(CNCCNC(=O)c2ccc(C)cc2)cc1OCCCC#N ZINC000147181176 GG On-Demand Mild REN 30 46 COc1ccc(CNCCNC(=O)c2ccc(C)cc2)cc1OCCCC#N ZINC000147181176 GG On-Demand Mild S1PR2 43 35 COc1ccc(CNCCNC(=O)c2ccc(C)cc2)cc1OCCCC#N ZINC000147181176 GG On-Demand Mild MT-ND1 26 45 C=CCNC(=O)Nc1ccc(NC(=O)[C@H](C)OCCCC)cc1 ZINC000147181221 DG On-Demand Mild SCN2A 17 40 C=CCNC(=O)Nc1ccc(NC(=O)[C@@H](C)OCCCC)cc1 ZINC000147181415 DG On-Demand Mild SCN2A 17 40 CCCCCCOc1ccc(C(=N)NO)cc1Br ZINC000147181483 DH For-Sale Anodyne LPAR2 50 48 CCCCCCOc1ccc(C(=N)NO)cc1Br ZINC000147181483 DH For-Sale Anodyne S1PR3 15 48 CCCCCCOc1ccc(C(=N)NO)cc1Br ZINC000147181483 DH For-Sale Anodyne PLA2G4B 63 38 CCCCCCOc1ccc(C(=N)NO)cc1Br ZINC000147181483 DH For-Sale Anodyne S1PR2 50 48 CCCCCCOc1ccc(C(=N)NO)cc1Br ZINC000147181483 DH For-Sale Anodyne ACR 49 60 CC(C)(C)OC(=O)N1CCC[C@@H]1C(C)(C)C ZINC000147181489 BG For-Sale Anodyne PREP 18 58 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147181492 EE On-Demand Anodyne KCNQ2 50 34 C[C@H](NC(=O)Nc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147181588 DD On-Demand Mild CCR1 41 39 C[C@H](NC(=O)Nc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147181588 DD On-Demand Mild EPHX2 21 41 C=C1C(=O)O[C@H]2C/C(C)=C/CC/C(C)=C/CC[C@@]3(COC(C)=O)O[C@@H]3C[C@H]12 ZINC000147181618 FI Annotated Mild MYB 0 41 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147181688 EE On-Demand Anodyne KCNQ2 50 34 O=S(=O)(c1cc(F)cc(C(F)(F)F)c1)c1sc2ncccc2c1-c1ccc(Cl)cc1 ZINC000147181702 JK Annotated Anodyne GRM5 40 73 Cc1ccc(C(=O)N2C[C@@H](C)C[C@@H](C)C2)cc1NC(=O)c1ccc2c(c1)COC2 ZINC000147181744 GI On-Demand Anodyne MAPK11 31 40 Cc1ccc(C(=O)N2C[C@@H](C)C[C@@H](C)C2)cc1NC(=O)c1ccc2c(c1)COC2 ZINC000147181744 GI On-Demand Anodyne MAPK14 26 43 C[C@@H](NC(=O)Nc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147181793 DD On-Demand Mild CCR1 41 39 C[C@@H](NC(=O)Nc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147181793 DD On-Demand Mild EPHX2 21 41 C=C1C(=O)O[C@@H]2[C@@H]1C[C@H]1O[C@]1(COC(C)=O)CC/C=C(\C)CC/C=C(\C)[C@H]2O ZINC000147181823 GG Annotated Mild MYB 0 40 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147181892 EE On-Demand Anodyne KCNQ2 50 34 NC(=O)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147181923 GC On-Demand Anodyne EPHX2 17 48 NC(=O)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147181923 GC On-Demand Anodyne TGM2 57 51 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@@H](C)CC ZINC000147181934 CI For-Sale Mild S1PR3 18 53 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@@H](C)CC ZINC000147181934 CI For-Sale Mild S1PR2 27 53 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@@H](C)CC ZINC000147181934 CI For-Sale Mild TPP2 29 46 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@@H](C)CC ZINC000147181934 CI For-Sale Mild LPAR3 18 40 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@@H](C)CC ZINC000147181934 CI For-Sale Mild ASAH1 87 36 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@@H](C)CC ZINC000147181934 CI For-Sale Mild NOD1 88 44 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@@H](C)CC ZINC000147181934 CI For-Sale Mild CQSS 65 46 Cc1ccc(C(=O)N2C[C@H](C)C[C@@H](C)C2)cc1NC(=O)c1ccc2c(c1)COC2 ZINC000147181957 GI On-Demand Anodyne MAPK11 31 40 Cc1ccc(C(=O)N2C[C@H](C)C[C@@H](C)C2)cc1NC(=O)c1ccc2c(c1)COC2 ZINC000147181957 GI On-Demand Anodyne MAPK14 26 43 C=C1C(=O)O[C@H]2[C@@H](O)/C(C)=C/CC/C(C)=C/CC[C@@]3(COC(C)=O)O[C@@H]3C[C@H]12 ZINC000147182010 GG Annotated Mild MYB 0 40 COCc1nc(C(=O)NC[C@@H]2COc3ccccc3O2)cs1 ZINC000147182072 DD On-Demand Anodyne ADRA2B 19 41 COCc1nc(C(=O)NC[C@@H]2COc3ccccc3O2)cs1 ZINC000147182072 DD On-Demand Anodyne ADRA2C 15 41 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147182074 EE On-Demand Anodyne KCNQ2 50 34 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@H](C)CC ZINC000147182138 CI For-Sale Mild S1PR3 18 53 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@H](C)CC ZINC000147182138 CI For-Sale Mild S1PR2 27 53 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@H](C)CC ZINC000147182138 CI For-Sale Mild TPP2 29 46 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@H](C)CC ZINC000147182138 CI For-Sale Mild LPAR3 18 40 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@H](C)CC ZINC000147182138 CI For-Sale Mild ASAH1 87 36 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@H](C)CC ZINC000147182138 CI For-Sale Mild NOD1 88 44 CCCCCCCCCCCCNC(=O)[C@@H](N)[C@H](C)CC ZINC000147182138 CI For-Sale Mild CQSS 65 46 CC(C)CN(c1ccc(F)cc1)S(=O)(=O)c1ccc(Br)cn1 ZINC000147182178 GH For-Sale Anodyne RORC 18 45 C=C1C(=O)O[C@H]2[C@@H](OC(C)=O)/C(C)=C/CC/C(C)=C/CC[C@@]3(C)O[C@@H]3C[C@H]12 ZINC000147182198 FI Annotated Mild MYB 0 51 CSCC[C@H](NC(=O)c1ccco1)C(=O)N1CCC(C#N)CC1 ZINC000147182224 ED On-Demand Mild GHRHR 40 32 CSCC[C@H](NC(=O)c1ccco1)C(=O)N1CCC(C#N)CC1 ZINC000147182224 ED On-Demand Mild P2RY12 69 34 CSCC[C@H](NC(=O)c1ccco1)C(=O)N1CCC(C#N)CC1 ZINC000147182224 ED On-Demand Mild KISS1R 48 32 COCc1nc(C(=O)NC[C@H]2COc3ccccc3O2)cs1 ZINC000147182267 DD On-Demand Anodyne ADRA2B 19 41 COCc1nc(C(=O)NC[C@H]2COc3ccccc3O2)cs1 ZINC000147182267 DD On-Demand Anodyne ADRA2C 15 41 CNC(=O)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147182312 GD On-Demand Anodyne EPHX2 21 50 CNC(=O)c1ccc(S(=O)(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147182312 GD On-Demand Anodyne TGM2 58 52 CC(=O)N1CCc2cc(NC(=O)C(=O)NC[C@@H]3CCCCO3)ccc21 ZINC000147182424 ED On-Demand Anodyne NOS1 15 40 CC(=O)N1CCc2cc(NC(=O)C(=O)NC[C@@H]3CCCCO3)ccc21 ZINC000147182424 ED On-Demand Anodyne NAMPT 30 40 CSCC[C@@H](NC(=O)c1ccco1)C(=O)N1CCC(C#N)CC1 ZINC000147182436 ED On-Demand Mild GHRHR 40 32 CSCC[C@@H](NC(=O)c1ccco1)C(=O)N1CCC(C#N)CC1 ZINC000147182436 ED On-Demand Mild P2RY12 69 34 CSCC[C@@H](NC(=O)c1ccco1)C(=O)N1CCC(C#N)CC1 ZINC000147182436 ED On-Demand Mild KISS1R 48 32 CC(C)CCO[C@@H](C)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147182512 EG On-Demand Anodyne KCNQ2 65 39 CC(=O)N1CCc2cc(NC(=O)C(=O)NC[C@H]3CCCCO3)ccc21 ZINC000147182627 ED On-Demand Anodyne NOS1 15 40 CC(=O)N1CCc2cc(NC(=O)C(=O)NC[C@H]3CCCCO3)ccc21 ZINC000147182627 ED On-Demand Anodyne NAMPT 30 40 C[C@H]1CN(Cc2ccccc2NC(=O)COc2ccc(C(N)=O)cc2)C[C@@H](C)O1 ZINC000147182661 GE On-Demand Anodyne CYSLTR2 45 33 C[C@H]1CN(Cc2ccccc2NC(=O)COc2ccc(C(N)=O)cc2)C[C@@H](C)O1 ZINC000147182661 GE On-Demand Anodyne ITGA4 43 33 NC(=O)c1cncc2cccc(Br)c12 ZINC000147182668 CE For-Sale Anodyne PARP1 25 40 CCOC(=O)c1cnc(-c2ccncc2)nc1N1CCCC1 ZINC000147182676 CE For-Sale Anodyne P2RY12 55 38 CCOC(=O)c1cnc(-c2ccncc2)nc1N1CCCC1 ZINC000147182676 CE For-Sale Anodyne JUN 18 43 CCOC(=O)c1cnc(-c2ccncc2)nc1N1CCCC1 ZINC000147182676 CE For-Sale Anodyne ROCK2 16 40 COCc1nc(C(=O)Nc2cccc3ncccc23)cs1 ZINC000147182683 CG On-Demand Anodyne G2YM83_BOTF4 63 33 CC(C)CCO[C@H](C)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147182720 EG On-Demand Anodyne KCNQ2 65 39 C[C@H]1CN(Cc2ccccc2NC(=O)COc2ccc(C(N)=O)cc2)C[C@H](C)O1 ZINC000147182853 GE On-Demand Anodyne CYSLTR2 45 33 C[C@H]1CN(Cc2ccccc2NC(=O)COc2ccc(C(N)=O)cc2)C[C@H](C)O1 ZINC000147182853 GE On-Demand Anodyne ITGA4 43 33 COCc1nc(C(=O)Nc2nc(-c3ccc(Br)cc3)cs2)cs1 ZINC000147182926 HI On-Demand Anodyne ROCK1 21 41 COCc1nc(C(=O)Nc2nc(-c3ccc(Br)cc3)cs2)cs1 ZINC000147182926 HI On-Demand Anodyne HDAC9 15 40 COCc1nc(C(=O)Nc2nc(-c3ccc(Br)cc3)cs2)cs1 ZINC000147182926 HI On-Demand Anodyne TRPA1 15 43 Nc1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)n1 ZINC000147182996 JA Annotated Anodyne POLA1 47 55 Nc1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)n1 ZINC000147182996 JA Annotated Anodyne P2RY6 129 47 Nc1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)n1 ZINC000147182996 JA Annotated Anodyne POLB 58 55 Nc1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)n1 ZINC000147182996 JA Annotated Anodyne P2RX4 42 38 Nc1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)n1 ZINC000147182996 JA Annotated Anodyne P2RX1 58 38 Nc1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)n1 ZINC000147182996 JA Annotated Anodyne P2RY4 134 47 Nc1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)n1 ZINC000147182996 JA Annotated Anodyne P2RY1 31 40 Nc1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)n1 ZINC000147182996 JA Annotated Anodyne P2RY2 170 51 Nc1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)n1 ZINC000147182996 JA Annotated Anodyne P2RY14 54 39 Nc1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)n1 ZINC000147182996 JA Annotated Anodyne GPR17 46 35 C[C@@H]1CN(Cc2ccccc2NC(=O)COc2ccc(C(N)=O)cc2)C[C@@H](C)O1 ZINC000147183056 GE On-Demand Anodyne CYSLTR2 45 33 C[C@@H]1CN(Cc2ccccc2NC(=O)COc2ccc(C(N)=O)cc2)C[C@@H](C)O1 ZINC000147183056 GE On-Demand Anodyne ITGA4 43 33 CC[C@H](NCc1ccc(OC)c(OCCCC#N)c1)c1ccc2c(c1)OCCO2 ZINC000147183221 GI On-Demand Mild PDE10A 22 43 Cc1cc(C)nc(NC(=O)N2CCO[C@@H](COc3ccccc3)C2)c1 ZINC000147183245 EG On-Demand Anodyne COLA 40 34 Cc1cc(C)cc(S(=O)(=O)c2sc3ncccc3c2-c2ccc(Cl)cc2)c1 ZINC000147183313 HK Annotated Anodyne GRM5 40 84 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N[C@H]1CCCC[C@H]1C ZINC000147183417 HF On-Demand Mild L3MBTL3 64 34 Cc1cc(C)nc(NC(=O)N2CCO[C@H](COc3ccccc3)C2)c1 ZINC000147183422 EG On-Demand Anodyne ADAM17 54 37 Cc1cc(C)nc(NC(=O)N2CCO[C@H](COc3ccccc3)C2)c1 ZINC000147183422 EG On-Demand Anodyne COLA 40 34 Cc1cc(C)nc(NC(=O)N2CCO[C@H](COc3ccccc3)C2)c1 ZINC000147183422 EG On-Demand Anodyne ITGA4 40 33 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCC(C(N)=O)CC3)c2)cc1 ZINC000147183456 HD On-Demand Anodyne ACHE 26 41 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCC(C(N)=O)CC3)c2)cc1 ZINC000147183456 HD On-Demand Anodyne HRH2 59 43 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCC(C(N)=O)CC3)c2)cc1 ZINC000147183456 HD On-Demand Anodyne LTA4H 40 46 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCC(C(N)=O)CC3)c2)cc1 ZINC000147183456 HD On-Demand Anodyne SIGMAR1 29 44 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCC(C(N)=O)CC3)c2)cc1 ZINC000147183456 HD On-Demand Anodyne CHEK2 38 41 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCC(C(N)=O)CC3)c2)cc1 ZINC000147183456 HD On-Demand Anodyne CCR3 55 45 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCC(C(N)=O)CC3)c2)cc1 ZINC000147183456 HD On-Demand Anodyne ST14 41 39 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCC(C(N)=O)CC3)c2)cc1 ZINC000147183456 HD On-Demand Anodyne MCHR1 55 45 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCC(C(N)=O)CC3)c2)cc1 ZINC000147183456 HD On-Demand Anodyne HIF1A 26 44 NC(=O)c1ccc(OCC(=O)Nc2cccc(CN3CCC(C(N)=O)CC3)c2)cc1 ZINC000147183456 HD On-Demand Anodyne NPFFR1 43 35 CCOC(=O)c1cnc(-c2ccccc2C)nc1N1CCCCC1 ZINC000147183501 EH For-Sale Anodyne P2RY12 61 43 CCOC(=O)c1cnc(-c2ccccc2C)nc1N1CCCCC1 ZINC000147183501 EH For-Sale Anodyne JUN 17 40 C[C@H]1CN[C@H](C(=O)O)[C@@H](CC(=O)O)C1 ZINC000147183514 BC For-Sale Anodyne GRIK3 18 66 C[C@H]1CN[C@H](C(=O)O)[C@@H](CC(=O)O)C1 ZINC000147183514 BC For-Sale Anodyne GRIK2 100 50 C[C@H]1CN[C@H](C(=O)O)[C@@H](CC(=O)O)C1 ZINC000147183514 BC For-Sale Anodyne GRIK4 0 50 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N[C@H]1CCCC[C@@H]1C ZINC000147183619 HF On-Demand Mild L3MBTL3 64 34 Cc1ccc(Br)cc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147183655 FF On-Demand Anodyne HIF1A 24 41 CC(C)C[C@H](Nc1nc(CCl)nc2ccccc12)C(N)=O ZINC000147183704 DF For-Sale Reactive CAPNS1 56 33 CC(C)C[C@H](Nc1nc(CCl)nc2ccccc12)C(N)=O ZINC000147183704 DF For-Sale Reactive HLA-DRB1 47 34 CC(C)C[C@H](Nc1nc(CCl)nc2ccccc12)C(N)=O ZINC000147183704 DF For-Sale Reactive CAPN2 52 35 CC(C)C[C@H](Nc1nc(CCl)nc2ccccc12)C(N)=O ZINC000147183704 DF For-Sale Reactive NPR 57 34 CC(C)C[C@H](Nc1nc(CCl)nc2ccccc12)C(N)=O ZINC000147183704 DF For-Sale Reactive CX3CR1 37 46 CC(C)C[C@H](Nc1nc(CCl)nc2ccccc12)C(N)=O ZINC000147183704 DF For-Sale Reactive KISS1R 61 34 C[C@@H]1CN[C@H](C(=O)O)[C@@H](CC(=O)O)C1 ZINC000147183719 BC For-Sale Anodyne GRIK3 18 66 C[C@@H]1CN[C@H](C(=O)O)[C@@H](CC(=O)O)C1 ZINC000147183719 BC For-Sale Anodyne GRIK2 100 50 C[C@@H]1CN[C@H](C(=O)O)[C@@H](CC(=O)O)C1 ZINC000147183719 BC For-Sale Anodyne GRIK4 0 50 COc1ccc(C)cc1-n1ccc(C(=O)Nc2ccccn2)n1 ZINC000147183789 DF On-Demand Anodyne GRM4 35 44 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N[C@@H]1CCCC[C@H]1C ZINC000147183812 HF On-Demand Mild L3MBTL3 64 34 COc1ccccc1[C@H](C)NC(=O)N(C)Cc1cscn1 ZINC000147183884 DG On-Demand Anodyne CYP3A4 19 45 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(Cl)ccc1N1CCCCC1 ZINC000147184012 GF On-Demand Anodyne CNR1 52 32 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(Cl)ccc1N1CCCCC1 ZINC000147184012 GF On-Demand Anodyne KCNQ2 59 39 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N[C@@H]1CCCC[C@@H]1C ZINC000147184016 HF On-Demand Mild L3MBTL3 64 34 CCCC[C@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184060 FG On-Demand Anodyne GHRHR 43 34 CCCC[C@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184060 FG On-Demand Anodyne CTSB 40 31 CCCC[C@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184060 FG On-Demand Anodyne CTSK 27 41 CCCC[C@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184060 FG On-Demand Anodyne MMP3 37 42 CCCC[C@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184060 FG On-Demand Anodyne HLA-DRB1 44 34 CCCC[C@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184060 FG On-Demand Anodyne CTRB_BOVIN 45 33 CCCC[C@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184060 FG On-Demand Anodyne PLM2_PLAFA 39 42 CCCC[C@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184060 FG On-Demand Anodyne AMP1_PLAFQ 22 44 CCCC[C@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184060 FG On-Demand Anodyne POLG_WNV 47 33 CCCC[C@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184060 FG On-Demand Anodyne NPFFR1 40 31 COc1ccccc1[C@@H](C)NC(=O)N(C)Cc1cscn1 ZINC000147184090 DG On-Demand Anodyne CYP3A4 19 45 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147184162 FH On-Demand Anodyne KCNQ2 80 47 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147184162 FH On-Demand Anodyne TRY2_BOVIN 55 35 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147184162 FH On-Demand Anodyne CCKAR 46 38 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147184162 FH On-Demand Anodyne ACPS 0 47 CCCCCCOc1ccc(C(=N)NO)cc1C(F)(F)F ZINC000147184185 DH For-Sale Anodyne S1PR4 20 42 CCCCCCOc1ccc(C(=N)NO)cc1C(F)(F)F ZINC000147184185 DH For-Sale Anodyne PLA2G4B 54 39 CCCCCCOc1ccc(C(=N)NO)cc1C(F)(F)F ZINC000147184185 DH For-Sale Anodyne S1PR2 40 36 CCCCCCOc1ccc(C(=N)NO)cc1C(F)(F)F ZINC000147184185 DH For-Sale Anodyne ACR 26 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(Cl)ccc1N1CCCCC1 ZINC000147184197 GF On-Demand Anodyne CNR1 52 32 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(Cl)ccc1N1CCCCC1 ZINC000147184197 GF On-Demand Anodyne KCNQ2 59 39 N#CC1CCN(C(=O)c2cccc(NS(=O)(=O)c3ccccc3)c2)CC1 ZINC000147184245 FF On-Demand Mild CACNA1B 19 40 N#CC1CCN(C(=O)c2cccc(NS(=O)(=O)c3ccccc3)c2)CC1 ZINC000147184245 FF On-Demand Mild ST14 82 38 N#CC1CCN(C(=O)c2cccc(NS(=O)(=O)c3ccccc3)c2)CC1 ZINC000147184245 FF On-Demand Mild AKR1C3 33 44 N#CC1CCN(C(=O)c2cccc(NS(=O)(=O)c3ccccc3)c2)CC1 ZINC000147184245 FF On-Demand Mild SFRP1 93 41 N#CC1CCN(C(=O)c2cccc(NS(=O)(=O)c3ccccc3)c2)CC1 ZINC000147184245 FF On-Demand Mild LIMK2 37 42 N#CC1CCN(C(=O)c2cccc(NS(=O)(=O)c3ccccc3)c2)CC1 ZINC000147184245 FF On-Demand Mild WNT3 71 37 N#CC1CCN(C(=O)c2cccc(NS(=O)(=O)c3ccccc3)c2)CC1 ZINC000147184245 FF On-Demand Mild L3MBTL3 59 41 CCCC[C@@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184254 FG On-Demand Anodyne GHRHR 43 34 CCCC[C@@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184254 FG On-Demand Anodyne CTSB 40 31 CCCC[C@@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184254 FG On-Demand Anodyne CTSK 27 41 CCCC[C@@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184254 FG On-Demand Anodyne MMP3 37 42 CCCC[C@@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184254 FG On-Demand Anodyne HLA-DRB1 44 34 CCCC[C@@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184254 FG On-Demand Anodyne CTRB_BOVIN 45 33 CCCC[C@@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184254 FG On-Demand Anodyne PLM2_PLAFA 39 42 CCCC[C@@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184254 FG On-Demand Anodyne AMP1_PLAFQ 22 44 CCCC[C@@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184254 FG On-Demand Anodyne POLG_WNV 47 33 CCCC[C@@H](NC(N)=O)C(=O)N(CCc1ccccc1)Cc1ccccc1 ZINC000147184254 FG On-Demand Anodyne NPFFR1 40 31 COc1cccc(CN(C)C(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147184277 DG On-Demand Bother CACNA1D 71 36 COc1cccc(CN(C)C(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147184277 DG On-Demand Bother ROCK1 28 45 COc1cccc(CN(C)C(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147184277 DG On-Demand Bother ROCK2 33 40 COc1cccc(CN(C)C(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147184277 DG On-Demand Bother HSP90AB1 16 41 COc1cccc(CN(C)C(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147184277 DG On-Demand Bother HSD17B2 42 63 O=C(c1ccc2c(c1)COC2)N1CCC[C@H]1C1CCCCC1 ZINC000147184300 CH On-Demand Anodyne PREP 25 40 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne ACE 69 46 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne OPRM1 19 41 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne OPRD1 27 44 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne MME 98 44 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne ANPEP 63 38 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne CTSB 17 42 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne CPA1 53 44 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne ITGA4 73 37 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne NAALAD2 33 47 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne ECE1 38 41 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne CAPN1 51 43 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne CAPN2 16 42 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne ACE2 100 43 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne LAP3 15 40 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne FPR1 60 40 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne BLA1_STEMA 70 38 O=C(N[C@H](Cc1ccccc1)C(=O)O)[C@@H]1Cc2ccccc2S1 ZINC000147184378 EF On-Demand Anodyne BRCA1 44 32 CCN(CC)C(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147184388 FD On-Demand Anodyne OXTR 26 40 CCN(CC)C(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147184584 FD On-Demand Anodyne OXTR 26 40 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne ACE 69 46 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne OPRM1 19 41 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne OPRD1 27 44 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne MME 98 44 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne ANPEP 63 38 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne CTSB 17 42 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne CPA1 53 44 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne ITGA4 73 37 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne NAALAD2 33 47 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne ECE1 38 41 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne CAPN1 51 43 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne CAPN2 16 42 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne ACE2 100 43 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne LAP3 15 40 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne FPR1 60 40 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne BLA1_STEMA 70 38 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1Cc2ccccc2S1 ZINC000147184588 EF On-Demand Anodyne BRCA1 44 32 COc1ccc2c(c1)OC[C@H](C(=O)N1CCC(C(=O)Nc3nncs3)CC1)C2 ZINC000147184703 HD On-Demand Anodyne ROCK2 35 45 CC(C)Cc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147184732 EI On-Demand Anodyne BMP1 57 36 CC(C)Cc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147184732 EI On-Demand Anodyne ACACA 40 36 CC(C)Cc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147184732 EI On-Demand Anodyne CYP3A4 21 48 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne ACE 69 46 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne OPRM1 19 41 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne OPRD1 27 44 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne MME 98 44 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne ANPEP 63 38 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne CTSB 17 42 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne CPA1 53 44 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne ITGA4 73 37 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne NAALAD2 33 47 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne ECE1 38 41 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne CAPN1 51 43 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne CAPN2 16 42 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne ACE2 100 43 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne LAP3 15 40 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne FPR1 60 40 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne BLA1_STEMA 70 38 O=C(O)[C@H](Cc1ccccc1)NC(=O)[C@H]1Cc2ccccc2S1 ZINC000147184768 EF On-Demand Anodyne BRCA1 44 32 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne LTA4H 32 42 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne LDHA 32 43 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne HDAC8 24 42 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne HDAC10 27 41 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne HDAC1 18 50 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne HDAC2 25 50 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne HDAC3 30 41 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne HDAC6 26 41 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne ALOX15 0 43 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne PTPRF 44 38 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne SLC1A2 40 34 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne HCAR2 31 41 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne HDA106 0 41 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne AKR1C2 47 33 Cc1cc(NC(=O)CCCc2ccccc2)ccc1C(=O)O ZINC000147184799 CH On-Demand Anodyne PFHDAC1 0 41 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC(C(=O)Nc3nncs3)CC1)C2 ZINC000147184874 HD On-Demand Anodyne ROCK2 35 45 CC(C)CN(c1ccc(F)cc1)S(=O)(=O)c1ccc(Cl)nc1 ZINC000147184910 EH For-Sale Anodyne RORC 26 48 CC(C)Cc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147184917 EI On-Demand Anodyne BMP1 57 36 CC(C)Cc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147184917 EI On-Demand Anodyne ACACA 40 36 CC(C)Cc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147184917 EI On-Demand Anodyne CYP3A4 21 48 CCc1ccc2nc(NC(=O)c3cnc(CC)s3)sc2c1 ZINC000147185059 DI On-Demand Anodyne LCK 38 42 CCc1ccc2nc(NC(=O)c3cnc(CC)s3)sc2c1 ZINC000147185059 DI On-Demand Anodyne CSNK1D 49 46 CCc1ccc2nc(NC(=O)c3cnc(CC)s3)sc2c1 ZINC000147185059 DI On-Demand Anodyne PIK3CA 21 43 CCc1ccc2nc(NC(=O)c3cnc(CC)s3)sc2c1 ZINC000147185059 DI On-Demand Anodyne HSD17B1 29 42 C[C@@H](NC(=O)OC(C)(C)C)/C(Cl)=N/O ZINC000147185064 BD For-Sale Mild CTSK 27 49 CC(C)(C)NC(=O)c1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147185116 HF On-Demand Bother TAAR1 35 42 CC(C)(C)NC(=O)c1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147185116 HF On-Demand Bother AKR1C3 17 40 CC(C)(C)NC(=O)c1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147185116 HF On-Demand Bother UREA_CANEN 16 42 CC(C)(C)NC(=O)c1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147185116 HF On-Demand Bother KCNK3 96 39 CC(C)(C)NC(=O)c1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147185116 HF On-Demand Bother KCNK9 48 39 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild F2 35 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild PLG 34 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild ACE 53 45 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild OPRM1 22 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild P2RY12 104 36 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild MME 59 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild UGCG 49 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild MC4R 141 51 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CTRA_BOVIN 24 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CTSB 36 49 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild TRY2_BOVIN 82 35 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild PAPA1_CARPA 27 48 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CCKAR 56 38 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CTSL 37 48 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CCR1 54 56 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CCR3 0 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CYP51A1 27 48 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild TIMP3 41 36 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild PYGL 15 53 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild DPP4 19 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild PREP 19 55 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild MC3R 66 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild MC5R 89 44 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CCKBR 33 47 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CTSS 29 48 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CAPN1 40 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild ACE2 66 38 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild MC1R 28 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild DPP7 49 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CTSV 49 48 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild ST14 104 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild CTRB_BOVIN 51 36 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild AMP1_PLAFQ 19 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild DPP8 22 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild DPP9 15 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild FAP 0 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild BLA1_STEMA 60 37 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild UTS2 50 43 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccc(Cl)cc2)CC1 ZINC000147185179 GG On-Demand Mild TMPRSS6 57 38 O=C(Nc1nncs1)C1CCN(C(=O)c2ccc3c(c2)COC3)CC1 ZINC000147185265 FE On-Demand Anodyne L3MBTL3 65 36 CC(C)c1nccn1Cc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147185300 GG On-Demand Anodyne ADORA2B 34 40 CCOc1cc(C(=O)N2CCC(C#N)CC2)ccc1OCC(=O)N1CCCCC1 ZINC000147185422 GF On-Demand Mild L3MBTL3 76 37 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(-n3cccn3)c(F)c1)C2 ZINC000147185494 FG On-Demand Anodyne NPY2R 40 36 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(-n3cccn3)c(F)c1)C2 ZINC000147185494 FG On-Demand Anodyne ROCK2 35 49 CN1CCCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147185502 GD On-Demand Anodyne HTR1B 22 43 CN1CCCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147185502 GD On-Demand Anodyne ADORA2B 44 45 CN1CCCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147185502 GD On-Demand Anodyne LCK 18 40 CN1CCCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147185502 GD On-Demand Anodyne PRNP 42 46 CN1CCCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147185502 GD On-Demand Anodyne HCK 16 40 CN1CCCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147185502 GD On-Demand Anodyne ACR 62 39 CN1CCCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147185502 GD On-Demand Anodyne FLT3 22 41 CN1CCCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147185502 GD On-Demand Anodyne MCHR1 20 49 CN1CCCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147185502 GD On-Demand Anodyne AURKA 18 41 CN1CCCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147185502 GD On-Demand Anodyne HIF1A 25 40 CN1CCCN(c2ccc(NC(=O)COc3ccc(C(N)=O)cc3)cc2)CC1 ZINC000147185502 GD On-Demand Anodyne STAT6 26 40 Cc1nnc(C)n1-c1ccccc1N ZINC000147185540 AD For-Sale Anodyne SLC6A5 28 46 COCc1nc(C(=O)Nc2ccc3c(c2)Cc2ccccc2-3)cs1 ZINC000147185551 EI On-Demand Anodyne GRM4 42 37 COCc1nc(C(=O)Nc2ccc3c(c2)Cc2ccccc2-3)cs1 ZINC000147185551 EI On-Demand Anodyne SLC1A1 25 46 COCc1nc(C(=O)Nc2ccc3c(c2)Cc2ccccc2-3)cs1 ZINC000147185551 EI On-Demand Anodyne SLC1A3 29 46 COCc1nc(C(=O)Nc2ccc3c(c2)Cc2ccccc2-3)cs1 ZINC000147185551 EI On-Demand Anodyne SLC1A2 23 46 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(-n3cccn3)c(F)c1)C2 ZINC000147185702 FG On-Demand Anodyne NPY2R 40 36 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(-n3cccn3)c(F)c1)C2 ZINC000147185702 FG On-Demand Anodyne ROCK2 35 49 CCOc1ccc(Oc2ccccc2NC(=O)c2csc(COC)n2)cc1 ZINC000147185753 GJ On-Demand Anodyne PYGM 31 44 CC(C)CN(C)C(=O)c1nc2ccccc2nc1O ZINC000147186021 CE For-Sale Anodyne TSPO 23 47 COc1ccc(CNCc2ccc([C@@H](C)O)cc2)cc1OCCCC#N ZINC000147186093 FH On-Demand Mild MT-ND1 16 41 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild OPRM1 18 52 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild OPRD1 25 52 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild ANPEP 16 44 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild NPR1 53 47 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild EDNRB 27 42 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild EDNRA 24 42 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild HLA-DRB3 15 43 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild MC4R 44 55 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild KLK3 45 30 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild CTSB 37 51 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild PAPA1_CARPA 76 51 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild RIR1_HHV11 55 34 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild NTSR1 144 63 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild NTSR2 106 45 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild F2R 48 47 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild ADRBK1 18 53 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild C3AR1 39 42 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild HLA-A 101 47 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild MC3R 49 55 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild MC5R 71 55 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild HLA-DRB1 73 45 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild REN 16 41 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild LNPEP 22 42 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild FURIN 53 47 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild SORT1 58 41 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild CAPN1 25 49 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild CAPN2 55 33 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild ENPEP 71 36 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild MC1R 88 55 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild FPR1 43 34 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild SIRT1 26 41 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild PSMB2 45 39 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild F2RL1 67 42 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild WDR5 16 46 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild Q9NAW4_PLAFA 16 49 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild HPN 58 41 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147186100 KA For-Sale Mild H9B8T9_CAPHI 47 49 N#Cc1c(-c2ccccc2)[nH]c(SCc2cccc(F)c2F)nc1=O ZINC000147186255 FH Annotated Mild CTSB 18 45 N#Cc1c(-c2ccccc2)[nH]c(SCc2cccc(F)c2F)nc1=O ZINC000147186255 FH Annotated Mild NS5B 21 41 NC(=O)[C@H]1CCCN(C(=O)c2ccc(S(=O)(=O)NCc3ccco3)cc2)C1 ZINC000147186273 GD On-Demand Anodyne SFRP1 41 34 NC(=O)[C@@H]1CCCN(C(=O)c2ccc(S(=O)(=O)NCc3ccco3)cc2)C1 ZINC000147186482 GD On-Demand Anodyne SFRP1 41 34 O=S(=O)(c1ccc(C(F)(F)F)cc1)c1sc2ncccc2c1-c1ccc(Cl)cc1 ZINC000147186496 JK Annotated Anodyne GRM5 45 83 N#Cc1ccc(-c2c(S(=O)(=O)c3cccc(C#N)c3)sc3ncccc23)cc1 ZINC000147186685 HJ Annotated Mild GRM5 47 88 COC(=O)CNC(=O)c1cc(Br)c(O)c(Br)c1 ZINC000147186756 FD On-Demand Anodyne SLC22A12 74 36 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCCC3)cc2)s1 ZINC000147186781 GH On-Demand Anodyne GSK3B 15 42 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCCC3)cc2)s1 ZINC000147186781 GH On-Demand Anodyne GRM4 20 49 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCCC3)cc2)s1 ZINC000147186781 GH On-Demand Anodyne EPHX2 19 40 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCCC3)cc2)s1 ZINC000147186781 GH On-Demand Anodyne TGM2 80 43 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCCC3)cc2)s1 ZINC000147186781 GH On-Demand Anodyne F13A1 93 47 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCCC3)cc2)s1 ZINC000147186781 GH On-Demand Anodyne MERTK 31 44 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCCC3)cc2)s1 ZINC000147186781 GH On-Demand Anodyne NAMPT 60 48 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCCCCC3)cc2)s1 ZINC000147186781 GH On-Demand Anodyne USP47 41 34 N#CC1CCN(C(=O)CSc2nnc(-c3cccnc3)n2-c2ccccc2)CC1 ZINC000147187035 HG On-Demand Mild PTAFR 27 42 N#CC1CCN(C(=O)CSc2nnc(-c3cccnc3)n2-c2ccccc2)CC1 ZINC000147187035 HG On-Demand Mild C3AR1 40 34 N#CC1CCN(C(=O)CSc2nnc(-c3cccnc3)n2-c2ccccc2)CC1 ZINC000147187035 HG On-Demand Mild VCP 47 34 CC1(C)Cc2cc(Cl)ccc2N[C@@H]1c1cccc([N+](=O)[O-])c1 ZINC000147187175 DJ For-Sale Anodyne CACNA1C 59 38 CC1(C)Cc2cc(Cl)ccc2N[C@@H]1c1cccc([N+](=O)[O-])c1 ZINC000147187175 DJ For-Sale Anodyne CACNA1D 93 38 CC1(C)Cc2cc(Cl)ccc2N[C@H]1c1cccc([N+](=O)[O-])c1 ZINC000147187349 DJ For-Sale Anodyne CACNA1C 59 38 CC1(C)Cc2cc(Cl)ccc2N[C@H]1c1cccc([N+](=O)[O-])c1 ZINC000147187349 DJ For-Sale Anodyne CACNA1D 93 38 O=C(O)CN1N[C@H](Cc2nc3cc(C(F)(F)F)ccc3s2)C(=O)C2=C1[C@@H]1CCCC[C@@H]21 ZINC000147187356 JH For-Sale Anodyne AKR1B1 20 44 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147187460 HG On-Demand Anodyne LPL 65 37 CCn1c(SCC(=O)N2CCC(C#N)CC2)nnc1-c1cccs1 ZINC000147187508 FF On-Demand Mild ETHR 43 38 CCOC(=O)c1cnc(-c2ccccc2Cl)nc1NC ZINC000147187527 CG For-Sale Anodyne ADORA1 16 42 CCOC(=O)c1cnc(-c2ccccc2Cl)nc1NC ZINC000147187527 CG For-Sale Anodyne JUN 19 48 CCOC(=O)c1cnc(-c2ccccc2Cl)nc1NC ZINC000147187527 CG For-Sale Anodyne ADORA3 17 42 CN(Cc1cscn1)C(=O)NCC1(N2CCOCC2)CCCCC1 ZINC000147187555 FE On-Demand Anodyne HCN1 57 36 CN(Cc1cscn1)C(=O)NCC1(N2CCOCC2)CCCCC1 ZINC000147187555 FE On-Demand Anodyne HCN4 54 36 O=C(Nc1cccnc1)c1ccccc1N1CCCCC1 ZINC000147187660 CG On-Demand Anodyne AVPR2 42 39 O=C(Nc1cccnc1)c1ccccc1N1CCCCC1 ZINC000147187660 CG On-Demand Anodyne KCNQ2 78 38 O=C(Nc1cccnc1)c1ccccc1N1CCCCC1 ZINC000147187660 CG On-Demand Anodyne NPY2R 25 42 O=C(Nc1cccnc1)c1ccccc1N1CCCCC1 ZINC000147187660 CG On-Demand Anodyne RPS6KA3 28 42 O=C(Nc1cccnc1)c1ccccc1N1CCCCC1 ZINC000147187660 CG On-Demand Anodyne CSF1R 31 44 O=C(Nc1cccnc1)c1ccccc1N1CCCCC1 ZINC000147187660 CG On-Demand Anodyne PIM2 15 44 O=C(Nc1cccnc1)c1ccccc1N1CCCCC1 ZINC000147187660 CG On-Demand Anodyne NAMPT 29 43 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147187680 HG On-Demand Anodyne LPL 65 37 CC(=O)N[C@@H]1Cc2ccccc2[C@H]1C ZINC000147187756 AD For-Sale Anodyne MTNR1B 0 47 CC(C)(C)OC(=O)N[C@@H]1CCCN(c2ccccc2[N+](=O)[O-])C1 ZINC000147187796 DG In-Stock Bother KCNQ2 43 31 CC(C)(C)OC(=O)N[C@@H]1CCCN(c2ccccc2[N+](=O)[O-])C1 ZINC000147187796 DG In-Stock Bother SFRP1 46 36 CC(C)(C)OC(=O)N[C@@H]1CCCN(c2ccccc2[N+](=O)[O-])C1 ZINC000147187796 DG In-Stock Bother WNT3 52 36 CCCCCCCCO[C@H](CCC)C(=O)O ZINC000147187864 BH For-Sale Mild PLA2G4B 68 37 CCCCCCCCO[C@H](CCC)C(=O)O ZINC000147187864 BH For-Sale Mild NOD1 71 37 CCCCCCCCO[C@H](CCC)C(=O)O ZINC000147187864 BH For-Sale Mild CQSS 58 40 Cc1cc(-c2ccc(C(F)(F)F)cc2)n[nH]1 ZINC000147187871 BG For-Sale Anodyne DHODH 18 41 Cc1cc(-c2ccc(C(F)(F)F)cc2)n[nH]1 ZINC000147187871 BG For-Sale Anodyne KIF11 17 44 C[C@@H](NC(=O)c1ccc2c(c1)COC2)c1cccc(OCc2ccccn2)c1 ZINC000147187921 FI On-Demand Anodyne SMO 22 41 CC(C)(C)OC(=O)N[C@H]1CCCN(c2ccccc2[N+](=O)[O-])C1 ZINC000147188009 DG In-Stock Bother KCNQ2 43 31 CC(C)(C)OC(=O)N[C@H]1CCCN(c2ccccc2[N+](=O)[O-])C1 ZINC000147188009 DG In-Stock Bother SFRP1 46 36 CC(C)(C)OC(=O)N[C@H]1CCCN(c2ccccc2[N+](=O)[O-])C1 ZINC000147188009 DG In-Stock Bother WNT3 52 36 CC(=O)N[C@H]1Cc2ccccc2[C@@H]1C ZINC000147188160 AD For-Sale Anodyne MTNR1B 0 47 NC(=O)c1ccc(OCC(=O)N2CCC(=Cc3cccc(F)c3)CC2)cc1 ZINC000147188259 FG On-Demand Anodyne COLA 15 40 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne LTA4H 36 42 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne HDAC8 22 50 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne HDAC10 20 48 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne MTNR1B 15 42 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne HDAC1 20 50 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne HDAC2 15 48 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne HDAC3 18 49 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne SLC1A2 19 45 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne HCAR2 34 50 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne MCHR1 15 41 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne VIPR1 24 40 Cc1ccc(NC(=O)CCc2ccc3ccccc3c2)cc1 ZINC000147188286 CJ On-Demand Anodyne FFAR1 23 41 CCOC(=O)c1cnc(-c2ccccc2C)nc1NC ZINC000147188341 CF For-Sale Anodyne ADORA1 16 43 CCOC(=O)c1cnc(-c2ccccc2C)nc1NC ZINC000147188341 CF For-Sale Anodyne JUN 19 49 CCOC(=O)c1cnc(-c2ccccc2C)nc1NC ZINC000147188341 CF For-Sale Anodyne ADORA3 18 43 Cc1cc(C(N)=O)c(N)nc1C ZINC000147188385 AC For-Sale Anodyne EEF2K 18 42 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccccc3F)CC2)CC1 ZINC000147188493 GD On-Demand Mild EPHX2 28 54 CC(=O)N1CC(NC(=O)[C@@H]2N[C@H](CC(C)(C)C)[C@]3(C(=O)Nc4cc(Cl)ccc43)[C@H]2c2cccc(Cl)c2F)C1 ZINC000147188556 KI Annotated Anodyne MDM2 105 70 COc1ccc(CNC[C@@H](O)COc2ccc(F)cc2)cc1OCCCC#N ZINC000147188568 GG On-Demand Mild ADRB2 38 49 COc1ccc(CNC[C@@H](O)COc2ccc(F)cc2)cc1OCCCC#N ZINC000147188568 GG On-Demand Mild ADRB1 51 45 COc1ccc(CNC[C@@H](O)COc2ccc(F)cc2)cc1OCCCC#N ZINC000147188568 GG On-Demand Mild GRIN1 16 42 COc1ccc(CNC[C@@H](O)COc2ccc(F)cc2)cc1OCCCC#N ZINC000147188568 GG On-Demand Mild ADRB3 35 42 CCC[C@@H](NC(N)=O)C(=O)N1CCC(=Cc2cccc(F)c2)CC1 ZINC000147188667 EF On-Demand Anodyne P2RY12 76 31 CCC[C@@H](NC(N)=O)C(=O)N1CCC(=Cc2cccc(F)c2)CC1 ZINC000147188667 EF On-Demand Anodyne TRY2_BOVIN 61 31 C[C@H](Sc1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147188687 DH On-Demand Mild CCR1 52 40 O=C(Nc1cnccn1)C1CCN(C(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147188749 GG On-Demand Anodyne TYK2 62 38 Cc1nn(Cc2ccccc2)c(C)c1CNC(=O)[C@@H](C)Cc1cccc(F)c1 ZINC000147188765 GI On-Demand Anodyne P2RX7 48 58 Cc1nn(Cc2ccccc2)c(C)c1CNC(=O)[C@@H](C)Cc1cccc(F)c1 ZINC000147188765 GI On-Demand Anodyne CARM1 49 36 CC(C)(C)Oc1cc(-c2ccc(CNC(=O)c3c(F)ccc(F)c3Cl)cc2)ccn1 ZINC000147188809 IK For-Sale Anodyne SUCNR1 40 39 CC(=O)N(C(C)=O)c1ccc(C(=O)c2ccc(N(C(C)=O)C(C)=O)cc2)cc1 ZINC000147188881 GF For-Sale Anodyne SRD5A2 15 46 C[C@@H](Sc1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147188886 DH On-Demand Mild CCR1 52 40 CCOC(=O)/C=C/Cc1cccc(-c2cccc(OC)c2)c1 ZINC000147188891 CI For-Sale Anodyne HSD17B2 25 44 O=C(Nc1cnccn1)C1CCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147188935 GG On-Demand Anodyne TYK2 62 38 Cc1ccc(NC(=O)c2ccccc2)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147189067 GF On-Demand Anodyne MAPK14 41 48 Cc1ccc(NC(=O)c2ccccc2)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147189067 GF On-Demand Anodyne KCNK3 86 42 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne ACE 43 41 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne OPRM1 28 42 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CELA1 30 42 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne ELANE 25 41 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne MME 45 44 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne TACR1 17 59 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CASP3 17 40 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne KLK3 76 35 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CTSB 60 41 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne PAPA1_CARPA 65 37 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CYSP_TRYCR 45 39 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CTSK 41 42 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CTSL 42 41 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne PREP 22 45 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne AMY2 43 29 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CAPNS1 78 36 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne REN 51 45 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne LGMN 46 37 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CTSS 28 41 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne GHSR 42 40 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CAPN1 97 41 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CAPN2 129 40 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne ACE2 46 32 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CTSC 35 49 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne NPR 80 36 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne CALCRL 37 44 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne XIAP 43 35 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne PSMB5 42 38 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne SLC12A5 52 34 C[C@H](NC(=O)[C@@H]1CCCN1)C(=O)OCc1ccccc1 ZINC000147189125 CC For-Sale Anodyne PFKFB3 46 37 O=C(Nc1cnccn1)C1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147189137 GG On-Demand Anodyne TYK2 62 38 COc1ccc(CNC[C@@H](O)COc2cccc(C)c2)cc1OCCCC#N ZINC000147189142 GG On-Demand Mild ADRB2 32 47 COc1ccc(CNC[C@@H](O)COc2cccc(C)c2)cc1OCCCC#N ZINC000147189142 GG On-Demand Mild ADRB1 29 47 CCOc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1OCC ZINC000147189159 FH On-Demand Anodyne BMP1 59 37 CCOc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1OCC ZINC000147189159 FH On-Demand Anodyne CYP3A4 16 44 Cc1ccc(NC(=O)c2ccccc2)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147189239 GF On-Demand Anodyne MAPK14 41 48 Cc1ccc(NC(=O)c2ccccc2)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147189239 GF On-Demand Anodyne KCNK3 86 42 CC(C)c1ccc(S(=O)(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)cc1 ZINC000147189266 HF On-Demand Mild EPHX2 21 54 CC(C)c1ccc(S(=O)(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)cc1 ZINC000147189266 HF On-Demand Mild TGM2 51 43 CC(C)c1ccc(S(=O)(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)cc1 ZINC000147189266 HF On-Demand Mild F13A1 53 43 CC(C)c1ccc(S(=O)(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)cc1 ZINC000147189266 HF On-Demand Mild NAMPT 15 44 O=C(Nc1cnccn1)C1CCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147189332 GG On-Demand Anodyne TYK2 62 38 CCOc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1OCC ZINC000147189356 FH On-Demand Anodyne BMP1 59 37 CCOc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1OCC ZINC000147189356 FH On-Demand Anodyne CYP3A4 16 44 CN(Cc1ccc(F)cc1Cl)C(=O)c1ccc(Br)cc1 ZINC000147189365 FJ On-Demand Anodyne P2RX7 58 40 O=C(NCC[C@H](O)CO)[C@@H]1N[C@H](CCC2CCCC2)[C@]2(C(=O)Nc3cc(Cl)c(F)cc32)[C@H]1c1cccc(Cl)c1 ZINC000147189411 KI Annotated Anodyne MDM2 72 79 CC(C)(C)NS(=O)(=O)c1cc(C(=O)N2CCC(C#N)CC2)ccc1Cl ZINC000147189471 GF On-Demand Mild L3MBTL3 58 34 CS(=O)(=O)c1ccc(-c2c(S(=O)(=O)c3ccc(Cl)cc3)sc3ncccc23)cc1 ZINC000147189494 JJ Annotated Anodyne PTGS1 21 41 CS(=O)(=O)c1ccc(-c2c(S(=O)(=O)c3ccc(Cl)cc3)sc3ncccc23)cc1 ZINC000147189494 JJ Annotated Anodyne PTGS2 63 45 CS(=O)(=O)c1ccc(-c2c(S(=O)(=O)c3ccc(Cl)cc3)sc3ncccc23)cc1 ZINC000147189494 JJ Annotated Anodyne GRM5 46 88 CCN1C(=O)Cn2c1nc1nc(N3CCC[C@@H](N)C3)n(Cc3cc(F)ccc3F)c1c2=O ZINC000147189547 ID Annotated Anodyne DPP4 46 51 Cc1cccc(OCc2ccc(CC#N)cc2)c1 ZINC000147189551 BH On-Demand Mild MAOB 43 42 Cc1cccc(OCc2ccc(CC#N)cc2)c1 ZINC000147189551 BH On-Demand Mild DRTS_LEIMA 33 44 Cc1cccc(OCc2ccc(CC#N)cc2)c1 ZINC000147189551 BH On-Demand Mild ACR 17 44 CCc1ccc(N2CCNCC2)c(Cl)c1 ZINC000147189704 BE For-Sale Anodyne HTR3A 29 42 CCc1ccc(N2CCNCC2)c(Cl)c1 ZINC000147189704 BE For-Sale Anodyne HTR6 22 52 CC(C)NS(=O)(=O)c1ccc(C(=O)N2CCN(C(=O)c3cccs3)CC2)cc1 ZINC000147189748 HE On-Demand Anodyne MMP13 15 44 CC(C)NS(=O)(=O)c1ccc(C(=O)N2CCN(C(=O)c3cccs3)CC2)cc1 ZINC000147189748 HE On-Demand Anodyne TRY2_BOVIN 78 39 Cc1ccc(Nc2ccc(N)cc2S(N)(=O)=O)cc1 ZINC000147189870 CD For-Sale Anodyne CA2 17 43 O=C(O)c1cc(Cl)cc(S(=O)(=O)NCCc2ccc(Cl)cc2)c1 ZINC000147189967 FG On-Demand Anodyne CA2 15 44 O=C(O)c1cc(Cl)cc(S(=O)(=O)NCCc2ccc(Cl)cc2)c1 ZINC000147189967 FG On-Demand Anodyne TBXA2R 64 50 O=C(O)c1cc(Cl)cc(S(=O)(=O)NCCc2ccc(Cl)cc2)c1 ZINC000147189967 FG On-Demand Anodyne TBXAS1 39 50 O=C(O)c1cc(Cl)cc(S(=O)(=O)NCCc2ccc(Cl)cc2)c1 ZINC000147189967 FG On-Demand Anodyne CA1 16 44 O=C(O)c1cc(Cl)cc(S(=O)(=O)NCCc2ccc(Cl)cc2)c1 ZINC000147189967 FG On-Demand Anodyne CCR1 15 44 O=C(O)c1cc(Cl)cc(S(=O)(=O)NCCc2ccc(Cl)cc2)c1 ZINC000147189967 FG On-Demand Anodyne AKR1C3 20 75 O=C(O)c1cc(Cl)cc(S(=O)(=O)NCCc2ccc(Cl)cc2)c1 ZINC000147189967 FG On-Demand Anodyne A6YCJ1_9METZ 16 41 Cc1nn(Cc2ccccc2)c(C)c1CNC(=O)[C@@H](C)OCCC(C)C ZINC000147190197 FH On-Demand Anodyne P2RX7 21 46 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)OCCO4)CC2)CC1 ZINC000147190260 HD On-Demand Mild EPHX2 15 57 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)OCCO4)CC2)CC1 ZINC000147190260 HD On-Demand Mild PKM 47 55 N#CC1CCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)OCCO4)CC2)CC1 ZINC000147190260 HD On-Demand Mild NAMPT 17 42 NC(=O)[C@H]1CCCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)OCCO4)CC2)C1 ZINC000147190321 IC On-Demand Anodyne EPHX2 15 60 NC(=O)[C@H]1CCCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)OCCO4)CC2)C1 ZINC000147190321 IC On-Demand Anodyne PKM 46 53 Cc1nn(Cc2ccccc2)c(C)c1CNC(=O)[C@H](C)OCCC(C)C ZINC000147190380 FH On-Demand Anodyne P2RX7 21 46 NC(=O)[C@@H]1CCCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)OCCO4)CC2)C1 ZINC000147190496 IC On-Demand Anodyne EPHX2 15 60 NC(=O)[C@@H]1CCCN(C(=O)C2CCN(S(=O)(=O)c3ccc4c(c3)OCCO4)CC2)C1 ZINC000147190496 IC On-Demand Anodyne PKM 46 53 CCN1C(=O)Cn2c1nc1nc(N3CCC[C@@H](N)C3)n(Cc3cc(F)ccc3C(F)(F)F)c1c2=O ZINC000147190611 JE Annotated Anodyne DPP4 42 48 O=C(N[C@H](CO)Cc1ccccc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147190633 HE On-Demand Anodyne CA2 16 43 O=C(N[C@H](CO)Cc1ccccc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147190633 HE On-Demand Anodyne MAP1 71 38 O=C(N[C@H](CO)Cc1ccccc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147190633 HE On-Demand Anodyne LIMK2 46 36 Cc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147190689 GF On-Demand Mild TGM2 16 40 Cc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147190689 GF On-Demand Mild ST14 58 34 Cc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147190689 GF On-Demand Mild F13A1 20 40 Cc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147190689 GF On-Demand Mild CCR8 62 32 Cc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147190689 GF On-Demand Mild SFRP1 103 36 Cc1ccc(S(=O)(=O)NCc2ccccc2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147190689 GF On-Demand Mild WNT3 69 33 COc1cc(CN(C(=O)Cc2cccc(OC(C)C)c2)C2CC2)ccc1OC(F)F ZINC000147190793 HJ On-Demand Anodyne SLC6A9 24 40 CCCCCCO[C@@H](C)c1cccc(-c2csc(NC(=O)c3cc(Cl)c(/C=C(/C)C(=O)O)c(Cl)c3)n2)c1OC ZINC000147190840 KK In-Stock Anodyne MPL 49 40 O=c1cc(O)c2cc(O)c(O)cc2o1 ZINC000147190875 AC For-Sale Clean HSD17B3 27 44 CCN(CC(=O)NCc1ccc(F)cc1)C(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147190901 FF On-Demand Bother MMP8 19 42 CCN(CC(=O)NCc1ccc(F)cc1)C(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147190901 FF On-Demand Bother MMP1 20 42 O=C(NCc1ccc(OCc2ccccn2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147191013 GJ On-Demand Anodyne SCN9A 21 42 N#CC1CCN(C(=O)Cc2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2)CC1 ZINC000147191135 HF On-Demand Mild TBXA2R 15 40 N#CC1CCN(C(=O)Cc2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2)CC1 ZINC000147191135 HF On-Demand Mild HTR6 16 41 N#CC1CCN(C(=O)Cc2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2)CC1 ZINC000147191135 HF On-Demand Mild MLNR 46 48 N#CC1CCN(C(=O)Cc2ccc(NS(=O)(=O)c3ccc(F)cc3)cc2)CC1 ZINC000147191135 HF On-Demand Mild LIMK2 27 41 O=C(NCc1ccc(OCc2ccccn2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147191167 GJ On-Demand Anodyne SCN9A 21 42 CN1C(=O)Cn2c1nc1nc(N3CCC[C@@H](N)C3)n(Cc3cc(F)ccc3C#N)c1c2=O ZINC000147191211 IC Annotated Mild DPP4 52 65 O=C(NCc1ccc(OCc2ccccn2)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147191316 GJ On-Demand Anodyne SCN9A 21 42 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc(OC[C@@H]2CCCO2)cc1 ZINC000147191397 HH On-Demand Anodyne PRTN3 40 35 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc(OC[C@@H]2CCCO2)cc1 ZINC000147191397 HH On-Demand Anodyne CCR8 44 33 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCCC[C@@H]1C ZINC000147191399 EH For-Sale Anodyne P2RY12 72 39 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCCC[C@@H]1C ZINC000147191399 EH For-Sale Anodyne JUN 18 47 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCCC[C@@H]1C ZINC000147191399 EH For-Sale Anodyne COLA 76 39 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCCC[C@@H]1C ZINC000147191399 EH For-Sale Anodyne CPT1A 75 39 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCCC[C@@H]1C ZINC000147191399 EH For-Sale Anodyne ADORA3 28 40 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCCC[C@H]1C ZINC000147191567 EH For-Sale Anodyne P2RY12 72 39 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCCC[C@H]1C ZINC000147191567 EH For-Sale Anodyne JUN 18 47 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCCC[C@H]1C ZINC000147191567 EH For-Sale Anodyne COLA 76 39 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCCC[C@H]1C ZINC000147191567 EH For-Sale Anodyne CPT1A 75 39 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCCC[C@H]1C ZINC000147191567 EH For-Sale Anodyne ADORA3 28 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(OCc3ccccn3)cc1)C2 ZINC000147191568 HH On-Demand Anodyne ROCK2 29 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(OCc3ccccn3)cc1)C2 ZINC000147191568 HH On-Demand Anodyne FAAH 15 49 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne F2 15 41 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne ACE 47 35 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne OPRM1 46 46 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne OPRD1 41 46 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne OPRK1 0 45 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne MME 68 42 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne ANPEP 50 33 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne TRY2_BOVIN 51 33 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne SLC15A1 0 46 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne AKT3 24 45 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne TPH1 45 31 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne DPP4 23 53 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne DNPEP 0 42 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne DPP7 88 48 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne LAP3 56 39 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne AKT1 27 53 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne AMP1_PLAFQ 38 43 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne DPP8 51 49 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne DPP9 27 49 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne FAP 0 44 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne SLC15A2 0 44 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne AKT1S1 0 45 N[C@@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147191576 BC For-Sale Anodyne BLAIMP-1 0 41 CCCCC(C)(C)C[C@H]1N[C@@H](C(=O)NCC[C@H](O)CO)[C@H](c2cccc(Cl)c2)[C@@]12C(=O)Nc1cc(Cl)c(F)cc12 ZINC000147191694 KJ Annotated Anodyne MDM2 79 84 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(-c3nccs3)c1)C2 ZINC000147191781 FI On-Demand Anodyne ROCK2 37 48 CNCCCc1nc2c(C(=O)OC)cccc2[nH]1 ZINC000147191943 BD For-Sale Anodyne PARP1 52 41 CC(C)[C@@H](NCc1ccc(-c2ccccc2C#N)cc1)C(=O)OCc1ccccc1 ZINC000147192096 GK For-Sale Mild MME 20 42 CC(C)[C@@H](NCc1ccc(-c2ccccc2C#N)cc1)C(=O)OCc1ccccc1 ZINC000147192096 GK For-Sale Mild CTSB 53 38 CC(C)[C@@H](NCc1ccc(-c2ccccc2C#N)cc1)C(=O)OCc1ccccc1 ZINC000147192096 GK For-Sale Mild PAPA1_CARPA 55 38 CC(C)[C@@H](NCc1ccc(-c2ccccc2C#N)cc1)C(=O)OCc1ccccc1 ZINC000147192096 GK For-Sale Mild CTSK 20 44 CC(C)[C@@H](NCc1ccc(-c2ccccc2C#N)cc1)C(=O)OCc1ccccc1 ZINC000147192096 GK For-Sale Mild ADAMTS4 45 36 CC(C)[C@@H](NCc1ccc(-c2ccccc2C#N)cc1)C(=O)OCc1ccccc1 ZINC000147192096 GK For-Sale Mild NPR 56 35 COCCOCc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147192169 HE On-Demand Bother CACNA1D 48 39 COCCOCc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147192169 HE On-Demand Bother TAAR1 30 47 COCCOCc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147192169 HE On-Demand Bother KCNK3 59 33 CC(=O)c1cccc(NC(=O)Cc2ccc(Cl)cc2)c1O ZINC000147192171 DG On-Demand Anodyne KCNQ2 27 49 COc1ccc(N2CCOCC2)c2sc(NC(=O)c3ccc(OC(F)(F)F)cc3)nc12 ZINC000147192231 JI For-Sale Clean ADORA2B 21 54 COc1ccc(N2CCOCC2)c2sc(NC(=O)c3ccc(OC(F)(F)F)cc3)nc12 ZINC000147192231 JI For-Sale Clean PPARD 17 41 COc1ccc(N2CCOCC2)c2sc(NC(=O)c3ccc(OC(F)(F)F)cc3)nc12 ZINC000147192231 JI For-Sale Clean SHH 49 37 CCOC(=O)c1cnc(-c2ccccc2C)nc1N1CCCC1 ZINC000147192261 DG For-Sale Anodyne P2RY12 62 43 CCOC(=O)c1cnc(-c2ccccc2C)nc1N1CCCC1 ZINC000147192261 DG For-Sale Anodyne JUN 17 40 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147192527 GC On-Demand Anodyne BDKRB1 15 50 CN[C@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147192529 BE For-Sale Anodyne DRD2 19 46 CN[C@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147192529 BE For-Sale Anodyne DRD4 19 48 CN[C@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147192529 BE For-Sale Anodyne DRD3 16 48 CN[C@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147192529 BE For-Sale Anodyne SLC6A3 29 49 CN[C@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147192529 BE For-Sale Anodyne SLC18A2 41 37 CN[C@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147192529 BE For-Sale Anodyne KCNH2 28 43 CN[C@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147192529 BE For-Sale Anodyne SIGMAR1 41 56 CN[C@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147192529 BE For-Sale Anodyne ACHP_LYMST 22 49 CN[C@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147192529 BE For-Sale Anodyne ARG1 30 42 CN[C@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147192529 BE For-Sale Anodyne ARG2 30 42 CN[C@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147192529 BE For-Sale Anodyne Q8WSF8_APLCA 24 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne FOLH1 19 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne MME 19 44 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne NPR1 41 33 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne CA1 49 36 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne KLK3 64 39 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne CTSK 40 45 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne NPFFR2 45 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne TIMP3 65 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne C3AR1 44 31 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne HDAC8 27 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne HDAC10 47 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne MMP2 23 52 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne MMP3 49 51 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne HLA-DRB1 33 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne SOAT1 27 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne HDAC1 22 45 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne HDAC2 32 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne HDAC3 31 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne HDAC6 33 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne PCSK5 41 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne FURIN 69 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne CCKBR 16 44 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne ACE2 41 39 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne HDAC11 62 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne POLG_WNV 69 33 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne MTCA1 25 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne P96878_MYCTU 36 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192557 GG On-Demand Anodyne NPFFR1 62 34 N=C(N)Nc1ccc(CC(=O)Cl)cc1 ZINC000147192617 BD For-Sale Reactive FURIN 23 43 N=C(N)Nc1ccc(CC(=O)Cl)cc1 ZINC000147192617 BD For-Sale Reactive SPHK1 15 40 N=C(N)Nc1ccc(CC(=O)Cl)cc1 ZINC000147192617 BD For-Sale Reactive ACR 57 45 N=C(N)Nc1ccc(CC(=O)Cl)cc1 ZINC000147192617 BD For-Sale Reactive AOC3 25 43 N=C(N)Nc1ccc(CC(=O)Cl)cc1 ZINC000147192617 BD For-Sale Reactive Q9GPQ4_TRYVI 0 43 CCc1ncc(C(=O)NCCc2ccc3c(c2)OCCO3)s1 ZINC000147192627 DE On-Demand Anodyne NOS2 50 40 CC(C)NS(=O)(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147192699 GC On-Demand Anodyne BDKRB1 15 50 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne FOLH1 19 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne MME 19 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne NPR1 41 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne CA1 49 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne KLK3 64 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne CTSK 40 45 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne NPFFR2 45 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne TIMP3 65 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne C3AR1 44 31 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne HDAC8 27 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne HDAC10 47 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne MMP2 23 52 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne MMP3 49 51 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne HLA-DRB1 33 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne SOAT1 27 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne HDAC1 22 45 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne HDAC2 32 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne HDAC3 31 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne HDAC6 33 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne PCSK5 41 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne FURIN 69 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne CCKBR 16 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne ACE2 41 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne HDAC11 62 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne POLG_WNV 69 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne MTCA1 25 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne P96878_MYCTU 36 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192740 GG On-Demand Anodyne NPFFR1 62 34 CO[C@@H](C)c1ccc([N+](=O)[O-])cc1 ZINC000147192766 AE For-Sale Bother KCNJ1 15 40 COCc1nc(C(=O)NCCc2ccc3c(c2)OCCO3)cs1 ZINC000147192836 EE On-Demand Anodyne NOS2 59 38 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCC1 ZINC000147192872 DG For-Sale Anodyne ADORA1 26 52 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCC1 ZINC000147192872 DG For-Sale Anodyne P2RY12 86 42 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCC1 ZINC000147192872 DG For-Sale Anodyne TSPO 19 40 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCC1 ZINC000147192872 DG For-Sale Anodyne SOAT1 20 47 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCC1 ZINC000147192872 DG For-Sale Anodyne NPY5R 18 43 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCC1 ZINC000147192872 DG For-Sale Anodyne ADORA3 39 52 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCC1 ZINC000147192872 DG For-Sale Anodyne DGAT1 29 47 C[C@@H](NC(=O)c1ccc(Br)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147192887 FE On-Demand Mild CCR1 28 41 C[C@@H](NC(=O)c1ccc(Br)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147192887 FE On-Demand Mild JAK3 41 36 Cc1nn(C(F)F)c(C)c1CC(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192931 HJ On-Demand Anodyne P2RX7 29 46 Cc1nn(C(F)F)c(C)c1CC(=O)Nc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147192931 HJ On-Demand Anodyne FPR2 46 35 CO[C@H](C)c1ccc([N+](=O)[O-])cc1 ZINC000147192975 AE For-Sale Bother KCNJ1 15 40 COCCOc1cc(Cl)c(C(=O)NCc2ccc(Br)cc2)c(Cl)c1 ZINC000147193178 IJ For-Sale Anodyne PDS 44 38 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne POLA1 40 35 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne P2RY6 56 35 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne HPRT1 60 37 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne P2RX5 0 40 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne POLB 49 50 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne PNP 26 49 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne P2RX4 43 40 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne P2RX1 60 40 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne P2RX6 0 40 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne P2RY4 74 46 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne P2RY1 152 41 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne P2RY2 79 46 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne EIF4E 0 48 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne RNASE1 44 34 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne RAC1 0 56 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne GPR17 51 37 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne Q3ZDS5_9HEPC 0 65 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne CNGA2 0 41 C[C@]12OC[C@](CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147193236 KA Annotated Anodyne ROCR 0 41 Cn1ncc2c(-c3cccc4[nH]ncc34)nc(N3CCOCC3)nc21 ZINC000147193268 ED For-Sale Anodyne PIK3CA 17 48 Cn1ncc2c(-c3cccc4[nH]ncc34)nc(N3CCOCC3)nc21 ZINC000147193268 ED For-Sale Anodyne MTOR 15 46 CN(Cc1cscn1)C(=O)NC[C@@H]1CN(Cc2ccccc2)CCO1 ZINC000147193271 FE On-Demand Anodyne DRD4 21 43 CN(Cc1cscn1)C(=O)NC[C@@H]1CN(Cc2ccccc2)CCO1 ZINC000147193271 FE On-Demand Anodyne CYP3A4 17 40 CN(Cc1cscn1)C(=O)NC[C@H]1CN(Cc2ccccc2)CCO1 ZINC000147193472 FE On-Demand Anodyne DRD4 21 43 CN(Cc1cscn1)C(=O)NC[C@H]1CN(Cc2ccccc2)CCO1 ZINC000147193472 FE On-Demand Anodyne CYP3A4 17 40 CCOC(=O)c1cnc(-c2ccccn2)nc1NC ZINC000147193482 CD For-Sale Anodyne ADORA1 19 42 CCOC(=O)c1cnc(-c2ccccn2)nc1NC ZINC000147193482 CD For-Sale Anodyne JUN 23 48 CCOC(=O)c1cnc(-c2ccccn2)nc1NC ZINC000147193482 CD For-Sale Anodyne METAP1 29 42 CCOC(=O)c1cnc(-c2ccccn2)nc1NC ZINC000147193482 CD For-Sale Anodyne ADORA3 22 42 CN1C(=O)Cn2c1nc1nc(N3CCC[C@@H](N)C3)n(Cc3cc(F)ccc3C(F)(F)F)c1c2=O ZINC000147193533 JD Annotated Anodyne DPP4 44 53 COc1ccc2c(c1)OC[C@@H](C(=O)N(Cc1ccccc1OC)C1CC1)C2 ZINC000147193565 FG On-Demand Anodyne MBTPS1 40 34 Cc1cc(C(=O)N(C)Cc2ccccc2Br)cc([N+](=O)[O-])c1 ZINC000147193675 FH On-Demand Bother COLA 80 35 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1N1C[C@H](C)O[C@H](C)C1)C2 ZINC000147193728 GG On-Demand Anodyne KCNQ2 67 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1N1C[C@H](C)O[C@H](C)C1)C2 ZINC000147193728 GG On-Demand Anodyne ROCK2 30 45 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)NC1CCCC1 ZINC000147193776 GE On-Demand Mild CPT1A 20 44 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)NC1CCCC1 ZINC000147193776 GE On-Demand Mild CCR8 83 39 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)NC1CCCC1 ZINC000147193776 GE On-Demand Mild SFRP1 110 38 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)NC1CCCC1 ZINC000147193776 GE On-Demand Mild WNT3 76 33 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)NC1CCCC1 ZINC000147193776 GE On-Demand Mild L3MBTL3 71 37 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc(C(C)C)cc3)CC2)s1 ZINC000147193851 HF On-Demand Anodyne TGM2 65 36 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc(C(C)C)cc3)CC2)s1 ZINC000147193851 HF On-Demand Anodyne F13A1 65 36 CCOC(=O)c1cnc(-c2ccc(Cl)cc2)nc1N1CCCCC1 ZINC000147193889 EH For-Sale Anodyne P2RY12 58 45 CCOC(=O)c1cnc(-c2ccc(Cl)cc2)nc1N1CCCCC1 ZINC000147193889 EH For-Sale Anodyne JUN 17 41 CCOC(=O)c1cnc(-c2ccc(Cl)cc2)nc1N1CCCCC1 ZINC000147193889 EH For-Sale Anodyne SCN2A 18 40 CCOC(=O)c1cnc(-c2ccc(Cl)cc2)nc1N1CCCCC1 ZINC000147193889 EH For-Sale Anodyne SCN10A 28 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1N1C[C@H](C)O[C@@H](C)C1)C2 ZINC000147193924 GG On-Demand Anodyne KCNQ2 67 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1N1C[C@H](C)O[C@@H](C)C1)C2 ZINC000147193924 GG On-Demand Anodyne ROCK2 30 45 N#CC1CCN(C(=O)Cn2c(C(F)(F)F)nc3ccccc32)CC1 ZINC000147193947 EF On-Demand Mild ETHR 54 37 CCOC(=O)c1cnc(-c2ccc(Br)cc2)nc1N1CCCCC1 ZINC000147194063 GI For-Sale Anodyne P2RY12 51 37 CCOC(=O)c1cnc(-c2ccc(Br)cc2)nc1N1CCCCC1 ZINC000147194063 GI For-Sale Anodyne JUN 18 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1N1C[C@@H](C)O[C@H](C)C1)C2 ZINC000147194115 GG On-Demand Anodyne KCNQ2 67 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1N1C[C@@H](C)O[C@H](C)C1)C2 ZINC000147194115 GG On-Demand Anodyne ROCK2 30 45 Cc1cc(C(=O)NCCc2ccc3c(c2)OCCO3)cc([N+](=O)[O-])c1 ZINC000147194256 EF On-Demand Bother PLK1 15 41 O=C(OCCl)c1ccc2ccccc2c1 ZINC000147194318 BG For-Sale Reactive TRYP_PIG 15 40 O=C(OCCl)c1ccc2ccccc2c1 ZINC000147194318 BG For-Sale Reactive PLAU 17 40 O=C(OCCl)c1ccc2ccccc2c1 ZINC000147194318 BG For-Sale Reactive POLG_HRV16 16 50 C[C@H]1CN(c2ccccc2NC(=O)c2ccc3c(c2)COC3)C[C@@H](C)O1 ZINC000147194330 FH On-Demand Anodyne KCNQ2 68 33 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild ACE 22 48 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild SSTR2 60 43 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild OPRM1 20 54 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild OPRD1 22 50 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild GHRHR 36 49 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild MME 25 43 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild EDNRB 54 44 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild EDNRA 81 47 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild TACR1 52 44 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild MC4R 66 43 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild TACR2 34 46 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild CCKAR 82 42 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild CTSL 25 41 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild BRS3 42 44 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild CYP51A1 24 40 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild UTS2R 15 44 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild MC3R 62 40 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild MC5R 58 39 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild MMP2 22 43 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild MMP8 57 40 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild MMP14 89 40 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild GRPR 74 38 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild ECE1 59 46 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild MMP11 68 40 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild CCKBR 68 46 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild GHSR 72 50 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild CCR2 51 34 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild MMP9 23 52 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild MC1R 71 43 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild ADAM9 39 40 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild CTSC 18 45 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild C5AR1 60 44 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild MMP1 20 41 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild NPR 31 43 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild KISS1R 60 33 CC(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194445 ED On-Demand Mild ERAP2 41 36 C[C@@H]1CN(c2ccccc2NC(=O)c2ccc3c(c2)COC3)C[C@@H](C)O1 ZINC000147194534 FH On-Demand Anodyne KCNQ2 68 33 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild ACE 22 48 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild SSTR2 60 43 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild OPRM1 17 42 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild GHRHR 36 49 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild MME 25 43 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild EDNRA 46 47 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild TACR1 29 52 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild MC4R 66 43 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild CCKAR 82 42 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild BRS3 24 44 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild CYP51A1 24 40 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild MC3R 62 40 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild MC5R 58 39 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild MMP2 22 43 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild MMP8 34 43 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild GRPR 74 38 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild ECE1 59 46 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild MMP11 68 40 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild CCKBR 68 46 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild GHSR 72 50 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild MMP9 23 52 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild MC1R 71 43 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild ADAM9 39 40 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild CTSC 18 45 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild C5AR1 46 44 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild MMP1 20 41 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild NPR 31 43 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild KISS1R 60 33 CC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC(C#N)CC1 ZINC000147194660 ED On-Demand Mild ERAP2 41 36 CC(=O)N1CCc2cc(S(=O)(=O)O)ccc21 ZINC000147194716 BC For-Sale Anodyne CYP11B2 15 52 CC(=O)N1CCc2cc(S(=O)(=O)O)ccc21 ZINC000147194716 BC For-Sale Anodyne HSD17B3 58 38 CC(=O)N1CCc2cc(S(=O)(=O)O)ccc21 ZINC000147194716 BC For-Sale Anodyne BETA-TUBULIN 0 41 CNC(=O)c1cc(NC(=O)c2cnn(-c3ccccc3Cl)c2)ccc1Cl ZINC000147194719 GH On-Demand Anodyne MAOB 17 41 CNC(=O)c1cc(NC(=O)c2cnn(-c3ccccc3Cl)c2)ccc1Cl ZINC000147194719 GH On-Demand Anodyne GRM4 55 36 CNC(=O)c1cc(NC(=O)c2cnn(-c3ccccc3Cl)c2)ccc1Cl ZINC000147194719 GH On-Demand Anodyne MAPK10 19 42 CNC(=O)c1cc(NC(=O)c2cnn(-c3ccccc3Cl)c2)ccc1Cl ZINC000147194719 GH On-Demand Anodyne CSF1R 20 44 CNC(=O)c1cc(NC(=O)c2cnn(-c3ccccc3Cl)c2)ccc1Cl ZINC000147194719 GH On-Demand Anodyne NR2E3 63 37 CNC(=O)c1cc(NC(=O)c2cnn(-c3ccccc3Cl)c2)ccc1Cl ZINC000147194719 GH On-Demand Anodyne SHH 42 39 CNC(=O)c1cc(NC(=O)c2cnn(-c3ccccc3Cl)c2)ccc1Cl ZINC000147194719 GH On-Demand Anodyne SMO 23 40 CNC(=O)c1cc(NC(=O)c2cnn(-c3ccccc3Cl)c2)ccc1Cl ZINC000147194719 GH On-Demand Anodyne IMDH_CRYPV 21 40 CNC(=O)c1cc(NC(=O)c2cnn(-c3ccccc3Cl)c2)ccc1Cl ZINC000147194719 GH On-Demand Anodyne KCNK3 61 40 CCCC(=O)Nc1nc2ccc(NC(=O)c3cc(OC)ccc3[N+](=O)[O-])cc2s1 ZINC000147194793 HI On-Demand Bother LDHA 40 39 CCCC(=O)Nc1nc2ccc(NC(=O)c3cc(OC)ccc3[N+](=O)[O-])cc2s1 ZINC000147194793 HI On-Demand Bother CSNK1D 49 52 CCCC(=O)Nc1nc2ccc(NC(=O)c3cc(OC)ccc3[N+](=O)[O-])cc2s1 ZINC000147194793 HI On-Demand Bother NMT1 20 41 CCCC(=O)Nc1nc2ccc(NC(=O)c3cc(OC)ccc3[N+](=O)[O-])cc2s1 ZINC000147194793 HI On-Demand Bother MTNR1B 15 40 CCCC(=O)Nc1nc2ccc(NC(=O)c3cc(OC)ccc3[N+](=O)[O-])cc2s1 ZINC000147194793 HI On-Demand Bother TAAR1 21 41 CNC(=O)c1cc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)ccc1Cl ZINC000147194911 FF On-Demand Anodyne Q8MMZ8_EIMTE 16 42 CC(C)Oc1cccc(OCC2CC2)c1 ZINC000147194979 BG On-Demand Anodyne PDE4D 24 43 CC(C)Oc1cccc(OCC2CC2)c1 ZINC000147194979 BG On-Demand Anodyne CHRNA10 74 39 CC(C)Oc1cccc(OCC2CC2)c1 ZINC000147194979 BG On-Demand Anodyne DUT 44 39 CCCCC[C@H](N)C(=O)NC ZINC000147195054 AC For-Sale Anodyne DPP7 51 63 CCCCC[C@H](N)C(=O)NC ZINC000147195054 AC For-Sale Anodyne DPP8 44 49 CCCCC[C@H](N)C(=O)NC ZINC000147195054 AC For-Sale Anodyne DPP9 37 49 O=C(CNC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)Nc1ccccc1 ZINC000147195126 EG On-Demand Anodyne CCKBR 19 41 O=C(CNC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)Nc1ccccc1 ZINC000147195126 EG On-Demand Anodyne MDM2 79 40 CC(C)COc1cccc(OC(C)C)c1 ZINC000147195177 BH On-Demand Anodyne ACACA 15 41 CC(C)COc1cccc(OC(C)C)c1 ZINC000147195177 BH On-Demand Anodyne PDS 64 34 CNc1ccccc1CC[C@@H]1CCCCN1C ZINC000147195179 BG For-Sale Anodyne SLC18A2 46 45 CNc1ccccc1CC[C@@H]1CCCCN1C ZINC000147195179 BG For-Sale Anodyne CHRNA10 50 41 CC#CCn1c(N2CCC[C@@H](N)C2)nc2nc3n(c(=O)c21)CC(=O)N3C ZINC000147195228 FB Annotated Mild DPP4 44 63 O=C(CNC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)Nc1ccccc1 ZINC000147195309 EG On-Demand Anodyne CCKBR 19 41 O=C(CNC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)Nc1ccccc1 ZINC000147195309 EG On-Demand Anodyne MDM2 79 40 COc1ccccc1OCCNC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147195327 EF On-Demand Bother ADRA1A 20 40 COc1ccccc1OCCNC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147195327 EF On-Demand Bother CACNA1D 51 36 CNc1ccccc1CC[C@H]1CCCCN1C ZINC000147195381 BG For-Sale Anodyne SLC18A2 46 45 CNc1ccccc1CC[C@H]1CCCCN1C ZINC000147195381 BG For-Sale Anodyne CHRNA10 50 41 O=C(CNC(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1)Nc1ccccc1 ZINC000147195485 EG On-Demand Anodyne CCKBR 19 41 O=C(CNC(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1)Nc1ccccc1 ZINC000147195485 EG On-Demand Anodyne MDM2 79 40 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild FABP2 0 48 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild FABP4 16 48 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild FAAH 24 53 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild CES2 47 42 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild CES1 36 42 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild EST1_PIG 63 42 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild CES2C 52 32 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild CPT1 68 33 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild JHE 0 57 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild FABP5 16 48 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild SLC22A20 0 48 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild Q9GPG0_MANSE 0 42 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild FPPS 57 34 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild NOD1 73 39 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild CQSS 94 63 CCCCCCCC(=O)[C@@H](C)C(C)=O ZINC000147195512 AG Annotated Mild EST5_RAT 48 29 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCN(CC)CC1 ZINC000147195591 FD On-Demand Anodyne KCNQ2 88 48 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCN(CC)CC1 ZINC000147195591 FD On-Demand Anodyne PCSK5 40 32 COCc1nc(C(=O)N2CCN(c3ccccc3[N+](=O)[O-])CC2)cs1 ZINC000147195630 FE On-Demand Bother TRPC6 55 35 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild FABP2 0 48 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild FABP4 16 48 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild FAAH 24 53 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild CES2 47 42 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild CES1 36 42 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild EST1_PIG 63 42 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild CES2C 52 32 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild CPT1 68 33 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild JHE 0 57 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild FABP5 16 48 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild SLC22A20 0 48 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild Q9GPG0_MANSE 0 42 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild FPPS 57 34 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild NOD1 73 39 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild CQSS 94 63 CCCCCCCC(=O)[C@H](C)C(C)=O ZINC000147195696 AG Annotated Mild EST5_RAT 48 29 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCN(CC)CC1 ZINC000147195788 FD On-Demand Anodyne KCNQ2 88 48 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCN(CC)CC1 ZINC000147195788 FD On-Demand Anodyne PCSK5 40 32 CCCN(Cc1ccccc1)C(=O)c1cnc(CC)s1 ZINC000147195820 CH On-Demand Anodyne TSPO 35 40 Cc1nc2cc(NC(=O)OC(C)(C)C)ccc2s1 ZINC000147195863 CH For-Sale Anodyne ACOX1 64 38 Cc1nc2cc(NC(=O)OC(C)(C)C)ccc2s1 ZINC000147195863 CH For-Sale Anodyne AGPAT2 40 49 Cc1nc2cc(NC(=O)OC(C)(C)C)ccc2s1 ZINC000147195863 CH For-Sale Anodyne LEF1 0 40 CNC(=O)NCc1ccc(Cl)cc1F ZINC000147195974 BD On-Demand Anodyne P2RX7 78 45 C[C@@H](O)N1CCc2ccccc21 ZINC000147196047 AD For-Sale Anodyne DRD1 24 44 C[C@@H](O)N1CCc2ccccc21 ZINC000147196047 AD For-Sale Anodyne DRD5 51 44 CCc1ncc(C(=O)Nc2nc(-c3ccc(F)cc3)c(C)s2)s1 ZINC000147196184 EJ On-Demand Anodyne MPL 18 40 CCc1ncc(C(=O)Nc2nc(-c3ccc(F)cc3)c(C)s2)s1 ZINC000147196184 EJ On-Demand Anodyne MAPK14 18 43 CN[C@@H]1CCN(Cc2ccc(OCC(=O)OC)cc2)C1 ZINC000147196226 CD On-Demand Anodyne DRD4 34 46 CN[C@@H]1CCN(Cc2ccc(OCC(=O)OC)cc2)C1 ZINC000147196226 CD On-Demand Anodyne LTA4H 46 45 CN[C@@H]1CCN(Cc2ccc(OCC(=O)OC)cc2)C1 ZINC000147196226 CD On-Demand Anodyne SIGMAR1 43 42 CN[C@@H]1CCN(Cc2ccc(OCC(=O)OC)cc2)C1 ZINC000147196226 CD On-Demand Anodyne SSTR5 53 36 CN[C@@H]1CCN(Cc2ccc(OCC(=O)OC)cc2)C1 ZINC000147196226 CD On-Demand Anodyne CCR3 33 43 CN[C@@H]1CCN(Cc2ccc(OCC(=O)OC)cc2)C1 ZINC000147196226 CD On-Demand Anodyne UTS2R 20 48 CN[C@@H]1CCN(Cc2ccc(OCC(=O)OC)cc2)C1 ZINC000147196226 CD On-Demand Anodyne MLNR 69 38 CN[C@@H]1CCN(Cc2ccc(OCC(=O)OC)cc2)C1 ZINC000147196226 CD On-Demand Anodyne SLC6A5 31 42 CN[C@@H]1CCN(Cc2ccc(OCC(=O)OC)cc2)C1 ZINC000147196226 CD On-Demand Anodyne MMP1 16 40 CN[C@@H]1CCN(Cc2ccc(OCC(=O)OC)cc2)C1 ZINC000147196226 CD On-Demand Anodyne MCHR1 45 45 C[C@H](O)N1CCc2ccccc21 ZINC000147196233 AD For-Sale Anodyne DRD1 24 44 C[C@H](O)N1CCc2ccccc21 ZINC000147196233 AD For-Sale Anodyne DRD5 51 44 N#Cc1cn(-c2ccc(C(=O)O)c(O)c2)c2ccc(OCc3ccccc3)cc12 ZINC000147196294 GI Annotated Anodyne MAOB 24 45 N#Cc1cn(-c2ccc(C(=O)O)c(O)c2)c2ccc(OCc3ccccc3)cc12 ZINC000147196294 GI Annotated Anodyne EDNRA 21 41 N#Cc1cn(-c2ccc(C(=O)O)c(O)c2)c2ccc(OCc3ccccc3)cc12 ZINC000147196294 GI Annotated Anodyne PLA2G2A 22 41 N#Cc1cn(-c2ccc(C(=O)O)c(O)c2)c2ccc(OCc3ccccc3)cc12 ZINC000147196294 GI Annotated Anodyne PFKFB3 46 41 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)Nc1ccccc1)C2 ZINC000147196295 EE On-Demand Anodyne MTNR1A 70 44 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)Nc1ccccc1)C2 ZINC000147196295 EE On-Demand Anodyne MTNR1B 62 39 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)Nc1ccccc1)C2 ZINC000147196295 EE On-Demand Anodyne ROCK2 32 47 CN1CCN(CC(=O)Nc2cccnc2)CC1 ZINC000147196375 BC In-Stock Anodyne CHRNA7 39 47 CN1CCN(CC(=O)Nc2cccnc2)CC1 ZINC000147196375 BC In-Stock Anodyne PRNP 27 42 CN1CCN(CC(=O)Nc2cccnc2)CC1 ZINC000147196375 BC In-Stock Anodyne NAMPT 41 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCC(=O)Nc1ccccc1)C2 ZINC000147196460 EE On-Demand Anodyne MTNR1A 70 44 COc1ccc2c(c1)OC[C@@H](C(=O)NCC(=O)Nc1ccccc1)C2 ZINC000147196460 EE On-Demand Anodyne MTNR1B 62 39 COc1ccc2c(c1)OC[C@@H](C(=O)NCC(=O)Nc1ccccc1)C2 ZINC000147196460 EE On-Demand Anodyne ROCK2 32 47 NC(=O)c1ccc(OCC(=O)N2CCCc3cc(Cl)ccc32)cc1 ZINC000147196598 EF On-Demand Anodyne CNR1 41 32 NC(=O)c1ccc(OCC(=O)N2CCCc3cc(Cl)ccc32)cc1 ZINC000147196598 EF On-Demand Anodyne AVPR2 21 48 NC(=O)c1ccc(OCC(=O)N2CCCc3cc(Cl)ccc32)cc1 ZINC000147196598 EF On-Demand Anodyne EIF2AK3 42 34 CCC(C)(C)NC(=O)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147196652 GH On-Demand Anodyne ROCK2 26 50 Nc1c(C(=O)c2ccc(Cl)c(Cl)c2)sc2nc3c(cc12)CCCCCC3 ZINC000147196864 HK In-Stock Anodyne EEF2K 72 50 C[C@H]1CCCCN1C(=O)c1ccc(NC(=O)c2ccc3c(c2)COC3)cc1Cl ZINC000147196890 GJ On-Demand Anodyne AVPR2 61 37 C[C@H]1CCCCN1C(=O)c1ccc(NC(=O)c2ccc3c(c2)COC3)cc1Cl ZINC000147196890 GJ On-Demand Anodyne CPT1A 25 41 Nc1cn2ccnc2c(Oc2cccc(F)c2)n1 ZINC000147196909 BE For-Sale Anodyne HIVRT 0 40 COc1ccccc1CN(C)C(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147197063 DG On-Demand Bother CACNA1D 47 33 Cc1ccc(C(=O)NNC(=O)NCC2(N(C)C)CCCC2)s1 ZINC000147197112 DD On-Demand Reactive SLC6A5 15 43 CCNc1cn2ccnc2c(Oc2cccc(F)c2)n1 ZINC000147197140 CG For-Sale Anodyne HIVRT 0 43 COc1nc(N)nc(Oc2cccc3ccccc23)n1 ZINC000147197326 CE For-Sale Anodyne ALS 40 36 O=C(CCc1ccccc1)OCCl ZINC000147197626 AE For-Sale Reactive NA 15 40 O=C(CCc1ccccc1)OCCl ZINC000147197626 AE For-Sale Reactive FAAH 50 35 O=C(CCc1ccccc1)OCCl ZINC000147197626 AE For-Sale Reactive CES1 60 38 O=C(CCc1ccccc1)OCCl ZINC000147197626 AE For-Sale Reactive HCAR2 21 43 O=C(CCc1ccccc1)OCCl ZINC000147197626 AE For-Sale Reactive FFAR1 62 45 O=C(CCc1ccccc1)OCCl ZINC000147197626 AE For-Sale Reactive FFAR4 44 38 NC(=O)c1ccc(OCC(=O)N2CCCc3cc(F)c(F)cc32)cc1 ZINC000147197802 EE On-Demand Anodyne PLA2G4B 40 32 CN1CCN(Nc2ccc(C(F)(F)F)cc2)CC1 ZINC000147197811 CE For-Sale Anodyne EPHX2 19 50 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1N1CCCC1 ZINC000147198064 ED On-Demand Anodyne KCNQ2 93 48 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1N1CCCC1 ZINC000147198064 ED On-Demand Anodyne CSF1R 20 45 CN(CCCCc1ccccc1)C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147198210 GG On-Demand Bother LIMK2 41 38 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccccc1N1CCCC1 ZINC000147198250 ED On-Demand Anodyne KCNQ2 93 48 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccccc1N1CCCC1 ZINC000147198250 ED On-Demand Anodyne CSF1R 20 45 CC(C)(C)Oc1cc(-c2ccc(CNC(=O)c3c(Cl)cccc3Cl)cc2)ccn1 ZINC000147198339 IK For-Sale Anodyne TYK2 52 38 CC(C)(C)Oc1cc(-c2ccc(CNC(=O)c3c(Cl)cccc3Cl)cc2)ccn1 ZINC000147198339 IK For-Sale Anodyne SUCNR1 41 37 NC(=O)c1ccc(OCC(=O)N2CCCc3cc(F)ccc32)cc1 ZINC000147198428 EE On-Demand Anodyne EIF2AK3 60 39 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne F2 15 41 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne ACE 47 35 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne OPRM1 46 46 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne OPRD1 41 46 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne OPRK1 0 45 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne MME 68 42 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne ANPEP 50 33 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne TRY2_BOVIN 51 33 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne SLC15A1 0 46 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne AKT3 24 45 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne TPH1 45 31 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne DPP4 23 53 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne DNPEP 0 42 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne DPP7 88 48 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne LAP3 56 39 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne AKT1 27 53 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne AMP1_PLAFQ 38 43 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne DPP8 51 49 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne DPP9 27 49 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne FAP 0 44 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne SLC15A2 0 44 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne AKT1S1 0 45 N[C@H](Cc1ccccc1)C(=O)N1CCC(=O)CC1 ZINC000147198454 BC For-Sale Anodyne BLAIMP-1 0 41 CC(C)Oc1ccc(CC[C@@H](C)NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147198501 FI On-Demand Anodyne ACACB 20 44 O=C(NCC1CCOCC1)c1cccc2ccccc12 ZINC000147198592 CF On-Demand Anodyne CNR1 31 71 O=C(NCC1CCOCC1)c1cccc2ccccc12 ZINC000147198592 CF On-Demand Anodyne CNR2 23 56 O=C(NCC1CCOCC1)c1cccc2ccccc12 ZINC000147198592 CF On-Demand Anodyne ACACB 26 42 O=C(NCC1CCOCC1)c1cccc2ccccc12 ZINC000147198592 CF On-Demand Anodyne FAP 0 48 COc1cc([C@@H](C)NC(=O)c2ccc3c(c2)COC3)ccc1OCc1ccccc1 ZINC000147198709 HJ On-Demand Anodyne AGTR2 46 38 COc1cc([C@@H](C)NC(=O)c2ccc3c(c2)COC3)ccc1OCc1ccccc1 ZINC000147198709 HJ On-Demand Anodyne CTSB 17 40 COc1cc([C@@H](C)NC(=O)c2ccc3c(c2)COC3)ccc1OCc1ccccc1 ZINC000147198709 HJ On-Demand Anodyne MTNR1B 20 42 COc1cc([C@@H](C)NC(=O)c2ccc3c(c2)COC3)ccc1OCc1ccccc1 ZINC000147198709 HJ On-Demand Anodyne CAPN1 30 40 COc1cc([C@@H](C)NC(=O)c2ccc3c(c2)COC3)ccc1OCc1ccccc1 ZINC000147198709 HJ On-Demand Anodyne CAPN2 35 40 COc1cc([C@@H](C)NC(=O)c2ccc3c(c2)COC3)ccc1OCc1ccccc1 ZINC000147198709 HJ On-Demand Anodyne F7 17 46 N#CC1CCN(C(=O)COc2ccc(I)cc2)CC1 ZINC000147198810 FE On-Demand Mild HTR1B 17 41 N#CC1CCN(C(=O)COc2ccc(I)cc2)CC1 ZINC000147198810 FE On-Demand Mild COLA 45 40 N#CC1CCN(C(=O)COc2ccc(I)cc2)CC1 ZINC000147198810 FE On-Demand Mild CPT1A 41 40 N#CC1CCN(C(=O)COc2ccc(I)cc2)CC1 ZINC000147198810 FE On-Demand Mild TRAR 21 40 NC(=O)c1ccc(OCC(=O)N2CCCc3c(C(N)=O)cccc32)cc1 ZINC000147198849 FD On-Demand Anodyne COLA 44 43 NC(=O)c1ccc(OCC(=O)N2CCCc3c(C(N)=O)cccc32)cc1 ZINC000147198849 FD On-Demand Anodyne PLA2G4B 46 34 CNC(=O)c1cc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)ccc1Cl ZINC000147198931 FI On-Demand Anodyne IMDH_CRYPV 16 41 CCOc1cc(C(=O)N2CCC(C#N)CC2)ccc1OCCOc1ccccc1 ZINC000147199001 GH On-Demand Mild AVPR1A 22 41 CCOc1cc(C(=O)N2CCC(C#N)CC2)ccc1OCCOc1ccccc1 ZINC000147199001 GH On-Demand Mild HRH3 26 41 CCOc1cc(C(=O)N2CCC(C#N)CC2)ccc1OCCOc1ccccc1 ZINC000147199001 GH On-Demand Mild L3MBTL3 53 42 CCc1ncc(C(=O)N(C)Cc2ccccc2C)s1 ZINC000147199090 CG On-Demand Anodyne HSP90AB1 15 41 CNC(=O)c1cc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)ccc1Cl ZINC000147199130 FI On-Demand Anodyne IMDH_CRYPV 16 41 CNC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147199207 DC On-Demand Anodyne TNK2 23 41 N#CC1CCN(C(=O)C[C@H](NC(N)=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000147199279 GG On-Demand Mild PTAFR 29 40 N#CC1CCN(C(=O)C[C@H](NC(N)=O)c2cccc(Oc3ccccc3)c2)CC1 ZINC000147199279 GG On-Demand Mild LGMN 44 35 CNC(=O)c1cc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)ccc1Cl ZINC000147199314 FI On-Demand Anodyne IMDH_CRYPV 16 41 COc1ccc(CNC[C@@H](O)c2cccc(F)c2)cc1OCCCC#N ZINC000147199391 FG On-Demand Mild PHES 0 43 CNC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147199405 DC On-Demand Anodyne TNK2 23 41 CS(=O)(=O)c1cc(C(=O)Nc2ccc3nccnc3c2)cc([N+](=O)[O-])c1 ZINC000147199459 FE On-Demand Bother SHH 15 45 CNC(=O)c1cc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)ccc1Cl ZINC000147199521 HI On-Demand Anodyne TYK2 40 38 NC(=O)c1cccc2c1CCCN2C(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147199660 GF On-Demand Anodyne AVPR2 57 38 NC(=O)c1cccc2c1CCCN2C(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147199660 GF On-Demand Anodyne FABP4 54 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc3nccnc3c2)c1 ZINC000147199682 DF On-Demand Bother KDR 44 39 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc3nccnc3c2)c1 ZINC000147199682 DF On-Demand Bother PDGFRA 45 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc3nccnc3c2)c1 ZINC000147199682 DF On-Demand Bother TAAR1 27 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc3nccnc3c2)c1 ZINC000147199682 DF On-Demand Bother AKR1C3 20 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc3nccnc3c2)c1 ZINC000147199682 DF On-Demand Bother AKR1C2 51 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc3nccnc3c2)c1 ZINC000147199682 DF On-Demand Bother USP7 27 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc3nccnc3c2)c1 ZINC000147199682 DF On-Demand Bother USP47 34 40 CNC(=O)c1cc(NC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)ccc1Cl ZINC000147199717 HI On-Demand Anodyne TYK2 40 38 CNc1nc(OC)nc(Oc2cccc3ccccc23)n1 ZINC000147199806 CF For-Sale Anodyne ALS 42 35 CNC(=O)c1cc(NC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)ccc1Cl ZINC000147199880 HI On-Demand Anodyne TYK2 40 38 O=C(Nc1ccc2nccnc2c1)c1ccn(-c2cccc(F)c2)n1 ZINC000147199907 EG On-Demand Anodyne GRM4 41 36 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147199968 FG On-Demand Anodyne MPL 40 33 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147199968 FG On-Demand Anodyne ROCK1 19 43 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147199968 FG On-Demand Anodyne ROCK2 15 43 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147199968 FG On-Demand Anodyne HDAC9 17 46 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147199968 FG On-Demand Anodyne TRPA1 15 43 CN1C(=O)C(c2ccccc2)=C(N2CCN(c3ccccc3)CC2)C1=O ZINC000147199987 EE For-Sale Anodyne HTR1A 21 47 CN1C(=O)C(c2ccccc2)=C(N2CCN(c3ccccc3)CC2)C1=O ZINC000147199987 EE For-Sale Anodyne PRNP 22 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCC1 ZINC000147199992 GF On-Demand Anodyne MC4R 15 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCC1 ZINC000147199992 GF On-Demand Anodyne KCNQ2 46 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCC1 ZINC000147199992 GF On-Demand Anodyne TEK 21 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCC1 ZINC000147199992 GF On-Demand Anodyne LIPG 50 36 O=C1NCCn2c1cccc2=O ZINC000147200010 AB For-Sale Anodyne PARP1 19 44 CNC(=O)c1cc(NC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)ccc1Cl ZINC000147200030 HI On-Demand Anodyne TYK2 40 38 CCOC[C@H]1[C@@H](c2ccc(Cl)c(Cl)c2)C[C@@H]2CC[C@H]1N2C ZINC000147200049 EJ Annotated Anodyne SLC6A2 35 41 CCOC[C@H]1[C@@H](c2ccc(Cl)c(Cl)c2)C[C@@H]2CC[C@H]1N2C ZINC000147200049 EJ Annotated Anodyne SLC6A4 56 70 CCOC[C@H]1[C@@H](c2ccc(Cl)c(Cl)c2)C[C@@H]2CC[C@H]1N2C ZINC000147200049 EJ Annotated Anodyne SLC6A3 125 70 CCOC[C@H]1[C@@H](c2ccc(Cl)c(Cl)c2)C[C@@H]2CC[C@H]1N2C ZINC000147200049 EJ Annotated Anodyne CHRNA9 0 48 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200120 FG On-Demand Anodyne MPL 40 33 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200120 FG On-Demand Anodyne ROCK1 19 43 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200120 FG On-Demand Anodyne ROCK2 15 43 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200120 FG On-Demand Anodyne HDAC9 17 46 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200120 FG On-Demand Anodyne TRPA1 15 43 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCC1 ZINC000147200136 GF On-Demand Anodyne MC4R 15 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCC1 ZINC000147200136 GF On-Demand Anodyne KCNQ2 46 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCC1 ZINC000147200136 GF On-Demand Anodyne TEK 21 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCC1 ZINC000147200136 GF On-Demand Anodyne LIPG 50 36 CCN1C(=O)Cn2c1nc1nc(N3CCC[C@@H](N)C3)n(Cc3cc(F)ccc3C#N)c1c2=O ZINC000147200178 JC Annotated Mild DPP4 50 63 CCCCCC[C@@H](CCCCCCCCCCC(=O)OC)OS(C)(=O)=O ZINC000147200227 GK For-Sale Mild NOD1 51 34 CCCCCC[C@@H](CCCCCCCCCCC(=O)OC)OS(C)(=O)=O ZINC000147200227 GK For-Sale Mild CQSS 58 37 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200257 FG On-Demand Anodyne MPL 40 33 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200257 FG On-Demand Anodyne ROCK1 19 43 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200257 FG On-Demand Anodyne ROCK2 15 43 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200257 FG On-Demand Anodyne HDAC9 17 46 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200257 FG On-Demand Anodyne TRPA1 15 43 CCOC[C@H]1[C@@H](c2ccc(Cl)c(Cl)c2)C[C@@H]2CC[C@@H]1N2C ZINC000147200362 EJ Annotated Anodyne SLC6A2 35 41 CCOC[C@H]1[C@@H](c2ccc(Cl)c(Cl)c2)C[C@@H]2CC[C@@H]1N2C ZINC000147200362 EJ Annotated Anodyne SLC6A4 56 70 CCOC[C@H]1[C@@H](c2ccc(Cl)c(Cl)c2)C[C@@H]2CC[C@@H]1N2C ZINC000147200362 EJ Annotated Anodyne SLC6A3 125 70 CCOC[C@H]1[C@@H](c2ccc(Cl)c(Cl)c2)C[C@@H]2CC[C@@H]1N2C ZINC000147200362 EJ Annotated Anodyne CHRNA9 0 48 CCCCCC[C@H](CCCCCCCCCCC(=O)OC)OS(C)(=O)=O ZINC000147200389 GK For-Sale Mild NOD1 51 34 CCCCCC[C@H](CCCCCCCCCCC(=O)OC)OS(C)(=O)=O ZINC000147200389 GK For-Sale Mild CQSS 58 37 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200394 FG On-Demand Anodyne MPL 40 33 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200394 FG On-Demand Anodyne ROCK1 19 43 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200394 FG On-Demand Anodyne ROCK2 15 43 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200394 FG On-Demand Anodyne HDAC9 17 46 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1nc(-c2cccc(F)c2)cs1 ZINC000147200394 FG On-Demand Anodyne TRPA1 15 43 CC(=O)Nc1ccc2cccc(S(=O)(=O)CCO)c2c1 ZINC000147200448 CD For-Sale Anodyne NQO2 25 45 CC(=O)Nc1ccc2cccc(S(=O)(=O)CCO)c2c1 ZINC000147200448 CD For-Sale Anodyne MTNR1A 26 45 CC(=O)Nc1ccc2cccc(S(=O)(=O)CCO)c2c1 ZINC000147200448 CD For-Sale Anodyne MTNR1B 17 45 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne SRD5A2 0 46 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne RARG 23 40 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne ECR 16 40 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne NR1H4 23 48 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne HDAC1 28 58 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne HDAC2 24 58 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne HDAC3 0 40 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne NEU3 0 42 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne KCNMA1 20 44 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne FABH 0 42 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne AKR1C3 28 43 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne GPR35 55 46 Cc1ccc(C(=O)Nc2cc(C(=O)O)ccc2O)cc1 ZINC000147200449 CF For-Sale Anodyne KCNK3 73 39 Cc1ccc(C)c(S(=O)(=O)NCCC(=O)N2CCC(C#N)CC2)c1 ZINC000147200578 ED On-Demand Mild CCR8 46 36 c1cnc(N2CCN(Cc3ccc(-c4cccs4)cc3)CC2)nc1 ZINC000147200707 EH On-Demand Anodyne DRD2 15 55 c1cnc(N2CCN(Cc3ccc(-c4cccs4)cc3)CC2)nc1 ZINC000147200707 EH On-Demand Anodyne DRD4 38 55 c1cnc(N2CCN(Cc3ccc(-c4cccs4)cc3)CC2)nc1 ZINC000147200707 EH On-Demand Anodyne DRD3 15 55 NC(=O)c1cccc2c1CCCN2C(=O)c1csc(-c2ccccc2F)n1 ZINC000147200797 GH On-Demand Anodyne AVPR2 45 35 CN1C(=O)Cn2c1nc1nc(N3CCC[C@@H](N)C3)n(Cc3cc(F)ccc3F)c1c2=O ZINC000147200803 IC Annotated Anodyne DPP4 50 53 COc1ccc(N2CCOCC2)c2sc(NC(=O)c3ccc(CN4CCC4)cc3)nc12 ZINC000147200940 IH For-Sale Clean DRD2 16 40 COc1ccc(N2CCOCC2)c2sc(NC(=O)c3ccc(CN4CCC4)cc3)nc12 ZINC000147200940 IH For-Sale Clean DRD3 21 40 COc1ccc(N2CCOCC2)c2sc(NC(=O)c3ccc(CN4CCC4)cc3)nc12 ZINC000147200940 IH For-Sale Clean ADORA2B 20 54 COc1ccc(N2CCOCC2)c2sc(NC(=O)c3ccc(CN4CCC4)cc3)nc12 ZINC000147200940 IH For-Sale Clean CASR 19 42 COc1ccc(N2CCOCC2)c2sc(NC(=O)c3ccc(CN4CCC4)cc3)nc12 ZINC000147200940 IH For-Sale Clean CPT1B 43 34 COc1ccc(N2CCOCC2)c2sc(NC(=O)c3ccc(CN4CCC4)cc3)nc12 ZINC000147200940 IH For-Sale Clean NOD2 40 37 Cc1ccc(C(=O)NNC(=O)NCc2ccc3c(c2)OCCO3)s1 ZINC000147201083 ED On-Demand Reactive NOS2 65 34 CN(Cc1cscn1)C(=O)NCc1ccc2c(c1)OCCO2 ZINC000147201270 DE On-Demand Anodyne NOS2 57 33 N#Cc1ccc(O)c(NC(=O)c2ccccc2C(F)(F)F)c1 ZINC000147201294 DH On-Demand Mild KCNMA1 31 46 CN(C)c1nc(-c2ccccc2)ncc1C(=O)OC[C@@H]1CCCCO1 ZINC000147201334 EF For-Sale Anodyne OXTR 24 41 CN(C)c1nc(-c2ccccc2)ncc1C(=O)OC[C@@H]1CCCCO1 ZINC000147201334 EF For-Sale Anodyne AVPR1A 15 41 CN(C)c1nc(-c2ccccc2)ncc1C(=O)OC[C@H]1CCCCO1 ZINC000147201437 EF For-Sale Anodyne OXTR 24 41 CN(C)c1nc(-c2ccccc2)ncc1C(=O)OC[C@H]1CCCCO1 ZINC000147201437 EF For-Sale Anodyne AVPR1A 15 41 COc1ccc([C@H](CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)N2CCCC2)cc1 ZINC000147201609 GG On-Demand Bother DRD4 40 32 COc1ccc([C@H](CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)N2CCCC2)cc1 ZINC000147201609 GG On-Demand Bother CYP24A1 23 41 COc1ccc([C@H](CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)N2CCCC2)cc1 ZINC000147201609 GG On-Demand Bother CYP27B1 27 41 COc1ccc([C@@H](CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)N2CCCC2)cc1 ZINC000147201696 GG On-Demand Bother DRD4 40 32 COc1ccc([C@@H](CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)N2CCCC2)cc1 ZINC000147201696 GG On-Demand Bother CYP24A1 23 41 COc1ccc([C@@H](CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)N2CCCC2)cc1 ZINC000147201696 GG On-Demand Bother CYP27B1 27 41 CC(C)(C)C[C@H]1N[C@@H](C(=O)NCC(C)(C)O)[C@H](c2cccc(Cl)c2F)[C@@]12C(=O)Nc1cc(Cl)ccc12 ZINC000147201699 KJ Annotated Anodyne MDM2 67 59 CSCC[C@H](NC(=O)c1cccc([N+](=O)[O-])c1)C(=O)N1CCC(C#N)CC1 ZINC000147201841 GE On-Demand Mild P2RY12 128 35 CSCC[C@@H](NC(=O)c1cccc([N+](=O)[O-])c1)C(=O)N1CCC(C#N)CC1 ZINC000147201994 GE On-Demand Mild P2RY12 128 35 Cc1cc2cccnc2cn1 ZINC000147202097 AD In-Stock Anodyne CCR1 0 47 Nc1nccc(Oc2cccc3ccccc23)n1 ZINC000147202101 BG For-Sale Anodyne DFR1 17 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(CN2CCCCC2)c1 ZINC000147202107 FE On-Demand Anodyne HRH2 52 44 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(CN2CCCCC2)c1 ZINC000147202107 FE On-Demand Anodyne SIGMAR1 17 40 N#Cc1ccc(O)c(NC(=O)c2c(Cl)cccc2Cl)c1 ZINC000147202121 DH On-Demand Mild KCNMA1 25 43 N#Cc1ccc(O)c(NC(=O)c2c(Cl)cccc2Cl)c1 ZINC000147202121 DH On-Demand Mild TYK2 27 40 COCCOc1cc(C)ccc1NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147202143 FG On-Demand Anodyne ROCK2 45 55 COc1ccccc1C(=O)N[C@@H](CCSC)C(=O)N1CCC(C#N)CC1 ZINC000147202198 GE On-Demand Mild P2RY12 175 38 COc1ccccc1C(=O)N[C@@H](CCSC)C(=O)N1CCC(C#N)CC1 ZINC000147202198 GE On-Demand Mild CCR1 20 41 COc1ccccc1C(=O)N[C@@H](CCSC)C(=O)N1CCC(C#N)CC1 ZINC000147202198 GE On-Demand Mild KCNA3 40 36 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(CN2CCCCC2)c1 ZINC000147202247 FE On-Demand Anodyne HRH2 52 44 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(CN2CCCCC2)c1 ZINC000147202247 FE On-Demand Anodyne SIGMAR1 17 40 CCc1ncc(C(=O)N(C)Cc2ccc(Cl)cc2)s1 ZINC000147202283 CH On-Demand Anodyne KLKB1 21 41 CCc1ncc(C(=O)N(C)Cc2ccc(Cl)cc2)s1 ZINC000147202283 CH On-Demand Anodyne TSPO 15 44 COc1ccccc1C(=O)N[C@H](CCSC)C(=O)N1CCC(C#N)CC1 ZINC000147202326 GE On-Demand Mild P2RY12 175 38 COc1ccccc1C(=O)N[C@H](CCSC)C(=O)N1CCC(C#N)CC1 ZINC000147202326 GE On-Demand Mild CCR1 20 41 COc1ccccc1C(=O)N[C@H](CCSC)C(=O)N1CCC(C#N)CC1 ZINC000147202326 GE On-Demand Mild KCNA3 40 36 COc1ccc(CNC[C@H]2CCN(c3ccc(Cl)cc3)C2)cc1OCCCC#N ZINC000147202602 HJ On-Demand Mild PDE5A 19 40 CCCCCS(=O)(=O)NCC(=O)NCC(=O)O ZINC000147202612 CB On-Demand Anodyne CPT1A 27 41 CSCC[C@@H](NC(=O)c1cccc(C)c1)C(=O)N1CCC(C#N)CC1 ZINC000147202653 FF On-Demand Mild P2RY12 123 37 CSCC[C@@H](NC(=O)c1cccc(C)c1)C(=O)N1CCC(C#N)CC1 ZINC000147202653 FF On-Demand Mild CCKAR 31 47 CSCC[C@@H](NC(=O)c1cccc(C)c1)C(=O)N1CCC(C#N)CC1 ZINC000147202653 FF On-Demand Mild CCKBR 94 47 CSCC[C@@H](NC(=O)c1cccc(C)c1)C(=O)N1CCC(C#N)CC1 ZINC000147202653 FF On-Demand Mild CTSV 21 41 CSCC[C@@H](NC(=O)c1cccc(C)c1)C(=O)N1CCC(C#N)CC1 ZINC000147202653 FF On-Demand Mild ST14 41 32 CCCOCC(=O)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000147202950 DE On-Demand Anodyne MLNR 46 42 CCCOCC(=O)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000147202950 DE On-Demand Anodyne CACNA1G 41 42 CCNc1nc(Cl)nc(Oc2cccc3ccccc23)n1 ZINC000147203027 DH For-Sale Anodyne Q31945_CHEAL 0 40 CCNc1nc(Cl)nc(Oc2cccc3ccccc23)n1 ZINC000147203027 DH For-Sale Anodyne PPX1 0 47 COCCOc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1OC ZINC000147203125 FD On-Demand Anodyne QRFPR 40 34 COCCOc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1OC ZINC000147203125 FD On-Demand Anodyne ENPP1 49 30 CCCCO[C@@H](C)C(=O)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000147203188 EG On-Demand Anodyne HRH3 29 42 CCCCO[C@@H](C)C(=O)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000147203188 EG On-Demand Anodyne MLNR 36 41 CCCCO[C@@H](C)C(=O)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000147203188 EG On-Demand Anodyne CACNA1G 39 41 O=C(Cn1cnnn1)Nc1cnn(C[C@@H]2CCCO2)c1 ZINC000147203214 CB On-Demand Anodyne PANC 44 31 CSCC[C@@H](NS(=O)(=O)c1ccccc1F)C(=O)N1CCC(C#N)CC1 ZINC000147203266 GD On-Demand Mild F2 42 42 CSCC[C@@H](NS(=O)(=O)c1ccccc1F)C(=O)N1CCC(C#N)CC1 ZINC000147203266 GD On-Demand Mild TRY2_BOVIN 48 34 CSCC[C@@H](NS(=O)(=O)c1ccccc1F)C(=O)N1CCC(C#N)CC1 ZINC000147203266 GD On-Demand Mild ST14 81 37 CSCC[C@@H](NS(=O)(=O)c1ccccc1F)C(=O)N1CCC(C#N)CC1 ZINC000147203266 GD On-Demand Mild TMPRSS6 41 31 COCCOc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1OC ZINC000147203275 FD On-Demand Anodyne QRFPR 40 34 COCCOc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1OC ZINC000147203275 FD On-Demand Anodyne ENPP1 49 30 CCCCO[C@H](C)C(=O)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000147203298 EG On-Demand Anodyne HRH3 29 42 CCCCO[C@H](C)C(=O)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000147203298 EG On-Demand Anodyne MLNR 36 41 CCCCO[C@H](C)C(=O)N1CCCN(Cc2ccc(F)cc2)CC1 ZINC000147203298 EG On-Demand Anodyne CACNA1G 39 41 O=C(Cn1cnnn1)Nc1cnn(C[C@H]2CCCO2)c1 ZINC000147203335 CB On-Demand Anodyne PANC 44 31 COc1cccc(COC(=O)c2cnc(-c3ccccc3)nc2N(C)C)c1 ZINC000147203346 FH For-Sale Anodyne PRKCZ 15 41 COc1cccc(COC(=O)c2cnc(-c3ccccc3)nc2N(C)C)c1 ZINC000147203346 FH For-Sale Anodyne HSD17B2 21 41 COC(=O)/C=C(/c1ccc(Cl)cc1)C(F)(F)F ZINC000147203352 CG On-Demand Anodyne KMO 0 40 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne ADORA1 18 67 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne DHODH 37 44 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne TSPO 36 47 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne TACR3 61 52 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne ADORA3 25 51 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne ALS 44 33 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne LUCI_LUCLA 32 49 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne ABCG2 47 55 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne LUCI_PHOPY 23 41 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne LUCI_PHOPE 28 41 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne MT-CO2 50 41 COc1ccc(-c2nc(C(=O)O)c3ccccc3n2)cc1 ZINC000147203371 CG For-Sale Anodyne RPA1 17 40 Cc1ccccc1C(=O)N[C@H](C(=O)N1CCC(C#N)CC1)C(C)C ZINC000147203507 EF On-Demand Mild CCR1 59 67 Cc1ccccc1C(=O)N[C@H](C(=O)N1CCC(C#N)CC1)C(C)C ZINC000147203507 EF On-Demand Mild CCR8 58 36 C#Cc1cccc(NC(=O)CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147203736 FD On-Demand Mild MTNR1A 42 41 C#Cc1cccc(NC(=O)CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147203736 FD On-Demand Mild ROCK2 27 43 CCOC(=O)c1cnc(-c2ccccc2Cl)nc1N1CCCCC1 ZINC000147203763 EH For-Sale Anodyne P2RY12 67 45 CCOC(=O)c1cnc(-c2ccccc2Cl)nc1N1CCCCC1 ZINC000147203763 EH For-Sale Anodyne PDE2A 37 45 CC(C)[C@H](NS(=O)(=O)c1ccccc1F)C(=O)N1CCC(C#N)CC1 ZINC000147203878 FD On-Demand Mild CCR1 44 43 CC(C)[C@H](NS(=O)(=O)c1ccccc1F)C(=O)N1CCC(C#N)CC1 ZINC000147203878 FD On-Demand Mild LEF 18 42 C#Cc1cccc(NC(=O)CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147203890 FD On-Demand Mild MTNR1A 42 41 C#Cc1cccc(NC(=O)CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147203890 FD On-Demand Mild ROCK2 27 43 CCOc1c(Cl)cc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1OC ZINC000147204118 HH On-Demand Anodyne ROCK2 21 40 CCOc1c(Cl)cc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1OC ZINC000147204118 HH On-Demand Anodyne PDE6A 40 31 COc1cc(OCC(=O)N[C@@H](CC(C)C)c2nc3ccccc3[nH]2)ccc1[N+](=O)[O-] ZINC000147204127 HH On-Demand Bother MMP7 22 49 CCOC(=O)c1cnc(-c2cccs2)nc1N(C)C ZINC000147204151 CE For-Sale Anodyne JUN 24 59 CCC[C@H](C(=O)N1CCC(C#N)CC1)c1ccccc1 ZINC000147204192 CG On-Demand Mild P2RY12 63 33 CCC[C@H](C(=O)N1CCC(C#N)CC1)c1ccccc1 ZINC000147204192 CG On-Demand Mild GRIN2B 20 42 CCC[C@H](C(=O)N1CCC(C#N)CC1)c1ccccc1 ZINC000147204192 CG On-Demand Mild PTAFR 30 44 CCC[C@H](C(=O)N1CCC(C#N)CC1)c1ccccc1 ZINC000147204192 CG On-Demand Mild KCNQ2 16 43 CCC[C@H](C(=O)N1CCC(C#N)CC1)c1ccccc1 ZINC000147204192 CG On-Demand Mild DPP4 31 41 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cnn(C[C@@H]2CCCO2)c1 ZINC000147204223 GE On-Demand Anodyne CCR8 64 36 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cnn(C[C@@H]2CCCO2)c1 ZINC000147204223 GE On-Demand Anodyne PANC 56 38 CCOc1c(Cl)cc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1OC ZINC000147204288 HH On-Demand Anodyne ROCK2 21 40 CCOc1c(Cl)cc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1OC ZINC000147204288 HH On-Demand Anodyne PDE6A 40 31 CCc1ncc(C(=O)N(CC)CC(=O)Nc2cccc(OC)c2)s1 ZINC000147204353 EF On-Demand Anodyne PDGFRB 19 40 CCc1ncc(C(=O)N(CC)CC(=O)Nc2cccc(OC)c2)s1 ZINC000147204353 EF On-Demand Anodyne MTNR1A 30 40 CCc1ncc(C(=O)N(CC)CC(=O)Nc2cccc(OC)c2)s1 ZINC000147204353 EF On-Demand Anodyne MTNR1B 37 43 CCc1ncc(C(=O)N(CC)CC(=O)Nc2cccc(OC)c2)s1 ZINC000147204353 EF On-Demand Anodyne FLT4 21 40 CCc1ncc(C(=O)N(CC)CC(=O)Nc2cccc(OC)c2)s1 ZINC000147204353 EF On-Demand Anodyne HSD17B2 20 40 CN(CC(=O)N1CCOCC1)C(=O)c1cccc(NC(=O)c2cccs2)c1 ZINC000147204374 GD On-Demand Anodyne EPHX2 20 41 CN(CC(=O)N1CCOCC1)C(=O)c1cccc(NC(=O)c2cccs2)c1 ZINC000147204374 GD On-Demand Anodyne KCNK3 44 48 CN(CC(=O)N1CCOCC1)C(=O)c1cccc(NC(=O)c2cccs2)c1 ZINC000147204374 GD On-Demand Anodyne KCNK9 30 48 CCC[C@@H](C(=O)N1CCC(C#N)CC1)c1ccccc1 ZINC000147204388 CG On-Demand Mild P2RY12 63 33 CCC[C@@H](C(=O)N1CCC(C#N)CC1)c1ccccc1 ZINC000147204388 CG On-Demand Mild GRIN2B 20 42 CCC[C@@H](C(=O)N1CCC(C#N)CC1)c1ccccc1 ZINC000147204388 CG On-Demand Mild PTAFR 30 44 CCC[C@@H](C(=O)N1CCC(C#N)CC1)c1ccccc1 ZINC000147204388 CG On-Demand Mild KCNQ2 16 43 CCC[C@@H](C(=O)N1CCC(C#N)CC1)c1ccccc1 ZINC000147204388 CG On-Demand Mild DPP4 31 41 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cnn(C[C@H]2CCCO2)c1 ZINC000147204426 GE On-Demand Anodyne CCR8 64 36 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cnn(C[C@H]2CCCO2)c1 ZINC000147204426 GE On-Demand Anodyne PANC 56 38 N#Cc1cc2ccccc2c(-c2ccccc2)c1C#N ZINC000147204566 CI For-Sale Mild FASN 15 40 COc1ccc(CNCCC(=O)N2CCOCC2)cc1OCCCC#N ZINC000147204582 FD On-Demand Mild REN 21 50 CSCC[C@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147204884 GF On-Demand Mild P2RY12 159 36 CSCC[C@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147204884 GF On-Demand Mild UGCG 47 35 CSCC[C@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147204884 GF On-Demand Mild MC4R 50 36 CSCC[C@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147204884 GF On-Demand Mild CCR1 40 46 CSCC[C@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147204884 GF On-Demand Mild PREP 15 53 CSCC[C@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147204884 GF On-Demand Mild CCKBR 22 41 C[C@@H]1Cc2cc([N+](=O)[O-])cc(I)c2N1 ZINC000147204928 DF For-Sale Bother PNMT 21 48 Cc1ccc(C)n1-c1c(C(=O)Nc2cnn(C[C@@H]3CCCO3)c2)cnn1C ZINC000147205042 FE On-Demand Anodyne PANC 55 38 CSCC[C@@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147205085 GF On-Demand Mild P2RY12 159 36 CSCC[C@@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147205085 GF On-Demand Mild UGCG 47 35 CSCC[C@@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147205085 GF On-Demand Mild MC4R 50 36 CSCC[C@@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147205085 GF On-Demand Mild CCR1 40 46 CSCC[C@@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147205085 GF On-Demand Mild PREP 15 53 CSCC[C@@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147205085 GF On-Demand Mild CCKBR 22 41 C[C@H]1Cc2cc([N+](=O)[O-])cc(I)c2N1 ZINC000147205127 DF For-Sale Bother PNMT 21 48 Cc1ccc(NC2=C(c3ccc(C)cc3)C(=O)N(c3ccc(C)cc3)C2=O)cc1 ZINC000147205171 GK For-Sale Anodyne NR1H2 0 49 Cc1ccc(C)n1-c1c(C(=O)Nc2cnn(C[C@H]3CCCO3)c2)cnn1C ZINC000147205202 FE On-Demand Anodyne PANC 55 38 CSCC[C@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147205248 GE On-Demand Mild P2RY12 210 41 CSCC[C@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147205248 GE On-Demand Mild CCR1 17 42 CSCC[C@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147205248 GE On-Demand Mild CPT1A 40 38 CN(C)c1nc(N)nc(Oc2cccc3ccccc23)n1 ZINC000147205265 CE For-Sale Anodyne DHFR 18 40 CN(C)c1nc(N)nc(Oc2cccc3ccccc23)n1 ZINC000147205265 CE For-Sale Anodyne DYR_PNECA 33 40 Nc1ncc(N2CCOCC2)cn1 ZINC000147205371 AB For-Sale Anodyne ADK 18 42 Nc1ncc(N2CCOCC2)cn1 ZINC000147205371 AB For-Sale Anodyne PIK3CA 28 48 Nc1ncc(N2CCOCC2)cn1 ZINC000147205371 AB For-Sale Anodyne PIK3CB 15 44 Nc1ncc(N2CCOCC2)cn1 ZINC000147205371 AB For-Sale Anodyne AKR1C3 0 43 NC(=O)COc1ccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147205388 HD On-Demand Anodyne ROCK2 24 41 NC(=O)c1ccc(OCC(=O)Nc2cnn(C[C@@H]3CCCO3)c2)cc1 ZINC000147205389 ED On-Demand Anodyne HIF1A 24 41 NC(=O)c1ccc(OCC(=O)Nc2cnn(C[C@@H]3CCCO3)c2)cc1 ZINC000147205389 ED On-Demand Anodyne PANC 52 34 CSCC[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147205460 GE On-Demand Mild P2RY12 210 41 CSCC[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147205460 GE On-Demand Mild CCR1 17 42 CSCC[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147205460 GE On-Demand Mild CPT1A 40 38 Cc1cc(C)nc(NNC(=O)c2nn(-c3ccccc3C)c3c2CCC3)n1 ZINC000147205480 FF On-Demand Reactive CNR1 40 31 NC(=O)COc1ccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147205564 HD On-Demand Anodyne ROCK2 24 41 NC(=O)c1ccc(OCC(=O)Nc2cnn(C[C@H]3CCCO3)c2)cc1 ZINC000147205593 ED On-Demand Anodyne HIF1A 24 41 NC(=O)c1ccc(OCC(=O)Nc2cnn(C[C@H]3CCCO3)c2)cc1 ZINC000147205593 ED On-Demand Anodyne PANC 52 34 CCOc1nc(N)nc(Oc2cccc3ccccc23)n1 ZINC000147205628 CF For-Sale Anodyne DHFR 20 40 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(c3ncc(Cl)cc3Cl)CC2)c1 ZINC000147205684 HG On-Demand Bother P2RY12 27 43 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(c3ncc(Cl)cc3Cl)CC2)c1 ZINC000147205684 HG On-Demand Bother SLC6A9 18 44 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne ACHE 30 43 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne EDNRB 32 40 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne EDNRA 54 44 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne TACR1 41 46 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MC4R 58 42 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne TACR2 23 41 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne CCKAR 75 43 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne CTSL 29 40 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MPO 55 44 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne BRS3 42 43 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne NMBR 43 33 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MC5R 44 31 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MTNR1A 17 40 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MMP2 22 40 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MMP8 43 40 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne GRIA1 21 43 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MMP14 72 40 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne GRPR 56 32 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne ECE1 43 37 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne HDAC3 15 40 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MMP11 51 33 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne CCKBR 59 39 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne GHSR 59 35 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne ALOX15 22 40 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MMP9 19 41 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MC1R 59 39 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MMP7 17 40 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne MMP1 21 40 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne AANAT 57 34 CC(C)OC(=O)CCNC(=O)CCCc1c[nH]c2ccccc12 ZINC000147205705 DF On-Demand Anodyne KISS1R 58 33 Cc1cc2c([nH]1)c(I)cc1nc(N)nc(N)c12 ZINC000147205707 EE For-Sale Anodyne DFR1 78 47 Cc1cc2c([nH]1)c(I)cc1nc(N)nc(N)c12 ZINC000147205707 EE For-Sale Anodyne HT1 23 41 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(OCC(N)=O)cc3)c2)CCO1 ZINC000147205807 HE On-Demand Anodyne HRH2 32 44 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(OCC(N)=O)cc3)c2)CCO1 ZINC000147205807 HE On-Demand Anodyne CCR3 17 42 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(OCC(N)=O)cc3)c2)CCO1 ZINC000147205807 HE On-Demand Anodyne EPHX2 26 42 COc1cc(F)ccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147205907 DD On-Demand Anodyne GRIN2B 23 47 COc1cc(F)ccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147205907 DD On-Demand Anodyne ACKR3 46 32 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ncc(Cc3ccc(Cl)cc3C)s2)c1 ZINC000147205929 HJ On-Demand Bother F10 50 33 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ncc(Cc3ccc(Cl)cc3C)s2)c1 ZINC000147205929 HJ On-Demand Bother SCD1 38 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ncc(Cc3ccc(Cl)cc3C)s2)c1 ZINC000147205929 HJ On-Demand Bother SCD 31 41 C[C@@H]1C[C@@H](c2cccc(Cl)c2)[C@@H](c2ccc(Cl)cc2)OC1=O ZINC000147205941 EK For-Sale Anodyne MDM2 142 39 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(OCC(N)=O)cc3)c2)CCO1 ZINC000147205982 HE On-Demand Anodyne HRH2 32 44 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(OCC(N)=O)cc3)c2)CCO1 ZINC000147205982 HE On-Demand Anodyne CCR3 17 42 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(OCC(N)=O)cc3)c2)CCO1 ZINC000147205982 HE On-Demand Anodyne EPHX2 26 42 COc1ccc2nc(N(C)CCN)sc2c1 ZINC000147206010 BD For-Sale Anodyne CSNK1D 21 43 COc1ccc2nc(N(C)CCN)sc2c1 ZINC000147206010 BD For-Sale Anodyne LUCI_PHOPY 16 47 COc1ccc2nc(N(C)CCN)sc2c1 ZINC000147206010 BD For-Sale Anodyne LUCI_PHOPE 37 47 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne HPRT1 56 38 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne P2RX5 0 41 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne POLB 37 48 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne PNP 24 42 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne P2RX4 43 41 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne P2RX1 60 41 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne P2RX6 0 41 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne P2RY4 39 46 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne P2RY1 117 41 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne MAT1A 0 42 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne P2RY2 57 46 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne IMPDH2 0 41 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne EIF4E 0 48 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne RNASE1 43 34 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne RAC1 0 55 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne GPR17 48 38 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne Q3ZDS5_9HEPC 0 52 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne CNGA2 0 46 C[C@H](O[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)[C@]12CO[C@H]([C@@H]1O)[C@H](n1cnc3c(=O)[nH]c(N)nc31)O2 ZINC000147206022 KA Annotated Anodyne ROCR 0 46 COc1cc(F)ccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147206072 DD On-Demand Anodyne GRIN2B 23 47 COc1cc(F)ccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147206072 DD On-Demand Anodyne ACKR3 46 32 Nc1cn2ccnc2c(Oc2cccc3ccccc23)n1 ZINC000147206078 CG For-Sale Anodyne HIVRT 0 41 C[C@H]1C[C@@H](c2cccc(Cl)c2)[C@@H](c2ccc(Cl)cc2)OC1=O ZINC000147206136 EK For-Sale Anodyne MDM2 142 39 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)c3ccc(C)c(OC)c3)CC2)c1 ZINC000147206172 HF On-Demand Bother AKR1C3 16 41 Cc1cc(C)n(Cc2ccc(C(=O)[C@@H](C#N)c3nc4ccccc4n3C(F)F)cc2)n1 ZINC000147206208 HJ On-Demand Mild PDE6D 57 34 CN(C)C(=O)c1ccccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147206267 ED On-Demand Anodyne CXCR2 63 35 CN(C)C(=O)c1ccccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147206267 ED On-Demand Anodyne CXCR1 63 34 CC(=O)Nc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206367 GD On-Demand Mild ST14 57 38 Cc1cc(C)n(Cc2ccc(C(=O)[C@H](C#N)c3nc4ccccc4n3C(F)F)cc2)n1 ZINC000147206382 HJ On-Demand Mild PDE6D 57 34 CCOC[C@H](C)NC(=O)Nc1ccc(OCC(N)=O)cc1 ZINC000147206402 CD On-Demand Anodyne CA12 16 40 CCOC[C@H](C)NC(=O)Nc1ccc(OCC(N)=O)cc1 ZINC000147206402 CD On-Demand Anodyne CA9 17 40 CCOC[C@H](C)NC(=O)Nc1ccc(OCC(N)=O)cc1 ZINC000147206402 CD On-Demand Anodyne NCE103 15 40 CN(C)C(=O)c1ccccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147206485 ED On-Demand Anodyne CXCR2 63 35 CN(C)C(=O)c1ccccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147206485 ED On-Demand Anodyne CXCR1 63 34 C[C@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147206522 DD On-Demand Mild P2RY12 86 36 C[C@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147206522 DD On-Demand Mild COLA 74 39 C[C@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147206522 DD On-Demand Mild CPT1A 68 39 C[C@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147206522 DD On-Demand Mild DPP4 16 40 C[C@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147206522 DD On-Demand Mild CAPN2 40 39 O=C(Nc1cnn(C[C@@H]2CCCO2)c1)C(=O)c1ccc2c(c1)CCC2 ZINC000147206547 EE On-Demand Anodyne PANC 53 35 O=C(Nc1cnn(C[C@H]2CCCO2)c1)C(=O)c1ccc2c(c1)CCC2 ZINC000147206683 EE On-Demand Anodyne PANC 53 35 CC[C@@H](N)CCn1ccnc1 ZINC000147206685 AD For-Sale Anodyne CYP11B1 28 40 CC[C@@H](N)CCn1ccnc1 ZINC000147206685 AD For-Sale Anodyne TBXAS1 33 50 CC[C@@H](N)CCn1ccnc1 ZINC000147206685 AD For-Sale Anodyne CYP11B2 23 40 C[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147206686 DD On-Demand Mild P2RY12 86 36 C[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147206686 DD On-Demand Mild CPT1A 68 39 C[C@@H](NC(=O)COc1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147206686 DD On-Demand Mild DPP4 16 40 Cc1cc(C(=O)NCC2(N(C)C)CCCCC2)cc([N+](=O)[O-])c1 ZINC000147206693 DF On-Demand Bother SLC6A5 17 47 N#Cc1nc(Cl)nc2[nH]cnc12 ZINC000147206754 AC For-Sale Mild PRIM_HHV11 40 35 N#Cc1nc(Cl)nc2[nH]cnc12 ZINC000147206754 AC For-Sale Mild AHK4 0 44 N#Cc1nc(Cl)nc2[nH]cnc12 ZINC000147206754 AC For-Sale Mild AHK3 0 40 N#Cc1nc(Cl)nc2[nH]cnc12 ZINC000147206754 AC For-Sale Mild CKX2 0 42 CC[C@H](N)CCn1ccnc1 ZINC000147206871 AD For-Sale Anodyne CYP11B1 28 40 CC[C@H](N)CCn1ccnc1 ZINC000147206871 AD For-Sale Anodyne TBXAS1 33 50 CC[C@H](N)CCn1ccnc1 ZINC000147206871 AD For-Sale Anodyne CYP11B2 23 40 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild F2 23 44 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild CHRM2 50 40 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild BMP1 30 40 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild MMP13 68 50 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild TRY2_BOVIN 60 35 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild MMP2 42 52 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild MMP3 58 53 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild MMP8 49 53 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild MMP9 45 48 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild MMP12 20 41 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild ST14 45 34 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild MMP7 60 44 COc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147206888 FD On-Demand Mild MMP1 57 45 CN1CC(C(=O)c2ccc(Br)cc2)C1 ZINC000147207073 CE For-Sale Anodyne SLC18A3 26 44 Cc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147207078 ED On-Demand Mild F2 18 44 Cc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147207078 ED On-Demand Mild MMP13 31 46 Cc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147207078 ED On-Demand Mild MMP2 24 42 Cc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147207078 ED On-Demand Mild MMP8 16 42 Cc1ccc(S(=O)(=O)N[C@@H](C)C(=O)N2CCC(C#N)CC2)cc1 ZINC000147207078 ED On-Demand Mild ST14 61 42 COC(=O)c1cnc(-c2ccc3ccccc3c2)s1 ZINC000147207297 CH For-Sale Anodyne CYP11B2 16 46 NC(=O)COc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147207350 HG On-Demand Anodyne ROCK2 28 49 NC(=O)COc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147207350 HG On-Demand Anodyne MET 53 46 NC(=O)COc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147207350 HG On-Demand Anodyne NAMPT 57 52 COc1ccc(CNC2CCN(C(=O)c3ccncc3)CC2)cc1OCCCC#N ZINC000147207387 HG On-Demand Mild SSTR5 53 37 COCCNC(=O)c1cccc(SC)c1 ZINC000147207665 BD On-Demand Anodyne DRD4 49 37 NC(=O)COc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147207681 GF On-Demand Anodyne EPHX2 15 40 N#CC1CCN(C(=O)c2ccc(OC[C@H]3CCCO3)cc2)CC1 ZINC000147207842 DF On-Demand Mild L3MBTL3 66 38 NC(=O)COc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147207865 GF On-Demand Anodyne EPHX2 15 40 CC(C)(C)C(=O)Oc1cccc(O)c1 ZINC000147207906 AE For-Sale Anodyne ELANE 30 55 CC(C)(C)C(=O)Oc1cccc(O)c1 ZINC000147207906 AE For-Sale Anodyne PRTN3 58 38 CC(C)(C)C(=O)Oc1cccc(O)c1 ZINC000147207906 AE For-Sale Anodyne HSD17B1 47 40 CC(C)(C)C(=O)Oc1cccc(O)c1 ZINC000147207906 AE For-Sale Anodyne KYNU 42 30 CC(C)(C)C(=O)Oc1cccc(O)c1 ZINC000147207906 AE For-Sale Anodyne HSD17B2 37 40 COC(=O)c1cnc(Cc2ccc(Cl)c(Cl)c2)s1 ZINC000147207973 DH For-Sale Anodyne SCD1 25 42 Cc1cc(OCC(=O)N2CCC(C#N)CC2)ccc1C(C)C ZINC000147208032 DG On-Demand Mild HTR1D 15 40 Cc1cc(OCC(=O)N2CCC(C#N)CC2)ccc1C(C)C ZINC000147208032 DG On-Demand Mild HTR1B 19 40 NC(=O)COc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147208079 GF On-Demand Anodyne EPHX2 15 40 COC(=O)c1cnc(CCc2ccccc2)s1 ZINC000147208167 BF For-Sale Anodyne FAAH 63 47 COC(=O)c1cnc(CCc2ccccc2)s1 ZINC000147208167 BF For-Sale Anodyne CES1 60 43 COC(=O)c1cnc(CCc2ccccc2)s1 ZINC000147208167 BF For-Sale Anodyne FAS 57 37 NC(=O)COc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147208268 GF On-Demand Anodyne EPHX2 15 40 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(-c2ccccc2)cc1 ZINC000147208288 FJ On-Demand Anodyne BMP1 58 39 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(-c2ccccc2)cc1 ZINC000147208288 FJ On-Demand Anodyne ACACA 26 43 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(-c2ccccc2)cc1 ZINC000147208288 FJ On-Demand Anodyne ACACB 31 43 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(-c2ccccc2)cc1 ZINC000147208288 FJ On-Demand Anodyne CYP3A4 22 48 Cc1cc(C(=O)OC(C)C)cc(C(=O)OC(C)C)c1 ZINC000147208348 CG On-Demand Anodyne CA14 18 64 C/C=C1/CN(C)[C@H]2Cc3c([nH]c4ccccc34)[C@H](O)C[C@H]1[C@@H]2C(=O)OC ZINC000147208354 FF Annotated Anodyne PDE5A 0 43 C/C=C1/CN(C)[C@H]2Cc3c([nH]c4ccccc34)[C@H](O)C[C@H]1[C@@H]2C(=O)OC ZINC000147208354 FF Annotated Anodyne SLC6A1 77 39 COC=C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147208465 DH For-Sale Anodyne GRIN2B 21 44 COC=C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147208465 DH For-Sale Anodyne PREP 23 40 COC=C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147208465 DH For-Sale Anodyne TGM2 42 41 COC=C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147208465 DH For-Sale Anodyne F13A1 43 41 COC=C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147208465 DH For-Sale Anodyne SLC12A5 77 43 C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(-c2ccccc2)cc1 ZINC000147208467 FJ On-Demand Anodyne BMP1 58 39 C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(-c2ccccc2)cc1 ZINC000147208467 FJ On-Demand Anodyne ACACA 26 43 C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(-c2ccccc2)cc1 ZINC000147208467 FJ On-Demand Anodyne ACACB 31 43 C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(-c2ccccc2)cc1 ZINC000147208467 FJ On-Demand Anodyne CYP3A4 22 48 C/C=C1/CN(C)[C@H]2Cc3c([nH]c4ccccc34)[C@H](OC)C[C@H]1[C@@H]2C(=O)OC ZINC000147208526 FG Annotated Anodyne PDE5A 0 43 C/C=C1/CN(C)[C@H]2Cc3c([nH]c4ccccc34)[C@H](OC)C[C@H]1[C@@H]2C(=O)OC ZINC000147208526 FG Annotated Anodyne SLC6A1 73 39 COC(=O)Nc1ccc2c(c1)NC(=O)[C@H](C)CCC[C@H](N1CC[C@@H](c3nccc(Cl)c3F)N(C)C1=O)c1nc-2c[nH]1 ZINC000147208590 KK Annotated Anodyne KLKB1 21 58 COC(=O)Nc1ccc2c(c1)NC(=O)[C@H](C)CCC[C@H](N1CC[C@@H](c3nccc(Cl)c3F)N(C)C1=O)c1nc-2c[nH]1 ZINC000147208590 KK Annotated Anodyne F11 28 54 O=C(NCC(F)(F)F)Nc1cccc(-c2cnc3cc(-c4nccc(C(F)(F)F)n4)ccn23)c1 ZINC000147208598 JK Annotated Anodyne GYRB 0 40 O=C(NCC(F)(F)F)Nc1cccc(-c2cnc3cc(-c4nccc(C(F)(F)F)n4)ccn23)c1 ZINC000147208598 JK Annotated Anodyne BRAF 44 41 CC(C)Oc1cccc(CC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000147208610 GH On-Demand Anodyne HRH2 30 40 CC(C)Oc1cccc(CC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000147208610 GH On-Demand Anodyne MMP13 20 44 CC(C)Oc1cccc(CC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000147208610 GH On-Demand Anodyne PREP 18 42 CC(C)Oc1cccc(CC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000147208610 GH On-Demand Anodyne FURIN 51 34 CC(C)Oc1cccc(CC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000147208610 GH On-Demand Anodyne DPP7 50 42 CC(C)Oc1cccc(CC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000147208610 GH On-Demand Anodyne TAAR1 19 41 CC(C)Oc1cccc(CC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000147208610 GH On-Demand Anodyne L3MBTL3 49 36 CC(C)Oc1cccc(CC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000147208610 GH On-Demand Anodyne HPGD 36 40 CC(C)Oc1cccc(CC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000147208610 GH On-Demand Anodyne NAMPT 20 45 CC(C)Oc1cccc(CC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)c1 ZINC000147208610 GH On-Demand Anodyne PDS 43 33 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)N(C)Cc1ccccc1)C2 ZINC000147208616 FE On-Demand Anodyne MTNR1A 51 43 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)N(C)Cc1ccccc1)C2 ZINC000147208616 FE On-Demand Anodyne MTNR1B 42 42 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)N(C)Cc1ccccc1)C2 ZINC000147208616 FE On-Demand Anodyne ROCK2 33 40 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)N(C)Cc1ccccc1)C2 ZINC000147208616 FE On-Demand Anodyne ADAM9 50 36 CCc1nc(CN(C)C(=O)N[C@@H](C)c2ccc(-c3ccccc3)cc2)cs1 ZINC000147208665 GK On-Demand Anodyne ACACA 22 40 CCc1nc(CN(C)C(=O)N[C@@H](C)c2ccc(-c3ccccc3)cc2)cs1 ZINC000147208665 GK On-Demand Anodyne ACACB 21 40 CCC[C@@H](NC(N)=O)C(=O)Nc1cnn(C[C@@H]2CCCO2)c1 ZINC000147208708 DC On-Demand Anodyne PANC 54 36 CNc1cn2ccnc2c(Oc2ccc(OC)cc2)n1 ZINC000147208776 CF For-Sale Anodyne HIVRT 0 45 CN1C(=O)Cn2c1nc1nc(N3CCC[C@@H](N)C3)n(Cc3ccccc3C#N)c1c2=O ZINC000147208864 HC Annotated Mild DPP4 58 69 CCc1nc(CN(C)C(=O)N[C@H](C)c2ccc(-c3ccccc3)cc2)cs1 ZINC000147208881 GK On-Demand Anodyne ACACA 22 40 CCc1nc(CN(C)C(=O)N[C@H](C)c2ccc(-c3ccccc3)cc2)cs1 ZINC000147208881 GK On-Demand Anodyne ACACB 21 40 CNc1ncc(Cl)c(Oc2ccc(OC)cc2)n1 ZINC000147209009 CF For-Sale Anodyne NPBWR1 78 35 CCC[C@@H](NC(N)=O)C(=O)Nc1cnn(C[C@H]2CCCO2)c1 ZINC000147209089 DC On-Demand Anodyne PANC 54 36 CS(=O)(=O)c1cc(C(=O)Nc2ccccc2OC2CCCC2)cc([N+](=O)[O-])c1 ZINC000147209120 HH On-Demand Bother PYGL 22 41 NC(=O)[C@H]1CCCN1Cl ZINC000147209124 AC For-Sale Anodyne TPP2 15 46 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147209212 GH On-Demand Anodyne TRY2_BOVIN 57 38 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147209212 GH On-Demand Anodyne F2R 51 33 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147209212 GH On-Demand Anodyne FURIN 53 34 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147209212 GH On-Demand Anodyne DPP7 49 36 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147209212 GH On-Demand Anodyne PROC 43 34 NC(=O)[C@@H]1CCCN1Cl ZINC000147209307 AC For-Sale Anodyne TPP2 15 46 N#CC1CCN(C(=O)CCC(=O)c2ccccc2)CC1 ZINC000147209355 CE On-Demand Mild DPP4 17 40 N#CC1CCN(C(=O)CCC(=O)c2ccccc2)CC1 ZINC000147209355 CE On-Demand Mild PREP 37 49 N#CC1CCN(C(=O)CCC(=O)c2ccccc2)CC1 ZINC000147209355 CE On-Demand Mild CYP2J2 47 33 N#CC1CCN(C(=O)CCC(=O)c2ccccc2)CC1 ZINC000147209355 CE On-Demand Mild ETHR 42 38 C[C@H](Cc1cccc(F)c1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147209400 GH On-Demand Anodyne TRY2_BOVIN 57 38 C[C@H](Cc1cccc(F)c1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147209400 GH On-Demand Anodyne F2R 51 33 C[C@H](Cc1cccc(F)c1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147209400 GH On-Demand Anodyne FURIN 53 34 C[C@H](Cc1cccc(F)c1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147209400 GH On-Demand Anodyne DPP7 49 36 C[C@H](Cc1cccc(F)c1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147209400 GH On-Demand Anodyne PROC 43 34 CN(C)C(=O)c1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1Cl ZINC000147209457 FD On-Demand Anodyne ENV 44 36 CN(Cc1ccccc1)C(=O)CNC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147209587 FG On-Demand Anodyne LIMK2 24 42 CN(Cc1ccccc1)C(=O)CNC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147209587 FG On-Demand Anodyne GPR88 0 41 CCCNc1ncc(Cl)c(Oc2ccc(OC)cc2)n1 ZINC000147209614 CH For-Sale Anodyne NPBWR1 77 34 CN(C)C(=O)c1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1Cl ZINC000147209658 FD On-Demand Anodyne ENV 44 36 COC(=O)c1cnc(Cc2cccc(OC)c2)s1 ZINC000147209710 CF For-Sale Anodyne ROCK1 41 41 COC(=O)c1cnc(Cc2cccc(OC)c2)s1 ZINC000147209710 CF For-Sale Anodyne MTNR1A 44 44 COC(=O)c1cnc(Cc2cccc(OC)c2)s1 ZINC000147209710 CF For-Sale Anodyne MTNR1B 46 44 COC(=O)c1cnc(Cc2cccc(OC)c2)s1 ZINC000147209710 CF For-Sale Anodyne ROCK2 47 41 COC(=O)c1cnc(Cc2cccc(OC)c2)s1 ZINC000147209710 CF For-Sale Anodyne HSD17B2 23 41 COC(=O)c1cnc(Cc2cccc(OC)c2)s1 ZINC000147209710 CF For-Sale Anodyne SCD1 24 43 CN(Cc1ccccc1)C(=O)CNC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147209786 FG On-Demand Anodyne LIMK2 24 42 CN(Cc1ccccc1)C(=O)CNC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147209786 FG On-Demand Anodyne GPR88 0 41 CC(=O)Nc1cc(NC(C)=O)cc(C(=O)Nc2nc(-c3c[nH]c(C(N)=O)c3)cs2)c1 ZINC000147209808 IE On-Demand Anodyne MPL 44 39 CN(Cc1ccccc1)C(=O)CNC(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147209969 FG On-Demand Anodyne LIMK2 24 42 CN(Cc1ccccc1)C(=O)CNC(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147209969 FG On-Demand Anodyne GPR88 0 41 CC(C)(C)OC(=O)c1ccc(CN2CCC(CO)CC2)cc1 ZINC000147209976 DF In-Stock Anodyne ACHE 40 44 CC(C)(C)OC(=O)c1ccc(CN2CCC(CO)CC2)cc1 ZINC000147209976 DF In-Stock Anodyne SIGMAR1 51 50 CC(C)(C)OC(=O)c1ccc(CN2CCC(CO)CC2)cc1 ZINC000147209976 DF In-Stock Anodyne CCR3 24 43 CC(C)(C)OC(=O)c1ccc(CN2CCC(CO)CC2)cc1 ZINC000147209976 DF In-Stock Anodyne MCHR1 36 41 CC(C)(C)OC(=O)c1ccc(CN2CCC(CO)CC2)cc1 ZINC000147209976 DF In-Stock Anodyne CACNA1I 59 38 CC(C)(C)OC(=O)c1ccc(CN2CCC(CO)CC2)cc1 ZINC000147209976 DF In-Stock Anodyne PANC 24 40 CC(C)(C)OC(=O)c1ccc(CN2CCC(CO)CC2)cc1 ZINC000147209976 DF In-Stock Anodyne NOD2 41 36 Cc1cc(C(=O)N(C)Cc2ccc(Br)cc2)cc([N+](=O)[O-])c1 ZINC000147210171 FH On-Demand Bother MMP8 24 41 Cc1cc(C(=O)N(C)Cc2ccc(Br)cc2)cc([N+](=O)[O-])c1 ZINC000147210171 FH On-Demand Bother MMP1 24 41 O=C(Nc1ccc(C(=O)N2CCOCC2)c(Cl)c1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147210179 HI On-Demand Anodyne AVPR2 40 38 Cn1ccc(-c2ccc(CNC(=O)c3c(Cl)cccc3Cl)cc2)cc1=O ZINC000147210236 GI Annotated Anodyne UL54 76 35 Cn1ccc(-c2ccc(CNC(=O)c3c(Cl)cccc3Cl)cc2)cc1=O ZINC000147210236 GI Annotated Anodyne RPA1 54 37 CCc1ncc(C(=O)NCCc2ccc(C(F)(F)F)cc2)s1 ZINC000147210377 EH On-Demand Anodyne PPARD 23 41 O=C(Nc1ccc(C(=O)N2CCOCC2)c(Cl)c1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147210394 HI On-Demand Anodyne AVPR2 40 38 COc1ccc(CN[C@H](c2ccc3c(c2)OCCO3)C2CC2)cc1OCCCC#N ZINC000147210405 HI On-Demand Mild PDE10A 22 42 Cn1cc(C(=O)NC2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)cn1 ZINC000147210586 GC On-Demand Anodyne PLG 18 40 Cn1cc(C(=O)NC2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)cn1 ZINC000147210586 GC On-Demand Anodyne SSTR5 43 37 Cn1cc(C(=O)NC2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)cn1 ZINC000147210586 GC On-Demand Anodyne CPT1A 59 42 Cn1cc(C(=O)NC2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)cn1 ZINC000147210586 GC On-Demand Anodyne SLC6A5 38 43 Cn1cc(C(=O)NC2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)cn1 ZINC000147210586 GC On-Demand Anodyne PLAU 27 43 Cn1cc(C(=O)NC2CCN(C(=O)COc3ccc(C(N)=O)cc3)CC2)cn1 ZINC000147210586 GC On-Demand Anodyne ST14 25 43 O=C(Nc1ccc(C(=O)N2CCOCC2)c(Cl)c1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147210601 HI On-Demand Anodyne AVPR2 40 38 COC(=O)Nc1ccc2c(c1)NC(=O)[C@H](C)CCC[C@H](N1CC[C@H](c3nccc(Cl)c3F)NC1=O)c1nc-2c[nH]1 ZINC000147210605 KK Annotated Anodyne KLKB1 22 59 COC(=O)Nc1ccc2c(c1)NC(=O)[C@H](C)CCC[C@H](N1CC[C@H](c3nccc(Cl)c3F)NC1=O)c1nc-2c[nH]1 ZINC000147210605 KK Annotated Anodyne F11 29 56 Cc1ccc(C(=O)N(C)C)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147210608 ED On-Demand Anodyne MAPK11 32 43 Cc1ccc(C(=O)N(C)C)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147210608 ED On-Demand Anodyne MAPK14 17 43 COC(=O)c1cnc(-c2ccccc2[N+](=O)[O-])s1 ZINC000147210642 CF For-Sale Bother CACNA1D 24 41 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210650 EH On-Demand Anodyne MAPK14 41 39 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210650 EH On-Demand Anodyne CCR3 65 45 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210650 EH On-Demand Anodyne BACE2 16 43 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210650 EH On-Demand Anodyne TIMP3 54 33 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210650 EH On-Demand Anodyne EPHX2 23 45 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210650 EH On-Demand Anodyne ST14 64 38 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210650 EH On-Demand Anodyne MCHR1 22 41 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210650 EH On-Demand Anodyne KCNK3 69 42 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210650 EH On-Demand Anodyne KCNK9 41 42 Cc1ccc(C(=O)N(C)C)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147210782 ED On-Demand Anodyne MAPK11 32 43 Cc1ccc(C(=O)N(C)C)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147210782 ED On-Demand Anodyne MAPK14 17 43 COC(=O)Nc1ccc2c(c1)NC(=O)[C@H](C)CCC[C@H](N1CC[C@@H](c3nccc(Cl)c3F)NC1=O)c1nc-2c[nH]1 ZINC000147210807 KK Annotated Anodyne KLKB1 22 59 COC(=O)Nc1ccc2c(c1)NC(=O)[C@H](C)CCC[C@H](N1CC[C@@H](c3nccc(Cl)c3F)NC1=O)c1nc-2c[nH]1 ZINC000147210807 KK Annotated Anodyne F11 29 56 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210823 EH On-Demand Anodyne MAPK14 41 39 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210823 EH On-Demand Anodyne CCR3 65 45 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210823 EH On-Demand Anodyne BACE2 16 43 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210823 EH On-Demand Anodyne TIMP3 54 33 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210823 EH On-Demand Anodyne EPHX2 23 45 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210823 EH On-Demand Anodyne ST14 64 38 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210823 EH On-Demand Anodyne MCHR1 22 41 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210823 EH On-Demand Anodyne KCNK3 69 42 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147210823 EH On-Demand Anodyne KCNK9 41 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(C(=O)N(C)c3ccccc3)c1)C2 ZINC000147210849 HI On-Demand Anodyne MTNR1A 25 48 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(C(=O)N(C)c3ccccc3)c1)C2 ZINC000147210849 HI On-Demand Anodyne MTNR1B 26 48 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(C(=O)N(C)c3ccccc3)c1)C2 ZINC000147210849 HI On-Demand Anodyne ROCK2 29 47 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(C(=O)N(C)c3ccccc3)c1)C2 ZINC000147210849 HI On-Demand Anodyne HSD17B2 19 44 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(C(=O)N(C)c3ccccc3)c1)C2 ZINC000147210849 HI On-Demand Anodyne AKR1C3 15 40 Cc1ccc(Oc2ccc(Cl)c(Cl)c2)c(C#N)c1 ZINC000147210860 CJ For-Sale Mild AR 17 57 N#CC1CCN(C(=O)COc2ccc3ccc(=O)oc3c2)CC1 ZINC000147210882 DD On-Demand Mild HTR1B 18 40 N#CC1CCN(C(=O)COc2ccc3ccc(=O)oc3c2)CC1 ZINC000147210882 DD On-Demand Mild CA7 25 46 O=C(NCc1ccc(-c2cc(=O)[nH]cc2F)cc1)c1c(Cl)cccc1Cl ZINC000147210895 GI Annotated Anodyne MAPK1 16 41 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne DRD2 21 45 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne DRD4 43 36 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne ACHE 36 42 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne HRH2 20 46 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne DRD3 26 41 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne OPRL1 23 43 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne CHRM3 15 40 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne SIGMAR1 76 41 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne BCHE 19 43 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne NPFFR2 44 48 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne ADAM17 18 41 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne CACNA1G 34 40 CC(C)(C)OC(=O)NCCC1(O)CCN(Cc2ccccc2)CC1 ZINC000147210981 EF In-Stock Anodyne NPFFR1 66 42 NC(=O)c1ccc(OCC(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)cc1 ZINC000147210997 HD On-Demand Anodyne CA2 15 41 NC(=O)c1ccc(OCC(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)cc1 ZINC000147210997 HD On-Demand Anodyne MMP13 42 36 NC(=O)c1ccc(OCC(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)cc1 ZINC000147210997 HD On-Demand Anodyne ADAM17 46 36 NC(=O)c1ccc(OCC(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)cc1 ZINC000147210997 HD On-Demand Anodyne TGM2 60 39 NC(=O)c1ccc(OCC(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)cc1 ZINC000147210997 HD On-Demand Anodyne MMP7 44 34 NC(=O)c1ccc(OCC(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)cc1 ZINC000147210997 HD On-Demand Anodyne CA9 23 41 NC(=O)c1ccc(OCC(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)cc1 ZINC000147210997 HD On-Demand Anodyne MMP1 40 34 NC(=O)c1ccc(OCC(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)cc1 ZINC000147210997 HD On-Demand Anodyne F13A1 61 38 NC(=O)c1ccc(OCC(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)cc1 ZINC000147210997 HD On-Demand Anodyne NAMPT 73 51 NC(=O)c1ccc(OCC(=O)NCc2ccc(S(=O)(=O)N3CCCC3)cc2)cc1 ZINC000147210997 HD On-Demand Anodyne TMPRSS11D 45 32 CNc1ncc(Br)c(Oc2ccc(OC)cc2)n1 ZINC000147211223 DG For-Sale Anodyne TBK1 17 44 COc1ccc(CN[C@@H](C)C(=O)NCc2ccccc2)cc1OCCCC#N ZINC000147211284 GG On-Demand Mild CTSD 15 48 COc1ccc(CN[C@@H](C)C(=O)NCc2ccccc2)cc1OCCCC#N ZINC000147211284 GG On-Demand Mild REN 31 45 COc1ccc(CN[C@@H](C)C(=O)NCc2ccccc2)cc1OCCCC#N ZINC000147211284 GG On-Demand Mild FURIN 52 35 COc1ccc(CN[C@@H](C)C(=O)NCc2ccccc2)cc1OCCCC#N ZINC000147211284 GG On-Demand Mild HCRTR2 18 41 COc1ccc(CN[C@@H](C)C(=O)NCc2ccccc2)cc1OCCCC#N ZINC000147211284 GG On-Demand Mild PDS 49 35 CCc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147211312 DH On-Demand Anodyne BMP1 57 36 CCc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147211312 DH On-Demand Anodyne ACACA 50 39 CCc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147211312 DH On-Demand Anodyne CYP3A4 17 45 COc1cc(/C=C/C(=O)N2CCC(C#N)CC2)ccc1OCC#N ZINC000147211351 EE On-Demand Mild ACKR3 45 33 COc1ccc2nc(NC(=O)c3ccc(F)c(Br)c3)sc2c1 ZINC000147211480 GI On-Demand Anodyne LCK 36 48 COc1ccc2nc(NC(=O)c3ccc(F)c(Br)c3)sc2c1 ZINC000147211480 GI On-Demand Anodyne CSNK1D 60 58 COc1ccc2nc(NC(=O)c3ccc(F)c(Br)c3)sc2c1 ZINC000147211480 GI On-Demand Anodyne NMT1 32 47 COc1ccc2nc(NC(=O)c3ccc(F)c(Br)c3)sc2c1 ZINC000147211480 GI On-Demand Anodyne PIK3CA 20 43 COc1ccc2nc(NC(=O)c3ccc(F)c(Br)c3)sc2c1 ZINC000147211480 GI On-Demand Anodyne HSD17B1 15 58 COc1ccc2nc(NC(=O)c3ccc(F)c(Br)c3)sc2c1 ZINC000147211480 GI On-Demand Anodyne PIK3CG 18 44 COc1ccc2nc(NC(=O)c3ccc(F)c(Br)c3)sc2c1 ZINC000147211480 GI On-Demand Anodyne TAAR1 31 56 COc1ccc2nc(NC(=O)c3ccc(F)c(Br)c3)sc2c1 ZINC000147211480 GI On-Demand Anodyne LUCI_PHOPE 32 45 COc1ccc2nc(NC(=O)c3ccc(F)c(Br)c3)sc2c1 ZINC000147211480 GI On-Demand Anodyne SCD 25 40 CCc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147211505 DH On-Demand Anodyne BMP1 57 36 CCc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147211505 DH On-Demand Anodyne ACACA 50 39 CCc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147211505 DH On-Demand Anodyne CYP3A4 17 45 COC(=O)c1cnc(-c2ccc3ccccc3n2)s1 ZINC000147211536 CG For-Sale Anodyne ALOX5AP 21 40 C[C@]12OC[C@](CO)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147211717 DA Annotated Anodyne HPRT1 54 36 C[C@]12OC[C@](CO)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147211717 DA Annotated Anodyne NS5B 0 58 C[C@]12OC[C@](CO)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147211717 DA Annotated Anodyne EIF4E 0 40 C[C@]12OC[C@](CO)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147211717 DA Annotated Anodyne Q4VQ11_PIG 72 33 C[C@]12OC[C@](CO)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147211717 DA Annotated Anodyne Q3ZDS5_9HEPC 0 50 C[C@]12OC[C@](CO)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147211717 DA Annotated Anodyne UL97 0 43 C[C@]12OC[C@](CO)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147211717 DA Annotated Anodyne CNGA2 0 43 C[C@]12OC[C@](CO)(O[C@H]1n1cnc3c(=O)[nH]c(N)nc31)[C@H]2O ZINC000147211717 DA Annotated Anodyne ROCR 0 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(N2CCCC2=O)ccc1Cl ZINC000147211737 GE On-Demand Anodyne F10 18 46 N#Cc1ccc(C(=O)N[C@@H](c2ccccc2)c2ccc3nc(C(F)(F)F)[nH]c3c2)cc1 ZINC000147211781 HJ On-Demand Mild CTSG 17 42 N#Cc1ccc(C(=O)N[C@@H](c2ccccc2)c2ccc3nc(C(F)(F)F)[nH]c3c2)cc1 ZINC000147211781 HJ On-Demand Mild CELA2A 15 42 N#Cc1ccc(C(=O)N[C@@H](c2ccccc2)c2ccc3nc(C(F)(F)F)[nH]c3c2)cc1 ZINC000147211781 HJ On-Demand Mild CTRB_BOVIN 48 36 Cc1ccc(/C=C/C(=O)N2CCC(C#N)CC2)cc1 ZINC000147211788 CF On-Demand Mild CCR2 61 44 Cc1ccc(/C=C/C(=O)N2CCC(C#N)CC2)cc1 ZINC000147211788 CF On-Demand Mild GPR183 0 54 CC(C)CCO[C@@H](C)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147211884 FG On-Demand Anodyne DPP7 46 38 CC(C)CCO[C@@H](C)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147211884 FG On-Demand Anodyne PROC 42 33 CC(C)CCO[C@@H](C)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147211884 FG On-Demand Anodyne L3MBTL3 46 35 C=CC[C@@]1(C)C[C@H](c2cccc(Cl)c2)[C@H](c2ccc(Cl)cc2)OC1=O ZINC000147211929 GK For-Sale Anodyne TP53 27 44 C=CC[C@@]1(C)C[C@H](c2cccc(Cl)c2)[C@H](c2ccc(Cl)cc2)OC1=O ZINC000147211929 GK For-Sale Anodyne MDM2 161 44 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(N2CCCC2=O)ccc1Cl ZINC000147211941 GE On-Demand Anodyne F10 18 46 CCCOc1ccc(C(=O)CCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147211972 EG On-Demand Mild THRA 33 45 CCCOc1ccc(C(=O)CCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147211972 EG On-Demand Mild THRB 17 44 CCCOc1ccc(C(=O)CCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147211972 EG On-Demand Mild HRH3 18 50 CCCOc1ccc(C(=O)CCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147211972 EG On-Demand Mild PLA2G4B 46 34 COC(=O)c1cnc(-c2cccc([N+](=O)[O-])c2)s1 ZINC000147211976 CF For-Sale Bother CACNA1C 64 40 COC(=O)c1cnc(-c2cccc([N+](=O)[O-])c2)s1 ZINC000147211976 CF For-Sale Bother P2RX7 0 42 COC(=O)c1cnc(-c2cccc([N+](=O)[O-])c2)s1 ZINC000147211976 CF For-Sale Bother CACNA1D 99 40 NC(=O)/C=C/c1ccc(Cl)c(F)c1 ZINC000147211994 AD For-Sale Anodyne PYGL 16 42 N#Cc1ccc(C(=O)N[C@H](c2ccccc2)c2ccc3nc(C(F)(F)F)[nH]c3c2)cc1 ZINC000147211999 HJ On-Demand Mild CTSG 17 42 N#Cc1ccc(C(=O)N[C@H](c2ccccc2)c2ccc3nc(C(F)(F)F)[nH]c3c2)cc1 ZINC000147211999 HJ On-Demand Mild CELA2A 15 42 N#Cc1ccc(C(=O)N[C@H](c2ccccc2)c2ccc3nc(C(F)(F)F)[nH]c3c2)cc1 ZINC000147211999 HJ On-Demand Mild CTRB_BOVIN 48 36 O=C(Nc1cccc2c1C[C@H](O)CC2)N[C@@H]1CC[C@H](c2ccccc2)C1 ZINC000147212036 FH Annotated Anodyne TRPV1 24 49 CC(C)CCO[C@H](C)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147212064 FG On-Demand Anodyne DPP7 46 38 CC(C)CCO[C@H](C)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147212064 FG On-Demand Anodyne PROC 42 33 CC(C)CCO[C@H](C)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147212064 FG On-Demand Anodyne L3MBTL3 46 35 C[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147212168 CD On-Demand Mild ACE 23 44 C[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147212168 CD On-Demand Mild CTSB 15 42 C[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147212168 CD On-Demand Mild CCR1 41 48 C[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147212168 CD On-Demand Mild PREP 25 42 O=C(Nc1cccc2c1C[C@H](O)CC2)N[C@H]1CC[C@H](c2ccccc2)C1 ZINC000147212242 FH Annotated Anodyne TRPV1 24 49 C[C@H](OC[C@@H]1CCCO1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147212270 FF On-Demand Anodyne PROC 47 34 O=C(Nc1cccc(-c2cnco2)c1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147212334 EJ On-Demand Anodyne IMPDH2 0 44 O=C(O)/C=C\c1ccc(Cl)cc1Br ZINC000147212357 CG For-Sale Anodyne APP 40 40 O=C(O)/C=C\c1ccc(Cl)cc1Br ZINC000147212357 CG For-Sale Anodyne BOTA 26 51 COC(=O)CCCCCCCCCCC/C=C/CCCCCCCCCCCC(=O)OC ZINC000147212383 JK For-Sale Anodyne FAAH 16 46 COC(=O)CCCCCCCCCCC/C=C/CCCCCCCCCCCC(=O)OC ZINC000147212383 JK For-Sale Anodyne LPAR3 32 42 COC(=O)CCCCCCCCCCC/C=C/CCCCCCCCCCCC(=O)OC ZINC000147212383 JK For-Sale Anodyne FABP3 42 50 COC(=O)CCCCCCCCCCC/C=C/CCCCCCCCCCCC(=O)OC ZINC000147212383 JK For-Sale Anodyne FABP5 15 50 COC(=O)CCCCCCCCCCC/C=C/CCCCCCCCCCCC(=O)OC ZINC000147212383 JK For-Sale Anodyne FABP1 16 50 O=C(Nc1cccc2c1C[C@H](O)CC2)N[C@@H]1CC[C@@H](c2ccccc2)C1 ZINC000147212445 FH Annotated Anodyne TRPV1 24 49 C[C@@H](OC[C@@H]1CCCO1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147212484 FF On-Demand Anodyne PROC 47 34 O=C(Nc1cccc(-c2cnco2)c1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147212525 EJ On-Demand Anodyne IMPDH2 0 44 C[C@H](OC[C@H]1CCCO1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147212686 FF On-Demand Anodyne PROC 47 34 CCC(CC)C1=NO[C@H]2[C@H]1[C@H](NC(=O)OC(C)(C)C)C[C@H]2C(=O)O ZINC000147212698 EF Annotated Anodyne PAPA1_CARPA 41 32 O=C(Nc1cccc(-c2cnco2)c1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147212758 EJ On-Demand Anodyne IMPDH2 0 44 C[C@@H](OC[C@H]1CCCO1)C(=O)NCc1ccc(C(=O)N2CCCCC2)cc1 ZINC000147212868 FF On-Demand Anodyne PROC 47 34 CC(C)c1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147212930 DI On-Demand Anodyne BMP1 48 34 CC(C)c1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147212930 DI On-Demand Anodyne ACACA 48 39 CC(C)c1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147212930 DI On-Demand Anodyne CYP3A4 18 45 COC(=O)c1cnc([C@@H]2COc3ccccc3O2)s1 ZINC000147212933 CE For-Sale Anodyne ADRA2B 20 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(-c3cnco3)c1)C2 ZINC000147212956 FH On-Demand Anodyne ROCK2 44 53 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(-c3cnco3)c1)C2 ZINC000147212956 FH On-Demand Anodyne IMPDH2 0 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(-c3cnco3)c1)C2 ZINC000147212956 FH On-Demand Anodyne CDC42BPA 0 44 COc1ccc(C(=O)NNC(=O)c2occ(-c3ccccc3)c2-c2ccccc2)cc1 ZINC000147213036 HJ Annotated Reactive GCGR 56 74 CC(C)c1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147213121 DI On-Demand Anodyne BMP1 48 34 CC(C)c1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147213121 DI On-Demand Anodyne ACACA 48 39 CC(C)c1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147213121 DI On-Demand Anodyne CYP3A4 18 45 COC(=O)c1cnc([C@H]2COc3ccccc3O2)s1 ZINC000147213128 CE For-Sale Anodyne ADRA2B 20 40 O=C(Nc1ccc(-c2cn3cccnc3n2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147213184 HI On-Demand Anodyne GRM4 51 36 O=C(Nc1ccc(-c2cn3cccnc3n2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147213184 HI On-Demand Anodyne SMO 18 42 O=C1CC2(CCCC2)CCN1CCO ZINC000147213305 AD For-Sale Anodyne ADRA1D 22 48 COC(=O)c1cnc(CSc2cccc(Br)c2)s1 ZINC000147213315 EH For-Sale Anodyne FAS 58 36 COc1ccc(Oc2nc(N)nc3ccccc23)cc1 ZINC000147213353 CG For-Sale Anodyne DHFR 34 41 COc1ccc(Oc2nc(N)nc3ccccc23)cc1 ZINC000147213353 CG For-Sale Anodyne DFR1 26 43 COc1ccc(Oc2nc(N)nc3ccccc23)cc1 ZINC000147213353 CG For-Sale Anodyne DRTS_TOXGO 48 39 COc1ccc(Oc2nc(N)nc3ccccc23)cc1 ZINC000147213353 CG For-Sale Anodyne TUBB3 33 46 COc1ccc(Oc2nc(N)nc3ccccc23)cc1 ZINC000147213353 CG For-Sale Anodyne NPBWR1 44 35 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(-c3cn4cccnc4n3)cc1)C2 ZINC000147213372 HH On-Demand Anodyne ROCK2 49 53 COC(=O)c1cnc(-c2ccc(OC)c(OC)c2)s1 ZINC000147213541 CF On-Demand Anodyne KIT 0 40 C[C@]1(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@@H](c2ccc(Cl)cc2)N([C@H](CS(=O)(=O)N2CCCCC2)C2CC2)C1=O ZINC000147213553 KK Annotated Anodyne TP53 39 61 Cc1cc(C)c(C)c(S(=O)(=O)N2CCC(C(=O)N3CCC(C#N)CC3)CC2)c1C ZINC000147213565 HG On-Demand Mild EPHX2 33 42 CCOC(=O)C1CCN(C(=O)/C=C/c2cc3ccccc3o2)CC1 ZINC000147213691 EG On-Demand Anodyne GYRB 19 42 CCOC(=O)C1CCN(C(=O)/C=C/c2cc3ccccc3o2)CC1 ZINC000147213691 EG On-Demand Anodyne CCR2 46 34 COC(=O)c1cnc(Cc2ccc(OC)cc2)s1 ZINC000147213970 CF For-Sale Anodyne MAPK10 0 44 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne ACE 64 54 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne OPRM1 83 61 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne OPRD1 88 61 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne MME 156 70 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne ANPEP 96 45 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne EDNRA 17 44 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne TACR1 21 54 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne CTSD 34 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne FCER2 86 36 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne TACR2 27 49 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne RNPEP 38 47 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne KLK3 107 54 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne CTSB 83 55 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne PAPA1_CARPA 85 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne CYSP_TRYCR 78 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne CTSL 47 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne CPA1 42 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne PGA 47 42 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne NPFFR2 61 36 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne C3AR1 51 57 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne HLA-A 140 59 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne CTRB1 30 41 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne CAPNS1 74 41 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne MMP3 42 39 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne ECE1 32 45 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne HLA-DRB1 102 46 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne REN 45 42 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne REN1 54 38 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne LNPEP 27 47 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne PCSK5 46 39 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne FURIN 63 42 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne YARS 67 43 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne CAPN1 107 49 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne CASP1 38 44 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne CAPN2 134 44 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne ACE2 87 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne PLAU 39 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne BACE1 31 49 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne LAP3 56 47 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne CTSC 31 48 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne ST14 42 35 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne MMP1 35 47 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne FPR1 83 45 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne NPR 84 45 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne AMP1_PLAFQ 35 47 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne GAG-PRO 43 34 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne XIAP 31 41 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne SIRT1 39 46 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne PSMB2 36 44 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne PSMB5 45 39 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne BLA1_STEMA 73 35 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne QRFPR 57 39 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne PSMB8 59 33 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne DLG4 68 41 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne BRCA1 46 38 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne NPFFR1 69 36 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne TMPRSS6 52 39 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@H](C)O)C(=O)O ZINC000147213981 HA For-Sale Anodyne HPN 46 36 N#CC1CCN(C(=O)CSc2nnc(-c3ccc(Cl)cc3)o2)CC1 ZINC000147214025 FG On-Demand Mild ALOX15 15 43 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(C(=O)NC(C)(C)C)cc1 ZINC000147214055 EE On-Demand Anodyne MMP2 15 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(C(=O)NC(C)(C)C)cc1 ZINC000147214055 EE On-Demand Anodyne MMP3 25 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(C(=O)NC(C)(C)C)cc1 ZINC000147214055 EE On-Demand Anodyne FURIN 30 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne ACE 64 54 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne OPRM1 83 61 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne OPRD1 88 61 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne MME 156 70 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne ANPEP 96 45 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne EDNRA 17 44 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne TACR1 21 54 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne CTSD 34 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne FCER2 86 36 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne TACR2 27 49 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne RNPEP 38 47 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne KLK3 107 54 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne CTSB 83 55 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne PAPA1_CARPA 85 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne CYSP_TRYCR 78 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne CTSL 47 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne CPA1 42 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne PGA 47 42 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne NPFFR2 61 36 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne C3AR1 51 57 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne HLA-A 140 59 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne CTRB1 30 41 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne CAPNS1 74 41 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne MMP3 42 39 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne ECE1 32 45 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne HLA-DRB1 102 46 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne REN 45 42 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne REN1 54 38 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne LNPEP 27 47 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne PCSK5 46 39 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne FURIN 63 42 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne YARS 67 43 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne CAPN1 107 49 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne CASP1 38 44 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne CAPN2 134 44 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne ACE2 87 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne PLAU 39 40 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne BACE1 31 49 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne LAP3 56 47 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne CTSC 31 48 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne ST14 42 35 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne MMP1 35 47 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne FPR1 83 45 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne NPR 84 45 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne AMP1_PLAFQ 35 47 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne GAG-PRO 43 34 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne XIAP 31 41 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne SIRT1 39 46 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne PSMB2 36 44 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne PSMB5 45 39 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne BLA1_STEMA 73 35 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne QRFPR 57 39 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne PSMB8 59 33 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne DLG4 68 41 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne BRCA1 46 38 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne NPFFR1 69 36 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne TMPRSS6 52 39 C[C@H](NC(=O)[C@H](CO)NC(=O)[C@H](NC(=O)[C@H](N)Cc1ccccc1)[C@@H](C)O)C(=O)O ZINC000147214170 HA For-Sale Anodyne HPN 46 36 COC(=O)c1cnc(Cc2cccc(Cl)c2)s1 ZINC000147214203 CG For-Sale Anodyne MAOB 23 40 COC(=O)c1cnc(Cc2cccc(Cl)c2)s1 ZINC000147214203 CG For-Sale Anodyne PTGER1 31 52 COC(=O)c1cnc(Cc2cccc(Cl)c2)s1 ZINC000147214203 CG For-Sale Anodyne SCD1 25 43 COC(=O)c1cnc(Cc2cccc(Cl)c2)s1 ZINC000147214203 CG For-Sale Anodyne SCD 25 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(C(=O)NC(C)(C)C)cc1 ZINC000147214251 EE On-Demand Anodyne MMP2 15 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(C(=O)NC(C)(C)C)cc1 ZINC000147214251 EE On-Demand Anodyne MMP3 25 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(C(=O)NC(C)(C)C)cc1 ZINC000147214251 EE On-Demand Anodyne FURIN 30 40 CNc1cc(Oc2ccc(OC)cc2)cc([N+](=O)[O-])c1 ZINC000147214256 CG For-Sale Bother TAAR1 15 40 CNc1cc(Oc2ccc(OC)cc2)cc([N+](=O)[O-])c1 ZINC000147214256 CG For-Sale Bother AKR1C2 15 41 O=[N+]([O-])c1ccc(NC[C@H](O)COc2ccc(I)cc2)cc1 ZINC000147214309 HG On-Demand Bother ADRB2 44 45 O=[N+]([O-])c1ccc(NC[C@H](O)COc2ccc(I)cc2)cc1 ZINC000147214309 HG On-Demand Bother ADRB1 56 49 O=[N+]([O-])c1ccc(NC[C@H](O)COc2ccc(I)cc2)cc1 ZINC000147214309 HG On-Demand Bother ADRB3 39 44 O=C(NCC[C@H](O)CO)[C@@H]1N[C@H](CCc2cccs2)[C@]2(C(=O)Nc3cc(Cl)c(F)cc32)[C@H]1c1cccc(Cl)c1 ZINC000147214335 KI Annotated Anodyne MDM2 58 75 COC(=O)c1cnc(Cc2cccc(F)c2)s1 ZINC000147214413 CF For-Sale Anodyne SCD1 26 43 Cc1cc(Cl)ccc1O[C@@H](C)C(=O)N1CCC(C#N)CC1 ZINC000147214431 DG On-Demand Mild CCR1 41 37 CCCOc1nc(N)nc(Oc2ccc(OC)cc2)n1 ZINC000147214444 CE For-Sale Anodyne DHFR 20 40 CCCOc1nc(N)nc(Oc2ccc(OC)cc2)n1 ZINC000147214444 CE For-Sale Anodyne DRTS_PLAFK 21 40 O=[N+]([O-])c1ccc(NC[C@@H](O)COc2ccc(I)cc2)cc1 ZINC000147214483 HG On-Demand Bother ADRB2 44 45 O=[N+]([O-])c1ccc(NC[C@@H](O)COc2ccc(I)cc2)cc1 ZINC000147214483 HG On-Demand Bother ADRB1 56 49 O=[N+]([O-])c1ccc(NC[C@@H](O)COc2ccc(I)cc2)cc1 ZINC000147214483 HG On-Demand Bother ADRB3 39 44 CCOC(=O)C1CCN(C(=O)/C=C\c2cc3ccccc3o2)CC1 ZINC000147214501 EG On-Demand Anodyne GYRB 19 42 CCOC(=O)C1CCN(C(=O)/C=C\c2cc3ccccc3o2)CC1 ZINC000147214501 EG On-Demand Anodyne CCR2 46 34 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne CHRM2 25 47 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne DRD2 29 56 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne DRD4 55 40 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne ACHE 42 43 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne HRH1 19 46 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne ADRA1B 22 41 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne DRD3 37 56 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne OPRD1 18 42 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne OPRK1 26 44 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne OPRL1 36 44 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne CHRM3 31 51 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne HRH3 15 41 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne SIGMAR1 109 49 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne MMP13 19 50 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne KCNA3 26 41 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne NPFFR2 46 44 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne ADAM17 28 50 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne MMP9 16 50 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne MCHR1 27 45 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne MCHR2 57 38 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne CCR8 51 41 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne NPFFR1 71 44 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne SLC12A5 77 42 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne PA 18 43 COC(=O)C1(C)CCN(Cc2ccccc2)CC1 ZINC000147214559 BE On-Demand Anodyne NOD2 40 36 COC(=O)c1cnc(-c2ccc([N+](=O)[O-])cc2)s1 ZINC000147214617 CF For-Sale Bother CACNA1D 42 32 O=C(Nc1cccc(C(=O)N2CCCCC2)c1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147214650 GJ On-Demand Anodyne NPY2R 18 44 O=C(Nc1cccc(C(=O)N2CCCCC2)c1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147214650 GJ On-Demand Anodyne HPGD 35 44 O=C(Nc1cccc(C(=O)N2CCCCC2)c1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147214821 GJ On-Demand Anodyne NPY2R 18 44 O=C(Nc1cccc(C(=O)N2CCCCC2)c1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147214821 GJ On-Demand Anodyne HPGD 35 44 COC(=O)c1cnc(-c2ccc(F)c(Cl)c2)s1 ZINC000147214827 CG For-Sale Anodyne KMO 0 40 COc1ccc(Oc2nc(N)ncc2Br)cc1 ZINC000147214866 CF For-Sale Anodyne FOLA 42 46 COc1ccc(Oc2nc(N)ncc2Br)cc1 ZINC000147214866 CF For-Sale Anodyne DRTS_PLAFK 28 46 COc1ccc(Oc2nc(N)ncc2Br)cc1 ZINC000147214866 CF For-Sale Anodyne P2RX2 40 43 COc1ccc(Oc2nc(N)ncc2Br)cc1 ZINC000147214866 CF For-Sale Anodyne DFRA17 0 46 COc1ccc(CNCc2ccnc(-n3ccnc3)c2)cc1OCCCC#N ZINC000147214902 GG On-Demand Mild NOS2 20 41 COc1cc(CN(C)C(=O)c2cc(C)cc([N+](=O)[O-])c2)ccc1OC(F)F ZINC000147214969 GH On-Demand Bother MT-ND1 24 44 COc1cc(OC[C@@H](O)CO)cc(OC)c1OC ZINC000147214980 CC For-Sale Anodyne TUBB1 46 34 O=C(Nc1cccc(C(=O)N2CCCCC2)c1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147215022 GJ On-Demand Anodyne NPY2R 18 44 O=C(Nc1cccc(C(=O)N2CCCCC2)c1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147215022 GJ On-Demand Anodyne HPGD 35 44 CCOc1cccc(-c2ncc(C(=O)OC)s2)c1 ZINC000147215035 CF For-Sale Anodyne GYRB 0 40 CCOc1cccc(-c2ncc(C(=O)OC)s2)c1 ZINC000147215035 CF For-Sale Anodyne DHODH 37 46 CCOc1cccc(-c2ncc(C(=O)OC)s2)c1 ZINC000147215035 CF For-Sale Anodyne HSD17B2 18 47 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild SRD5A2 0 45 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild AVPR1A 25 40 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild GRIN2B 46 38 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild LTA4H 31 47 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild HRH3 25 45 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild COLA 29 40 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild CPT1A 30 40 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild GRM5 24 47 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild FAAH 15 41 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild SLC6A5 34 44 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild FAP 0 40 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild FFAR1 24 40 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild L3MBTL1 0 41 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild L3MBTL3 78 41 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild MBTD1 0 41 N#CC1CCN(C(=O)c2ccc(COc3ccccc3)cc2)CC1 ZINC000147215107 DH On-Demand Mild SLC6A7 0 54 CCOP(=O)(OCC)Oc1nn(C)c(Cl)c1Cl ZINC000147215196 DG For-Sale Anodyne MGLL 16 49 COc1ccccc1[C@H](CNC(=O)N(C)Cc1cscn1)N(C)C ZINC000147215220 EF On-Demand Anodyne BMP1 46 32 Cc1ccc([C@]23CNC[C@H]2C3)s1 ZINC000147215298 AD For-Sale Anodyne NET 0 67 CCN1CC[C@H](NS(=O)(=O)c2ccc(C)cc2)C1 ZINC000147215303 CD On-Demand Anodyne HRH2 18 55 CCN1CC[C@H](NS(=O)(=O)c2ccc(C)cc2)C1 ZINC000147215303 CD On-Demand Anodyne HTR6 15 49 CCN1CC[C@H](NS(=O)(=O)c2ccc(C)cc2)C1 ZINC000147215303 CD On-Demand Anodyne CCR8 46 36 COC(=O)[C@@H]1CC=C(c2ccccc2)CC1 ZINC000147215364 BG For-Sale Anodyne SLC6A3 18 40 COc1ccc(C)cc1-n1ccc(C(=O)N2CCN(c3cc(C#N)ccn3)CC2)n1 ZINC000147215372 HE On-Demand Mild TACR3 17 42 Nc1cc(-c2ccncc2NC(=O)c2nc(-c3c(F)cccc3F)ccc2N)ncn1 ZINC000147215387 HG Annotated Anodyne PIM1 36 46 Nc1cc(-c2ccncc2NC(=O)c2nc(-c3c(F)cccc3F)ccc2N)ncn1 ZINC000147215387 HG Annotated Anodyne PIM2 17 46 Nc1cc(-c2ccncc2NC(=O)c2nc(-c3c(F)cccc3F)ccc2N)ncn1 ZINC000147215387 HG Annotated Anodyne PIM3 24 46 Cc1cccc2sc(NC(=O)c3ccc(NC(=O)c4cccs4)cc3)nc12 ZINC000147215399 GK On-Demand Anodyne LCK 41 55 Cc1cccc2sc(NC(=O)c3ccc(NC(=O)c4cccs4)cc3)nc12 ZINC000147215399 GK On-Demand Anodyne SHH 55 38 Cc1cccc2sc(NC(=O)c3ccc(NC(=O)c4cccs4)cc3)nc12 ZINC000147215399 GK On-Demand Anodyne KCNK3 42 48 Cc1cccc2sc(NC(=O)c3ccc(NC(=O)c4cccs4)cc3)nc12 ZINC000147215399 GK On-Demand Anodyne KCNK9 30 48 COc1ccccc1[C@@H](CNC(=O)N(C)Cc1cscn1)N(C)C ZINC000147215427 EF On-Demand Anodyne BMP1 46 32 Cc1ccc([C@@]23CNC[C@H]2C3)s1 ZINC000147215491 AD For-Sale Anodyne NET 0 67 N#CC1CCN(C(=O)c2cccc(OCc3ccccc3)c2)CC1 ZINC000147215560 DH For-Sale Mild PTGER2 24 42 N#CC1CCN(C(=O)c2cccc(OCc3ccccc3)c2)CC1 ZINC000147215560 DH For-Sale Mild GRIN2B 40 37 N#CC1CCN(C(=O)c2cccc(OCc3ccccc3)c2)CC1 ZINC000147215560 DH For-Sale Mild EDNRA 0 45 N#CC1CCN(C(=O)c2cccc(OCc3ccccc3)c2)CC1 ZINC000147215560 DH For-Sale Mild GRM5 26 42 N#CC1CCN(C(=O)c2cccc(OCc3ccccc3)c2)CC1 ZINC000147215560 DH For-Sale Mild L3MBTL1 0 42 N#CC1CCN(C(=O)c2cccc(OCc3ccccc3)c2)CC1 ZINC000147215560 DH For-Sale Mild L3MBTL3 45 42 N#CC1CCN(C(=O)c2cccc(OCc3ccccc3)c2)CC1 ZINC000147215560 DH For-Sale Mild MBTD1 0 42 N#CC1CCN(C(=O)c2cccc(OCc3ccccc3)c2)CC1 ZINC000147215560 DH For-Sale Mild SLC6A7 0 47 CC(=O)N1CCN(S(=O)(=O)c2cccc(C(=O)N(C)Cc3cccc(F)c3)c2)CC1 ZINC000147215595 ID On-Demand Anodyne PKM 36 43 CC(=O)N1CCN(S(=O)(=O)c2cccc(C(=O)N(C)Cc3cccc(F)c3)c2)CC1 ZINC000147215595 ID On-Demand Anodyne TGM2 25 41 CC(=O)N1CCN(S(=O)(=O)c2cccc(C(=O)N(C)Cc3cccc(F)c3)c2)CC1 ZINC000147215595 ID On-Demand Anodyne HSD17B2 20 42 CC(=O)N1CCN(S(=O)(=O)c2cccc(C(=O)N(C)Cc3cccc(F)c3)c2)CC1 ZINC000147215595 ID On-Demand Anodyne AKR1C3 57 44 CC(=O)N1CCN(S(=O)(=O)c2cccc(C(=O)N(C)Cc3cccc(F)c3)c2)CC1 ZINC000147215595 ID On-Demand Anodyne LIMK2 23 45 CCN1C[C@]2(C)CC[C@H](O)[C@]34[C@H]1[C@](O)([C@@H](OC)[C@H]23)[C@@]1(O)C[C@H](OC)[C@H]2C[C@]4(O)[C@@H]1[C@H]2OC(=O)c1ccccc1 ZINC000147215635 KC Annotated Anodyne CHRNA4 15 41 Cc1ccc([C@]23CNC[C@@H]2C3)s1 ZINC000147215697 AD For-Sale Anodyne NET 0 67 COc1ccc(Oc2nc(N)nc(N3CCCC3)n2)cc1 ZINC000147215757 CD For-Sale Anodyne HRH4 17 40 COc1ccc(Oc2nc(N)nc(N3CCCC3)n2)cc1 ZINC000147215757 CD For-Sale Anodyne ERM 0 51 COc1ccc(Oc2nc(N)nc(N3CCCC3)n2)cc1 ZINC000147215757 CD For-Sale Anodyne GALR2 44 42 Cc1ccc([C@@]23CNC[C@@H]2C3)s1 ZINC000147215880 AD For-Sale Anodyne NET 0 67 CCN(CC)c1nc(N)nc(Oc2ccc(OC)cc2)n1 ZINC000147216035 CE For-Sale Anodyne DHFR 18 40 CCN(CC)c1nc(N)nc(Oc2ccc(OC)cc2)n1 ZINC000147216035 CE For-Sale Anodyne DRTS_TOXGO 33 40 CCN(CC)c1nc(N)nc(Oc2ccc(OC)cc2)n1 ZINC000147216035 CE For-Sale Anodyne DYR_PNECA 29 40 Cc1ccccc1C(=O)N[C@@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216227 EF On-Demand Mild P2RY12 166 36 Cc1ccccc1C(=O)N[C@@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216227 EF On-Demand Mild ANPEP 16 41 Cc1ccccc1C(=O)N[C@@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216227 EF On-Demand Mild CTSK 23 43 Cc1ccccc1C(=O)N[C@@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216227 EF On-Demand Mild CTSL 29 43 Cc1ccccc1C(=O)N[C@@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216227 EF On-Demand Mild CACNA1B 17 41 Cc1ccccc1C(=O)N[C@@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216227 EF On-Demand Mild CCR1 42 69 Cc1ccccc1C(=O)N[C@@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216227 EF On-Demand Mild CCR8 63 37 COC(=O)c1cnc(-c2ccc3nccnc3c2)s1 ZINC000147216245 CF For-Sale Anodyne TGFBR1 18 44 NC1CCC(c2nc3c(C(=O)O)cccc3[nH]2)CC1 ZINC000147216381 CE Annotated Anodyne PARP2 82 59 NC1CCC(c2nc3c(C(=O)O)cccc3[nH]2)CC1 ZINC000147216381 CE Annotated Anodyne PARP1 75 62 COc1ccc(Oc2nc(N)ncc2C)cc1 ZINC000147216419 BE For-Sale Anodyne FOLA 43 46 COc1ccc(Oc2nc(N)ncc2C)cc1 ZINC000147216419 BE For-Sale Anodyne DRTS_PLAFK 28 46 COc1ccc(Oc2nc(N)ncc2C)cc1 ZINC000147216419 BE For-Sale Anodyne P2RX2 39 43 COc1ccc(Oc2nc(N)ncc2C)cc1 ZINC000147216419 BE For-Sale Anodyne DFRA17 0 46 Cc1ccccc1C(=O)N[C@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216436 EF On-Demand Mild P2RY12 166 36 Cc1ccccc1C(=O)N[C@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216436 EF On-Demand Mild ANPEP 16 41 Cc1ccccc1C(=O)N[C@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216436 EF On-Demand Mild CTSK 23 43 Cc1ccccc1C(=O)N[C@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216436 EF On-Demand Mild CTSL 29 43 Cc1ccccc1C(=O)N[C@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216436 EF On-Demand Mild CACNA1B 17 41 Cc1ccccc1C(=O)N[C@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216436 EF On-Demand Mild CCR1 42 69 Cc1ccccc1C(=O)N[C@H](CC(C)C)C(=O)N1CCC(C#N)CC1 ZINC000147216436 EF On-Demand Mild CCR8 63 37 COC(=O)c1cnc(CSc2ccccc2Br)s1 ZINC000147216451 EH For-Sale Anodyne FAS 50 34 CCCCCCCCCCCC[S@@+](C)[C@@H](C)C(=O)O ZINC000147216502 CJ For-Sale Anodyne Q8WS26_TRYCR 20 41 CCCCCCCCCCCC[S@@+](C)[C@@H](C)C(=O)O ZINC000147216502 CJ For-Sale Anodyne NOD1 72 38 CCCCCCCCCCCC[S@@+](C)[C@@H](C)C(=O)O ZINC000147216502 CJ For-Sale Anodyne CQSS 59 39 CNCCCc1nc2cc(C(=O)OC)ccc2[nH]1 ZINC000147216591 BD For-Sale Anodyne F9 26 44 CNCCCc1nc2cc(C(=O)OC)ccc2[nH]1 ZINC000147216591 BD For-Sale Anodyne CYSP_TRYCR 15 41 CNCCCc1nc2cc(C(=O)OC)ccc2[nH]1 ZINC000147216591 BD For-Sale Anodyne CHEK2 63 39 CNCCCc1nc2cc(C(=O)OC)ccc2[nH]1 ZINC000147216591 BD For-Sale Anodyne CACNA1G 29 43 CNc1nc(Cl)nc(Oc2ccc(OC)cc2)n1 ZINC000147216604 CE For-Sale Anodyne NPBWR1 46 31 CCCCCCCCCCCC[S@+](C)[C@@H](C)C(=O)O ZINC000147216687 CJ For-Sale Anodyne Q8WS26_TRYCR 20 41 CCCCCCCCCCCC[S@+](C)[C@@H](C)C(=O)O ZINC000147216687 CJ For-Sale Anodyne NOD1 72 38 CCCCCCCCCCCC[S@+](C)[C@@H](C)C(=O)O ZINC000147216687 CJ For-Sale Anodyne CQSS 59 39 CC(C)N(Cc1ccccn1)C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147216712 EI On-Demand Anodyne MDM2 92 39 CNCc1ccc(NS(C)(=O)=O)cc1 ZINC000147216802 BC For-Sale Anodyne TRPV1 34 55 CNCc1ccc(NS(C)(=O)=O)cc1 ZINC000147216802 BC For-Sale Anodyne PTPRB 43 36 CCNc1cc(Oc2ccc(OC)cc2)cc([N+](=O)[O-])c1 ZINC000147216807 CH For-Sale Bother TBXA2R 17 42 CCNc1cc(Oc2ccc(OC)cc2)cc([N+](=O)[O-])c1 ZINC000147216807 CH For-Sale Bother ENR 0 40 CCOc1ccc(C(=O)NNC(=O)Nc2nc(C)cs2)cc1OC ZINC000147216850 FE On-Demand Reactive GCK 19 49 CCCCCCCCCCCC[S@@+](C)[C@H](C)C(=O)O ZINC000147216883 CJ For-Sale Anodyne Q8WS26_TRYCR 20 41 CCCCCCCCCCCC[S@@+](C)[C@H](C)C(=O)O ZINC000147216883 CJ For-Sale Anodyne NOD1 72 38 CCCCCCCCCCCC[S@@+](C)[C@H](C)C(=O)O ZINC000147216883 CJ For-Sale Anodyne CQSS 59 39 CC(C)N(Cc1ccccn1)C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147216887 EI On-Demand Anodyne MDM2 92 39 c1cc2c(cc1CCN1CCCC1)OCO2 ZINC000147216901 BE For-Sale Anodyne KCNH2 19 50 c1cc2c(cc1CCN1CCCC1)OCO2 ZINC000147216901 BE For-Sale Anodyne HRH3 20 53 c1cc2c(cc1CCN1CCCC1)OCO2 ZINC000147216901 BE For-Sale Anodyne SIGMAR1 40 68 c1cc2c(cc1CCN1CCCC1)OCO2 ZINC000147216901 BE For-Sale Anodyne F2R 22 46 c1cc2c(cc1CCN1CCCC1)OCO2 ZINC000147216901 BE For-Sale Anodyne NOS2 42 33 c1cc2c(cc1CCN1CCCC1)OCO2 ZINC000147216901 BE For-Sale Anodyne SSTR3 47 34 c1cc2c(cc1CCN1CCCC1)OCO2 ZINC000147216901 BE For-Sale Anodyne MCHR1 20 42 c1cc2c(cc1CCN1CCCC1)OCO2 ZINC000147216901 BE For-Sale Anodyne L3MBTL3 32 40 c1cc2c(cc1CCN1CCCC1)OCO2 ZINC000147216901 BE For-Sale Anodyne KCNJ1 61 43 CCCCCC(=O)/C=C/[C@@H]1CC1(C(=O)OCC)C(=O)OCC ZINC000147216908 DF For-Sale Mild CQSS 50 33 COC(=O)c1cnc(-c2ccc(Cl)c(F)c2)s1 ZINC000147216932 CG For-Sale Anodyne KMO 0 40 COC(=O)c1cnc(-c2ccc(Cl)c(F)c2)s1 ZINC000147216932 CG For-Sale Anodyne ENV 42 33 COC(=O)c1cnc(-c2ccc(Cl)c(F)c2)s1 ZINC000147216932 CG For-Sale Anodyne ERCC5 25 44 O=C(NCC[C@H](O)CO)[C@@H]1N[C@H](CCc2ccccc2)[C@]2(C(=O)Nc3cc(Cl)c(F)cc32)[C@H]1c1cccc(Cl)c1 ZINC000147217013 KH Annotated Anodyne MDM2 72 79 C[C@H](NC(=O)c1ccco1)C(=O)N1CCC(C#N)CC1 ZINC000147217029 CD On-Demand Mild KISS1R 45 31 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217043 GH On-Demand Anodyne CTSK 15 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217043 GH On-Demand Anodyne PCSK5 42 35 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217043 GH On-Demand Anodyne FURIN 58 35 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217043 GH On-Demand Anodyne POLG_WNV 59 32 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217043 GH On-Demand Anodyne NPFFR1 43 33 CC(C)[C@@H](C(=O)Nc1cnn(C[C@@H]2CCCO2)c1)N1C(=O)c2ccccc2C1=O ZINC000147217053 GE On-Demand Anodyne PANC 52 36 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(COCc3ccco3)c2)c1 ZINC000147217066 GI On-Demand Bother TAAR1 31 45 CCCCCCCCCCCC[S@+](C)[C@H](C)C(=O)O ZINC000147217077 CJ For-Sale Anodyne Q8WS26_TRYCR 20 41 CCCCCCCCCCCC[S@+](C)[C@H](C)C(=O)O ZINC000147217077 CJ For-Sale Anodyne NOD1 72 38 CCCCCCCCCCCC[S@+](C)[C@H](C)C(=O)O ZINC000147217077 CJ For-Sale Anodyne CQSS 59 39 CC(C)N(Cc1ccccn1)C(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147217086 EI On-Demand Anodyne MDM2 92 39 CCCCCC(=O)/C=C/[C@H]1CC1(C(=O)OCC)C(=O)OCC ZINC000147217102 DF For-Sale Mild CQSS 50 33 C[C@H](Cc1cccc(F)c1)C(=O)N(C)CCOc1ccccc1F ZINC000147217133 EH On-Demand Anodyne SLC6A9 15 44 COc1ccc(Oc2nc(N)ncc2F)cc1 ZINC000147217210 BD For-Sale Anodyne FOLA 33 45 COc1ccc(Oc2nc(N)ncc2F)cc1 ZINC000147217210 BD For-Sale Anodyne P2RX2 38 42 COc1ccc(Oc2nc(N)ncc2F)cc1 ZINC000147217210 BD For-Sale Anodyne DFRA17 0 45 C[C@@H](NC(=O)c1ccco1)C(=O)N1CCC(C#N)CC1 ZINC000147217212 CD On-Demand Mild KISS1R 45 31 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217228 GH On-Demand Anodyne CTSK 15 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217228 GH On-Demand Anodyne PCSK5 42 35 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217228 GH On-Demand Anodyne FURIN 58 35 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217228 GH On-Demand Anodyne POLG_WNV 59 32 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217228 GH On-Demand Anodyne NPFFR1 43 33 CC(C)[C@H](C(=O)Nc1cnn(C[C@@H]2CCCO2)c1)N1C(=O)c2ccccc2C1=O ZINC000147217250 GE On-Demand Anodyne PANC 52 36 CCCC[C@H](NC(N)=O)C(=O)NC[C@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217421 GH On-Demand Anodyne CTSK 15 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217421 GH On-Demand Anodyne PCSK5 42 35 CCCC[C@H](NC(N)=O)C(=O)NC[C@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217421 GH On-Demand Anodyne FURIN 58 35 CCCC[C@H](NC(N)=O)C(=O)NC[C@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217421 GH On-Demand Anodyne POLG_WNV 59 32 CCCC[C@H](NC(N)=O)C(=O)NC[C@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217421 GH On-Demand Anodyne NPFFR1 43 33 Cc1cc(C(=O)N(C)Cc2ccc(C(F)(F)F)cc2)cc([N+](=O)[O-])c1 ZINC000147217424 FI On-Demand Bother MLYCD 16 43 CC(C)[C@@H](C(=O)Nc1cnn(C[C@H]2CCCO2)c1)N1C(=O)c2ccccc2C1=O ZINC000147217471 GE On-Demand Anodyne PANC 52 36 CNC(=O)CCCNCc1ccc(OC)c(OCCCC#N)c1 ZINC000147217514 DD On-Demand Mild LPAR2 51 39 CNC(=O)CCCNCc1ccc(OC)c(OCCCC#N)c1 ZINC000147217514 DD On-Demand Mild REN 23 48 CNC(=O)CCCNCc1ccc(OC)c(OCCCC#N)c1 ZINC000147217514 DD On-Demand Mild S1PR2 54 39 CNC(=O)CCCNCc1ccc(OC)c(OCCCC#N)c1 ZINC000147217514 DD On-Demand Mild DRTS_TRYCR 40 36 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCCCC3)cc1)C2 ZINC000147217554 HH On-Demand Anodyne MTNR1A 19 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCCCC3)cc1)C2 ZINC000147217554 HH On-Demand Anodyne MTNR1B 22 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCCCC3)cc1)C2 ZINC000147217554 HH On-Demand Anodyne ROCK2 31 52 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCCCC3)cc1)C2 ZINC000147217554 HH On-Demand Anodyne EPHX2 16 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCCCC3)cc1)C2 ZINC000147217554 HH On-Demand Anodyne L3MBTL3 48 36 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne PPIA 43 33 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne MME 26 40 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne CTSB 29 42 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne PAPA1_CARPA 45 36 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne CYSP_TRYCR 42 35 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne CTSL 25 41 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne CAPNS1 48 33 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne SLC1A6 0 42 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne PAM 0 43 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne CAPN1 41 35 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne SLC1A7 0 42 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne CAPN2 71 39 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne POL 0 41 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne NPR 54 34 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne 17HSDCL 0 46 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne RHODESAIN 0 48 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne NAAA 22 42 NC(=S)CC(=O)OCc1ccccc1 ZINC000147217575 BD For-Sale Anodyne SLC12A5 59 37 COC(=O)c1cnc(-c2ccc(C3CC3)cc2)s1 ZINC000147217593 CG For-Sale Anodyne DGAT1 17 41 C/C=C\C(=O)NCCCN(C)C ZINC000147217614 AC For-Sale Anodyne DNM1 0 50 C/C=C\C(=O)NCCCN(C)C ZINC000147217614 AC For-Sale Anodyne FOXO1 0 40 O=C(O)c1ccc(NC(=O)C2[C@H]3CCCC[C@H]23)cc1 ZINC000147217636 CF On-Demand Anodyne SRD5A2 22 43 O=C(O)c1ccc(NC(=O)C2[C@H]3CCCC[C@H]23)cc1 ZINC000147217636 CF On-Demand Anodyne DHODH 45 45 O=C(O)c1ccc(NC(=O)C2[C@H]3CCCC[C@H]23)cc1 ZINC000147217636 CF On-Demand Anodyne EPHX2 27 42 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217650 GH On-Demand Anodyne CTSK 15 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217650 GH On-Demand Anodyne PCSK5 42 35 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217650 GH On-Demand Anodyne FURIN 58 35 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217650 GH On-Demand Anodyne POLG_WNV 59 32 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H]1CC2c3ccccc3C1c1ccccc12 ZINC000147217650 GH On-Demand Anodyne NPFFR1 43 33 CC(C)[C@H](C(=O)Nc1cnn(C[C@H]2CCCO2)c1)N1C(=O)c2ccccc2C1=O ZINC000147217651 GE On-Demand Anodyne PANC 52 36 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne HTR1A 35 57 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne DRD2 55 57 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne DRD1 0 41 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne DRD4 40 33 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne ADRA1D 48 38 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne HTR2A 41 43 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne HTR2C 47 44 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne SLC6A1 45 33 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne ADRA1A 53 37 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne ADRA1B 42 41 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne DRD3 72 42 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne HTR4 47 43 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne HRH3 36 44 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne CHRNA7 38 57 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne HNMT 70 39 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne HCN1 51 33 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne HCN4 48 33 Nc1ccccc1C(=O)NCCCN1CCCCCC1 ZINC000147217755 CE On-Demand Anodyne POLR1A 32 44 COC(=O)c1cnc(-c2ccc(Cl)cc2Cl)s1 ZINC000147217799 CH For-Sale Anodyne CNR1 24 41 COC(=O)c1cnc(-c2ccc(Cl)cc2Cl)s1 ZINC000147217799 CH For-Sale Anodyne AGPAT2 15 40 COC(=O)c1cnc(-c2ccc(Cl)cc2Cl)s1 ZINC000147217799 CH For-Sale Anodyne ALPL 48 50 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne ADH1A 0 49 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne IMPDH1 0 48 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne ADORA1 36 42 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne P2RY12 27 65 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne ADORA2A 22 42 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne P2RY6 47 35 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne P2RX5 0 65 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne POLB 44 35 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne P2RX3 15 65 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne AK3 0 60 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne AHCY 82 42 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne P2RX4 68 65 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne P2RX1 87 65 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne P2RX6 0 65 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne P2RY4 53 65 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne P2RY1 217 65 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne P2RY11 0 65 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne MAT1A 0 55 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne MAT2A 0 52 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne ENTPD1 0 41 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne RNASEL 0 49 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne ASNS 0 44 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne ITPR1 61 45 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne P2RY2 100 65 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne PRKACA 43 33 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne AK2 0 60 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne ADORA3 26 42 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne OXGR1 126 42 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne DTYMK 0 48 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne PARG 0 54 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne QARS 0 42 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne IMPDH2 0 48 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne GLUD1 0 49 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne AANAT 64 37 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne ABL 0 53 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne PANE 0 46 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne RNASE1 61 46 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne RNASE2 0 46 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne CYA 0 54 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne ADCY10 0 51 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne GPR17 60 49 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne MENB 0 40 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne CNGA2 0 46 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne DOT1L 61 37 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne HLCS 0 41 Nc1ncnc2c1ncn2[C@@H]1O[C@@]2(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]1[C@@H]2O ZINC000147217820 KA Annotated Anodyne BIRA 0 41 Ic1ncc(-c2cccnc2)o1 ZINC000147217823 CE For-Sale Anodyne CYP2E1 61 51 Ic1ncc(-c2cccnc2)o1 ZINC000147217823 CE For-Sale Anodyne CYP2A6 54 51 CS(=O)(=O)Nc1ccc(F)cc1C(=O)Nc1cnn(C[C@@H]2CCCO2)c1 ZINC000147217831 GD On-Demand Anodyne PANC 57 42 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild HMGCR 0 65 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild TOP1 0 88 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild CNR1 22 57 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild PPARA 0 62 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild PTGER1 0 41 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild PLA2G4C 0 49 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild FABP2 0 74 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild PLA2G2C 0 47 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild PLA2G4A 0 50 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild PLA2G2A 0 48 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild CPT1A 0 41 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild LPAR1 41 50 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild LPAR2 15 48 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild PLA2G4B 55 49 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild FAAH 29 63 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild CES2 47 42 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild CES1 34 42 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild EST1_PIG 62 42 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild PRKCA 19 48 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild EPHX2 36 74 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild CDC25C 0 57 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild PLCG1 0 44 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild CES2C 53 32 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild Q6UB75_PIG 0 46 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild CPT1 0 43 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild JHE 0 42 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild LPAR3 71 44 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild LOX1.1 20 88 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild MGLL 0 49 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild FFAR1 0 88 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild TLR2 0 74 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild ENPP2 36 44 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild SLC22A20 0 74 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild LPAR4 0 44 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild LPAR5 0 44 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild ACAT 0 50 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild Q9GPG0_MANSE 0 42 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild NOD1 50 39 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild SAE1 0 44 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild OXER1 42 58 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild CQSS 68 42 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild SLCO2A1 57 40 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild LPAR6 0 44 CCCCCCC/C=C\CCCCCC(=O)O ZINC000147217871 BJ For-Sale Mild EST1 0 47 O=C(O)c1ccc(NC(=O)C2[C@H]3CCCC[C@@H]23)cc1 ZINC000147217913 CF For-Sale Anodyne SRD5A2 22 43 O=C(O)c1ccc(NC(=O)C2[C@H]3CCCC[C@@H]23)cc1 ZINC000147217913 CF For-Sale Anodyne DHODH 45 45 CCN(CC)C(=O)N1CC(NC(=O)[C@@H]2N[C@H](CC(C)(C)C)[C@]3(C(=O)Nc4cc(Cl)ccc43)[C@H]2c2cccc(Cl)c2F)C1 ZINC000147217979 KK Annotated Anodyne MDM2 101 67 CS(=O)(=O)Nc1ccc(F)cc1C(=O)Nc1cnn(C[C@H]2CCCO2)c1 ZINC000147218008 GD On-Demand Anodyne PANC 57 42 O=C(O)c1ccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)cc1 ZINC000147218145 CF On-Demand Anodyne SRD5A2 22 43 O=C(O)c1ccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)cc1 ZINC000147218145 CF On-Demand Anodyne DHODH 45 45 O=C(O)c1ccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)cc1 ZINC000147218145 CF On-Demand Anodyne EPHX2 27 42 CC(C)CC(C)(C)C[C@H]1N[C@@H](C(=O)NCC[C@H](O)CO)[C@H](c2cccc(Cl)c2)[C@@]12C(=O)Nc1cc(Cl)c(F)cc12 ZINC000147218218 KJ Annotated Anodyne MDM2 80 86 O=C(Nc1ccccc1Br)c1ccc(CSc2ccc(Cl)cc2)cc1 ZINC000147218267 IK In-Stock Anodyne F10 28 42 O=C(Nc1ccccc1Br)c1ccc(CSc2ccc(Cl)cc2)cc1 ZINC000147218267 IK In-Stock Anodyne KCNJ11 30 40 O=C(Nc1ccccc1Br)c1ccc(CSc2ccc(Cl)cc2)cc1 ZINC000147218267 IK In-Stock Anodyne HDAC1 45 48 O=C(Nc1ccccc1Br)c1ccc(CSc2ccc(Cl)cc2)cc1 ZINC000147218267 IK In-Stock Anodyne HDAC2 28 43 O=C(Nc1ccccc1Br)c1ccc(CSc2ccc(Cl)cc2)cc1 ZINC000147218267 IK In-Stock Anodyne HAO1 15 41 Cc1ncoc1C(=O)Nc1ccc(C(=O)O)cc1 ZINC000147218370 BD On-Demand Anodyne RARA 17 41 Cc1ncoc1C(=O)Nc1ccc(C(=O)O)cc1 ZINC000147218370 BD On-Demand Anodyne TRPV1 19 42 Cc1ncoc1C(=O)Nc1ccc(C(=O)O)cc1 ZINC000147218370 BD On-Demand Anodyne PRNP 55 40 Cc1ncoc1C(=O)Nc1ccc(C(=O)O)cc1 ZINC000147218370 BD On-Demand Anodyne P4HTM 0 46 Cc1ncoc1C(=O)Nc1ccc(C(=O)O)cc1 ZINC000147218370 BD On-Demand Anodyne AKR1C3 21 41 Cc1ncoc1C(=O)Nc1ccc(C(=O)O)cc1 ZINC000147218370 BD On-Demand Anodyne SHH 42 36 Cc1ncoc1C(=O)Nc1ccc(C(=O)O)cc1 ZINC000147218370 BD On-Demand Anodyne KCNK3 67 36 Cc1cc(C(=O)N(C)CC(=O)Nc2cccc(F)c2)cc([N+](=O)[O-])c1 ZINC000147218408 EF On-Demand Bother KCNK3 41 41 Cc1cc(C(=O)N(C)CC(=O)Nc2cccc(F)c2)cc([N+](=O)[O-])c1 ZINC000147218408 EF On-Demand Bother KCNK9 32 41 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218442 EF On-Demand Mild P2RY12 105 33 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218442 EF On-Demand Mild ELANE 32 40 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218442 EF On-Demand Mild CCKAR 0 42 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218442 EF On-Demand Mild CCR1 48 66 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218442 EF On-Demand Mild CTRB1 37 44 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218442 EF On-Demand Mild CELA2A 30 44 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218442 EF On-Demand Mild CCKBR 35 42 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218442 EF On-Demand Mild ACE2 44 33 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218442 EF On-Demand Mild CTRB_BOVIN 47 34 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218442 EF On-Demand Mild FAP 0 42 CC[C@@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218442 EF On-Demand Mild F2RL1 29 43 Cn1ncc(C(=O)Oc2cccc(C(=O)NC3CC3)c2)c1C1CC1 ZINC000147218479 EE On-Demand Anodyne DRD4 42 32 Cn1ncc(C(=O)Oc2cccc(C(=O)NC3CC3)c2)c1C1CC1 ZINC000147218479 EE On-Demand Anodyne MAPK14 46 39 Cn1ncc(C(=O)Oc2cccc(C(=O)NC3CC3)c2)c1C1CC1 ZINC000147218479 EE On-Demand Anodyne MAPK13 56 35 CNc1cc(Oc2ccc(OC)cc2)ncn1 ZINC000147218554 BE For-Sale Anodyne CDKL2 39 40 O=C(O)CC1CCN(C(=O)c2cccc(F)c2Cl)CC1 ZINC000147218565 CF On-Demand Anodyne P2RX7 43 41 O=C(Cc1csc(Cc2ccc(F)cc2)n1)NC1CCN(C(=O)C2CC2)CC1 ZINC000147218572 HF On-Demand Anodyne SIGMAR1 15 44 O=C(Cc1csc(Cc2ccc(F)cc2)n1)NC1CCN(C(=O)C2CC2)CC1 ZINC000147218572 HF On-Demand Anodyne CCR3 21 40 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCCC1 ZINC000147218632 EH For-Sale Anodyne ADORA1 22 51 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCCC1 ZINC000147218632 EH For-Sale Anodyne P2RY12 83 43 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCCC1 ZINC000147218632 EH For-Sale Anodyne SOAT1 20 48 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCCC1 ZINC000147218632 EH For-Sale Anodyne NPY5R 23 45 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCCC1 ZINC000147218632 EH For-Sale Anodyne ADORA3 34 51 CCOC(=O)c1c(C)nc(-c2ccccc2)nc1N1CCCCC1 ZINC000147218632 EH For-Sale Anodyne DGAT1 29 48 Cc1ccc(NS(C)(=O)=O)c(C(=O)Nc2cnn(C[C@@H]3CCCO3)c2)c1 ZINC000147218667 GD On-Demand Anodyne PANC 54 37 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218682 EF On-Demand Mild P2RY12 105 33 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218682 EF On-Demand Mild ELANE 32 40 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218682 EF On-Demand Mild CCKAR 0 42 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218682 EF On-Demand Mild CCR1 48 66 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218682 EF On-Demand Mild CTRB1 37 44 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218682 EF On-Demand Mild CELA2A 30 44 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218682 EF On-Demand Mild CCKBR 35 42 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218682 EF On-Demand Mild ACE2 44 33 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218682 EF On-Demand Mild CTRB_BOVIN 47 34 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218682 EF On-Demand Mild FAP 0 42 CC[C@H](C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218682 EF On-Demand Mild F2RL1 29 43 CNC(=O)c1ccc(C)c(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147218694 EC On-Demand Anodyne MAPK14 42 40 COC(=O)c1cnc(-c2ccc(OC)c(F)c2)s1 ZINC000147218702 CF For-Sale Anodyne MET 28 41 COC(=O)c1cnc(-c2ccc(OC)c(F)c2)s1 ZINC000147218702 CF For-Sale Anodyne CSF1R 21 43 O=C(O)CC1CCN(C(=O)[C@H]2C[C@H]2c2ccccc2)CC1 ZINC000147218793 CF For-Sale Anodyne ERBB2 28 40 O=C(O)CC1CCN(C(=O)[C@H]2C[C@H]2c2ccccc2)CC1 ZINC000147218793 CF For-Sale Anodyne PREP 35 51 O=C(O)CC1CCN(C(=O)[C@H]2C[C@H]2c2ccccc2)CC1 ZINC000147218793 CF For-Sale Anodyne MMP2 0 40 O=C(O)CC1CCN(C(=O)[C@H]2C[C@H]2c2ccccc2)CC1 ZINC000147218793 CF For-Sale Anodyne ADAM10 37 40 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(C(=O)C2CC2)CC1 ZINC000147218832 DC On-Demand Anodyne EPHX2 20 40 CCOC(=O)c1cnc(-c2cccnc2)nc1N1CCCC1 ZINC000147218844 CE For-Sale Anodyne P2RY12 54 36 CCOC(=O)c1cnc(-c2cccnc2)nc1N1CCCC1 ZINC000147218844 CE For-Sale Anodyne JUN 17 43 CCOC(=O)c1cnc(-c2cccnc2)nc1N1CCCC1 ZINC000147218844 CE For-Sale Anodyne PDE4B 15 43 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218854 EF On-Demand Mild P2RY12 105 33 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218854 EF On-Demand Mild ELANE 32 40 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218854 EF On-Demand Mild CCKAR 0 42 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218854 EF On-Demand Mild CCR1 48 66 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218854 EF On-Demand Mild CTRB1 37 44 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218854 EF On-Demand Mild CELA2A 30 44 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218854 EF On-Demand Mild CCKBR 35 42 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218854 EF On-Demand Mild ACE2 44 33 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218854 EF On-Demand Mild CTRB_BOVIN 47 34 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218854 EF On-Demand Mild FAP 0 42 CC[C@@H](C)[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147218854 EF On-Demand Mild F2RL1 29 43 Cc1ccc(NS(C)(=O)=O)c(C(=O)Nc2cnn(C[C@H]3CCCO3)c2)c1 ZINC000147218875 GD On-Demand Anodyne PANC 54 37 CCc1ncc(C(=O)N(C)CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)s1 ZINC000147218891 HI On-Demand Anodyne RAF1 31 42 CCc1ncc(C(=O)N(C)CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)s1 ZINC000147218891 HI On-Demand Anodyne Q8MMZ8_EIMTE 48 44 CCc1ncc(C(=O)N(C)CC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)s1 ZINC000147218891 HI On-Demand Anodyne IMDH_CRYPV 18 42 CNC(=O)c1ccc(C)c(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147218893 EC On-Demand Anodyne MAPK14 42 40 COC(=O)c1cnc(-c2ccc3c(c2)CCN3C)s1 ZINC000147218921 CF For-Sale Anodyne CYP11B2 25 40 COC(=O)c1cnc(-c2ccc3c(c2)CCN3C)s1 ZINC000147218921 CF For-Sale Anodyne EIF2AK3 64 34 CN1CC[C@]23CC(=O)CC[C@@]2(O)[C@H]1Cc1ccc(C(=O)NCCc2ccc(-c4ccnc(O)c4)cc2)c(O)c13 ZINC000147218930 KG Annotated Anodyne OPRM1 34 53 CN1CC[C@]23CC(=O)CC[C@@]2(O)[C@H]1Cc1ccc(C(=O)NCCc2ccc(-c4ccnc(O)c4)cc2)c(O)c13 ZINC000147218930 KG Annotated Anodyne OPRD1 36 48 CN1CC[C@]23CC(=O)CC[C@@]2(O)[C@H]1Cc1ccc(C(=O)NCCc2ccc(-c4ccnc(O)c4)cc2)c(O)c13 ZINC000147218930 KG Annotated Anodyne OPRK1 32 53 O=C(O)CC1CCN(C(=O)[C@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147218996 CF For-Sale Anodyne ERBB2 28 40 O=C(O)CC1CCN(C(=O)[C@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147218996 CF For-Sale Anodyne PREP 35 51 O=C(O)CC1CCN(C(=O)[C@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147218996 CF For-Sale Anodyne MMP2 0 40 O=C(O)CC1CCN(C(=O)[C@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147218996 CF For-Sale Anodyne ADAM10 37 40 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(C(=O)C2CC2)CC1 ZINC000147219095 DC On-Demand Anodyne EPHX2 20 40 O=C(O)CC1CCN(C(=O)[C@@H]2C[C@H]2c2ccccc2)CC1 ZINC000147219197 CF For-Sale Anodyne ERBB2 28 40 O=C(O)CC1CCN(C(=O)[C@@H]2C[C@H]2c2ccccc2)CC1 ZINC000147219197 CF For-Sale Anodyne PREP 35 51 O=C(O)CC1CCN(C(=O)[C@@H]2C[C@H]2c2ccccc2)CC1 ZINC000147219197 CF For-Sale Anodyne MMP2 0 40 O=C(O)CC1CCN(C(=O)[C@@H]2C[C@H]2c2ccccc2)CC1 ZINC000147219197 CF For-Sale Anodyne ADAM10 37 40 COc1ccc(Br)c(CNCc2ccc(OC)c(OCCCC#N)c2)c1 ZINC000147219248 HI On-Demand Mild MT-ND1 23 41 CS(=O)(=O)c1ccc(N2CC[C@H](Br)C2)c(S(C)(=O)=O)c1 ZINC000147219295 GD For-Sale Reactive SLC6A9 29 40 CS(=O)(=O)c1ccc(N2CC[C@H](Br)C2)c(S(C)(=O)=O)c1 ZINC000147219295 GD For-Sale Reactive GPR119 44 41 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne ACE 49 40 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne OPRM1 24 40 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne OPRD1 23 40 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne CACNA2D1 17 43 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne MME 116 48 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne LTA4H 25 49 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne ANPEP 103 44 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne RNPEP 35 41 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne PAPA1_CARPA 42 37 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne CTSL 34 43 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne CPA1 58 36 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne SLC15A1 0 48 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne CTRB1 34 54 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne CA5B 32 40 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne CA5A 37 40 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne CAPNS1 58 35 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne MMP2 21 44 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne MMP3 29 41 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne LNPEP 17 41 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne PAM 0 41 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne FURIN 52 38 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne DNPEP 0 43 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne CAPN1 73 45 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne MMP9 18 44 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne CAPN2 76 35 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne ACE2 56 36 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne LAP3 66 43 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne CDK5 15 42 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne MMP1 23 44 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne FPR1 40 38 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne POL 0 44 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne NPR 94 39 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne AMP1_PLAFQ 64 41 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne AMPX_VIBPR 0 41 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne SLC15A2 0 45 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne BIRC2 19 40 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne CARM1 46 35 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne METAP2 0 40 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne BLAIMP-1 0 43 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne VM1B1_BOTAS 0 40 C[C@H](N)C(=O)NC(=O)Cc1ccccc1 ZINC000147219322 BC For-Sale Anodyne H9B8T9_CAPHI 15 53 N#CC1CCN(C(=O)[C@@H]2CC(=O)N(Cc3ccccc3)C2)CC1 ZINC000147219337 DD On-Demand Mild SAP2 36 46 COc1ccc(CNCC(=O)N2CCN(C)CC2)cc1OCCCC#N ZINC000147219366 FD On-Demand Mild REN 21 40 COc1ccc(CNCC(=O)N2CCN(C)CC2)cc1OCCCC#N ZINC000147219366 FD On-Demand Mild DRTS_TRYCR 40 35 CNS(=O)(=O)c1cc(NS(=O)(=O)c2ccc3[nH]c(=O)[nH]c3c2)ccc1C ZINC000147219372 GC On-Demand Anodyne PKM 43 41 O=C(O)CC1CCN(C(=O)[C@@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147219416 CF For-Sale Anodyne ERBB2 28 40 O=C(O)CC1CCN(C(=O)[C@@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147219416 CF For-Sale Anodyne PREP 35 51 O=C(O)CC1CCN(C(=O)[C@@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147219416 CF For-Sale Anodyne MMP2 0 40 O=C(O)CC1CCN(C(=O)[C@@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147219416 CF For-Sale Anodyne ADAM10 37 40 O=C(O[C@@H]1CCCNC1)c1ccc(-c2ccccc2)cc1 ZINC000147219470 CG For-Sale Anodyne GLRA1 66 33 O=C(O[C@@H]1CCCNC1)c1ccc(-c2ccccc2)cc1 ZINC000147219470 CG For-Sale Anodyne ACHP_LYMST 18 47 O=C(O[C@@H]1CCCNC1)c1ccc(-c2ccccc2)cc1 ZINC000147219470 CG For-Sale Anodyne Q8WSF8_APLCA 47 37 O=C(Nc1cnn(C[C@@H]2CCCO2)c1)c1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147219490 HE On-Demand Anodyne CCR8 47 32 O=C(Nc1cnn(C[C@@H]2CCCO2)c1)c1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147219490 HE On-Demand Anodyne PANC 56 39 CS(=O)(=O)c1ccc(N2CC[C@@H](Br)C2)c(S(C)(=O)=O)c1 ZINC000147219515 GD For-Sale Reactive SLC6A9 29 40 CS(=O)(=O)c1ccc(N2CC[C@@H](Br)C2)c(S(C)(=O)=O)c1 ZINC000147219515 GD For-Sale Reactive GPR119 44 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219523 EG On-Demand Anodyne KCNQ2 110 58 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219523 EG On-Demand Anodyne KLK3 46 37 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219523 EG On-Demand Anodyne NPFFR2 48 31 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219523 EG On-Demand Anodyne CSF1R 23 44 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219523 EG On-Demand Anodyne POLG_WNV 58 30 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219523 EG On-Demand Anodyne NPFFR1 41 31 N#CC1CCN(C(=O)[C@H]2CC(=O)N(Cc3ccccc3)C2)CC1 ZINC000147219531 DD On-Demand Mild SAP2 36 46 Cc1ccc(C(=O)N2CCC(CC(=O)O)CC2)cc1Br ZINC000147219638 EG On-Demand Anodyne L3MBTL1 0 46 Cc1ccc(C(=O)N2CCC(CC(=O)O)CC2)cc1Br ZINC000147219638 EG On-Demand Anodyne L3MBTL3 73 40 Cc1ccc(C(=O)N2CCC(CC(=O)O)CC2)cc1Br ZINC000147219638 EG On-Demand Anodyne MBTD1 0 46 O=C(O[C@H]1CCCNC1)c1ccc(-c2ccccc2)cc1 ZINC000147219649 CG For-Sale Anodyne GLRA1 66 33 O=C(O[C@H]1CCCNC1)c1ccc(-c2ccccc2)cc1 ZINC000147219649 CG For-Sale Anodyne ACHP_LYMST 18 47 O=C(O[C@H]1CCCNC1)c1ccc(-c2ccccc2)cc1 ZINC000147219649 CG For-Sale Anodyne Q8WSF8_APLCA 47 37 O=C(Nc1cnn(C[C@H]2CCCO2)c1)c1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147219671 HE On-Demand Anodyne CCR8 47 32 O=C(Nc1cnn(C[C@H]2CCCO2)c1)c1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147219671 HE On-Demand Anodyne PANC 56 39 CN(C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc(F)cc1 ZINC000147219681 DI On-Demand Anodyne MDM2 43 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219713 EG On-Demand Anodyne KCNQ2 110 58 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219713 EG On-Demand Anodyne KLK3 46 37 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219713 EG On-Demand Anodyne NPFFR2 48 31 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219713 EG On-Demand Anodyne CSF1R 23 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219713 EG On-Demand Anodyne POLG_WNV 58 30 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147219713 EG On-Demand Anodyne NPFFR1 41 31 CCOC(=O)c1cnc(-c2ccc(CC)cc2)nc1N(C)C ZINC000147219732 CF For-Sale Anodyne JUN 19 45 CCOc1ccc(C(=O)NNC(=O)Nc2nc(C)c(C)s2)cc1OC ZINC000147219855 FF On-Demand Reactive ADORA2B 22 40 CN(C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc(F)cc1 ZINC000147219880 DI On-Demand Anodyne MDM2 43 33 COC(=O)c1cnc(-c2ccnc3ccccc23)s1 ZINC000147219988 CG For-Sale Anodyne GABRA1 27 42 COC(=O)c1cnc(-c2ccnc3ccccc23)s1 ZINC000147219988 CG For-Sale Anodyne TGFBR1 25 41 CN(C(=O)[C@H]1C[C@H]1c1cccc(Cl)c1)c1ccc(F)cc1 ZINC000147220076 DI On-Demand Anodyne MDM2 43 33 COc1ccc(Oc2nc(N)ncc2Cl)cc1 ZINC000147220177 CF For-Sale Anodyne FOLA 35 45 COc1ccc(Oc2nc(N)ncc2Cl)cc1 ZINC000147220177 CF For-Sale Anodyne DRTS_PLAFK 31 45 COc1ccc(Oc2nc(N)ncc2Cl)cc1 ZINC000147220177 CF For-Sale Anodyne P2RX2 48 45 COc1ccc(Oc2nc(N)ncc2Cl)cc1 ZINC000147220177 CF For-Sale Anodyne DFRA17 0 45 COc1ccc(Oc2nc(N)ncc2Cl)cc1 ZINC000147220177 CF For-Sale Anodyne NPBWR1 86 36 COc1ccc2c(c1)OC[C@H](C(=O)N(C)c1ccc(F)cc1)C2 ZINC000147220201 DG On-Demand Anodyne ROCK2 25 40 O=c1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147220458 JA Annotated Anodyne POLA1 44 42 O=c1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147220458 JA Annotated Anodyne P2RY6 163 62 O=c1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147220458 JA Annotated Anodyne POLB 54 37 O=c1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147220458 JA Annotated Anodyne P2RX1 51 32 O=c1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147220458 JA Annotated Anodyne P2RY4 163 62 O=c1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147220458 JA Annotated Anodyne P2RY2 187 62 O=c1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147220458 JA Annotated Anodyne P2RY14 96 59 O=c1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147220458 JA Annotated Anodyne RNASE1 49 40 O=c1ccn([C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147220458 JA Annotated Anodyne GPR17 41 32 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild MAOB 28 46 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild AVPR1A 25 42 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild GRIN2B 53 40 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild LTA4H 39 50 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild HRH3 29 45 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild CHEK2 17 41 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild ADAM17 32 43 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild SLC18A3 18 41 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild PREP 31 40 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild SLC6A5 34 43 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild EPHX2 15 40 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild FFAR1 29 42 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild CCR8 23 40 N#CC1CCN(C(=O)c2ccc(OCc3ccccc3)cc2)CC1 ZINC000147220481 DH On-Demand Mild L3MBTL3 78 39 NS(=O)(=O)c1cc(Br)ccc1OCCc1cccnc1 ZINC000147220560 FE For-Sale Anodyne CA14 0 41 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147220580 HD On-Demand Anodyne DRD4 30 47 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147220580 HD On-Demand Anodyne TGM2 21 42 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147220580 HD On-Demand Anodyne F13A1 34 42 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147220580 HD On-Demand Anodyne IDO1 28 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)NC(C)C)cc1)C2 ZINC000147220753 FG On-Demand Anodyne MTNR1A 20 43 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)NC(C)C)cc1)C2 ZINC000147220753 FG On-Demand Anodyne MTNR1B 21 43 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)NC(C)C)cc1)C2 ZINC000147220753 FG On-Demand Anodyne ROCK2 32 54 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147220767 HD On-Demand Anodyne DRD4 30 47 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147220767 HD On-Demand Anodyne TGM2 21 42 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147220767 HD On-Demand Anodyne F13A1 34 42 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H]2CN(Cc3ccccc3)CCO2)cc1 ZINC000147220767 HD On-Demand Anodyne IDO1 28 41 Cc1cc(NC(=O)[C@@H]2C[C@@H]2c2ccccc2)sc1C(=O)O ZINC000147221017 DG For-Sale Anodyne ITK 0 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(-n2cccn2)cc1C(F)(F)F ZINC000147221078 GF On-Demand Anodyne AMP1_PLAFQ 43 31 COC(=O)[C@H]1Cc2c([nH]c3ccccc23)[C@@H](c2ccc(Cl)nc2)N1 ZINC000147221153 EF For-Sale Anodyne PDE5A 38 40 COC(=O)[C@H]1Cc2c([nH]c3ccccc23)[C@@H](c2ccc(Cl)nc2)N1 ZINC000147221153 EF For-Sale Anodyne PDE11A 48 32 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@H]3C)cc1)C2 ZINC000147221184 HH On-Demand Anodyne MTNR1A 17 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@H]3C)cc1)C2 ZINC000147221184 HH On-Demand Anodyne MTNR1B 19 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@H]3C)cc1)C2 ZINC000147221184 HH On-Demand Anodyne ROCK2 26 49 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@H]3C)cc1)C2 ZINC000147221184 HH On-Demand Anodyne CFTR 42 39 Cc1cc(NC(=O)[C@H]2C[C@@H]2c2ccccc2)sc1C(=O)O ZINC000147221220 DG For-Sale Anodyne ITK 0 42 N#Cc1ccc(COc2ccc(Br)cc2S(N)(=O)=O)cc1 ZINC000147221235 FF For-Sale Mild CYP19A1 16 42 N#Cc1ccc(COc2ccc(Br)cc2S(N)(=O)=O)cc1 ZINC000147221235 FF For-Sale Mild CCR5 22 52 COc1ccccc1[C@H](C)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147221262 DG On-Demand Bother KCNMA1 19 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(-n2cccn2)cc1C(F)(F)F ZINC000147221278 GF On-Demand Anodyne AMP1_PLAFQ 43 31 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147221311 HJ On-Demand Anodyne MAPK11 36 43 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147221311 HJ On-Demand Anodyne MAPK14 35 43 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147221311 HJ On-Demand Anodyne KCNK3 79 37 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147221311 HJ On-Demand Anodyne KCNK9 41 37 Cc1cc(Cl)ccc1NC(=S)Nc1cccc2ccccc12 ZINC000147221362 EK For-Sale Anodyne TRPV1 15 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@@H]3C)cc1)C2 ZINC000147221377 HH On-Demand Anodyne MTNR1A 17 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@@H]3C)cc1)C2 ZINC000147221377 HH On-Demand Anodyne MTNR1B 19 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@@H]3C)cc1)C2 ZINC000147221377 HH On-Demand Anodyne ROCK2 26 49 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@@H]3C)cc1)C2 ZINC000147221377 HH On-Demand Anodyne CFTR 42 39 Cc1cc(NC(=O)[C@@H]2C[C@H]2c2ccccc2)sc1C(=O)O ZINC000147221418 DG For-Sale Anodyne ITK 0 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)CC(C)C)cc1 ZINC000147221453 EF On-Demand Anodyne MMP2 16 44 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)CC(C)C)cc1 ZINC000147221453 EF On-Demand Anodyne MMP3 38 45 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)CC(C)C)cc1 ZINC000147221453 EF On-Demand Anodyne FURIN 30 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)CC(C)C)cc1 ZINC000147221453 EF On-Demand Anodyne NOD1 50 34 COc1ccccc1[C@@H](C)NC(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147221454 DG On-Demand Bother KCNMA1 19 40 COC(=O)c1cnc(-c2cccc(Cl)c2Cl)s1 ZINC000147221504 CH For-Sale Anodyne TYK2 27 40 COC(=O)c1cnc(-c2cccc(Cl)c2Cl)s1 ZINC000147221504 CH For-Sale Anodyne CSF1R 15 40 CCNc1cn2ccnc2c(Oc2ccc(OC)cc2)n1 ZINC000147221539 CF For-Sale Anodyne HIVRT 0 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@@H]3C)cc1)C2 ZINC000147221598 HH On-Demand Anodyne MTNR1A 17 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@@H]3C)cc1)C2 ZINC000147221598 HH On-Demand Anodyne MTNR1B 19 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@@H]3C)cc1)C2 ZINC000147221598 HH On-Demand Anodyne ROCK2 26 49 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCCC[C@@H]3C)cc1)C2 ZINC000147221598 HH On-Demand Anodyne CFTR 42 39 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne POLA1 43 37 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne P2RY12 0 44 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne P2RY6 107 40 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne HPRT1 60 40 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne P2RX5 0 44 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne POLB 62 54 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne AK3 0 40 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne PNP 30 51 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne P2RX4 50 44 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne P2RX1 70 45 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne P2RX6 0 44 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne P2RY4 103 51 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne P2RY1 184 46 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne P2RY11 0 44 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne P2RY2 128 51 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne AK2 0 40 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne DTYMK 0 40 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne FUT6 0 44 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne IMPDH2 0 44 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne EIF4E 0 54 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne URA3 0 41 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne RNASE1 49 38 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne CYA 0 40 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne RAC1 0 65 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne GPR17 65 44 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne Q3ZDS5_9HEPC 0 59 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne CNGA2 0 49 Nc1nc2c(ncn2[C@@H]2O[C@@]3(CO[P@](=O)(O)O[P@](=O)(O)OP(=O)(O)O)CO[C@@H]2[C@@H]3O)c(=O)[nH]1 ZINC000147221601 KA Annotated Anodyne ROCR 0 49 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)CC(C)C)cc1 ZINC000147221631 EF On-Demand Anodyne MMP2 16 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)CC(C)C)cc1 ZINC000147221631 EF On-Demand Anodyne MMP3 38 45 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)CC(C)C)cc1 ZINC000147221631 EF On-Demand Anodyne FURIN 30 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)CC(C)C)cc1 ZINC000147221631 EF On-Demand Anodyne NOD1 50 34 Cc1cc(NC(=O)[C@H]2C[C@H]2c2ccccc2)sc1C(=O)O ZINC000147221641 DG For-Sale Anodyne ITK 0 42 CCCCCCCCCCCCOC(=O)C(Br)(Br)Br ZINC000147221666 JK For-Sale Mild AMY2 44 31 CCCCCCCCCCCCOC(=O)C(Br)(Br)Br ZINC000147221666 JK For-Sale Mild PLA2G4B 85 39 CCCCCCCCCCCCOC(=O)C(Br)(Br)Br ZINC000147221666 JK For-Sale Mild CES2 51 44 CCCCCCCCCCCCOC(=O)C(Br)(Br)Br ZINC000147221666 JK For-Sale Mild EST1_PIG 68 44 CCCCCCCCCCCCOC(=O)C(Br)(Br)Br ZINC000147221666 JK For-Sale Mild GBA2 28 40 CCCCCCCCCCCCOC(=O)C(Br)(Br)Br ZINC000147221666 JK For-Sale Mild CES2C 61 44 CCCCCCCCCCCCOC(=O)C(Br)(Br)Br ZINC000147221666 JK For-Sale Mild LPAR3 29 41 CCCCCCCCCCCCOC(=O)C(Br)(Br)Br ZINC000147221666 JK For-Sale Mild CQSS 54 34 COC(=O)c1cnc(-c2c(Cl)cccc2Cl)s1 ZINC000147221749 CH For-Sale Anodyne LCK 15 41 COC(=O)c1cnc(-c2c(Cl)cccc2Cl)s1 ZINC000147221749 CH For-Sale Anodyne TYK2 33 40 CNc1cncc(Oc2ccc3c(C)cc(=O)oc3c2)n1 ZINC000147221759 CF For-Sale Anodyne MAOA 61 46 CNc1cncc(Oc2ccc3c(C)cc(=O)oc3c2)n1 ZINC000147221759 CF For-Sale Anodyne MAOB 37 48 CC(C)NC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147221802 FI On-Demand Anodyne PRNP 16 43 CC(C)NC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147221802 FI On-Demand Anodyne MDM2 52 36 CC(C)NC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147221802 FI On-Demand Anodyne NAMPT 23 41 COc1cccc(O)c1CC(C)=O ZINC000147221809 AD For-Sale Anodyne ESR2 0 41 COc1cccc(O)c1CC(C)=O ZINC000147221809 AD For-Sale Anodyne CA14 0 48 Cc1ccc(C(=O)Nc2cc(C)c(C(=O)O)s2)cc1Br ZINC000147221841 FI For-Sale Anodyne GPR35 43 37 COc1ccc(CN[C@@H](C)C(=O)NC(C)(C)C)cc1OCCCC#N ZINC000147221887 EF On-Demand Mild DRTS_TRYCR 40 36 Cc1cc(=O)oc2cc(Oc3cc(N)ncn3)ccc12 ZINC000147221966 CE For-Sale Anodyne MAOA 66 50 Cc1cc(=O)oc2cc(Oc3cc(N)ncn3)ccc12 ZINC000147221966 CE For-Sale Anodyne MAOB 46 50 C[C@H]1C[C@@H](C)CN(S(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)C1 ZINC000147221968 GF On-Demand Mild CNR1 0 45 C[C@H]1C[C@@H](C)CN(S(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)C1 ZINC000147221968 GF On-Demand Mild L3MBTL1 0 50 C[C@H]1C[C@@H](C)CN(S(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)C1 ZINC000147221968 GF On-Demand Mild L3MBTL3 61 50 C[C@H]1C[C@@H](C)CN(S(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)C1 ZINC000147221968 GF On-Demand Mild MBTD1 0 50 C[C@@H](OC[C@@H]1CCCO1)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147221975 EF On-Demand Anodyne MTNR1B 25 40 CC(C)NC(=O)c1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147221998 FI On-Demand Anodyne PRNP 16 43 CC(C)NC(=O)c1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147221998 FI On-Demand Anodyne MDM2 52 36 CC(C)NC(=O)c1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147221998 FI On-Demand Anodyne NAMPT 23 41 CN(C)C(=O)NCCNc1nc2cc([N+](=O)[O-])ccc2[nH]1 ZINC000147222091 CD On-Demand Bother GYRB 47 42 C[C@@H]1C[C@@H](C)CN(S(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)C1 ZINC000147222133 GF On-Demand Mild CNR1 0 45 C[C@@H]1C[C@@H](C)CN(S(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)C1 ZINC000147222133 GF On-Demand Mild L3MBTL1 0 50 C[C@@H]1C[C@@H](C)CN(S(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)C1 ZINC000147222133 GF On-Demand Mild L3MBTL3 61 50 C[C@@H]1C[C@@H](C)CN(S(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)C1 ZINC000147222133 GF On-Demand Mild MBTD1 0 50 C[C@H](OC[C@H]1CCCO1)C(=O)NCCOc1ccc2ccccc2c1 ZINC000147222145 EF On-Demand Anodyne MTNR1B 25 40 CCOC(=O)c1cnc(-c2ccccc2Cl)nc1N1CCCC1 ZINC000147222171 EH For-Sale Anodyne P2RY12 68 45 CCOC(=O)c1cnc(-c2ccccc2Cl)nc1N1CCCC1 ZINC000147222171 EH For-Sale Anodyne JUN 17 40 CCOC(=O)c1cnc(-c2ccccc2Cl)nc1N1CCCC1 ZINC000147222171 EH For-Sale Anodyne PDE2A 37 46 Cc1cc(=O)oc2cc(Oc3cc(N)nc(N)n3)ccc12 ZINC000147222192 CD For-Sale Anodyne MAOA 63 47 Cc1cc(=O)oc2cc(Oc3cc(N)nc(N)n3)ccc12 ZINC000147222192 CD For-Sale Anodyne MAOB 43 47 CC(C)NC(=O)c1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147222240 FI On-Demand Anodyne PRNP 16 43 CC(C)NC(=O)c1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147222240 FI On-Demand Anodyne MDM2 52 36 CC(C)NC(=O)c1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147222240 FI On-Demand Anodyne NAMPT 23 41 CC(C)Oc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147222305 FF On-Demand Anodyne ENV 40 33 N#CC1CCN(C(=O)C[C@@H](NC(=O)c2ccccc2Cl)c2ccccc2)CC1 ZINC000147222411 GH On-Demand Mild PTAFR 32 44 Cc1cc(=O)oc2cc(Oc3ccnc(N)n3)ccc12 ZINC000147222423 CE For-Sale Anodyne MAOA 65 49 Cc1cc(=O)oc2cc(Oc3ccnc(N)n3)ccc12 ZINC000147222423 CE For-Sale Anodyne MAOB 46 49 CC(C)Oc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147222493 FF On-Demand Anodyne ENV 40 33 CN(C)C(=O)NCCNc1ccc([N+](=O)[O-])cc1[N+](=O)[O-] ZINC000147222511 CD On-Demand Bother BDKRB1 21 40 C[C@H](NC(=O)c1cccc(OC(F)F)c1)c1cccc(C(F)(F)F)c1 ZINC000147222517 FJ On-Demand Anodyne PTGER4 17 41 C[C@H](NC(=O)c1cccc(OC(F)F)c1)c1cccc(C(F)(F)F)c1 ZINC000147222517 FJ On-Demand Anodyne CCR2 48 38 C[C@H](NC(=O)c1cccc(OC(F)F)c1)c1cccc(C(F)(F)F)c1 ZINC000147222517 FJ On-Demand Anodyne KCNK3 26 41 C[C@H](NC(=O)c1cccc(OC(F)F)c1)c1cccc(C(F)(F)F)c1 ZINC000147222517 FJ On-Demand Anodyne PDS 44 37 N#CC1CCN(C(=O)C[C@H](NC(=O)c2ccccc2Cl)c2ccccc2)CC1 ZINC000147222596 GH On-Demand Mild PTAFR 32 44 Cc1c(N)ncnc1Oc1ccc2c(C)cc(=O)oc2c1 ZINC000147222619 CF For-Sale Anodyne MAOA 65 49 Cc1c(N)ncnc1Oc1ccc2c(C)cc(=O)oc2c1 ZINC000147222619 CF For-Sale Anodyne MAOB 50 49 CCOC(=O)c1cnc(-c2ccccn2)nc1N1CCCC1 ZINC000147222630 CE For-Sale Anodyne ADORA1 17 46 CCOC(=O)c1cnc(-c2ccccn2)nc1N1CCCC1 ZINC000147222630 CE For-Sale Anodyne P2RY12 61 39 CCOC(=O)c1cnc(-c2ccccn2)nc1N1CCCC1 ZINC000147222630 CE For-Sale Anodyne JUN 17 40 CCOC(=O)c1cnc(-c2ccccn2)nc1N1CCCC1 ZINC000147222630 CE For-Sale Anodyne METAP1 37 47 CCOC(=O)c1cnc(-c2ccccn2)nc1N1CCCC1 ZINC000147222630 CE For-Sale Anodyne ADORA3 15 47 C[C@@H](NC(=O)c1cccc(OC(F)F)c1)c1cccc(C(F)(F)F)c1 ZINC000147222729 FJ On-Demand Anodyne PTGER4 17 41 C[C@@H](NC(=O)c1cccc(OC(F)F)c1)c1cccc(C(F)(F)F)c1 ZINC000147222729 FJ On-Demand Anodyne CCR2 48 38 C[C@@H](NC(=O)c1cccc(OC(F)F)c1)c1cccc(C(F)(F)F)c1 ZINC000147222729 FJ On-Demand Anodyne KCNK3 26 41 C[C@@H](NC(=O)c1cccc(OC(F)F)c1)c1cccc(C(F)(F)F)c1 ZINC000147222729 FJ On-Demand Anodyne PDS 44 37 COc1cc(C(=O)N2CCC(C#N)CC2)ccc1OCc1ccccc1Cl ZINC000147222784 GI On-Demand Mild HRH3 26 40 COc1cc(C(=O)N2CCC(C#N)CC2)ccc1OCc1ccccc1Cl ZINC000147222784 GI On-Demand Mild CCR8 21 40 COc1cc(C(=O)N2CCC(C#N)CC2)ccc1OCc1ccccc1Cl ZINC000147222784 GI On-Demand Mild L3MBTL3 57 37 Cc1cc(=O)oc2cc(Oc3nc(N)nc(Cl)n3)ccc12 ZINC000147222836 DE For-Sale Anodyne MAOA 62 46 Cc1cc(=O)oc2cc(Oc3nc(N)nc(Cl)n3)ccc12 ZINC000147222836 DE For-Sale Anodyne MAOB 30 46 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](c2ccccc2)C2CCCC2)c1 ZINC000147222856 FI On-Demand Bother TAAR1 21 40 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](c2ccccc2)C2CCCC2)c1 ZINC000147222856 FI On-Demand Bother AKR1C2 33 44 O=C(c1ccccc1)N(CCc1ccccc1)Cc1ccccc1 ZINC000147222940 DJ On-Demand Anodyne OPRD1 16 45 O=C(c1ccccc1)N(CCc1ccccc1)Cc1ccccc1 ZINC000147222940 DJ On-Demand Anodyne TSPO 27 40 O=C(c1ccccc1)N(CCc1ccccc1)Cc1ccccc1 ZINC000147222940 DJ On-Demand Anodyne ALOX15 15 50 O=C(c1ccccc1)N(CCc1ccccc1)Cc1ccccc1 ZINC000147222940 DJ On-Demand Anodyne CES1 50 38 O=C(c1ccccc1)N(CCc1ccccc1)Cc1ccccc1 ZINC000147222940 DJ On-Demand Anodyne PLM2_PLAFA 47 50 O=C(c1ccccc1)N(CCc1ccccc1)Cc1ccccc1 ZINC000147222940 DJ On-Demand Anodyne MLYCD 17 49 O=C(c1ccccc1)N(CCc1ccccc1)Cc1ccccc1 ZINC000147222940 DJ On-Demand Anodyne LIMK2 46 49 Cc1cc(=O)oc2cc(Oc3nc(N)ncc3Br)ccc12 ZINC000147223039 EG For-Sale Anodyne MAOA 71 47 Cc1cc(=O)oc2cc(Oc3nc(N)ncc3Br)ccc12 ZINC000147223039 EG For-Sale Anodyne MAOB 43 47 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](c2ccccc2)C2CCCC2)c1 ZINC000147223042 FI On-Demand Bother TAAR1 21 40 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](c2ccccc2)C2CCCC2)c1 ZINC000147223042 FI On-Demand Bother AKR1C2 33 44 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne RARA 21 42 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne MAOB 19 41 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne AVPR2 50 40 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne AVPR1A 26 49 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne MAPK14 24 40 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne COLA 39 43 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne CPT1A 55 47 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne CPT2 44 43 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne PYGL 22 41 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne PRNP 30 40 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne F3 47 31 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne NR1H4 17 46 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne P4HTM 0 41 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne CPT1B 18 43 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne CSF1R 24 46 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne TAAR1 25 43 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne AKR1C3 37 40 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne SHH 47 36 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne AKR1C2 42 40 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne SMO 27 40 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne KCNK3 96 42 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(Cl)c2)cc1Br ZINC000147223071 FI On-Demand Anodyne KCNK9 48 38 COc1cc(OC)cc(C(=O)N[C@@H](C(=O)N2CCC(C#N)CC2)C(C)C)c1 ZINC000147223177 FE On-Demand Mild ELANE 35 43 COc1cc(OC)cc(C(=O)N[C@@H](C(=O)N2CCC(C#N)CC2)C(C)C)c1 ZINC000147223177 FE On-Demand Mild CCR1 48 46 C[C@@H]1C[C@H]2c3cccc(O)c3CC[C@H]2N(CCO)C1 ZINC000147223250 CE For-Sale Anodyne DRD1 32 41 C[C@@H]1C[C@H]2c3cccc(O)c3CC[C@H]2N(CCO)C1 ZINC000147223250 CE For-Sale Anodyne DRD5 36 41 Cc1nc(N)cc(Oc2ccc3c(C)cc(=O)oc3c2)n1 ZINC000147223316 CF For-Sale Anodyne MAOA 63 47 Cc1nc(N)cc(Oc2ccc3c(C)cc(=O)oc3c2)n1 ZINC000147223316 CF For-Sale Anodyne MAOB 39 47 O=C(O)c1ccc(NC(=O)C2[C@H]3CCCC[C@H]23)cc1Cl ZINC000147223325 CG On-Demand Anodyne NPY2R 33 44 O=C(O)c1ccc(NC(=O)C2[C@H]3CCCC[C@H]23)cc1Cl ZINC000147223325 CG On-Demand Anodyne GRM4 18 41 CCOc1ccc(C(=O)NNC(=O)Nc2cccc(CN(C)C)c2)cc1OC ZINC000147223386 GF On-Demand Reactive ROCK2 15 52 CCOc1ccc(C(=O)NNC(=O)Nc2cccc(CN(C)C)c2)cc1OC ZINC000147223386 GF On-Demand Reactive KCNK3 53 45 CCOc1ccc(C(=O)NNC(=O)Nc2cccc(CN(C)C)c2)cc1OC ZINC000147223386 GF On-Demand Reactive KCNK9 45 45 CCc1cc(NC[C@@H]2CNCCO2)ncn1 ZINC000147223426 BC For-Sale Anodyne EPHA2 41 35 CC(C)[C@H](NC(=O)c1ccco1)C(=O)N1CCC(C#N)CC1 ZINC000147223464 DD On-Demand Mild CCR1 51 45 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(OC(F)F)c(Cl)c1 ZINC000147223518 FF On-Demand Anodyne ENV 41 33 Cc1cnc(N)nc1Oc1ccc2c(C)cc(=O)oc2c1 ZINC000147223523 CF For-Sale Anodyne MAOA 75 50 Cc1cnc(N)nc1Oc1ccc2c(C)cc(=O)oc2c1 ZINC000147223523 CF For-Sale Anodyne MAOB 48 50 O=C(O)c1ccc(NC(=O)C2[C@H]3CCCC[C@@H]23)cc1Cl ZINC000147223536 CG For-Sale Anodyne NPY2R 28 44 CCOc1ccc(C(=O)NNC(=O)Nc2ccc(=O)n(CC)c2)cc1OC ZINC000147223621 FD On-Demand Reactive ENPP1 64 37 CN(Cc1cscn1)C(=O)NC[C@H](Cc1ccccc1)N(C)C ZINC000147223629 EE On-Demand Anodyne BMP1 53 37 CN(Cc1cscn1)C(=O)NC[C@H](Cc1ccccc1)N(C)C ZINC000147223629 EE On-Demand Anodyne CYP3A4 21 47 CN(Cc1cscn1)C(=O)NC[C@H](Cc1ccccc1)N(C)C ZINC000147223629 EE On-Demand Anodyne GPR142 43 40 CCc1cc(NC[C@H]2CNCCO2)ncn1 ZINC000147223632 BC For-Sale Anodyne EPHA2 41 35 CC(C)[C@@H](NC(=O)c1ccco1)C(=O)N1CCC(C#N)CC1 ZINC000147223675 DD On-Demand Mild CCR1 51 45 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(OC(F)F)c(Cl)c1 ZINC000147223709 FF On-Demand Anodyne ENV 41 33 Cc1cc(=O)oc2cc(Oc3nc(N)ncc3F)ccc12 ZINC000147223735 CE For-Sale Anodyne MAOA 63 47 Cc1cc(=O)oc2cc(Oc3nc(N)ncc3F)ccc12 ZINC000147223735 CE For-Sale Anodyne MAOB 41 47 O=C(O)c1ccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)cc1Cl ZINC000147223763 CG On-Demand Anodyne NPY2R 33 44 O=C(O)c1ccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)cc1Cl ZINC000147223763 CG On-Demand Anodyne GRM4 18 41 CN(Cc1cscn1)C(=O)NC[C@@H](Cc1ccccc1)N(C)C ZINC000147223809 EE On-Demand Anodyne CYP3A4 21 47 CN(Cc1cscn1)C(=O)NC[C@@H](Cc1ccccc1)N(C)C ZINC000147223809 EE On-Demand Anodyne GPR142 43 40 CCCOc1ccc(C(F)(F)F)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147223896 GG On-Demand Anodyne PPARD 20 40 CCCCOc1ccc(C(=O)N2CCC(C#N)CC2)cc1OC ZINC000147223929 DG On-Demand Mild THRA 39 46 CCCCOc1ccc(C(=O)N2CCC(C#N)CC2)cc1OC ZINC000147223929 DG On-Demand Mild AVPR1A 19 41 CCCCOc1ccc(C(=O)N2CCC(C#N)CC2)cc1OC ZINC000147223929 DG On-Demand Mild THRB 26 46 CCCCOc1ccc(C(=O)N2CCC(C#N)CC2)cc1OC ZINC000147223929 DG On-Demand Mild PLA2G4B 33 45 CCCCOc1ccc(C(=O)N2CCC(C#N)CC2)cc1OC ZINC000147223929 DG On-Demand Mild L3MBTL3 56 35 Brc1cncnc1NC[C@@H]1CNCCO1 ZINC000147223930 CC On-Demand Anodyne EPHA2 41 38 CNc1cc(Oc2ccc3c(C)cc(=O)oc3c2)ncn1 ZINC000147223931 CF For-Sale Anodyne MAOA 66 49 CNc1cc(Oc2ccc3c(C)cc(=O)oc3c2)ncn1 ZINC000147223931 CF For-Sale Anodyne MAOB 46 49 COCc1cccc(-c2ncc(C(=O)OC)s2)c1 ZINC000147223975 CF For-Sale Anodyne HSD17B2 17 45 COCc1nc(C(=O)N2CCN(C(=O)[C@@H]3CCCO3)CC2)cs1 ZINC000147223995 EC On-Demand Anodyne TRPC6 55 37 Cc1cc(=O)oc2cc(Oc3nc(N)ncc3Cl)ccc12 ZINC000147224048 DF For-Sale Anodyne MAOA 63 47 Cc1cc(=O)oc2cc(Oc3nc(N)ncc3Cl)ccc12 ZINC000147224048 DF For-Sale Anodyne MAOB 46 47 CCCOc1ccc(C(F)(F)F)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147224077 GG On-Demand Anodyne PPARD 20 40 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccc(C(F)(F)F)c1 ZINC000147224092 EI On-Demand Anodyne BMP1 0 45 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccc(C(F)(F)F)c1 ZINC000147224092 EI On-Demand Anodyne CYP3A4 15 43 Brc1cncnc1NC[C@H]1CNCCO1 ZINC000147224109 CC On-Demand Anodyne EPHA2 41 38 Cn1cc(C#N)c2ccc([N+](=O)[O-])cc21 ZINC000147224143 BD For-Sale Mild IMPDH2 31 56 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild FOLH1 50 45 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild FABP2 0 45 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild FABP4 16 45 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild PLA2G2C 0 49 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild CCKAR 0 43 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild CPT1A 47 55 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild FAAH 0 42 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild EPHX2 68 55 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild Q6UB75_PIG 0 52 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild FABP5 15 45 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild ASAH1 84 35 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild SLC22A20 0 45 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild ACAT 0 40 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild NOD1 95 44 CCCCCCCCNC(=O)N[C@@H](C)CCC(=O)O ZINC000147224185 CF For-Sale Mild CQSS 56 37 CCCOc1cccc(-c2ncc(C(=O)OC)s2)c1 ZINC000147224193 CG For-Sale Anodyne PPARA 20 40 CCCOc1cccc(-c2ncc(C(=O)OC)s2)c1 ZINC000147224193 CG For-Sale Anodyne HSD17B2 16 46 COCc1nc(C(=O)N2CCN(C(=O)[C@H]3CCCO3)CC2)cs1 ZINC000147224210 EC On-Demand Anodyne TRPC6 55 37 CC[C@H](CNC(=O)Nc1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147224227 CE For-Sale Bother NMBR 42 33 CNc1nccc(Oc2ccc3c(C)cc(=O)oc3c2)n1 ZINC000147224276 CF For-Sale Anodyne MAOA 73 48 CNc1nccc(Oc2ccc3c(C)cc(=O)oc3c2)n1 ZINC000147224276 CF For-Sale Anodyne MAOB 44 48 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccc(C(F)(F)F)c1 ZINC000147224294 EI On-Demand Anodyne BMP1 0 45 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccc(C(F)(F)F)c1 ZINC000147224294 EI On-Demand Anodyne CYP3A4 15 43 CC(C)C[C@@H]1OC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](C(C)C)NC(=O)CNC1=O ZINC000147224344 KC Annotated Anodyne AVPR2 22 40 CC(C)C[C@@H]1OC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](C(C)C)NC(=O)CNC1=O ZINC000147224344 KC Annotated Anodyne OPRD1 15 47 CC(C)C[C@@H]1OC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](C(C)C)NC(=O)CNC1=O ZINC000147224344 KC Annotated Anodyne EDNRA 0 51 CC(C)C[C@@H]1OC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](C(C)C)NC(=O)CNC1=O ZINC000147224344 KC Annotated Anodyne TACR2 33 44 CC(C)C[C@@H]1OC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](C(C)C)NC(=O)CNC1=O ZINC000147224344 KC Annotated Anodyne GALR1 61 46 CC(C)C[C@@H]1OC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](C(C)C)NC(=O)CNC1=O ZINC000147224344 KC Annotated Anodyne CXCR4 47 39 CC(C)C[C@@H]1OC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](C(C)C)NC(=O)CNC1=O ZINC000147224344 KC Annotated Anodyne HDAC10 20 42 CC(C)C[C@@H]1OC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](C(C)C)NC(=O)CNC1=O ZINC000147224344 KC Annotated Anodyne MLNR 44 43 CC(C)C[C@@H]1OC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](C(C)C)NC(=O)CNC1=O ZINC000147224344 KC Annotated Anodyne GALR2 28 46 CC(C)C[C@@H]1OC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](C(C)C)NC(=O)CNC1=O ZINC000147224344 KC Annotated Anodyne ITGAV 17 40 CC(C)C[C@@H]1OC(=O)[C@@H](CC(C)C)NC(=O)CNC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](C(C)C)NC(=O)CNC1=O ZINC000147224344 KC Annotated Anodyne GHRL 75 45 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147224403 FE On-Demand Mild MMP13 49 52 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147224403 FE On-Demand Mild CCR1 29 43 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147224403 FE On-Demand Mild MMP2 32 52 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147224403 FE On-Demand Mild MMP3 17 52 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147224403 FE On-Demand Mild MMP8 20 40 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147224403 FE On-Demand Mild CAPN1 22 41 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147224403 FE On-Demand Mild MMP12 51 34 Cc1ccc(S(=O)(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147224403 FE On-Demand Mild ST14 48 41 COC(=O)c1cnc(-c2ccc(OC)c(Cl)c2)s1 ZINC000147224433 CG For-Sale Anodyne KMO 0 46 CC[C@@H](CNC(=O)Nc1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147224440 CE For-Sale Bother NMBR 42 33 Nc1cc(Oc2ccc(Oc3ccccc3)cc2)ncn1 ZINC000147224479 CH For-Sale Anodyne LCK 22 41 Nc1cc(Oc2ccc(Oc3ccccc3)cc2)ncn1 ZINC000147224479 CH For-Sale Anodyne TEK 15 41 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild FOLH1 50 45 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild FABP2 0 45 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild FABP4 16 45 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild PLA2G2C 0 49 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild CCKAR 0 43 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild CPT1A 47 55 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild FAAH 0 42 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild EPHX2 68 55 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild Q6UB75_PIG 0 52 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild FABP5 15 45 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild ASAH1 84 35 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild SLC22A20 0 45 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild ACAT 0 40 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild NOD1 95 44 CCCCCCCCNC(=O)N[C@H](C)CCC(=O)O ZINC000147224492 CF For-Sale Mild CQSS 56 37 CC[C@H](CNC(=O)Nc1cccc(C)c1)CC(=O)O ZINC000147224658 CF For-Sale Anodyne CCKAR 26 52 CC[C@H](CNC(=O)Nc1cccc(C)c1)CC(=O)O ZINC000147224658 CF For-Sale Anodyne ACAT 0 49 CC[C@H](CNC(=O)Nc1cccc(C)c1)CC(=O)O ZINC000147224658 CF For-Sale Anodyne KCNK3 71 41 CC[C@H](CNC(=O)Nc1cccc(C)c1)CC(=O)O ZINC000147224658 CF For-Sale Anodyne KCNK9 50 41 CCCCCCCCNC(=O)NC[C@H](C(=O)O)C(C)C ZINC000147224726 CG For-Sale Mild CPT1A 24 44 CCCCCCCCNC(=O)NC[C@H](C(=O)O)C(C)C ZINC000147224726 CG For-Sale Mild EPHX2 60 51 CCCCCCCCNC(=O)NC[C@H](C(=O)O)C(C)C ZINC000147224726 CG For-Sale Mild ASAH1 88 35 CCCCCCCCNC(=O)NC[C@H](C(=O)O)C(C)C ZINC000147224726 CG For-Sale Mild NOD1 60 38 CCCCCCCCNC(=O)NC[C@H](C(=O)O)C(C)C ZINC000147224726 CG For-Sale Mild CQSS 50 33 COC(=O)c1cnc(-c2cccc(OC(C)C)c2)s1 ZINC000147224733 CG For-Sale Anodyne ACACA 31 40 COC(=O)c1cnc(-c2cccc(OC(C)C)c2)s1 ZINC000147224733 CG For-Sale Anodyne ACACB 29 40 COC(=O)c1cnc(-c2cccc(OC(C)C)c2)s1 ZINC000147224733 CG For-Sale Anodyne HSD17B2 20 47 CCOC(=O)c1cnc(-c2ccncc2)nc1NC ZINC000147224768 CD For-Sale Anodyne JUN 20 53 CC[C@@H](CNC(=O)Nc1cccc(C)c1)CC(=O)O ZINC000147224795 CF For-Sale Anodyne CCKAR 26 52 CC[C@@H](CNC(=O)Nc1cccc(C)c1)CC(=O)O ZINC000147224795 CF For-Sale Anodyne ACAT 0 49 CC[C@@H](CNC(=O)Nc1cccc(C)c1)CC(=O)O ZINC000147224795 CF For-Sale Anodyne KCNK3 71 41 CC[C@@H](CNC(=O)Nc1cccc(C)c1)CC(=O)O ZINC000147224795 CF For-Sale Anodyne KCNK9 50 41 NS(=O)(=O)c1cc(Br)ccc1OCC(=O)N1CCCC1 ZINC000147224858 FD For-Sale Anodyne GPR183 0 40 COc1cc(NC[C@@H]2CNCCO2)c([N+](=O)[O-])cc1F ZINC000147224874 CD On-Demand Bother EPHA2 44 41 CCCCCCCCNC(=O)NC[C@@H](C(=O)O)C(C)C ZINC000147224944 CG For-Sale Mild CPT1A 24 44 CCCCCCCCNC(=O)NC[C@@H](C(=O)O)C(C)C ZINC000147224944 CG For-Sale Mild EPHX2 60 51 CCCCCCCCNC(=O)NC[C@@H](C(=O)O)C(C)C ZINC000147224944 CG For-Sale Mild ASAH1 88 35 CCCCCCCCNC(=O)NC[C@@H](C(=O)O)C(C)C ZINC000147224944 CG For-Sale Mild NOD1 60 38 CCCCCCCCNC(=O)NC[C@@H](C(=O)O)C(C)C ZINC000147224944 CG For-Sale Mild CQSS 50 33 CCOc1ccc(S(=O)(=O)Nc2ccc([C@@H](C#N)c3ccccc3)c(Cl)c2)cc1 ZINC000147225037 IK On-Demand Mild ALPL 16 50 COc1cc(NC[C@H]2CNCCO2)c([N+](=O)[O-])cc1F ZINC000147225066 CD On-Demand Bother EPHA2 44 41 CCOC(=O)Cc1cccc(C(=O)c2ccc(Br)cc2)c1N ZINC000147225136 FG For-Sale Anodyne SHC 40 30 Cc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)c1 ZINC000147225138 FG On-Demand Anodyne RAF1 28 45 Cc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)c1 ZINC000147225138 FG On-Demand Anodyne PFKFB3 54 33 CCCCCCCCNC(=O)N[C@@H]1COC[C@@H]1C(=O)O ZINC000147225152 CD For-Sale Mild EPHX2 25 50 CCCCCCCCNC(=O)N[C@@H]1COC[C@@H]1C(=O)O ZINC000147225152 CD For-Sale Mild ASAH1 42 32 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCC(CBr)CC1 ZINC000147225153 GE For-Sale Reactive PKM 62 71 CCOC(=O)c1cnc(-c2ccccn2)nc1N(C)C ZINC000147225187 CD For-Sale Anodyne JUN 18 42 CCOC(=O)c1cnc(-c2ccccn2)nc1N(C)C ZINC000147225187 CD For-Sale Anodyne ADORA3 15 42 Nc1ccc2c(NCC(F)F)ncnc2c1 ZINC000147225189 BD For-Sale Anodyne EGFR 25 49 CCOc1ccc(S(=O)(=O)Nc2ccc([C@H](C#N)c3ccccc3)c(Cl)c2)cc1 ZINC000147225216 IK On-Demand Mild ALPL 16 50 CCCCCCCCNC(=O)N[C@H]1COC[C@@H]1C(=O)O ZINC000147225312 CD For-Sale Mild EPHX2 25 50 CCCCCCCCNC(=O)N[C@H]1COC[C@@H]1C(=O)O ZINC000147225312 CD For-Sale Mild ASAH1 42 32 Cc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)c1 ZINC000147225326 FG On-Demand Anodyne RAF1 28 45 Cc1cccc(Oc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)c1 ZINC000147225326 FG On-Demand Anodyne PFKFB3 54 33 N#Cc1ccnnc1NC[C@@H]1CNCCO1 ZINC000147225404 BB For-Sale Mild EPHA2 40 35 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H]1C[C@@H]1C(=O)O ZINC000147225463 CD For-Sale Bother CACNA1D 47 35 CNC(=O)COc1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147225464 HF On-Demand Anodyne PDS 49 40 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1C[C@@H](C)C[C@@H](C)C1 ZINC000147225478 HF On-Demand Mild L3MBTL3 58 35 CCCCCCCCNC(=O)N[C@@H]1COC[C@H]1C(=O)O ZINC000147225513 CD For-Sale Mild EPHX2 25 50 CCCCCCCCNC(=O)N[C@@H]1COC[C@H]1C(=O)O ZINC000147225513 CD For-Sale Mild ASAH1 42 32 N#Cc1ccnnc1NC[C@H]1CNCCO1 ZINC000147225597 BB For-Sale Mild EPHA2 40 35 CCC(CC)N(CCOC)C(=O)C1CCN(C(=O)Nc2cccc(C)c2)CC1 ZINC000147225618 GH On-Demand Anodyne CCKAR 16 41 CCC(CC)N(CCOC)C(=O)C1CCN(C(=O)Nc2cccc(C)c2)CC1 ZINC000147225618 GH On-Demand Anodyne CCKBR 20 41 CCC(CC)N(CCOC)C(=O)C1CCN(C(=O)Nc2cccc(C)c2)CC1 ZINC000147225618 GH On-Demand Anodyne KCNK3 57 36 CCC(CC)N(CCOC)C(=O)C1CCN(C(=O)Nc2cccc(C)c2)CC1 ZINC000147225618 GH On-Demand Anodyne KCNK9 46 36 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H]1C[C@@H]1C(=O)O ZINC000147225633 CD For-Sale Bother CACNA1D 47 35 CNC(=O)COc1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147225664 HF On-Demand Anodyne PDS 49 40 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1C[C@@H](C)C[C@H](C)C1 ZINC000147225722 HF On-Demand Mild L3MBTL3 58 35 CCCCCCCCNC(=O)N[C@H]1COC[C@H]1C(=O)O ZINC000147225735 CD For-Sale Mild EPHX2 25 50 CCCCCCCCNC(=O)N[C@H]1COC[C@H]1C(=O)O ZINC000147225735 CD For-Sale Mild ASAH1 42 32 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H]1C[C@@H]1C(=O)O ZINC000147225808 CD For-Sale Bother CACNA1D 47 35 Fc1cc(Cl)cnc1NC[C@@H]1CNCCO1 ZINC000147225820 BD On-Demand Anodyne EPHA2 41 42 CNC(=O)COc1cccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147225847 HF On-Demand Anodyne PDS 49 40 CC[C@H](CNC(=O)Nc1ccc(Cl)cc1)CC(=O)O ZINC000147225863 CF For-Sale Anodyne GUAB 0 42 CC[C@H](CNC(=O)Nc1ccc(Cl)cc1)CC(=O)O ZINC000147225863 CF For-Sale Anodyne P95276_MYCTO 0 41 CC[C@H](CNC(=O)Nc1ccc(Cl)cc1)CC(=O)O ZINC000147225863 CF For-Sale Anodyne PSBA 0 40 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1C[C@H](C)C[C@@H](C)C1 ZINC000147225928 HF On-Demand Mild L3MBTL3 58 35 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild PPARA 0 43 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild FABP2 0 68 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild FABP4 23 68 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild PLA2G2C 0 45 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild PLA2G4A 0 66 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild CPT1A 47 51 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild DNM1 0 47 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild PLA2G4B 43 35 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild FAAH 0 55 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild S1PR2 30 44 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild EPHX2 41 81 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild Q6UB75_PIG 0 48 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild PA2A1_NAJMO 0 40 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild FABP3 42 55 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild FABP5 23 68 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild GNAI1 0 41 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild GNAI3 0 41 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild GNAO1 0 41 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild FFAR1 0 50 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild FABP1 18 55 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild ASAH1 99 36 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild SLC22A20 0 68 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild KDM4A 0 41 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild ACAT 0 46 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild KDM4C 0 41 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild LASR 44 31 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild NOD1 62 40 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild SLC22A8 0 68 CCCCCCCCNC(=O)NCCCCCCC(=O)O ZINC000147225935 DH For-Sale Mild CQSS 64 39 COc1ccc(OC)c(CN2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)c1 ZINC000147225952 GF On-Demand Bother MGLL 0 46 COc1ccc(OC)c(CN2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)c1 ZINC000147225952 GF On-Demand Bother ABHD6 0 46 COc1ccc(OC)c(CN2CCN(C(=O)c3cc(C)cc([N+](=O)[O-])c3)CC2)c1 ZINC000147225952 GF On-Demand Bother GPR183 0 40 CCNC(=O)c1ccc(C)c(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147225953 ED On-Demand Anodyne MAPK14 40 45 N#Cc1ccc(Nc2nc(C(=O)O)cs2)c(F)c1 ZINC000147225978 CF For-Sale Mild PTGER1 15 45 N#Cc1ccc(Nc2nc(C(=O)O)cs2)c(F)c1 ZINC000147225978 CF For-Sale Mild TRPC6 60 48 N#Cc1ccc(Nc2nc(C(=O)O)cs2)c(F)c1 ZINC000147225978 CF For-Sale Mild TRPC3 52 33 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H]1C[C@@H]1C(=O)O ZINC000147225989 CD For-Sale Bother CACNA1D 47 35 Fc1cc(Cl)cnc1NC[C@H]1CNCCO1 ZINC000147226006 BD On-Demand Anodyne EPHA2 41 42 Cc1ccnc(-c2ccn3c(-c4cccc(NC(=O)NCC(F)(F)F)c4)cnc3c2)n1 ZINC000147226008 II Annotated Anodyne GYRB 0 40 Cc1ccnc(-c2ccn3c(-c4cccc(NC(=O)NCC(F)(F)F)c4)cnc3c2)n1 ZINC000147226008 II Annotated Anodyne BRAF 41 39 O=C(NCC1CC1)[C@@H]1CCC(=O)N(Cc2ccccc2)[C@@H]1c1ccccc1 ZINC000147226052 FH On-Demand Anodyne P2RX7 24 48 CNC(=O)COc1cccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147226058 HF On-Demand Anodyne PDS 49 40 CC[C@@H](CNC(=O)Nc1ccc(Cl)cc1)CC(=O)O ZINC000147226068 CF For-Sale Anodyne GUAB 0 42 CC[C@@H](CNC(=O)Nc1ccc(Cl)cc1)CC(=O)O ZINC000147226068 CF For-Sale Anodyne P95276_MYCTO 0 41 CC[C@@H](CNC(=O)Nc1ccc(Cl)cc1)CC(=O)O ZINC000147226068 CF For-Sale Anodyne PSBA 0 40 CCCCCCCCNC(=O)NC1(C(=O)O)CC1 ZINC000147226144 CE For-Sale Mild CPT1A 26 42 CCCCCCCCNC(=O)NC1(C(=O)O)CC1 ZINC000147226144 CE For-Sale Mild EPHX2 40 55 CCCCCCCCNC(=O)NC1(C(=O)O)CC1 ZINC000147226144 CE For-Sale Mild ASAH1 83 35 CCNC(=O)c1ccc(C)c(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147226158 ED On-Demand Anodyne MAPK14 40 45 OC[C@H]1O[C@H](Oc2ccc(Cl)cc2)[C@H](O)[C@@H](O)[C@@H]1O ZINC000147226167 CB Annotated Anodyne TYR 40 57 OC[C@H]1O[C@H](Oc2ccc(Cl)cc2)[C@H](O)[C@@H](O)[C@@H]1O ZINC000147226167 CB Annotated Anodyne VEGFA 37 40 OC[C@H]1O[C@H](Oc2ccc(Cl)cc2)[C@H](O)[C@@H](O)[C@@H]1O ZINC000147226167 CB Annotated Anodyne IL2 29 46 OC[C@H]1O[C@H](Oc2ccc(Cl)cc2)[C@H](O)[C@@H](O)[C@@H]1O ZINC000147226167 CB Annotated Anodyne SLC5A1 92 44 OC[C@H]1O[C@H](Oc2ccc(Cl)cc2)[C@H](O)[C@@H](O)[C@@H]1O ZINC000147226167 CB Annotated Anodyne SLC5A2 141 52 OC[C@H]1O[C@H](Oc2ccc(Cl)cc2)[C@H](O)[C@@H](O)[C@@H]1O ZINC000147226167 CB Annotated Anodyne FIMH 146 72 OC[C@H]1O[C@H](Oc2ccc(Cl)cc2)[C@H](O)[C@@H](O)[C@@H]1O ZINC000147226167 CB Annotated Anodyne SLC5A4 23 50 COC(=O)CCN1CCN(CCCF)CC1 ZINC000147226185 BC On-Demand Anodyne PAOX 19 44 Cc1nc(Nc2ccc(C#N)cc2F)sc1C(=O)O ZINC000147226188 CF For-Sale Mild DHODH 20 40 O=C(NCC1CC1)[C@@H]1CCC(=O)N(Cc2ccccc2)[C@H]1c1ccccc1 ZINC000147226253 FH On-Demand Anodyne P2RX7 24 48 CNC(=O)COc1cccc(CNC(=O)c2cnn(-c3ccccc3Cl)c2)c1 ZINC000147226272 GF On-Demand Anodyne UPP1 42 32 CNC(=O)COc1cccc(CNC(=O)c2cnn(-c3ccccc3Cl)c2)c1 ZINC000147226272 GF On-Demand Anodyne PDS 55 34 c1ccc(CN[C@@H]2CCCNCC2)cc1 ZINC000147226295 BD In-Stock Anodyne SLC6A3 0 45 CC[C@H](CNC(=O)N1CCCCC1)CC(=O)O ZINC000147226328 BD For-Sale Anodyne RIR1_HHV11 44 38 CCCCCCCCNC(=O)N(CC)CCC(=O)O ZINC000147226367 CF For-Sale Mild FABP2 0 47 CCCCCCCCNC(=O)N(CC)CCC(=O)O ZINC000147226367 CF For-Sale Mild FABP4 17 47 CCCCCCCCNC(=O)N(CC)CCC(=O)O ZINC000147226367 CF For-Sale Mild DNM1 0 45 CCCCCCCCNC(=O)N(CC)CCC(=O)O ZINC000147226367 CF For-Sale Mild EPHX2 30 55 CCCCCCCCNC(=O)N(CC)CCC(=O)O ZINC000147226367 CF For-Sale Mild FABP5 16 47 CCCCCCCCNC(=O)N(CC)CCC(=O)O ZINC000147226367 CF For-Sale Mild ASAH1 83 33 CCCCCCCCNC(=O)N(CC)CCC(=O)O ZINC000147226367 CF For-Sale Mild SLC22A20 0 47 CCCCCCCCNC(=O)N(CC)CCC(=O)O ZINC000147226367 CF For-Sale Mild KDM4A 0 40 CCCCCCCCNC(=O)N(CC)CCC(=O)O ZINC000147226367 CF For-Sale Mild CQSS 50 31 Cc1ccc(C(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147226368 EF On-Demand Mild ELANE 45 42 Cc1ccc(C(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147226368 EF On-Demand Mild CCR1 66 64 COC(=O)c1sc(Nc2ccc(C#N)cc2F)nc1C ZINC000147226413 CF For-Sale Mild DHODH 26 41 CN[C@@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147226417 BE For-Sale Anodyne DRD2 19 46 CN[C@@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147226417 BE For-Sale Anodyne DRD4 19 48 CN[C@@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147226417 BE For-Sale Anodyne DRD3 16 48 CN[C@@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147226417 BE For-Sale Anodyne SLC6A3 29 49 CN[C@@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147226417 BE For-Sale Anodyne SLC18A2 41 37 CN[C@@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147226417 BE For-Sale Anodyne KCNH2 28 43 CN[C@@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147226417 BE For-Sale Anodyne SIGMAR1 41 56 CN[C@@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147226417 BE For-Sale Anodyne ACHP_LYMST 22 49 CN[C@@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147226417 BE For-Sale Anodyne ARG1 30 42 CN[C@@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147226417 BE For-Sale Anodyne ARG2 30 42 CN[C@@H]1C[C@@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147226417 BE For-Sale Anodyne Q8WSF8_APLCA 24 40 O=C(NCC1CC1)[C@H]1CCC(=O)N(Cc2ccccc2)[C@@H]1c1ccccc1 ZINC000147226464 FH On-Demand Anodyne P2RX7 24 48 c1ccc(CN[C@H]2CCCNCC2)cc1 ZINC000147226502 BD In-Stock Anodyne SLC6A3 0 45 CC[C@@H](CNC(=O)N1CCCCC1)CC(=O)O ZINC000147226527 BD For-Sale Anodyne RIR1_HHV11 44 38 CC[C@@H](C)[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1nc2ccccc2[nH]1 ZINC000147226530 GF On-Demand Anodyne ADORA2B 32 41 CC[C@@H](C)[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1nc2ccccc2[nH]1 ZINC000147226530 GF On-Demand Anodyne CHEK2 74 42 Cc1ccc(C(=O)N[C@@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147226574 EF On-Demand Mild ELANE 45 42 Cc1ccc(C(=O)N[C@@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147226574 EF On-Demand Mild CCR1 66 64 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne ALOX5 15 60 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne PTGS2 0 47 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne PTGER2 23 46 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne AKR1B1 21 40 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne PTGER4 0 46 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne CYP1B1 49 42 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne P2RX3 16 44 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne LTB4R 32 40 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne AHR 35 44 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne HDAC8 27 42 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne CA14 0 49 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne MTNR1A 31 51 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne MTNR1B 32 51 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne CYP1A1 36 40 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne HDAC6 15 42 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne CYP1A2 15 45 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne ALS 48 32 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne AKR1C3 46 43 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne PTPA 0 46 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne ABCG2 20 49 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne RHOA 0 57 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne CYSP_PLAFA 40 34 COc1ccc(Oc2cccc(/C=C\C(=O)O)c2)cc1 ZINC000147226589 CH For-Sale Anodyne GPR183 0 40 CCCCCCCCNC(=O)N[C@@H](CO)C(=O)O ZINC000147226595 CD For-Sale Mild FOLH1 56 49 CCCCCCCCNC(=O)N[C@@H](CO)C(=O)O ZINC000147226595 CD For-Sale Mild CPT1A 44 52 CCCCCCCCNC(=O)N[C@@H](CO)C(=O)O ZINC000147226595 CD For-Sale Mild EPHX2 25 53 CCCCCCCCNC(=O)N[C@@H](CO)C(=O)O ZINC000147226595 CD For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N[C@@H](CO)C(=O)O ZINC000147226595 CD For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N[C@@H](CO)C(=O)O ZINC000147226595 CD For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N[C@@H](CO)C(=O)O ZINC000147226595 CD For-Sale Mild TLR2 0 42 CCCCCCCCNC(=O)N[C@@H](CO)C(=O)O ZINC000147226595 CD For-Sale Mild ASAH1 87 36 CCCCCCCCNC(=O)N[C@@H](CO)C(=O)O ZINC000147226595 CD For-Sale Mild NOD1 94 45 CCCCCCCCNC(=O)N[C@@H](CO)C(=O)O ZINC000147226595 CD For-Sale Mild CQSS 50 31 Cc1cc(CNC(=O)Nc2ccc(NC(=O)c3ccoc3)cc2C(F)(F)F)no1 ZINC000147226596 HI On-Demand Anodyne ABL1 41 34 Cc1cc(CNC(=O)Nc2ccc(NC(=O)c3ccoc3)cc2C(F)(F)F)no1 ZINC000147226596 HI On-Demand Anodyne Q8MMZ8_EIMTE 44 33 Br[C@H]1CCN(c2ncnc3c2cnn3-c2ccccc2)C1 ZINC000147226636 EF For-Sale Reactive PDE3B 57 33 O=C(NCC1CC1)[C@H]1CCC(=O)N(Cc2ccccc2)[C@H]1c1ccccc1 ZINC000147226643 FH On-Demand Anodyne P2RX7 24 48 COC(=O)c1cnc(-c2ccc(Cl)c(Cl)c2)s1 ZINC000147226696 CH For-Sale Anodyne KMO 0 41 CNC(=O)COc1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147226709 FF On-Demand Anodyne MAOB 15 42 CNC(=O)COc1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147226709 FF On-Demand Anodyne PDS 62 40 CC[C@H](C)[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1nc2ccccc2[nH]1 ZINC000147226715 GF On-Demand Anodyne ADORA2B 32 41 CC[C@H](C)[C@H](NC(=O)COc1ccc(C(N)=O)cc1)c1nc2ccccc2[nH]1 ZINC000147226715 GF On-Demand Anodyne CHEK2 74 42 CC[C@@H]([C@@H]1CCCO1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147226757 KK Annotated Anodyne TP53 44 68 CC[C@@H]([C@@H]1CCCO1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147226757 KK Annotated Anodyne MDM2 264 68 CCCCCCCCNC(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147226760 CF On-Demand Mild SLC6A1 103 38 CCCCCCCCNC(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147226760 CF On-Demand Mild F2R 0 42 CCCCCCCCNC(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147226760 CF On-Demand Mild EPHX2 15 46 CCCCCCCCNC(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147226760 CF On-Demand Mild TPP2 21 41 CCCCCCCCNC(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147226760 CF On-Demand Mild GNAI1 0 43 CCCCCCCCNC(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147226760 CF On-Demand Mild GNAI3 0 43 CCCCCCCCNC(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147226760 CF On-Demand Mild GNAO1 0 43 CCCCCCCCNC(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147226760 CF On-Demand Mild ASAH1 102 40 CCCCOc1ccc(OC)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147226768 FE On-Demand Anodyne MTNR1A 26 40 CCCCOc1ccc(OC)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147226768 FE On-Demand Anodyne MTNR1B 23 40 Cc1cc(C)n(-c2ccc(C(=O)N3CCC(C#N)CC3)cc2)n1 ZINC000147226842 DF On-Demand Mild L3MBTL3 63 38 Br[C@@H]1CCN(c2ncnc3c2cnn3-c2ccccc2)C1 ZINC000147226890 EF For-Sale Reactive PDE3B 57 33 CCNc1cccc(NCc2ccccc2)n1 ZINC000147226893 BG For-Sale Anodyne PETD 0 46 CCNc1cccc(NCc2ccccc2)n1 ZINC000147226893 BG For-Sale Anodyne Q31945_CHEAL 0 40 O=[N+]([O-])c1ccc2[nH]c(NC[C@@H]3CNCCO3)nc2c1 ZINC000147226913 CC On-Demand Bother GYRB 41 37 CNC(=O)COc1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147226921 FF On-Demand Anodyne MAOB 15 42 CNC(=O)COc1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147226921 FF On-Demand Anodyne PDS 62 40 CC[C@@H](C)[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1nc2ccccc2[nH]1 ZINC000147226926 GF On-Demand Anodyne ADORA2B 32 41 CC[C@@H](C)[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1nc2ccccc2[nH]1 ZINC000147226926 GF On-Demand Anodyne CHEK2 74 42 CCCCCCCCNC(=O)N[C@@H](CCOC)C(=O)O ZINC000147226942 CE For-Sale Mild FOLH1 68 53 CCCCCCCCNC(=O)N[C@@H](CCOC)C(=O)O ZINC000147226942 CE For-Sale Mild CPT1A 46 47 CCCCCCCCNC(=O)N[C@@H](CCOC)C(=O)O ZINC000147226942 CE For-Sale Mild EPHX2 61 47 CCCCCCCCNC(=O)N[C@@H](CCOC)C(=O)O ZINC000147226942 CE For-Sale Mild ASAH1 59 32 CCCCCCCCNC(=O)N[C@@H](CCOC)C(=O)O ZINC000147226942 CE For-Sale Mild NOD1 101 46 CCCCOc1ccc(OC)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147226967 FE On-Demand Anodyne MTNR1A 26 40 CCCCOc1ccc(OC)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147226967 FE On-Demand Anodyne MTNR1B 23 40 CCOC(=O)c1cnc(-c2ccc(Br)cc2)nc1N1CCCC1 ZINC000147226969 GH For-Sale Anodyne P2RY12 52 37 CCOC(=O)c1cnc(-c2ccc(Br)cc2)nc1N1CCCC1 ZINC000147226969 GH For-Sale Anodyne JUN 18 44 CCOC(=O)c1cnc(-c2ccc(Br)cc2)nc1N1CCCC1 ZINC000147226969 GH For-Sale Anodyne PRS 43 32 Cc1ccc(CC(=O)NCCCCCCN)cc1 ZINC000147227005 BE On-Demand Anodyne CA5B 18 40 Cc1ccc(CC(=O)NCCCCCCN)cc1 ZINC000147227005 BE On-Demand Anodyne CA5A 15 40 Cc1ccc(CC(=O)NCCCCCCN)cc1 ZINC000147227005 BE On-Demand Anodyne GRIA1 83 45 Cc1ccc(CC(=O)NCCCCCCN)cc1 ZINC000147227005 BE On-Demand Anodyne FURIN 28 40 Cc1ccc(CC(=O)NCCCCCCN)cc1 ZINC000147227005 BE On-Demand Anodyne CHRND 0 46 Cc1ccc(CC(=O)NCCCCCCN)cc1 ZINC000147227005 BE On-Demand Anodyne NCE103 22 41 Cc1ccc(CC(=O)NCCCCCCN)cc1 ZINC000147227005 BE On-Demand Anodyne POLG_WNV 57 37 Cc1ccc(CC(=O)NCCCCCCN)cc1 ZINC000147227005 BE On-Demand Anodyne PAO 44 36 Cc1ccc(CC(=O)NCCCCCCN)cc1 ZINC000147227005 BE On-Demand Anodyne CAN2 0 41 N#CC1CCN(C(=O)c2ccc3ncsc3c2)CC1 ZINC000147227012 CF On-Demand Mild L3MBTL3 57 36 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CA2 69 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CA6 20 45 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CA1 59 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CA7 52 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CA13 20 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CA4 65 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CA14 35 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CA12 34 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CA9 39 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CAH_METTE 64 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CYNT 56 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne NCE103 33 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CA15 30 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne MTCA1 21 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne P96878_MYCTU 20 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne CA 0 46 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne A6YCJ1_9METZ 39 45 Nc1cc(S(N)(=O)=O)ccc1NCC(F)F ZINC000147227106 CC For-Sale Anodyne Q5TU56_ANOGA 0 46 O=[N+]([O-])c1ccc2[nH]c(NC[C@H]3CNCCO3)nc2c1 ZINC000147227130 CC On-Demand Bother GYRB 41 37 CC[C@H](C)[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1nc2ccccc2[nH]1 ZINC000147227132 GF On-Demand Anodyne ADORA2B 32 41 CC[C@H](C)[C@@H](NC(=O)COc1ccc(C(N)=O)cc1)c1nc2ccccc2[nH]1 ZINC000147227132 GF On-Demand Anodyne CHEK2 74 42 CNC(=O)COc1cccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147227134 FF On-Demand Anodyne MAOB 15 42 CNC(=O)COc1cccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147227134 FF On-Demand Anodyne PDS 62 40 Cc1cc(C(=O)N(C)Cc2ccc(F)cc2)cc([N+](=O)[O-])c1 ZINC000147227148 DG On-Demand Bother MMP8 22 40 Cc1cc(C(=O)N(C)Cc2ccc(F)cc2)cc([N+](=O)[O-])c1 ZINC000147227148 DG On-Demand Bother LIMK2 36 42 CCCCCCCCNC(=O)N[C@H](CCOC)C(=O)O ZINC000147227155 CE For-Sale Mild FOLH1 68 53 CCCCCCCCNC(=O)N[C@H](CCOC)C(=O)O ZINC000147227155 CE For-Sale Mild EPHX2 23 47 CCCCCCCCNC(=O)N[C@H](CCOC)C(=O)O ZINC000147227155 CE For-Sale Mild ASAH1 59 32 CCCCCCCCNC(=O)N[C@H](CCOC)C(=O)O ZINC000147227155 CE For-Sale Mild NOD1 101 46 CSCC[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147227217 EE On-Demand Mild GHRHR 48 32 CSCC[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147227217 EE On-Demand Mild P2RY12 189 37 CSCC[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147227217 EE On-Demand Mild CCR1 27 40 CSCC[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147227217 EE On-Demand Mild PREP 17 44 CSCC[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147227217 EE On-Demand Mild CCKBR 29 41 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne CA2 16 46 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne CA7 15 40 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne CXCR2 15 45 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne GRM4 18 40 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne MTTP 19 40 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne EPHX2 17 43 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne PTGDR 20 46 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne CA9 15 46 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne IDO1 35 43 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne LIMK2 20 40 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne KDM1A 22 49 O=C(Nc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227233 HH On-Demand Anodyne KCNK3 43 46 CCOC(=O)c1csc(Nc2ccc(C#N)cc2F)n1 ZINC000147227262 CG For-Sale Mild TRPC6 39 43 COC(=O)c1cnc(-c2ccc(OC)cc2OC)s1 ZINC000147227270 CF For-Sale Anodyne CYP1B1 24 40 COC(=O)c1cnc(-c2ccc(OC)cc2OC)s1 ZINC000147227270 CF For-Sale Anodyne LUCI_LUCLA 16 41 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive CA2 17 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive CA1 15 42 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive TGM1 24 43 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive EPHX2 51 46 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive TGM2 100 47 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive CA12 15 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive MMP7 15 40 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive CA9 16 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive F13A1 120 48 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive AKR1C3 23 43 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive IDO1 33 41 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive NAMPT 52 47 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive TGM6 0 43 CC(=O)Nc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147227280 GE For-Sale Reactive DDIT3 0 47 CNC(=O)COc1cccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147227331 FF On-Demand Anodyne MAOB 15 42 CNC(=O)COc1cccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147227331 FF On-Demand Anodyne PDS 62 40 CCCCCCCCNC(=O)N(C)[C@@H](C)C(=O)O ZINC000147227373 CE For-Sale Mild EPHX2 29 45 CCCCCCCCNC(=O)N(C)[C@@H](C)C(=O)O ZINC000147227373 CE For-Sale Mild ASAH1 75 35 CCCCCCCCNC(=O)N(C)[C@@H](C)C(=O)O ZINC000147227373 CE For-Sale Mild NOD1 86 42 CCCCCCCCNC(=O)N(C)[C@@H](C)C(=O)O ZINC000147227373 CE For-Sale Mild CQSS 51 34 CSCC[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147227431 EE On-Demand Mild GHRHR 48 32 CSCC[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147227431 EE On-Demand Mild P2RY12 189 37 CSCC[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147227431 EE On-Demand Mild CCKAR 31 42 CSCC[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147227431 EE On-Demand Mild CCR1 27 40 CSCC[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147227431 EE On-Demand Mild PREP 17 44 CSCC[C@@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147227431 EE On-Demand Mild CCKBR 102 45 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne CA2 16 46 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne CA7 15 40 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne CXCR2 15 45 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne GRM4 18 40 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne MTTP 19 40 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne EPHX2 17 43 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne PTGDR 20 46 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne CA9 15 46 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne IDO1 35 43 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne LIMK2 20 40 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne KDM1A 22 49 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227439 HH On-Demand Anodyne KCNK3 43 46 COC(=O)c1cnc(-c2cc(Br)ccc2OC)s1 ZINC000147227469 EG For-Sale Anodyne HTR2A 19 42 CNC(=O)COc1cccc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147227547 GD On-Demand Anodyne MTNR1A 49 38 CNC(=O)COc1cccc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147227547 GD On-Demand Anodyne MTNR1B 40 38 CNC(=O)COc1cccc(CNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147227547 GD On-Demand Anodyne ROCK2 56 39 Clc1ccc(Br)c(Cn2cncn2)c1 ZINC000147227554 CF For-Sale Anodyne CYP19A1 28 41 CCCCCCCCNC(=O)N(C)[C@H](C)C(=O)O ZINC000147227592 CE For-Sale Mild EPHX2 29 45 CCCCCCCCNC(=O)N(C)[C@H](C)C(=O)O ZINC000147227592 CE For-Sale Mild ASAH1 87 35 CCCCCCCCNC(=O)N(C)[C@H](C)C(=O)O ZINC000147227592 CE For-Sale Mild NOD1 86 42 CCCCCCCCNC(=O)N(C)[C@H](C)C(=O)O ZINC000147227592 CE For-Sale Mild CQSS 51 34 Cc1c(NC(=O)c2cccc(F)c2Cl)cccc1C(=O)O ZINC000147227607 DH On-Demand Anodyne FABP2 0 40 Cc1c(NC(=O)c2cccc(F)c2Cl)cccc1C(=O)O ZINC000147227607 DH On-Demand Anodyne NR1H4 15 54 Cc1c(NC(=O)c2cccc(F)c2Cl)cccc1C(=O)O ZINC000147227607 DH On-Demand Anodyne ACPS 0 43 Cc1c(NC(=O)c2cccc(F)c2Cl)cccc1C(=O)O ZINC000147227607 DH On-Demand Anodyne AKR1C3 24 41 Cc1c(NC(=O)c2cccc(F)c2Cl)cccc1C(=O)O ZINC000147227607 DH On-Demand Anodyne AKR1C2 52 41 Cc1c(NC(=O)c2cccc(F)c2Cl)cccc1C(=O)O ZINC000147227607 DH On-Demand Anodyne WDR5 18 40 Cc1c(NC(=O)c2cccc(F)c2Cl)cccc1C(=O)O ZINC000147227607 DH On-Demand Anodyne G2YM83_BOTF4 68 36 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne CA2 16 46 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne CA7 15 40 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne CXCR2 15 45 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne GRM4 18 40 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne MTTP 19 40 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne EPHX2 17 43 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne PTGDR 20 46 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne CA9 15 46 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne IDO1 35 43 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne LIMK2 20 40 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne KDM1A 22 49 O=C(Nc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1)c1ccc(F)cc1 ZINC000147227630 HH On-Demand Anodyne KCNK3 43 46 CN(C)C(=O)NCCNC1=NS(=O)(=O)c2ccccc21 ZINC000147227640 CB On-Demand Anodyne KCNA3 37 40 CC(C)[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147227648 FH On-Demand Mild ELANE 46 43 CC(C)[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147227648 FH On-Demand Mild CCR1 52 48 CC(C)[C@H](NC(=O)c1ccc(C(C)(C)C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147227648 FH On-Demand Mild CELA2A 17 41 CC[C@H](CNC(=O)Nc1ccccc1Cl)CC(=O)O ZINC000147227650 CF For-Sale Anodyne ANPEP 16 49 CC[C@H](CNC(=O)Nc1ccccc1Cl)CC(=O)O ZINC000147227650 CF For-Sale Anodyne CXCL8 59 44 CC[C@H](CNC(=O)Nc1ccccc1Cl)CC(=O)O ZINC000147227650 CF For-Sale Anodyne KCNQ2 46 35 CNC(=O)COc1cccc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147227737 GD On-Demand Anodyne MTNR1A 49 38 CNC(=O)COc1cccc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147227737 GD On-Demand Anodyne MTNR1B 40 38 CNC(=O)COc1cccc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147227737 GD On-Demand Anodyne ROCK2 56 39 CCc1ncc(C(=O)NCC2(N3CCOCC3)CCCCC2)s1 ZINC000147227742 EE On-Demand Anodyne HCN1 67 41 CCc1ncc(C(=O)NCC2(N3CCOCC3)CCCCC2)s1 ZINC000147227742 EE On-Demand Anodyne HCN4 65 41 CCOC(=O)c1cccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)c1 ZINC000147227763 HG On-Demand Anodyne CHRM3 20 42 CCOC(=O)c1cccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)c1 ZINC000147227763 HG On-Demand Anodyne CCR3 46 44 CCOC(=O)c1cccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)c1 ZINC000147227763 HG On-Demand Anodyne EPHX2 23 46 Cc1ccc(C(=O)Nc2cccc(C(=O)O)c2C)cc1Br ZINC000147227796 EI On-Demand Anodyne PPARG 0 48 Cc1ccc(C(=O)Nc2cccc(C(=O)O)c2C)cc1Br ZINC000147227796 EI On-Demand Anodyne PPARA 0 44 Cc1ccc(C(=O)Nc2cccc(C(=O)O)c2C)cc1Br ZINC000147227796 EI On-Demand Anodyne PPARD 28 41 Cc1ccc(C(=O)Nc2cccc(C(=O)O)c2C)cc1Br ZINC000147227796 EI On-Demand Anodyne NR1H4 25 58 Cc1ccc(C(=O)Nc2cccc(C(=O)O)c2C)cc1Br ZINC000147227796 EI On-Demand Anodyne FABH 0 50 Cc1ccc(C(=O)Nc2cccc(C(=O)O)c2C)cc1Br ZINC000147227796 EI On-Demand Anodyne AKR1C3 35 46 Cc1ccc(C(=O)Nc2cccc(C(=O)O)c2C)cc1Br ZINC000147227796 EI On-Demand Anodyne AKR1C2 48 43 Cc1ccc(C(=O)Nc2cccc(C(=O)O)c2C)cc1Br ZINC000147227796 EI On-Demand Anodyne GPR35 61 40 Cc1ccc(C(=O)Nc2cccc(C(=O)O)c2C)cc1Br ZINC000147227796 EI On-Demand Anodyne KCNK3 82 40 Cc1ccc(C(=O)Nc2cccc(C(=O)O)c2C)cc1Br ZINC000147227796 EI On-Demand Anodyne KCNK9 46 38 CCCCCCCCNC(=O)N(CC(=O)O)CC(F)(F)F ZINC000147227797 DG For-Sale Mild CES2 50 40 CCCCCCCCNC(=O)N(CC(=O)O)CC(F)(F)F ZINC000147227797 DG For-Sale Mild EST1_PIG 73 40 CCCCCCCCNC(=O)N(CC(=O)O)CC(F)(F)F ZINC000147227797 DG For-Sale Mild EPHX2 0 41 CCCCCCCCNC(=O)N(CC(=O)O)CC(F)(F)F ZINC000147227797 DG For-Sale Mild CES2C 59 40 CCCCCCCCNC(=O)N(CC(=O)O)CC(F)(F)F ZINC000147227797 DG For-Sale Mild JHE 0 40 CCCCCCCCNC(=O)N(CC(=O)O)CC(F)(F)F ZINC000147227797 DG For-Sale Mild ASAH1 84 34 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147227805 IH On-Demand Mild PRNP 41 36 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147227805 IH On-Demand Mild GRM4 61 45 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147227805 IH On-Demand Mild GRM5 18 44 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147227805 IH On-Demand Mild TGM2 47 39 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147227805 IH On-Demand Mild F13A1 49 39 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147227805 IH On-Demand Mild SHH 18 41 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147227805 IH On-Demand Mild NAMPT 42 40 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147227805 IH On-Demand Mild KCNK3 59 42 CCc1c(NC)ncnc1Nc1ccc(C#N)cc1F ZINC000147227863 CF For-Sale Mild FLT1 0 44 O=S(=O)(N[C@H]1C[C@H]1c1ccccc1)c1cccc2cnccc12 ZINC000147227880 DG On-Demand Anodyne PDE10A 16 40 CCCOc1ccc(-c2ncc(C(=O)OC)s2)cc1 ZINC000147227881 CG For-Sale Anodyne ACACA 44 41 CCCOc1ccc(-c2ncc(C(=O)OC)s2)cc1 ZINC000147227881 CG For-Sale Anodyne ACACB 24 41 CCCOc1ccc(-c2ncc(C(=O)OC)s2)cc1 ZINC000147227881 CG For-Sale Anodyne PLA2G4B 58 33 CC[C@@H](CNC(=O)Nc1ccccc1Cl)CC(=O)O ZINC000147227892 CF For-Sale Anodyne ANPEP 16 49 CC[C@@H](CNC(=O)Nc1ccccc1Cl)CC(=O)O ZINC000147227892 CF For-Sale Anodyne CXCL8 59 44 CC[C@@H](CNC(=O)Nc1ccccc1Cl)CC(=O)O ZINC000147227892 CF For-Sale Anodyne KCNQ2 46 35 CC(C)[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147227903 FH On-Demand Mild ELANE 46 43 CC(C)[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147227903 FH On-Demand Mild CCR1 52 48 CC(C)[C@@H](NC(=O)c1ccc(C(C)(C)C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147227903 FH On-Demand Mild CELA2A 17 41 CNC(=O)COc1cccc(CNC(=O)c2ccc3c(c2)COC3)c1 ZINC000147227958 ED On-Demand Anodyne MMP13 19 46 CCOC(=O)c1cccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)c1 ZINC000147227981 HG On-Demand Anodyne CHRM3 20 42 CCOC(=O)c1cccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)c1 ZINC000147227981 HG On-Demand Anodyne CCKAR 21 42 CCOC(=O)c1cccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)c1 ZINC000147227981 HG On-Demand Anodyne CCR3 46 44 CCOC(=O)c1cccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)c1 ZINC000147227981 HG On-Demand Anodyne CCKBR 17 42 CCOC(=O)c1cccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)c1 ZINC000147227981 HG On-Demand Anodyne EPHX2 23 46 NS(=O)(=O)c1cc(Br)ccc1OCCc1ccncc1 ZINC000147227997 FE For-Sale Anodyne CA14 0 42 CCCCOc1ccc(C(=O)Nc2cccc(C(C)=O)c2O)cc1 ZINC000147228007 EI On-Demand Anodyne CYSLTR1 20 41 CCCCOc1ccc(C(=O)Nc2cccc(C(C)=O)c2O)cc1 ZINC000147228007 EI On-Demand Anodyne CYSLTR2 54 38 CCCCOc1ccc(C(=O)Nc2cccc(C(C)=O)c2O)cc1 ZINC000147228007 EI On-Demand Anodyne SCN2A 18 40 CCCCOc1ccc(C(=O)Nc2cccc(C(C)=O)c2O)cc1 ZINC000147228007 EI On-Demand Anodyne PLA2G4B 92 40 CCCCOc1ccc(C(=O)Nc2cccc(C(C)=O)c2O)cc1 ZINC000147228007 EI On-Demand Anodyne NR1H4 15 42 CCCCOc1ccc(C(=O)Nc2cccc(C(C)=O)c2O)cc1 ZINC000147228007 EI On-Demand Anodyne FAAH 22 41 CCCCOc1ccc(C(=O)Nc2cccc(C(C)=O)c2O)cc1 ZINC000147228007 EI On-Demand Anodyne KCNK3 51 34 CCCCCCCCNC(=O)N(CC)C(C)(C)C(=O)O ZINC000147228022 CG For-Sale Mild EST1_PIG 52 32 CCCCCCCCNC(=O)N(CC)C(C)(C)C(=O)O ZINC000147228022 CG For-Sale Mild EPHX2 25 41 CCCCCCCCNC(=O)N(CC)C(C)(C)C(=O)O ZINC000147228022 CG For-Sale Mild ASAH1 78 32 Cc1nc(C)c(C(=O)Nc2cccc(C(=O)O)c2C)o1 ZINC000147228031 CF On-Demand Anodyne AKR1C2 40 41 Cc1nc(C)c(C(=O)Nc2cccc(C(=O)O)c2C)o1 ZINC000147228031 CF On-Demand Anodyne G2YM83_BOTF4 50 31 O=S(=O)(N[C@H]1C[C@@H]1c1ccccc1)c1cccc2cnccc12 ZINC000147228077 DG On-Demand Anodyne PDE10A 16 40 CCCNc1cccc(NCc2ccccc2)n1 ZINC000147228138 BH For-Sale Anodyne PETD 0 44 COC(=O)c1cnc(-c2ccc(OC(C)C)cc2)s1 ZINC000147228146 CG For-Sale Anodyne ACACA 49 45 COC(=O)c1cnc(-c2ccc(OC(C)C)cc2)s1 ZINC000147228146 CG For-Sale Anodyne ACACB 39 45 CCOc1ccc(OCCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147228149 DG On-Demand Mild LTA4H 15 45 CCOc1ccc(OCCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147228149 DG On-Demand Mild HRH3 22 48 CCOc1ccc(OCCCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147228149 DG On-Demand Mild PLA2G4B 50 34 CCCNc1ncnc(Nc2ccc(C#N)cc2F)c1C ZINC000147228155 CG For-Sale Mild FLT1 0 44 CC[C@H](CNC(=O)Nc1cccc(C#N)c1)CC(=O)O ZINC000147228158 CE For-Sale Mild CCR3 21 45 CC[C@H](CNC(=O)Nc1cccc(C#N)c1)CC(=O)O ZINC000147228158 CE For-Sale Mild MCHR1 19 46 Cc1c(NC(=O)C2[C@H]3CCCC[C@H]23)cccc1C(=O)O ZINC000147228234 CG On-Demand Anodyne AKR1C3 15 41 Cc1c(NC(=O)C2[C@H]3CCCC[C@H]23)cccc1C(=O)O ZINC000147228234 CG On-Demand Anodyne AKR1C2 39 41 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)nc1 ZINC000147228245 CG For-Sale Mild EPHX2 17 61 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)nc1 ZINC000147228245 CG For-Sale Mild ASAH1 88 35 COc1ccc2c(c1)OC[C@H](C(=O)NCCCOCCc1ccccc1)C2 ZINC000147228269 FG On-Demand Anodyne SCNN1A 48 35 COc1ccc2c(c1)OC[C@H](C(=O)NCCCOCCc1ccccc1)C2 ZINC000147228269 FG On-Demand Anodyne NQO2 30 41 COc1ccc2c(c1)OC[C@H](C(=O)NCCCOCCc1ccccc1)C2 ZINC000147228269 FG On-Demand Anodyne MTNR1A 92 43 COc1ccc2c(c1)OC[C@H](C(=O)NCCCOCCc1ccccc1)C2 ZINC000147228269 FG On-Demand Anodyne MTNR1B 86 43 O=S(=O)(N[C@@H]1C[C@H]1c1ccccc1)c1cccc2cnccc12 ZINC000147228330 DG On-Demand Anodyne PDE10A 16 40 CC[C@@H](CNC(=O)Nc1cccc(C#N)c1)CC(=O)O ZINC000147228359 CE For-Sale Mild CCR3 21 45 CC[C@@H](CNC(=O)Nc1cccc(C#N)c1)CC(=O)O ZINC000147228359 CE For-Sale Mild MCHR1 19 46 CC1(C)Oc2ncnc(N)c2N=C1c1ccc([C@@H]2CC[C@H](CC(=O)O)CC2)cc1 ZINC000147228368 GI In-Stock Anodyne DGAT1 60 54 CCNc1ncnc(Nc2ccc(C#N)cc2F)c1C ZINC000147228376 CF For-Sale Mild FLT1 0 44 O=C(NCc1cccc(CN2CCOCC2)c1)C(=O)c1ccc2c(c1)CCC2 ZINC000147228388 GF On-Demand Anodyne CHRM3 16 43 CCCCCCCCNC(=O)N[C@H](C(=O)O)c1cccs1 ZINC000147228390 DH For-Sale Mild FOLH1 27 41 CCCCCCCCNC(=O)N[C@H](C(=O)O)c1cccs1 ZINC000147228390 DH For-Sale Mild CPT1A 22 43 CCCCCCCCNC(=O)N[C@H](C(=O)O)c1cccs1 ZINC000147228390 DH For-Sale Mild EPHX2 47 40 CCCCCCCCNC(=O)N[C@H](C(=O)O)c1cccs1 ZINC000147228390 DH For-Sale Mild ASAH1 88 37 CCCCCCCCNC(=O)N[C@H](C(=O)O)c1cccs1 ZINC000147228390 DH For-Sale Mild ACAT 0 45 CCCOc1ccc(C(=O)NNC(=O)Nc2nc(C)cs2)cc1OC ZINC000147228399 FF On-Demand Reactive GCK 22 48 Cc1c(NC(=O)C2[C@H]3CCCC[C@@H]23)cccc1C(=O)O ZINC000147228436 CG For-Sale Anodyne AKR1C3 15 41 Cc1c(NC(=O)C2[C@H]3CCCC[C@@H]23)cccc1C(=O)O ZINC000147228436 CG For-Sale Anodyne AKR1C2 39 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCCCOCCc1ccccc1)C2 ZINC000147228448 FG On-Demand Anodyne SCNN1A 48 35 COc1ccc2c(c1)OC[C@@H](C(=O)NCCCOCCc1ccccc1)C2 ZINC000147228448 FG On-Demand Anodyne NQO2 30 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCCCOCCc1ccccc1)C2 ZINC000147228448 FG On-Demand Anodyne MTNR1A 92 43 COc1ccc2c(c1)OC[C@@H](C(=O)NCCCOCCc1ccccc1)C2 ZINC000147228448 FG On-Demand Anodyne MTNR1B 86 43 O=S(=O)(c1cccc2cnccc12)N1CCC(CBr)CC1 ZINC000147228484 FG For-Sale Reactive P2RX7 48 42 O=S(=O)(c1cccc2cnccc12)N1CCC(CBr)CC1 ZINC000147228484 FG For-Sale Reactive NPY2R 0 46 O=S(=O)(c1cccc2cnccc12)N1CCC(CBr)CC1 ZINC000147228484 FG For-Sale Reactive ROCK2 0 61 O=S(=O)(c1cccc2cnccc12)N1CCC(CBr)CC1 ZINC000147228484 FG For-Sale Reactive Q95J97_RABIT 0 52 CCCCCCCCNC(=O)N[C@@H](C(=O)O)c1cccs1 ZINC000147228526 DH For-Sale Mild FOLH1 27 41 CCCCCCCCNC(=O)N[C@@H](C(=O)O)c1cccs1 ZINC000147228526 DH For-Sale Mild CPT1A 22 43 CCCCCCCCNC(=O)N[C@@H](C(=O)O)c1cccs1 ZINC000147228526 DH For-Sale Mild EPHX2 47 40 CCCCCCCCNC(=O)N[C@@H](C(=O)O)c1cccs1 ZINC000147228526 DH For-Sale Mild ASAH1 88 37 CCCCCCCCNC(=O)N[C@@H](C(=O)O)c1cccs1 ZINC000147228526 DH For-Sale Mild ACAT 0 45 CN(CCNC(=O)OC(C)(C)C)c1ccc(C#N)cn1 ZINC000147228536 CD On-Demand Mild PAPA1_CARPA 44 34 O=S(=O)(N[C@@H]1C[C@@H]1c1ccccc1)c1cccc2cnccc12 ZINC000147228546 DG On-Demand Anodyne PDE10A 16 40 CCOc1ccc(C(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147228598 FF On-Demand Mild ELANE 45 42 CCOc1ccc(C(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147228598 FF On-Demand Mild CCR1 50 48 CCOc1ccc(C(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147228598 FF On-Demand Mild CELA2A 20 42 Cc1c(NC(=O)C2[C@@H]3CCCC[C@@H]23)cccc1C(=O)O ZINC000147228622 CG On-Demand Anodyne AKR1C3 15 41 Cc1c(NC(=O)C2[C@@H]3CCCC[C@@H]23)cccc1C(=O)O ZINC000147228622 CG On-Demand Anodyne AKR1C2 39 41 CCCOc1ccc(C(=O)NNC(=O)Nc2ncc(C)s2)cc1OC ZINC000147228678 FF On-Demand Reactive SCD1 42 44 CCCOc1ccc(C(=O)NNC(=O)Nc2ncc(C)s2)cc1OC ZINC000147228678 FF On-Demand Reactive SCD 36 44 CCCOc1ccc(C(=O)NNC(=O)Nc2ncc(C)s2)cc1OC ZINC000147228678 FF On-Demand Reactive ENPP1 56 35 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228708 GI On-Demand Anodyne NPY1R 26 41 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228708 GI On-Demand Anodyne CCKAR 31 45 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228708 GI On-Demand Anodyne CCKBR 34 45 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228708 GI On-Demand Anodyne EPHX2 16 41 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228708 GI On-Demand Anodyne KCNK3 73 35 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228708 GI On-Demand Anodyne KCNK9 47 34 CCCCCCCCNC(=O)NCC[C@@H](C)C(=O)O ZINC000147228721 CF For-Sale Mild FOLH1 25 44 CCCCCCCCNC(=O)NCC[C@@H](C)C(=O)O ZINC000147228721 CF For-Sale Mild CPT1A 25 47 CCCCCCCCNC(=O)NCC[C@@H](C)C(=O)O ZINC000147228721 CF For-Sale Mild EPHX2 29 54 CCCCCCCCNC(=O)NCC[C@@H](C)C(=O)O ZINC000147228721 CF For-Sale Mild ASAH1 88 34 CCCCCCCCNC(=O)NCC[C@@H](C)C(=O)O ZINC000147228721 CF For-Sale Mild ACAT 0 42 CCCCCCCCNC(=O)NCC[C@@H](C)C(=O)O ZINC000147228721 CF For-Sale Mild NOD1 99 46 CCCCCCCCNC(=O)NCC[C@@H](C)C(=O)O ZINC000147228721 CF For-Sale Mild CQSS 54 35 CCC(CC)N(CCOC)C(=O)c1cc2cc(C)ccc2[nH]1 ZINC000147228740 DH On-Demand Anodyne PYGL 68 43 CCC(CC)N(CCOC)C(=O)c1cc2cc(C)ccc2[nH]1 ZINC000147228740 DH On-Demand Anodyne TUBB2B 33 44 CCOc1ccc(C(=O)N[C@@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147228759 FF On-Demand Mild ELANE 45 42 CCOc1ccc(C(=O)N[C@@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147228759 FF On-Demand Mild CCR1 50 48 CCOc1ccc(C(=O)N[C@@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147228759 FF On-Demand Mild CELA2A 20 42 CN(C(=O)OC(C)(C)C)[C@@](C)(C(=O)O)c1ccc(-c2ccccc2)cc1 ZINC000147228828 FJ For-Sale Anodyne PAPA1_CARPA 26 40 O=S(=O)(NC1CC1)c1ccccc1NC[C@@H]1CNCCO1 ZINC000147228831 DC For-Sale Anodyne CCR8 42 32 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1C ZINC000147228833 CE On-Demand Anodyne AKR1C2 32 40 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1C ZINC000147228833 CE On-Demand Anodyne G2YM83_BOTF4 65 33 O=C(CBr)c1ccc(Cl)c(C(=O)O)c1 ZINC000147228898 CF For-Sale Anodyne AKR1C2 60 36 O=C(CBr)c1ccc(Cl)c(C(=O)O)c1 ZINC000147228898 CF For-Sale Anodyne AKR1C1 59 36 CCCCCCCCNC(=O)NCC[C@H](C)C(=O)O ZINC000147228923 CF For-Sale Mild FOLH1 25 44 CCCCCCCCNC(=O)NCC[C@H](C)C(=O)O ZINC000147228923 CF For-Sale Mild CPT1A 25 47 CCCCCCCCNC(=O)NCC[C@H](C)C(=O)O ZINC000147228923 CF For-Sale Mild EPHX2 29 54 CCCCCCCCNC(=O)NCC[C@H](C)C(=O)O ZINC000147228923 CF For-Sale Mild ASAH1 88 34 CCCCCCCCNC(=O)NCC[C@H](C)C(=O)O ZINC000147228923 CF For-Sale Mild ACAT 0 42 CCCCCCCCNC(=O)NCC[C@H](C)C(=O)O ZINC000147228923 CF For-Sale Mild NOD1 99 46 CCCCCCCCNC(=O)NCC[C@H](C)C(=O)O ZINC000147228923 CF For-Sale Mild CQSS 54 35 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228926 GI On-Demand Anodyne NPY1R 26 41 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228926 GI On-Demand Anodyne CCKAR 31 45 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228926 GI On-Demand Anodyne CCKBR 34 45 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228926 GI On-Demand Anodyne EPHX2 16 41 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228926 GI On-Demand Anodyne KCNK3 73 35 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147228926 GI On-Demand Anodyne KCNK9 47 34 CC(C)[C@@H](NC(=O)c1ccccc1F)C(=O)N1CCC(C#N)CC1 ZINC000147228959 EE On-Demand Mild ELANE 43 39 CC(C)[C@@H](NC(=O)c1ccccc1F)C(=O)N1CCC(C#N)CC1 ZINC000147228959 EE On-Demand Mild CCR1 61 48 CCCNc1ncc(C)c(Nc2ccc(C#N)cc2F)n1 ZINC000147229009 CG For-Sale Mild SYK 15 42 CC(C)(NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147229041 CE On-Demand Anodyne E3UJZ5_SPOLI 42 42 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne CCKAR 25 49 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne CCR3 15 45 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne MTNR1A 52 48 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne MTNR1B 52 49 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne ROCK2 20 44 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne CCKBR 0 49 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne EPHX2 15 45 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne FLT4 18 41 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne TAAR1 34 42 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne AKR1C3 18 43 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne AKR1C2 43 36 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne ACAT 0 52 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne KCNK3 48 36 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne KCNK9 45 36 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne PDS 40 39 CC[C@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229044 CE For-Sale Anodyne PARP10 0 40 O=S(=O)(NC1CC1)c1ccccc1NC[C@H]1CNCCO1 ZINC000147229048 DC For-Sale Anodyne CCR8 42 32 CCOC(=O)c1cn(C(C)(C)C)c2nc(NC(=O)c3ccc(C)cc3)ccc12 ZINC000147229056 GJ For-Sale Anodyne MAP3K5 68 44 CC(C)N1c2ccccc2[C@H](c2ccc(F)cc2)[C@@H]1/C=C/[C@@H](O)C[C@@H](O)CC(=O)O ZINC000147229093 HH Annotated Anodyne HMGCR 177 48 CCCCCCCCNC(=O)N[C@H]1C=C[C@@H](C(=O)O)C1 ZINC000147229098 CF For-Sale Mild EPHX2 30 51 CCCCCCCCNC(=O)N[C@H]1C=C[C@@H](C(=O)O)C1 ZINC000147229098 CF For-Sale Mild ASAH1 74 33 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229105 GI On-Demand Anodyne NPY1R 26 41 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229105 GI On-Demand Anodyne CCKAR 31 45 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229105 GI On-Demand Anodyne CCKBR 34 45 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229105 GI On-Demand Anodyne EPHX2 16 41 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229105 GI On-Demand Anodyne KCNK3 73 35 CCOC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229105 GI On-Demand Anodyne KCNK9 47 34 CSCC[C@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147229172 GE On-Demand Mild F2 41 47 CSCC[C@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147229172 GE On-Demand Mild MMP13 15 41 CSCC[C@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147229172 GE On-Demand Mild TRY2_BOVIN 72 36 CSCC[C@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147229172 GE On-Demand Mild ST14 93 37 CSCC[C@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147229172 GE On-Demand Mild TMPRSS6 52 33 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne CCKAR 25 49 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne CCR3 15 45 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne MTNR1A 52 48 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne MTNR1B 52 49 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne ROCK2 20 44 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne CCKBR 0 49 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne EPHX2 15 45 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne FLT4 18 41 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne TAAR1 34 42 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne AKR1C3 18 43 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne AKR1C2 43 36 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne ACAT 0 52 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne KCNK3 48 36 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne KCNK9 45 36 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne PDS 40 39 CC[C@@H](CNC(=O)Nc1cccc(OC)c1)CC(=O)O ZINC000147229209 CE For-Sale Anodyne PARP10 0 40 N#CCCOC(=O)c1cccs1 ZINC000147229214 AD For-Sale Mild CTSC 34 40 CC(C)(NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147229243 BD For-Sale Anodyne FFAR1 0 43 CC(C)(NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147229243 BD For-Sale Anodyne NAMPT 22 41 CC(C)(NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147229243 BD For-Sale Anodyne GPR88 0 43 CCc1nc(CN(C)C(=O)NCCN2CCN(Cc3ccccc3)CC2)cs1 ZINC000147229244 HF On-Demand Anodyne HTR1A 21 45 CCc1nc(CN(C)C(=O)NCCN2CCN(Cc3ccccc3)CC2)cs1 ZINC000147229244 HF On-Demand Anodyne DRD3 23 41 CCc1nc(CN(C)C(=O)NCCN2CCN(Cc3ccccc3)CC2)cs1 ZINC000147229244 HF On-Demand Anodyne SIGMAR1 25 42 CNc1cn2ccnc2c(Nc2ccc(C#N)cc2F)n1 ZINC000147229249 CF For-Sale Mild HIVRT 0 48 CCCCO[C@@H](C)C(=O)NCCc1nccn1Cc1ccccc1 ZINC000147229251 EF On-Demand Anodyne AGTR1B 57 33 CCCCO[C@@H](C)C(=O)NCCc1nccn1Cc1ccccc1 ZINC000147229251 EF On-Demand Anodyne CAPN2 62 34 CCC1CCN(C(=O)c2ccccc2Cc2ccccc2)CC1 ZINC000147229262 DJ On-Demand Anodyne CHRM2 26 44 CCC1CCN(C(=O)c2ccccc2Cc2ccccc2)CC1 ZINC000147229262 DJ On-Demand Anodyne ACHE 18 40 CCC1CCN(C(=O)c2ccccc2Cc2ccccc2)CC1 ZINC000147229262 DJ On-Demand Anodyne GRIN2B 79 46 CCC1CCN(C(=O)c2ccccc2Cc2ccccc2)CC1 ZINC000147229262 DJ On-Demand Anodyne SIGMAR1 28 40 CCC1CCN(C(=O)c2ccccc2Cc2ccccc2)CC1 ZINC000147229262 DJ On-Demand Anodyne CCR3 44 39 CCC1CCN(C(=O)c2ccccc2Cc2ccccc2)CC1 ZINC000147229262 DJ On-Demand Anodyne CCR5 22 43 CCC1CCN(C(=O)c2ccccc2Cc2ccccc2)CC1 ZINC000147229262 DJ On-Demand Anodyne AMP1_PLAFQ 16 40 CCC1CCN(C(=O)c2ccccc2Cc2ccccc2)CC1 ZINC000147229262 DJ On-Demand Anodyne L3MBTL3 54 53 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229283 GI On-Demand Anodyne NPY1R 26 41 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229283 GI On-Demand Anodyne CCKAR 31 45 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229283 GI On-Demand Anodyne CCKBR 34 45 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229283 GI On-Demand Anodyne EPHX2 16 41 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229283 GI On-Demand Anodyne KCNK3 73 35 CCOC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147229283 GI On-Demand Anodyne KCNK9 47 34 CCCCCCCCNC(=O)N[C@@H]1C=C[C@@H](C(=O)O)C1 ZINC000147229287 CF For-Sale Mild EPHX2 30 51 CCCCCCCCNC(=O)N[C@@H]1C=C[C@@H](C(=O)O)C1 ZINC000147229287 CF For-Sale Mild ASAH1 74 33 CSCC[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147229382 GE On-Demand Mild F2 41 47 CSCC[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147229382 GE On-Demand Mild MMP13 15 41 CSCC[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147229382 GE On-Demand Mild TRY2_BOVIN 72 36 CSCC[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147229382 GE On-Demand Mild ST14 93 37 CSCC[C@@H](NS(=O)(=O)c1ccc(C)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147229382 GE On-Demand Mild TMPRSS6 52 33 CC(C)(NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147229383 BD For-Sale Anodyne FFAR1 0 43 CC(C)(NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147229383 BD For-Sale Anodyne NAMPT 22 41 CC(C)(NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147229383 BD For-Sale Anodyne GPR88 0 43 CCCCO[C@H](C)C(=O)NCCc1nccn1Cc1ccccc1 ZINC000147229384 EF On-Demand Anodyne AGTR1B 57 33 CCCCO[C@H](C)C(=O)NCCc1nccn1Cc1ccccc1 ZINC000147229384 EF On-Demand Anodyne CAPN2 62 34 CC[C@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229474 CE For-Sale Anodyne ADRB1 15 40 CC[C@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229474 CE For-Sale Anodyne CA1 43 35 CC[C@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229474 CE For-Sale Anodyne MTNR1B 33 40 CC[C@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229474 CE For-Sale Anodyne NPY5R 16 41 CC[C@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229474 CE For-Sale Anodyne F7 18 43 CC[C@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229474 CE For-Sale Anodyne ACR 42 41 CC[C@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229474 CE For-Sale Anodyne CA12 20 44 CC[C@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229474 CE For-Sale Anodyne CA9 21 44 CC[C@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229474 CE For-Sale Anodyne AKR1C2 40 38 CC[C@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229474 CE For-Sale Anodyne PQSD 0 40 CCCCCCCCNC(=O)N[C@H]1C=C[C@H](C(=O)O)C1 ZINC000147229487 CF For-Sale Mild EPHX2 30 51 CCCCCCCCNC(=O)N[C@H]1C=C[C@H](C(=O)O)C1 ZINC000147229487 CF For-Sale Mild ASAH1 74 33 CC(C)(NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147229586 BD For-Sale Anodyne FFAR1 0 43 CC(C)(NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147229586 BD For-Sale Anodyne NAMPT 22 41 CC(C)(NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147229586 BD For-Sale Anodyne GPR88 0 43 O=S(=O)(c1ccccc1C(F)(F)F)N1CCC(CBr)CC1 ZINC000147229632 GH For-Sale Reactive EPHX2 31 45 O=S(=O)(c1ccccc1C(F)(F)F)N1CCC(CBr)CC1 ZINC000147229632 GH For-Sale Reactive RBP4 64 37 O=S(=O)(c1ccccc1C(F)(F)F)N1CCC(CBr)CC1 ZINC000147229632 GH For-Sale Reactive SFRP1 103 43 O=S(=O)(c1ccccc1C(F)(F)F)N1CCC(CBr)CC1 ZINC000147229632 GH For-Sale Reactive WNT3 62 33 CCCCCCCCNC(=O)N[C@@H]1C=C[C@H](C(=O)O)C1 ZINC000147229679 CF For-Sale Mild EPHX2 30 51 CCCCCCCCNC(=O)N[C@@H]1C=C[C@H](C(=O)O)C1 ZINC000147229679 CF For-Sale Mild ASAH1 74 33 CCOC[C@H](C)NC(=O)Nc1cccc(C)c1C(=O)N1CCCC1 ZINC000147229682 EF On-Demand Anodyne KCNQ2 42 33 CCCC[C@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229683 DD On-Demand Anodyne PPARD 17 41 CCCC[C@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229683 DD On-Demand Anodyne MTNR1A 41 41 CCCC[C@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229683 DD On-Demand Anodyne MTNR1B 29 43 CCCC[C@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229683 DD On-Demand Anodyne GRIA1 64 31 CCCC[C@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229683 DD On-Demand Anodyne PCSK5 58 36 CCCC[C@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229683 DD On-Demand Anodyne FURIN 69 36 CCCC[C@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229683 DD On-Demand Anodyne MT-ND1 17 45 CCCC[C@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229683 DD On-Demand Anodyne POLG_WNV 54 39 CC[C@@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229687 CE For-Sale Anodyne ADRB1 15 40 CC[C@@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229687 CE For-Sale Anodyne CA1 43 35 CC[C@@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229687 CE For-Sale Anodyne MTNR1B 33 40 CC[C@@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229687 CE For-Sale Anodyne NPY5R 16 41 CC[C@@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229687 CE For-Sale Anodyne F7 18 43 CC[C@@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229687 CE For-Sale Anodyne ACR 42 41 CC[C@@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229687 CE For-Sale Anodyne CA12 20 44 CC[C@@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229687 CE For-Sale Anodyne CA9 21 44 CC[C@@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229687 CE For-Sale Anodyne AKR1C2 40 38 CC[C@@H](CNC(=O)Nc1ccc(OC)cc1)CC(=O)O ZINC000147229687 CE For-Sale Anodyne PQSD 0 40 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1OCC(N)=O ZINC000147229712 FC On-Demand Anodyne QRFPR 40 33 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1OCC(N)=O ZINC000147229712 FC On-Demand Anodyne ENPP1 54 31 COc1ccc(CNC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147229749 FE On-Demand Anodyne TSHR 40 29 COc1ccc(CNC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147229749 FE On-Demand Anodyne MTNR1B 23 44 CC(C)(NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147229809 BD For-Sale Anodyne FFAR1 0 43 CC(C)(NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147229809 BD For-Sale Anodyne NAMPT 22 41 CC(C)(NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147229809 BD For-Sale Anodyne GPR88 0 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229881 DD On-Demand Anodyne PPARD 17 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229881 DD On-Demand Anodyne MTNR1A 41 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229881 DD On-Demand Anodyne MTNR1B 29 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229881 DD On-Demand Anodyne GRIA1 64 31 CCCC[C@@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229881 DD On-Demand Anodyne PCSK5 58 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229881 DD On-Demand Anodyne FURIN 69 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229881 DD On-Demand Anodyne MT-ND1 17 45 CCCC[C@@H](NC(N)=O)C(=O)NCc1cc(OC)ccc1OC ZINC000147229881 DD On-Demand Anodyne POLG_WNV 54 39 CC[C@H](CNC(=O)Nc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147229886 CE For-Sale Bother CACNA1D 56 33 CC[C@H](CNC(=O)Nc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147229886 CE For-Sale Bother DDX3X 0 50 CC[C@H](CNC(=O)Nc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147229886 CE For-Sale Bother OSIGBA0132E09-OSIGBA0108L24.11 0 41 CCCCCCCCNC(=O)NCC1(CC(=O)O)CCC1 ZINC000147229896 CG For-Sale Mild CACNA2D1 0 40 CCCCCCCCNC(=O)NCC1(CC(=O)O)CCC1 ZINC000147229896 CG For-Sale Mild CPT1A 35 44 CCCCCCCCNC(=O)NCC1(CC(=O)O)CCC1 ZINC000147229896 CG For-Sale Mild EPHX2 25 47 CCCCCCCCNC(=O)NCC1(CC(=O)O)CCC1 ZINC000147229896 CG For-Sale Mild ASAH1 78 32 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1OCC(N)=O ZINC000147229907 FC On-Demand Anodyne QRFPR 40 33 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1OCC(N)=O ZINC000147229907 FC On-Demand Anodyne ENPP1 54 31 Nc1nc2c3ccccc3nc(Cc3ccc(O)cc3O)n2n1 ZINC000147229926 DD Annotated Anodyne HSP90AB1 20 56 COc1ccc(CNC(C)=O)cc1S(=O)(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147229945 FE On-Demand Anodyne TSHR 40 29 COc1ccc(CNC(C)=O)cc1S(=O)(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147229945 FE On-Demand Anodyne MTNR1B 23 44 CN1CCO[C@H](COc2ccc(Br)cc2S(N)(=O)=O)C1 ZINC000147229967 FC For-Sale Anodyne EPHA2 25 49 COCC(=O)N1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147229971 EB On-Demand Anodyne HTR1D 16 42 COCC(=O)N1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147229971 EB On-Demand Anodyne HTR1B 19 42 COCC(=O)N1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147229971 EB On-Demand Anodyne CPT1A 53 42 COCC(=O)N1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147229971 EB On-Demand Anodyne PLA2G4B 47 36 CCCCCCCCNC(=O)NC1(C(=O)O)CCOCC1 ZINC000147230088 DE For-Sale Mild EPHX2 34 49 CCCCCCCCNC(=O)NC1(C(=O)O)CCOCC1 ZINC000147230088 DE For-Sale Mild ASAH1 50 35 CCCCCCCCNC(=O)NC1(C(=O)O)CCOCC1 ZINC000147230088 DE For-Sale Mild ACAT 0 40 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1OCC(=O)NC1CC1 ZINC000147230099 HC On-Demand Anodyne ENPP1 54 31 CC[C@@H](CNC(=O)Nc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147230101 CE For-Sale Bother CACNA1D 56 33 CC[C@@H](CNC(=O)Nc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147230101 CE For-Sale Bother DDX3X 0 50 CC[C@@H](CNC(=O)Nc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147230101 CE For-Sale Bother OSIGBA0132E09-OSIGBA0108L24.11 0 41 COc1ccc(CNC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147230112 FE On-Demand Anodyne TSHR 40 29 COc1ccc(CNC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147230112 FE On-Demand Anodyne MTNR1B 23 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccccc2OC(F)F)CC1 ZINC000147230117 HD On-Demand Anodyne GHRHR 41 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccccc2OC(F)F)CC1 ZINC000147230117 HD On-Demand Anodyne P2RY12 197 39 COc1ccc(C(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147230136 EE On-Demand Mild CHRM2 21 40 COc1ccc(C(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147230136 EE On-Demand Mild ELANE 53 49 COc1ccc(C(=O)N[C@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147230136 EE On-Demand Mild CCR1 49 51 NC(=O)c1ccc(OCC(=O)Nc2cccc(C(=O)N3CCOCC3)c2)cc1 ZINC000147230164 GD On-Demand Anodyne EPHX2 32 53 NC(=O)c1ccc(OCC(=O)Nc2cccc(C(=O)N3CCOCC3)c2)cc1 ZINC000147230164 GD On-Demand Anodyne MCHR1 18 48 NC(=O)c1ccc(OCC(=O)Nc2cccc(C(=O)N3CCOCC3)c2)cc1 ZINC000147230164 GD On-Demand Anodyne BTK 40 37 NC(=O)c1ccc(OCC(=O)Nc2cccc(C(=O)N3CCOCC3)c2)cc1 ZINC000147230164 GD On-Demand Anodyne HIF1A 32 48 CN1CCO[C@@H](COc2ccc(Br)cc2S(N)(=O)=O)C1 ZINC000147230165 FC For-Sale Anodyne EPHA2 25 49 CCCCCCCCNC(=O)NCC1(C(=O)O)CCCC1 ZINC000147230278 CG For-Sale Mild CPT1A 0 40 CCCCCCCCNC(=O)NCC1(C(=O)O)CCCC1 ZINC000147230278 CG For-Sale Mild EPHX2 27 47 CCCCCCCCNC(=O)NCC1(C(=O)O)CCCC1 ZINC000147230278 CG For-Sale Mild ASAH1 84 33 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1OCC(=O)NC1CC1 ZINC000147230306 HC On-Demand Anodyne ENPP1 54 31 COc1ccc(CNC(C)=O)cc1S(=O)(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147230314 FE On-Demand Anodyne TSHR 40 29 COc1ccc(CNC(C)=O)cc1S(=O)(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147230314 FE On-Demand Anodyne MTNR1B 23 44 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCC[C@@H](O)C1 ZINC000147230319 EE For-Sale Anodyne SLC6A1 43 31 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCC[C@@H](O)C1 ZINC000147230319 EE For-Sale Anodyne ADORA1 17 41 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCC[C@@H](O)C1 ZINC000147230319 EE For-Sale Anodyne P2RY12 107 47 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCC[C@@H](O)C1 ZINC000147230319 EE For-Sale Anodyne JUN 18 49 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCC[C@@H](O)C1 ZINC000147230319 EE For-Sale Anodyne ADORA3 22 41 COc1ccc(C(=O)N[C@@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147230322 EE On-Demand Mild CHRM2 21 40 COc1ccc(C(=O)N[C@@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147230322 EE On-Demand Mild ELANE 53 49 COc1ccc(C(=O)N[C@@H](C(=O)N2CCC(C#N)CC2)C(C)C)cc1 ZINC000147230322 EE On-Demand Mild CCR1 49 51 CC[C@H](CNC(=O)NC1CCCCC1)CC(=O)O ZINC000147230328 CE For-Sale Anodyne EPHX2 19 44 CC(C)(C)C[C@H]1N[C@@H](C(=O)NC2CN(CC(C)(C)O)C2)[C@H](c2cccc(Cl)c2F)[C@@]12C(=O)Nc1cc(Cl)ccc12 ZINC000147230357 KI Annotated Anodyne MDM2 105 71 CCCNC(=O)c1cccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147230423 GF On-Demand Anodyne MAPK14 16 41 CCCNC(=O)c1cccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147230423 GF On-Demand Anodyne EPHX2 27 42 CCCNC(=O)c1cccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147230423 GF On-Demand Anodyne KCNK3 24 44 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCC[C@H](O)C1 ZINC000147230461 EE For-Sale Anodyne SLC6A1 43 31 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCC[C@H](O)C1 ZINC000147230461 EE For-Sale Anodyne ADORA1 17 41 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCC[C@H](O)C1 ZINC000147230461 EE For-Sale Anodyne P2RY12 107 47 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCC[C@H](O)C1 ZINC000147230461 EE For-Sale Anodyne JUN 18 49 CCOC(=O)c1cnc(-c2ccccc2)nc1N1CCC[C@H](O)C1 ZINC000147230461 EE For-Sale Anodyne ADORA3 22 41 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1OCc1cccnc1 ZINC000147230470 GE On-Demand Anodyne PDE4A 26 40 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1OCc1cccnc1 ZINC000147230470 GE On-Demand Anodyne ENPP1 47 34 CCCCCCCCNC(=O)N[C@H](C(=O)O)[C@@H](C)O ZINC000147230476 CD For-Sale Mild CPT1A 51 55 CCCCCCCCNC(=O)N[C@H](C(=O)O)[C@@H](C)O ZINC000147230476 CD For-Sale Mild EPHX2 59 48 CCCCCCCCNC(=O)N[C@H](C(=O)O)[C@@H](C)O ZINC000147230476 CD For-Sale Mild ASAH1 82 35 CCCCCCCCNC(=O)N[C@H](C(=O)O)[C@@H](C)O ZINC000147230476 CD For-Sale Mild NOD1 85 41 CCCCCCCCNC(=O)N[C@H](C(=O)O)[C@@H](C)O ZINC000147230476 CD For-Sale Mild CQSS 54 37 Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147230517 FD On-Demand Mild FKBP1A 18 43 Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147230517 FD On-Demand Mild MMP13 28 41 Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147230517 FD On-Demand Mild ITGA4 41 43 Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147230517 FD On-Demand Mild CAPNS1 22 45 Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147230517 FD On-Demand Mild MMP3 26 44 Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147230517 FD On-Demand Mild MMP7 38 41 Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147230517 FD On-Demand Mild MMP1 30 44 Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147230517 FD On-Demand Mild SFRP1 44 33 Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N2CCC(C#N)CC2)cc1 ZINC000147230517 FD On-Demand Mild WNT3 54 34 CC[C@@H](CNC(=O)NC1CCCCC1)CC(=O)O ZINC000147230534 CE For-Sale Anodyne EPHX2 19 44 O=C1CC[C@@]2(O)[C@H]3Cc4ccc(C(=O)NCCc5ccc(-c6c[nH]c(=O)[nH]c6=O)cc5)c(O)c4[C@@]2(CCN3CCc2ccccc2)C1 ZINC000147230535 KG Annotated Anodyne OPRM1 49 47 O=C1CC[C@@]2(O)[C@H]3Cc4ccc(C(=O)NCCc5ccc(-c6c[nH]c(=O)[nH]c6=O)cc5)c(O)c4[C@@]2(CCN3CCc2ccccc2)C1 ZINC000147230535 KG Annotated Anodyne OPRD1 53 47 O=C1CC[C@@]2(O)[C@H]3Cc4ccc(C(=O)NCCc5ccc(-c6c[nH]c(=O)[nH]c6=O)cc5)c(O)c4[C@@]2(CCN3CCc2ccccc2)C1 ZINC000147230535 KG Annotated Anodyne OPRK1 56 47 CN(C)C(=O)NCCNc1ccnc2cc(Cl)ccc12 ZINC000147230552 CF On-Demand Anodyne RBP_CHICK 0 43 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)Cc3cccc(F)c3)c(F)c2)CC1 ZINC000147230613 JH Annotated Clean SSTR3 40 37 CCCCCCCCNC(=O)N[C@@H](C(=O)O)[C@@H](C)O ZINC000147230663 CD For-Sale Mild CPT1A 51 55 CCCCCCCCNC(=O)N[C@@H](C(=O)O)[C@@H](C)O ZINC000147230663 CD For-Sale Mild EPHX2 59 48 CCCCCCCCNC(=O)N[C@@H](C(=O)O)[C@@H](C)O ZINC000147230663 CD For-Sale Mild ASAH1 82 35 CCCCCCCCNC(=O)N[C@@H](C(=O)O)[C@@H](C)O ZINC000147230663 CD For-Sale Mild NOD1 85 41 CCCCCCCCNC(=O)N[C@@H](C(=O)O)[C@@H](C)O ZINC000147230663 CD For-Sale Mild CQSS 54 37 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1OCc1cccnc1 ZINC000147230671 GE On-Demand Anodyne PDE4A 26 40 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1OCc1cccnc1 ZINC000147230671 GE On-Demand Anodyne ENPP1 47 34 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCC(CBr)CC1 ZINC000147230673 GH For-Sale Reactive HSD11B1 16 53 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCC(CBr)CC1 ZINC000147230673 GH For-Sale Reactive CACNA1B 63 44 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCC(CBr)CC1 ZINC000147230673 GH For-Sale Reactive BDKRB1 22 40 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCC(CBr)CC1 ZINC000147230673 GH For-Sale Reactive EPHX2 17 44 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCC(CBr)CC1 ZINC000147230673 GH For-Sale Reactive PKM 36 56 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCC(CBr)CC1 ZINC000147230673 GH For-Sale Reactive AKR1C3 54 37 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCC(CBr)CC1 ZINC000147230673 GH For-Sale Reactive SFRP1 28 40 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCC(CBr)CC1 ZINC000147230673 GH For-Sale Reactive RHOA 0 42 COc1nc(N)nc(Oc2ccc3ccccc3c2)n1 ZINC000147230686 CE For-Sale Anodyne CYP2A5 0 52 N#Cc1ccc(Nc2cc(N)ncn2)c(F)c1 ZINC000147230697 BD For-Sale Mild CDC7 18 41 CC[C@H](CNC(=O)Oc1ccccc1)CC(=O)O ZINC000147230729 CE For-Sale Anodyne FAAH 27 47 CC[C@H](CNC(=O)Oc1ccccc1)CC(=O)O ZINC000147230729 CE For-Sale Anodyne CAPN2 57 32 CC[C@H](CNC(=O)Oc1ccccc1)CC(=O)O ZINC000147230729 CE For-Sale Anodyne ACE2 43 35 CC[C@H](CNC(=O)Oc1ccccc1)CC(=O)O ZINC000147230729 CE For-Sale Anodyne PDS 71 41 CC(C)[C@H](NC(=O)c1ccccc1Br)C(=O)N1CCC(C#N)CC1 ZINC000147230768 GF On-Demand Mild CCR1 69 52 CCCNC(=O)c1cccc(NC(=O)NCc2ccc(-n3ccnc3C)c(F)c2)c1 ZINC000147230778 HH On-Demand Anodyne ROCK2 28 41 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne FOLH1 52 36 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne MME 27 46 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne ANPEP 42 43 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne RNPEP 23 42 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne CCKAR 41 47 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne CTSK 26 40 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne CTSL 29 44 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne CTSS 24 44 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne CAPN1 39 40 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne CAPN2 55 33 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne FPR1 52 38 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne SLC15A2 0 40 CC(C)C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230805 CF On-Demand Anodyne DAC 51 40 CN(C)C(=O)NCCNc1nc(Cl)nc(-n2ccnc2)n1 ZINC000147230823 DC For-Sale Anodyne NOS2 56 32 CCCCCCCCNC(=O)N[C@H](C(=O)O)[C@H](C)O ZINC000147230844 CD For-Sale Mild CPT1A 51 55 CCCCCCCCNC(=O)N[C@H](C(=O)O)[C@H](C)O ZINC000147230844 CD For-Sale Mild EPHX2 59 48 CCCCCCCCNC(=O)N[C@H](C(=O)O)[C@H](C)O ZINC000147230844 CD For-Sale Mild ASAH1 82 35 CCCCCCCCNC(=O)N[C@H](C(=O)O)[C@H](C)O ZINC000147230844 CD For-Sale Mild NOD1 85 41 CCCCCCCCNC(=O)N[C@H](C(=O)O)[C@H](C)O ZINC000147230844 CD For-Sale Mild CQSS 54 37 NC(=O)c1ccc(OCC(=O)N2CCC(NC(=O)c3ccncc3)CC2)cc1 ZINC000147230864 GC On-Demand Anodyne PLG 19 42 NC(=O)c1ccc(OCC(=O)N2CCC(NC(=O)c3ccncc3)CC2)cc1 ZINC000147230864 GC On-Demand Anodyne SSTR5 43 36 NC(=O)c1ccc(OCC(=O)N2CCC(NC(=O)c3ccncc3)CC2)cc1 ZINC000147230864 GC On-Demand Anodyne CPT1A 41 45 NC(=O)c1ccc(OCC(=O)N2CCC(NC(=O)c3ccncc3)CC2)cc1 ZINC000147230864 GC On-Demand Anodyne C3AR1 40 35 NC(=O)c1ccc(OCC(=O)N2CCC(NC(=O)c3ccncc3)CC2)cc1 ZINC000147230864 GC On-Demand Anodyne SLC6A5 40 45 NC(=O)c1ccc(OCC(=O)N2CCC(NC(=O)c3ccncc3)CC2)cc1 ZINC000147230864 GC On-Demand Anodyne EPHX2 27 42 NC(=O)c1ccc(OCC(=O)N2CCC(NC(=O)c3ccncc3)CC2)cc1 ZINC000147230864 GC On-Demand Anodyne PLAU 28 44 NC(=O)c1ccc(OCC(=O)N2CCC(NC(=O)c3ccncc3)CC2)cc1 ZINC000147230864 GC On-Demand Anodyne ST14 32 43 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1OCc1ccncc1 ZINC000147230878 GE On-Demand Anodyne PDE4A 31 44 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1OCc1ccncc1 ZINC000147230878 GE On-Demand Anodyne ENPP1 56 33 CC[C@@H](CNC(=O)Oc1ccccc1)CC(=O)O ZINC000147230919 CE For-Sale Anodyne FAAH 27 47 CC[C@@H](CNC(=O)Oc1ccccc1)CC(=O)O ZINC000147230919 CE For-Sale Anodyne CAPN2 57 32 CC[C@@H](CNC(=O)Oc1ccccc1)CC(=O)O ZINC000147230919 CE For-Sale Anodyne ACE2 43 35 CC[C@@H](CNC(=O)Oc1ccccc1)CC(=O)O ZINC000147230919 CE For-Sale Anodyne PDS 71 41 CC(C)[C@@H](NC(=O)c1ccccc1Br)C(=O)N1CCC(C#N)CC1 ZINC000147230930 GF On-Demand Mild CCR1 69 52 CC(C)C[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230941 CF On-Demand Anodyne FOLH1 52 36 CC(C)C[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230941 CF On-Demand Anodyne CCKAR 41 47 CC(C)C[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147230941 CF On-Demand Anodyne SLC15A2 0 40 O=C(Cl)[C@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147230965 CI For-Sale Reactive CHRM2 20 42 O=C(Cl)[C@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147230965 CI For-Sale Reactive CHRM1 23 42 O=C(Cl)[C@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147230965 CI For-Sale Reactive CHRM4 18 41 O=C(Cl)[C@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147230965 CI For-Sale Reactive CHRM5 19 41 O=C(Cl)[C@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147230965 CI For-Sale Reactive CHRM3 36 42 O=C(Cl)[C@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147230965 CI For-Sale Reactive AMY2 58 40 N#Cc1ccc(Nc2nc(N)ncc2F)c(F)c1 ZINC000147230972 BD For-Sale Mild SYK 15 48 CCCc1ccc(S(=O)(=O)N2CCC(CBr)CC2)cc1 ZINC000147230993 FG For-Sale Reactive TGM2 42 37 CCCCCCCCNC(=O)N[C@@H](C(=O)O)[C@H](C)O ZINC000147231038 CD For-Sale Mild CPT1A 51 55 CCCCCCCCNC(=O)N[C@@H](C(=O)O)[C@H](C)O ZINC000147231038 CD For-Sale Mild EPHX2 59 48 CCCCCCCCNC(=O)N[C@@H](C(=O)O)[C@H](C)O ZINC000147231038 CD For-Sale Mild ASAH1 82 35 CCCCCCCCNC(=O)N[C@@H](C(=O)O)[C@H](C)O ZINC000147231038 CD For-Sale Mild NOD1 85 41 CCCCCCCCNC(=O)N[C@@H](C(=O)O)[C@H](C)O ZINC000147231038 CD For-Sale Mild CQSS 54 37 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1OCc1ccncc1 ZINC000147231040 GE On-Demand Anodyne PDE4A 31 44 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1OCc1ccncc1 ZINC000147231040 GE On-Demand Anodyne ENPP1 56 33 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(CN3CCOC3=O)cc1)C2 ZINC000147231045 GF On-Demand Anodyne ROCK2 30 49 CCCNC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147231110 GI On-Demand Anodyne KCNK3 88 38 CCCNC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147231110 GI On-Demand Anodyne KCNK9 49 36 O=C(Cl)[C@@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147231151 CI For-Sale Reactive CHRM2 20 42 O=C(Cl)[C@@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147231151 CI For-Sale Reactive CHRM1 23 42 O=C(Cl)[C@@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147231151 CI For-Sale Reactive CHRM4 18 41 O=C(Cl)[C@@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147231151 CI For-Sale Reactive CHRM5 19 41 O=C(Cl)[C@@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147231151 CI For-Sale Reactive CHRM3 36 42 O=C(Cl)[C@@](Cl)(c1ccccc1)C1CCCCC1 ZINC000147231151 CI For-Sale Reactive AMY2 58 40 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne ACE 41 45 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne FOLH1 52 36 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne MME 62 49 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne ANPEP 50 42 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne EDNRB 49 60 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne RNPEP 25 45 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne CTSB 24 42 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne RIR1_HHV11 46 30 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne PLD1 15 40 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne CAPNS1 58 36 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne CAPN1 76 45 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne CAPN2 93 39 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne ACE2 65 39 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne LAP3 21 45 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne FPR1 81 42 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne NPR 77 38 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne AMP1_PLAFQ 27 45 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne AMPX_VIBPR 0 45 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne SLC15A2 0 44 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne Q9N6S8_PLAFA 41 32 CC(C)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231162 CE For-Sale Anodyne GPR88 0 50 NS(=O)(=O)c1cc(F)ccc1OCC(=O)NC1CCCC1 ZINC000147231190 DC For-Sale Anodyne LUXN 0 42 N#CC1CCN(C(=O)CCCNC(=O)c2ccc(Cl)cc2)CC1 ZINC000147231209 EF On-Demand Mild PREP 16 43 N#CC1CCN(C(=O)CCCNC(=O)c2ccc(Cl)cc2)CC1 ZINC000147231209 EF On-Demand Mild CACNA1G 15 40 CCCCCCCCNC(=O)N1C[C@H](O)C[C@@H]1C(=O)O ZINC000147231219 CD For-Sale Mild EPHX2 33 42 CCCCCCCCNC(=O)N1C[C@H](O)C[C@@H]1C(=O)O ZINC000147231219 CD For-Sale Mild ASAH1 104 41 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)Cc3ccc(Cl)cc3)c(F)c2)CC1 ZINC000147231256 JI Annotated Clean SSTR3 55 38 CCCNC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147231277 GI On-Demand Anodyne KCNK3 88 38 CCCNC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147231277 GI On-Demand Anodyne KCNK9 49 36 O=C(c1cccc2c1OCCN2)N1CCN2CCC[C@@H]2C1 ZINC000147231296 CD For-Sale Anodyne HRH3 18 41 O=C(c1cccc2c1OCCN2)N1CCN2CCC[C@@H]2C1 ZINC000147231296 CD For-Sale Anodyne L3MBTL1 0 42 O=C(c1cccc2c1OCCN2)N1CCN2CCC[C@@H]2C1 ZINC000147231296 CD For-Sale Anodyne L3MBTL3 76 42 O=C(c1cccc2c1OCCN2)N1CCN2CCC[C@@H]2C1 ZINC000147231296 CD For-Sale Anodyne TP53BP1 0 42 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](c1ccccc1)c1nccn1C ZINC000147231297 FH On-Demand Anodyne ACE2 55 35 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne ACE 41 45 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne FOLH1 52 36 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne MME 62 49 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne ANPEP 50 42 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne EDNRB 49 60 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne RNPEP 25 45 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne CTSB 24 42 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne RIR1_HHV11 46 30 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne PLD1 15 40 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne CAPNS1 58 36 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne CAPN1 76 45 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne CAPN2 93 39 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne ACE2 65 39 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne LAP3 21 45 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne FPR1 81 42 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne NPR 77 38 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne AMP1_PLAFQ 27 45 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne AMPX_VIBPR 0 45 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne SLC15A2 0 44 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne Q9N6S8_PLAFA 41 32 CC(C)C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231328 CE For-Sale Anodyne GPR88 0 50 CCCCCCCCNC(=O)N1C[C@@H](O)C[C@@H]1C(=O)O ZINC000147231395 CD For-Sale Mild EPHX2 33 42 CCCCCCCCNC(=O)N1C[C@@H](O)C[C@@H]1C(=O)O ZINC000147231395 CD For-Sale Mild ASAH1 104 41 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](c1ccccc1)c1nccn1C ZINC000147231470 FH On-Demand Anodyne ACE2 55 35 CCCNC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147231472 GI On-Demand Anodyne KCNK3 88 38 CCCNC(=O)c1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147231472 GI On-Demand Anodyne KCNK9 49 36 O=C(c1cccc2c1OCCN2)N1CCN2CCC[C@H]2C1 ZINC000147231479 CD For-Sale Anodyne HRH3 18 41 O=C(c1cccc2c1OCCN2)N1CCN2CCC[C@H]2C1 ZINC000147231479 CD For-Sale Anodyne L3MBTL1 0 42 O=C(c1cccc2c1OCCN2)N1CCN2CCC[C@H]2C1 ZINC000147231479 CD For-Sale Anodyne L3MBTL3 76 42 O=C(c1cccc2c1OCCN2)N1CCN2CCC[C@H]2C1 ZINC000147231479 CD For-Sale Anodyne TP53BP1 0 42 CCCCCCCCNC(=O)N1C[C@H](O)C[C@H]1C(=O)O ZINC000147231534 CD For-Sale Mild EPHX2 33 42 CCCCCCCCNC(=O)N1C[C@H](O)C[C@H]1C(=O)O ZINC000147231534 CD For-Sale Mild ASAH1 104 41 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne ACE 41 45 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne FOLH1 52 36 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne MME 62 49 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne ANPEP 50 42 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne EDNRB 49 60 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne RNPEP 25 45 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne CTSB 24 42 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne RIR1_HHV11 46 30 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne PLD1 15 40 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne CAPNS1 58 36 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne CAPN1 76 45 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne CAPN2 93 39 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne ACE2 65 39 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne LAP3 21 45 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne FPR1 81 42 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne NPR 77 38 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne AMP1_PLAFQ 27 45 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne AMPX_VIBPR 0 45 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne SLC15A2 0 44 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne Q9N6S8_PLAFA 41 32 CC(C)C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231537 CE For-Sale Anodyne GPR88 0 50 CN(CCNC(=O)OC(C)(C)C)Cc1ccc(C#N)cn1 ZINC000147231595 CD On-Demand Mild PAPA1_CARPA 43 34 CNc1cc(Oc2ccc3ccccc3c2)nc(C)n1 ZINC000147231601 CH For-Sale Anodyne CYP2A5 0 41 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1nccn1C ZINC000147231627 FH On-Demand Anodyne ACE2 55 35 CC[C@H](CNC(=O)Nc1cccc(F)c1)CC(=O)O ZINC000147231630 CE For-Sale Anodyne KCNK3 29 40 CCCCCCCCNC(=O)N1C[C@@H](O)C[C@H]1C(=O)O ZINC000147231666 CD For-Sale Mild EPHX2 33 42 CCCCCCCCNC(=O)N1C[C@@H](O)C[C@H]1C(=O)O ZINC000147231666 CD For-Sale Mild ASAH1 104 41 CCCNC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147231673 GI On-Demand Anodyne KCNK3 88 38 CCCNC(=O)c1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147231673 GI On-Demand Anodyne KCNK9 49 36 COc1cc(C(=O)N2CCC(C#N)CC2)ccc1OC(C)C ZINC000147231685 DF On-Demand Mild L3MBTL3 52 36 O=c1[nH]c2ccccc2n1C1CCC1 ZINC000147231732 AE For-Sale Anodyne OPRL1 39 64 O=c1[nH]c2ccccc2n1C1CCC1 ZINC000147231732 AE For-Sale Anodyne AKT2 28 42 O=c1[nH]c2ccccc2n1C1CCC1 ZINC000147231732 AE For-Sale Anodyne PLD1 127 50 O=c1[nH]c2ccccc2n1C1CCC1 ZINC000147231732 AE For-Sale Anodyne PLD2 87 50 O=c1[nH]c2ccccc2n1C1CCC1 ZINC000147231732 AE For-Sale Anodyne AKT1 15 49 O=c1[nH]c2ccccc2n1C1CCC1 ZINC000147231732 AE For-Sale Anodyne GRIN3A 0 40 O=c1[nH]c2ccccc2n1C1CCC1 ZINC000147231732 AE For-Sale Anodyne CALCRL 29 46 O=c1[nH]c2ccccc2n1C1CCC1 ZINC000147231732 AE For-Sale Anodyne TNKS 28 40 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne ACE 41 45 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne FOLH1 52 36 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne MME 62 49 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne ANPEP 50 42 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne EDNRB 49 60 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne RNPEP 25 45 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne CTSB 24 42 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne RIR1_HHV11 46 30 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne PLD1 15 40 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne CAPNS1 58 36 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne CAPN1 76 45 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne CAPN2 93 39 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne ACE2 65 39 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne LAP3 21 45 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne FPR1 81 42 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne NPR 77 38 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne AMP1_PLAFQ 27 45 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne AMPX_VIBPR 0 45 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne SLC15A2 0 44 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne Q9N6S8_PLAFA 41 32 CC(C)C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147231737 CE For-Sale Anodyne GPR88 0 50 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](c1ccccc1)c1nccn1C ZINC000147231790 FH On-Demand Anodyne ACE2 55 35 CCCCCCCCNC(=O)N[C@H](CO)C(=O)O ZINC000147231840 CD For-Sale Mild FOLH1 56 49 CCCCCCCCNC(=O)N[C@H](CO)C(=O)O ZINC000147231840 CD For-Sale Mild CPT1A 44 52 CCCCCCCCNC(=O)N[C@H](CO)C(=O)O ZINC000147231840 CD For-Sale Mild EPHX2 25 53 CCCCCCCCNC(=O)N[C@H](CO)C(=O)O ZINC000147231840 CD For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N[C@H](CO)C(=O)O ZINC000147231840 CD For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N[C@H](CO)C(=O)O ZINC000147231840 CD For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N[C@H](CO)C(=O)O ZINC000147231840 CD For-Sale Mild TLR2 0 42 CCCCCCCCNC(=O)N[C@H](CO)C(=O)O ZINC000147231840 CD For-Sale Mild ASAH1 87 36 CCCCCCCCNC(=O)N[C@H](CO)C(=O)O ZINC000147231840 CD For-Sale Mild NOD1 94 45 CCCCCCCCNC(=O)N[C@H](CO)C(=O)O ZINC000147231840 CD For-Sale Mild CQSS 50 31 CCCn1c(SCC(=O)Nc2ccc(C(=O)OCC)cc2)nnc1-c1cccc(C)c1 ZINC000147231844 IJ On-Demand Anodyne ADORA2B 28 42 CCCn1c(SCC(=O)Nc2ccc(C(=O)OCC)cc2)nnc1-c1cccc(C)c1 ZINC000147231844 IJ On-Demand Anodyne ACR 49 34 CCCn1c(SCC(=O)Nc2ccc(C(=O)OCC)cc2)nnc1-c1cccc(C)c1 ZINC000147231844 IJ On-Demand Anodyne ENPP1 65 32 CCCn1c(SCC(=O)Nc2ccc(C(=O)OCC)cc2)nnc1-c1cccc(C)c1 ZINC000147231844 IJ On-Demand Anodyne SLC27A1 27 57 CC[C@@H](CNC(=O)Nc1cccc(F)c1)CC(=O)O ZINC000147231873 CE For-Sale Anodyne KCNK3 29 40 N#CC1CCN(C(=O)CCCc2nc3ccccc3s2)CC1 ZINC000147231886 DG On-Demand Mild PREP 33 42 N#CC1CCN(C(=O)CCCc2nc3ccccc3s2)CC1 ZINC000147231886 DG On-Demand Mild ETHR 63 35 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne CA2 26 58 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne FOLH1 57 39 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne MME 20 43 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne ANPEP 41 40 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne CTSK 23 43 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne CTSL 29 44 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne CA4 17 58 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne CTSS 18 43 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne FPR1 51 38 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne NPR 53 37 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne AMP1_PLAFQ 18 40 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne SLC15A2 0 44 Cc1ccc(C(=O)N[C@@H](CC(C)C)C(=O)O)cc1Br ZINC000147231973 EF On-Demand Anodyne ERAP1 0 42 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccc(F)cc3)c(F)c2)CC1 ZINC000147231978 JG Annotated Clean SSTR3 45 36 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccc(F)cc3)c(F)c2)CC1 ZINC000147231978 JG Annotated Clean RORC 15 44 CCC(CC)N(CCOC)C(=O)[C@H](C)NS(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147232039 HD On-Demand Anodyne IDO1 32 40 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild CPT1A 53 62 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild FAAH 0 41 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild EPHX2 65 54 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild Q6UB75_PIG 0 46 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild ASAH1 88 36 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild ACAT 0 42 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild NOD1 74 40 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild OXER1 46 31 CCCCCCCCNC(=O)N[C@@H](C)CC(=O)O ZINC000147232051 CF For-Sale Mild CQSS 52 35 Cc1ccccc1NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147232081 GG On-Demand Mild PRTN3 50 32 Cc1ccccc1NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147232081 GG On-Demand Mild CCR8 73 36 Cc1ccccc1NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147232081 GG On-Demand Mild SFRP1 66 37 Cc1ccccc1NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147232081 GG On-Demand Mild LIMK2 26 40 Cc1ccccc1NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147232081 GG On-Demand Mild WNT3 43 33 Cc1ccccc1NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147232081 GG On-Demand Mild L3MBTL3 82 40 COC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147232109 DD On-Demand Anodyne CASR 17 44 COC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147232109 DD On-Demand Anodyne HIF1A 20 40 O=C(O)c1cc2ccccc2cc1F ZINC000147232119 AF In-Stock Anodyne DHODH 29 40 O=C(O)c1cc2ccccc2cc1F ZINC000147232119 AF In-Stock Anodyne AKR1C2 60 36 O=C(O)c1cc2ccccc2cc1F ZINC000147232119 AF In-Stock Anodyne AKR1C1 42 48 O=C(O)c1cc2ccccc2cc1F ZINC000147232119 AF In-Stock Anodyne SLC16A3 59 36 CCCOc1ccc(C(=O)NNC(=O)Nc2ccc(=O)n(CC)c2)cc1OC ZINC000147232128 GE On-Demand Reactive ENPP1 62 36 COc1ccc(S(=O)(=O)N(CC(=O)Nc2ccccc2C(=O)NC2CCCCC2)c2ccccc2)cc1 ZINC000147232147 KJ In-Stock Anodyne CNR2 18 41 COc1ccc(S(=O)(=O)N(CC(=O)Nc2ccccc2C(=O)NC2CCCCC2)c2ccccc2)cc1 ZINC000147232147 KJ In-Stock Anodyne BMP1 77 41 COc1ccc(S(=O)(=O)N(CC(=O)Nc2ccccc2C(=O)NC2CCCCC2)c2ccccc2)cc1 ZINC000147232147 KJ In-Stock Anodyne MMP13 58 49 COc1ccc(S(=O)(=O)N(CC(=O)Nc2ccccc2C(=O)NC2CCCCC2)c2ccccc2)cc1 ZINC000147232147 KJ In-Stock Anodyne ADAM17 41 40 COc1ccc(S(=O)(=O)N(CC(=O)Nc2ccccc2C(=O)NC2CCCCC2)c2ccccc2)cc1 ZINC000147232147 KJ In-Stock Anodyne MMP2 37 49 COc1ccc(S(=O)(=O)N(CC(=O)Nc2ccccc2C(=O)NC2CCCCC2)c2ccccc2)cc1 ZINC000147232147 KJ In-Stock Anodyne MMP3 46 49 COc1ccc(S(=O)(=O)N(CC(=O)Nc2ccccc2C(=O)NC2CCCCC2)c2ccccc2)cc1 ZINC000147232147 KJ In-Stock Anodyne MMP8 34 40 COc1ccc(S(=O)(=O)N(CC(=O)Nc2ccccc2C(=O)NC2CCCCC2)c2ccccc2)cc1 ZINC000147232147 KJ In-Stock Anodyne PRTN3 46 35 COc1ccc(S(=O)(=O)N(CC(=O)Nc2ccccc2C(=O)NC2CCCCC2)c2ccccc2)cc1 ZINC000147232147 KJ In-Stock Anodyne MMP9 55 49 COc1ccc(S(=O)(=O)N(CC(=O)Nc2ccccc2C(=O)NC2CCCCC2)c2ccccc2)cc1 ZINC000147232147 KJ In-Stock Anodyne MMP12 28 43 COc1ccc(S(=O)(=O)N(CC(=O)Nc2ccccc2C(=O)NC2CCCCC2)c2ccccc2)cc1 ZINC000147232147 KJ In-Stock Anodyne MMP1 51 46 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccccc3)c(F)c2)CC1 ZINC000147232193 IG Annotated Clean SSTR1 35 40 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccccc3)c(F)c2)CC1 ZINC000147232193 IG Annotated Clean SSTR3 38 40 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccccc3)c(F)c2)CC1 ZINC000147232193 IG Annotated Clean SFRP1 42 33 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccccc3)c(F)c2)CC1 ZINC000147232193 IG Annotated Clean WNT3 50 33 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccccc3)c(F)c2)CC1 ZINC000147232193 IG Annotated Clean RORC 18 46 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne CA2 26 58 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne FOLH1 57 39 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne MME 20 43 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne ANPEP 41 40 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne CTSK 23 43 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne CTSL 29 44 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne CA4 17 58 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne CTSS 18 43 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne FPR1 51 38 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne NPR 53 37 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne AMP1_PLAFQ 18 40 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne SLC15A2 0 44 Cc1ccc(C(=O)N[C@H](CC(C)C)C(=O)O)cc1Br ZINC000147232197 EF On-Demand Anodyne ERAP1 0 42 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild CPT1A 53 62 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild FAAH 0 41 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild EPHX2 65 54 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild Q6UB75_PIG 0 46 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild ASAH1 88 36 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild ACAT 0 42 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild NOD1 74 40 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild OXER1 46 31 CCCCCCCCNC(=O)N[C@H](C)CC(=O)O ZINC000147232255 CF For-Sale Mild CQSS 52 35 COC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147232304 DD On-Demand Anodyne CASR 17 44 COC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147232304 DD On-Demand Anodyne HIF1A 20 40 O=C(/C=N/O)Nc1cccc2ccccc12 ZINC000147232385 BE For-Sale Mild KCNJ11 91 35 O=C(/C=N/O)Nc1cccc2ccccc12 ZINC000147232385 BE For-Sale Mild TRPV1 21 44 O=C(/C=N/O)Nc1cccc2ccccc12 ZINC000147232385 BE For-Sale Mild HDAH 28 47 CC(C)Oc1cccc(CC(=O)Nc2nc(C(C)C)cs2)c1 ZINC000147232411 DI On-Demand Anodyne CSNK1D 37 47 CC(C)Oc1cccc(CC(=O)Nc2nc(C(C)C)cs2)c1 ZINC000147232411 DI On-Demand Anodyne ROCK1 15 41 CC(C)Oc1cccc(CC(=O)Nc2nc(C(C)C)cs2)c1 ZINC000147232411 DI On-Demand Anodyne CDK5 18 40 CC(C)Oc1cccc(CC(=O)Nc2nc(C(C)C)cs2)c1 ZINC000147232411 DI On-Demand Anodyne GCK 15 43 Cc1nc(N(CCc2ccccc2)C2CCN(C(=O)OC(C)(C)C)CC2)no1 ZINC000147232428 GH For-Sale Anodyne GPR119 45 41 CC(C)C[C@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147232453 CE On-Demand Anodyne FOLH1 25 41 CC(C)C[C@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147232453 CE On-Demand Anodyne RIR1_HHV11 83 36 CC(C)C[C@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147232453 CE On-Demand Anodyne CAPN1 28 40 CC(C)C[C@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147232453 CE On-Demand Anodyne LAP3 17 44 CC(C)C[C@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147232453 CE On-Demand Anodyne SLC15A2 0 47 CCCCCCCCNC(=O)N(C)C(C)(C)C(=O)O ZINC000147232475 CF For-Sale Mild EST1_PIG 52 31 CCCCCCCCNC(=O)N(C)C(C)(C)C(=O)O ZINC000147232475 CF For-Sale Mild EPHX2 26 45 CCCCCCCCNC(=O)N(C)C(C)(C)C(=O)O ZINC000147232475 CF For-Sale Mild ASAH1 82 33 Cc1cccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1C(=O)N1CCCC1 ZINC000147232517 HD On-Demand Anodyne LPL 43 34 CC[C@@H](C)NC(=O)[C@@H](C)Oc1ccc(F)cc1S(N)(=O)=O ZINC000147232656 DD For-Sale Anodyne SDH1 0 41 CC(C)C[C@@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147232668 CE On-Demand Anodyne FOLH1 25 41 CC(C)C[C@@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147232668 CE On-Demand Anodyne RIR1_HHV11 83 36 CC(C)C[C@@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147232668 CE On-Demand Anodyne CAPN1 28 40 CC(C)C[C@@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147232668 CE On-Demand Anodyne LAP3 17 44 CC(C)C[C@@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147232668 CE On-Demand Anodyne SLC15A2 0 47 CCCCCCCCNC(=O)N[C@@H](COC)C(=O)O ZINC000147232692 CD For-Sale Mild FOLH1 48 40 CCCCCCCCNC(=O)N[C@@H](COC)C(=O)O ZINC000147232692 CD For-Sale Mild CPT1A 48 49 CCCCCCCCNC(=O)N[C@@H](COC)C(=O)O ZINC000147232692 CD For-Sale Mild EPHX2 65 49 CCCCCCCCNC(=O)N[C@@H](COC)C(=O)O ZINC000147232692 CD For-Sale Mild ASAH1 74 33 CCCCCCCCNC(=O)N[C@@H](COC)C(=O)O ZINC000147232692 CD For-Sale Mild ACAT 0 41 CCCCCCCCNC(=O)N[C@@H](COC)C(=O)O ZINC000147232692 CD For-Sale Mild NOD1 92 45 Cc1cccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1C(=O)N1CCCC1 ZINC000147232700 HD On-Demand Anodyne LPL 43 34 CC(C)=CCC/C(C)=C/CC/C(C)=C/CC/C(C)=C/CCc1ccco1 ZINC000147232748 FK Annotated Anodyne GGPS1 44 36 CC(C)=CCC/C(C)=C/CC/C(C)=C/CC/C(C)=C/CCc1ccco1 ZINC000147232748 FK Annotated Anodyne FDFT1 24 44 CC(C)=CCC/C(C)=C/CC/C(C)=C/CC/C(C)=C/CCc1ccco1 ZINC000147232748 FK Annotated Anodyne TRPA1 24 41 O[C@H](CNN1CCOCC1)COc1ccccc1 ZINC000147232760 CC For-Sale Anodyne ADRB2 55 55 O[C@H](CNN1CCOCC1)COc1ccccc1 ZINC000147232760 CC For-Sale Anodyne ADRB1 63 49 O[C@H](CNN1CCOCC1)COc1ccccc1 ZINC000147232760 CC For-Sale Anodyne ADRB3 58 42 O[C@H](CNN1CCOCC1)COc1ccccc1 ZINC000147232760 CC For-Sale Anodyne CYP2D6 0 40 CCOc1cc(NCCNC(=O)N(C)C)cc([N+](=O)[O-])c1 ZINC000147232802 CD For-Sale Bother PSBA 0 42 CN(Cc1cccc(C(F)(F)F)c1)C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147232807 HG On-Demand Bother CACNA1B 47 35 CN(Cc1cccc(C(F)(F)F)c1)C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147232807 HG On-Demand Bother COLA 23 46 CCCCCCCCNC(=O)N[C@H](COC)C(=O)O ZINC000147232859 CD For-Sale Mild FOLH1 48 40 CCCCCCCCNC(=O)N[C@H](COC)C(=O)O ZINC000147232859 CD For-Sale Mild CPT1A 48 49 CCCCCCCCNC(=O)N[C@H](COC)C(=O)O ZINC000147232859 CD For-Sale Mild EPHX2 65 49 CCCCCCCCNC(=O)N[C@H](COC)C(=O)O ZINC000147232859 CD For-Sale Mild ASAH1 74 33 CCCCCCCCNC(=O)N[C@H](COC)C(=O)O ZINC000147232859 CD For-Sale Mild ACAT 0 41 CCCCCCCCNC(=O)N[C@H](COC)C(=O)O ZINC000147232859 CD For-Sale Mild NOD1 92 45 CC[C@H](C)NC(=O)[C@@H](C)Oc1ccc(F)cc1S(N)(=O)=O ZINC000147232877 DD For-Sale Anodyne SDH1 0 41 CCc1ncc(C(=O)NC[C@@H](c2ccc(OC)cc2)N2CCCCC2)s1 ZINC000147232885 FH On-Demand Anodyne CCR3 18 45 CC(C)C[C@H](NC(=O)C1[C@H]2CCCC[C@@H]12)C(=O)O ZINC000147232937 CE For-Sale Anodyne FOLH1 25 41 CC(C)C[C@H](NC(=O)C1[C@H]2CCCC[C@@H]12)C(=O)O ZINC000147232937 CE For-Sale Anodyne RIR1_HHV11 67 35 CC(C)C[C@H](NC(=O)C1[C@H]2CCCC[C@@H]12)C(=O)O ZINC000147232937 CE For-Sale Anodyne SLC15A2 0 47 CC[C@@H](C)[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147232975 FG On-Demand Mild CACNA1H 20 41 CC[C@@H](C)[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147232975 FG On-Demand Mild CCR1 62 52 CC[C@@H](C)[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147232975 FG On-Demand Mild CCKBR 41 34 CC[C@@H](C)[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147232975 FG On-Demand Mild UTS2 44 35 CCNc1ncc(C)c(Nc2ccc(C#N)cc2F)n1 ZINC000147232980 CF For-Sale Mild SYK 16 42 O[C@@H](CNN1CCOCC1)COc1ccccc1 ZINC000147232990 CC For-Sale Anodyne ADRB2 55 55 O[C@@H](CNN1CCOCC1)COc1ccccc1 ZINC000147232990 CC For-Sale Anodyne ADRB1 63 49 O[C@@H](CNN1CCOCC1)COc1ccccc1 ZINC000147232990 CC For-Sale Anodyne ADRB3 58 42 O[C@@H](CNN1CCOCC1)COc1ccccc1 ZINC000147232990 CC For-Sale Anodyne CYP2D6 0 40 CN(Cc1cccc(C(F)(F)F)c1)C(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147233029 GI On-Demand Anodyne HSD17B2 22 40 CCCCCCCCNC(=O)N1CC[C@H](CCC(=O)O)C1 ZINC000147233069 CG For-Sale Mild F2R 0 41 CCCCCCCCNC(=O)N1CC[C@H](CCC(=O)O)C1 ZINC000147233069 CG For-Sale Mild EPHX2 27 43 CCCCCCCCNC(=O)N1CC[C@H](CCC(=O)O)C1 ZINC000147233069 CG For-Sale Mild ASAH1 100 41 CC[C@@H](C)NC(=O)[C@H](C)Oc1ccc(F)cc1S(N)(=O)=O ZINC000147233073 DD For-Sale Anodyne SDH1 0 41 CCNc1cncc(Oc2ccc3ccccc3c2)n1 ZINC000147233082 CH For-Sale Anodyne CYP11B2 21 40 CCc1ncc(C(=O)NC[C@H](c2ccc(OC)cc2)N2CCCCC2)s1 ZINC000147233099 FH On-Demand Anodyne CCR3 18 45 O=S(=O)(c1ccc2c(c1)CCC2)N1CCC(CBr)CC1 ZINC000147233130 FF For-Sale Reactive AKR1C3 59 37 COc1cc(C[C@@H](OC(=O)/C=C/c2ccc3c(c2)O[C@H](C(=O)O)[C@H](c2ccc(O)c(O)c2)O3)C(=O)O)ccc1O ZINC000147233131 KG Annotated Clean MMP12 0 51 CN1CCC(Nc2ccc(-c3ccn4c(-c5cccc(NC(=O)NCC(F)(F)F)c5)cnc4c3)nn2)CC1 ZINC000147233148 KJ Annotated Anodyne PRKD1 45 31 CC(C)C[C@@H](NC(=O)C1[C@H]2CCCC[C@@H]12)C(=O)O ZINC000147233166 CE For-Sale Anodyne FOLH1 25 41 CC(C)C[C@@H](NC(=O)C1[C@H]2CCCC[C@@H]12)C(=O)O ZINC000147233166 CE For-Sale Anodyne RIR1_HHV11 67 35 CC(C)C[C@@H](NC(=O)C1[C@H]2CCCC[C@@H]12)C(=O)O ZINC000147233166 CE For-Sale Anodyne SLC15A2 0 47 CC[C@@H](C)[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147233189 FG On-Demand Mild CACNA1H 20 41 CC[C@@H](C)[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147233189 FG On-Demand Mild CCR1 62 52 CC[C@@H](C)[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147233189 FG On-Demand Mild CCKBR 41 34 CC[C@@H](C)[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147233189 FG On-Demand Mild UTS2 44 35 O=C(CNN1CCOCC1)Nc1ccccc1 ZINC000147233236 BC For-Sale Anodyne LPL 33 43 O=C(CNN1CCOCC1)Nc1ccccc1 ZINC000147233236 BC For-Sale Anodyne PIK3CA 16 44 O=C(CNN1CCOCC1)Nc1ccccc1 ZINC000147233236 BC For-Sale Anodyne MTOR 27 44 O=C(CNN1CCOCC1)Nc1ccccc1 ZINC000147233236 BC For-Sale Anodyne EPHX2 32 49 O=C(CNN1CCOCC1)Nc1ccccc1 ZINC000147233236 BC For-Sale Anodyne PIK3CG 15 44 O=C(CNN1CCOCC1)Nc1ccccc1 ZINC000147233236 BC For-Sale Anodyne DGAT1 27 40 O=C(CNN1CCOCC1)Nc1ccccc1 ZINC000147233236 BC For-Sale Anodyne PFHDAC1 0 40 CCCCCCCCNC(=O)N1CC[C@@H](CCC(=O)O)C1 ZINC000147233310 CG For-Sale Mild F2R 0 41 CCCCCCCCNC(=O)N1CC[C@@H](CCC(=O)O)C1 ZINC000147233310 CG For-Sale Mild EPHX2 27 43 CCCCCCCCNC(=O)N1CC[C@@H](CCC(=O)O)C1 ZINC000147233310 CG For-Sale Mild ASAH1 100 41 CC[C@H](C)NC(=O)[C@H](C)Oc1ccc(F)cc1S(N)(=O)=O ZINC000147233311 DD For-Sale Anodyne SDH1 0 41 COc1ccc(NC(C)=O)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147233330 ED On-Demand Anodyne QRFPR 41 35 Cc1ncoc1C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147233393 BD On-Demand Anodyne FOLH1 53 39 Cc1ncoc1C(=O)N[C@@H](CC(C)C)C(=O)O ZINC000147233393 BD On-Demand Anodyne NPR 40 34 O=CCc1c[nH]c2cc(F)c(F)cc12 ZINC000147233398 AE For-Sale Mild MPO 81 39 CC[C@H](C)[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147233407 FG On-Demand Mild CACNA1H 20 41 CC[C@H](C)[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147233407 FG On-Demand Mild CCR1 62 52 CC[C@H](C)[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147233407 FG On-Demand Mild CCKBR 41 34 CC[C@H](C)[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147233407 FG On-Demand Mild UTS2 44 35 CC(C)Oc1cccc(CC(=O)N[C@@H]2CCSc3ccc(F)cc32)c1 ZINC000147233454 FJ On-Demand Anodyne LUXR 42 39 CNc1nc(OC)nc(Oc2ccc3ccccc3c2)n1 ZINC000147233506 CF For-Sale Anodyne CYP2A5 0 49 CCCCCCCCNC(=O)NC[C@@H](CC)CC(=O)O ZINC000147233533 CG For-Sale Mild CPT1A 48 53 CCCCCCCCNC(=O)NC[C@@H](CC)CC(=O)O ZINC000147233533 CG For-Sale Mild EPHX2 59 54 CCCCCCCCNC(=O)NC[C@@H](CC)CC(=O)O ZINC000147233533 CG For-Sale Mild ASAH1 70 34 CCCCCCCCNC(=O)NC[C@@H](CC)CC(=O)O ZINC000147233533 CG For-Sale Mild NOD1 44 35 CCCCCCCCNC(=O)NC[C@@H](CC)CC(=O)O ZINC000147233533 CG For-Sale Mild CQSS 42 33 COc1ccc(NC(C)=O)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147233551 ED On-Demand Anodyne QRFPR 41 35 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCCC1 ZINC000147233553 DD For-Sale Anodyne HTR2A 28 43 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCCC1 ZINC000147233553 DD For-Sale Anodyne HTR2C 15 47 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCCC1 ZINC000147233553 DD For-Sale Anodyne LTA4H 36 47 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCCC1 ZINC000147233553 DD For-Sale Anodyne HRH3 32 46 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCCC1 ZINC000147233553 DD For-Sale Anodyne MCHR1 0 43 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCCC1 ZINC000147233553 DD For-Sale Anodyne PSMB2 39 40 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCCC1 ZINC000147233553 DD For-Sale Anodyne PSMB1 43 40 C[C@H]1CCC[C@@H](C)N1C(=O)COc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147233622 GG On-Demand Mild HRH3 25 48 C[C@H]1CCC[C@@H](C)N1C(=O)COc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147233622 GG On-Demand Mild COLA 45 39 C[C@H]1CCC[C@@H](C)N1C(=O)COc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147233622 GG On-Demand Mild CPT1A 45 39 C[C@H]1CCC[C@@H](C)N1C(=O)COc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147233622 GG On-Demand Mild L3MBTL3 66 37 CNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147233641 CF For-Sale Mild INSR 39 42 CNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147233641 CF For-Sale Mild MAPK9 45 45 CNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147233641 CF For-Sale Mild MAPK10 46 45 CNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147233641 CF For-Sale Mild ALK 34 42 COc1ccc(CN2CCC(Nc3nc4cc(Cl)ccc4o3)CC2)cc1OCCF ZINC000147233674 IJ For-Sale Anodyne DRD4 23 40 COc1ccc(CN2CCC(Nc3nc4cc(Cl)ccc4o3)CC2)cc1OCCF ZINC000147233674 IJ For-Sale Anodyne HRH1 18 65 COc1ccc(CN2CCC(Nc3nc4cc(Cl)ccc4o3)CC2)cc1OCCF ZINC000147233674 IJ For-Sale Anodyne SSTR5 117 84 COc1ccc(CN2CCC(Nc3nc4cc(Cl)ccc4o3)CC2)cc1OCCF ZINC000147233674 IJ For-Sale Anodyne MCHR1 36 47 COc1ccc(CN2CCC(Nc3nc4cc(Cl)ccc4o3)CC2)cc1OCCF ZINC000147233674 IJ For-Sale Anodyne EHMT2 79 38 CCCCCCCCNC(=O)NC[C@H](CC)CC(=O)O ZINC000147233726 CG For-Sale Mild CPT1A 48 53 CCCCCCCCNC(=O)NC[C@H](CC)CC(=O)O ZINC000147233726 CG For-Sale Mild EPHX2 59 54 CCCCCCCCNC(=O)NC[C@H](CC)CC(=O)O ZINC000147233726 CG For-Sale Mild ASAH1 70 34 CCCCCCCCNC(=O)NC[C@H](CC)CC(=O)O ZINC000147233726 CG For-Sale Mild NOD1 44 35 CCCCCCCCNC(=O)NC[C@H](CC)CC(=O)O ZINC000147233726 CG For-Sale Mild CQSS 42 33 CC[C@@H](C)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147233812 CF On-Demand Anodyne ACE 30 43 CC[C@@H](C)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147233812 CF On-Demand Anodyne TPP2 43 30 C[C@@H]1CCC[C@@H](C)N1C(=O)COc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147233828 GG On-Demand Mild HRH3 25 48 C[C@@H]1CCC[C@@H](C)N1C(=O)COc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147233828 GG On-Demand Mild COLA 45 39 C[C@@H]1CCC[C@@H](C)N1C(=O)COc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147233828 GG On-Demand Mild CPT1A 45 39 C[C@@H]1CCC[C@@H](C)N1C(=O)COc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147233828 GG On-Demand Mild L3MBTL3 66 37 C=CCN(C(=O)c1cccc2c1OCCN2)C1CCCC1 ZINC000147233846 CG For-Sale Mild ACE 42 41 O=S(=O)(c1c(F)cc(F)cc1F)N1CCC(CBr)CC1 ZINC000147233849 FF For-Sale Reactive EPHX2 29 44 O=S(=O)(c1c(F)cc(F)cc1F)N1CCC(CBr)CC1 ZINC000147233849 FF For-Sale Reactive PKM 28 45 C[C@H](CNS(=O)(=O)c1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147233943 DC On-Demand Bother NADE 0 40 C[C@H](CNS(=O)(=O)c1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147233943 DC On-Demand Bother COLA 57 38 C[C@H](CNS(=O)(=O)c1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147233943 DC On-Demand Bother MMP2 25 52 Nc1cc(Oc2ccc3ccccc3c2)ncn1 ZINC000147233947 BG For-Sale Anodyne CYP2A5 0 40 CCCCCCCCNC(=O)NC1(C(=O)O)CCC1 ZINC000147233949 CF For-Sale Mild CPT1A 0 40 CCCCCCCCNC(=O)NC1(C(=O)O)CCC1 ZINC000147233949 CF For-Sale Mild EPHX2 38 52 CCCCCCCCNC(=O)NC1(C(=O)O)CCC1 ZINC000147233949 CF For-Sale Mild ASAH1 67 34 CSc1ccccc1CNC(=O)c1ccccc1 ZINC000147234030 CG For-Sale Anodyne ECR 31 41 CSc1ccccc1CNC(=O)c1ccccc1 ZINC000147234030 CG For-Sale Anodyne CTSG 18 42 CSc1ccccc1CNC(=O)c1ccccc1 ZINC000147234030 CG For-Sale Anodyne CTRB1 36 42 CSc1ccccc1CNC(=O)c1ccccc1 ZINC000147234030 CG For-Sale Anodyne AMP1_PLAFQ 42 38 CC[C@H](C)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147234064 CF On-Demand Anodyne ACE 30 43 CC[C@H](C)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147234064 CF On-Demand Anodyne TPP2 43 30 NC(=O)c1ccccc1CNN1CCOCC1 ZINC000147234084 BC For-Sale Anodyne STAT6 68 39 CCCCCCCCNC(=O)NCC(=O)NCC(=O)O ZINC000147234112 CC For-Sale Mild EPHX2 25 58 CCCCCCCCNC(=O)NCC(=O)NCC(=O)O ZINC000147234112 CC For-Sale Mild ASAH1 84 33 C[C@@H](CNS(=O)(=O)c1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147234120 DC On-Demand Bother NADE 0 40 C[C@@H](CNS(=O)(=O)c1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147234120 DC On-Demand Bother COLA 57 38 C[C@@H](CNS(=O)(=O)c1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147234120 DC On-Demand Bother MMP2 25 52 CCO[C@@H]1CCCN(C(=O)Nc2cc(C(F)(F)F)ccc2-n2nc(C)cc2C)C1 ZINC000147234240 HJ On-Demand Anodyne LIPG 56 43 CC[C@@H](C)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147234263 CF On-Demand Anodyne ACE 30 43 CC[C@@H](C)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147234263 CF On-Demand Anodyne TPP2 43 30 CCN(CC)[C@@H](CNC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147234272 EG On-Demand Anodyne BMP1 41 33 CCCC[C@H](NC(N)=O)C(=O)N[C@@H]1CCC[C@H](C(F)(F)F)C1 ZINC000147234320 DE On-Demand Anodyne HDAC4 15 40 CCCCCCCCNC(=O)N1CC(C(=O)O)C1 ZINC000147234348 CE On-Demand Mild EPHX2 39 40 CCCCCCCCNC(=O)N1CC(C(=O)O)C1 ZINC000147234348 CE On-Demand Mild ASAH1 106 43 CCCCCCCCNC(=O)N1CC(C(=O)O)C1 ZINC000147234348 CE On-Demand Mild NOD1 40 36 O=C(Nc1ncccc1O)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147234367 FD On-Demand Anodyne GSK3B 15 46 O=C(Nc1ncccc1O)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147234367 FD On-Demand Anodyne PRNP 44 34 O=C(Nc1ncccc1O)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147234367 FD On-Demand Anodyne TGM2 68 44 O=C(Nc1ncccc1O)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147234367 FD On-Demand Anodyne F13A1 78 44 O=C(Nc1ncccc1O)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147234367 FD On-Demand Anodyne MERTK 26 44 O=C(Nc1ncccc1O)c1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147234367 FD On-Demand Anodyne NAMPT 48 48 CN1CCN(CCOc2ccc(F)cc2S(N)(=O)=O)CC1 ZINC000147234376 DC For-Sale Anodyne DRD2 16 48 CN1CCN(CCOc2ccc(F)cc2S(N)(=O)=O)CC1 ZINC000147234376 DC For-Sale Anodyne HTR6 15 40 COc1cnc2ncccc2c1 ZINC000147234412 AD For-Sale Anodyne CYP11B2 29 43 CN(C)C(=O)NCCNc1ccc([N+](=O)[O-])c2nonc12 ZINC000147234428 CC On-Demand Bother GSTM2 80 40 CN(C)C(=O)NCCNc1ccc([N+](=O)[O-])c2nonc12 ZINC000147234428 CC On-Demand Bother GSTP1 79 48 CSc1nc(N)cc(Oc2ccc3ccccc3c2)n1 ZINC000147234429 CH For-Sale Anodyne CYP2A5 0 41 CC[C@H](C)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147234454 CF On-Demand Anodyne ACE 30 43 CC[C@H](C)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147234454 CF On-Demand Anodyne TPP2 43 30 CCO[C@H]1CCCN(C(=O)Nc2cc(C(F)(F)F)ccc2-n2nc(C)cc2C)C1 ZINC000147234469 HJ On-Demand Anodyne LIPG 56 43 CCN(CC)[C@H](CNC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147234487 EG On-Demand Anodyne BMP1 41 33 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne TBXAS1 17 48 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne FABP4 15 67 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne FAAH 18 46 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne CES2 47 41 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne CES1 26 41 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne EST1_PIG 63 41 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne CES2C 53 33 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne FABP3 52 67 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne FABP5 24 67 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne FABP1 22 67 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne NOD1 42 36 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne OXER1 32 42 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne CQSS 60 37 CCCCCC/C=C(/C)CCCCCCCCCC(=O)O ZINC000147234505 CK For-Sale Anodyne SLCO2A1 48 35 CCCCCCCCNC(=O)N(CCC(=O)O)C(C)(C)C ZINC000147234539 DH For-Sale Mild FABP2 0 44 CCCCCCCCNC(=O)N(CCC(=O)O)C(C)(C)C ZINC000147234539 DH For-Sale Mild EPHX2 33 52 CCCCCCCCNC(=O)N(CCC(=O)O)C(C)(C)C ZINC000147234539 DH For-Sale Mild FABP5 15 44 CCCCCCCCNC(=O)N(CCC(=O)O)C(C)(C)C ZINC000147234539 DH For-Sale Mild ASAH1 82 34 CCCCCCCCNC(=O)N(CCC(=O)O)C(C)(C)C ZINC000147234539 DH For-Sale Mild SLC22A20 0 44 CCN(CC)C(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147234654 GE On-Demand Anodyne ENV 41 33 Nc1ccc2nc(NCC(F)F)sc2c1 ZINC000147234677 BF For-Sale Anodyne MAPT 19 43 CCCCCCCCNC(=O)N(CC(=O)O)[C@@H](C)CC ZINC000147234731 CG For-Sale Mild CPT1A 39 43 CCCCCCCCNC(=O)N(CC(=O)O)[C@@H](C)CC ZINC000147234731 CG For-Sale Mild EPHX2 42 47 CCCCCCCCNC(=O)N(CC(=O)O)[C@@H](C)CC ZINC000147234731 CG For-Sale Mild ASAH1 90 34 CCCCCCCCNC(=O)N(CC(=O)O)[C@@H](C)CC ZINC000147234731 CG For-Sale Mild NOD1 53 38 CCCCCCCCNC(=O)N(CC(=O)O)[C@@H](C)CC ZINC000147234731 CG For-Sale Mild CQSS 42 33 CCCC[C@H](NC(N)=O)C(=O)N[C@H]1CCC[C@H](C(F)(F)F)C1 ZINC000147234742 DE On-Demand Anodyne HDAC4 15 40 COC(=O)c1cccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)c1 ZINC000147234821 DC On-Demand Anodyne CASP3 21 40 COC(=O)c1cccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)c1 ZINC000147234821 DC On-Demand Anodyne ADAMTS4 15 42 COC(=O)c1cccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)c1 ZINC000147234821 DC On-Demand Anodyne AKR1C3 17 45 CCN(CC)C(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147234867 GE On-Demand Anodyne ENV 41 33 CCCCCCCCNC(=O)N(CC(=O)O)[C@H](C)CC ZINC000147234925 CG For-Sale Mild CPT1A 39 43 CCCCCCCCNC(=O)N(CC(=O)O)[C@H](C)CC ZINC000147234925 CG For-Sale Mild EPHX2 42 47 CCCCCCCCNC(=O)N(CC(=O)O)[C@H](C)CC ZINC000147234925 CG For-Sale Mild ASAH1 90 34 CCCCCCCCNC(=O)N(CC(=O)O)[C@H](C)CC ZINC000147234925 CG For-Sale Mild NOD1 53 38 CCCCCCCCNC(=O)N(CC(=O)O)[C@H](C)CC ZINC000147234925 CG For-Sale Mild CQSS 42 33 Cc1ccc(C)c(-c2ccccc2C(F)(F)F)c1 ZINC000147234999 CJ For-Sale Anodyne TRPA1 28 51 NS(=O)(=O)c1cc(F)ccc1OCC(=O)NC1CC1 ZINC000147235004 CC For-Sale Anodyne NPY2R 29 40 NS(=O)(=O)c1cc(F)ccc1OCC(=O)NC1CC1 ZINC000147235004 CC For-Sale Anodyne NPY5R 18 40 CC(C)CN(Cc1ccc(OC2CCN(S(C)(=O)=O)CC2)cc1)S(=O)(=O)Cc1ccccc1 ZINC000147235031 JG Annotated Anodyne PRSS2 56 36 COC(=O)c1cccc(S(=O)(=O)NC[C@H](C)CC(=O)O)c1 ZINC000147235034 DC On-Demand Anodyne CASP3 21 40 COC(=O)c1cccc(S(=O)(=O)NC[C@H](C)CC(=O)O)c1 ZINC000147235034 DC On-Demand Anodyne ADAMTS4 15 42 COC(=O)c1cccc(S(=O)(=O)NC[C@H](C)CC(=O)O)c1 ZINC000147235034 DC On-Demand Anodyne AKR1C3 17 45 CCC(CC)N(CCOC)C(=O)c1cc2cc(Cl)ccc2[nH]1 ZINC000147235066 DI On-Demand Anodyne PYGL 92 54 COc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1NC(=O)c1cccnc1 ZINC000147235089 HD On-Demand Anodyne ROCK2 22 42 CCCCCCCCNC(=O)N[C@@H](CCC(N)=O)C(=O)O ZINC000147235128 DD For-Sale Mild FOLH1 78 51 CCCCCCCCNC(=O)N[C@@H](CCC(N)=O)C(=O)O ZINC000147235128 DD For-Sale Mild CPT1A 27 47 CCCCCCCCNC(=O)N[C@@H](CCC(N)=O)C(=O)O ZINC000147235128 DD For-Sale Mild C3AR1 59 36 CCCCCCCCNC(=O)N[C@@H](CCC(N)=O)C(=O)O ZINC000147235128 DD For-Sale Mild NAALAD2 64 44 CCCCCCCCNC(=O)N[C@@H](CCC(N)=O)C(=O)O ZINC000147235128 DD For-Sale Mild EPHX2 57 50 CCCCCCCCNC(=O)N[C@@H](CCC(N)=O)C(=O)O ZINC000147235128 DD For-Sale Mild ASAH1 86 35 CCCCCCCCNC(=O)N[C@@H](CCC(N)=O)C(=O)O ZINC000147235128 DD For-Sale Mild NOD1 120 55 CCCCCCCCNC(=O)N[C@@H](CCC(N)=O)C(=O)O ZINC000147235128 DD For-Sale Mild CQSS 51 32 CC(C)NC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147235217 CC For-Sale Anodyne SDH1 0 44 CCN(CC)S(=O)(=O)c1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147235227 HG On-Demand Anodyne BMP1 41 32 COc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1NC(=O)c1cccnc1 ZINC000147235298 HD On-Demand Anodyne ROCK2 22 42 CCCCCCCCNC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147235328 CC For-Sale Mild FOLH1 46 40 CCCCCCCCNC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147235328 CC For-Sale Mild GRIA1 69 35 CCCCCCCCNC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147235328 CC For-Sale Mild EPHX2 20 55 CCCCCCCCNC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147235328 CC For-Sale Mild ASAH1 67 33 CCCCCCCCNC(=O)N[C@@H](CC(N)=O)C(=O)O ZINC000147235328 CC For-Sale Mild NOD1 96 45 CCOC(=O)c1cnc(-c2cccnc2)nc1NC ZINC000147235414 CD For-Sale Anodyne JUN 19 52 CCOC(=O)c1cnc(-c2cccnc2)nc1NC ZINC000147235414 CD For-Sale Anodyne CYP11B2 20 41 CCOC(=O)c1cnc(-c2cccnc2)nc1NC ZINC000147235414 CD For-Sale Anodyne ADORA3 18 42 CCN(CC)S(=O)(=O)c1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147235427 HG On-Demand Anodyne BMP1 41 32 CCC(CC)N(CCOC)C(=O)c1cc2ccc(Cl)cc2[nH]1 ZINC000147235464 DI On-Demand Anodyne PYGL 62 45 CNc1nc(C)cc(Oc2ccc3ccccc3c2)n1 ZINC000147235476 CH For-Sale Anodyne CYP2A5 0 41 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne DRD2 27 48 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne CNR1 23 41 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne DRD4 61 63 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne ACHE 25 54 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne HRH1 24 57 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne DRD3 18 45 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne KCNH2 22 42 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne HTR4 39 40 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne F10 17 47 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne CNR2 22 44 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne HRH3 16 43 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne SIGMAR1 35 50 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne SSTR5 105 57 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne CCR1 35 42 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne CCR3 33 42 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne CCR5 15 50 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne UTS2R 32 58 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne CCR2 18 46 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne SLC6A5 40 46 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne PTGDR 19 42 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne PDK1 41 38 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne CXCR3 48 43 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne MCHR1 72 58 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne PTGDR2 18 42 CCCOc1ccc(C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cc1OCC ZINC000147235552 IJ On-Demand Anodyne CACNA1I 53 43 CCCCN(CCBr)S(=O)(=O)c1ccc2c(c1)OCCO2 ZINC000147235607 GF For-Sale Reactive PKM 36 43 CCCCCCCCNC(=O)N(CC(=O)O)C(C)(C)C ZINC000147235612 CG For-Sale Mild EPHX2 28 44 CCCCCCCCNC(=O)N(CC(=O)O)C(C)(C)C ZINC000147235612 CG For-Sale Mild ASAH1 75 32 Cc1cc(NCCNC(=O)N(C)C)c2ccccc2n1 ZINC000147235621 CE On-Demand Anodyne ADAM17 54 35 Cc1cc(NCCNC(=O)N(C)C)c2ccccc2n1 ZINC000147235621 CE On-Demand Anodyne SLC2A1 0 46 Cc1cc(NCCNC(=O)N(C)C)c2ccccc2n1 ZINC000147235621 CE On-Demand Anodyne HT1 0 46 Cc1cc(NCCNC(=O)N(C)C)c2ccccc2n1 ZINC000147235621 CE On-Demand Anodyne LMGT2 0 46 Cc1ncc([N+](=O)[O-])n1CCN1CCN(C(=O)OC(C)(C)C)CC1 ZINC000147235719 ED On-Demand Bother TYMS 33 40 CCC(CC)N(CCOC)C(=O)c1cnn2c(-c3ccccc3)ccnc12 ZINC000147235752 FH On-Demand Anodyne BRAF 23 41 CCCc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147235755 CE On-Demand Anodyne CA2 23 43 CCCc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147235755 CE On-Demand Anodyne TBXA2R 48 36 CCCc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147235755 CE On-Demand Anodyne CA1 17 40 CCCc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147235755 CE On-Demand Anodyne CA4 19 40 CCCc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147235755 CE On-Demand Anodyne LIMK2 37 40 CCCc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147235755 CE On-Demand Anodyne OXER1 43 35 CCNc1nc(Cl)nc(Nc2ccc(C#N)cc2F)n1 ZINC000147235811 CF For-Sale Mild PETD 0 48 CCNc1nc(Cl)nc(Nc2ccc(C#N)cc2F)n1 ZINC000147235811 CF For-Sale Mild Q31945_CHEAL 0 40 CCNc1nc(Cl)nc(Nc2ccc(C#N)cc2F)n1 ZINC000147235811 CF For-Sale Mild PPX1 0 48 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc2c(c1)Cc1ccccc1-2 ZINC000147235824 FF On-Demand Anodyne SLC1A1 24 44 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc2c(c1)Cc1ccccc1-2 ZINC000147235824 FF On-Demand Anodyne SLC1A3 28 44 CC(C)[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147235865 EF On-Demand Mild ELANE 41 41 CC(C)[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147235865 EF On-Demand Mild CCR1 75 60 CC(C)[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147235865 EF On-Demand Mild UTS2 44 35 Nc1nccc(Oc2ccc3ccccc3c2)n1 ZINC000147235925 BG For-Sale Anodyne CYP2A5 0 40 CCCc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147235939 CE On-Demand Anodyne CA2 23 43 CCCc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147235939 CE On-Demand Anodyne TBXA2R 48 36 CCCc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147235939 CE On-Demand Anodyne CA1 17 40 CCCc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147235939 CE On-Demand Anodyne CA4 19 40 CCCc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147235939 CE On-Demand Anodyne LIMK2 37 40 CCCc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147235939 CE On-Demand Anodyne OXER1 43 35 CCOC(=O)[C@@]1(C)C[C@H]1c1ccccc1 ZINC000147235944 BF For-Sale Anodyne CACNA1C 38 41 CCOC(=O)[C@@]1(C)C[C@H]1c1ccccc1 ZINC000147235944 BF For-Sale Anodyne CACNA1D 50 34 CCOC(=O)[C@@]1(C)C[C@H]1c1ccccc1 ZINC000147235944 BF For-Sale Anodyne KDM1A 38 45 C#CCNC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147235948 CB For-Sale Mild CA2 25 41 CCCCCCCCNC(=O)N(CC)C[C@@H](C)C(=O)O ZINC000147235958 CG For-Sale Mild EPHX2 40 39 CCCCCCCCNC(=O)N(CC)C[C@@H](C)C(=O)O ZINC000147235958 CG For-Sale Mild ASAH1 60 32 CCCCCCCCNC(=O)N(CC)C[C@@H](C)C(=O)O ZINC000147235958 CG For-Sale Mild NOD1 75 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc2c(c1)Cc1ccccc1-2 ZINC000147236028 FF On-Demand Anodyne SLC1A1 24 44 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc2c(c1)Cc1ccccc1-2 ZINC000147236028 FF On-Demand Anodyne SLC1A3 28 44 C[C@@H]1O[C@H](Oc2ccc([N+](=O)[O-])cc2Cl)[C@H](O)[C@H](O)[C@H]1O ZINC000147236050 DC For-Sale Anodyne FIMH 67 44 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccc2ccccc12 ZINC000147236095 EI On-Demand Anodyne BMP1 49 33 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccc2ccccc12 ZINC000147236095 EI On-Demand Anodyne CYP3A4 18 44 CC(C)C[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236119 FG On-Demand Mild P2RY12 46 34 CC(C)C[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236119 FG On-Demand Mild MC4R 102 42 CC(C)C[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236119 FG On-Demand Mild CTSK 20 43 CC(C)C[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236119 FG On-Demand Mild CTSL 32 45 CC(C)C[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236119 FG On-Demand Mild CCR1 56 43 CC(C)C[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236119 FG On-Demand Mild MC3R 42 39 CC(C)C[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236119 FG On-Demand Mild MC5R 70 40 CC(C)C[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236119 FG On-Demand Mild CCKBR 30 46 CC(C)C[C@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236119 FG On-Demand Mild UTS2 45 35 COCCN(CC(=O)O)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147236120 CD For-Sale Anodyne GPR88 0 43 COc1ccc([N+](=O)[O-])cc1SC ZINC000147236122 AE In-Stock Bother KCNMA1 20 44 COc1ccc([N+](=O)[O-])cc1SC ZINC000147236122 AE In-Stock Bother TRXR2 0 43 C[C@H](CNS(=O)(=O)c1ccc(C(C)(C)C)cc1)CC(=O)O ZINC000147236132 DE On-Demand Anodyne CYNT 50 42 C[C@H](CNS(=O)(=O)c1ccc(C(C)(C)C)cc1)CC(=O)O ZINC000147236132 DE On-Demand Anodyne UQCRB 0 42 CCCCCCCCNC(=O)N(CC)C[C@H](C)C(=O)O ZINC000147236157 CG For-Sale Mild EPHX2 40 39 CCCCCCCCNC(=O)N(CC)C[C@H](C)C(=O)O ZINC000147236157 CG For-Sale Mild ASAH1 60 32 CCCCCCCCNC(=O)N(CC)C[C@H](C)C(=O)O ZINC000147236157 CG For-Sale Mild NOD1 75 40 CCCCCC(=O)C(F)(F)C(F)(F)F ZINC000147236172 BG For-Sale Anodyne CES2 67 65 CCCCCC(=O)C(F)(F)C(F)(F)F ZINC000147236172 BG For-Sale Anodyne CES1 80 65 CCCCCC(=O)C(F)(F)C(F)(F)F ZINC000147236172 BG For-Sale Anodyne EST1_PIG 99 65 CCCCCC(=O)C(F)(F)C(F)(F)F ZINC000147236172 BG For-Sale Anodyne CES2C 73 42 CCCCCC(=O)C(F)(F)C(F)(F)F ZINC000147236172 BG For-Sale Anodyne FABP5 15 44 CCCCCC(=O)C(F)(F)C(F)(F)F ZINC000147236172 BG For-Sale Anodyne CQSS 63 39 O=C1Cc2cc(OCc3ccccc3)ccc2N1 ZINC000147236178 BF In-Stock Anodyne MAOA 29 52 O=C1Cc2cc(OCc3ccccc3)ccc2N1 ZINC000147236178 BF In-Stock Anodyne MAOB 77 49 O=C1Cc2cc(OCc3ccccc3)ccc2N1 ZINC000147236178 BF In-Stock Anodyne GRM1 25 47 O=C1Cc2cc(OCc3ccccc3)ccc2N1 ZINC000147236178 BF In-Stock Anodyne FFAR1 26 43 O=C1Cc2cc(OCc3ccccc3)ccc2N1 ZINC000147236178 BF In-Stock Anodyne HPGD 24 44 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(-c2cn3ccccc3n2)cc1 ZINC000147236224 FG On-Demand Anodyne P2RY12 60 33 COc1ccc(CN[C@@H]2CCN(Cc3ccccc3)C2=O)cc1OCCCC#N ZINC000147236263 GG On-Demand Mild ACHE 17 43 COc1ccc(CN[C@@H]2CCN(Cc3ccccc3)C2=O)cc1OCCCC#N ZINC000147236263 GG On-Demand Mild SIGMAR1 15 43 COc1cccc(CNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)c1 ZINC000147236293 HF On-Demand Anodyne KCNA5 15 43 COc1cccc(CNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)c1 ZINC000147236293 HF On-Demand Anodyne MMP13 41 50 COc1cccc(CNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)c1 ZINC000147236293 HF On-Demand Anodyne MAP1 81 34 COc1cccc(CNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)c1 ZINC000147236293 HF On-Demand Anodyne ROCK1 38 44 COc1cccc(CNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)c1 ZINC000147236293 HF On-Demand Anodyne ROCK2 42 38 COc1cccc(CNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)c1 ZINC000147236293 HF On-Demand Anodyne LIMK2 26 46 COc1cccc(CNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)c1 ZINC000147236293 HF On-Demand Anodyne NAMPT 68 36 C[C@@H](CNS(=O)(=O)c1ccc(C(C)(C)C)cc1)CC(=O)O ZINC000147236302 DE On-Demand Anodyne CA2 20 42 C[C@@H](CNS(=O)(=O)c1ccc(C(C)(C)C)cc1)CC(=O)O ZINC000147236302 DE On-Demand Anodyne CYNT 50 42 C[C@@H](CNS(=O)(=O)c1ccc(C(C)(C)C)cc1)CC(=O)O ZINC000147236302 DE On-Demand Anodyne UQCRB 0 42 COCCN(CC(=O)O)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147236304 CD For-Sale Anodyne GPR88 0 43 C#CCNC(=O)[C@H](C)Oc1ccc(F)cc1S(N)(=O)=O ZINC000147236328 DB For-Sale Mild CA2 29 40 CC(C)C[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236347 FG On-Demand Mild P2RY12 46 34 CC(C)C[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236347 FG On-Demand Mild MC4R 102 42 CC(C)C[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236347 FG On-Demand Mild CTSK 20 43 CC(C)C[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236347 FG On-Demand Mild CTSL 32 45 CC(C)C[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236347 FG On-Demand Mild CCR1 56 43 CC(C)C[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236347 FG On-Demand Mild MC3R 42 39 CC(C)C[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236347 FG On-Demand Mild MC5R 70 40 CC(C)C[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236347 FG On-Demand Mild CCKBR 30 46 CC(C)C[C@@H](NC(=O)c1ccc(Cl)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147236347 FG On-Demand Mild UTS2 45 35 CCCCCCCCNC(=O)N1C[C@@H](C(=O)O)[C@@H](C)C1 ZINC000147236352 CF For-Sale Mild ASAH1 100 38 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccc2ccccc12 ZINC000147236354 EI On-Demand Anodyne CYP3A4 18 44 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne DRD2 23 47 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne DRD4 48 47 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne ACHE 46 43 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne HRH1 39 41 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne DRD3 26 47 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne KCNH2 16 41 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne LTA4H 20 40 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne HRH3 22 56 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne SIGMAR1 67 52 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne BCHE 15 40 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne CCR3 58 41 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne SLC18A3 25 44 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne SCN9A 17 41 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne MLNR 41 41 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne SCN5A 65 38 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne MCHR1 28 41 O=C(C1CCN(Cc2ccccc2)CC1)N1CCC(Oc2c(F)cc(F)cc2F)CC1 ZINC000147236402 II For-Sale Anodyne CACNA1G 39 44 COc1ccc(CN[C@H]2CCN(Cc3ccccc3)C2=O)cc1OCCCC#N ZINC000147236430 GG On-Demand Mild ACHE 17 43 COc1ccc(CN[C@H]2CCN(Cc3ccccc3)C2=O)cc1OCCCC#N ZINC000147236430 GG On-Demand Mild SIGMAR1 15 43 Cc1nc(N)c(C)c(Oc2ccc3ccccc3c2)n1 ZINC000147236439 CH For-Sale Anodyne CYP2A5 0 42 COc1cc(C(=O)NNC(=O)Nc2nc(C)cs2)ccc1OC(C)C ZINC000147236464 FF On-Demand Reactive GCK 22 48 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(-c2cn3ccccc3n2)cc1 ZINC000147236477 FG On-Demand Anodyne P2RY12 60 33 Cc1cccc(NNC=O)c1 ZINC000147236479 AD For-Sale Anodyne IDO1 16 46 Cc1cccc(NNC=O)c1 ZINC000147236479 AD For-Sale Anodyne KCNK3 53 41 Cc1cccc(NNC=O)c1 ZINC000147236479 AD For-Sale Anodyne KCNK9 43 41 COCCN(CC(=O)O)C(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147236486 CD For-Sale Anodyne GPR88 0 43 N#CC1CCN(C(=O)c2ccc3c(c2)C(=O)N(CCc2ccccc2)C3=O)CC1 ZINC000147236546 GF On-Demand Mild L3MBTL3 49 39 CCCCCCCCNC(=O)N1C[C@@H](C)[C@H](C(=O)O)C1 ZINC000147236551 CF For-Sale Mild ASAH1 100 38 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne MAOB 33 43 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne CYSLTR1 19 41 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne LTA4H 22 44 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne CYSLTR2 51 37 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne SCN2A 16 42 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne ADAM17 24 43 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne PRNP 46 38 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne NR1H4 18 47 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne HDAC1 41 42 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne HDAC2 24 42 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne FFAR1 39 41 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne ADCYAP1R1 31 40 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne SMO 27 42 CC(=O)c1cccc(NC(=O)c2ccc(OCc3ccccc3)cc2)c1O ZINC000147236554 FI On-Demand Anodyne KCNK3 69 37 C#CCNC(=O)[C@@H](C)Oc1ccc(F)cc1S(N)(=O)=O ZINC000147236586 DB For-Sale Mild CA2 29 40 NC(=O)NCCNc1ccccc1S(=O)(=O)NC1CC1 ZINC000147236617 CC For-Sale Anodyne CCR8 97 40 NC(=O)NCCNc1ccccc1S(=O)(=O)NC1CC1 ZINC000147236617 CC For-Sale Anodyne SFRP1 87 37 NC(=O)NCCNc1ccccc1S(=O)(=O)NC1CC1 ZINC000147236617 CC For-Sale Anodyne WNT3 50 33 COCCN(CC(=O)O)C(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147236684 CD For-Sale Anodyne GPR88 0 43 CCCCCCCCNC(=O)N1C[C@H](C)[C@@H](C(=O)O)C1 ZINC000147236759 CF For-Sale Mild ASAH1 100 38 CCOc1ccc(NS(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147236809 HG On-Demand Mild AVPR1A 19 43 CCOc1ccc(NS(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147236809 HG On-Demand Mild MMP13 45 44 CCOc1ccc(NS(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147236809 HG On-Demand Mild ADAM17 37 40 CCOc1ccc(NS(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147236809 HG On-Demand Mild MMP1 24 40 CCOc1ccc(NS(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147236809 HG On-Demand Mild LIMK2 28 43 CCOc1ccc(NS(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147236809 HG On-Demand Mild L3MBTL3 62 38 CCNc1ncc(F)c(Nc2ccc(C#N)cc2F)n1 ZINC000147236827 CF For-Sale Mild SYK 36 52 CCOC(=O)C(C(=O)OCC)[C@H](c1ccccc1)N(CC)CC ZINC000147236841 DF For-Sale Anodyne AOC3 19 40 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147236843 EE On-Demand Bother BMP1 19 40 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147236843 EE On-Demand Bother MTNR1A 18 40 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147236843 EE On-Demand Bother MMP8 21 42 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147236843 EE On-Demand Bother ROCK2 28 42 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147236843 EE On-Demand Bother MMP1 20 42 CCc1ncc(C(=O)N2CCc3cc(OC)c(OC)cc3[C@@H]2c2ccccc2)s1 ZINC000147236848 HJ On-Demand Anodyne HCRTR1 15 40 CCc1ncc(C(=O)N2CCc3cc(OC)c(OC)cc3[C@@H]2c2ccccc2)s1 ZINC000147236848 HJ On-Demand Anodyne MTNR1B 28 46 CCNc1nc(Cl)nc(Oc2ccc3ccccc3c2)n1 ZINC000147236861 DH For-Sale Anodyne Q31945_CHEAL 0 40 CCNc1nc(Cl)nc(Oc2ccc3ccccc3c2)n1 ZINC000147236861 DH For-Sale Anodyne PPX1 0 47 CCc1ccc(OC[C@H](O)CNN2CCOCC2)cc1 ZINC000147236881 CC For-Sale Anodyne ADRB2 53 48 CCc1ccc(OC[C@H](O)CNN2CCOCC2)cc1 ZINC000147236881 CC For-Sale Anodyne ADRB1 67 60 CCc1ccc(OC[C@H](O)CNN2CCOCC2)cc1 ZINC000147236881 CC For-Sale Anodyne ADRB3 54 42 CCc1ccc(OC[C@H](O)CNN2CCOCC2)cc1 ZINC000147236881 CC For-Sale Anodyne ABCB1 0 42 COc1cc(C(=O)NNC(=O)Nc2ncc(C)s2)ccc1OC(C)C ZINC000147236908 FF On-Demand Reactive ENPP1 47 36 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147236932 EE On-Demand Bother BMP1 19 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147236932 EE On-Demand Bother MTNR1A 18 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147236932 EE On-Demand Bother MMP8 21 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147236932 EE On-Demand Bother ROCK2 28 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147236932 EE On-Demand Bother MMP1 20 42 Cc1cc(N(C)C)ccc1NC(=O)NC[C@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147236972 HH On-Demand Anodyne ADRB1 23 43 Cc1cc(N(C)C)ccc1NC(=O)NC[C@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147236972 HH On-Demand Anodyne PDS 53 42 CCOC(=O)C(C(=O)OCC)[C@@H](c1ccccc1)N(CC)CC ZINC000147237006 DF For-Sale Anodyne AOC3 19 40 CCc1ncc(C(=O)N2CCc3cc(OC)c(OC)cc3[C@H]2c2ccccc2)s1 ZINC000147237007 HJ On-Demand Anodyne HCRTR1 15 40 CCc1ncc(C(=O)N2CCc3cc(OC)c(OC)cc3[C@H]2c2ccccc2)s1 ZINC000147237007 HJ On-Demand Anodyne MTNR1B 28 46 CN(Cc1cscn1)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000147237047 EF On-Demand Anodyne DRD4 31 46 CN(Cc1cscn1)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000147237047 EF On-Demand Anodyne ACHE 22 41 CN(Cc1cscn1)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000147237047 EF On-Demand Anodyne SIGMAR1 34 46 CN(Cc1cscn1)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000147237047 EF On-Demand Anodyne CCR3 25 43 CN(Cc1cscn1)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000147237047 EF On-Demand Anodyne CYP3A4 17 40 CN(Cc1cscn1)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000147237047 EF On-Demand Anodyne MCHR1 30 48 CN(Cc1cscn1)C(=O)N[C@@H]1CCN(Cc2ccccc2)C1 ZINC000147237047 EF On-Demand Anodyne BIRC2 32 41 CCCCCCCCNC(=O)N1C[C@@H](C)[C@@H](C(=O)O)C1 ZINC000147237054 CF For-Sale Mild ASAH1 100 38 CNc1ncc(F)c(Nc2ccc(C#N)cc2F)n1 ZINC000147237063 CE For-Sale Mild SYK 32 55 CNc1ncc(F)c(Nc2ccc(C#N)cc2F)n1 ZINC000147237063 CE For-Sale Mild AURKA 15 40 Cn1ncc2c(-c3cccc4[nH]ccc34)nc(N3CCOCC3)nc21 ZINC000147237064 EE For-Sale Anodyne PIK3CA 19 48 Cn1ncc2c(-c3cccc4[nH]ccc34)nc(N3CCOCC3)nc21 ZINC000147237064 EE For-Sale Anodyne MTOR 22 49 Cn1ncc2c(-c3cccc4[nH]ccc34)nc(N3CCOCC3)nc21 ZINC000147237064 EE For-Sale Anodyne ATR 57 47 CCc1ccc(OC[C@@H](O)CNN2CCOCC2)cc1 ZINC000147237068 CC For-Sale Anodyne ADRB2 53 48 CCc1ccc(OC[C@@H](O)CNN2CCOCC2)cc1 ZINC000147237068 CC For-Sale Anodyne ADRB1 67 60 CCc1ccc(OC[C@@H](O)CNN2CCOCC2)cc1 ZINC000147237068 CC For-Sale Anodyne ADRB3 54 42 CCc1ccc(OC[C@@H](O)CNN2CCOCC2)cc1 ZINC000147237068 CC For-Sale Anodyne ABCB1 0 42 CCCCN(CCBr)S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147237119 GF For-Sale Reactive CA2 18 47 CCCCN(CCBr)S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147237119 GF For-Sale Reactive CA1 17 52 CCCCN(CCBr)S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147237119 GF For-Sale Reactive CA4 17 43 CCCCN(CCBr)S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147237119 GF For-Sale Reactive CA12 16 52 CCCCN(CCBr)S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147237119 GF For-Sale Reactive CA9 18 52 CCCCN(CCBr)S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147237119 GF For-Sale Reactive IDO1 33 41 CCCCN(CCBr)S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147237119 GF For-Sale Reactive MTCA1 28 40 CCCCN(CCBr)S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147237119 GF For-Sale Reactive P96878_MYCTU 39 41 CCCCN(CCBr)S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147237119 GF For-Sale Reactive RORC 18 41 CCCCN(CCBr)S(=O)(=O)c1ccc(NC(C)=O)cc1 ZINC000147237119 GF For-Sale Reactive Q9JN24_ECOLX 0 51 CCOC(=O)Cc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000147237129 BE For-Sale Anodyne GSTM2 40 38 O=C(NCc1ccc([N+](=O)[O-])cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147237150 FG On-Demand Bother NAMPT 48 40 Cc1cc(N(C)C)ccc1NC(=O)NC[C@@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147237168 HH On-Demand Anodyne ADRB1 23 43 Cc1cc(N(C)C)ccc1NC(=O)NC[C@@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147237168 HH On-Demand Anodyne PDS 53 42 CN(Cc1cscn1)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000147237225 EF On-Demand Anodyne DRD4 31 46 CN(Cc1cscn1)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000147237225 EF On-Demand Anodyne ACHE 22 41 CN(Cc1cscn1)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000147237225 EF On-Demand Anodyne DRD3 22 43 CN(Cc1cscn1)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000147237225 EF On-Demand Anodyne SIGMAR1 34 46 CN(Cc1cscn1)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000147237225 EF On-Demand Anodyne CCR3 25 43 CN(Cc1cscn1)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000147237225 EF On-Demand Anodyne CYP3A4 17 40 CN(Cc1cscn1)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000147237225 EF On-Demand Anodyne MCHR1 30 48 CN(Cc1cscn1)C(=O)N[C@H]1CCN(Cc2ccccc2)C1 ZINC000147237225 EF On-Demand Anodyne BIRC2 32 41 CCNc1ncnc(Nc2ccc(C#N)cc2F)c1CC ZINC000147237254 CG For-Sale Mild FLT1 0 44 CCCCCCCCNC(=O)N1CC(CC(=O)O)C1 ZINC000147237260 CE For-Sale Mild ASAH1 102 41 O=C(NCC(F)(F)F)Nc1cccc(-c2cnc3cc(-c4cccnc4)ccn23)c1 ZINC000147237264 HJ Annotated Anodyne GYRB 0 43 O=C(NCC(F)(F)F)Nc1cccc(-c2cnc3cc(-c4cccnc4)ccn23)c1 ZINC000147237264 HJ Annotated Anodyne BRAF 48 42 Nc1cc(NCC(F)F)cc(S(N)(=O)=O)c1 ZINC000147237277 CC For-Sale Anodyne CAH_METTE 40 37 O=C(NCc1ccc([N+](=O)[O-])cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147237340 EH On-Demand Bother CACNA1D 55 36 O=C(NCc1ccc([N+](=O)[O-])cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147237340 EH On-Demand Bother MDM2 49 31 COCCN(CC(=O)O)C(=O)C1[C@H]2CCCC[C@H]12 ZINC000147237396 CC On-Demand Anodyne ACE 0 47 N#Cc1ccc(NCCCCn2ccnc2)cn1 ZINC000147237422 BE On-Demand Mild CYP19A1 0 44 N#Cc1ccc(NCCCCn2ccnc2)cn1 ZINC000147237422 BE On-Demand Mild TBXAS1 45 43 N#Cc1ccc(NCCCCn2ccnc2)cn1 ZINC000147237422 BE On-Demand Mild HMOX1 15 44 N#Cc1ccc(NCCCCn2ccnc2)cn1 ZINC000147237422 BE On-Demand Mild HMOX2 50 43 N#Cc1ccc(NCCCCn2ccnc2)cn1 ZINC000147237422 BE On-Demand Mild QPCT 41 43 CCCCCCCCNC(=O)N[C@@](C)(C(=O)O)C(F)(F)F ZINC000147237479 DG For-Sale Mild CES2 53 41 CCCCCCCCNC(=O)N[C@@](C)(C(=O)O)C(F)(F)F ZINC000147237479 DG For-Sale Mild CES1 55 36 CCCCCCCCNC(=O)N[C@@](C)(C(=O)O)C(F)(F)F ZINC000147237479 DG For-Sale Mild EST1_PIG 75 41 CCCCCCCCNC(=O)N[C@@](C)(C(=O)O)C(F)(F)F ZINC000147237479 DG For-Sale Mild EPHX2 44 43 CCCCCCCCNC(=O)N[C@@](C)(C(=O)O)C(F)(F)F ZINC000147237479 DG For-Sale Mild CES2C 62 41 CCCCCCCCNC(=O)N[C@@](C)(C(=O)O)C(F)(F)F ZINC000147237479 DG For-Sale Mild JHE 0 41 CCCCCCCCNC(=O)N[C@@](C)(C(=O)O)C(F)(F)F ZINC000147237479 DG For-Sale Mild ASAH1 85 35 CNc1ncnc(Nc2ccc(C#N)cc2F)c1C ZINC000147237483 CF For-Sale Mild FLT1 0 44 CN(C)CCOc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147237529 HE On-Demand Bother USP7 47 43 CN(C)CCOc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147237529 HE On-Demand Bother USP47 59 43 O=C(NCc1ccc([N+](=O)[O-])cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147237547 EH On-Demand Bother CACNA1D 55 36 O=C(NCc1ccc([N+](=O)[O-])cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147237547 EH On-Demand Bother MDM2 49 31 COCCN(CC(=O)O)C(=O)C1[C@H]2CCCC[C@@H]12 ZINC000147237599 CC For-Sale Anodyne ACE 0 47 CCCCCCCCNC(=O)N[C@](C)(C(=O)O)C(F)(F)F ZINC000147237679 DG For-Sale Mild CES2 53 41 CCCCCCCCNC(=O)N[C@](C)(C(=O)O)C(F)(F)F ZINC000147237679 DG For-Sale Mild CES1 55 36 CCCCCCCCNC(=O)N[C@](C)(C(=O)O)C(F)(F)F ZINC000147237679 DG For-Sale Mild EST1_PIG 75 41 CCCCCCCCNC(=O)N[C@](C)(C(=O)O)C(F)(F)F ZINC000147237679 DG For-Sale Mild EPHX2 44 43 CCCCCCCCNC(=O)N[C@](C)(C(=O)O)C(F)(F)F ZINC000147237679 DG For-Sale Mild CES2C 62 41 CCCCCCCCNC(=O)N[C@](C)(C(=O)O)C(F)(F)F ZINC000147237679 DG For-Sale Mild JHE 0 41 CCCCCCCCNC(=O)N[C@](C)(C(=O)O)C(F)(F)F ZINC000147237679 DG For-Sale Mild ASAH1 85 35 O=C(NCc1ccc([N+](=O)[O-])cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147237768 EH On-Demand Bother CACNA1D 55 36 O=C(NCc1ccc([N+](=O)[O-])cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147237768 EH On-Demand Bother MDM2 49 31 C[C@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147237801 CD On-Demand Anodyne MME 49 39 C[C@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147237801 CD On-Demand Anodyne CPA1 25 40 C[C@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147237801 CD On-Demand Anodyne CAPN2 55 33 C[C@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147237801 CD On-Demand Anodyne CPA3 0 40 C[C@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147237801 CD On-Demand Anodyne Q9JN24_ECOLX 0 41 C[C@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147237801 CD On-Demand Anodyne TMPRSS11D 45 36 CN(c1cccc(Cl)c1)S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147237810 HH On-Demand Mild CACNA1B 30 49 CN(c1cccc(Cl)c1)S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147237810 HH On-Demand Mild SFRP1 15 40 COCCN(CC(=O)O)C(=O)C1[C@@H]2CCCC[C@@H]12 ZINC000147237815 CC On-Demand Anodyne ACE 0 47 CCCCCCCCNC(=O)N1CCOC[C@@H]1C(=O)O ZINC000147237882 CD For-Sale Mild ASAH1 101 47 O=C(NCc1ccc([N+](=O)[O-])cc1)[C@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147237985 GH On-Demand Bother CACNA1D 48 32 COc1cc(C(=O)NCc2ccccc2C)ccc1OCC(C)C ZINC000147237999 EH On-Demand Anodyne PPARG 15 43 COc1cc(C(=O)NCc2ccccc2C)ccc1OCC(C)C ZINC000147237999 EH On-Demand Anodyne PPARA 18 43 COc1cc(C(=O)NCc2ccccc2C)ccc1OCC(C)C ZINC000147237999 EH On-Demand Anodyne PPARD 23 43 COc1cc(C(=O)NCc2ccccc2C)ccc1OCC(C)C ZINC000147237999 EH On-Demand Anodyne SCN10A 19 43 COc1cc(C(=O)NCc2ccccc2C)ccc1OCC(C)C ZINC000147237999 EH On-Demand Anodyne MT-ND1 15 42 COc1cc(C(=O)NCc2ccccc2C)ccc1OCC(C)C ZINC000147237999 EH On-Demand Anodyne KCNK3 42 34 CCCC[C@H](N)C(=O)NN(C)C ZINC000147238002 AC For-Sale Reactive DPP4 0 53 CCCC[C@H](N)C(=O)NN(C)C ZINC000147238002 AC For-Sale Reactive DPP7 20 53 CCCC[C@H](N)C(=O)NN(C)C ZINC000147238002 AC For-Sale Reactive DPP8 0 48 CCCC[C@H](N)C(=O)NN(C)C ZINC000147238002 AC For-Sale Reactive DPP9 0 48 CCCC[C@H](N)C(=O)NN(C)C ZINC000147238002 AC For-Sale Reactive PLC 52 37 CCCC[C@H](N)C(=O)NN(C)C ZINC000147238002 AC For-Sale Reactive NOD1 70 37 CCCC[C@H](N)C(=O)NN(C)C ZINC000147238002 AC For-Sale Reactive CQSS 43 40 COC(=O)CCCCn1c(C(=O)O)cc2ccccc21 ZINC000147238028 CF For-Sale Anodyne CCR2 17 55 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)Nc3ccc(F)cc3)cc2)CC1 ZINC000147238045 GG On-Demand Mild SFRP1 42 36 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)Nc3ccc(F)cc3)cc2)CC1 ZINC000147238045 GG On-Demand Mild LIMK2 25 42 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)Nc3ccc(F)cc3)cc2)CC1 ZINC000147238045 GG On-Demand Mild L3MBTL3 73 41 C[C@@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147238056 CD On-Demand Anodyne MME 49 39 C[C@@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147238056 CD On-Demand Anodyne CPA1 25 40 C[C@@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147238056 CD On-Demand Anodyne CAPN2 55 33 C[C@@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147238056 CD On-Demand Anodyne CPA3 0 40 C[C@@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147238056 CD On-Demand Anodyne Q9JN24_ECOLX 0 41 C[C@@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147238056 CD On-Demand Anodyne TMPRSS11D 45 36 CCCCCCCCNC(=O)N1CCOC[C@H]1C(=O)O ZINC000147238111 CD For-Sale Mild ASAH1 101 47 CCCC[C@@H](N)C(=O)NN(C)C ZINC000147238201 AC For-Sale Reactive DPP4 0 53 CCCC[C@@H](N)C(=O)NN(C)C ZINC000147238201 AC For-Sale Reactive DPP7 20 53 CCCC[C@@H](N)C(=O)NN(C)C ZINC000147238201 AC For-Sale Reactive DPP8 0 48 CCCC[C@@H](N)C(=O)NN(C)C ZINC000147238201 AC For-Sale Reactive DPP9 0 48 CCCC[C@@H](N)C(=O)NN(C)C ZINC000147238201 AC For-Sale Reactive PLC 52 37 CCCC[C@@H](N)C(=O)NN(C)C ZINC000147238201 AC For-Sale Reactive NOD1 70 37 CCCC[C@@H](N)C(=O)NN(C)C ZINC000147238201 AC For-Sale Reactive CQSS 43 40 O=C(c1cccc2c1OCCN2)N(CCO)C1CCCC1 ZINC000147238205 CD For-Sale Anodyne ACE 42 42 O=C(NCc1ccc([N+](=O)[O-])cc1)[C@@H]1C[C@H]1c1cccc(Br)c1 ZINC000147238213 GH On-Demand Bother CACNA1D 48 32 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCOCC2)cc1C(F)(F)F ZINC000147238220 HE On-Demand Anodyne TTK 20 42 C[C@H](CNS(=O)(=O)Cc1ccccc1[N+](=O)[O-])CC(=O)O ZINC000147238247 DD On-Demand Bother COLA 123 50 C[C@H](CNS(=O)(=O)Cc1ccccc1[N+](=O)[O-])CC(=O)O ZINC000147238247 DD On-Demand Bother PQSD 0 42 CC(=O)CC#Cc1ccccc1 ZINC000147238263 AE For-Sale Mild FFAR1 29 45 CCCCCCCCNC(=O)NCC[C@@H](C)CCC(=O)O ZINC000147238343 DH For-Sale Mild FOLH1 35 41 CCCCCCCCNC(=O)NCC[C@@H](C)CCC(=O)O ZINC000147238343 DH For-Sale Mild FABP2 0 44 CCCCCCCCNC(=O)NCC[C@@H](C)CCC(=O)O ZINC000147238343 DH For-Sale Mild PLA2G2C 0 44 CCCCCCCCNC(=O)NCC[C@@H](C)CCC(=O)O ZINC000147238343 DH For-Sale Mild CPT1A 40 47 CCCCCCCCNC(=O)NCC[C@@H](C)CCC(=O)O ZINC000147238343 DH For-Sale Mild EPHX2 24 57 CCCCCCCCNC(=O)NCC[C@@H](C)CCC(=O)O ZINC000147238343 DH For-Sale Mild Q6UB75_PIG 0 48 CCCCCCCCNC(=O)NCC[C@@H](C)CCC(=O)O ZINC000147238343 DH For-Sale Mild FABP5 15 44 CCCCCCCCNC(=O)NCC[C@@H](C)CCC(=O)O ZINC000147238343 DH For-Sale Mild ASAH1 82 34 CCCCCCCCNC(=O)NCC[C@@H](C)CCC(=O)O ZINC000147238343 DH For-Sale Mild SLC22A20 0 44 CCCCCCCCNC(=O)NCC[C@@H](C)CCC(=O)O ZINC000147238343 DH For-Sale Mild NOD1 75 40 CCCCCCCCNC(=O)NCC[C@@H](C)CCC(=O)O ZINC000147238343 DH For-Sale Mild CQSS 55 36 CC(C)C(=O)NC12C[C@H]3C[C@@H](CC(O)(C3)C1)C2 ZINC000147238382 BD On-Demand Anodyne EPHX2 22 40 O=C(NCc1ccc([N+](=O)[O-])cc1)[C@@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147238391 GH On-Demand Bother CACNA1D 48 32 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCOCC2)cc1C(F)(F)F ZINC000147238396 HE On-Demand Anodyne TTK 20 42 C[C@@H](CNS(=O)(=O)Cc1ccccc1[N+](=O)[O-])CC(=O)O ZINC000147238402 DD On-Demand Bother COLA 123 50 C[C@@H](CNS(=O)(=O)Cc1ccccc1[N+](=O)[O-])CC(=O)O ZINC000147238402 DD On-Demand Bother PQSD 0 42 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccs1 ZINC000147238433 CG On-Demand Anodyne BMP1 47 33 OCCN1CCN(c2cc(F)ccc2F)CC1 ZINC000147238442 BD On-Demand Anodyne HTR1A 28 48 OCCN1CCN(c2cc(F)ccc2F)CC1 ZINC000147238442 BD On-Demand Anodyne DRD2 30 48 OCCN1CCN(c2cc(F)ccc2F)CC1 ZINC000147238442 BD On-Demand Anodyne DRD1 28 44 OCCN1CCN(c2cc(F)ccc2F)CC1 ZINC000147238442 BD On-Demand Anodyne DRD4 31 41 OCCN1CCN(c2cc(F)ccc2F)CC1 ZINC000147238442 BD On-Demand Anodyne HTR2C 16 44 OCCN1CCN(c2cc(F)ccc2F)CC1 ZINC000147238442 BD On-Demand Anodyne ADRA1A 17 41 OCCN1CCN(c2cc(F)ccc2F)CC1 ZINC000147238442 BD On-Demand Anodyne ADRA1B 21 44 OCCN1CCN(c2cc(F)ccc2F)CC1 ZINC000147238442 BD On-Demand Anodyne DRD3 21 41 CCN(CCC(=O)O)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147238459 CE For-Sale Anodyne GPR88 0 48 COc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1NC(C)=O ZINC000147238489 ED On-Demand Anodyne QRFPR 40 33 CC1(C)C[C@@H]1C(=O)c1ccccn1 ZINC000147238519 AE For-Sale Anodyne GRM4 50 40 CCCCCCCCNC(=O)NCC[C@H](C)CCC(=O)O ZINC000147238555 DH For-Sale Mild FOLH1 35 41 CCCCCCCCNC(=O)NCC[C@H](C)CCC(=O)O ZINC000147238555 DH For-Sale Mild FABP2 0 44 CCCCCCCCNC(=O)NCC[C@H](C)CCC(=O)O ZINC000147238555 DH For-Sale Mild PLA2G2C 0 44 CCCCCCCCNC(=O)NCC[C@H](C)CCC(=O)O ZINC000147238555 DH For-Sale Mild CPT1A 40 47 CCCCCCCCNC(=O)NCC[C@H](C)CCC(=O)O ZINC000147238555 DH For-Sale Mild EPHX2 24 57 CCCCCCCCNC(=O)NCC[C@H](C)CCC(=O)O ZINC000147238555 DH For-Sale Mild Q6UB75_PIG 0 48 CCCCCCCCNC(=O)NCC[C@H](C)CCC(=O)O ZINC000147238555 DH For-Sale Mild FABP5 15 44 CCCCCCCCNC(=O)NCC[C@H](C)CCC(=O)O ZINC000147238555 DH For-Sale Mild ASAH1 82 34 CCCCCCCCNC(=O)NCC[C@H](C)CCC(=O)O ZINC000147238555 DH For-Sale Mild SLC22A20 0 44 CCCCCCCCNC(=O)NCC[C@H](C)CCC(=O)O ZINC000147238555 DH For-Sale Mild NOD1 75 40 CCCCCCCCNC(=O)NCC[C@H](C)CCC(=O)O ZINC000147238555 DH For-Sale Mild CQSS 55 36 C[C@H](CNS(=O)(=O)c1cc(Cl)ccc1C#N)CC(=O)O ZINC000147238575 DD On-Demand Mild TRPV4 44 35 O=C1CCCc2cc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)ccc2N1 ZINC000147238618 FF On-Demand Anodyne PKM 38 50 COc1ccc(OCCN2[C@@H]3CC[C@@H]2CC(Br)C3)cc1 ZINC000147238627 EG For-Sale Reactive LTA4H 33 44 CCN(CCC(=O)O)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147238639 CE For-Sale Anodyne GPR88 0 48 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccs1 ZINC000147238643 CG On-Demand Anodyne BMP1 47 33 COc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1NC(C)=O ZINC000147238671 ED On-Demand Anodyne QRFPR 40 33 O=C(c1cccc2c1OCCN2)N1CCN(C2CC2)CC1 ZINC000147238680 CD For-Sale Anodyne L3MBTL1 0 46 O=C(c1cccc2c1OCCN2)N1CCN(C2CC2)CC1 ZINC000147238680 CD For-Sale Anodyne L3MBTL3 80 46 O=C(c1cccc2c1OCCN2)N1CCN(C2CC2)CC1 ZINC000147238680 CD For-Sale Anodyne MBTD1 0 40 O=C(c1cccc2c1OCCN2)N1CCN(C2CC2)CC1 ZINC000147238680 CD For-Sale Anodyne TP53BP1 0 46 CCCCCCCCNC(=O)NC[C@](C)(O)CC(=O)O ZINC000147238774 CD For-Sale Mild CPT1A 24 44 CCCCCCCCNC(=O)NC[C@](C)(O)CC(=O)O ZINC000147238774 CD For-Sale Mild EPHX2 50 51 CCCCCCCCNC(=O)NC[C@](C)(O)CC(=O)O ZINC000147238774 CD For-Sale Mild ASAH1 73 35 C[C@@H](CNS(=O)(=O)c1cc(Cl)ccc1C#N)CC(=O)O ZINC000147238786 DD On-Demand Mild TRPV4 44 35 O=C(O)CCc1ncccc1F ZINC000147238797 AD For-Sale Anodyne TBXAS1 18 40 O=C(O)CCc1ncccc1F ZINC000147238797 AD For-Sale Anodyne FFAR1 59 41 O=C(O)CCc1ncccc1F ZINC000147238797 AD For-Sale Anodyne FFAR4 47 35 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N(C)Cc3ccccc3)cc2)s1 ZINC000147238809 HH On-Demand Anodyne GRM4 18 40 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N(C)Cc3ccccc3)cc2)s1 ZINC000147238809 HH On-Demand Anodyne LIMK2 42 36 COc1ccc(OCCN2[C@H]3CC[C@@H]2CC(Br)C3)cc1 ZINC000147238820 EG For-Sale Reactive LTA4H 33 44 O=C1CCCc2cc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)ccc2N1 ZINC000147238829 FF On-Demand Anodyne PKM 38 50 CC(C)[C@H](Nc1ccc(C(F)(F)F)cc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147238851 GJ On-Demand Mild CCR1 43 39 CCN(CCC(=O)O)C(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147238860 CE For-Sale Anodyne GPR88 0 48 O=C1CN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2Cl)CCN1 ZINC000147238869 GC On-Demand Anodyne NPY2R 38 43 COc1ccccc1CNC(=O)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147238874 HF On-Demand Anodyne EDNRB 15 41 COc1ccccc1CNC(=O)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147238874 HF On-Demand Anodyne MAP1 100 41 COc1ccccc1CNC(=O)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147238874 HF On-Demand Anodyne LIMK2 28 41 CCNC(=O)c1ccc(NCCNC(N)=O)c([N+](=O)[O-])c1 ZINC000147238935 CC For-Sale Bother DRTS_TOXGO 15 41 CCNC(=O)c1ccc(NCCNC(N)=O)c([N+](=O)[O-])c1 ZINC000147238935 CC For-Sale Bother TAAR1 20 49 CCCCCCCCNC(=O)NC[C@@](C)(O)CC(=O)O ZINC000147239010 CD For-Sale Mild CPT1A 24 44 CCCCCCCCNC(=O)NC[C@@](C)(O)CC(=O)O ZINC000147239010 CD For-Sale Mild EPHX2 50 51 CCCCCCCCNC(=O)NC[C@@](C)(O)CC(=O)O ZINC000147239010 CD For-Sale Mild ASAH1 73 35 C[C@H](CNS(=O)(=O)c1ccccc1C(F)(F)F)CC(=O)O ZINC000147239017 EE On-Demand Anodyne RBP4 40 34 C[C@H](CNS(=O)(=O)c1ccccc1C(F)(F)F)CC(=O)O ZINC000147239017 EE On-Demand Anodyne SFRP1 79 35 C[C@H](CNS(=O)(=O)c1ccccc1C(F)(F)F)CC(=O)O ZINC000147239017 EE On-Demand Anodyne WNT3 57 35 COc1ccc(OCCN2[C@H]3CC[C@H]2CC(Br)C3)cc1 ZINC000147239031 EG For-Sale Reactive LTA4H 33 44 O=C1CCCc2cc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)ccc2N1 ZINC000147239040 FF On-Demand Anodyne PKM 38 50 CC1=NN(c2cccnc2)C(=O)C1 ZINC000147239042 AD For-Sale Anodyne CHRNA4 15 40 CC1=NN(c2cccnc2)C(=O)C1 ZINC000147239042 AD For-Sale Anodyne CYP2A6 18 43 CCCNC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147239077 CC For-Sale Anodyne CA2 25 41 CCCNC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147239077 CC For-Sale Anodyne CA1 22 41 CCCNC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147239077 CC For-Sale Anodyne CA9 15 41 CCN(CCC(=O)O)C(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147239090 CE For-Sale Anodyne GPR88 0 48 O=C1CN(c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2Cl)CCN1 ZINC000147239113 GC On-Demand Anodyne NPY2R 38 43 C[C@@H](CNS(=O)(=O)c1ccccc1C(F)(F)F)CC(=O)O ZINC000147239225 EE On-Demand Anodyne RBP4 40 34 C[C@@H](CNS(=O)(=O)c1ccccc1C(F)(F)F)CC(=O)O ZINC000147239225 EE On-Demand Anodyne SFRP1 79 35 C[C@@H](CNS(=O)(=O)c1ccccc1C(F)(F)F)CC(=O)O ZINC000147239225 EE On-Demand Anodyne WNT3 57 35 CCCCCCCCNC(=O)NC[C@H](O)C(=O)O ZINC000147239228 CD For-Sale Mild CPT1A 25 47 CCCCCCCCNC(=O)NC[C@H](O)C(=O)O ZINC000147239228 CD For-Sale Mild FAAH 0 40 CCCCCCCCNC(=O)NC[C@H](O)C(=O)O ZINC000147239228 CD For-Sale Mild S1PR2 30 40 CCCCCCCCNC(=O)NC[C@H](O)C(=O)O ZINC000147239228 CD For-Sale Mild EPHX2 62 54 CCCCCCCCNC(=O)NC[C@H](O)C(=O)O ZINC000147239228 CD For-Sale Mild ASAH1 87 34 CCCCCCCCNC(=O)NC[C@H](O)C(=O)O ZINC000147239228 CD For-Sale Mild NOD1 46 37 CCCCCCCCNC(=O)NC[C@H](O)C(=O)O ZINC000147239228 CD For-Sale Mild CQSS 60 38 O=C1CCCc2cc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)ccc2N1 ZINC000147239262 FF On-Demand Anodyne PKM 38 50 CN(C)c1nc(N)nc(Oc2ccc3ccccc3c2)n1 ZINC000147239295 CE For-Sale Anodyne DYR_PNECA 17 42 CN(C)c1nc(N)nc(Oc2ccc3ccccc3c2)n1 ZINC000147239295 CE For-Sale Anodyne CYP2A5 0 43 Cc1ccc(NS(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1C ZINC000147239300 GG On-Demand Mild PKM 34 47 Cc1ccc(NS(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1C ZINC000147239300 GG On-Demand Mild LIMK2 19 41 Cc1ccc(NS(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1C ZINC000147239300 GG On-Demand Mild L3MBTL3 79 39 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne F2 94 48 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne PLG 46 42 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne PRSS1 40 44 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne ACE 80 48 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne FKBP1A 50 42 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne LHCGR 42 42 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne OPRM1 57 53 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne OPRD1 49 53 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CELA1 61 42 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne ELANE 76 52 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne MME 31 42 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne ANPEP 16 49 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne TACR1 25 50 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne TRHR 95 54 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CTSD 17 41 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne HLA-DRB3 61 38 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CMA1 43 47 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CTRA_BOVIN 75 42 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne KLK3 68 35 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CTSB 53 45 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne PAPA1_CARPA 55 37 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne TRY1_BOVIN 118 42 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne NTSR1 165 53 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne NTSR2 113 45 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CTSG 53 42 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CTSK 42 47 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CTSL 40 47 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CPA1 29 44 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CACNA1B 56 37 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne NPFFR2 47 47 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne C3AR1 28 52 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne HLA-A 82 44 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne PREP 51 54 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CAPNS1 73 36 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CELA2A 63 42 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne REN 40 44 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne REN1 68 47 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne LNPEP 23 40 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne LGMN 98 49 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne PLAT 17 43 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne SORT1 60 45 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne TGM1 17 51 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CTSS 20 47 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CAPN1 105 46 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CASP1 18 44 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CTRC 41 47 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CAPN2 131 40 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne CTSE 27 41 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne ACE2 47 44 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne TGM2 23 51 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne LAP3 22 43 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne KLK5 45 49 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne C5AR1 17 43 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne MARS 41 35 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne KLK1 28 48 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne FPR1 42 35 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne NPR 74 38 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne XIAP 78 56 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne BRCA1 79 43 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne NPFFR1 20 44 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne Q9NAW4_PLAFA 37 40 CC(C)C[C@H](NC(=O)[C@H]1CCC(=O)N1C(=O)OCc1ccccc1)C(=O)N1CCC[C@H]1C(N)=O ZINC000147239322 JD For-Sale Anodyne TMPRSS11D 75 48 CCCCN(CCBr)S(=O)(=O)c1cccc2cnccc12 ZINC000147239374 FG For-Sale Reactive TRPV1 0 43 CCCCN(CCBr)S(=O)(=O)c1cccc2cnccc12 ZINC000147239374 FG For-Sale Reactive P2RX7 28 43 CCCCN(CCBr)S(=O)(=O)c1cccc2cnccc12 ZINC000147239374 FG For-Sale Reactive Q95J97_RABIT 0 46 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(N2CCOCC2)cn1 ZINC000147239416 ED On-Demand Anodyne STAT6 62 35 CCCCCCCCNC(=O)NC[C@@H](O)C(=O)O ZINC000147239437 CD For-Sale Mild CPT1A 25 47 CCCCCCCCNC(=O)NC[C@@H](O)C(=O)O ZINC000147239437 CD For-Sale Mild FAAH 0 40 CCCCCCCCNC(=O)NC[C@@H](O)C(=O)O ZINC000147239437 CD For-Sale Mild S1PR2 30 40 CCCCCCCCNC(=O)NC[C@@H](O)C(=O)O ZINC000147239437 CD For-Sale Mild EPHX2 62 54 CCCCCCCCNC(=O)NC[C@@H](O)C(=O)O ZINC000147239437 CD For-Sale Mild ASAH1 87 34 CCCCCCCCNC(=O)NC[C@@H](O)C(=O)O ZINC000147239437 CD For-Sale Mild NOD1 46 37 CCCCCCCCNC(=O)NC[C@@H](O)C(=O)O ZINC000147239437 CD For-Sale Mild CQSS 60 38 CCc1ncc(C(=O)NCC(=O)Nc2c(C)cccc2C)s1 ZINC000147239458 DF On-Demand Anodyne LCK 18 44 CCc1ncc(C(=O)NCC(=O)Nc2c(C)cccc2C)s1 ZINC000147239458 DF On-Demand Anodyne FYN 18 40 CCc1ncc(C(=O)NCC(=O)Nc2c(C)cccc2C)s1 ZINC000147239458 DF On-Demand Anodyne FGR 19 40 Cc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1F ZINC000147239496 DF On-Demand Anodyne LEF 49 38 CCOC[C@H](C)NC(=O)Nc1ccc(OCC(F)(F)F)c(C#N)c1 ZINC000147239546 EG On-Demand Mild ADRB1 44 35 CCOC[C@H](C)NC(=O)Nc1ccc(OCC(F)(F)F)c(C#N)c1 ZINC000147239546 EG On-Demand Mild XDH 40 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(N2CCOCC2)cn1 ZINC000147239614 ED On-Demand Anodyne STAT6 62 35 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild ACE 41 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild GHRHR 70 33 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild P2RY12 122 33 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild MME 42 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild MC4R 71 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild TRY2_BOVIN 85 36 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild CCKAR 37 48 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild NPFFR2 45 33 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild CYP51A1 24 47 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild DPP4 28 43 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild MC3R 39 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild MC5R 56 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild CTSS 24 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild CAPN1 28 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild ACE2 51 39 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild ST14 101 37 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild AMP1_PLAFQ 18 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild DPP8 30 44 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild DPP9 21 44 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild BLA1_STEMA 45 36 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239624 FF On-Demand Mild TMPRSS6 52 33 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild CPT1A 48 49 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild PLA2G4B 63 37 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild CES2 18 41 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild EST1_PIG 15 41 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild EPHX2 29 53 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild CES2C 23 41 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild JHE 0 41 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild ASAH1 83 33 CCCCCCCCNC(=O)NCCOCC(=O)O ZINC000147239627 CD For-Sale Mild ACAT 0 41 Cn1cc(Cc2c[nH]cn2)c2cc(N)ccc21 ZINC000147239628 BE For-Sale Anodyne ADRA1D 26 40 Cc1cc(C(=O)NCC(=O)Nc2c(C)cccc2C)cc([N+](=O)[O-])c1 ZINC000147239685 EF On-Demand Bother METC 0 55 Cc1ccc(S(=O)(=O)N[C@H]2C[C@@H]2c2ccccc2)cc1F ZINC000147239715 DF On-Demand Anodyne LEF 49 38 Cc1c(NC(=O)c2ccccc2)cccc1NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147239758 HK On-Demand Anodyne KCNK3 62 43 CC(C)NS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147239820 DC For-Sale Anodyne CA2 39 42 CC(C)NS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147239820 DC For-Sale Anodyne CA1 35 42 CC(C)NS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147239820 DC For-Sale Anodyne CA7 16 40 CC(C)NS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147239820 DC For-Sale Anodyne CA14 25 40 CC(C)NS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147239820 DC For-Sale Anodyne CA12 24 42 CC(C)NS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147239820 DC For-Sale Anodyne ADAMTS4 41 37 CC(C)NS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147239820 DC For-Sale Anodyne CA9 25 42 CC(C)NS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147239820 DC For-Sale Anodyne LEF 48 37 CC(C)NS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147239820 DC For-Sale Anodyne CYNT 40 36 Cc1nn(C(F)F)c(C)c1CC(=O)Nc1ccc(N2CCOCC2)cn1 ZINC000147239821 FE On-Demand Anodyne STAT6 56 34 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild ACE 41 42 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild GHRHR 70 33 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild P2RY12 122 33 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild MME 42 42 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild MC4R 71 41 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild TRY2_BOVIN 85 36 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild CCKAR 37 48 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild NPFFR2 45 33 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild CYP51A1 24 47 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild DPP4 28 43 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild MC3R 39 41 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild MC5R 56 41 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild CTSS 24 40 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild CAPN1 28 42 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild ACE2 51 39 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild ST14 101 37 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild AMP1_PLAFQ 18 40 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild DPP8 30 44 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild DPP9 21 44 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild BLA1_STEMA 45 36 N#CC1CCN(C(=O)[C@@H](Cc2ccccc2)NC(=O)c2cccs2)CC1 ZINC000147239828 FF On-Demand Mild TMPRSS6 52 33 COc1ccccc1CCNC(=O)N(C)Cc1cscn1 ZINC000147239850 DF On-Demand Anodyne BMP1 41 33 CCCCCCCCNC(=O)N1CCCC[C@@H]1CC(=O)O ZINC000147239860 CG For-Sale Mild TPP2 22 43 CCCCCCCCNC(=O)N1CCCC[C@@H]1CC(=O)O ZINC000147239860 CG For-Sale Mild ASAH1 100 40 Cc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1F ZINC000147239909 DF On-Demand Anodyne LEF 49 38 CCCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147239910 DD On-Demand Anodyne ACACA 38 42 CCCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147239910 DD On-Demand Anodyne ADAM17 27 40 CCCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147239910 DD On-Demand Anodyne PLA2G4B 61 34 CCCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147239910 DD On-Demand Anodyne MMP9 31 41 CCCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147239910 DD On-Demand Anodyne MMP7 35 42 CCCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147239910 DD On-Demand Anodyne ADAMTS4 60 37 CCCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147239910 DD On-Demand Anodyne MMP1 29 52 c1ccc([C@H](Cc2ncc[nH]2)c2ccccn2)cc1 ZINC000147239914 BG For-Sale Anodyne HRH1 23 46 Cc1c(NC(=O)c2ccccc2)cccc1NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147239969 HK On-Demand Anodyne KCNK3 62 43 COC[C@H](C)NC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147239983 DC For-Sale Anodyne SDH1 0 40 CCCCCCCCNC(=O)N1CCCC[C@H]1CC(=O)O ZINC000147240068 CG For-Sale Mild TPP2 22 43 CCCCCCCCNC(=O)N1CCCC[C@H]1CC(=O)O ZINC000147240068 CG For-Sale Mild ASAH1 100 40 CCCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147240069 DD On-Demand Anodyne ACACA 38 42 CCCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147240069 DD On-Demand Anodyne ADAM17 27 40 CCCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147240069 DD On-Demand Anodyne PLA2G4B 61 34 CCCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147240069 DD On-Demand Anodyne MMP9 31 41 CCCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147240069 DD On-Demand Anodyne MMP7 35 42 CCCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147240069 DD On-Demand Anodyne ADAMTS4 60 37 CCCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147240069 DD On-Demand Anodyne MMP1 29 52 CN(C)NC(=O)[C@@H]1Cc2ccccc2CN1 ZINC000147240102 BC For-Sale Reactive MC4R 37 42 CN(C)NC(=O)[C@@H]1Cc2ccccc2CN1 ZINC000147240102 BC For-Sale Reactive PNMT 16 45 c1ccc([C@@H](Cc2ncc[nH]2)c2ccccn2)cc1 ZINC000147240120 BG For-Sale Anodyne HRH1 23 46 O=S(=O)(c1ccccc1N1CCC(CBr)CC1)C(F)(F)F ZINC000147240131 GH For-Sale Reactive SFRP1 59 34 COC[C@@H](C)NC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147240149 DC For-Sale Anodyne SDH1 0 40 Cc1c(NC(=O)c2ccccc2)cccc1NC(=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147240219 HK On-Demand Anodyne KCNK3 62 43 C[C@H](CNS(=O)(=O)CCc1ccccc1)CC(=O)O ZINC000147240290 CD On-Demand Anodyne MMP8 25 55 C[C@H](CNS(=O)(=O)CCc1ccccc1)CC(=O)O ZINC000147240290 CD On-Demand Anodyne CASP1 20 47 C[C@H](CNS(=O)(=O)CCc1ccccc1)CC(=O)O ZINC000147240290 CD On-Demand Anodyne CAPN2 45 31 C[C@H](CNS(=O)(=O)CCc1ccccc1)CC(=O)O ZINC000147240290 CD On-Demand Anodyne MMP12 27 52 CCC[C@@H](NC(N)=O)C(=O)NCc1cccc(N2CCOC2=O)c1 ZINC000147240301 ED On-Demand Anodyne PCSK5 52 33 CCC[C@@H](NC(N)=O)C(=O)NCc1cccc(N2CCOC2=O)c1 ZINC000147240301 ED On-Demand Anodyne FURIN 51 34 CCC[C@@H](NC(N)=O)C(=O)NCc1cccc(N2CCOC2=O)c1 ZINC000147240301 ED On-Demand Anodyne CARM1 43 35 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild FABP4 23 68 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild CPT1A 47 51 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild PLA2G4B 43 35 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild FAAH 0 55 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild S1PR2 30 44 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild EPHX2 41 81 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild FABP3 42 55 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild FABP5 23 68 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild FABP1 18 55 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild ASAH1 99 36 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild LASR 44 31 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild NOD1 62 40 CCCCCCCCNC(=O)NCCCCCC(=O)O ZINC000147240305 CG For-Sale Mild CQSS 64 39 CN(C)C(=O)NCCNc1nc(Cl)nc2ccccc12 ZINC000147240314 CD On-Demand Anodyne SLC2A1 0 40 CN(C)C(=O)NCCNc1nc(Cl)nc2ccccc12 ZINC000147240314 CD On-Demand Anodyne HT1 0 40 CN(C)NC(=O)[C@H]1Cc2ccccc2CN1 ZINC000147240325 BC For-Sale Reactive MC4R 37 42 CN(C)NC(=O)[C@H]1Cc2ccccc2CN1 ZINC000147240325 BC For-Sale Reactive PNMT 16 45 N#Cc1ccc(OCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147240339 CD On-Demand Mild HTR1B 17 42 N#Cc1ccc(OCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147240339 CD On-Demand Mild CPT1A 39 51 N#Cc1ccc(OCC(=O)N2CCC(C#N)CC2)cc1 ZINC000147240339 CD On-Demand Mild MEN1 42 35 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(NC(=O)c3ccccc3)c1C)C2 ZINC000147240443 HI On-Demand Anodyne ROCK2 32 46 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(NC(=O)c3ccccc3)c1C)C2 ZINC000147240443 HI On-Demand Anodyne GPR35 28 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(NC(=O)c3ccccc3)c1C)C2 ZINC000147240443 HI On-Demand Anodyne KCNK3 32 41 C[C@@H](CNS(=O)(=O)CCc1ccccc1)CC(=O)O ZINC000147240484 CD On-Demand Anodyne MMP8 25 55 C[C@@H](CNS(=O)(=O)CCc1ccccc1)CC(=O)O ZINC000147240484 CD On-Demand Anodyne CASP1 20 47 C[C@@H](CNS(=O)(=O)CCc1ccccc1)CC(=O)O ZINC000147240484 CD On-Demand Anodyne CAPN2 45 31 C[C@@H](CNS(=O)(=O)CCc1ccccc1)CC(=O)O ZINC000147240484 CD On-Demand Anodyne MMP12 27 52 CCCCCCCCNC(=O)N(CC(=O)O)CC(C)C ZINC000147240486 CG For-Sale Mild CPT1A 37 40 CCCCCCCCNC(=O)N(CC(=O)O)CC(C)C ZINC000147240486 CG For-Sale Mild S1PR2 47 36 CCCCCCCCNC(=O)N(CC(=O)O)CC(C)C ZINC000147240486 CG For-Sale Mild EPHX2 25 42 CCCCCCCCNC(=O)N(CC(=O)O)CC(C)C ZINC000147240486 CG For-Sale Mild ASAH1 60 31 CCOC(=O)c1c(-c2ccccc2)nc(-c2ccccc2)nc1N(C)C ZINC000147240515 EI For-Sale Anodyne DHODH 24 44 CCOC(=O)c1c(-c2ccccc2)nc(-c2ccccc2)nc1N(C)C ZINC000147240515 EI For-Sale Anodyne TSPO 35 44 CCOC(=O)c1c(-c2ccccc2)nc(-c2ccccc2)nc1N(C)C ZINC000147240515 EI For-Sale Anodyne SOAT1 17 42 CCOC(=O)c1c(-c2ccccc2)nc(-c2ccccc2)nc1N(C)C ZINC000147240515 EI For-Sale Anodyne ADORA3 18 48 CCOC(=O)c1c(-c2ccccc2)nc(-c2ccccc2)nc1N(C)C ZINC000147240515 EI For-Sale Anodyne DGAT1 24 42 C[C@H](N)C(=O)NN(C)C ZINC000147240530 AA For-Sale Reactive SLC15A2 0 44 CCNc1ncc(Br)c(Nc2ccc(C#N)cc2F)n1 ZINC000147240545 EG For-Sale Mild SYK 16 41 CCCCN(CCBr)S(=O)(=O)c1ccccc1C(F)(F)F ZINC000147240608 GH For-Sale Reactive AGTR2 47 34 NC(=O)NCCNc1nc(Cl)nc(N2CCOCC2)n1 ZINC000147240612 DB For-Sale Anodyne STAT6 51 33 COc1nc(N)nc(Oc2ccc(Cl)cc2C)n1 ZINC000147240618 CE For-Sale Anodyne AGPAT2 44 40 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147240647 FD On-Demand Anodyne MAPK11 44 45 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147240647 FD On-Demand Anodyne MAPK14 68 45 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147240647 FD On-Demand Anodyne MAPK13 45 39 C[C@H](CNS(=O)(=O)N(C)Cc1ccccc1)CC(=O)O ZINC000147240694 DD For-Sale Anodyne MME 46 36 C[C@H](CNS(=O)(=O)N(C)Cc1ccccc1)CC(=O)O ZINC000147240694 DD For-Sale Anodyne MMP3 19 45 C[C@H](CNS(=O)(=O)N(C)Cc1ccccc1)CC(=O)O ZINC000147240694 DD For-Sale Anodyne POL 0 40 C[C@H](CNS(=O)(=O)N(C)Cc1ccccc1)CC(=O)O ZINC000147240694 DD For-Sale Anodyne PTGES 22 41 C[C@H](CNS(=O)(=O)N(C)Cc1ccccc1)CC(=O)O ZINC000147240694 DD For-Sale Anodyne LIMK2 29 40 CCCCCCCCNC(=O)N1[C@@H](CC)SC[C@H]1C(=O)O ZINC000147240701 DG For-Sale Mild ASAH1 93 37 C[C@@H](N)C(=O)NN(C)C ZINC000147240744 AA For-Sale Reactive SLC15A2 0 44 CCN(CC)C(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147240778 FH On-Demand Bother EXSA 0 40 CCN(CC)C(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147240778 FH On-Demand Bother SENP1 0 41 CNc1cccc(NCCc2ccc(OC)cc2)n1 ZINC000147240790 CF For-Sale Anodyne PTGDR 33 49 COc1cc(OCC(=O)N[C@H](C)c2ccc(S(C)(=O)=O)cc2)ccc1[N+](=O)[O-] ZINC000147240809 HE In-Stock Bother COLA 59 37 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1NC(=O)c1ccco1 ZINC000147240838 EG On-Demand Mild MAPK11 29 40 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1NC(=O)c1ccco1 ZINC000147240838 EG On-Demand Mild MAPK14 16 40 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1NC(=O)c1ccco1 ZINC000147240838 EG On-Demand Mild KISS1R 46 34 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1NC(=O)c1ccco1 ZINC000147240838 EG On-Demand Mild L3MBTL3 43 32 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147240846 FD On-Demand Anodyne MAPK11 44 45 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147240846 FD On-Demand Anodyne MAPK14 68 45 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147240846 FD On-Demand Anodyne MAPK13 45 39 CN(Cc1cscn1)C(=O)N[C@@H](c1ccccc1)c1ccccn1 ZINC000147240912 EG On-Demand Anodyne CYP3A4 18 43 C[C@@H](CNS(=O)(=O)N(C)Cc1ccccc1)CC(=O)O ZINC000147240916 DD For-Sale Anodyne MME 46 36 C[C@@H](CNS(=O)(=O)N(C)Cc1ccccc1)CC(=O)O ZINC000147240916 DD For-Sale Anodyne MMP3 19 45 C[C@@H](CNS(=O)(=O)N(C)Cc1ccccc1)CC(=O)O ZINC000147240916 DD For-Sale Anodyne POL 0 40 C[C@@H](CNS(=O)(=O)N(C)Cc1ccccc1)CC(=O)O ZINC000147240916 DD For-Sale Anodyne PTGES 22 41 C[C@@H](CNS(=O)(=O)N(C)Cc1ccccc1)CC(=O)O ZINC000147240916 DD For-Sale Anodyne LIMK2 29 40 CCCCCCCCNC(=O)N1[C@@H](C(=O)O)CS[C@@H]1CC ZINC000147240927 DG For-Sale Mild ASAH1 93 37 CCC[C@H](N)C(=O)NN(C)C ZINC000147240936 AB For-Sale Reactive DPP7 0 46 CCC[C@H](N)C(=O)NN(C)C ZINC000147240936 AB For-Sale Reactive DPP8 0 46 CCC[C@H](N)C(=O)NN(C)C ZINC000147240936 AB For-Sale Reactive DPP9 0 46 CC(C)NS(=O)(=O)c1ccccc1NCCNC(N)=O ZINC000147240941 DC For-Sale Anodyne PRTN3 44 32 CC(C)NS(=O)(=O)c1ccccc1NCCNC(N)=O ZINC000147240941 DC For-Sale Anodyne ITGAV 34 40 CCc1cc(C)cc(C)c1OC ZINC000147240946 AF For-Sale Anodyne DRTS_PLABA 15 44 Nc1cnccc1NCC(F)F ZINC000147240975 AD For-Sale Anodyne AOC1 19 40 Nc1cnccc1NCC(F)F ZINC000147240975 AD For-Sale Anodyne AMO_PEA 41 34 N#Cc1c(N)[nH]c(=O)[nH]c1=O ZINC000147241015 AA For-Sale Mild DEOA 15 46 CCc1ncc(C(=O)N2CCN(c3ccc(C(F)(F)F)cc3[N+](=O)[O-])CC2)s1 ZINC000147241017 HH On-Demand Bother SERPINE1 23 41 CCc1ncc(C(=O)N2CCN(c3ccc(C(F)(F)F)cc3[N+](=O)[O-])CC2)s1 ZINC000147241017 HH On-Demand Bother SLC6A9 30 43 COC(=O)C(C)(C)[C@H](N)Cc1ccc(OC)cc1 ZINC000147241041 CD For-Sale Anodyne MMP13 19 41 COC(=O)C(C)(C)[C@H](N)Cc1ccc(OC)cc1 ZINC000147241041 CD For-Sale Anodyne PTPRB 43 43 COC(=O)C(C)(C)[C@H](N)Cc1ccc(OC)cc1 ZINC000147241041 CD For-Sale Anodyne MMP9 22 41 COC(=O)C(C)(C)[C@H](N)Cc1ccc(OC)cc1 ZINC000147241041 CD For-Sale Anodyne CA9 20 41 COC(=O)C(C)(C)[C@H](N)Cc1ccc(OC)cc1 ZINC000147241041 CD For-Sale Anodyne MMP1 32 41 COC(=O)C(C)(C)[C@H](N)Cc1ccc(OC)cc1 ZINC000147241041 CD For-Sale Anodyne CYP26A1 24 41 COC(=O)C(C)(C)[C@H](N)Cc1ccc(OC)cc1 ZINC000147241041 CD For-Sale Anodyne PROKR1 58 32 CN(Cc1cscn1)C(=O)N[C@H](c1ccccc1)c1ccccn1 ZINC000147241068 EG On-Demand Anodyne CYP3A4 18 43 CCCCCCCCNC(=O)N1[C@H](CC)SC[C@H]1C(=O)O ZINC000147241074 DG For-Sale Mild ASAH1 93 37 CCC[C@@H](N)C(=O)NN(C)C ZINC000147241076 AB For-Sale Reactive DPP7 0 46 CCC[C@@H](N)C(=O)NN(C)C ZINC000147241076 AB For-Sale Reactive DPP8 0 46 CCC[C@@H](N)C(=O)NN(C)C ZINC000147241076 AB For-Sale Reactive DPP9 0 46 CNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147241105 DC On-Demand Mild TRY2_BOVIN 40 36 CNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147241105 DC On-Demand Mild PREP 19 40 CNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147241105 DC On-Demand Mild ST14 79 36 CNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147241105 DC On-Demand Mild AKR1C3 47 38 CNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147241105 DC On-Demand Mild SFRP1 45 41 CNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147241105 DC On-Demand Mild L3MBTL3 43 42 CNS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147241105 DC On-Demand Mild TMPRSS6 63 33 NC(=O)NCCNc1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000147241184 CC For-Sale Anodyne SFRP1 93 38 NC(=O)NCCNc1ccc(S(=O)(=O)NC2CC2)cc1 ZINC000147241184 CC For-Sale Anodyne WNT3 59 33 COc1ccc([C@@H]2CCCCCN2C(=O)[C@H](C)OC[C@@H]2CCCO2)cc1 ZINC000147241199 FH On-Demand Anodyne CPT1A 56 38 CCCc1c(N)ncnc1Nc1ccc(C#N)cc1F ZINC000147241235 CF For-Sale Mild FLT1 0 44 COC(=O)C(C)(C)[C@@H](N)Cc1ccc(OC)cc1 ZINC000147241249 CD For-Sale Anodyne MMP13 19 41 COC(=O)C(C)(C)[C@@H](N)Cc1ccc(OC)cc1 ZINC000147241249 CD For-Sale Anodyne PTPRB 43 43 COC(=O)C(C)(C)[C@@H](N)Cc1ccc(OC)cc1 ZINC000147241249 CD For-Sale Anodyne MMP9 22 41 COC(=O)C(C)(C)[C@@H](N)Cc1ccc(OC)cc1 ZINC000147241249 CD For-Sale Anodyne CA9 20 41 COC(=O)C(C)(C)[C@@H](N)Cc1ccc(OC)cc1 ZINC000147241249 CD For-Sale Anodyne MMP1 32 41 COC(=O)C(C)(C)[C@@H](N)Cc1ccc(OC)cc1 ZINC000147241249 CD For-Sale Anodyne CYP26A1 24 41 COC(=O)C(C)(C)[C@@H](N)Cc1ccc(OC)cc1 ZINC000147241249 CD For-Sale Anodyne PROKR1 58 32 Cc1cccnc1-c1ccc(Cl)cc1Cl ZINC000147241251 BI For-Sale Anodyne CNR1 25 41 Cc1cccnc1-c1ccc(Cl)cc1Cl ZINC000147241251 BI For-Sale Anodyne CRHR1 30 43 Cc1cccnc1-c1ccc(Cl)cc1Cl ZINC000147241251 BI For-Sale Anodyne DPP4 24 45 CCn1cc(NC(=O)NNC(=O)c2ccc(OC(C)C)c(OC)c2)ccc1=O ZINC000147241252 GE On-Demand Reactive CPT1A 47 33 CCn1cc(NC(=O)NNC(=O)c2ccc(OC(C)C)c(OC)c2)ccc1=O ZINC000147241252 GE On-Demand Reactive ENPP1 69 37 CC(C)C[C@H](N)C(=O)NN(C)C ZINC000147241261 AB For-Sale Reactive RNPEP 41 32 CC(C)C[C@H](N)C(=O)NN(C)C ZINC000147241261 AB For-Sale Reactive DNPEP 0 42 CC(C)C[C@H](N)C(=O)NN(C)C ZINC000147241261 AB For-Sale Reactive LAP3 31 42 CC(C)C[C@H](N)C(=O)NN(C)C ZINC000147241261 AB For-Sale Reactive AMPX_VIBPR 0 61 NC(=O)c1ccc(OCC(=O)N2CCNC(=O)C[C@H]2c2ccccc2)cc1 ZINC000147241273 FD On-Demand Anodyne CPT1A 129 51 NC(=O)c1ccc(OCC(=O)N2CCNC(=O)C[C@H]2c2ccccc2)cc1 ZINC000147241273 FD On-Demand Anodyne CPT2 45 39 CCCCCCCCNC(=O)N1[C@H](CC)SC[C@@H]1C(=O)O ZINC000147241281 DG For-Sale Mild ASAH1 93 37 CCNc1ncnc(Oc2ccc(Cl)cc2C)c1[N+](=O)[O-] ZINC000147241308 DH For-Sale Bother S1PR4 21 40 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147241337 HG On-Demand Mild F2 17 41 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147241337 HG On-Demand Mild PLG 22 41 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147241337 HG On-Demand Mild MMP13 43 42 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147241337 HG On-Demand Mild TRY2_BOVIN 54 34 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147241337 HG On-Demand Mild ADAM17 43 41 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147241337 HG On-Demand Mild ST14 77 41 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147241337 HG On-Demand Mild MMP1 19 41 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147241337 HG On-Demand Mild GPR119 19 40 CCOc1ccc(S(=O)(=O)Nc2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147241337 HG On-Demand Mild LIMK2 30 41 COc1ccc([C@@H]2CCCCCN2C(=O)[C@@H](C)OC[C@@H]2CCCO2)cc1 ZINC000147241380 FH On-Demand Anodyne CPT1A 56 38 N[C@@H]1CC[C@H](c2cccc(F)c2F)CN(CC(F)(F)F)C1=O ZINC000147241427 DF For-Sale Anodyne CALCRL 33 52 NC(=O)c1ccc(OCC(=O)N2CCNC(=O)C[C@@H]2c2ccccc2)cc1 ZINC000147241467 FD On-Demand Anodyne CPT1A 129 51 NC(=O)c1ccc(OCC(=O)N2CCNC(=O)C[C@@H]2c2ccccc2)cc1 ZINC000147241467 FD On-Demand Anodyne CPT2 45 39 CC(C)C[C@@H](N)C(=O)NN(C)C ZINC000147241495 AB For-Sale Reactive RNPEP 41 32 CC(C)C[C@@H](N)C(=O)NN(C)C ZINC000147241495 AB For-Sale Reactive DNPEP 0 42 CC(C)C[C@@H](N)C(=O)NN(C)C ZINC000147241495 AB For-Sale Reactive LAP3 31 42 CC(C)C[C@@H](N)C(=O)NN(C)C ZINC000147241495 AB For-Sale Reactive AMPX_VIBPR 0 61 COc1ccc(C)cc1-n1ccc(C(=O)NC2CCC(C(F)(F)F)CC2)n1 ZINC000147241613 GI On-Demand Anodyne MAPK13 67 34 N#Cc1ccccc1OCC(=O)N1CCC(C#N)CC1 ZINC000147241640 CD On-Demand Mild ADRB1 42 32 N#Cc1ccccc1OCC(=O)N1CCC(C#N)CC1 ZINC000147241640 CD On-Demand Mild COLA 0 41 N#Cc1ccccc1OCC(=O)N1CCC(C#N)CC1 ZINC000147241640 CD On-Demand Mild FAP 0 41 CCCOc1cc(NCC(F)F)ccc1N ZINC000147241645 BF For-Sale Anodyne DRTS_TRYCR 46 33 COc1cc(NCCNC(N)=O)c([N+](=O)[O-])cc1OC ZINC000147241697 CC On-Demand Bother SCMU_MYCTU 0 41 CC(C)NC(=O)[C@@H](C)Oc1ccc(F)cc1S(N)(=O)=O ZINC000147241748 DC For-Sale Anodyne SDH1 0 45 CN(C)NC(=O)[C@H](N)c1ccccc1 ZINC000147241749 AC For-Sale Reactive CACNA2D1 23 53 CN(C)NC(=O)[C@H](N)c1ccccc1 ZINC000147241749 AC For-Sale Reactive SLC15A1 56 35 CN(C)NC(=O)[C@H](N)c1ccccc1 ZINC000147241749 AC For-Sale Reactive KYNU 41 29 C[C@@H](CNC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147241756 CG On-Demand Anodyne BMP1 50 35 CC(C)NC(=O)[C@H](C)Oc1ccc(F)cc1S(N)(=O)=O ZINC000147241943 DC For-Sale Anodyne SDH1 0 45 CN(C)NC(=O)[C@@H](N)c1ccccc1 ZINC000147241950 AC For-Sale Reactive CACNA2D1 23 53 CN(C)NC(=O)[C@@H](N)c1ccccc1 ZINC000147241950 AC For-Sale Reactive SLC15A1 56 35 CN(C)NC(=O)[C@@H](N)c1ccccc1 ZINC000147241950 AC For-Sale Reactive KYNU 41 29 O=C(O)C1(NCc2ccc3c(c2)OCO3)CCC1 ZINC000147241997 BD For-Sale Anodyne NOS2 94 37 COC(=O)c1cncc(N[C@@H]2c3ccccc3C[C@H]2O)n1 ZINC000147242070 CD On-Demand Anodyne PLM2_PLAFA 40 35 NS(=O)(=O)c1cc(F)ccc1OCCN1CCOCC1 ZINC000147242150 DC For-Sale Anodyne HTR2A 27 44 NS(=O)(=O)c1cc(F)ccc1OCCN1CCOCC1 ZINC000147242150 DC For-Sale Anodyne MAPK14 0 48 NS(=O)(=O)c1cc(F)ccc1OCCN1CCOCC1 ZINC000147242150 DC For-Sale Anodyne EPHX2 16 45 CN(C)NC(=O)CCCCCCN ZINC000147242203 AC For-Sale Reactive PAOX 18 41 CN(C)NC(=O)CCCCCCN ZINC000147242203 AC For-Sale Reactive APHA 0 44 CN(C)NC(=O)CCCCCCN ZINC000147242203 AC For-Sale Reactive KDM7A 0 52 COC(=O)c1cncc(N[C@H]2c3ccccc3C[C@H]2O)n1 ZINC000147242252 CD On-Demand Anodyne PLM2_PLAFA 40 35 NS(=O)(=O)c1cc(F)ccc1OCCCN1CCCC1 ZINC000147242374 DD For-Sale Anodyne DRD2 20 43 NS(=O)(=O)c1cc(F)ccc1OCCCN1CCCC1 ZINC000147242374 DD For-Sale Anodyne HTR2A 30 40 NS(=O)(=O)c1cc(F)ccc1OCCCN1CCCC1 ZINC000147242374 DD For-Sale Anodyne HTR2C 15 40 NS(=O)(=O)c1cc(F)ccc1OCCCN1CCCC1 ZINC000147242374 DD For-Sale Anodyne KCNH2 0 41 NS(=O)(=O)c1cc(F)ccc1OCCCN1CCCC1 ZINC000147242374 DD For-Sale Anodyne LTA4H 23 41 NS(=O)(=O)c1cc(F)ccc1OCCCN1CCCC1 ZINC000147242374 DD For-Sale Anodyne HRH3 66 53 CCCCCCCCNC(=O)NC[C@@H]1CCC[C@@H]1C(=O)O ZINC000147242377 CG For-Sale Mild EPHX2 25 50 CN(C)NC(=O)CNC1CCCC1 ZINC000147242424 AC For-Sale Reactive DPP7 15 40 O=C(O)C1(NCCOc2cccc(Cl)c2)CCC1 ZINC000147242447 CE For-Sale Anodyne DRD4 16 54 O=C(O)C1(NCCOc2cccc(Cl)c2)CCC1 ZINC000147242447 CE For-Sale Anodyne HRH2 26 44 CCc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147242483 CD On-Demand Anodyne CA2 17 40 CCc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147242483 CD On-Demand Anodyne TBXA2R 42 35 CCc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147242483 CD On-Demand Anodyne ADAMTS4 44 37 CCc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147242483 CD On-Demand Anodyne LIMK2 37 45 BrC1C[C@H]2CC[C@H](C1)N2C[C@@H]1OCCc2ccccc21 ZINC000147242491 EH For-Sale Reactive ACHP_LYMST 21 40 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147242512 HD On-Demand Anodyne F13A1 40 36 CCCNS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147242583 DC For-Sale Anodyne CA2 35 44 CCCNS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147242583 DC For-Sale Anodyne CA1 33 44 CCCNS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147242583 DC For-Sale Anodyne CA4 28 44 CCCNS(=O)(=O)c1ccc(NCCNC(N)=O)cc1 ZINC000147242583 DC For-Sale Anodyne CYNT 46 36 CCCCCCCCNC(=O)NC[C@H]1CCC[C@@H]1C(=O)O ZINC000147242593 CG For-Sale Mild EPHX2 25 50 CN(C)NC(=O)CNC1CC1 ZINC000147242626 AB For-Sale Reactive KDM7A 0 42 CCCc1c(NCC)ncnc1Oc1ccc(Cl)cc1C ZINC000147242644 DJ For-Sale Anodyne PDE6A 41 32 CCCC[C@H](NC(N)=O)C(=O)NC1CCC(C(F)(F)F)CC1 ZINC000147242678 DE On-Demand Anodyne HDAC4 15 40 BrC1C[C@@H]2CC[C@H](C1)N2C[C@H]1OCCc2ccccc21 ZINC000147242685 EH For-Sale Reactive ACHP_LYMST 21 40 CCc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147242700 CD On-Demand Anodyne CA2 17 40 CCc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147242700 CD On-Demand Anodyne TBXA2R 42 35 CCc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147242700 CD On-Demand Anodyne ADAMTS4 44 37 CCc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147242700 CD On-Demand Anodyne LIMK2 37 45 C[C@@H](OC[C@@H]1CCCO1)C(=O)N1CCCN(S(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147242707 HD On-Demand Anodyne F13A1 40 36 CCOC[C@H](C)NC(=O)Nc1cc(C(=O)NC2CC2)ccc1C ZINC000147242757 DE On-Demand Anodyne MAPK11 45 45 CCOC[C@H](C)NC(=O)Nc1cc(C(=O)NC2CC2)ccc1C ZINC000147242757 DE On-Demand Anodyne MAPK14 68 45 CCOC[C@H](C)NC(=O)Nc1cc(C(=O)NC2CC2)ccc1C ZINC000147242757 DE On-Demand Anodyne MAPK13 44 37 CCCCCCCCNC(=O)NC[C@@H]1CCC[C@H]1C(=O)O ZINC000147242781 CG For-Sale Mild EPHX2 25 50 O=C(O)CCN(C(=O)c1cccc(F)c1Cl)C1CC1 ZINC000147242816 CF On-Demand Anodyne ACE 45 40 O=C(O)CCN(C(=O)c1cccc(F)c1Cl)C1CC1 ZINC000147242816 CF On-Demand Anodyne C5AR1 27 46 CCCC[C@@H](NC(N)=O)C(=O)NC1CCC(C(F)(F)F)CC1 ZINC000147242858 DE On-Demand Anodyne HDAC4 15 40 CCOC(=O)c1cnc(-c2ccc(Br)cc2)nc1N(CC)CC ZINC000147242870 GH For-Sale Anodyne JUN 18 44 CCN1CCC(NC(=O)c2cccc3c2OCCN3)CC1 ZINC000147242872 CD For-Sale Anodyne DRD4 21 44 CCN1CCC(NC(=O)c2cccc3c2OCCN3)CC1 ZINC000147242872 CD For-Sale Anodyne HTR4 31 44 CCN1CCC(NC(=O)c2cccc3c2OCCN3)CC1 ZINC000147242872 CD For-Sale Anodyne SIGMAR1 17 42 BrC1C[C@@H]2CC[C@H](C1)N2C[C@@H]1OCCc2ccccc21 ZINC000147242873 EH For-Sale Reactive ACHP_LYMST 21 40 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@@H](O)COc1c(C)cccc1C ZINC000147242980 HG On-Demand Anodyne ADRB1 40 34 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@@H](O)COc1c(C)cccc1C ZINC000147242980 HG On-Demand Anodyne MAPK11 43 44 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@@H](O)COc1c(C)cccc1C ZINC000147242980 HG On-Demand Anodyne MAPK14 71 44 CCCCCCCCNC(=O)NC[C@H]1CCC[C@H]1C(=O)O ZINC000147242995 CG For-Sale Mild EPHX2 25 50 N#CC1CCN(C(=O)CCN2c3ccccc3Sc3ccccc32)CC1 ZINC000147243005 FI On-Demand Mild BCHE 21 44 O=C(O)CCN(C(=O)[C@H]1C[C@H]1c1ccccc1)C1CC1 ZINC000147243039 CE For-Sale Anodyne FFAR1 0 41 O=C(O)CCN(C(=O)[C@H]1C[C@H]1c1ccccc1)C1CC1 ZINC000147243039 CE For-Sale Anodyne GPR88 0 47 O=C(O)[C@@H]1CN(Cc2ccccc2)C[C@]12CCCc1ccccc12 ZINC000147243065 DG For-Sale Anodyne SIGMAR1 54 51 Cc1nn(C(F)F)c(C)c1CC(=O)NC1CCC(C(F)(F)F)CC1 ZINC000147243075 FH On-Demand Anodyne P2RX7 15 45 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)NCC(C)C)c(Cl)c1)C2 ZINC000147243083 HH On-Demand Anodyne ROCK2 27 46 CNc1cn2ccnc2c(Oc2ccc(Cl)cc2C)n1 ZINC000147243094 CH For-Sale Anodyne HIVRT 0 58 CCc1nc(CN(C)C(=O)NC[C@@H](c2cccc(OC)c2)N2CCCC2)cs1 ZINC000147243097 HH On-Demand Anodyne DRD4 40 30 CCc1nc(CN(C)C(=O)NC[C@@H](c2cccc(OC)c2)N2CCCC2)cs1 ZINC000147243097 HH On-Demand Anodyne KCNQ2 15 41 O=C(Nc1cccc(F)c1F)c1cc([N+](=O)[O-])n[nH]1 ZINC000147243138 CD On-Demand Bother PLA2G7 15 44 O=C(Nc1cccc(F)c1F)c1cc([N+](=O)[O-])n[nH]1 ZINC000147243138 CD On-Demand Bother ALPL 44 35 O=C(O)C1(NCc2nc(-c3cccs3)no2)CCC1 ZINC000147243151 CD For-Sale Anodyne ETHR 31 42 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@H](O)COc1c(C)cccc1C ZINC000147243170 HG On-Demand Anodyne ADRB1 40 34 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@H](O)COc1c(C)cccc1C ZINC000147243170 HG On-Demand Anodyne MAPK11 43 44 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@H](O)COc1c(C)cccc1C ZINC000147243170 HG On-Demand Anodyne MAPK14 71 44 CC(C)[C@H](NC(=O)c1ccc(F)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147243224 EE On-Demand Mild ELANE 52 52 CC(C)[C@H](NC(=O)c1ccc(F)cc1)C(=O)N1CCC(C#N)CC1 ZINC000147243224 EE On-Demand Mild CCR1 51 52 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(OCC(=O)N2CCCC2)c1 ZINC000147243234 GD On-Demand Anodyne CPT1A 118 45 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(OCC(=O)N2CCCC2)c1 ZINC000147243234 GD On-Demand Anodyne CPT2 47 36 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(OCC(=O)N2CCCC2)c1 ZINC000147243234 GD On-Demand Anodyne EPHX2 21 43 O=C(O)CCN(C(=O)[C@H]1C[C@@H]1c1ccccc1)C1CC1 ZINC000147243250 CE For-Sale Anodyne FFAR1 0 41 O=C(O)CCN(C(=O)[C@H]1C[C@@H]1c1ccccc1)C1CC1 ZINC000147243250 CE For-Sale Anodyne GPR88 0 47 COCCNC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147243283 DB For-Sale Anodyne CA2 24 42 COCCNC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147243283 DB For-Sale Anodyne CA1 16 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1CN1CCOCC1)C2 ZINC000147243284 GF On-Demand Anodyne CCR3 20 45 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1CN1CCOCC1)C2 ZINC000147243284 GF On-Demand Anodyne ROCK2 35 44 CCOC(=O)c1cnc(-c2cccnc2)nc1N(CC)CC ZINC000147243299 DF For-Sale Anodyne JUN 17 42 CCOC(=O)c1cnc(-c2cccnc2)nc1N(CC)CC ZINC000147243299 DF For-Sale Anodyne KLK7 25 40 CCc1nc(CN(C)C(=O)NC[C@H](c2cccc(OC)c2)N2CCCC2)cs1 ZINC000147243317 HH On-Demand Anodyne DRD4 40 30 CCc1nc(CN(C)C(=O)NC[C@H](c2cccc(OC)c2)N2CCCC2)cs1 ZINC000147243317 HH On-Demand Anodyne KCNQ2 15 41 CN(C)C(=O)c1ccc(NCCNC(N)=O)c([N+](=O)[O-])c1 ZINC000147243327 CC For-Sale Bother DRTS_TOXGO 17 48 O=C(O)CCN(C(=O)[C@@H]1C[C@H]1c1ccccc1)C1CC1 ZINC000147243422 CE For-Sale Anodyne FFAR1 0 41 O=C(O)CCN(C(=O)[C@@H]1C[C@H]1c1ccccc1)C1CC1 ZINC000147243422 CE For-Sale Anodyne GPR88 0 47 CCc1c(N)ncnc1Nc1ccc(C#N)cc1F ZINC000147243426 CE For-Sale Mild FLT1 0 43 CNC(=O)Oc1ccc(S)cc1 ZINC000147243433 AD For-Sale Anodyne AO-ACHE 0 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(OCC(=O)N2CCCC2)c1 ZINC000147243449 GD On-Demand Anodyne CPT1A 118 45 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(OCC(=O)N2CCCC2)c1 ZINC000147243449 GD On-Demand Anodyne CPT2 47 36 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(OCC(=O)N2CCCC2)c1 ZINC000147243449 GD On-Demand Anodyne EPHX2 21 43 CC[C@@H](C)NC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147243516 DC For-Sale Anodyne SDH1 0 41 COc1ccc2c(c1)OC[C@H](C(=O)NCc1cc(F)ccc1Br)C2 ZINC000147243535 GG On-Demand Anodyne MTNR1A 23 40 COc1ccc2c(c1)OC[C@H](C(=O)NCc1cc(F)ccc1Br)C2 ZINC000147243535 GG On-Demand Anodyne ROCK2 23 42 CCCNc1cc(Oc2ccc(Cl)cc2C)nc(N)n1 ZINC000147243548 CH For-Sale Anodyne AGPAT2 75 45 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne PPIA 46 45 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne PTGER1 52 41 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne BMP1 46 35 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne CTSB 42 39 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne PAPA1_CARPA 43 34 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne CYSP_TRYCR 52 36 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne GRM4 41 37 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne CAPNS1 54 33 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne CAPN1 60 38 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne CAPN2 97 39 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne TYK2 64 35 O=C(Nc1ccnc(Cl)c1)OCc1ccccc1 ZINC000147243576 CG For-Sale Anodyne NPR 59 35 O=C(O)C1(NCc2cc(-c3ccccc3)on2)CCC1 ZINC000147243585 CE For-Sale Anodyne NPPA 45 35 CCOC(=O)CCC(=O)C1CCC(COCc2ccccc2)CC1 ZINC000147243594 EH For-Sale Anodyne VCP 45 34 O=C(O)c1cccnc1C(=O)NCC(F)F ZINC000147243595 BC For-Sale Anodyne OSIGBA0132E09-OSIGBA0108L24.11 0 48 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(OC)c(OC)c2)CC1 ZINC000147243596 HD On-Demand Anodyne F2 23 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(OC)c(OC)c2)CC1 ZINC000147243596 HD On-Demand Anodyne P2RY12 200 43 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(OC)c(OC)c2)CC1 ZINC000147243596 HD On-Demand Anodyne PTAFR 15 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(OC)c(OC)c2)CC1 ZINC000147243596 HD On-Demand Anodyne TRY2_BOVIN 64 37 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(OC)c(OC)c2)CC1 ZINC000147243596 HD On-Demand Anodyne HPGD 16 40 O=C(O)CCN(C(=O)[C@@H]1C[C@@H]1c1ccccc1)C1CC1 ZINC000147243638 CE For-Sale Anodyne FFAR1 0 41 O=C(O)CCN(C(=O)[C@@H]1C[C@@H]1c1ccccc1)C1CC1 ZINC000147243638 CE For-Sale Anodyne GPR88 0 47 CCNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147243642 CG For-Sale Mild INSR 39 42 CCNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147243642 CG For-Sale Mild MAPK9 38 43 CCNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147243642 CG For-Sale Mild MAPK10 39 43 CCNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147243642 CG For-Sale Mild ALK 41 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(OCc2ccc(F)cc2)c1 ZINC000147243657 GG On-Demand Anodyne CCR3 45 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(OCc2ccc(F)cc2)c1 ZINC000147243657 GG On-Demand Anodyne EPHX2 17 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cc(F)ccc1Br)C2 ZINC000147243663 GG On-Demand Anodyne MTNR1A 23 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cc(F)ccc1Br)C2 ZINC000147243663 GG On-Demand Anodyne ROCK2 23 42 CN(C)NC(=O)COCCN ZINC000147243676 AA For-Sale Reactive KDM7A 0 45 CC[C@H](C)NC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147243709 DC For-Sale Anodyne SDH1 0 41 CCCCN(CCBr)S(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000147243718 GH For-Sale Reactive CACNA1B 51 39 CCCCN(CCBr)S(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000147243718 GH For-Sale Reactive COLA 15 41 CCCCN(CCBr)S(=O)(=O)c1cccc(C(F)(F)F)c1 ZINC000147243718 GH For-Sale Reactive GALR3 44 31 O=C(Nc1cccc(F)c1F)c1cccc2c1OCCN2 ZINC000147243735 CG For-Sale Anodyne G2YM83_BOTF4 51 32 N#CC1CCN(C(=O)Cc2ccc([N+](=O)[O-])cc2)CC1 ZINC000147243757 CD On-Demand Mild KCNJ1 35 46 CCOC(=O)c1c(N)csc1C ZINC000147243763 AD For-Sale Anodyne PRKCZ 40 49 CCOC(=O)c1c(N)csc1C ZINC000147243763 AD For-Sale Anodyne PRKCI 0 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(OC)c(OC)c2)CC1 ZINC000147243781 HD On-Demand Anodyne F2 23 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(OC)c(OC)c2)CC1 ZINC000147243781 HD On-Demand Anodyne P2RY12 200 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(OC)c(OC)c2)CC1 ZINC000147243781 HD On-Demand Anodyne PTAFR 15 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(OC)c(OC)c2)CC1 ZINC000147243781 HD On-Demand Anodyne TRY2_BOVIN 64 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(OC)c(OC)c2)CC1 ZINC000147243781 HD On-Demand Anodyne HPGD 16 40 CCCCCCCCNC(=O)N1[C@H]2CC[C@H]1[C@H](C(=O)O)C2 ZINC000147243808 CF For-Sale Mild ASAH1 94 40 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NCc1ccc(-n2ccnc2)c(F)c1 ZINC000147243825 HH On-Demand Anodyne MAPK11 42 42 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NCc1ccc(-n2ccnc2)c(F)c1 ZINC000147243825 HH On-Demand Anodyne MAPK14 66 44 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NCc1ccc(-n2ccnc2)c(F)c1 ZINC000147243825 HH On-Demand Anodyne NOS2 79 33 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NCc1ccc(-n2ccnc2)c(F)c1 ZINC000147243825 HH On-Demand Anodyne MAPK13 96 38 O=C(O)c1ccccc1C(=O)NCC(F)F ZINC000147243840 BD For-Sale Anodyne PADI4 0 43 O=C(O)c1ccccc1C(=O)NCC(F)F ZINC000147243840 BD For-Sale Anodyne PADI1 0 43 O=C(O)c1ccccc1C(=O)NCC(F)F ZINC000147243840 BD For-Sale Anodyne PADI2 0 41 O=C(O)c1ccccc1C(=O)NCC(F)F ZINC000147243840 BD For-Sale Anodyne PADI3 0 41 CC(C)OCC(=O)N1CCNC(=O)C[C@@H]1c1ccccc1 ZINC000147243842 CD On-Demand Anodyne CPT1A 81 34 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(OCc2ccc(F)cc2)c1 ZINC000147243873 GG On-Demand Anodyne CCR3 45 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(OCc2ccc(F)cc2)c1 ZINC000147243873 GG On-Demand Anodyne EPHX2 17 42 COCCCNC(=O)COc1ccc(F)cc1S(N)(=O)=O ZINC000147243915 DC For-Sale Anodyne CA2 20 45 CCCCCCCCCCCCCCCCOC[C@@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147243978 IG Annotated Mild VEGFA 28 53 CCCCCCCCCCCCCCCCOC[C@@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147243978 IG Annotated Mild FGF1 0 53 CCCCCCCCCCCCCCCCOC[C@@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147243978 IG Annotated Mild SELP 49 45 CCCCCCCCCCCCCCCCOC[C@@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147243978 IG Annotated Mild FGF2 0 53 CCCCCCCCCCCCCCCCOC[C@@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147243978 IG Annotated Mild GBA2 50 37 CCCCCCCCCCCCCCCCOC[C@@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147243978 IG Annotated Mild SELL 0 45 CCCCCCCCCCCCCCCCOC[C@@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147243978 IG Annotated Mild ENV 17 52 CCCCCCCCCCCCCCCCOC[C@@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147243978 IG Annotated Mild FIMH 68 68 CCCCCCCCCCCCCCCCOC[C@@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147243978 IG Annotated Mild LGALS8 0 43 CCCCCCCCCCCCCCCCOC[C@@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147243978 IG Annotated Mild LGALS4 0 43 CC(C)OCC(=O)N1CCNC(=O)C[C@H]1c1ccccc1 ZINC000147243994 CD On-Demand Anodyne CPT1A 81 34 CCCCCCCCNC(=O)N(C)CCCC(=O)O ZINC000147244033 CF For-Sale Mild FABP2 0 50 CCCCCCCCNC(=O)N(C)CCCC(=O)O ZINC000147244033 CF For-Sale Mild FABP4 18 50 CCCCCCCCNC(=O)N(C)CCCC(=O)O ZINC000147244033 CF For-Sale Mild CPT1A 39 41 CCCCCCCCNC(=O)N(C)CCCC(=O)O ZINC000147244033 CF For-Sale Mild DNM1 0 48 CCCCCCCCNC(=O)N(C)CCCC(=O)O ZINC000147244033 CF For-Sale Mild EPHX2 33 77 CCCCCCCCNC(=O)N(C)CCCC(=O)O ZINC000147244033 CF For-Sale Mild FABP3 33 42 CCCCCCCCNC(=O)N(C)CCCC(=O)O ZINC000147244033 CF For-Sale Mild FABP5 17 50 CCCCCCCCNC(=O)N(C)CCCC(=O)O ZINC000147244033 CF For-Sale Mild ASAH1 82 34 CCCCCCCCNC(=O)N(C)CCCC(=O)O ZINC000147244033 CF For-Sale Mild SLC22A20 0 50 CCCCCCCCNC(=O)N(C)CCCC(=O)O ZINC000147244033 CF For-Sale Mild KDM4A 0 42 CCCCCCCCNC(=O)N(C)CCCC(=O)O ZINC000147244033 CF For-Sale Mild CQSS 49 30 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@@H]1CCCO[C@@H]1c1ccccc1 ZINC000147244132 HI On-Demand Anodyne MAPK11 40 43 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@@H]1CCCO[C@@H]1c1ccccc1 ZINC000147244132 HI On-Demand Anodyne MAPK14 61 44 CCCc1c(C(=O)O)c2cc(O)ccc2n1C ZINC000147244162 BF In-Stock Anodyne F2RL3 46 33 CCCc1c(C(=O)O)c2cc(O)ccc2n1C ZINC000147244162 BF In-Stock Anodyne OXER1 30 45 CCNc1cccc(NCc2ccccc2Cl)n1 ZINC000147244179 CH For-Sale Anodyne P2RX7 18 41 CCCCCCCCCCCCCCCCOC[C@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147244200 IG Annotated Mild VEGFA 28 53 CCCCCCCCCCCCCCCCOC[C@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147244200 IG Annotated Mild FGF1 0 53 CCCCCCCCCCCCCCCCOC[C@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147244200 IG Annotated Mild SELP 49 45 CCCCCCCCCCCCCCCCOC[C@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147244200 IG Annotated Mild FGF2 0 53 CCCCCCCCCCCCCCCCOC[C@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147244200 IG Annotated Mild GBA2 50 37 CCCCCCCCCCCCCCCCOC[C@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147244200 IG Annotated Mild SELL 0 45 CCCCCCCCCCCCCCCCOC[C@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147244200 IG Annotated Mild ENV 17 52 CCCCCCCCCCCCCCCCOC[C@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147244200 IG Annotated Mild FIMH 68 68 CCCCCCCCCCCCCCCCOC[C@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147244200 IG Annotated Mild LGALS8 0 43 CCCCCCCCCCCCCCCCOC[C@H](O)CO[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147244200 IG Annotated Mild LGALS4 0 43 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild CNR1 0 40 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild PTPN2 16 42 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild GRIA1 46 34 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild SOAT1 52 42 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild FAAH 15 43 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild PTPRA 51 42 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild PTPN1 17 50 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild EPHX2 37 43 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild HCAR2 44 41 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild AKR1C3 18 40 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild ASAH1 100 43 CCCCCCCCNC(=O)Nc1ccccc1C(=O)O ZINC000147244255 CH For-Sale Mild AKR1C2 41 41 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147244286 FE On-Demand Anodyne MMP13 51 45 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147244286 FE On-Demand Anodyne MMP2 41 45 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147244286 FE On-Demand Anodyne MMP3 29 45 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147244286 FE On-Demand Anodyne MMP14 28 45 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147244286 FE On-Demand Anodyne PRTN3 45 32 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147244286 FE On-Demand Anodyne MMP9 35 45 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147244286 FE On-Demand Anodyne EPHX2 15 40 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147244286 FE On-Demand Anodyne ADAMTS4 45 34 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147244286 FE On-Demand Anodyne IDO1 15 44 C[C@H]1C[C@H](C)CN(c2ccc(C(=O)N3CCC(C#N)CC3)cc2[N+](=O)[O-])C1 ZINC000147244296 FG On-Demand Mild L3MBTL1 0 44 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@H]1CCCO[C@@H]1c1ccccc1 ZINC000147244359 HI On-Demand Anodyne MAPK11 40 43 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@H]1CCCO[C@@H]1c1ccccc1 ZINC000147244359 HI On-Demand Anodyne MAPK14 61 44 O=C(O)CCC(=O)NCC(F)F ZINC000147244474 AC On-Demand Anodyne KDM4E 27 46 O=C(O)CCC(=O)NCC(F)F ZINC000147244474 AC On-Demand Anodyne KDM2A 44 46 O=C(O)CCC(=O)NCC(F)F ZINC000147244474 AC On-Demand Anodyne PHF8 0 46 O=C(O)CCC(=O)NCC(F)F ZINC000147244474 AC On-Demand Anodyne KDM5C 0 46 O=C(O)CCC(=O)NCC(F)F ZINC000147244474 AC On-Demand Anodyne KDM7A 0 40 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild PPIA 19 41 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild FOLH1 25 40 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild CCKAR 34 48 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild LTB4R 16 40 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild CCR3 42 47 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild CPT1A 0 43 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild PLA2G4B 73 44 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild SOAT1 36 42 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild FAAH 20 44 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild CCKBR 36 42 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild EPHX2 48 63 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild AKR1C3 39 49 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild ASAH1 91 38 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild IMDH_CRYPV 45 32 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild KCNK3 96 37 CCCCCCCCNC(=O)Nc1cccc(C(=O)O)c1 ZINC000147244485 CH For-Sale Mild KCNK9 60 37 C[C@@H]1C[C@@H](C)CN(c2ccc(C(=O)N3CCC(C#N)CC3)cc2[N+](=O)[O-])C1 ZINC000147244504 FG On-Demand Mild L3MBTL1 0 44 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244511 FE On-Demand Anodyne MMP13 51 45 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244511 FE On-Demand Anodyne MMP2 41 45 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244511 FE On-Demand Anodyne MMP3 29 45 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244511 FE On-Demand Anodyne MMP14 28 45 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244511 FE On-Demand Anodyne PRTN3 45 32 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244511 FE On-Demand Anodyne MMP9 35 45 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244511 FE On-Demand Anodyne EPHX2 15 40 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244511 FE On-Demand Anodyne ADAMTS4 45 34 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244511 FE On-Demand Anodyne IDO1 15 44 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@@H]1CCCO[C@H]1c1ccccc1 ZINC000147244545 HI On-Demand Anodyne MAPK11 40 43 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@@H]1CCCO[C@H]1c1ccccc1 ZINC000147244545 HI On-Demand Anodyne MAPK14 61 44 CCCCN(CCBr)S(=O)(=O)c1ccc(CCC)cc1 ZINC000147244581 FH For-Sale Reactive BMP1 16 42 CC[C@H]1CN(C(=O)c2ccc3c(c2)OCO3)CC[C@H]1N ZINC000147244610 CD On-Demand Anodyne SSTR3 58 30 CC[C@H]1CN(C(=O)c2ccc3c(c2)OCO3)CC[C@H]1N ZINC000147244610 CD On-Demand Anodyne L3MBTL3 61 35 C[C@H](CNS(=O)(=O)c1cc(C#N)ccc1Cl)CC(=O)O ZINC000147244634 DD On-Demand Mild TBXA2R 0 44 CC(C)[C@H](CCN)CCC(=O)NN(C)C ZINC000147244661 BC For-Sale Reactive KDM7A 0 45 O=C(O)[C@H]1CCCN1C(=O)c1cccc2c1OCCN2 ZINC000147244703 CD For-Sale Anodyne ACE 43 39 O=C(O)[C@H]1CCCN1C(=O)c1cccc2c1OCCN2 ZINC000147244703 CD For-Sale Anodyne PREP 62 39 CCCCCCCCNC(=O)N1CSC[C@@H]1C(=O)O ZINC000147244706 CF For-Sale Mild ASAH1 108 42 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@H]1CCCO[C@H]1c1ccccc1 ZINC000147244713 HI On-Demand Anodyne MAPK11 40 43 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)NC[C@H]1CCCO[C@H]1c1ccccc1 ZINC000147244713 HI On-Demand Anodyne MAPK14 61 44 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244719 FE On-Demand Anodyne MMP13 51 45 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244719 FE On-Demand Anodyne MMP2 41 45 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244719 FE On-Demand Anodyne MMP3 29 45 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244719 FE On-Demand Anodyne MMP14 28 45 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244719 FE On-Demand Anodyne PRTN3 45 32 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244719 FE On-Demand Anodyne MMP9 35 45 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244719 FE On-Demand Anodyne EPHX2 15 40 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244719 FE On-Demand Anodyne ADAMTS4 45 34 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147244719 FE On-Demand Anodyne IDO1 15 44 CCN(c1ccccc1)S(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147244757 GG On-Demand Mild NPY2R 18 42 CCN(c1ccccc1)S(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147244757 GG On-Demand Mild L3MBTL3 67 37 C[C@@H](CNS(=O)(=O)c1cc(C#N)ccc1Cl)CC(=O)O ZINC000147244853 DD On-Demand Mild TBXA2R 0 44 NS(=O)(=O)c1cc(F)ccc1OCCn1ccnc1 ZINC000147244857 CC For-Sale Anodyne CYP19A1 15 44 NS(=O)(=O)c1cc(F)ccc1OCCn1ccnc1 ZINC000147244857 CC For-Sale Anodyne CYP11B1 30 40 NS(=O)(=O)c1cc(F)ccc1OCCn1ccnc1 ZINC000147244857 CC For-Sale Anodyne TBXAS1 39 46 NS(=O)(=O)c1cc(F)ccc1OCCn1ccnc1 ZINC000147244857 CC For-Sale Anodyne CYP11B2 24 40 NS(=O)(=O)c1cc(F)ccc1OCCn1ccnc1 ZINC000147244857 CC For-Sale Anodyne CYP17A1 0 42 COc1ccc(Br)c(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147244861 GG On-Demand Bother TAAR1 21 46 COc1ccc(Br)c(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147244861 GG On-Demand Bother AKR1C2 29 41 CC(C)[C@@H](CCN)CCC(=O)NN(C)C ZINC000147244864 BC For-Sale Reactive KDM7A 0 45 CCCCCCCCNC(=O)N1CSC[C@H]1C(=O)O ZINC000147244910 CF For-Sale Mild ASAH1 108 42 O=C(O)[C@@H]1CCCN1C(=O)c1cccc2c1OCCN2 ZINC000147244913 CD For-Sale Anodyne ACE 43 39 O=C(O)[C@@H]1CCCN1C(=O)c1cccc2c1OCCN2 ZINC000147244913 CD For-Sale Anodyne PREP 62 39 CNc1cccc(NCc2ccccc2Cl)n1 ZINC000147244920 BG For-Sale Anodyne P2RX7 20 41 CNc1cccc(NCc2ccccc2Cl)n1 ZINC000147244920 BG For-Sale Anodyne GPR39 0 42 CN(C)/N=N/c1cn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)[nH]c1=O ZINC000147244927 DA For-Sale Clean ADORA1 18 44 CN(C)/N=N/c1cn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)[nH]c1=O ZINC000147244927 DA For-Sale Clean SLC29A1 44 33 CN(C)/N=N/c1cn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)[nH]c1=O ZINC000147244927 DA For-Sale Clean TK 76 36 CN(C)/N=N/c1cn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)[nH]c1=O ZINC000147244927 DA For-Sale Clean P2RY6 86 43 CN(C)/N=N/c1cn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)[nH]c1=O ZINC000147244927 DA For-Sale Clean TK1 64 56 CN(C)/N=N/c1cn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)[nH]c1=O ZINC000147244927 DA For-Sale Clean CDA 66 42 CN(C)/N=N/c1cn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)[nH]c1=O ZINC000147244927 DA For-Sale Clean P2RY4 65 41 CN(C)/N=N/c1cn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)[nH]c1=O ZINC000147244927 DA For-Sale Clean P2RY2 57 44 CN(C)/N=N/c1cn([C@@H]2O[C@H](CO)[C@@H](O)[C@H]2O)c(=O)[nH]c1=O ZINC000147244927 DA For-Sale Clean P2RY14 59 42 N#Cc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147244953 FG On-Demand Mild SFRP1 75 37 N#Cc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147244953 FG On-Demand Mild WNT3 48 37 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1CCOCC1 ZINC000147245020 GD On-Demand Mild CNR2 17 52 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1CCOCC1 ZINC000147245020 GD On-Demand Mild LRRK2 32 44 COc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1CCOCC1 ZINC000147245020 GD On-Demand Mild L3MBTL3 59 38 Cc1cc(Cl)ccc1Oc1cc(N)nc(N)n1 ZINC000147245077 CE For-Sale Anodyne AGPAT2 49 37 CCc1ncc(C(=O)NCc2ccc3c(c2)OCCO3)s1 ZINC000147245098 DE On-Demand Anodyne NOS2 85 37 O=C(O)C1=Cc2c(F)cccc2O[C@H]1C(F)(F)F ZINC000147245111 CF In-Stock Anodyne PTGS1 36 61 O=C(O)C1=Cc2c(F)cccc2O[C@H]1C(F)(F)F ZINC000147245111 CF In-Stock Anodyne PTGS2 45 61 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild FOLH1 112 65 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild FABP2 0 43 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild PLA2G2C 0 47 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild CCKAR 22 50 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild PLA2G4A 0 45 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild CPT1A 43 52 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild NAALAD2 80 59 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild CCKBR 0 41 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild GGH 0 40 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild EPHX2 25 56 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild Q6UB75_PIG 0 47 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild FABP5 15 43 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild TLR2 0 43 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild ASAH1 90 36 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild SLC22A20 0 43 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild NOD1 117 54 CCCCCCCCNC(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147245134 DD For-Sale Mild CQSS 53 33 N#Cc1ccc(S(=O)(=O)N[C@H]2C[C@@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147245139 FG On-Demand Mild SFRP1 75 37 N#Cc1ccc(S(=O)(=O)N[C@H]2C[C@@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147245139 FG On-Demand Mild WNT3 48 37 CC(C)CN(CC(=O)O)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147245176 CE For-Sale Anodyne ACE 15 41 CC(C)CN(CC(=O)O)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147245176 CE For-Sale Anodyne GPR88 0 51 NC(=O)NCCNc1ncnc2ccc([N+](=O)[O-])cc12 ZINC000147245253 CC On-Demand Bother CLK4 57 36 NC(=O)NCCNc1ncnc2ccc([N+](=O)[O-])cc12 ZINC000147245253 CC On-Demand Bother HTT 0 42 NS(=O)(=O)c1cc(F)ccc1OCCCn1ccnc1 ZINC000147245261 CD For-Sale Anodyne TBXAS1 44 42 NS(=O)(=O)c1cc(F)ccc1OCCCn1ccnc1 ZINC000147245261 CD For-Sale Anodyne CYP17A1 0 47 NS(=O)(=O)c1cc(F)ccc1OCCCn1ccnc1 ZINC000147245261 CD For-Sale Anodyne HMOX2 49 41 NS(=O)(=O)c1cc(F)ccc1OCCCn1ccnc1 ZINC000147245261 CD For-Sale Anodyne QPCT 38 40 CN1CCC(N(C)C(=O)Cc2cccc(OC(F)(F)F)c2)CC1 ZINC000147245328 EF On-Demand Anodyne HCRTR1 24 42 CN1CCC(N(C)C(=O)Cc2cccc(OC(F)(F)F)c2)CC1 ZINC000147245328 EF On-Demand Anodyne CCR5 24 56 CN1CCC(N(C)C(=O)Cc2cccc(OC(F)(F)F)c2)CC1 ZINC000147245328 EF On-Demand Anodyne SLC6A9 28 45 CN1CCC(N(C)C(=O)Cc2cccc(OC(F)(F)F)c2)CC1 ZINC000147245328 EF On-Demand Anodyne MCHR1 17 40 N#Cc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147245347 FG On-Demand Mild SFRP1 75 37 N#Cc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147245347 FG On-Demand Mild WNT3 48 37 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild FOLH1 112 65 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild FABP2 0 43 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild PLA2G2C 0 47 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild CCKAR 22 50 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild PLA2G4A 0 45 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild CPT1A 43 52 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild NAALAD2 80 59 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild CCKBR 0 41 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild GGH 0 40 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild EPHX2 25 56 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild Q6UB75_PIG 0 47 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild FABP5 15 43 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild TLR2 0 43 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild ASAH1 90 36 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild SLC22A20 0 43 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild NOD1 117 54 CCCCCCCCNC(=O)N[C@H](CCC(=O)O)C(=O)O ZINC000147245362 DD For-Sale Mild CQSS 53 33 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc(CS(C)(=O)=O)cc1)C2 ZINC000147245385 GE On-Demand Anodyne BMP1 44 33 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc(CS(C)(=O)=O)cc1)C2 ZINC000147245385 GE On-Demand Anodyne MTNR1A 27 44 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc(CS(C)(=O)=O)cc1)C2 ZINC000147245385 GE On-Demand Anodyne ROCK2 26 42 CC(C)CN(CC(=O)O)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147245422 CE For-Sale Anodyne ACE 15 41 CC(C)CN(CC(=O)O)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147245422 CE For-Sale Anodyne GPR88 0 51 COC(=O)c1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147245468 HF On-Demand Anodyne CA2 29 47 COC(=O)c1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147245468 HF On-Demand Anodyne BMP1 33 46 COC(=O)c1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147245468 HF On-Demand Anodyne CA1 32 47 COC(=O)c1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147245468 HF On-Demand Anodyne CA4 18 46 COC(=O)c1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147245468 HF On-Demand Anodyne CA12 27 47 COC(=O)c1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147245468 HF On-Demand Anodyne CA9 31 47 COC(=O)c1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147245468 HF On-Demand Anodyne NCE103 25 44 COC(=O)c1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147245468 HF On-Demand Anodyne PRMT3 17 40 COC(=O)c1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147245468 HF On-Demand Anodyne MTCA1 31 46 COC(=O)c1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147245468 HF On-Demand Anodyne P96878_MYCTU 41 36 COC(=O)c1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147245468 HF On-Demand Anodyne NAMPT 56 47 Cc1cc(C(=O)NCc2ccc3c(c2)OCCO3)cc([N+](=O)[O-])c1 ZINC000147245508 EF On-Demand Bother PLK1 15 42 N#Cc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147245544 FG On-Demand Mild SFRP1 75 37 N#Cc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147245544 FG On-Demand Mild WNT3 48 37 COc1cccc2c(NCc3ccc(Cl)cc3)cc(C)nc12 ZINC000147245546 DJ For-Sale Anodyne U38 0 42 COc1cccc2c(NCc3ccc(Cl)cc3)cc(C)nc12 ZINC000147245546 DJ For-Sale Anodyne PETD 0 42 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild FABP2 0 62 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild FABP4 22 62 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild PLA2G2C 0 41 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild CPT1A 49 51 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild DNM1 0 43 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild PLA2G4B 43 35 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild FAAH 0 50 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild S1PR2 29 48 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild EPHX2 36 75 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild Q6UB75_PIG 0 44 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild FABP3 38 50 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild FABP5 21 62 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild GNAI1 0 41 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild GNAI3 0 41 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild GNAO1 0 41 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild FABP1 16 50 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild ASAH1 99 36 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild SLC22A20 0 62 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild ACAT 0 46 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild NOD1 47 38 CCCCCCCCNC(=O)NCCCC(=O)O ZINC000147245555 CF For-Sale Mild CQSS 57 35 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(CS(C)(=O)=O)cc1)C2 ZINC000147245606 GE On-Demand Anodyne BMP1 44 33 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(CS(C)(=O)=O)cc1)C2 ZINC000147245606 GE On-Demand Anodyne MTNR1A 27 44 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(CS(C)(=O)=O)cc1)C2 ZINC000147245606 GE On-Demand Anodyne ROCK2 26 42 CC(C)CN(CC(=O)O)C(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147245614 CE For-Sale Anodyne ACE 15 41 CC(C)CN(CC(=O)O)C(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147245614 CE For-Sale Anodyne GPR88 0 51 COC(=O)c1ccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147245703 FE On-Demand Anodyne EPHX2 46 42 CCCCCCCCNC(=O)NC[C@@H](C)C(=O)O ZINC000147245716 CE On-Demand Mild FOLH1 17 41 CCCCCCCCNC(=O)NC[C@@H](C)C(=O)O ZINC000147245716 CE On-Demand Mild CPT1A 25 47 CCCCCCCCNC(=O)NC[C@@H](C)C(=O)O ZINC000147245716 CE On-Demand Mild EPHX2 30 54 CCCCCCCCNC(=O)NC[C@@H](C)C(=O)O ZINC000147245716 CE On-Demand Mild ASAH1 91 36 CCCCCCCCNC(=O)NC[C@@H](C)C(=O)O ZINC000147245716 CE On-Demand Mild NOD1 88 43 CCCCCCCCNC(=O)NC[C@@H](C)C(=O)O ZINC000147245716 CE On-Demand Mild CQSS 52 35 CC(C)CN(CC(=O)O)C(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147245782 CE For-Sale Anodyne ACE 15 41 CC(C)CN(CC(=O)O)C(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147245782 CE For-Sale Anodyne GPR88 0 51 COc1cc(C[C@@H](OC(=O)/C=C/c2ccc3c(c2)O[C@@H](C(=O)O)[C@@H](c2ccc(O)c(OC)c2)O3)C(=O)O)ccc1O ZINC000147245793 KG Annotated Anodyne MMP12 0 53 CCOc1ccccc1C(=O)N1CC[C@H](N)[C@H](CC)C1 ZINC000147245837 CE On-Demand Anodyne HCN1 51 39 CCOc1ccccc1C(=O)N1CC[C@H](N)[C@H](CC)C1 ZINC000147245837 CE On-Demand Anodyne HCN4 51 39 CCOc1ccccc1C(=O)N1CC[C@H](N)[C@H](CC)C1 ZINC000147245837 CE On-Demand Anodyne L3MBTL1 0 40 CCOc1ccccc1C(=O)N1CC[C@H](N)[C@H](CC)C1 ZINC000147245837 CE On-Demand Anodyne TP53BP1 0 40 N#Cc1ccc(-n2cnc3ccccc32)cn1 ZINC000147245839 BE For-Sale Mild PDGFRB 27 56 O=C(O)C1(NCc2ccc(-n3ccnc3)cc2)CCC1 ZINC000147245854 CD On-Demand Anodyne NOS2 79 36 O=C(O)C1(NCc2ccc(-n3ccnc3)cc2)CCC1 ZINC000147245854 CD On-Demand Anodyne UPPS 0 40 CN(C)C(=O)c1cccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)c1 ZINC000147245887 EE On-Demand Anodyne AKR1C3 23 44 CCCCCCCCNC(=O)NC[C@H](C)C(=O)O ZINC000147245906 CE On-Demand Mild FOLH1 17 41 CCCCCCCCNC(=O)NC[C@H](C)C(=O)O ZINC000147245906 CE On-Demand Mild CPT1A 25 47 CCCCCCCCNC(=O)NC[C@H](C)C(=O)O ZINC000147245906 CE On-Demand Mild EPHX2 30 54 CCCCCCCCNC(=O)NC[C@H](C)C(=O)O ZINC000147245906 CE On-Demand Mild ASAH1 91 36 CCCCCCCCNC(=O)NC[C@H](C)C(=O)O ZINC000147245906 CE On-Demand Mild NOD1 88 43 CCCCCCCCNC(=O)NC[C@H](C)C(=O)O ZINC000147245906 CE On-Demand Mild CQSS 52 35 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CC1 ZINC000147245908 BD In-Stock Bother CACNA1C 58 41 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CC1 ZINC000147245908 BD In-Stock Bother SIGMAR1 20 73 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CC1 ZINC000147245908 BD In-Stock Bother CACNA1D 93 41 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CC1 ZINC000147245908 BD In-Stock Bother FAAH 0 53 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CC1 ZINC000147245908 BD In-Stock Bother MGLL 0 41 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CC1 ZINC000147245908 BD In-Stock Bother APR 0 40 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CC1 ZINC000147245908 BD In-Stock Bother LUXR 52 65 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CC1 ZINC000147245908 BD In-Stock Bother TRPM8 25 47 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CC1 ZINC000147245908 BD In-Stock Bother TRAR 27 65 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CC1 ZINC000147245908 BD In-Stock Bother LASR 29 65 O=C(Cc1cccc([N+](=O)[O-])c1)NC1CC1 ZINC000147245908 BD In-Stock Bother OSIGBA0132E09-OSIGBA0108L24.11 0 40 CNc1nccc(Nc2ccc(C#N)cc2F)n1 ZINC000147245917 BE For-Sale Mild CDC7 0 46 N#CC1CCN(C(=O)COc2ccc(C(=O)c3ccccc3)cc2)CC1 ZINC000147245926 EG On-Demand Mild SRD5A2 33 42 N#CC1CCN(C(=O)COc2ccc(C(=O)c3ccccc3)cc2)CC1 ZINC000147245926 EG On-Demand Mild COLA 125 47 COC(=O)c1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147245957 HG On-Demand Anodyne ADRB2 34 41 COC(=O)c1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147245957 HG On-Demand Anodyne ADRB1 61 48 COC(=O)c1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147245957 HG On-Demand Anodyne ADRB3 43 48 COC(=O)c1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147245957 HG On-Demand Anodyne P2RY1 27 45 COC(=O)c1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147245957 HG On-Demand Anodyne RAF1 43 39 COC(=O)c1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147245957 HG On-Demand Anodyne F7 24 40 COC(=O)c1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147245957 HG On-Demand Anodyne ACR 50 52 COC(=O)c1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147245957 HG On-Demand Anodyne TEK 42 36 COC(=O)c1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147245957 HG On-Demand Anodyne Q8MMZ8_EIMTE 52 39 COC(=O)c1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147245957 HG On-Demand Anodyne PDS 64 50 CCOc1ccccc1C(=O)N1CC[C@H](N)[C@@H](CC)C1 ZINC000147246019 CE On-Demand Anodyne HCN1 51 39 CCOc1ccccc1C(=O)N1CC[C@H](N)[C@@H](CC)C1 ZINC000147246019 CE On-Demand Anodyne HCN4 51 39 CCOc1ccccc1C(=O)N1CC[C@H](N)[C@@H](CC)C1 ZINC000147246019 CE On-Demand Anodyne L3MBTL1 0 40 CCOc1ccccc1C(=O)N1CC[C@H](N)[C@@H](CC)C1 ZINC000147246019 CE On-Demand Anodyne TP53BP1 0 40 Cc1cccc(-c2[nH]c(SCc3cccc(F)c3F)nc(=O)c2C#N)c1 ZINC000147246051 FI Annotated Mild CXCR2 22 73 Cc1cccc(-c2[nH]c(SCc3cccc(F)c3F)nc(=O)c2C#N)c1 ZINC000147246051 FI Annotated Mild NS5B 22 46 CN(C)C(=O)c1cccc(S(=O)(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147246087 EE On-Demand Anodyne AKR1C3 23 44 N#Cc1ccc(Nc2ccnc(N)n2)c(F)c1 ZINC000147246127 BD For-Sale Mild HRH4 15 40 CCCCCCCCNC(=O)N(CCC(=O)O)C1CC1 ZINC000147246131 CF For-Sale Mild PPARA 0 43 CCCCCCCCNC(=O)N(CCC(=O)O)C1CC1 ZINC000147246131 CF For-Sale Mild FABP2 0 43 CCCCCCCCNC(=O)N(CCC(=O)O)C1CC1 ZINC000147246131 CF For-Sale Mild FABP4 15 43 CCCCCCCCNC(=O)N(CCC(=O)O)C1CC1 ZINC000147246131 CF For-Sale Mild EPHX2 40 51 CCCCCCCCNC(=O)N(CCC(=O)O)C1CC1 ZINC000147246131 CF For-Sale Mild FABP5 15 43 CCCCCCCCNC(=O)N(CCC(=O)O)C1CC1 ZINC000147246131 CF For-Sale Mild GNAI1 0 43 CCCCCCCCNC(=O)N(CCC(=O)O)C1CC1 ZINC000147246131 CF For-Sale Mild GNAI3 0 43 CCCCCCCCNC(=O)N(CCC(=O)O)C1CC1 ZINC000147246131 CF For-Sale Mild GNAO1 0 43 CCCCCCCCNC(=O)N(CCC(=O)O)C1CC1 ZINC000147246131 CF For-Sale Mild ASAH1 77 33 CCCCCCCCNC(=O)N(CCC(=O)O)C1CC1 ZINC000147246131 CF For-Sale Mild SLC22A20 0 43 CCCCCCCCNC(=O)N(CCC(=O)O)C1CC1 ZINC000147246131 CF For-Sale Mild LASR 48 34 CC(C)CCCCNC(=O)CCc1cccc(N)c1 ZINC000147246145 CG For-Sale Anodyne MTNR1A 23 41 CC(C)CCCCNC(=O)CCc1cccc(N)c1 ZINC000147246145 CG For-Sale Anodyne MTNR1B 21 41 CC(C)CCCCNC(=O)CCc1cccc(N)c1 ZINC000147246145 CG For-Sale Anodyne GRIA1 47 47 CC(C)CCCCNC(=O)CCc1cccc(N)c1 ZINC000147246145 CG For-Sale Anodyne PAM 0 43 CC(C)CCCCNC(=O)CCc1cccc(N)c1 ZINC000147246145 CG For-Sale Anodyne POLG_WNV 43 36 CC(C)CCCCNC(=O)CCc1cccc(N)c1 ZINC000147246145 CG For-Sale Anodyne CRTM 40 37 COC(=O)c1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147246169 HG On-Demand Anodyne ADRB2 34 41 COC(=O)c1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147246169 HG On-Demand Anodyne ADRB1 61 48 COC(=O)c1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147246169 HG On-Demand Anodyne ADRB3 43 48 COC(=O)c1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147246169 HG On-Demand Anodyne P2RY1 27 45 COC(=O)c1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147246169 HG On-Demand Anodyne RAF1 43 39 COC(=O)c1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147246169 HG On-Demand Anodyne F7 24 40 COC(=O)c1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147246169 HG On-Demand Anodyne ACR 50 52 COC(=O)c1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147246169 HG On-Demand Anodyne TEK 42 36 COC(=O)c1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147246169 HG On-Demand Anodyne Q8MMZ8_EIMTE 52 39 COC(=O)c1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1 ZINC000147246169 HG On-Demand Anodyne PDS 64 50 CCOc1ccccc1C(=O)N1CC[C@@H](N)[C@H](CC)C1 ZINC000147246236 CE On-Demand Anodyne HCN1 51 39 CCOc1ccccc1C(=O)N1CC[C@@H](N)[C@H](CC)C1 ZINC000147246236 CE On-Demand Anodyne HCN4 51 39 CCOc1ccccc1C(=O)N1CC[C@@H](N)[C@H](CC)C1 ZINC000147246236 CE On-Demand Anodyne L3MBTL1 0 40 CCOc1ccccc1C(=O)N1CC[C@@H](N)[C@H](CC)C1 ZINC000147246236 CE On-Demand Anodyne TP53BP1 0 40 CC(C)CN(CC(=O)O)C(=O)C1[C@H]2CCCC[C@H]12 ZINC000147246238 CD On-Demand Anodyne ACE 51 37 CN(C)C(=O)c1cccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)c1 ZINC000147246318 EE On-Demand Anodyne AKR1C3 23 44 CCCNc1ncc(F)c(Nc2ccc(C#N)cc2F)n1 ZINC000147246328 CG For-Sale Mild SYK 36 50 CCCCCCCCNC(=O)N1CCN(CC(=O)O)CC1 ZINC000147246338 CD For-Sale Mild PLA2G2A 28 41 CCCCCCCCNC(=O)N1CCN(CC(=O)O)CC1 ZINC000147246338 CD For-Sale Mild EPHX2 26 42 CCCCCCCCNC(=O)N1CCN(CC(=O)O)CC1 ZINC000147246338 CD For-Sale Mild ASAH1 102 39 CCCCCCCCNC(=O)N1CCN(CC(=O)O)CC1 ZINC000147246338 CD For-Sale Mild NMUR1 0 44 O=C(CN1CCC[C@H](O)C1)N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147246345 HC On-Demand Anodyne F10 23 42 O=C(CN1CCC[C@H](O)C1)N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147246345 HC On-Demand Anodyne APP 52 43 O=C(CN1CCC[C@H](O)C1)N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147246345 HC On-Demand Anodyne LSS 17 42 O=C(CN1CCC[C@H](O)C1)N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147246345 HC On-Demand Anodyne TGM2 51 38 O=C(CN1CCC[C@H](O)C1)N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147246345 HC On-Demand Anodyne F13A1 62 38 CCOC1CCN(C(=O)C2CCN(Cc3ccnnc3)CC2)CC1 ZINC000147246360 ED For-Sale Anodyne HRH3 17 46 CCOC1CCN(C(=O)C2CCN(Cc3ccnnc3)CC2)CC1 ZINC000147246360 ED For-Sale Anodyne SSTR5 51 34 Cc1ccc(C(=O)N2CCC(c3ccc(C(F)(F)F)cc3)CC2)cc1N ZINC000147246382 FJ On-Demand Anodyne SLC9A1 45 41 Cc1ccc(C(=O)N2CCC(c3ccc(C(F)(F)F)cc3)CC2)cc1N ZINC000147246382 FJ On-Demand Anodyne FASN 42 40 Cc1ccc(C(=O)N2CCC(c3ccc(C(F)(F)F)cc3)CC2)cc1N ZINC000147246382 FJ On-Demand Anodyne RBP4 26 46 Cc1ccc(C(=O)N2CCC(c3ccc(C(F)(F)F)cc3)CC2)cc1N ZINC000147246382 FJ On-Demand Anodyne L3MBTL3 66 42 Cc1ccc(C(=O)N2CCC(c3ccc(C(F)(F)F)cc3)CC2)cc1N ZINC000147246382 FJ On-Demand Anodyne HPGD 16 40 NC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147246388 ED On-Demand Anodyne ENV 40 33 CC(C)(C)OC(=O)N1CCC([C@@H](CO)n2c(-c3ccccc3)nc3ccccc32)CC1 ZINC000147246422 HJ For-Sale Anodyne P2RY12 51 33 CC(C)(C)OC(=O)N1CCC([C@@H](CO)n2c(-c3ccccc3)nc3ccccc32)CC1 ZINC000147246422 HJ For-Sale Anodyne PDE6D 111 51 CC(C)(C)OC(=O)N1CCC([C@@H](CO)n2c(-c3ccccc3)nc3ccccc32)CC1 ZINC000147246422 HJ For-Sale Anodyne GPR119 45 42 CCOc1cc(C)cc(C(=O)O)c1OC ZINC000147246425 BE For-Sale Anodyne ALS 20 41 CCOc1ccccc1C(=O)N1CC[C@@H](N)[C@@H](CC)C1 ZINC000147246445 CE On-Demand Anodyne HCN1 51 39 CCOc1ccccc1C(=O)N1CC[C@@H](N)[C@@H](CC)C1 ZINC000147246445 CE On-Demand Anodyne HCN4 51 39 CCOc1ccccc1C(=O)N1CC[C@@H](N)[C@@H](CC)C1 ZINC000147246445 CE On-Demand Anodyne L3MBTL1 0 40 CCOc1ccccc1C(=O)N1CC[C@@H](N)[C@@H](CC)C1 ZINC000147246445 CE On-Demand Anodyne TP53BP1 0 40 CC(C)Oc1ccc(-c2[nH]c(SCc3cccc(F)c3F)nc(=O)c2C#N)cc1 ZINC000147246455 HJ Annotated Mild CXCR2 28 75 CC(C)Oc1ccc(-c2[nH]c(SCc3cccc(F)c3F)nc(=O)c2C#N)cc1 ZINC000147246455 HJ Annotated Mild NS5B 23 42 C[C@@H]1CCN(C(=O)c2csc(-c3ccccc3)n2)[C@@H]2CCCC[C@@H]12 ZINC000147246471 EJ On-Demand Anodyne PTGER1 25 42 C[C@@H]1CCN(C(=O)c2csc(-c3ccccc3)n2)[C@@H]2CCCC[C@@H]12 ZINC000147246471 EJ On-Demand Anodyne CPT1A 37 41 C[C@@H]1CCN(C(=O)c2csc(-c3ccccc3)n2)[C@@H]2CCCC[C@@H]12 ZINC000147246471 EJ On-Demand Anodyne TRPC6 52 39 C[C@@H]1CCN(C(=O)c2csc(-c3ccccc3)n2)[C@@H]2CCCC[C@@H]12 ZINC000147246471 EJ On-Demand Anodyne TRPC3 46 39 O=C(O)[C@H]1CCCC[C@H]1C(=O)NCC(F)F ZINC000147246513 BD On-Demand Anodyne ACE 0 56 CN[C@@H]1CCN(c2ccc(C(N)=O)cc2)C1 ZINC000147246526 BC For-Sale Anodyne HRH4 65 45 CCCCCCCCNC(=O)N1CCC[C@@H]1CC(=O)O ZINC000147246534 CF For-Sale Mild TPP2 37 46 CCCCCCCCNC(=O)N1CCC[C@@H]1CC(=O)O ZINC000147246534 CF For-Sale Mild GNAI1 0 42 CCCCCCCCNC(=O)N1CCC[C@@H]1CC(=O)O ZINC000147246534 CF For-Sale Mild GNAI3 0 42 CCCCCCCCNC(=O)N1CCC[C@@H]1CC(=O)O ZINC000147246534 CF For-Sale Mild GNAO1 0 42 CCCCCCCCNC(=O)N1CCC[C@@H]1CC(=O)O ZINC000147246534 CF For-Sale Mild ASAH1 101 40 O=C(CN1CCC[C@@H](O)C1)N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147246560 HC On-Demand Anodyne F10 19 42 O=C(CN1CCC[C@@H](O)C1)N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147246560 HC On-Demand Anodyne APP 52 43 O=C(CN1CCC[C@@H](O)C1)N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147246560 HC On-Demand Anodyne LSS 16 42 O=C(CN1CCC[C@@H](O)C1)N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147246560 HC On-Demand Anodyne TGM2 51 38 O=C(CN1CCC[C@@H](O)C1)N1CCN(S(=O)(=O)c2ccc(Cl)cc2)CC1 ZINC000147246560 HC On-Demand Anodyne F13A1 57 38 NC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147246608 ED On-Demand Anodyne ENV 40 33 CC(C)(C)OC(=O)N1CCC([C@H](CO)n2c(-c3ccccc3)nc3ccccc32)CC1 ZINC000147246614 HJ For-Sale Anodyne P2RY12 51 33 CC(C)(C)OC(=O)N1CCC([C@H](CO)n2c(-c3ccccc3)nc3ccccc32)CC1 ZINC000147246614 HJ For-Sale Anodyne PDE6D 111 51 CC(C)(C)OC(=O)N1CCC([C@H](CO)n2c(-c3ccccc3)nc3ccccc32)CC1 ZINC000147246614 HJ For-Sale Anodyne NR1H4 28 40 CC(C)(C)OC(=O)N1CCC([C@H](CO)n2c(-c3ccccc3)nc3ccccc32)CC1 ZINC000147246614 HJ For-Sale Anodyne GPR119 45 42 CC(C)CCCCNC(=O)CCOc1cccc(N)c1 ZINC000147246644 CF For-Sale Anodyne HRH2 24 40 CC(C)CCCCNC(=O)CCOc1cccc(N)c1 ZINC000147246644 CF For-Sale Anodyne MTNR1A 38 40 CC(C)CCCCNC(=O)CCOc1cccc(N)c1 ZINC000147246644 CF For-Sale Anodyne MTNR1B 31 40 CC(C)CN(CC(=O)O)C(=O)C1[C@@H]2CCCC[C@@H]12 ZINC000147246646 CD On-Demand Anodyne ACE 51 37 CC(C)C[C@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147246660 CD For-Sale Anodyne CCKAR 31 45 CC(C)C[C@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147246660 CD For-Sale Anodyne FPR1 55 35 CC(C)C[C@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147246660 CD For-Sale Anodyne NPR 49 34 O=C(O)[C@@H]1CCCC[C@H]1C(=O)NCC(F)F ZINC000147246675 BD For-Sale Anodyne ACE 0 56 CCc1cc(C)cc(C(=O)O)c1OC ZINC000147246686 AE For-Sale Anodyne TPMT 49 38 N#Cc1ccc(Nc2nc(N)nc3ccccc23)c(F)c1 ZINC000147246718 CF For-Sale Mild ABCG2 25 46 Cn1c(=O)c2[nH]c(NCCNC(N)=O)nc2n(C)c1=O ZINC000147246732 CA For-Sale Anodyne ADORA1 27 44 CCCCCCCCNC(=O)N1CCC[C@H]1CC(=O)O ZINC000147246749 CF For-Sale Mild TPP2 37 46 CCCCCCCCNC(=O)N1CCC[C@H]1CC(=O)O ZINC000147246749 CF For-Sale Mild GNAI1 0 42 CCCCCCCCNC(=O)N1CCC[C@H]1CC(=O)O ZINC000147246749 CF For-Sale Mild GNAI3 0 42 CCCCCCCCNC(=O)N1CCC[C@H]1CC(=O)O ZINC000147246749 CF For-Sale Mild GNAO1 0 42 CCCCCCCCNC(=O)N1CCC[C@H]1CC(=O)O ZINC000147246749 CF For-Sale Mild ASAH1 101 40 CN[C@H]1CCN(c2ccc(C(N)=O)cc2)C1 ZINC000147246757 BC For-Sale Anodyne HRH4 65 45 C[C@@H]1CCN(C(=O)c2csc(-c3ccccc3)n2)[C@H]2CCCC[C@H]21 ZINC000147246771 EJ On-Demand Anodyne PTGER1 25 42 C[C@@H]1CCN(C(=O)c2csc(-c3ccccc3)n2)[C@H]2CCCC[C@H]21 ZINC000147246771 EJ On-Demand Anodyne CPT1A 37 41 C[C@@H]1CCN(C(=O)c2csc(-c3ccccc3)n2)[C@H]2CCCC[C@H]21 ZINC000147246771 EJ On-Demand Anodyne TRPC6 52 39 C[C@@H]1CCN(C(=O)c2csc(-c3ccccc3)n2)[C@H]2CCCC[C@H]21 ZINC000147246771 EJ On-Demand Anodyne TRPC3 46 39 O=C(O)[C@H]1CCCC[C@@H]1C(=O)NCC(F)F ZINC000147246815 BD For-Sale Anodyne ACE 0 56 O=C(CCCc1ccccc1)N1CCC[C@H](CCBr)C1 ZINC000147246831 EI For-Sale Reactive FKBP1A 34 42 O=C(CCCc1ccccc1)N1CCC[C@H](CCBr)C1 ZINC000147246831 EI For-Sale Reactive PREP 89 55 CC(C)C[C@@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147246842 CD For-Sale Anodyne CCKAR 31 45 CC(C)C[C@@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147246842 CD For-Sale Anodyne FPR1 55 35 CC(C)C[C@@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147246842 CD For-Sale Anodyne NPR 49 34 Cc1oc2ccccc2c1CNc1cccc(C(=O)O)c1 ZINC000147246861 CI On-Demand Anodyne AKR1C3 39 44 Cc1oc2ccccc2c1CNc1cccc(C(=O)O)c1 ZINC000147246861 CI On-Demand Anodyne REP 0 40 Cc1oc2ccccc2c1CNc1cccc(C(=O)O)c1 ZINC000147246861 CI On-Demand Anodyne KCNK3 48 34 CCCCCCCCNC(=O)N(C)[C@@H](CC)C(=O)O ZINC000147246900 CF For-Sale Mild DNM1 0 44 CCCCCCCCNC(=O)N(C)[C@@H](CC)C(=O)O ZINC000147246900 CF For-Sale Mild EPHX2 25 44 CCCCCCCCNC(=O)N(C)[C@@H](CC)C(=O)O ZINC000147246900 CF For-Sale Mild ASAH1 78 32 CCCCCCCCNC(=O)N(C)[C@@H](CC)C(=O)O ZINC000147246900 CF For-Sale Mild NOD1 74 39 CCCCCCCCNC(=O)N(C)[C@@H](CC)C(=O)O ZINC000147246900 CF For-Sale Mild CQSS 52 33 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne CHRM2 35 40 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne AVPR1A 23 45 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne GRM3 20 55 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne MMP13 35 44 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne SLC18A3 24 49 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne MMP3 33 43 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne MMP9 33 44 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne MMP7 36 43 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne MMP1 30 44 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne PTR1 41 35 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne L3MBTL1 0 41 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne L3MBTL3 70 41 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne GPR183 0 45 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147246916 CD On-Demand Anodyne SLC6A7 0 43 CC(C)CCCCNC(=O)c1ccc(N(C)C)c(N)c1 ZINC000147246922 CF For-Sale Anodyne FOLH1 30 41 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCC1 ZINC000147246985 CC For-Sale Anodyne HTR2A 29 42 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCC1 ZINC000147246985 CC For-Sale Anodyne LTA4H 37 48 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCC1 ZINC000147246985 CC For-Sale Anodyne HRH3 23 45 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCC1 ZINC000147246985 CC For-Sale Anodyne MCHR1 0 44 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCC1 ZINC000147246985 CC For-Sale Anodyne PSMB2 47 38 NS(=O)(=O)c1cc(F)ccc1OCCN1CCCC1 ZINC000147246985 CC For-Sale Anodyne PSMB1 41 38 O=[N+]([O-])c1cc(CCl)ccc1Oc1ccc(Cl)c(F)c1 ZINC000147246988 DJ For-Sale Reactive PPXII 0 40 CSCC[C@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147246991 DD For-Sale Anodyne CCKAR 0 47 O=C(CCCc1ccccc1)N1CCC[C@@H](CCBr)C1 ZINC000147246998 EI For-Sale Reactive FKBP1A 34 42 O=C(CCCc1ccccc1)N1CCC[C@@H](CCBr)C1 ZINC000147246998 EI For-Sale Reactive PREP 89 55 CCOc1ccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147247002 HG On-Demand Mild F2 17 44 CCOc1ccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147247002 HG On-Demand Mild PLG 24 44 CCOc1ccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147247002 HG On-Demand Mild MMP13 25 40 CCOc1ccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147247002 HG On-Demand Mild TRY2_BOVIN 54 34 CCOc1ccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147247002 HG On-Demand Mild ADAM17 20 40 CCOc1ccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147247002 HG On-Demand Mild ST14 89 44 CCOc1ccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)cc1 ZINC000147247002 HG On-Demand Mild TMPRSS6 55 40 O=C(NCC(F)F)[C@H]1CCCC[C@H]1C(=O)O ZINC000147247011 BD For-Sale Anodyne ACE 0 56 CCCCCCCCNC(=O)N(C)[C@H](CC)C(=O)O ZINC000147247020 CF For-Sale Mild DNM1 0 44 CCCCCCCCNC(=O)N(C)[C@H](CC)C(=O)O ZINC000147247020 CF For-Sale Mild EPHX2 25 44 CCCCCCCCNC(=O)N(C)[C@H](CC)C(=O)O ZINC000147247020 CF For-Sale Mild ASAH1 78 32 CCCCCCCCNC(=O)N(C)[C@H](CC)C(=O)O ZINC000147247020 CF For-Sale Mild NOD1 74 39 CCCCCCCCNC(=O)N(C)[C@H](CC)C(=O)O ZINC000147247020 CF For-Sale Mild CQSS 52 33 CS(=O)(=O)Cc1ccc(CNC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147247036 HG On-Demand Anodyne MAPK9 17 40 CS(=O)(=O)Cc1ccc(CNC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147247036 HG On-Demand Anodyne NAMPT 71 42 CC1(C)CC(=O)O[C@@H]1CC(=O)O ZINC000147247041 AC For-Sale Anodyne LANCL2 46 29 CN(C)C(=O)Nc1ccc(C(=O)c2ccc(Cl)cc2)cc1 ZINC000147247074 DH For-Sale Anodyne F10 16 45 CN(C)C(=O)Nc1ccc(C(=O)c2ccc(Cl)cc2)cc1 ZINC000147247074 DH For-Sale Anodyne ACR 19 40 CN(C)C(=O)Nc1ccc(C(=O)c2ccc(Cl)cc2)cc1 ZINC000147247074 DH For-Sale Anodyne UTS2 42 34 CN(C)C(=O)Nc1ccc(C(=O)c2ccc(Cl)cc2)cc1 ZINC000147247074 DH For-Sale Anodyne Q25615_ONCVO 25 40 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne CHRM2 35 40 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne AVPR1A 23 45 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne GRM3 20 55 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne MMP13 35 44 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne SLC18A3 24 49 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne MMP3 33 43 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne MMP9 33 44 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne MMP7 36 43 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne MMP1 30 44 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne PTR1 41 35 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne L3MBTL1 0 41 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne L3MBTL3 70 41 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne GPR183 0 45 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147247078 CD On-Demand Anodyne SLC6A7 0 43 CCNc1ccc([N+](=O)[O-])c(Oc2ccc(Cl)cc2C)n1 ZINC000147247126 DI For-Sale Bother S1PR4 24 40 COC(=O)CCN1C(=O)C=C(C(C)C)C1=O ZINC000147247141 BC Annotated Anodyne KAT2B 0 43 C[C@H](CNS(=O)(=O)c1cc(Cl)cc(Cl)c1)CC(=O)O ZINC000147247171 EE On-Demand Anodyne TBXA2R 42 33 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne CHRM2 35 40 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne AVPR1A 23 45 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne GRM3 20 55 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne MMP13 35 44 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne SLC18A3 24 49 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne MMP3 33 43 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne MMP9 33 44 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne MMP7 36 43 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne MMP1 30 44 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne PTR1 41 35 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne L3MBTL1 0 41 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne L3MBTL3 70 41 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne GPR183 0 45 CC[C@@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247201 CD On-Demand Anodyne SLC6A7 0 43 CC1(C)CC(=O)O[C@H]1CC(=O)O ZINC000147247220 AC For-Sale Anodyne LANCL2 46 29 CC[C@H](C)[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147247271 CE For-Sale Anodyne ACE2 48 37 CC[C@H](C)[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147247271 CE For-Sale Anodyne GPR88 0 50 CN(C)C(=O)Nc1ccc(C(=O)c2ccc(Cl)cc2)c(Cl)c1 ZINC000147247274 EI For-Sale Anodyne F10 17 42 CC12C[C@@H]3CC(C[C@H](C3)C1)N2C(=O)OCc1ccccc1 ZINC000147247297 CH For-Sale Anodyne PREP 24 41 CC12C[C@@H]3CC(C[C@H](C3)C1)N2C(=O)OCc1ccccc1 ZINC000147247297 CH For-Sale Anodyne EPHX2 29 45 CC12C[C@@H]3CC(C[C@H](C3)C1)N2C(=O)OCc1ccccc1 ZINC000147247297 CH For-Sale Anodyne SLC12A5 71 39 C[C@@H](CNS(=O)(=O)c1cc(Cl)cc(Cl)c1)CC(=O)O ZINC000147247306 EE On-Demand Anodyne TBXA2R 42 33 Cc1cccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)c1 ZINC000147247315 GG On-Demand Mild CACNA1B 20 40 Cc1cccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)c1 ZINC000147247315 GG On-Demand Mild ST14 76 38 Cc1cccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)c1 ZINC000147247315 GG On-Demand Mild AKR1C3 22 41 Cc1cccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)c1 ZINC000147247315 GG On-Demand Mild SFRP1 43 35 Cc1cccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)c1 ZINC000147247315 GG On-Demand Mild LIMK2 18 40 Cc1cccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)c1 ZINC000147247315 GG On-Demand Mild L3MBTL3 53 40 Cc1cccc(NS(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)c1 ZINC000147247315 GG On-Demand Mild TMPRSS6 42 36 CS(=O)(=O)Cc1ccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147247343 GG On-Demand Anodyne FBP1 22 42 CS(=O)(=O)Cc1ccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147247343 GG On-Demand Anodyne MDM2 90 36 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne CHRM2 35 40 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne AVPR1A 23 45 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne GRM3 20 55 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne MMP13 35 44 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne SLC18A3 24 49 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne MMP3 33 43 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne MMP9 33 44 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne MMP7 36 43 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne MMP1 30 44 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne PTR1 41 35 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne L3MBTL1 0 41 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne L3MBTL3 70 41 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne GPR183 0 45 CC[C@H]1CN(C(=O)c2ccc(OC)cc2)CC[C@H]1N ZINC000147247360 CD On-Demand Anodyne SLC6A7 0 43 CCOC(=O)c1c(NC)nc(-c2ccccc2)nc1-c1ccccc1 ZINC000147247382 EI For-Sale Anodyne ADORA1 39 59 CCOC(=O)c1c(NC)nc(-c2ccccc2)nc1-c1ccccc1 ZINC000147247382 EI For-Sale Anodyne DHODH 26 46 CCOC(=O)c1c(NC)nc(-c2ccccc2)nc1-c1ccccc1 ZINC000147247382 EI For-Sale Anodyne ADORA2A 20 51 CCOC(=O)c1c(NC)nc(-c2ccccc2)nc1-c1ccccc1 ZINC000147247382 EI For-Sale Anodyne PDE4B 21 41 CCOC(=O)c1c(NC)nc(-c2ccccc2)nc1-c1ccccc1 ZINC000147247382 EI For-Sale Anodyne TACR3 47 38 CCOC(=O)c1c(NC)nc(-c2ccccc2)nc1-c1ccccc1 ZINC000147247382 EI For-Sale Anodyne ADORA3 61 59 CCCc1c(NC)ncnc1Nc1ccc(C#N)cc1F ZINC000147247402 CG For-Sale Mild FLT1 0 45 CCCCCCCCNC(=O)N[C@@H](CC(=O)O)C(=O)O ZINC000147247405 CD For-Sale Mild FOLH1 64 49 CCCCCCCCNC(=O)N[C@@H](CC(=O)O)C(=O)O ZINC000147247405 CD For-Sale Mild CPT1A 52 60 CCCCCCCCNC(=O)N[C@@H](CC(=O)O)C(=O)O ZINC000147247405 CD For-Sale Mild ENPEP 42 31 CCCCCCCCNC(=O)N[C@@H](CC(=O)O)C(=O)O ZINC000147247405 CD For-Sale Mild EPHX2 25 67 CCCCCCCCNC(=O)N[C@@H](CC(=O)O)C(=O)O ZINC000147247405 CD For-Sale Mild Q6UB75_PIG 0 42 CCCCCCCCNC(=O)N[C@@H](CC(=O)O)C(=O)O ZINC000147247405 CD For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N[C@@H](CC(=O)O)C(=O)O ZINC000147247405 CD For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N[C@@H](CC(=O)O)C(=O)O ZINC000147247405 CD For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N[C@@H](CC(=O)O)C(=O)O ZINC000147247405 CD For-Sale Mild ASAH1 87 35 CCCCCCCCNC(=O)N[C@@H](CC(=O)O)C(=O)O ZINC000147247405 CD For-Sale Mild NOD1 94 45 CCCCCCCCNC(=O)N[C@@H](CC(=O)O)C(=O)O ZINC000147247405 CD For-Sale Mild CQSS 50 31 CC[C@H](C)[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147247456 CE For-Sale Anodyne ACE2 48 37 CC[C@H](C)[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147247456 CE For-Sale Anodyne GPR88 0 50 CS(=O)(=O)Cc1ccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147247489 GG On-Demand Anodyne FBP1 22 42 CS(=O)(=O)Cc1ccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147247489 GG On-Demand Anodyne MDM2 90 36 CCCCCCCCNC(=O)N1CC[C@@](C)(C(=O)O)C1 ZINC000147247548 CF On-Demand Mild ASAH1 99 37 C[C@H](CCCCCCCCc1ccccc1)C[C@@]1(C)C[C@@H](C)[C@](O)(CC(=O)O)OO1 ZINC000147247560 HK Annotated Reactive LTB4R 40 43 CC[C@H](C)[C@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147247576 CE For-Sale Anodyne ACE2 48 37 CC[C@H](C)[C@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147247576 CE For-Sale Anodyne GPR88 0 50 CS(=O)(=O)Cc1ccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147247586 GG On-Demand Anodyne FBP1 22 42 CS(=O)(=O)Cc1ccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147247586 GG On-Demand Anodyne MDM2 90 36 COc1ccc(CC(N)=O)c(C)c1 ZINC000147247602 AD In-Stock Anodyne PTGS2 26 44 COc1ccc(CC(N)=O)c(C)c1 ZINC000147247602 AD In-Stock Anodyne MTR1B_CHICK 80 34 COc1ccc(CC(N)=O)c(C)c1 ZINC000147247602 AD In-Stock Anodyne PLA2G2A 48 44 COc1ccc(CC(N)=O)c(C)c1 ZINC000147247602 AD In-Stock Anodyne MTNR1A 53 49 COc1ccc(CC(N)=O)c(C)c1 ZINC000147247602 AD In-Stock Anodyne MTNR1B 50 37 CCOC(=O)c1cnc(-c2ccc(Cl)cc2)nc1NC ZINC000147247628 CG For-Sale Anodyne JUN 19 52 CCOC(=O)c1cnc(-c2ccc(Cl)cc2)nc1NC ZINC000147247628 CG For-Sale Anodyne ADORA3 18 43 CCOC(=O)c1cnc(-c2ccc(Cl)cc2)nc1NC ZINC000147247628 CG For-Sale Anodyne SCN10A 44 34 CCCNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147247635 DH For-Sale Mild INSR 33 41 CCCNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147247635 DH For-Sale Mild MAPK9 32 42 CCCNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147247635 DH For-Sale Mild MAPK10 33 42 CCCNc1ncc(Cl)c(Nc2ccc(C#N)cc2F)n1 ZINC000147247635 DH For-Sale Mild ALK 33 41 Cc1cccc(OCCNC(=O)c2cnc3c(cnn3Cc3ccccc3)c2)c1 ZINC000147247649 GH On-Demand Anodyne DRD4 43 34 Cc1cccc(OCCNC(=O)c2cnc3c(cnn3Cc3ccccc3)c2)c1 ZINC000147247649 GH On-Demand Anodyne HRH2 46 40 O=C(O)C1CCN(C(=O)c2cccc3c2OCCN3)CC1 ZINC000147247669 CD For-Sale Anodyne L3MBTL1 0 40 O=C(O)C1CCN(C(=O)c2cccc3c2OCCN3)CC1 ZINC000147247669 CD For-Sale Anodyne L3MBTL3 56 40 O=C(O)C1CCN(C(=O)c2cccc3c2OCCN3)CC1 ZINC000147247669 CD For-Sale Anodyne TP53BP1 0 40 Cc1cc(Cl)ccc1Oc1nc(N)nc2ccccc12 ZINC000147247682 CH For-Sale Anodyne DHFR 31 42 Cc1cc(Cl)ccc1Oc1nc(N)nc2ccccc12 ZINC000147247682 CH For-Sale Anodyne FOLA 42 42 Cc1cc(Cl)ccc1Oc1nc(N)nc2ccccc12 ZINC000147247682 CH For-Sale Anodyne DRTS_TOXGO 34 40 Cc1cc(Cl)ccc1Oc1nc(N)nc2ccccc12 ZINC000147247682 CH For-Sale Anodyne DYR_PNECA 26 40 CCCCCCCCNC(=O)N1CC[C@](C)(C(=O)O)C1 ZINC000147247695 CF On-Demand Mild ASAH1 99 37 CC[C@@H](Cc1ccccc1)Nc1ccc(Cl)cc1Br ZINC000147247696 EK For-Sale Anodyne ACPS 0 42 CS(=O)(=O)Cc1ccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147247711 GG On-Demand Anodyne FBP1 22 42 CS(=O)(=O)Cc1ccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147247711 GG On-Demand Anodyne MDM2 90 36 CC[C@H](C)[C@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147247738 CE For-Sale Anodyne ACE2 48 37 CC[C@H](C)[C@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147247738 CE For-Sale Anodyne GPR88 0 50 CCOC(=O)COc1c(OC)cccc1C(=O)OCC ZINC000147247745 CD For-Sale Anodyne KCNK3 43 40 CCOC(=O)COc1c(OC)cccc1C(=O)OCC ZINC000147247745 CD For-Sale Anodyne KCNK9 33 40 CC(C)CCCCNC(=O)c1cc2cc(N)ccc2[nH]1 ZINC000147247789 CG For-Sale Anodyne CCKAR 25 46 CC(C)CCCCNC(=O)c1cc2cc(N)ccc2[nH]1 ZINC000147247789 CG For-Sale Anodyne PYGL 84 47 COc1cc(N)ccc1C(=O)c1ccc(Cl)cc1 ZINC000147247814 CG For-Sale Anodyne HTR4 43 38 COc1cc(N)ccc1C(=O)c1ccc(Cl)cc1 ZINC000147247814 CG For-Sale Anodyne CYSP_PLAFA 27 40 O=[N+]([O-])c1ccc(Oc2ccc(Cl)c(F)c2)c(CCl)c1 ZINC000147247839 DJ For-Sale Reactive TBXA2R 23 43 O=[N+]([O-])c1ccc(Oc2ccc(Cl)c(F)c2)c(CCl)c1 ZINC000147247839 DJ For-Sale Reactive ENR 0 46 O=[N+]([O-])c1ccc(Oc2ccc(Cl)c(F)c2)c(CCl)c1 ZINC000147247839 DJ For-Sale Reactive PPOX1 17 51 CCCCCCCCNC(=O)N1CCC(C)(C(=O)O)CC1 ZINC000147247851 CG On-Demand Mild ASAH1 102 38 CC[C@H](Cc1ccccc1)Nc1ccc(Cl)cc1Br ZINC000147247861 EK For-Sale Anodyne ACPS 0 42 N#Cc1ccc(Nc2nc(N)ncc2Cl)c(F)c1 ZINC000147247868 CE For-Sale Mild MAPK9 20 42 N#Cc1ccc(Nc2nc(N)ncc2Cl)c(F)c1 ZINC000147247868 CE For-Sale Mild MAPK10 18 42 O=C(O)C1(NCCc2ccccc2[N+](=O)[O-])CCC1 ZINC000147247877 CD For-Sale Bother COLA 114 38 O=C(O)C1(NCCc2ccccc2[N+](=O)[O-])CCC1 ZINC000147247877 CD For-Sale Bother PQSD 0 45 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147247971 FD On-Demand Anodyne NPY2R 16 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147247971 FD On-Demand Anodyne L3MBTL3 60 41 CS(=O)(=O)Cc1ccc(CNC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147247976 EE On-Demand Anodyne NAMPT 41 37 CN(C)C(=O)Nc1ccc(C(=O)c2ccccc2)c(Cl)c1 ZINC000147247993 DH For-Sale Anodyne ECR 27 40 CN(C)C(=O)Nc1ccc(C(=O)c2ccccc2)c(Cl)c1 ZINC000147247993 DH For-Sale Anodyne GRM4 37 40 CN(C)C(=O)Nc1ccc(C(=O)c2ccccc2)c(Cl)c1 ZINC000147247993 DH For-Sale Anodyne SMO 21 42 CN(C)C(=O)Nc1ccc(C(=O)c2ccccc2)c(Cl)c1 ZINC000147247993 DH For-Sale Anodyne KCNK3 70 43 CCCCCCCCNC(=O)N(CC)[C@@H](C)CC(=O)O ZINC000147248017 CG For-Sale Mild CPT1A 46 47 CCCCCCCCNC(=O)N(CC)[C@@H](C)CC(=O)O ZINC000147248017 CG For-Sale Mild EPHX2 26 43 CCCCCCCCNC(=O)N(CC)[C@@H](C)CC(=O)O ZINC000147248017 CG For-Sale Mild ASAH1 90 37 CCCCCCCCNC(=O)N(CC)[C@@H](C)CC(=O)O ZINC000147248017 CG For-Sale Mild NOD1 74 40 CCCCCCCCNC(=O)N(CC)[C@@H](C)CC(=O)O ZINC000147248017 CG For-Sale Mild OXER1 47 31 O=C(O)[C@H]1CCCN(C(=O)c2cccc3c2OCCN3)C1 ZINC000147248028 CD For-Sale Anodyne SLC6A1 130 37 OC[C@@H]1O[C@H](Oc2ccc(/C=C\c3cc(O)cc(O)c3)cc2)[C@@H](O)[C@H](O)[C@H]1O ZINC000147248060 GC For-Sale Anodyne TYR 42 58 OC[C@@H]1O[C@H](Oc2ccc(/C=C\c3cc(O)cc(O)c3)cc2)[C@@H](O)[C@H](O)[C@H]1O ZINC000147248060 GC For-Sale Anodyne IL2 38 43 OC[C@@H]1O[C@H](Oc2ccc(/C=C\c3cc(O)cc(O)c3)cc2)[C@@H](O)[C@H](O)[C@H]1O ZINC000147248060 GC For-Sale Anodyne GGTA1 0 40 OC[C@@H]1O[C@H](Oc2ccc(/C=C\c3cc(O)cc(O)c3)cc2)[C@@H](O)[C@H](O)[C@H]1O ZINC000147248060 GC For-Sale Anodyne CA12 0 50 OC[C@@H]1O[C@H](Oc2ccc(/C=C\c3cc(O)cc(O)c3)cc2)[C@@H](O)[C@H](O)[C@H]1O ZINC000147248060 GC For-Sale Anodyne B4GALT1 0 42 OC[C@@H]1O[C@H](Oc2ccc(/C=C\c3cc(O)cc(O)c3)cc2)[C@@H](O)[C@H](O)[C@H]1O ZINC000147248060 GC For-Sale Anodyne SLC5A1 73 45 OC[C@@H]1O[C@H](Oc2ccc(/C=C\c3cc(O)cc(O)c3)cc2)[C@@H](O)[C@H](O)[C@H]1O ZINC000147248060 GC For-Sale Anodyne SLC5A2 65 45 OC[C@@H]1O[C@H](Oc2ccc(/C=C\c3cc(O)cc(O)c3)cc2)[C@@H](O)[C@H](O)[C@H]1O ZINC000147248060 GC For-Sale Anodyne FIMH 108 60 OC[C@@H]1O[C@H](Oc2ccc(/C=C\c3cc(O)cc(O)c3)cc2)[C@@H](O)[C@H](O)[C@H]1O ZINC000147248060 GC For-Sale Anodyne IMA1 0 44 OC[C@@H]1O[C@H](Oc2ccc(/C=C\c3cc(O)cc(O)c3)cc2)[C@@H](O)[C@H](O)[C@H]1O ZINC000147248060 GC For-Sale Anodyne SLC28A3 0 43 OC[C@@H]1O[C@H](Oc2ccc(/C=C\c3cc(O)cc(O)c3)cc2)[C@@H](O)[C@H](O)[C@H]1O ZINC000147248060 GC For-Sale Anodyne SLC5A4 20 45 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147248084 FD On-Demand Anodyne NPY2R 16 43 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147248084 FD On-Demand Anodyne L3MBTL3 60 41 CC(C)[C@@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147248090 EF On-Demand Mild CCR1 66 52 CC(C)[C@@H](NC(=O)c1ccccc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147248090 EF On-Demand Mild JAK3 41 34 CC(=O)Nc1ccc2sc(Cl)nc2c1 ZINC000147248146 BF For-Sale Anodyne AGPAT2 49 49 CC(=O)Nc1ccc2sc(Cl)nc2c1 ZINC000147248146 BF For-Sale Anodyne P95276_MYCTO 0 41 CC(=O)Nc1ccc2sc(Cl)nc2c1 ZINC000147248146 BF For-Sale Anodyne PPX1 0 40 O=C(O)[C@@H]1CCCN(C(=O)c2cccc3c2OCCN3)C1 ZINC000147248167 CD For-Sale Anodyne SLC6A1 130 37 CCCCCCCCNC(=O)N(CC)[C@H](C)CC(=O)O ZINC000147248169 CG For-Sale Mild CPT1A 46 47 CCCCCCCCNC(=O)N(CC)[C@H](C)CC(=O)O ZINC000147248169 CG For-Sale Mild EPHX2 26 43 CCCCCCCCNC(=O)N(CC)[C@H](C)CC(=O)O ZINC000147248169 CG For-Sale Mild ASAH1 90 37 CCCCCCCCNC(=O)N(CC)[C@H](C)CC(=O)O ZINC000147248169 CG For-Sale Mild NOD1 74 40 CCCCCCCCNC(=O)N(CC)[C@H](C)CC(=O)O ZINC000147248169 CG For-Sale Mild OXER1 47 31 O=C(N[C@@H](Cc1ccc(O)cc1)c1nc2ccccc2[nH]1)c1ccc2c(c1)COC2 ZINC000147248227 GI On-Demand Anodyne F11 42 43 O=C(N[C@@H](Cc1ccc(O)cc1)c1nc2ccccc2[nH]1)c1ccc2c(c1)COC2 ZINC000147248227 GI On-Demand Anodyne PTPN1 41 51 O=C(N[C@@H](Cc1ccc(O)cc1)c1nc2ccccc2[nH]1)c1ccc2c(c1)COC2 ZINC000147248227 GI On-Demand Anodyne PIN1 32 43 CC[C@@H]1CN(C(=O)CCOc2ccccc2)CC[C@@H]1N ZINC000147248242 CE On-Demand Anodyne LTA4H 33 40 CC[C@@H]1CN(C(=O)CCOc2ccccc2)CC[C@@H]1N ZINC000147248242 CE On-Demand Anodyne COLA 79 40 CC[C@@H]1CN(C(=O)CCOc2ccccc2)CC[C@@H]1N ZINC000147248242 CE On-Demand Anodyne CPT1A 69 36 CC[C@@H]1CN(C(=O)CCOc2ccccc2)CC[C@@H]1N ZINC000147248242 CE On-Demand Anodyne PLA2G4B 43 32 COc1ccc(O)c(C(=O)N2CCC[C@H](CCBr)C2)c1 ZINC000147248246 EG For-Sale Reactive GRM3 16 48 C[C@@H]1CCCN(Cc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)C1 ZINC000147248286 FF On-Demand Anodyne PDE8B 16 41 CN(C)C(=O)Nc1cccc(C(=O)c2ccccc2)c1 ZINC000147248296 CG For-Sale Anodyne AKR1C3 32 45 CN(C)C(=O)Nc1cccc(C(=O)c2ccccc2)c1 ZINC000147248296 CG For-Sale Anodyne KCNK3 128 50 CN(C)C(=O)Nc1cccc(C(=O)c2ccccc2)c1 ZINC000147248296 CG For-Sale Anodyne KCNK9 84 45 CC(C)CCCCNC(=O)c1c[nH]c2ccc(N)cc12 ZINC000147248311 CG For-Sale Anodyne TPR 18 40 CC(C)CCCCNC(=O)c1c[nH]c2ccc(N)cc12 ZINC000147248311 CG For-Sale Anodyne KISS1R 63 36 O=C(O)[C@H]1CCCCN1C(=O)c1cccc2c1OCCN2 ZINC000147248369 CD For-Sale Anodyne ACE 41 38 O=C(O)[C@H]1CCCCN1C(=O)c1cccc2c1OCCN2 ZINC000147248369 CD For-Sale Anodyne PREP 60 42 CN(Cc1cscn1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147248371 FI On-Demand Anodyne BMP1 42 34 CN(Cc1cscn1)C(=O)NCC(c1ccccc1)c1ccccc1 ZINC000147248371 FI On-Demand Anodyne CYP3A4 15 43 Cc1cc(C(=O)Nc2ccc(C(=O)N(C)C)cc2)cc([N+](=O)[O-])c1 ZINC000147248379 EF On-Demand Bother EXSA 0 43 Cc1cc(C(=O)Nc2ccc(C(=O)N(C)C)cc2)cc([N+](=O)[O-])c1 ZINC000147248379 EF On-Demand Bother PSBA 0 48 Cc1cc(C(=O)Nc2ccc(C(=O)N(C)C)cc2)cc([N+](=O)[O-])c1 ZINC000147248379 EF On-Demand Bother KCNK3 41 37 CCCCCCCCNC(=O)NC1(CC(=O)O)CCCC1 ZINC000147248384 CG For-Sale Mild CPT1A 36 45 CCCCCCCCNC(=O)NC1(CC(=O)O)CCCC1 ZINC000147248384 CG For-Sale Mild EPHX2 35 50 CCCCCCCCNC(=O)NC1(CC(=O)O)CCCC1 ZINC000147248384 CG For-Sale Mild ASAH1 52 30 CC[C@H]1CN(C(=O)CCOc2ccccc2)CC[C@@H]1N ZINC000147248399 CE On-Demand Anodyne LTA4H 33 40 CC[C@H]1CN(C(=O)CCOc2ccccc2)CC[C@@H]1N ZINC000147248399 CE On-Demand Anodyne COLA 79 40 CC[C@H]1CN(C(=O)CCOc2ccccc2)CC[C@@H]1N ZINC000147248399 CE On-Demand Anodyne CPT1A 69 36 CC[C@H]1CN(C(=O)CCOc2ccccc2)CC[C@@H]1N ZINC000147248399 CE On-Demand Anodyne PLA2G4B 43 32 CCOC[C@H](C)NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147248410 DD On-Demand Anodyne MTOR 58 41 CCOC[C@H](C)NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147248410 DD On-Demand Anodyne DGAT1 59 47 C[C@H]1CCCN(Cc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)C1 ZINC000147248413 FF On-Demand Anodyne PDE8B 16 41 COc1ccc(O)c(C(=O)N2CCC[C@@H](CCBr)C2)c1 ZINC000147248424 EG For-Sale Reactive GRM3 16 48 CC[C@@H]1CCCCN1c1ccc(-c2nc(-c3ccc4c(c3)CN(CC(=O)OC(C)(C)C)CC4)no2)cc1COC ZINC000147248434 KK For-Sale Anodyne CPT1A 59 37 CC[C@@H]1CCCCN1c1ccc(-c2nc(-c3ccc4c(c3)CN(CC(=O)OC(C)(C)C)CC4)no2)cc1COC ZINC000147248434 KK For-Sale Anodyne S1PR1 25 40 O=C(NNC(=O)c1ccc(-n2cnnn2)cc1)Nc1nc2c(s1)CCCCC2 ZINC000147248499 GD On-Demand Reactive SLC27A1 32 43 CCCOCC(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147248509 DE On-Demand Anodyne DRD4 15 42 CCCOCC(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147248509 DE On-Demand Anodyne HRH3 20 46 CCCOCC(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147248509 DE On-Demand Anodyne SIGMAR1 17 43 CCCOCC(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147248509 DE On-Demand Anodyne MMP13 19 40 CCCOCC(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147248509 DE On-Demand Anodyne ADAM17 16 42 CCCOCC(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147248509 DE On-Demand Anodyne MMP9 20 42 CCCOCC(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147248509 DE On-Demand Anodyne MMP1 19 40 O=C(O)[C@@H]1CCCCN1C(=O)c1cccc2c1OCCN2 ZINC000147248530 CD For-Sale Anodyne ACE 41 38 O=C(O)[C@@H]1CCCCN1C(=O)c1cccc2c1OCCN2 ZINC000147248530 CD For-Sale Anodyne PREP 60 42 CC[C@@H]1CN(C(=O)CCOc2ccccc2)CC[C@H]1N ZINC000147248542 CE On-Demand Anodyne LTA4H 33 40 CC[C@@H]1CN(C(=O)CCOc2ccccc2)CC[C@H]1N ZINC000147248542 CE On-Demand Anodyne COLA 79 40 CC[C@@H]1CN(C(=O)CCOc2ccccc2)CC[C@H]1N ZINC000147248542 CE On-Demand Anodyne CPT1A 69 36 CC[C@@H]1CN(C(=O)CCOc2ccccc2)CC[C@H]1N ZINC000147248542 CE On-Demand Anodyne PLA2G4B 43 32 COc1cccc(CNC2(C(=O)O)CCC2)n1 ZINC000147248564 BD On-Demand Anodyne NPPA 40 32 COc1cccc(CNC2(C(=O)O)CCC2)n1 ZINC000147248564 BD On-Demand Anodyne ALS 61 31 Fc1cc(Oc2ccc(CCl)cc2Cl)ccc1Cl ZINC000147248574 DK For-Sale Reactive TTR 0 50 Fc1cc(Oc2ccc(CCl)cc2Cl)ccc1Cl ZINC000147248574 DK For-Sale Reactive FFAR1 0 40 CCCCCCCCNC(=O)NC(C)(C)C(C)(C)C(=O)O ZINC000147248582 DH For-Sale Mild CPT1A 0 42 CCCCCCCCNC(=O)NC(C)(C)C(C)(C)C(=O)O ZINC000147248582 DH For-Sale Mild EPHX2 24 46 CCCCCCCCNC(=O)NC(C)(C)C(C)(C)C(=O)O ZINC000147248582 DH For-Sale Mild ASAH1 79 33 Cc1ccc(Br)c(C(=O)Nc2cccc(S(C)(=O)=O)c2)c1 ZINC000147248590 FG On-Demand Anodyne F2R 0 61 Cc1ccc(Br)c(C(=O)Nc2cccc(S(C)(=O)=O)c2)c1 ZINC000147248590 FG On-Demand Anodyne CA4 17 43 Cc1ccc(Br)c(C(=O)Nc2cccc(S(C)(=O)=O)c2)c1 ZINC000147248590 FG On-Demand Anodyne F12 0 44 Cc1ccc(Br)c(C(=O)Nc2cccc(S(C)(=O)=O)c2)c1 ZINC000147248590 FG On-Demand Anodyne IDO1 18 42 Cc1ccc(Br)c(C(=O)Nc2cccc(S(C)(=O)=O)c2)c1 ZINC000147248590 FG On-Demand Anodyne PSBA 0 40 Cc1ccc(Br)c(C(=O)Nc2cccc(S(C)(=O)=O)c2)c1 ZINC000147248590 FG On-Demand Anodyne KCNK3 88 43 Cc1ccc(Br)c(C(=O)Nc2cccc(S(C)(=O)=O)c2)c1 ZINC000147248590 FG On-Demand Anodyne KCNK9 90 43 Cc1cc(C(=O)Nc2cc(Cl)ccc2N2CCN(C)CC2)cc([N+](=O)[O-])c1 ZINC000147248591 GH On-Demand Bother CNR1 51 33 Cc1cc(C(=O)Nc2cc(Cl)ccc2N2CCN(C)CC2)cc([N+](=O)[O-])c1 ZINC000147248591 GH On-Demand Bother DRD1 53 37 Cc1cc(C(=O)Nc2cc(Cl)ccc2N2CCN(C)CC2)cc([N+](=O)[O-])c1 ZINC000147248591 GH On-Demand Bother CNR2 15 43 Cc1cc(C(=O)Nc2cc(Cl)ccc2N2CCN(C)CC2)cc([N+](=O)[O-])c1 ZINC000147248591 GH On-Demand Bother CXCR3 19 40 Cc1cc(C(=O)Nc2cc(Cl)ccc2N2CCN(C)CC2)cc([N+](=O)[O-])c1 ZINC000147248591 GH On-Demand Bother WDR5 55 65 CC[C@H]1CCCCN1c1ccc(-c2nc(-c3ccc4c(c3)CN(CC(=O)OC(C)(C)C)CC4)no2)cc1COC ZINC000147248609 KK For-Sale Anodyne CPT1A 59 37 CC[C@H]1CCCCN1c1ccc(-c2nc(-c3ccc4c(c3)CN(CC(=O)OC(C)(C)C)CC4)no2)cc1COC ZINC000147248609 KK For-Sale Anodyne S1PR1 25 40 Cc1ccc(CCC(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147248627 EH For-Sale Reactive HRH3 0 42 Cc1cc(Cl)ccc1Oc1nc(N)nc(Cl)n1 ZINC000147248647 CF For-Sale Anodyne AGPAT2 44 35 CC[C@H]1CN(C(=O)CCOc2ccccc2)CC[C@H]1N ZINC000147248654 CE On-Demand Anodyne LTA4H 33 40 CC[C@H]1CN(C(=O)CCOc2ccccc2)CC[C@H]1N ZINC000147248654 CE On-Demand Anodyne COLA 79 40 CC[C@H]1CN(C(=O)CCOc2ccccc2)CC[C@H]1N ZINC000147248654 CE On-Demand Anodyne CPT1A 69 36 CC[C@H]1CN(C(=O)CCOc2ccccc2)CC[C@H]1N ZINC000147248654 CE On-Demand Anodyne PLA2G4B 43 32 CC[C@@H](C)[C@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147248720 CD For-Sale Anodyne ACE2 40 31 CCCCCCCCNC(=O)NCC(CC)(CC)C(=O)O ZINC000147248722 DH For-Sale Mild CPT1A 0 42 CCCCCCCCNC(=O)NCC(CC)(CC)C(=O)O ZINC000147248722 DH For-Sale Mild EPHX2 51 49 CCCCCCCCNC(=O)NCC(CC)(CC)C(=O)O ZINC000147248722 DH For-Sale Mild ASAH1 79 33 Cc1cc(CNC2(C(=O)O)CCC2)c2ccccc2n1 ZINC000147248775 CF For-Sale Anodyne ADAM17 93 44 Cc1cc(CNC2(C(=O)O)CCC2)c2ccccc2n1 ZINC000147248775 CF For-Sale Anodyne METG 43 32 Cc1cc(CNC2(C(=O)O)CCC2)c2ccccc2n1 ZINC000147248775 CF For-Sale Anodyne ADAMTS1 0 40 Cc1cc(CNC2(C(=O)O)CCC2)c2ccccc2n1 ZINC000147248775 CF For-Sale Anodyne ADAM33 0 41 Cc1ccc(CCC(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147248801 EH For-Sale Reactive HRH3 0 42 CCOC(=O)CC(=O)COc1ccc(Cl)c(F)c1 ZINC000147248839 CE For-Sale Anodyne PLA2G4B 58 34 CC[C@H](C)[C@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147248878 CD For-Sale Anodyne ACE2 40 31 CCCCCCCCNC(=O)N1CCC[C@@H]1C(=O)O ZINC000147248879 CF For-Sale Mild ACE 60 50 CCCCCCCCNC(=O)N1CCC[C@@H]1C(=O)O ZINC000147248879 CF For-Sale Mild TPP2 58 54 CCCCCCCCNC(=O)N1CCC[C@@H]1C(=O)O ZINC000147248879 CF For-Sale Mild GNAI1 0 41 CCCCCCCCNC(=O)N1CCC[C@@H]1C(=O)O ZINC000147248879 CF For-Sale Mild GNAI3 0 41 CCCCCCCCNC(=O)N1CCC[C@@H]1C(=O)O ZINC000147248879 CF For-Sale Mild GNAO1 0 41 CCCCCCCCNC(=O)N1CCC[C@@H]1C(=O)O ZINC000147248879 CF For-Sale Mild ASAH1 106 44 CCCCCCCCNC(=O)N1CCC[C@@H]1C(=O)O ZINC000147248879 CF For-Sale Mild DAPE 0 43 O=C(O)CN(CC1CC1)C(=O)c1cccc(F)c1Cl ZINC000147248941 CE On-Demand Anodyne ACE 43 37 CNc1cc(Oc2ccc(Cl)cc2C)cc([N+](=O)[O-])c1 ZINC000147248952 CI For-Sale Bother PPOX1 16 48 CC[C@@H](C)[C@@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147249004 CD For-Sale Anodyne ACE2 40 31 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc(S(=O)(=O)N(C)C)cc1 ZINC000147249013 HH On-Demand Anodyne MDM2 87 35 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249021 GD On-Demand Anodyne F2 21 40 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249021 GD On-Demand Anodyne P2RY12 197 39 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249021 GD On-Demand Anodyne HRH3 24 41 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249021 GD On-Demand Anodyne MMP13 22 42 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249021 GD On-Demand Anodyne TRY2_BOVIN 67 34 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249021 GD On-Demand Anodyne CACNA1B 19 40 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249021 GD On-Demand Anodyne ADAM17 17 42 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249021 GD On-Demand Anodyne MMP9 21 42 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249021 GD On-Demand Anodyne DPP7 45 45 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249021 GD On-Demand Anodyne CACNA1G 16 42 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249021 GD On-Demand Anodyne PROKR1 58 32 CCCOc1nc(N)nc(Oc2ccc(Cl)cc2C)n1 ZINC000147249142 CF For-Sale Anodyne FOLA 15 40 CCCOc1nc(N)nc(Oc2ccc(Cl)cc2C)n1 ZINC000147249142 CF For-Sale Anodyne AGPAT2 43 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249145 GD On-Demand Anodyne F2 21 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249145 GD On-Demand Anodyne P2RY12 197 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249145 GD On-Demand Anodyne HRH3 24 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249145 GD On-Demand Anodyne MMP13 22 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249145 GD On-Demand Anodyne TRY2_BOVIN 67 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249145 GD On-Demand Anodyne CACNA1B 19 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249145 GD On-Demand Anodyne ADAM17 17 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249145 GD On-Demand Anodyne MMP9 21 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249145 GD On-Demand Anodyne DPP7 45 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249145 GD On-Demand Anodyne CACNA1G 16 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(OC)cc2)CC1 ZINC000147249145 GD On-Demand Anodyne PROKR1 58 32 CC[C@H](C)[C@@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147249155 CD For-Sale Anodyne ACE2 40 31 O=C(O)CN(CC1CC1)C(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147249168 CE For-Sale Anodyne GPR88 0 46 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild F2 39 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild PLG 42 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild ACE 64 51 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild GHRHR 53 32 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild P2RY12 145 33 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild MME 82 46 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild MC4R 79 46 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CTRA_BOVIN 31 49 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CTSB 57 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild TRY2_BOVIN 95 39 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild PAPA1_CARPA 47 56 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CYSP_TRYCR 50 34 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CCKAR 51 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CTSF 46 37 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CTSL 44 45 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CCR1 33 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CCR3 15 49 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild NPFFR2 44 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CYP51A1 26 52 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild TIMP3 45 33 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild DPP4 26 42 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CTRB1 40 34 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild PREP 26 63 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild MC3R 41 36 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild MC5R 66 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CCKBR 94 44 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CTSS 33 50 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CAPN1 49 48 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild MMP9 17 41 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild ACE2 73 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CTSV 47 47 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild ST14 115 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild PIN1 15 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild CTRB_BOVIN 52 37 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild AMP1_PLAFQ 27 45 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild DPP8 22 44 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild BLA1_STEMA 64 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild BRCA1 54 36 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild NPFFR1 34 40 N#CC1CCN(C(=O)[C@H](Cc2ccccc2)NC(=O)c2ccccc2)CC1 ZINC000147249268 FF On-Demand Mild TMPRSS6 71 36 NC(=O)[C@@H]1CCC[C@@H]1NC(=O)c1ccc(N2CCCC2=O)cc1 ZINC000147249286 DD On-Demand Anodyne AKR1C3 22 44 CNc1ccc([N+](=O)[O-])c(Oc2ccc(Cl)cc2C)n1 ZINC000147249319 CH For-Sale Bother S1PR4 0 40 CNc1ccc([N+](=O)[O-])c(Oc2ccc(Cl)cc2C)n1 ZINC000147249319 CH For-Sale Bother ENR 0 40 O=C(O)CN(CC1CC1)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147249342 CE For-Sale Anodyne GPR88 0 46 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc(S(=O)(=O)N(C)C)cc1 ZINC000147249358 HH On-Demand Anodyne MDM2 87 35 CCCOc1cccc(C(=O)N2CCC[C@H](CCBr)C2)c1 ZINC000147249373 FI For-Sale Reactive HCRTR1 16 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1Cl ZINC000147249416 HG On-Demand Anodyne SSTR3 25 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1Cl ZINC000147249416 HG On-Demand Anodyne KCNK3 41 37 CCCCCCCCNC(=O)N[C@H](CC(=O)O)C(=O)O ZINC000147249437 CD For-Sale Mild FOLH1 64 49 CCCCCCCCNC(=O)N[C@H](CC(=O)O)C(=O)O ZINC000147249437 CD For-Sale Mild CPT1A 52 60 CCCCCCCCNC(=O)N[C@H](CC(=O)O)C(=O)O ZINC000147249437 CD For-Sale Mild ENPEP 42 31 CCCCCCCCNC(=O)N[C@H](CC(=O)O)C(=O)O ZINC000147249437 CD For-Sale Mild EPHX2 25 67 CCCCCCCCNC(=O)N[C@H](CC(=O)O)C(=O)O ZINC000147249437 CD For-Sale Mild Q6UB75_PIG 0 42 CCCCCCCCNC(=O)N[C@H](CC(=O)O)C(=O)O ZINC000147249437 CD For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N[C@H](CC(=O)O)C(=O)O ZINC000147249437 CD For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N[C@H](CC(=O)O)C(=O)O ZINC000147249437 CD For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N[C@H](CC(=O)O)C(=O)O ZINC000147249437 CD For-Sale Mild ASAH1 87 35 CCCCCCCCNC(=O)N[C@H](CC(=O)O)C(=O)O ZINC000147249437 CD For-Sale Mild NOD1 94 45 CCCCCCCCNC(=O)N[C@H](CC(=O)O)C(=O)O ZINC000147249437 CD For-Sale Mild CQSS 50 31 O=C(NCc1cccc(NC(=O)[C@@H]2CCCO2)c1)Nc1ccc(N2CCCC2)nc1 ZINC000147249469 HG On-Demand Anodyne DGAT1 44 41 O=C(NCc1cccc(NC(=O)[C@@H]2CCCO2)c1)Nc1ccc(N2CCCC2)nc1 ZINC000147249469 HG On-Demand Anodyne NAMPT 49 40 O=C(O)CN(CC1CC1)C(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147249517 CE For-Sale Anodyne GPR88 0 46 CC(C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147249522 DE On-Demand Mild ACE 16 40 CC(C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147249522 DE On-Demand Mild ELANE 60 43 CC(C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147249522 DE On-Demand Mild CTSB 20 40 CC(C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147249522 DE On-Demand Mild CCR1 59 63 CC(C)[C@H](NC(=O)c1ccccc1)C(=O)N1CCC(C#N)CC1 ZINC000147249522 DE On-Demand Mild PREP 17 48 CCCOc1cccc(C(=O)N2CCC[C@@H](CCBr)C2)c1 ZINC000147249523 FI For-Sale Reactive HCRTR1 16 41 Cc1cc(C(=O)NCC(=O)Nc2ccc(F)c(F)c2F)cc([N+](=O)[O-])c1 ZINC000147249559 FF On-Demand Bother METC 0 51 Cc1cc(Cl)ccc1Oc1nc(N)ncc1Br ZINC000147249563 DH For-Sale Anodyne AGPAT2 42 36 Cc1cc(Cl)ccc1Oc1nc(N)ncc1Br ZINC000147249563 DH For-Sale Anodyne MAP3K14 40 40 Cc1ccc(OCc2ccc(Cl)cc2C(=O)O)cc1 ZINC000147249569 CH For-Sale Anodyne PPARG 15 43 Cc1ccc(OCc2ccc(Cl)cc2C(=O)O)cc1 ZINC000147249569 CH For-Sale Anodyne OPRL1 17 41 Cc1ccc(OCc2ccc(Cl)cc2C(=O)O)cc1 ZINC000147249569 CH For-Sale Anodyne PTGER1 65 43 Cc1ccc(OCc2ccc(Cl)cc2C(=O)O)cc1 ZINC000147249569 CH For-Sale Anodyne PTGER4 40 54 Cc1ccc(OCc2ccc(Cl)cc2C(=O)O)cc1 ZINC000147249569 CH For-Sale Anodyne PTGER3 47 42 Cc1ccc(OCc2ccc(Cl)cc2C(=O)O)cc1 ZINC000147249569 CH For-Sale Anodyne GYS1 62 34 Cc1ccc(OCc2ccc(Cl)cc2C(=O)O)cc1 ZINC000147249569 CH For-Sale Anodyne NS5B 23 44 Cc1ccc(OCc2ccc(Cl)cc2C(=O)O)cc1 ZINC000147249569 CH For-Sale Anodyne PTGDR2 20 40 Cc1ccc(OCc2ccc(Cl)cc2C(=O)O)cc1 ZINC000147249569 CH For-Sale Anodyne FFAR1 43 58 Cc1ccc(OCc2ccc(Cl)cc2C(=O)O)cc1 ZINC000147249569 CH For-Sale Anodyne FFAR4 54 58 Cc1ccc(OCc2ccc(Cl)cc2C(=O)O)cc1 ZINC000147249569 CH For-Sale Anodyne AKR1C2 41 39 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1Cl ZINC000147249580 HG On-Demand Anodyne SSTR3 25 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1Cl ZINC000147249580 HG On-Demand Anodyne KCNK3 41 37 C=CCN(CC(=O)O)C(=O)NCCCCCCCC ZINC000147249598 CF For-Sale Mild EPHX2 25 44 C=CCN(CC(=O)O)C(=O)NCCCCCCCC ZINC000147249598 CF For-Sale Mild ASAH1 51 32 O=C(O)CN(CC1CC1)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147249599 CE For-Sale Anodyne GPR88 0 46 O=C(NCc1cccc(NC(=O)[C@H]2CCCO2)c1)Nc1ccc(N2CCCC2)nc1 ZINC000147249626 HG On-Demand Anodyne DGAT1 44 41 O=C(NCc1cccc(NC(=O)[C@H]2CCCO2)c1)Nc1ccc(N2CCCC2)nc1 ZINC000147249626 HG On-Demand Anodyne NAMPT 49 40 COc1cccc(F)c1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147249688 EG For-Sale Reactive CCR3 19 40 COc1cccc(F)c1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147249688 EG For-Sale Reactive ACKR3 59 34 COc1ccc(CNc2cc(NN)nc(C(C)C)n2)cc1 ZINC000147249702 CF For-Sale Anodyne PROKR1 43 32 CCCCCCCCCCCCCCCCOC[C@@H](CO)O[C@@H]1OC[C@@H](O)[C@@H](O)[C@@H]1O ZINC000147249736 IG Annotated Mild PTAFR 43 33 CCCCCCCCCCCCCCCCOC[C@@H](CO)O[C@@H]1OC[C@@H](O)[C@@H](O)[C@@H]1O ZINC000147249736 IG Annotated Mild UGCG 15 40 CCCCCCCCCCCCCCCCOC[C@@H](CO)O[C@@H]1OC[C@@H](O)[C@@H](O)[C@@H]1O ZINC000147249736 IG Annotated Mild GBA2 55 40 CCCCCCCCCCCCCCCCOC[C@@H](CO)O[C@@H]1OC[C@@H](O)[C@@H](O)[C@@H]1O ZINC000147249736 IG Annotated Mild SIS 0 40 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249762 GF On-Demand Anodyne DRD4 17 42 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249762 GF On-Demand Anodyne GHRHR 40 32 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249762 GF On-Demand Anodyne P2RY12 167 35 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249762 GF On-Demand Anodyne MC4R 108 41 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249762 GF On-Demand Anodyne TRY2_BOVIN 44 32 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249762 GF On-Demand Anodyne CCR1 44 42 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249762 GF On-Demand Anodyne MC5R 49 37 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249762 GF On-Demand Anodyne LSS 19 41 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249762 GF On-Demand Anodyne CCKBR 17 41 CCCC[C@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249762 GF On-Demand Anodyne DPP7 63 44 CCCCCCCCNC(=O)N[C@@H]1CCC[C@H](C(=O)O)C1 ZINC000147249771 CG For-Sale Mild EPHX2 40 69 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147249786 GF On-Demand Anodyne MAPK14 48 48 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147249786 GF On-Demand Anodyne KCNK3 77 37 Cc1ccc(C(=O)N(CC(=O)O)CC2CC2)cc1Br ZINC000147249819 EF On-Demand Anodyne OXTR 23 47 N#Cc1ccc(Nc2nc(NN)cn3ccnc23)c(F)c1 ZINC000147249836 CD For-Sale Mild HIVRT 0 48 COc1cccc(F)c1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147249842 EG For-Sale Reactive CCR3 19 40 COc1cccc(F)c1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147249842 EG For-Sale Reactive ACKR3 59 34 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne ACE 101 85 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne FKBP1A 47 38 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne MME 30 51 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne CTRA_BOVIN 41 32 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne CTSB 41 35 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne CYSP_TRYCR 45 40 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne PREP 21 40 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne CAPNS1 53 34 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne CELA2A 40 32 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne REN 17 47 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne CAPN1 54 36 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne CAPN2 93 38 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne ACE2 15 47 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne NPR 45 36 CCOC(=O)[C@H](CCc1ccccc1)N[C@@H](C)C(=O)N1[C@H]2CCCC[C@H]2C[C@@H]1C(=O)OCc1ccccc1 ZINC000147249881 KI For-Sale Anodyne BIRC2 45 38 COc1ccc(CNc2cc(NN)nc(C3CC3)n2)cc1 ZINC000147249907 CE For-Sale Anodyne PTGDR 32 45 CCCCCCCCCCCCCCCCOC[C@@H](COC(C)=O)O[C@@H]1OC[C@@H](O)[C@@H](O)[C@@H]1O ZINC000147249941 JH Annotated Mild PTAFR 62 39 CCCCCCCCCCCCCCCCOC[C@@H](COC(C)=O)O[C@@H]1OC[C@@H](O)[C@@H](O)[C@@H]1O ZINC000147249941 JH Annotated Mild GBA2 51 37 CC[C@@H]1CN(C(=O)c2ccc(C)c(C)c2)CC[C@@H]1N ZINC000147249949 CF On-Demand Anodyne L3MBTL3 74 38 Cc1ccc(C(=O)NNC(=O)N[C@@H](C)c2ccc3c(c2)OCCO3)s1 ZINC000147249955 FF On-Demand Reactive KCNQ2 21 40 CCCCCCCCNC(=O)N[C@H]1CCC[C@H](C(=O)O)C1 ZINC000147249967 CG For-Sale Mild EPHX2 40 69 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249971 GF On-Demand Anodyne DRD4 17 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249971 GF On-Demand Anodyne GHRHR 40 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249971 GF On-Demand Anodyne P2RY12 167 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249971 GF On-Demand Anodyne MC4R 108 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249971 GF On-Demand Anodyne TRY2_BOVIN 44 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249971 GF On-Demand Anodyne CCR1 44 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249971 GF On-Demand Anodyne MC5R 49 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249971 GF On-Demand Anodyne LSS 19 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249971 GF On-Demand Anodyne CCKBR 17 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147249971 GF On-Demand Anodyne DPP7 63 44 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147249973 GF On-Demand Anodyne MAPK14 48 48 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147249973 GF On-Demand Anodyne KCNK3 77 37 Cc1c[nH]c(=O)c2cccc(N)c12 ZINC000147249991 AD For-Sale Anodyne PARP2 50 50 C[C@@H]1CCCN(c2ccc(C(=O)N3CCC(C#N)CC3)cc2[N+](=O)[O-])C1 ZINC000147250005 FG On-Demand Mild L3MBTL3 43 34 NS(=O)(=O)c1cc(F)ccc1OCCc1cccnc1 ZINC000147250038 CD For-Sale Anodyne CA14 24 41 NS(=O)(=O)c1cc(F)ccc1OCCc1cccnc1 ZINC000147250038 CD For-Sale Anodyne ISPH 0 41 CC(C)c1nc(NN)cc(NC2CCCCCCC2)n1 ZINC000147250101 CG For-Sale Anodyne HRH4 17 40 CC(C)c1nc(NN)cc(NC2CCCCCCC2)n1 ZINC000147250101 CG For-Sale Anodyne PRKD1 52 34 COc1ccc(S(=O)(=O)NCC(F)F)c(CC(=O)O)c1 ZINC000147250129 DC On-Demand Anodyne MMP13 25 42 COc1ccc(S(=O)(=O)NCC(F)F)c(CC(=O)O)c1 ZINC000147250129 DC On-Demand Anodyne MMP16 0 42 COc1ccc(S(=O)(=O)NCC(F)F)c(CC(=O)O)c1 ZINC000147250129 DC On-Demand Anodyne MTNR1A 49 37 COc1ccc(S(=O)(=O)NCC(F)F)c(CC(=O)O)c1 ZINC000147250129 DC On-Demand Anodyne MMP9 17 43 CCCCCCCCCCCCCCCCCCOC[C@@H](CO)O[C@@H]1OC[C@@H](O)[C@@H](O)[C@@H]1O ZINC000147250145 JI Annotated Mild PTAFR 43 33 CCCCCCCCCCCCCCCCCCOC[C@@H](CO)O[C@@H]1OC[C@@H](O)[C@@H](O)[C@@H]1O ZINC000147250145 JI Annotated Mild UGCG 15 40 CCCCCCCCCCCCCCCCCCOC[C@@H](CO)O[C@@H]1OC[C@@H](O)[C@@H](O)[C@@H]1O ZINC000147250145 JI Annotated Mild GBA2 55 40 CCCCCCCCCCCCCCCCCCOC[C@@H](CO)O[C@@H]1OC[C@@H](O)[C@@H](O)[C@@H]1O ZINC000147250145 JI Annotated Mild SIS 0 40 Cc1ccc(C(=O)NNC(=O)N[C@H](C)c2ccc3c(c2)OCCO3)s1 ZINC000147250147 FF On-Demand Reactive KCNQ2 21 40 CC[C@H]1CN(C(=O)c2ccc(C)c(C)c2)CC[C@@H]1N ZINC000147250170 CF On-Demand Anodyne L3MBTL3 74 38 CCCCCCCCNC(=O)N[C@@H]1CCC[C@@H](C(=O)O)C1 ZINC000147250176 CG For-Sale Mild EPHX2 40 69 CCCNC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147250183 ED On-Demand Anodyne KCNK3 57 35 C[C@H]1CCCN(c2ccc(C(=O)N3CCC(C#N)CC3)cc2[N+](=O)[O-])C1 ZINC000147250198 FG On-Demand Mild L3MBTL3 43 34 Cc1nn(C(F)F)c(C)c1CC(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147250227 HH On-Demand Anodyne LSS 19 40 CCOc1cc(CNCC(=O)Nc2ccc(F)cc2)ccc1O[C@@H](C)C(=O)N(C)C ZINC000147250274 HF On-Demand Anodyne LEF 45 35 CCOc1cc(CNCC(=O)Nc2ccc(F)cc2)ccc1O[C@@H](C)C(=O)N(C)C ZINC000147250274 HF On-Demand Anodyne NR5A1 24 40 CC(=O)N1c2ccc(-c3ccc(C(=O)O)cc3)cc2[C@H](Nc2ccccc2)C[C@@H]1C ZINC000147250275 HK Annotated Anodyne ECR 36 58 NNc1cc(NC2CCCCCCC2)nc(C2CC2)n1 ZINC000147250294 CG For-Sale Anodyne HRH4 16 40 NNc1cc(NC2CCCCCCC2)nc(C2CC2)n1 ZINC000147250294 CG For-Sale Anodyne PRKD1 50 33 CC[C@@H]1CN(C(=O)c2ccc(C)c(C)c2)CC[C@H]1N ZINC000147250369 CF On-Demand Anodyne L3MBTL3 74 38 Cc1cc(Cl)ccc1Oc1nc(N)nc(N2CCCC2)n1 ZINC000147250374 DF For-Sale Anodyne HRH4 23 42 CCCCCCCCNC(=O)N[C@H]1CCC[C@@H](C(=O)O)C1 ZINC000147250382 CG For-Sale Mild EPHX2 40 69 CCCNC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147250400 ED On-Demand Anodyne KCNK3 57 35 CCOc1ccc(C(=O)COc2ccc(Cl)c(F)c2)cc1 ZINC000147250408 DI For-Sale Anodyne PLA2G4B 71 35 CC(C)(C)c1nc(NN)cc(NC2CCCCCCC2)n1 ZINC000147250474 CH For-Sale Anodyne HRH4 17 40 CC(C)(C)c1nc(NN)cc(NC2CCCCCCC2)n1 ZINC000147250474 CH For-Sale Anodyne PRKD1 55 33 O=C(NCc1ccc(F)cc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147250554 GG On-Demand Anodyne CA2 17 47 O=C(NCc1ccc(F)cc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147250554 GG On-Demand Anodyne MAP 0 46 O=C(NCc1ccc(F)cc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147250554 GG On-Demand Anodyne SCN3A 0 49 O=C(NCc1ccc(F)cc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147250554 GG On-Demand Anodyne MAP1 73 46 O=C(NCc1ccc(F)cc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147250554 GG On-Demand Anodyne SCN9A 0 47 O=C(NCc1ccc(F)cc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147250554 GG On-Demand Anodyne CYNT 18 42 O=C(NCc1ccc(F)cc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147250554 GG On-Demand Anodyne PFK 0 52 O=C(NCc1ccc(F)cc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147250554 GG On-Demand Anodyne NAMPT 72 45 CC[C@H]1CN(C(=O)c2ccc(C)c(C)c2)CC[C@H]1N ZINC000147250569 CF On-Demand Anodyne L3MBTL3 74 38 CN(C)NC(=O)CC[C@@H]1CCNC1 ZINC000147250579 AB For-Sale Reactive KDM7A 0 42 CCCCCCCCNC(=O)N(CCCC(=O)O)C(C)C ZINC000147250591 DH For-Sale Mild FABP2 0 46 CCCCCCCCNC(=O)N(CCCC(=O)O)C(C)C ZINC000147250591 DH For-Sale Mild PLA2G4A 0 48 CCCCCCCCNC(=O)N(CCCC(=O)O)C(C)C ZINC000147250591 DH For-Sale Mild EPHX2 28 53 CCCCCCCCNC(=O)N(CCCC(=O)O)C(C)C ZINC000147250591 DH For-Sale Mild Q6UB75_PIG 0 42 CCCCCCCCNC(=O)N(CCCC(=O)O)C(C)C ZINC000147250591 DH For-Sale Mild FABP5 15 46 CCCCCCCCNC(=O)N(CCCC(=O)O)C(C)C ZINC000147250591 DH For-Sale Mild ASAH1 95 35 CCCCCCCCNC(=O)N(CCCC(=O)O)C(C)C ZINC000147250591 DH For-Sale Mild SLC22A20 0 46 CCCCCCCCNC(=O)N(CCCC(=O)O)C(C)C ZINC000147250591 DH For-Sale Mild NOD1 69 39 CCCCCCCCNC(=O)N(CCCC(=O)O)C(C)C ZINC000147250591 DH For-Sale Mild CQSS 51 34 CCN(CC)c1nc(N)nc(Oc2ccc(Cl)cc2C)n1 ZINC000147250593 DG For-Sale Anodyne AGPAT2 43 36 Cc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250613 FJ On-Demand Mild DHODH 15 40 Cc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250613 FJ On-Demand Mild PRS 67 49 Cc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250613 FJ On-Demand Mild ACACB 24 42 Cc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250613 FJ On-Demand Mild PREP 16 50 Cc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250613 FJ On-Demand Mild TACR3 36 41 Cc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250613 FJ On-Demand Mild MT-CO2 56 48 CCCCCCCCNC(=O)N1C[C@H](OC)C[C@@H]1C(=O)O ZINC000147250776 DE For-Sale Mild ASAH1 102 40 CN(C)NC(=O)CC[C@H]1CCNC1 ZINC000147250779 AB For-Sale Reactive KDM7A 0 42 COc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250796 FI On-Demand Mild CCKAR 20 40 COc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250796 FI On-Demand Mild PRS 58 46 COc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250796 FI On-Demand Mild ACACB 22 42 COc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250796 FI On-Demand Mild TACR3 42 45 COc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250796 FI On-Demand Mild LUCI_PHOPY 17 54 COc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250796 FI On-Demand Mild MT-CO2 53 45 COc1ccc(-c2cc(C(=O)N3CCC(C#N)CC3)c3ccccc3n2)cc1 ZINC000147250796 FI On-Demand Mild VCP 18 41 CC(C)CCCCNC(=O)c1cc(N)n[nH]1 ZINC000147250807 BD For-Sale Anodyne ALPL 64 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCCC1 ZINC000147250902 FE On-Demand Anodyne KCNQ2 58 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCCC1 ZINC000147250902 FE On-Demand Anodyne HDAC10 41 33 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCCC1 ZINC000147250902 FE On-Demand Anodyne HDAC11 49 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCCC1 ZINC000147250902 FE On-Demand Anodyne DPP7 43 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCCC1 ZINC000147250902 FE On-Demand Anodyne NPSR1 16 45 CC(C)Cc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147250924 DE On-Demand Anodyne TBXA2R 49 37 CC(C)Cc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147250924 DE On-Demand Anodyne MMP9 21 41 CC(C)Cc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147250924 DE On-Demand Anodyne MMP10 15 41 CC(C)Cc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147250924 DE On-Demand Anodyne SLC22A20 0 42 O=C(NC1CCN(C(=O)Nc2ccc(N3CCCC3)nc2)CC1)c1ccoc1 ZINC000147250933 GF On-Demand Anodyne DGAT1 45 50 O=C(NC1CCN(C(=O)Nc2ccc(N3CCCC3)nc2)CC1)c1ccoc1 ZINC000147250933 GF On-Demand Anodyne HPGDS 33 52 C[C@@H]1CCN[C@H](C(=O)O)[C@H]1CC(=O)O ZINC000147250941 BC For-Sale Anodyne GRIK3 15 51 C[C@@H]1CCN[C@H](C(=O)O)[C@H]1CC(=O)O ZINC000147250941 BC For-Sale Anodyne GRIK2 101 50 CN(C)NC(=O)CCNC(C)(C)C ZINC000147250969 AC For-Sale Reactive KDM7A 0 52 CCCCCCCCNC(=O)N1C[C@@H](OC)C[C@@H]1C(=O)O ZINC000147251012 DE For-Sale Mild ASAH1 102 40 CCCC[C@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147251023 CD For-Sale Anodyne C3AR1 49 32 Cc1cc(Cl)ccc1Oc1nc(N)ncc1C ZINC000147251050 BG For-Sale Anodyne AGPAT2 48 35 Cc1cc(Cl)ccc1Oc1nc(N)ncc1C ZINC000147251050 BG For-Sale Anodyne MAP3K14 42 44 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1CCCCC1 ZINC000147251051 GF On-Demand Mild CNR2 23 74 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1CCCCC1 ZINC000147251051 GF On-Demand Mild EPHX2 32 43 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1CCCCC1 ZINC000147251051 GF On-Demand Mild L3MBTL3 87 43 CCCNC(=O)CN(CCC)C(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147251056 EE On-Demand Anodyne NQO2 36 42 CCCNC(=O)CN(CCC)C(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147251056 EE On-Demand Anodyne MTNR1A 52 38 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCOCC2)c1 ZINC000147251071 GC On-Demand Anodyne CASR 34 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCOCC2)c1 ZINC000147251071 GC On-Demand Anodyne NPY2R 16 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCOCC2)c1 ZINC000147251071 GC On-Demand Anodyne EPHX2 26 52 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCOCC2)c1 ZINC000147251071 GC On-Demand Anodyne TNK2 19 41 Cc1cc(NC(=O)C2(C)CC2)ccc1F ZINC000147251079 BF On-Demand Anodyne ENV 44 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCCC1 ZINC000147251119 FE On-Demand Anodyne KCNQ2 58 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCCC1 ZINC000147251119 FE On-Demand Anodyne HDAC10 41 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCCC1 ZINC000147251119 FE On-Demand Anodyne HDAC11 49 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCCC1 ZINC000147251119 FE On-Demand Anodyne DPP7 43 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCCC1 ZINC000147251119 FE On-Demand Anodyne NPSR1 16 45 CCCc1c(NN)ncnc1Nc1ccc(C#N)cc1F ZINC000147251130 CE For-Sale Mild FLT1 0 44 CC(C)Cc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147251136 DE On-Demand Anodyne TBXA2R 49 37 CC(C)Cc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147251136 DE On-Demand Anodyne MMP9 21 41 CC(C)Cc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147251136 DE On-Demand Anodyne MMP10 15 41 CC(C)Cc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147251136 DE On-Demand Anodyne SLC22A20 0 42 C[C@H]1CCN[C@H](C(=O)O)[C@H]1CC(=O)O ZINC000147251142 BC For-Sale Anodyne GRIK3 15 51 C[C@H]1CCN[C@H](C(=O)O)[C@H]1CC(=O)O ZINC000147251142 BC For-Sale Anodyne GRIK2 101 50 O=C(O)CN(C(=O)c1cccc(F)c1Cl)C1CC1 ZINC000147251146 CE In-Stock Anodyne ACE 74 55 O=C(O)CN(C(=O)c1cccc(F)c1Cl)C1CC1 ZINC000147251146 CE In-Stock Anodyne C5AR1 19 40 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(N3CCCC3)nc2)C1 ZINC000147251179 FD On-Demand Anodyne DGAT1 39 41 CN(C)NC(=O)c1ccc2c(c1)CNCC2 ZINC000147251184 BC For-Sale Reactive PNMT 31 44 CCCCCCCCNC(=O)N1C[C@H](OC)C[C@H]1C(=O)O ZINC000147251196 DE For-Sale Mild ASAH1 102 40 CCCC[C@@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147251206 CD For-Sale Anodyne C3AR1 49 32 O=C1S/C(=C/c2cc(-c3ccccc3)n(-c3ccc([N+](=O)[O-])cc3)c2-c2ccccc2)C(=O)N1c1ccccc1 ZINC000147251232 KK In-Stock Bother AKR1B1 22 42 O=C1S/C(=C/c2cc(-c3ccccc3)n(-c3ccc([N+](=O)[O-])cc3)c2-c2ccccc2)C(=O)N1c1ccccc1 ZINC000147251232 KK In-Stock Bother MDM2 25 46 CCCNC(=O)CN(CCC)C(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147251267 EE On-Demand Anodyne NQO2 36 42 CCCNC(=O)CN(CCC)C(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147251267 EE On-Demand Anodyne MTNR1A 52 38 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCOCC2)c1 ZINC000147251309 GC On-Demand Anodyne CASR 34 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCOCC2)c1 ZINC000147251309 GC On-Demand Anodyne NPY2R 16 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCOCC2)c1 ZINC000147251309 GC On-Demand Anodyne EPHX2 26 52 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(=O)N2CCOCC2)c1 ZINC000147251309 GC On-Demand Anodyne TNK2 19 41 C[C@H](CNS(=O)(=O)Cc1ccc(C#N)cc1)CC(=O)O ZINC000147251319 CD On-Demand Mild MMP12 0 48 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147251353 EE On-Demand Anodyne KCNQ2 59 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147251353 EE On-Demand Anodyne KLK3 41 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147251353 EE On-Demand Anodyne HDAC10 41 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147251353 EE On-Demand Anodyne HDAC11 42 34 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccc(N3CCCC3)nc2)C1 ZINC000147251369 FD On-Demand Anodyne DGAT1 39 41 O=C(O)CN(C(=O)[C@H]1C[C@H]1c1ccccc1)C1CC1 ZINC000147251395 CD For-Sale Anodyne ACE 56 44 O=C(O)CN(C(=O)[C@H]1C[C@H]1c1ccccc1)C1CC1 ZINC000147251395 CD For-Sale Anodyne GPR88 0 47 CCCCCCCCNC(=O)N1C[C@@H](OC)C[C@H]1C(=O)O ZINC000147251428 DE For-Sale Mild ASAH1 102 40 COc1ccc([N+](=O)[O-])c(C(=O)N2C[C@@H]3CCCN3Cc3ccccc32)c1 ZINC000147251430 FG On-Demand Bother AVPR2 37 45 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1CCOCC1 ZINC000147251495 GD On-Demand Mild CNR1 16 56 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1CCOCC1 ZINC000147251495 GD On-Demand Mild CNR2 22 68 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1CCOCC1 ZINC000147251495 GD On-Demand Mild NR1H4 17 40 Cc1ccc(C(=O)N2CCC(C#N)CC2)cc1S(=O)(=O)N1CCOCC1 ZINC000147251495 GD On-Demand Mild L3MBTL3 58 37 C[C@@H](CNS(=O)(=O)Cc1ccc(C#N)cc1)CC(=O)O ZINC000147251518 CD On-Demand Mild MMP12 0 48 CCNc1cc(Oc2ccc(Cl)cc2C)cc([N+](=O)[O-])c1 ZINC000147251530 DJ For-Sale Bother TBXA2R 15 40 CCNc1cc(Oc2ccc(Cl)cc2C)cc([N+](=O)[O-])c1 ZINC000147251530 DJ For-Sale Bother ENR 0 43 CCNc1cc(Oc2ccc(Cl)cc2C)cc([N+](=O)[O-])c1 ZINC000147251530 DJ For-Sale Bother PPOX1 15 45 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251559 GC On-Demand Anodyne PIK3CA 30 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251559 GC On-Demand Anodyne MTOR 59 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251559 GC On-Demand Anodyne EPHX2 20 51 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251559 GC On-Demand Anodyne PIK3CG 27 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251559 GC On-Demand Anodyne TNK2 21 45 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251559 GC On-Demand Anodyne L3MBTL3 58 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147251562 EE On-Demand Anodyne KCNQ2 59 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147251562 EE On-Demand Anodyne KLK3 41 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147251562 EE On-Demand Anodyne HDAC10 41 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N1CCCC1 ZINC000147251562 EE On-Demand Anodyne HDAC11 42 34 COc1ccc([N+](=O)[O-])c(C(=O)N2C[C@H]3CCCN3Cc3ccccc32)c1 ZINC000147251589 FG On-Demand Bother AVPR2 37 45 CC(C)CCCCNC(=O)c1sccc1N ZINC000147251608 BF For-Sale Anodyne HPN 65 33 CCCCCCCCNC(=O)N(CC(=O)O)C1CC1 ZINC000147251640 CF For-Sale Mild ACE 47 33 CCCCCCCCNC(=O)N(CC(=O)O)C1CC1 ZINC000147251640 CF For-Sale Mild EPHX2 41 43 CCCCCCCCNC(=O)N(CC(=O)O)C1CC1 ZINC000147251640 CF For-Sale Mild GNAI1 0 44 CCCCCCCCNC(=O)N(CC(=O)O)C1CC1 ZINC000147251640 CF For-Sale Mild GNAI3 0 44 CCCCCCCCNC(=O)N(CC(=O)O)C1CC1 ZINC000147251640 CF For-Sale Mild GNAO1 0 44 CCCCCCCCNC(=O)N(CC(=O)O)C1CC1 ZINC000147251640 CF For-Sale Mild ASAH1 68 34 CCCCCCCCNC(=O)N(CC(=O)O)C1CC1 ZINC000147251640 CF For-Sale Mild LASR 45 32 O=C(O)CN(C(=O)[C@H]1C[C@@H]1c1ccccc1)C1CC1 ZINC000147251641 CD For-Sale Anodyne ACE 56 44 O=C(O)CN(C(=O)[C@H]1C[C@@H]1c1ccccc1)C1CC1 ZINC000147251641 CD For-Sale Anodyne GPR88 0 47 CC[C@@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@@H]1N ZINC000147251652 CF On-Demand Anodyne CHRM1 22 42 CC[C@@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@@H]1N ZINC000147251652 CF On-Demand Anodyne CHRM3 32 42 CC[C@@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@@H]1N ZINC000147251652 CF On-Demand Anodyne NPY2R 36 40 CC[C@@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@@H]1N ZINC000147251652 CF On-Demand Anodyne AMY2 58 33 CC[C@@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@@H]1N ZINC000147251652 CF On-Demand Anodyne CYP2J2 41 35 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1ccc(N2CCCC2)nc1 ZINC000147251654 HI On-Demand Anodyne ROCK2 16 42 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1ccc(N2CCCC2)nc1 ZINC000147251654 HI On-Demand Anodyne MET 64 44 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1ccc(N2CCCC2)nc1 ZINC000147251654 HI On-Demand Anodyne NAMPT 61 45 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251729 GC On-Demand Anodyne PIK3CA 30 43 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251729 GC On-Demand Anodyne MTOR 59 43 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251729 GC On-Demand Anodyne EPHX2 20 51 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251729 GC On-Demand Anodyne PIK3CG 27 43 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251729 GC On-Demand Anodyne TNK2 21 45 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCOCC2)cc1 ZINC000147251729 GC On-Demand Anodyne L3MBTL3 58 36 COc1ccc([C@@H]2CCCCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)cc1 ZINC000147251787 HI On-Demand Bother FKBP1A 61 38 COc1ccc([C@@H]2CCCCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)cc1 ZINC000147251787 HI On-Demand Bother COLA 145 46 COc1ccc([C@@H]2CCCCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)cc1 ZINC000147251787 HI On-Demand Bother CPT1A 135 46 COc1ccc([C@@H]2CCCCCN2C(=O)COc2ccc([N+](=O)[O-])c(OC)c2)cc1 ZINC000147251787 HI On-Demand Bother CPT2 50 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(NC(=O)c3ccccn3)c1)C2 ZINC000147251830 HG On-Demand Anodyne GRM4 63 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(NC(=O)c3ccccn3)c1)C2 ZINC000147251830 HG On-Demand Anodyne ROCK2 55 42 O=C(O)CN(C(=O)[C@@H]1C[C@H]1c1ccccc1)C1CC1 ZINC000147251852 CD For-Sale Anodyne ACE 56 44 O=C(O)CN(C(=O)[C@@H]1C[C@H]1c1ccccc1)C1CC1 ZINC000147251852 CD For-Sale Anodyne GPR88 0 47 CCCCCCCCNC(=O)N(CC(=O)O)CC1CC1 ZINC000147251859 CF For-Sale Mild EPHX2 25 40 CCCCCCCCNC(=O)N(CC(=O)O)CC1CC1 ZINC000147251859 CF For-Sale Mild GNAI1 0 41 CCCCCCCCNC(=O)N(CC(=O)O)CC1CC1 ZINC000147251859 CF For-Sale Mild GNAI3 0 41 CCCCCCCCNC(=O)N(CC(=O)O)CC1CC1 ZINC000147251859 CF For-Sale Mild GNAO1 0 41 CCCCCCCCNC(=O)N(CC(=O)O)CC1CC1 ZINC000147251859 CF For-Sale Mild ASAH1 63 39 CC[C@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@@H]1N ZINC000147251874 CF On-Demand Anodyne CHRM1 22 42 CC[C@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@@H]1N ZINC000147251874 CF On-Demand Anodyne CHRM3 32 42 CC[C@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@@H]1N ZINC000147251874 CF On-Demand Anodyne NPY2R 36 40 CC[C@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@@H]1N ZINC000147251874 CF On-Demand Anodyne AMY2 58 33 CC[C@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@@H]1N ZINC000147251874 CF On-Demand Anodyne CYP2J2 41 35 CCCCCCCC/C=C/CCCCCCCC(=O)N(CCOCC)CCOCC ZINC000147251905 IK For-Sale Mild CNR1 15 59 CCCCCCCC/C=C/CCCCCCCC(=O)N(CCOCC)CCOCC ZINC000147251905 IK For-Sale Mild LPAR1 29 47 CCCCCCCC/C=C/CCCCCCCC(=O)N(CCOCC)CCOCC ZINC000147251905 IK For-Sale Mild LPAR2 15 47 CCCCCCCC/C=C/CCCCCCCC(=O)N(CCOCC)CCOCC ZINC000147251905 IK For-Sale Mild FAAH 21 51 CCCCCCCC/C=C/CCCCCCCC(=O)N(CCOCC)CCOCC ZINC000147251905 IK For-Sale Mild LPAR3 67 48 CCCCCCCC/C=C/CCCCCCCC(=O)N(CCOCC)CCOCC ZINC000147251905 IK For-Sale Mild FABP3 40 51 CCCCCCCC/C=C/CCCCCCCC(=O)N(CCOCC)CCOCC ZINC000147251905 IK For-Sale Mild FABP5 16 51 CCCCCCCC/C=C/CCCCCCCC(=O)N(CCOCC)CCOCC ZINC000147251905 IK For-Sale Mild ENPP2 19 41 CCCCCCCC/C=C/CCCCCCCC(=O)N(CCOCC)CCOCC ZINC000147251905 IK For-Sale Mild FABP1 17 51 CCCCCCCC/C=C/CCCCCCCC(=O)N(CCOCC)CCOCC ZINC000147251905 IK For-Sale Mild CQSS 52 32 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCCC2)nc1 ZINC000147251928 GH On-Demand Anodyne MTOR 47 39 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCCC2)nc1 ZINC000147251928 GH On-Demand Anodyne DGAT1 59 46 CC(C)CCCCNC(=O)c1c[nH]c2cc(N)ccc12 ZINC000147251936 CG For-Sale Anodyne TPR 17 44 CC(C)CCCCNC(=O)c1c[nH]c2cc(N)ccc12 ZINC000147251936 CG For-Sale Anodyne KISS1R 54 34 Cc1cc(Cl)ccc1Oc1nc(N)ncc1F ZINC000147251947 CF For-Sale Anodyne FOLA 19 40 Cc1cc(Cl)ccc1Oc1nc(N)ncc1F ZINC000147251947 CF For-Sale Anodyne AGPAT2 40 34 Cc1cc(Cl)ccc1Oc1nc(N)ncc1F ZINC000147251947 CF For-Sale Anodyne MAP3K14 40 40 C[C@H](N)CCC(=O)NN(C)C ZINC000147252032 AB For-Sale Reactive KDM7A 0 54 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1 ZINC000147252034 HF On-Demand Anodyne MLNR 18 41 CO[C@H](C(=O)N1CCC[C@@H]1c1ccccc1)c1ccccc1 ZINC000147252052 CH On-Demand Anodyne SLC6A3 22 40 CO[C@H](C(=O)N1CCC[C@@H]1c1ccccc1)c1ccccc1 ZINC000147252052 CH On-Demand Anodyne AGTR2 72 34 CO[C@H](C(=O)N1CCC[C@@H]1c1ccccc1)c1ccccc1 ZINC000147252052 CH On-Demand Anodyne ADAM17 55 46 CO[C@H](C(=O)N1CCC[C@@H]1c1ccccc1)c1ccccc1 ZINC000147252052 CH On-Demand Anodyne PREP 57 36 O=C(O)CN(C(=O)[C@@H]1C[C@@H]1c1ccccc1)C1CC1 ZINC000147252053 CD For-Sale Anodyne ACE 56 44 O=C(O)CN(C(=O)[C@@H]1C[C@@H]1c1ccccc1)C1CC1 ZINC000147252053 CD For-Sale Anodyne GPR88 0 47 O=C(COc1ccc(Cl)c(F)c1)c1ccc(Br)cc1 ZINC000147252077 EJ For-Sale Anodyne SHC 40 39 CCCCCCCCNC(=O)NCc1ccc(C(=O)O)o1 ZINC000147252102 CG For-Sale Mild S1PR2 46 39 CCCCCCCCNC(=O)NCc1ccc(C(=O)O)o1 ZINC000147252102 CG For-Sale Mild EPHX2 45 42 CCCCCCCCNC(=O)NCc1ccc(C(=O)O)o1 ZINC000147252102 CG For-Sale Mild ASAH1 90 36 COc1ccc2c(c1)OC[C@H](C(=O)NCc1cccc(NC(=O)C3CCCC3)c1)C2 ZINC000147252103 HH On-Demand Anodyne NQO2 25 42 COc1ccc2c(c1)OC[C@H](C(=O)NCc1cccc(NC(=O)C3CCCC3)c1)C2 ZINC000147252103 HH On-Demand Anodyne MTNR1A 46 42 COc1ccc2c(c1)OC[C@H](C(=O)NCc1cccc(NC(=O)C3CCCC3)c1)C2 ZINC000147252103 HH On-Demand Anodyne MTNR1B 41 42 COc1ccc2c(c1)OC[C@H](C(=O)NCc1cccc(NC(=O)C3CCCC3)c1)C2 ZINC000147252103 HH On-Demand Anodyne ROCK2 48 45 CC[C@@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@H]1N ZINC000147252110 CF On-Demand Anodyne CHRM1 22 42 CC[C@@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@H]1N ZINC000147252110 CF On-Demand Anodyne CHRM3 32 42 CC[C@@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@H]1N ZINC000147252110 CF On-Demand Anodyne NPY2R 36 40 CC[C@@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@H]1N ZINC000147252110 CF On-Demand Anodyne AMY2 58 33 CC[C@@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@H]1N ZINC000147252110 CF On-Demand Anodyne CYP2J2 41 35 O=C(C[C@@H]1CNc2ccccc21)N1CCCC1 ZINC000147252137 BE For-Sale Anodyne PREP 61 38 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCCC2)nc1 ZINC000147252153 GH On-Demand Anodyne MTOR 47 39 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCCC2)nc1 ZINC000147252153 GH On-Demand Anodyne DGAT1 59 46 COc1ccc(F)cc1CNC1(C(=O)O)CCC1 ZINC000147252159 CD On-Demand Anodyne NTSR2 25 42 CC(C)CCCCNC(=O)c1cc2cccc(N)c2[nH]1 ZINC000147252161 CG For-Sale Anodyne CCKAR 0 43 CC(C)CCCCNC(=O)c1cc2cccc(N)c2[nH]1 ZINC000147252161 CG For-Sale Anodyne PLCG2 0 43 C[C@H](CNS(=O)(=O)c1ccc2c(c1)OCCO2)CC(=O)O ZINC000147252181 DC On-Demand Anodyne PKM 29 41 COc1ccc(/C=C/C(=O)O)cc1S(=O)(=O)NCC(F)F ZINC000147252188 DD For-Sale Anodyne TUBB1 43 36 C[C@@H](OC[C@@H]1CCCO1)C(=O)N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1 ZINC000147252212 HF On-Demand Anodyne MLNR 18 41 CCc1c(NN)ncnc1Nc1ccc(C#N)cc1F ZINC000147252239 CE For-Sale Mild FLT1 0 43 C[C@@H](N)CCC(=O)NN(C)C ZINC000147252242 AB For-Sale Reactive KDM7A 0 54 Cc1ccc(C(=O)N(CC(=O)O)C2CC2)cc1Br ZINC000147252254 DE In-Stock Anodyne ACE 67 51 CO[C@H](C(=O)N1CCC[C@H]1c1ccccc1)c1ccccc1 ZINC000147252266 CH On-Demand Anodyne SLC6A3 22 40 CO[C@H](C(=O)N1CCC[C@H]1c1ccccc1)c1ccccc1 ZINC000147252266 CH On-Demand Anodyne AGTR2 72 34 CO[C@H](C(=O)N1CCC[C@H]1c1ccccc1)c1ccccc1 ZINC000147252266 CH On-Demand Anodyne ADAM17 55 46 CO[C@H](C(=O)N1CCC[C@H]1c1ccccc1)c1ccccc1 ZINC000147252266 CH On-Demand Anodyne PREP 57 36 N#CC1CCN(C(=O)CCc2ccc(S(=O)(=O)N3CCCCC3)cc2)CC1 ZINC000147252277 GF On-Demand Mild TGM2 41 45 N#CC1CCN(C(=O)CCc2ccc(S(=O)(=O)N3CCCCC3)cc2)CC1 ZINC000147252277 GF On-Demand Mild F13A1 48 45 N#CC1CCN(C(=O)CCc2ccc(S(=O)(=O)N3CCCCC3)cc2)CC1 ZINC000147252277 GF On-Demand Mild NAMPT 33 44 CCc1ccc(C(=O)COc2ccc(Cl)c(F)c2)s1 ZINC000147252286 CI For-Sale Anodyne ERCC5 23 41 CC[C@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@H]1N ZINC000147252324 CF On-Demand Anodyne CHRM1 22 42 CC[C@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@H]1N ZINC000147252324 CF On-Demand Anodyne CHRM3 32 42 CC[C@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@H]1N ZINC000147252324 CF On-Demand Anodyne NPY2R 36 40 CC[C@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@H]1N ZINC000147252324 CF On-Demand Anodyne AMY2 58 33 CC[C@H]1CN(C(=O)C(C)(C)c2ccccc2)CC[C@H]1N ZINC000147252324 CF On-Demand Anodyne CYP2J2 41 35 CCCCCCCCNC(=O)NCC(C)(C)C(=O)O ZINC000147252325 CF For-Sale Mild CPT1A 22 43 CCCCCCCCNC(=O)NCC(C)(C)C(=O)O ZINC000147252325 CF For-Sale Mild EPHX2 53 50 CCCCCCCCNC(=O)NCC(C)(C)C(=O)O ZINC000147252325 CF For-Sale Mild ASAH1 81 33 CCCCCCCCNC(=O)NCC(C)(C)C(=O)O ZINC000147252325 CF For-Sale Mild ACAT 0 44 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(NC(=O)C3CCCC3)c1)C2 ZINC000147252341 HH On-Demand Anodyne NQO2 25 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(NC(=O)C3CCCC3)c1)C2 ZINC000147252341 HH On-Demand Anodyne MTNR1A 46 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(NC(=O)C3CCCC3)c1)C2 ZINC000147252341 HH On-Demand Anodyne MTNR1B 41 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(NC(=O)C3CCCC3)c1)C2 ZINC000147252341 HH On-Demand Anodyne ROCK2 48 45 O=C(C[C@H]1CNc2ccccc21)N1CCCC1 ZINC000147252354 BE For-Sale Anodyne PREP 61 38 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCCC2)nc1 ZINC000147252371 GH On-Demand Anodyne MTOR 47 39 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCCC2)nc1 ZINC000147252371 GH On-Demand Anodyne DGAT1 59 46 C[C@@H](CNS(=O)(=O)c1ccc2c(c1)OCCO2)CC(=O)O ZINC000147252396 DC On-Demand Anodyne PKM 29 41 C[C@H](OC[C@H]1CCCO1)C(=O)N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1 ZINC000147252404 HF On-Demand Anodyne MLNR 18 41 CN(C)NC(=O)CCC(C)(C)CCN ZINC000147252432 BC For-Sale Reactive KDM7A 0 48 Cc1nc(C)c(C(=O)N(CC(=O)O)C2CC2)o1 ZINC000147252455 BC In-Stock Anodyne ACE 53 40 COc1cccc(C(F)F)c1 ZINC000147252475 AF For-Sale Anodyne MTNR1B 24 40 Cc1ccc(S(=O)(=O)N2CCCCC2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147252487 GF On-Demand Mild FASN 41 39 Cc1ccc(S(=O)(=O)N2CCCCC2)cc1C(=O)N1CCC(C#N)CC1 ZINC000147252487 GF On-Demand Mild L3MBTL3 59 43 O=C([C@@H]1COc2ccccc2C1)N1CCC[C@H](CCBr)C1 ZINC000147252508 FG For-Sale Reactive PREP 38 40 CCCCCCCCNC(=O)N1CCC[C@H](CC(=O)O)C1 ZINC000147252526 CG On-Demand Mild TPP2 25 40 CCCCCCCCNC(=O)N1CCC[C@H](CC(=O)O)C1 ZINC000147252526 CG On-Demand Mild ASAH1 99 41 CCCc1ccc(C(=O)COc2ccc(Cl)c(F)c2)cc1 ZINC000147252529 DJ For-Sale Anodyne PLA2G4B 65 33 CCCNC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147252569 FI On-Demand Anodyne GCGR 46 39 CCCNC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147252569 FI On-Demand Anodyne PRNP 15 41 CCCNC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147252569 FI On-Demand Anodyne NAMPT 25 40 O=C(C[C@@H]1CNc2ccccc21)NC1CCCCC1 ZINC000147252580 CG For-Sale Anodyne EPHX2 19 45 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCCC2)nc1 ZINC000147252581 GH On-Demand Anodyne MTOR 47 39 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCCC2)nc1 ZINC000147252581 GH On-Demand Anodyne DGAT1 59 46 C[C@@H](OC[C@H]1CCCO1)C(=O)N1CCN(Cc2ccc(C(F)(F)F)cc2)CC1 ZINC000147252585 HF On-Demand Anodyne MLNR 18 41 O=C(O)C1(NC[C@H]2COc3ccccc3O2)CCC1 ZINC000147252616 CD For-Sale Anodyne ADRA2B 21 41 CCOc1ccc(C(=O)NCCCCC(C)C)cc1N ZINC000147252625 CG For-Sale Anodyne FOLH1 44 35 CCOc1ccc(C(=O)NCCCCC(C)C)cc1N ZINC000147252625 CG For-Sale Anodyne ERAP2 44 31 COC(=O)c1ccccc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147252645 DC For-Sale Anodyne ILV2 0 40 CCCOc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1OCCC ZINC000147252648 GJ On-Demand Anodyne ACACA 16 40 CCCOc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1OCCC ZINC000147252648 GJ On-Demand Anodyne ACACB 17 40 O=C(O)CN(C(=O)C1[C@@H]2CCCC[C@@H]12)C1CC1 ZINC000147252665 BD On-Demand Anodyne ACE 58 41 O=C1S/C(=C/c2cc(-c3ccccc3)n(-c3ccc(Cl)cc3)c2-c2ccccc2)C(=O)N1c1ccccc1 ZINC000147252675 KK In-Stock Anodyne S1PR3 25 43 O=C1S/C(=C/c2cc(-c3ccccc3)n(-c3ccc(Cl)cc3)c2-c2ccccc2)C(=O)N1c1ccccc1 ZINC000147252675 KK In-Stock Anodyne MDM2 31 61 CCCCCCCCNC(=O)N1CCC[C@@H](CC(=O)O)C1 ZINC000147252697 CG On-Demand Mild TPP2 25 40 CCCCCCCCNC(=O)N1CCC[C@@H](CC(=O)O)C1 ZINC000147252697 CG On-Demand Mild ASAH1 99 41 O=C([C@H]1COc2ccccc2C1)N1CCC[C@H](CCBr)C1 ZINC000147252721 FG For-Sale Reactive PREP 38 40 CCCCNC(=O)C(C)(C)C(=O)NCCCC ZINC000147252739 BD For-Sale Anodyne ASAH1 40 31 Cc1ccc2[nH]c(CCc3ccncc3)nc2c1 ZINC000147252749 BG For-Sale Anodyne F9 23 44 CCCNC(=O)c1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147252752 FI On-Demand Anodyne GCGR 46 39 CCCNC(=O)c1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147252752 FI On-Demand Anodyne PRNP 15 41 CCCNC(=O)c1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147252752 FI On-Demand Anodyne NAMPT 25 40 O=C(C[C@H]1CNc2ccccc21)NC1CCCCC1 ZINC000147252812 CG For-Sale Anodyne EPHX2 19 45 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(OC(F)F)c1 ZINC000147252834 GJ On-Demand Anodyne CCR3 51 39 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(OC(F)F)c1 ZINC000147252834 GJ On-Demand Anodyne EPHX2 18 45 CCCOc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1OCCC ZINC000147252847 GJ On-Demand Anodyne ACACA 16 40 CCCOc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1OCCC ZINC000147252847 GJ On-Demand Anodyne ACACB 17 40 COc1cc(N)c(C(=O)NCCCCC(C)C)cc1OC ZINC000147252849 CF For-Sale Anodyne DRD3 21 44 COc1cc(N)c(C(=O)NCCCCC(C)C)cc1OC ZINC000147252849 CF For-Sale Anodyne HTR4 53 44 O=C(O)C1(NC[C@@H]2COc3ccccc3O2)CCC1 ZINC000147252854 CD For-Sale Anodyne ADRA2B 21 41 COC(=O)c1ccccc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147252869 DC For-Sale Anodyne ILV2 0 40 O=C(O)CN(C(=O)C1[C@H]2CCCC[C@@H]12)C1CC1 ZINC000147252876 BD For-Sale Anodyne ACE 58 41 CCCCCCCCNC(=O)N[C@@H](CC(=O)OC)C(=O)O ZINC000147252904 DD For-Sale Mild FOLH1 45 40 CCCCCCCCNC(=O)N[C@@H](CC(=O)OC)C(=O)O ZINC000147252904 DD For-Sale Mild CPT1A 50 51 CCCCCCCCNC(=O)N[C@@H](CC(=O)OC)C(=O)O ZINC000147252904 DD For-Sale Mild EPHX2 63 54 CCCCCCCCNC(=O)N[C@@H](CC(=O)OC)C(=O)O ZINC000147252904 DD For-Sale Mild ASAH1 70 33 CCCCCCCCNC(=O)N[C@@H](CC(=O)OC)C(=O)O ZINC000147252904 DD For-Sale Mild ACAT 0 40 CCCCCCCCNC(=O)N[C@@H](CC(=O)OC)C(=O)O ZINC000147252904 DD For-Sale Mild NOD1 89 42 O=C([C@@H]1COc2ccccc2C1)N1CCC[C@@H](CCBr)C1 ZINC000147252912 FG For-Sale Reactive PREP 38 40 CCCNC(=O)c1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147252955 FI On-Demand Anodyne GCGR 46 39 CCCNC(=O)c1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147252955 FI On-Demand Anodyne PRNP 15 41 CCCNC(=O)c1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147252955 FI On-Demand Anodyne NAMPT 25 40 O=C(C[C@@H]1CNc2ccccc21)Nc1ccccc1 ZINC000147253009 CG For-Sale Anodyne FUCA1 27 43 Cc1cccc(C(=O)COc2ccc(Cl)c(F)c2)c1 ZINC000147253014 CI For-Sale Anodyne KCNK3 52 38 Cc1cccc(C(=O)COc2ccc(Cl)c(F)c2)c1 ZINC000147253014 CI For-Sale Anodyne KCNK9 41 36 Cc1ccc2[nH]c(CCc3ccccn3)nc2c1 ZINC000147253022 BG For-Sale Anodyne CYSP_TRYCR 0 44 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(OC(F)F)c1 ZINC000147253051 GJ On-Demand Anodyne CCR3 51 39 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(OC(F)F)c1 ZINC000147253051 GJ On-Demand Anodyne EPHX2 18 45 O=C(O)CN(C(=O)C1[C@H]2CCCC[C@H]12)C1CC1 ZINC000147253053 BD On-Demand Anodyne ACE 58 41 O=C([C@H]1COc2ccccc2C1)N1CCC[C@@H](CCBr)C1 ZINC000147253073 FG For-Sale Reactive PREP 38 40 CCCCCCCCNC(=O)N1CC[C@@](CC)(C(=O)O)C1 ZINC000147253095 CG For-Sale Mild ASAH1 101 40 O=C(O)CCOc1ccc(S(=O)(=O)NCC(F)F)cc1 ZINC000147253106 DD On-Demand Anodyne TBXA2R 44 35 O=C(O)CCOc1ccc(S(=O)(=O)NCC(F)F)cc1 ZINC000147253106 DD On-Demand Anodyne MMP13 28 44 O=C(O)CCOc1ccc(S(=O)(=O)NCC(F)F)cc1 ZINC000147253106 DD On-Demand Anodyne ADAM17 18 44 O=C(O)CCOc1ccc(S(=O)(=O)NCC(F)F)cc1 ZINC000147253106 DD On-Demand Anodyne MMP2 23 42 O=C(O)CCOc1ccc(S(=O)(=O)NCC(F)F)cc1 ZINC000147253106 DD On-Demand Anodyne MMP14 18 44 O=C(O)CCOc1ccc(S(=O)(=O)NCC(F)F)cc1 ZINC000147253106 DD On-Demand Anodyne MMP9 28 42 O=C(O)CCOc1ccc(S(=O)(=O)NCC(F)F)cc1 ZINC000147253106 DD On-Demand Anodyne MMP7 19 42 O=C(O)CCOc1ccc(S(=O)(=O)NCC(F)F)cc1 ZINC000147253106 DD On-Demand Anodyne ADAMTS4 44 42 CC(C)CCCCNC(=O)c1cc2cc(N)ccc2o1 ZINC000147253137 CH For-Sale Anodyne PDGFRB 0 49 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(OC(F)F)c1 ZINC000147253164 GJ On-Demand Anodyne CCR3 51 39 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(OC(F)F)c1 ZINC000147253164 GJ On-Demand Anodyne EPHX2 18 45 CCc1cccc(C(C)(C)CC(=O)O)c1 ZINC000147253183 BG For-Sale Anodyne KIF11 18 45 O=C(C[C@H]1CNc2ccccc21)Nc1ccccc1 ZINC000147253190 CG For-Sale Anodyne FUCA1 27 43 CCCNC(=O)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147253201 FG On-Demand Anodyne DRD4 42 33 CCCNC(=O)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147253201 FG On-Demand Anodyne MTNR1A 50 41 CCCNC(=O)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147253201 FG On-Demand Anodyne MTNR1B 43 41 CCCNC(=O)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147253201 FG On-Demand Anodyne ROCK2 32 51 Cc1ccc2[nH]c(Cc3cccnc3)nc2c1 ZINC000147253218 BF For-Sale Anodyne TBXAS1 0 40 Cc1ccc2[nH]c(Cc3cccnc3)nc2c1 ZINC000147253218 BF For-Sale Anodyne ALKBH3 69 43 O=C(COc1ccc(Cl)c(F)c1)c1ccc(Cl)s1 ZINC000147253222 DI For-Sale Anodyne ERCC5 34 43 Cc1ncoc1C(=O)N(CC(=O)O)C1CC1 ZINC000147253275 BC On-Demand Anodyne ACE 62 40 CCCCCCCCNC(=O)N1CC[C@](CC)(C(=O)O)C1 ZINC000147253301 CG For-Sale Mild ASAH1 101 40 O=C(O)CN(C(=O)c1cccc2c1OCCN2)C1CC1 ZINC000147253377 CD For-Sale Anodyne ACE 60 52 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(OC(F)F)c1 ZINC000147253382 GJ On-Demand Anodyne CCR3 51 39 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(OC(F)F)c1 ZINC000147253382 GJ On-Demand Anodyne EPHX2 18 45 O=C(COc1ccc(CCNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1)NC1CC1 ZINC000147253388 HG On-Demand Anodyne PTPN22 16 40 CC(C)CCCCNC(=O)COc1ccccc1CN ZINC000147253390 CE For-Sale Anodyne GRIA1 57 33 CC(C)CCCCNC(=O)COc1ccccc1CN ZINC000147253390 CE For-Sale Anodyne FURIN 40 35 CC(C)CCCCNC(=O)COc1ccccc1CN ZINC000147253390 CE For-Sale Anodyne ST14 44 31 CC(C)CCCCNC(=O)COc1ccccc1CN ZINC000147253390 CE For-Sale Anodyne POLG_WNV 71 37 CC(C)CCCCNC(=O)COc1ccccc1CN ZINC000147253390 CE For-Sale Anodyne HPN 61 32 CCOC(=O)C1[C@@H]2CCCCC[C@@H]12 ZINC000147253504 AE For-Sale Anodyne Q8AWE3_CHICK 27 49 COc1ccccc1NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147253513 GF On-Demand Mild PRTN3 51 32 COc1ccccc1NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147253513 GF On-Demand Mild CCR8 47 35 COc1ccccc1NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147253513 GF On-Demand Mild SFRP1 46 35 COc1ccccc1NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147253513 GF On-Demand Mild LIMK2 21 48 COc1ccccc1NS(=O)(=O)c1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147253513 GF On-Demand Mild L3MBTL3 73 38 Cc1ncoc1C(=O)N1Cc2ccccc2C[C@@H]1C(=O)O ZINC000147253515 CD On-Demand Anodyne ACE 17 48 Cc1ncoc1C(=O)N1Cc2ccccc2C[C@@H]1C(=O)O ZINC000147253515 CD On-Demand Anodyne OPRM1 22 42 Cc1ncoc1C(=O)N1Cc2ccccc2C[C@@H]1C(=O)O ZINC000147253515 CD On-Demand Anodyne OPRD1 57 44 Cc1ncoc1C(=O)N1Cc2ccccc2C[C@@H]1C(=O)O ZINC000147253515 CD On-Demand Anodyne AGTR2 106 49 Cc1ncoc1C(=O)N1Cc2ccccc2C[C@@H]1C(=O)O ZINC000147253515 CD On-Demand Anodyne CFTR 56 38 Cc1ncoc1C(=O)N1Cc2ccccc2C[C@@H]1C(=O)O ZINC000147253515 CD On-Demand Anodyne ADAM9 42 32 CCCCCCCCNC(=O)N1CCC[C@@]1(C)C(=O)O ZINC000147253530 CF For-Sale Mild ASAH1 97 37 CNc1cc(Oc2ccc(Cl)cc2C)nc(N)n1 ZINC000147253538 CF For-Sale Anodyne AGPAT2 61 41 N#Cc1ccc(Nc2nc(NN)ncc2F)c(F)c1 ZINC000147253543 CD For-Sale Mild SYK 27 55 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc2c(c1)OCCO2 ZINC000147253571 EF On-Demand Anodyne CYP3A4 16 42 CC[C@@H]1CN(C(=O)c2ccc(C)nc2)CC[C@@H]1N ZINC000147253589 BD On-Demand Anodyne L3MBTL1 0 41 CC[C@@H]1CN(C(=O)c2ccc(C)nc2)CC[C@@H]1N ZINC000147253589 BD On-Demand Anodyne L3MBTL3 57 37 O=C(COc1ccc(CCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1)NC1CC1 ZINC000147253600 HG On-Demand Anodyne PTPN22 16 40 O=C(CNC1(C(=O)O)CCC1)N1CCc2ccccc2C1 ZINC000147253608 CD For-Sale Anodyne DPP8 25 43 N#Cc1ccc(Nc2nc(NN)ncc2Cl)c(F)c1 ZINC000147253715 CE For-Sale Mild INSR 31 40 N#Cc1ccc(Nc2nc(NN)ncc2Cl)c(F)c1 ZINC000147253715 CE For-Sale Mild MAPK9 53 48 N#Cc1ccc(Nc2nc(NN)ncc2Cl)c(F)c1 ZINC000147253715 CE For-Sale Mild MAPK10 53 48 N#Cc1ccc(Nc2nc(NN)ncc2Cl)c(F)c1 ZINC000147253715 CE For-Sale Mild ALK 21 40 CCCCCCCCNC(=O)N1CCC[C@]1(C)C(=O)O ZINC000147253716 CF For-Sale Mild ASAH1 97 37 C[C@@H](Cc1ccc(O)cc1)N(C)CCc1ccccc1 ZINC000147253743 CG On-Demand Anodyne ESR1 0 42 C[C@@H](Cc1ccc(O)cc1)N(C)CCc1ccccc1 ZINC000147253743 CG On-Demand Anodyne OPRM1 22 49 C[C@@H](Cc1ccc(O)cc1)N(C)CCc1ccccc1 ZINC000147253743 CG On-Demand Anodyne OPRD1 29 49 N#CC1CCN(C(=O)c2cc(S(=O)(=O)N3CCOCC3)ccc2F)CC1 ZINC000147253774 GD On-Demand Mild SLC6A9 30 43 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147253783 BB For-Sale Reactive TH 0 47 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147253783 BB For-Sale Reactive OPRM1 29 49 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147253783 BB For-Sale Reactive OPRD1 34 49 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147253783 BB For-Sale Reactive YARS 77 38 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147253783 BB For-Sale Reactive ALOX15 39 62 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147253783 BB For-Sale Reactive SLC15A2 0 43 CC[C@H]1CN(C(=O)c2ccc(C)nc2)CC[C@@H]1N ZINC000147253784 BD On-Demand Anodyne L3MBTL1 0 41 CC[C@H]1CN(C(=O)c2ccc(C)nc2)CC[C@@H]1N ZINC000147253784 BD On-Demand Anodyne L3MBTL3 57 37 C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc2c(c1)OCCO2 ZINC000147253798 EF On-Demand Anodyne CYP3A4 16 42 O=C(COc1ccc(CCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1)NC1CC1 ZINC000147253801 HG On-Demand Anodyne PTPN22 16 40 CC(C)CCCCNC(=O)C(=O)NCCN ZINC000147253832 BC For-Sale Anodyne DNPEP 0 43 CC(C)CCCCNC(=O)C(=O)NCCN ZINC000147253832 BC For-Sale Anodyne SIRT1 29 41 O=C(C[C@@H]1CNc2ccccc21)Nc1nccs1 ZINC000147253875 CF For-Sale Anodyne MAP 0 44 O=C(C[C@@H]1CNc2ccccc21)Nc1nccs1 ZINC000147253875 CF For-Sale Anodyne MAP1 123 40 CCOC(=O)C1[C@H]2CCCCC[C@H]12 ZINC000147253919 AE For-Sale Anodyne Q8AWE3_CHICK 27 49 CCCCCCCCNC(=O)N1CC[C@H](CC(=O)O)C1 ZINC000147253940 CF For-Sale Mild GNAI1 0 42 CCCCCCCCNC(=O)N1CC[C@H](CC(=O)O)C1 ZINC000147253940 CF For-Sale Mild GNAI3 0 43 CCCCCCCCNC(=O)N1CC[C@H](CC(=O)O)C1 ZINC000147253940 CF For-Sale Mild GNAO1 0 42 CCCCCCCCNC(=O)N1CC[C@H](CC(=O)O)C1 ZINC000147253940 CF For-Sale Mild ASAH1 102 43 CCCCCCCCNC(=O)N1CC[C@H](CC(=O)O)C1 ZINC000147253940 CF For-Sale Mild NR1D2 0 43 C[C@H](Cc1ccc(O)cc1)N(C)CCc1ccccc1 ZINC000147253943 CG On-Demand Anodyne ESR1 0 42 C[C@H](Cc1ccc(O)cc1)N(C)CCc1ccccc1 ZINC000147253943 CG On-Demand Anodyne OPRM1 22 49 C[C@H](Cc1ccc(O)cc1)N(C)CCc1ccccc1 ZINC000147253943 CG On-Demand Anodyne OPRD1 29 49 CC(C)(C)c1nc(NN)cc(NCCc2ccccc2)n1 ZINC000147253955 CF For-Sale Anodyne PTGDR 21 40 CC(C)(C)c1nc(NN)cc(NCCc2ccccc2)n1 ZINC000147253955 CF For-Sale Anodyne PETD 0 43 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2ccccn2)CC1 ZINC000147253967 ED On-Demand Anodyne P2RY12 184 37 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2ccccn2)CC1 ZINC000147253967 ED On-Demand Anodyne ST14 64 34 CC[C@@H]1CN(C(=O)c2ccc(C)nc2)CC[C@H]1N ZINC000147253975 BD On-Demand Anodyne L3MBTL1 0 41 CC[C@@H]1CN(C(=O)c2ccc(C)nc2)CC[C@H]1N ZINC000147253975 BD On-Demand Anodyne L3MBTL3 57 37 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1O ZINC000147253981 EG For-Sale Reactive GRM3 20 48 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1O ZINC000147253981 EG For-Sale Reactive L3MBTL3 40 33 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1O ZINC000147253981 EG For-Sale Reactive ACKR3 63 34 Cc1cc(NC(=O)c2cncs2)ccc1F ZINC000147253992 BF On-Demand Anodyne CSF1R 16 42 Cc1cc(NC(=O)c2cncs2)ccc1F ZINC000147253992 BF On-Demand Anodyne Q25615_ONCVO 53 32 Cc1cc(NC(=O)c2cncs2)ccc1F ZINC000147253992 BF On-Demand Anodyne KCNK3 43 32 O=C(COc1ccc(CCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1)NC1CC1 ZINC000147254029 HG On-Demand Anodyne PTPN22 16 40 O=C(CNC1(C(=O)O)CCC1)Nc1nc2ccccc2s1 ZINC000147254052 DD For-Sale Anodyne CSNK1D 46 58 O=C(CNC1(C(=O)O)CCC1)Nc1nc2ccccc2s1 ZINC000147254052 DD For-Sale Anodyne BCL2L1 59 39 O=C(CNC1(C(=O)O)CCC1)Nc1nc2ccccc2s1 ZINC000147254052 DD For-Sale Anodyne FABK 0 44 O=C(CNC1(C(=O)O)CCC1)Nc1nc2ccccc2s1 ZINC000147254052 DD For-Sale Anodyne PORCN 0 48 O=C(CNC1(C(=O)O)CCC1)Nc1nc2ccccc2s1 ZINC000147254052 DD For-Sale Anodyne ISPD 0 41 O=C(C[C@H]1CNc2ccccc21)Nc1nccs1 ZINC000147254090 CF For-Sale Anodyne MAP 0 44 O=C(C[C@H]1CNc2ccccc21)Nc1nccs1 ZINC000147254090 CF For-Sale Anodyne MAP1 123 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1NS(C)(=O)=O ZINC000147254096 ED On-Demand Anodyne PLA2G7 19 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1NS(C)(=O)=O ZINC000147254096 ED On-Demand Anodyne PCSK5 40 33 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1NS(C)(=O)=O ZINC000147254096 ED On-Demand Anodyne FURIN 45 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1NS(C)(=O)=O ZINC000147254096 ED On-Demand Anodyne POLG_WNV 72 33 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1NS(C)(=O)=O ZINC000147254096 ED On-Demand Anodyne NPFFR1 52 33 CCCCCCCCNC(=O)N1CC[C@@H](CC(=O)O)C1 ZINC000147254142 CF For-Sale Mild GNAI1 0 42 CCCCCCCCNC(=O)N1CC[C@@H](CC(=O)O)C1 ZINC000147254142 CF For-Sale Mild GNAI3 0 43 CCCCCCCCNC(=O)N1CC[C@@H](CC(=O)O)C1 ZINC000147254142 CF For-Sale Mild GNAO1 0 42 CCCCCCCCNC(=O)N1CC[C@@H](CC(=O)O)C1 ZINC000147254142 CF For-Sale Mild ASAH1 102 43 CCCCCCCCNC(=O)N1CC[C@@H](CC(=O)O)C1 ZINC000147254142 CF For-Sale Mild NR1D2 0 43 CC(C)CCCCNC(=O)COc1ccc(CN)cc1 ZINC000147254145 CE For-Sale Anodyne GRIA1 49 35 CC(C)CCCCNC(=O)COc1ccc(CN)cc1 ZINC000147254145 CE For-Sale Anodyne PLA2G4B 42 32 CC(C)CCCCNC(=O)COc1ccc(CN)cc1 ZINC000147254145 CE For-Sale Anodyne TPSAB1 43 38 CC(C)CCCCNC(=O)COc1ccc(CN)cc1 ZINC000147254145 CE For-Sale Anodyne POLG_WNV 46 36 O=C(N[C@@H](C(=O)O)c1ccccc1)c1cccc(F)c1Cl ZINC000147254182 DG On-Demand Anodyne AMP1_PLAFQ 18 40 O=C(N[C@@H](C(=O)O)c1ccccc1)c1cccc(F)c1Cl ZINC000147254182 DG On-Demand Anodyne VANX 0 46 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1O ZINC000147254196 EG For-Sale Reactive GRM3 20 48 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1O ZINC000147254196 EG For-Sale Reactive L3MBTL3 40 33 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1O ZINC000147254196 EG For-Sale Reactive ACKR3 63 34 CC[C@H]1CN(C(=O)c2ccc(C)nc2)CC[C@H]1N ZINC000147254201 BD On-Demand Anodyne L3MBTL1 0 41 CC[C@H]1CN(C(=O)c2ccc(C)nc2)CC[C@H]1N ZINC000147254201 BD On-Demand Anodyne L3MBTL3 57 37 CCNCCC(=O)NN(C)C ZINC000147254212 AB For-Sale Reactive KDM7A 0 54 COc1ccccc1CNC(=O)CNC1(C(=O)O)CCC1 ZINC000147254262 CC For-Sale Anodyne TACR1 22 43 COc1ccccc1CNC(=O)CNC1(C(=O)O)CCC1 ZINC000147254262 CC For-Sale Anodyne KCNA3 40 36 COc1ccccc1CNC(=O)CNC1(C(=O)O)CCC1 ZINC000147254262 CC For-Sale Anodyne MBTPS1 43 32 Cc1nccc(CNC(=O)CCCc2ccc3c(c2)-c2ccccc2C3)n1 ZINC000147254269 FH On-Demand Anodyne SUCNR1 56 39 Cc1cc(C(=O)Nc2ccc(NC(=O)C(C)C)cc2)cc([N+](=O)[O-])c1 ZINC000147254270 EH On-Demand Bother KCNK3 54 38 Cc1cc(C(=O)Nc2ccc(NC(=O)C(C)C)cc2)cc([N+](=O)[O-])c1 ZINC000147254270 EH On-Demand Bother KCNK9 42 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1NS(C)(=O)=O ZINC000147254289 ED On-Demand Anodyne PLA2G7 19 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1NS(C)(=O)=O ZINC000147254289 ED On-Demand Anodyne PCSK5 40 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1NS(C)(=O)=O ZINC000147254289 ED On-Demand Anodyne FURIN 45 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1NS(C)(=O)=O ZINC000147254289 ED On-Demand Anodyne POLG_WNV 72 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1NS(C)(=O)=O ZINC000147254289 ED On-Demand Anodyne NPFFR1 52 33 CCCCCCCCNC(=O)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000147254346 CF On-Demand Mild EPHX2 42 64 CCCCCCCCNC(=O)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000147254346 CF On-Demand Mild GNAI1 0 45 CCCCCCCCNC(=O)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000147254346 CF On-Demand Mild GNAI3 0 45 CCCCCCCCNC(=O)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000147254346 CF On-Demand Mild GNAO1 0 45 CCCCCCCCNC(=O)N[C@@H]1CC[C@H](C(=O)O)C1 ZINC000147254346 CF On-Demand Mild ASAH1 56 33 O=C(COc1ccc(Cl)c(F)c1)c1cc(Cl)ccc1Cl ZINC000147254349 EK For-Sale Anodyne ALPL 43 32 O=C(COc1ccc(Cl)c(F)c1)c1cc(Cl)ccc1Cl ZINC000147254349 EK For-Sale Anodyne FEN1 0 46 CC(C)CCCCNCc1ccc(Br)cc1 ZINC000147254370 CI For-Sale Anodyne FDFT1 0 41 CC(C)CCCCNCc1ccc(Br)cc1 ZINC000147254370 CI For-Sale Anodyne S1PR2 32 41 CC(C)CCCCNCc1ccc(Br)cc1 ZINC000147254370 CI For-Sale Anodyne LEF 94 39 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N[C@@H]1C[C@@H]1c1ccccc1)C(=O)C2 ZINC000147254392 EF On-Demand Anodyne CA5B 32 55 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N[C@@H]1C[C@@H]1c1ccccc1)C(=O)C2 ZINC000147254392 EF On-Demand Anodyne CA5A 34 55 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N[C@@H]1C[C@@H]1c1ccccc1)C(=O)C2 ZINC000147254392 EF On-Demand Anodyne CXCR3 41 43 O=C(Nc1cccc(O)c1)c1cccc2c1OCCN2 ZINC000147254398 CE For-Sale Anodyne KCNK3 92 37 O=C(Nc1cccc(O)c1)c1cccc2c1OCCN2 ZINC000147254398 CE For-Sale Anodyne KCNK9 72 37 Cc1ccc(C(=O)N[C@@H](C(=O)O)c2ccccc2)cc1Br ZINC000147254402 EG On-Demand Anodyne MTTP 67 39 Cc1ccc(C(=O)N[C@@H](C(=O)O)c2ccccc2)cc1Br ZINC000147254402 EG On-Demand Anodyne VANX 0 42 CC[C@@H]1CN(C(=O)c2ccc(C(F)(F)F)nc2)CC[C@@H]1N ZINC000147254462 DE On-Demand Anodyne SLC9A1 44 39 Cc1ccc(NC(=O)CNC2(C(=O)O)CCC2)cc1 ZINC000147254494 CD For-Sale Anodyne FUCA1 18 40 COCCc1ccc(-c2c(C)nc3c(-c4ccncc4)nccn23)cn1 ZINC000147254497 EG Annotated Anodyne PDE10A 16 52 Clc1cnc(-c2ccccc2)nc1N1CCCCC1 ZINC000147254516 CH For-Sale Anodyne NPY5R 19 42 C[C@H](Oc1ccc(Cl)cc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147254552 EH On-Demand Mild CCR1 41 36 CCCCCCCCNC(=O)N[C@H]1CC[C@H](C(=O)O)C1 ZINC000147254561 CF For-Sale Mild EPHX2 42 64 CCCCCCCCNC(=O)N[C@H]1CC[C@H](C(=O)O)C1 ZINC000147254561 CF For-Sale Mild GNAI1 0 45 CCCCCCCCNC(=O)N[C@H]1CC[C@H](C(=O)O)C1 ZINC000147254561 CF For-Sale Mild GNAI3 0 45 CCCCCCCCNC(=O)N[C@H]1CC[C@H](C(=O)O)C1 ZINC000147254561 CF For-Sale Mild GNAO1 0 45 CCCCCCCCNC(=O)N[C@H]1CC[C@H](C(=O)O)C1 ZINC000147254561 CF For-Sale Mild ASAH1 56 33 CCCCOCC(=O)CO ZINC000147254592 AC For-Sale Anodyne PLA2G2C 40 31 CCCCOCC(=O)CO ZINC000147254592 AC For-Sale Anodyne PLA2G4B 73 44 CCCCOCC(=O)CO ZINC000147254592 AC For-Sale Anodyne CES2 18 47 CCCCOCC(=O)CO ZINC000147254592 AC For-Sale Anodyne EST1_PIG 33 47 CCCCOCC(=O)CO ZINC000147254592 AC For-Sale Anodyne CES2C 22 47 CCCCOCC(=O)CO ZINC000147254592 AC For-Sale Anodyne JHE 0 47 CCN1CCC[C@H](NC(=O)c2cccc3c2OCCN3)C1 ZINC000147254639 CD For-Sale Anodyne DRD2 15 44 CCN1CCC[C@H](NC(=O)c2cccc3c2OCCN3)C1 ZINC000147254639 CD For-Sale Anodyne BIRC2 41 35 O=C(N[C@@H](C(=O)O)c1ccccc1)C1[C@H]2CCCC[C@H]12 ZINC000147254657 CE On-Demand Anodyne NAALAD2 19 41 CC[C@H]1CN(C(=O)c2ccc(C(F)(F)F)nc2)CC[C@@H]1N ZINC000147254692 DE On-Demand Anodyne SLC9A1 44 39 CN(C)C(=O)NCCNC(=O)c1cccc(/C(N)=N/O)c1 ZINC000147254707 CB For-Sale Mild DRD4 40 31 O=C(CNC1(C(=O)O)CCC1)Nc1ccc(F)c(F)c1 ZINC000147254733 CD For-Sale Anodyne SLC1A2 48 40 O=C(CNC1(C(=O)O)CCC1)Nc1ccc(F)c(F)c1 ZINC000147254733 CD For-Sale Anodyne ENV 41 33 C[C@@H](Oc1ccc(Cl)cc1Cl)C(=O)N1CCC(C#N)CC1 ZINC000147254761 EH On-Demand Mild CCR1 41 36 CCCCCCCCNC(=O)N[C@@H]1CC[C@@H](C(=O)O)C1 ZINC000147254767 CF For-Sale Mild EPHX2 42 64 CCCCCCCCNC(=O)N[C@@H]1CC[C@@H](C(=O)O)C1 ZINC000147254767 CF For-Sale Mild GNAI1 0 45 CCCCCCCCNC(=O)N[C@@H]1CC[C@@H](C(=O)O)C1 ZINC000147254767 CF For-Sale Mild GNAI3 0 45 CCCCCCCCNC(=O)N[C@@H]1CC[C@@H](C(=O)O)C1 ZINC000147254767 CF For-Sale Mild GNAO1 0 45 CCCCCCCCNC(=O)N[C@@H]1CC[C@@H](C(=O)O)C1 ZINC000147254767 CF For-Sale Mild ASAH1 56 33 C[C@H](Oc1ccc(Cl)c(F)c1)C(=O)c1ccc(F)cc1F ZINC000147254819 DI For-Sale Anodyne CES2 19 47 O=C(Cc1ccc(F)cc1F)N1CCC[C@H](CCBr)C1 ZINC000147254839 EH For-Sale Reactive HTR2A 18 43 CCN1CCC[C@@H](NC(=O)c2cccc3c2OCCN3)C1 ZINC000147254847 CD For-Sale Anodyne DRD2 15 44 CCN1CCC[C@@H](NC(=O)c2cccc3c2OCCN3)C1 ZINC000147254847 CD For-Sale Anodyne BIRC2 41 35 Cc1ccc2c(c1)c(-c1ccc(C(C)C)cc1)nc(=O)n2C(C)C ZINC000147254866 DK For-Sale Anodyne CASR 38 63 O=C(N[C@@H](C(=O)O)c1ccccc1)C1[C@H]2CCCC[C@@H]12 ZINC000147254880 CE For-Sale Anodyne NAALAD2 19 41 Cc1cc(Cl)ccc1Oc1nc(N)ncc1Cl ZINC000147254887 CG For-Sale Anodyne FOLA 22 41 Cc1cc(Cl)ccc1Oc1nc(N)ncc1Cl ZINC000147254887 CG For-Sale Anodyne DRTS_PLAFK 22 40 Cc1cc(Cl)ccc1Oc1nc(N)ncc1Cl ZINC000147254887 CG For-Sale Anodyne P2RX2 40 38 Cc1cc(Cl)ccc1Oc1nc(N)ncc1Cl ZINC000147254887 CG For-Sale Anodyne AGPAT2 46 35 Cc1cc(Cl)ccc1Oc1nc(N)ncc1Cl ZINC000147254887 CG For-Sale Anodyne MAP3K14 42 40 CC[C@@H]1CN(C(=O)c2ccc(C(F)(F)F)nc2)CC[C@H]1N ZINC000147254889 DE On-Demand Anodyne SLC9A1 44 39 CCCCCCCCNC(=O)N[C@H]1CC[C@@H](C(=O)O)C1 ZINC000147254993 CF For-Sale Mild EPHX2 42 64 CCCCCCCCNC(=O)N[C@H]1CC[C@@H](C(=O)O)C1 ZINC000147254993 CF For-Sale Mild GNAI1 0 45 CCCCCCCCNC(=O)N[C@H]1CC[C@@H](C(=O)O)C1 ZINC000147254993 CF For-Sale Mild GNAI3 0 45 CCCCCCCCNC(=O)N[C@H]1CC[C@@H](C(=O)O)C1 ZINC000147254993 CF For-Sale Mild GNAO1 0 45 CCCCCCCCNC(=O)N[C@H]1CC[C@@H](C(=O)O)C1 ZINC000147254993 CF For-Sale Mild ASAH1 56 33 C[C@@H](Oc1ccc(Cl)c(F)c1)C(=O)c1ccc(F)cc1F ZINC000147255041 DI For-Sale Anodyne CES2 19 47 CC(C)CNC(=O)/C=C/C=C/CC/C=C\[C@H](O)[C@H](C)O ZINC000147255090 CD Annotated Anodyne CNR2 15 66 CC[C@H]1CN(C(=O)c2ccc(C(F)(F)F)nc2)CC[C@H]1N ZINC000147255100 DE On-Demand Anodyne SLC9A1 44 39 CN(C)NC(=O)CCC1CCNCC1 ZINC000147255104 AC For-Sale Reactive PHF8 0 44 CN(C)NC(=O)CCC1CCNCC1 ZINC000147255104 AC For-Sale Reactive KDM7A 0 44 O=C(Cc1ccc(F)cc1F)N1CCC[C@@H](CCBr)C1 ZINC000147255107 EH For-Sale Reactive HTR2A 18 43 Cc1nccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)n1 ZINC000147255137 DF On-Demand Anodyne NAMPT 17 45 CCC[C@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147255140 DH On-Demand Anodyne BMP1 54 36 CCC[C@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147255140 DH On-Demand Anodyne TACR3 27 40 CCC[C@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147255140 DH On-Demand Anodyne CYP3A4 20 47 OCCCCCc1cnc(-c2ccccc2)c(-c2ccccc2)n1 ZINC000147255196 DJ For-Sale Anodyne FAAH 32 41 CCCCCCCCCNC1(C(=O)O)CCC1 ZINC000147255205 BG For-Sale Mild CES2 34 42 CCCCCCCCCNC1(C(=O)O)CCC1 ZINC000147255205 BG For-Sale Mild EST1_PIG 50 35 CCCCCCCCCNC1(C(=O)O)CCC1 ZINC000147255205 BG For-Sale Mild CES2C 40 42 CCCCCCCCNC(=O)N[C@@H]1COC[C@@]1(C)C(=O)O ZINC000147255221 DE For-Sale Mild EPHX2 58 45 C/C=C\C(=O)c1cccc(C(F)(F)F)c1 ZINC000147255251 BG For-Sale Mild CACNA1B 45 32 C/C=C\C(=O)c1cccc(C(F)(F)F)c1 ZINC000147255251 BG For-Sale Mild CCR2 46 38 C/C=C\C(=O)c1cccc(C(F)(F)F)c1 ZINC000147255251 BG For-Sale Mild BTK 15 41 C/C=C\C(=O)c1cccc(C(F)(F)F)c1 ZINC000147255251 BG For-Sale Mild KCNK3 20 50 COc1ccc(C(C)=O)cc1COc1ccc(Cl)c(F)c1 ZINC000147255263 DI For-Sale Anodyne TSHR 58 36 COc1ccc(C(C)=O)cc1COc1ccc(Cl)c(F)c1 ZINC000147255263 DI For-Sale Anodyne GYS1 41 33 Cc1nccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)n1 ZINC000147255309 DF On-Demand Anodyne NAMPT 17 45 CCC[C@@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147255310 DH On-Demand Anodyne BMP1 54 36 CCC[C@@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147255310 DH On-Demand Anodyne CYP3A4 20 47 C[C@H](CNS(=O)(=O)C[C@@H](C)c1ccccc1)CC(=O)O ZINC000147255327 CD For-Sale Anodyne GRIA4 23 45 COc1ccc(Nc2nc(-c3ccc4[nH]ncc4c3)cn3ccnc23)cc1OC ZINC000147255349 GI For-Sale Anodyne ROCK2 26 47 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H](CCBr)C1 ZINC000147255357 FI For-Sale Reactive SLC6A1 15 41 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H](CCBr)C1 ZINC000147255357 FI For-Sale Reactive RBP4 84 41 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H](CCBr)C1 ZINC000147255357 FI For-Sale Reactive SCD1 29 47 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H](CCBr)C1 ZINC000147255357 FI For-Sale Reactive SFRP1 58 35 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H](CCBr)C1 ZINC000147255357 FI For-Sale Reactive SCD 30 47 CN(C)NC(=O)CCC(C)(C)N ZINC000147255364 AC For-Sale Reactive KDM7A 0 52 CCCCCCCCNC(=O)N[C@H]1COC[C@@]1(C)C(=O)O ZINC000147255414 DE For-Sale Mild EPHX2 58 45 CCCOc1cccc(C(=O)N2CC[C@H](N)[C@H](CC)C2)c1 ZINC000147255484 CF On-Demand Anodyne L3MBTL1 0 41 Cc1nccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)n1 ZINC000147255494 DF On-Demand Anodyne NAMPT 17 45 C[C@@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147255510 CF For-Sale Anodyne PREP 112 37 C[C@H](CS(=O)(=O)NC[C@H](C)CC(=O)O)c1ccccc1 ZINC000147255520 CD For-Sale Anodyne GRIA4 23 45 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H](CCBr)C1 ZINC000147255540 FI For-Sale Reactive SLC6A1 15 41 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H](CCBr)C1 ZINC000147255540 FI For-Sale Reactive RBP4 84 41 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H](CCBr)C1 ZINC000147255540 FI For-Sale Reactive SCD1 29 47 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H](CCBr)C1 ZINC000147255540 FI For-Sale Reactive SFRP1 58 35 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H](CCBr)C1 ZINC000147255540 FI For-Sale Reactive SCD 30 47 CCC[C@H](NC(=O)N(C)Cc1csc(CC)n1)c1ccccc1 ZINC000147255560 EI On-Demand Anodyne TACR3 30 41 CN1CCC[C@H](NC(=O)c2cccc3c2OCCN3)C1 ZINC000147255579 CD For-Sale Anodyne HTR4 16 44 CCNc1cccc(NCCCN2CCCC[C@@H]2C)n1 ZINC000147255630 CG For-Sale Anodyne HRH3 59 39 CCCCCCCCNC(=O)N[C@@H]1COC[C@]1(C)C(=O)O ZINC000147255642 DE For-Sale Mild EPHX2 58 45 O=C(CNC1(C(=O)O)CCC1)Nc1ccc(Cl)cc1 ZINC000147255676 CD For-Sale Anodyne SLC1A2 35 40 O=C(CNC1(C(=O)O)CCC1)Nc1ccc(Cl)cc1 ZINC000147255676 CD For-Sale Anodyne IMDH_CRYPV 18 40 CCCOc1cccc(C(=O)N2CC[C@@H](N)[C@H](CC)C2)c1 ZINC000147255683 CF On-Demand Anodyne L3MBTL1 0 41 CCCOC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147255691 ED On-Demand Anodyne ACR 40 31 Cc1nccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)n1 ZINC000147255707 DF On-Demand Anodyne NAMPT 17 45 C[C@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147255728 CF For-Sale Anodyne PREP 112 37 C[C@H](CNS(=O)(=O)C[C@H](C)c1ccccc1)CC(=O)O ZINC000147255730 CD For-Sale Anodyne GRIA4 23 45 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@H](CCBr)C1 ZINC000147255755 FI For-Sale Reactive EPHX2 16 41 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@H](CCBr)C1 ZINC000147255755 FI For-Sale Reactive MCHR1 17 42 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@H](CCBr)C1 ZINC000147255755 FI For-Sale Reactive MLYCD 20 45 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@H](CCBr)C1 ZINC000147255755 FI For-Sale Reactive RHOA 0 41 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@H](CCBr)C1 ZINC000147255755 FI For-Sale Reactive L3MBTL3 57 39 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@H](CCBr)C1 ZINC000147255755 FI For-Sale Reactive SLC6A7 0 43 COc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1[N+](=O)[O-] ZINC000147255775 FH On-Demand Mild CPT1A 44 30 COc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1[N+](=O)[O-] ZINC000147255775 FH On-Demand Mild GRM4 20 42 COc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1[N+](=O)[O-] ZINC000147255775 FH On-Demand Mild TAAR1 38 49 COc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1[N+](=O)[O-] ZINC000147255775 FH On-Demand Mild DDR1 40 39 COc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1[N+](=O)[O-] ZINC000147255775 FH On-Demand Mild KCNK3 76 39 COc1ccc(C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1[N+](=O)[O-] ZINC000147255775 FH On-Demand Mild KCNK9 61 39 CN1CCC[C@@H](NC(=O)c2cccc3c2OCCN3)C1 ZINC000147255783 CD For-Sale Anodyne HTR4 16 44 CCC[C@@H](NC(=O)N(C)Cc1csc(CC)n1)c1ccccc1 ZINC000147255785 EI On-Demand Anodyne TACR3 30 41 CCNc1cccc(NCCCN2CCCC[C@H]2C)n1 ZINC000147255839 CG For-Sale Anodyne HRH3 59 39 CCCCCCCCNC(=O)N[C@H]1COC[C@]1(C)C(=O)O ZINC000147255867 DE For-Sale Mild EPHX2 58 45 O=C(c1ccc(S(=O)(=O)Nc2nccs2)cc1)N1CC[C@@H](Cc2ccccc2)C1 ZINC000147255893 IH On-Demand Anodyne GRIN2B 52 50 O=C(c1ccc(S(=O)(=O)Nc2nccs2)cc1)N1CC[C@@H](Cc2ccccc2)C1 ZINC000147255893 IH On-Demand Anodyne GCK 16 40 O=C(c1ccc(S(=O)(=O)Nc2nccs2)cc1)N1CC[C@@H](Cc2ccccc2)C1 ZINC000147255893 IH On-Demand Anodyne LIMK2 43 39 Cc1ccccc1CNCCCCC(C)C ZINC000147255901 BH For-Sale Anodyne LEF 71 42 Cc1ccccc1CNCCCCC(C)C ZINC000147255901 BH For-Sale Anodyne GPM3 0 72 CCCOc1cccc(C(=O)N2CC[C@H](N)[C@@H](CC)C2)c1 ZINC000147255912 CF On-Demand Anodyne L3MBTL1 0 41 CCCOC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147255921 ED On-Demand Anodyne ACR 40 31 CC(C)(C)C[C@H]1N[C@@H](C(=O)NCCN2CCOCC2)[C@H](c2cccc(Cl)c2F)[C@@]12C(=O)Nc1cc(F)c(F)cc12 ZINC000147255945 KH Annotated Anodyne MDM2 101 78 C[C@@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147255954 CF For-Sale Anodyne PREP 112 37 C[C@@H](CNS(=O)(=O)C[C@H](C)c1ccccc1)CC(=O)O ZINC000147255962 CD For-Sale Anodyne GRIA4 23 45 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147255967 FI For-Sale Reactive EPHX2 16 41 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147255967 FI For-Sale Reactive MCHR1 17 42 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147255967 FI For-Sale Reactive MLYCD 20 45 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147255967 FI For-Sale Reactive RHOA 0 41 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147255967 FI For-Sale Reactive L3MBTL3 57 39 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147255967 FI For-Sale Reactive SLC6A7 0 43 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccnc(C)n1)C2 ZINC000147255975 DD On-Demand Anodyne MTNR1A 19 40 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccnc(C)n1)C2 ZINC000147255975 DD On-Demand Anodyne ROCK2 31 43 CC[C@](C)(NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147256005 CE For-Sale Anodyne GPR88 0 45 O=C(c1ccc(S(=O)(=O)Nc2nccs2)cc1)N1CC[C@H](Cc2ccccc2)C1 ZINC000147256048 IH On-Demand Anodyne GRIN2B 52 50 O=C(c1ccc(S(=O)(=O)Nc2nccs2)cc1)N1CC[C@H](Cc2ccccc2)C1 ZINC000147256048 IH On-Demand Anodyne GCK 16 40 O=C(c1ccc(S(=O)(=O)Nc2nccs2)cc1)N1CC[C@H](Cc2ccccc2)C1 ZINC000147256048 IH On-Demand Anodyne LIMK2 43 39 Cc1cccc(Cl)c1C(=O)NCc1ccc(-c2cc[nH]c(=O)c2)cc1 ZINC000147256075 FH For-Sale Anodyne RPA1 41 36 CCCCCCCCNC(=O)NC1(CC(=O)O)CCC1 ZINC000147256106 CG For-Sale Mild CPT1A 36 45 CCCCCCCCNC(=O)NC1(CC(=O)O)CCC1 ZINC000147256106 CG For-Sale Mild EPHX2 35 50 CCCCCCCCNC(=O)NC1(CC(=O)O)CCC1 ZINC000147256106 CG For-Sale Mild ASAH1 52 30 CCCOc1cccc(C(=O)N2CC[C@@H](N)[C@@H](CC)C2)c1 ZINC000147256122 CF On-Demand Anodyne L3MBTL1 0 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccnc(C)n1)C2 ZINC000147256144 DD On-Demand Anodyne MTNR1A 19 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccnc(C)n1)C2 ZINC000147256144 DD On-Demand Anodyne ROCK2 31 43 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild ACE 28 40 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild OPRM1 25 48 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild MME 109 49 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild ANPEP 85 49 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild FCER2 59 36 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild PAPA1_CARPA 55 36 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild CPA1 46 35 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild SLC15A1 0 43 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild NPFFR2 46 36 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild CTRB1 31 42 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild TACR3 15 40 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild CAPNS1 52 33 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild HLA-DRB1 52 33 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild DNPEP 0 45 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild CAPN1 47 38 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild CAPN2 45 32 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild LAP3 49 45 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild FPR1 15 40 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild NPR 46 41 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild AMP1_PLAFQ 97 55 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild SLC15A2 0 41 NC(=O)NCCNC(=O)[C@@H](Cc1ccccc1)/C(N)=N/O ZINC000147256179 CB For-Sale Mild NPFFR1 67 36 CCC[C@H](CCN)CCC(=O)NN(C)C ZINC000147256187 BD For-Sale Reactive KDM7A 0 43 CC[C@@](C)(NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147256198 CE For-Sale Anodyne GPR88 0 45 C[C@H](CNS(=O)(=O)c1ccc(O)c([N+](=O)[O-])c1)CC(=O)O ZINC000147256207 DC For-Sale Bother CASP3 22 41 C[C@H](CNS(=O)(=O)c1ccc(O)c([N+](=O)[O-])c1)CC(=O)O ZINC000147256207 DC For-Sale Bother COLA 76 34 C[C@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147256222 CF For-Sale Anodyne PREP 112 37 CC(C)Oc1ccc(-c2cnc(-c3ccc(CN4CC(C(=O)O)C4)cc3)s2)cc1 ZINC000147256236 HJ For-Sale Anodyne ACACB 32 40 CC(C)Oc1ccc(-c2cnc(-c3ccc(CN4CC(C(=O)O)C4)cc3)s2)cc1 ZINC000147256236 HJ For-Sale Anodyne S1PR4 25 63 CC(C)Oc1ccc(-c2cnc(-c3ccc(CN4CC(C(=O)O)C4)cc3)s2)cc1 ZINC000147256236 HJ For-Sale Anodyne S1PR3 19 54 CC(C)Oc1ccc(-c2cnc(-c3ccc(CN4CC(C(=O)O)C4)cc3)s2)cc1 ZINC000147256236 HJ For-Sale Anodyne S1PR1 68 70 CC(C)Oc1ccc(-c2cnc(-c3ccc(CN4CC(C(=O)O)C4)cc3)s2)cc1 ZINC000147256236 HJ For-Sale Anodyne S1PR5 52 63 CC(C)Oc1ccc(-c2cnc(-c3ccc(CN4CC(C(=O)O)C4)cc3)s2)cc1 ZINC000147256236 HJ For-Sale Anodyne LUCI_LUCLA 16 41 CCCCCCCCNC(=O)NC[C@@H](CC(C)C)C(=O)O ZINC000147256264 DG For-Sale Mild CPT1A 22 43 CCCCCCCCNC(=O)NC[C@@H](CC(C)C)C(=O)O ZINC000147256264 DG For-Sale Mild EPHX2 52 49 CCCCCCCCNC(=O)NC[C@@H](CC(C)C)C(=O)O ZINC000147256264 DG For-Sale Mild Q6UB75_PIG 0 42 CCCCCCCCNC(=O)NC[C@@H](CC(C)C)C(=O)O ZINC000147256264 DG For-Sale Mild ASAH1 60 31 CCCCCCCCNC(=O)NC[C@@H](CC(C)C)C(=O)O ZINC000147256264 DG For-Sale Mild NOD1 46 37 COCc1nc(C(=O)Nc2ccccc2C(=O)N2CCCCC2)cs1 ZINC000147256286 FG On-Demand Anodyne NPSR1 17 56 COCc1nc(C(=O)Nc2ccccc2C(=O)N2CCCCC2)cs1 ZINC000147256286 FG On-Demand Anodyne TRPC6 45 32 N#CC1CCN(C(=O)c2ccc3c(c2)S(=O)(=O)c2ccccc2C3=O)CC1 ZINC000147256291 GE On-Demand Mild MAOA 15 50 N#CC1CCN(C(=O)c2ccc3c(c2)S(=O)(=O)c2ccccc2C3=O)CC1 ZINC000147256291 GE On-Demand Mild L3MBTL3 57 36 O=S(=O)(N[C@H]1C[C@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256299 HE On-Demand Anodyne EPHX2 22 41 O=S(=O)(N[C@H]1C[C@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256299 HE On-Demand Anodyne TGM2 59 48 O=S(=O)(N[C@H]1C[C@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256299 HE On-Demand Anodyne F13A1 86 45 O=S(=O)(N[C@H]1C[C@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256299 HE On-Demand Anodyne NAMPT 29 46 CS(=O)(=O)c1cc(C(=O)Nc2ccn(Cc3ccccc3)n2)cc([N+](=O)[O-])c1 ZINC000147256304 HE On-Demand Bother GCK 22 41 Cc1ccc(CNCCCCC(C)C)cc1 ZINC000147256312 BH For-Sale Anodyne FDFT1 0 42 Cc1ccc(CNCCCCC(C)C)cc1 ZINC000147256312 BH For-Sale Anodyne S1PR2 39 42 Cc1ccc(CNCCCCC(C)C)cc1 ZINC000147256312 BH For-Sale Anodyne LEF 94 47 Cc1ccc(CNCCCCC(C)C)cc1 ZINC000147256312 BH For-Sale Anodyne GPM3 0 70 O=C(COc1ccc(Cl)c(F)c1)c1ccc(Br)s1 ZINC000147256321 EJ For-Sale Anodyne ERCC5 23 42 CC[C@@H]1CN(C(=O)c2ccc(C)c(O)c2)CC[C@@H]1N ZINC000147256347 CD On-Demand Anodyne L3MBTL3 67 37 CC[C@](C)(NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147256390 CE For-Sale Anodyne GPR88 0 45 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild ACE 28 40 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild OPRM1 25 48 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild MME 109 49 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild ANPEP 85 49 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild FCER2 59 36 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild PAPA1_CARPA 55 36 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild CPA1 46 35 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild SLC15A1 0 43 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild NPFFR2 46 36 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild CTRB1 31 42 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild TACR3 15 40 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild CAPNS1 52 33 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild HLA-DRB1 52 33 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild DNPEP 0 45 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild CAPN1 47 38 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild CAPN2 45 32 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild LAP3 49 45 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild FPR1 15 40 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild NPR 46 41 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild AMP1_PLAFQ 97 55 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild SLC15A2 0 41 NC(=O)NCCNC(=O)[C@H](Cc1ccccc1)/C(N)=N/O ZINC000147256407 CB For-Sale Mild NPFFR1 67 36 CCC[C@@H](CCN)CCC(=O)NN(C)C ZINC000147256413 BD For-Sale Reactive KDM7A 0 43 C[C@@H](CNS(=O)(=O)c1ccc(O)c([N+](=O)[O-])c1)CC(=O)O ZINC000147256417 DC For-Sale Bother CASP3 22 41 C[C@@H](CNS(=O)(=O)c1ccc(O)c([N+](=O)[O-])c1)CC(=O)O ZINC000147256417 DC For-Sale Bother COLA 76 34 CCCCCCCCNC(=O)NC[C@H](CC(C)C)C(=O)O ZINC000147256489 DG For-Sale Mild CPT1A 22 43 CCCCCCCCNC(=O)NC[C@H](CC(C)C)C(=O)O ZINC000147256489 DG For-Sale Mild EPHX2 52 49 CCCCCCCCNC(=O)NC[C@H](CC(C)C)C(=O)O ZINC000147256489 DG For-Sale Mild Q6UB75_PIG 0 42 CCCCCCCCNC(=O)NC[C@H](CC(C)C)C(=O)O ZINC000147256489 DG For-Sale Mild ASAH1 60 31 CCCCCCCCNC(=O)NC[C@H](CC(C)C)C(=O)O ZINC000147256489 DG For-Sale Mild NOD1 46 37 O=S(=O)(N[C@@H]1C[C@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256507 HE On-Demand Anodyne EPHX2 22 41 O=S(=O)(N[C@@H]1C[C@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256507 HE On-Demand Anodyne TGM2 59 48 O=S(=O)(N[C@@H]1C[C@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256507 HE On-Demand Anodyne F13A1 86 45 O=S(=O)(N[C@@H]1C[C@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256507 HE On-Demand Anodyne NAMPT 29 46 CCNc1cn2ccnc2c(Oc2ccc(Cl)cc2C)n1 ZINC000147256515 DH For-Sale Anodyne HIVRT 0 55 CCc1ncc(C(=O)N(Cc2cccs2)Cc2ccccc2OC)s1 ZINC000147256530 FJ On-Demand Anodyne ADAM17 15 40 CS(=O)(=O)c1cc(C(=O)N2CCC[C@@H]2c2cccc(Cl)c2)cc([N+](=O)[O-])c1 ZINC000147256550 HH On-Demand Bother MDM2 49 31 CC[C@H]1CN(C(=O)c2ccc(C)c(O)c2)CC[C@@H]1N ZINC000147256574 CD On-Demand Anodyne L3MBTL3 67 37 CC(=O)Nc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147256576 CE On-Demand Mild AVPR1A 44 36 CC(=O)Nc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147256576 CE On-Demand Mild EPHX2 24 45 CC(=O)Nc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147256576 CE On-Demand Mild L3MBTL1 0 43 CC(=O)Nc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147256576 CE On-Demand Mild L3MBTL3 85 43 CC(=O)Nc1ccc(C(=O)N2CCC(C#N)CC2)cc1 ZINC000147256576 CE On-Demand Mild MBTD1 0 42 N#Cc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147256590 DD On-Demand Mild DHODH 17 40 N#Cc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147256590 DD On-Demand Mild ENV 40 33 CC[C@@](C)(NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147256605 CE For-Sale Anodyne GPR88 0 45 O=S(=O)(N[C@@H]1C[C@@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256706 HE On-Demand Anodyne EPHX2 22 41 O=S(=O)(N[C@@H]1C[C@@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256706 HE On-Demand Anodyne TGM2 59 48 O=S(=O)(N[C@@H]1C[C@@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256706 HE On-Demand Anodyne F13A1 86 45 O=S(=O)(N[C@@H]1C[C@@H]1c1ccccc1)c1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147256706 HE On-Demand Anodyne NAMPT 29 46 CS(=O)(=O)c1cc(C(=O)N2CCC[C@H]2c2cccc(Cl)c2)cc([N+](=O)[O-])c1 ZINC000147256717 HH On-Demand Bother MDM2 49 31 CCCCCCCCNC(=O)N(CCOC)CC(=O)O ZINC000147256746 CE For-Sale Mild EPHX2 23 43 CCCCCCCCNC(=O)N(CCOC)CC(=O)O ZINC000147256746 CE For-Sale Mild ASAH1 55 31 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@H](C)C3)cc2)s1 ZINC000147256750 GG On-Demand Anodyne TGM2 54 37 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@H](C)C3)cc2)s1 ZINC000147256750 GG On-Demand Anodyne F13A1 74 38 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@H](C)C3)cc2)s1 ZINC000147256750 GG On-Demand Anodyne MERTK 29 40 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@H](C)C3)cc2)s1 ZINC000147256750 GG On-Demand Anodyne NAMPT 43 54 CC[C@@H]1CN(C(=O)c2ccc(C)c(O)c2)CC[C@H]1N ZINC000147256784 CD On-Demand Anodyne L3MBTL3 67 37 N#Cc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147256802 DD On-Demand Mild DHODH 17 40 N#Cc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147256802 DD On-Demand Mild ENV 40 33 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3ccccc3Cl)c2)CC1 ZINC000147256805 HH On-Demand Mild PREP 25 40 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3ccccc3Cl)c2)CC1 ZINC000147256805 HH On-Demand Mild ST14 78 39 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3ccccc3Cl)c2)CC1 ZINC000147256805 HH On-Demand Mild SFRP1 95 43 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3ccccc3Cl)c2)CC1 ZINC000147256805 HH On-Demand Mild WNT3 66 35 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3ccccc3Cl)c2)CC1 ZINC000147256805 HH On-Demand Mild L3MBTL3 66 42 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3ccccc3Cl)c2)CC1 ZINC000147256805 HH On-Demand Mild TMPRSS6 55 36 CCCS(=O)(=O)Nc1ccccc1C(=O)N(C)CCCCc1ccccc1 ZINC000147256858 GH On-Demand Anodyne LIMK2 40 38 CN1CCN(C(=O)C[C@@H]2CNc3ccccc32)CC1 ZINC000147256908 CD For-Sale Anodyne SSTR1 40 39 CCCCCCCCNC(=O)N[C@H](C(=O)O)C1CC1 ZINC000147256949 CF For-Sale Mild CPT1A 40 49 CCCCCCCCNC(=O)N[C@H](C(=O)O)C1CC1 ZINC000147256949 CF For-Sale Mild EPHX2 32 50 CCCCCCCCNC(=O)N[C@H](C(=O)O)C1CC1 ZINC000147256949 CF For-Sale Mild GNAI1 0 47 CCCCCCCCNC(=O)N[C@H](C(=O)O)C1CC1 ZINC000147256949 CF For-Sale Mild GNAI3 0 47 CCCCCCCCNC(=O)N[C@H](C(=O)O)C1CC1 ZINC000147256949 CF For-Sale Mild GNAO1 0 47 CCCCCCCCNC(=O)N[C@H](C(=O)O)C1CC1 ZINC000147256949 CF For-Sale Mild ASAH1 60 33 CCCCCCCCNC(=O)N[C@H](C(=O)O)C1CC1 ZINC000147256949 CF For-Sale Mild NOD1 46 37 CCCCNCCCCC(C)C ZINC000147256953 AG For-Sale Anodyne ADH1A 0 42 CCCCNCCCCC(C)C ZINC000147256953 AG For-Sale Anodyne S1PR3 15 42 CCCCNCCCCC(C)C ZINC000147256953 AG For-Sale Anodyne S1PR2 36 42 CCCCNCCCCC(C)C ZINC000147256953 AG For-Sale Anodyne FPPS 43 38 CCCCNCCCCC(C)C ZINC000147256953 AG For-Sale Anodyne SPPS 42 38 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@@H](C)C3)cc2)s1 ZINC000147256958 GG On-Demand Anodyne TGM2 54 37 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@@H](C)C3)cc2)s1 ZINC000147256958 GG On-Demand Anodyne F13A1 74 38 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@@H](C)C3)cc2)s1 ZINC000147256958 GG On-Demand Anodyne MERTK 29 40 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@@H](C)C3)cc2)s1 ZINC000147256958 GG On-Demand Anodyne NAMPT 43 54 CC(=O)c1ccccc1OCCOc1ccc(Cl)c(F)c1 ZINC000147256996 DI For-Sale Anodyne PPARA 22 40 CC(=O)c1ccccc1OCCOc1ccc(Cl)c(F)c1 ZINC000147256996 DI For-Sale Anodyne TSPO 40 32 CC[C@H]1CN(C(=O)c2ccc(C)c(O)c2)CC[C@H]1N ZINC000147256997 CD On-Demand Anodyne L3MBTL3 67 37 CCOC(=O)CCCN1CCC[C@@H](CC)C1 ZINC000147257009 BE On-Demand Anodyne SLC6A1 52 34 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3cccc(Cl)c3)c2)CC1 ZINC000147257024 HH On-Demand Mild PLG 17 40 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3cccc(Cl)c3)c2)CC1 ZINC000147257024 HH On-Demand Mild ST14 79 40 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3cccc(Cl)c3)c2)CC1 ZINC000147257024 HH On-Demand Mild AKR1C3 22 41 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3cccc(Cl)c3)c2)CC1 ZINC000147257024 HH On-Demand Mild SFRP1 34 45 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3cccc(Cl)c3)c2)CC1 ZINC000147257024 HH On-Demand Mild L3MBTL3 46 40 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)Nc3cccc(Cl)c3)c2)CC1 ZINC000147257024 HH On-Demand Mild TMPRSS6 55 36 C[C@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257044 CD On-Demand Anodyne TBXA2R 59 43 C[C@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257044 CD On-Demand Anodyne TBXAS1 34 43 C[C@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257044 CD On-Demand Anodyne MMP2 17 49 C[C@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257044 CD On-Demand Anodyne MMP9 15 53 C[C@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257044 CD On-Demand Anodyne MMP7 16 53 C[C@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257044 CD On-Demand Anodyne IDO1 15 40 C[C@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257044 CD On-Demand Anodyne OXER1 40 34 O=C1CC[C@@H](C(=O)N[C@@H]2CN3CCC2CC3)CN1 ZINC000147257083 CB For-Sale Anodyne HTR3A 17 42 O=C1CC[C@@H](C(=O)N[C@@H]2CN3CCC2CC3)CN1 ZINC000147257083 CB For-Sale Anodyne CHRNA7 15 43 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C1CC1 ZINC000147257117 CF For-Sale Mild CPT1A 40 49 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C1CC1 ZINC000147257117 CF For-Sale Mild EPHX2 32 50 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C1CC1 ZINC000147257117 CF For-Sale Mild GNAI1 0 47 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C1CC1 ZINC000147257117 CF For-Sale Mild GNAI3 0 47 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C1CC1 ZINC000147257117 CF For-Sale Mild GNAO1 0 47 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C1CC1 ZINC000147257117 CF For-Sale Mild ASAH1 60 33 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C1CC1 ZINC000147257117 CF For-Sale Mild NOD1 46 37 CN1CCN(C(=O)C[C@H]2CNc3ccccc32)CC1 ZINC000147257134 CD For-Sale Anodyne SSTR1 40 39 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2Cc2c(F)cccc2Cl)cc1 ZINC000147257144 GG On-Demand Anodyne CPT1A 127 49 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2Cc2c(F)cccc2Cl)cc1 ZINC000147257144 GG On-Demand Anodyne CPT2 49 44 COCc1nc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@H](C)C3)cc2)cs1 ZINC000147257197 HF On-Demand Anodyne TGM2 54 34 COCc1nc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@H](C)C3)cc2)cs1 ZINC000147257197 HF On-Demand Anodyne F13A1 84 36 COCc1nc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@H](C)C3)cc2)cs1 ZINC000147257197 HF On-Demand Anodyne NAMPT 28 49 COCc1nc(C(=O)Nc2ccc(S(=O)(=O)N3CCC[C@H](C)C3)cc2)cs1 ZINC000147257197 HF On-Demand Anodyne TRPC6 48 36 COc1ccccc1NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147257246 GF On-Demand Mild PLG 19 40 COc1ccccc1NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147257246 GF On-Demand Mild ST14 82 40 COc1ccccc1NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147257246 GF On-Demand Mild SFRP1 55 36 COc1ccccc1NS(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147257246 GF On-Demand Mild TMPRSS6 64 38 C[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257254 CD On-Demand Anodyne TBXA2R 59 43 C[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257254 CD On-Demand Anodyne TBXAS1 34 43 C[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257254 CD On-Demand Anodyne MMP2 17 49 C[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257254 CD On-Demand Anodyne MMP9 15 53 C[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257254 CD On-Demand Anodyne MMP7 16 53 C[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257254 CD On-Demand Anodyne IDO1 15 40 C[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147257254 CD On-Demand Anodyne OXER1 40 34 O=C1CC[C@H](C(=O)N[C@@H]2CN3CCC2CC3)CN1 ZINC000147257290 CB For-Sale Anodyne HTR3A 17 42 O=C1CC[C@H](C(=O)N[C@@H]2CN3CCC2CC3)CN1 ZINC000147257290 CB For-Sale Anodyne CHRNA7 15 43 CCCCCCCCNC(=O)N[C@@H](CCCOC)C(=O)O ZINC000147257322 DF For-Sale Mild FOLH1 72 55 CCCCCCCCNC(=O)N[C@@H](CCCOC)C(=O)O ZINC000147257322 DF For-Sale Mild CPT1A 41 46 CCCCCCCCNC(=O)N[C@@H](CCCOC)C(=O)O ZINC000147257322 DF For-Sale Mild C3AR1 50 34 CCCCCCCCNC(=O)N[C@@H](CCCOC)C(=O)O ZINC000147257322 DF For-Sale Mild EPHX2 57 48 CCCCCCCCNC(=O)N[C@@H](CCCOC)C(=O)O ZINC000147257322 DF For-Sale Mild ASAH1 42 30 CCCCCCCCNC(=O)N[C@@H](CCCOC)C(=O)O ZINC000147257322 DF For-Sale Mild NOD1 109 48 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2Cc2c(F)cccc2Cl)cc1 ZINC000147257377 GG On-Demand Anodyne CPT1A 127 49 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2Cc2c(F)cccc2Cl)cc1 ZINC000147257377 GG On-Demand Anodyne CPT2 49 44 CC(C)C[C@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147257385 DI On-Demand Anodyne BMP1 56 39 CC(C)C[C@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147257385 DI On-Demand Anodyne PTGER3 48 37 CC(C)C[C@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147257385 DI On-Demand Anodyne CYP3A4 20 46 CCOc1ccc(-c2nnc(SCC(=O)Nc3cccc(C)c3C)[nH]2)cc1 ZINC000147257404 GI Annotated Anodyne ENPP1 68 34 C[C@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257457 CD On-Demand Anodyne HMGCR 45 37 C[C@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257457 CD On-Demand Anodyne TBXA2R 45 40 C[C@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257457 CD On-Demand Anodyne CA4 15 45 C[C@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257457 CD On-Demand Anodyne MMP2 16 49 C[C@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257457 CD On-Demand Anodyne MMP14 21 40 C[C@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257457 CD On-Demand Anodyne MMP9 17 40 C[C@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257457 CD On-Demand Anodyne MMP7 15 53 C[C@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257457 CD On-Demand Anodyne LIMK2 30 43 COc1ccc(C(=O)COc2ccc(Cl)c(F)c2)cc1Br ZINC000147257458 FJ For-Sale Anodyne PDE4D 15 41 Cc1nn(C(F)F)c(C)c1CC(=O)NCCNS(C)(=O)=O ZINC000147257468 DC On-Demand Anodyne P2RX7 36 43 O=C1CC[C@@H](C(=O)N[C@H]2CN3CCC2CC3)CN1 ZINC000147257497 CB For-Sale Anodyne HTR3A 17 42 O=C1CC[C@@H](C(=O)N[C@H]2CN3CCC2CC3)CN1 ZINC000147257497 CB For-Sale Anodyne CHRNA7 15 43 CCCCCCCCNC(=O)N[C@H](CCCOC)C(=O)O ZINC000147257531 DF For-Sale Mild FOLH1 72 55 CCCCCCCCNC(=O)N[C@H](CCCOC)C(=O)O ZINC000147257531 DF For-Sale Mild CPT1A 41 46 CCCCCCCCNC(=O)N[C@H](CCCOC)C(=O)O ZINC000147257531 DF For-Sale Mild C3AR1 50 34 CCCCCCCCNC(=O)N[C@H](CCCOC)C(=O)O ZINC000147257531 DF For-Sale Mild EPHX2 57 48 CCCCCCCCNC(=O)N[C@H](CCCOC)C(=O)O ZINC000147257531 DF For-Sale Mild ASAH1 42 30 CCCCCCCCNC(=O)N[C@H](CCCOC)C(=O)O ZINC000147257531 DF For-Sale Mild NOD1 109 48 Cc1cccc(F)c1C1CCNCC1 ZINC000147257570 AF For-Sale Anodyne SLC6A2 17 59 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147257585 FE On-Demand Anodyne TSHR 55 32 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147257585 FE On-Demand Anodyne COLA 57 38 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147257585 FE On-Demand Anodyne CPT1A 53 38 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147257585 FE On-Demand Anodyne CPT2 45 34 CC(C)C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147257595 DI On-Demand Anodyne BMP1 56 39 CC(C)C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147257595 DI On-Demand Anodyne PTGER3 48 37 CC(C)C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147257595 DI On-Demand Anodyne CYP3A4 20 46 C[C@@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257652 CD On-Demand Anodyne HMGCR 45 37 C[C@@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257652 CD On-Demand Anodyne TBXA2R 45 40 C[C@@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257652 CD On-Demand Anodyne CA4 15 45 C[C@@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257652 CD On-Demand Anodyne MMP2 16 49 C[C@@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257652 CD On-Demand Anodyne MMP14 21 40 C[C@@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257652 CD On-Demand Anodyne MMP9 17 40 C[C@@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257652 CD On-Demand Anodyne MMP7 15 53 C[C@@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147257652 CD On-Demand Anodyne LIMK2 30 43 CCc1ccc(C(=O)COc2ccc(Cl)c(F)c2)cc1 ZINC000147257671 CI For-Sale Anodyne PLA2G4B 49 32 O=C1CC[C@H](C(=O)N[C@H]2CN3CCC2CC3)CN1 ZINC000147257681 CB For-Sale Anodyne HTR3A 17 42 O=C1CC[C@H](C(=O)N[C@H]2CN3CCC2CC3)CN1 ZINC000147257681 CB For-Sale Anodyne CHRNA7 15 43 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cc(C(N)=O)ccc1N1CCCCC1)C2 ZINC000147257699 HF On-Demand Anodyne ROCK2 28 44 CC(C)(C)c1nc(NN)cc(NCc2ccc(F)cc2)n1 ZINC000147257747 CF For-Sale Anodyne PETD 0 45 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild THRA 37 41 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild FOLH1 22 43 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild RARB 27 48 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild THRB 0 44 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild CCR3 22 41 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild SCN2A 18 40 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild PLA2G4A 21 43 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild CPT1A 37 40 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild PLA2G4B 53 43 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild SOAT1 23 40 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild FAAH 21 43 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild S1PR2 47 37 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild EPHX2 47 64 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild CA9 17 40 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild ASAH1 100 39 CCCCCCCCNC(=O)Nc1ccc(C(=O)O)cc1 ZINC000147257749 CH For-Sale Mild P96878_MYCTU 16 43 FC(F)CNC[C@H]1CCCNC1 ZINC000147257775 AC For-Sale Anodyne CPN1 0 40 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147257783 FE On-Demand Anodyne TSHR 55 32 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147257783 FE On-Demand Anodyne CPT1A 53 38 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147257783 FE On-Demand Anodyne CPT2 45 34 COC(=O)C[C@]1(O)OO[C@@](C)(C[C@H](C)CCCCCCCCc2ccccc2)C[C@H]1C ZINC000147257813 IK Annotated Reactive NAAA 36 41 O=C(NCc1ccc(F)cc1)c1cccnc1F ZINC000147257865 BE On-Demand Anodyne CALCA 0 44 O=C(NCc1ccc(F)cc1)c1cccnc1F ZINC000147257865 BE On-Demand Anodyne EGLN1 0 48 O=C(NCc1ccc(F)cc1)c1cccnc1F ZINC000147257865 BE On-Demand Anodyne NAMPT 54 40 O=C(NCc1ccc(F)cc1)c1cccnc1F ZINC000147257865 BE On-Demand Anodyne Q76353_9HIV1 0 43 O=C(COc1ccc(Cl)c(F)c1)c1ccc(Cl)cc1Cl ZINC000147257897 EK For-Sale Anodyne ALPL 40 33 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild FABP2 0 45 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild CPT1A 42 41 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild DNM1 0 47 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild FAAH 0 43 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild EPHX2 46 61 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild FABP5 15 45 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild GNAI1 0 41 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild GNAI3 0 41 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild GNAO1 0 41 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild ASAH1 89 34 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild SLC22A20 0 45 CCCCCCCCNC(=O)N(C)CC(=O)O ZINC000147257956 BE For-Sale Mild CQSS 53 32 FC(F)CNC[C@@H]1CCCNC1 ZINC000147257961 AC For-Sale Anodyne CPN1 0 40 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147257994 FE On-Demand Anodyne TSHR 55 32 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147257994 FE On-Demand Anodyne COLA 57 38 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147257994 FE On-Demand Anodyne CPT1A 53 38 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147257994 FE On-Demand Anodyne CPT2 45 34 NS(=O)(=O)c1cc(F)ccc1OCCc1ccncc1 ZINC000147258113 CD For-Sale Anodyne CA14 22 42 BrC1C[C@H]2CC[C@H](C1)N2Cc1ccc2ncccc2c1 ZINC000147258114 EI For-Sale Reactive CCR3 26 41 BrC1C[C@H]2CC[C@H](C1)N2Cc1ccc2ncccc2c1 ZINC000147258114 EI For-Sale Reactive MET 0 45 CCCCO[C@@H](C)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147258119 FH On-Demand Anodyne HRH3 30 43 CCCCO[C@@H](C)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147258119 FH On-Demand Anodyne LSS 20 45 CCCCO[C@@H](C)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147258119 FH On-Demand Anodyne DPP7 34 40 CCCCCCCCNC(=O)N[C@@H](CCCC)C(=O)O ZINC000147258131 CG For-Sale Mild FOLH1 79 59 CCCCCCCCNC(=O)N[C@@H](CCCC)C(=O)O ZINC000147258131 CG For-Sale Mild CPT1A 43 52 CCCCCCCCNC(=O)N[C@@H](CCCC)C(=O)O ZINC000147258131 CG For-Sale Mild C3AR1 56 34 CCCCCCCCNC(=O)N[C@@H](CCCC)C(=O)O ZINC000147258131 CG For-Sale Mild NAALAD2 55 42 CCCCCCCCNC(=O)N[C@@H](CCCC)C(=O)O ZINC000147258131 CG For-Sale Mild EPHX2 25 54 CCCCCCCCNC(=O)N[C@@H](CCCC)C(=O)O ZINC000147258131 CG For-Sale Mild ASAH1 87 35 CCCCCCCCNC(=O)N[C@@H](CCCC)C(=O)O ZINC000147258131 CG For-Sale Mild NOD1 119 54 CCCCCCCCNC(=O)N[C@@H](CCCC)C(=O)O ZINC000147258131 CG For-Sale Mild CQSS 51 33 NC(=O)NCCNC(=O)[C@H](/C(N)=N/O)c1ccccc1 ZINC000147258138 CB For-Sale Mild C3AR1 54 34 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147258183 FE On-Demand Anodyne TSHR 55 32 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147258183 FE On-Demand Anodyne COLA 57 38 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147258183 FE On-Demand Anodyne CPT1A 53 38 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147258183 FE On-Demand Anodyne CPT2 45 34 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147258265 DD On-Demand Anodyne CA2 27 46 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147258265 DD On-Demand Anodyne CA1 35 44 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147258265 DD On-Demand Anodyne CA4 35 53 CC(=O)Nc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147258265 DD On-Demand Anodyne IDO1 40 45 BrC1C[C@@H]2CC[C@H](C1)N2Cc1ccc2ncccc2c1 ZINC000147258326 EI For-Sale Reactive CCR3 26 41 BrC1C[C@@H]2CC[C@H](C1)N2Cc1ccc2ncccc2c1 ZINC000147258326 EI For-Sale Reactive MET 0 45 CCCCO[C@H](C)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147258331 FH On-Demand Anodyne HRH3 30 43 CCCCO[C@H](C)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147258331 FH On-Demand Anodyne LSS 20 45 CCCCO[C@H](C)C(=O)N1CCCN(Cc2ccc(Cl)cc2)CC1 ZINC000147258331 FH On-Demand Anodyne DPP7 34 40 CCCCCCCCNC(=O)N[C@H](CCCC)C(=O)O ZINC000147258352 CG For-Sale Mild FOLH1 79 59 CCCCCCCCNC(=O)N[C@H](CCCC)C(=O)O ZINC000147258352 CG For-Sale Mild CPT1A 43 52 CCCCCCCCNC(=O)N[C@H](CCCC)C(=O)O ZINC000147258352 CG For-Sale Mild C3AR1 56 34 CCCCCCCCNC(=O)N[C@H](CCCC)C(=O)O ZINC000147258352 CG For-Sale Mild NAALAD2 55 42 CCCCCCCCNC(=O)N[C@H](CCCC)C(=O)O ZINC000147258352 CG For-Sale Mild EPHX2 25 54 CCCCCCCCNC(=O)N[C@H](CCCC)C(=O)O ZINC000147258352 CG For-Sale Mild ASAH1 87 35 CCCCCCCCNC(=O)N[C@H](CCCC)C(=O)O ZINC000147258352 CG For-Sale Mild NOD1 119 54 CCCCCCCCNC(=O)N[C@H](CCCC)C(=O)O ZINC000147258352 CG For-Sale Mild CQSS 51 33 NC(=O)NCCNC(=O)[C@@H](/C(N)=N/O)c1ccccc1 ZINC000147258389 CB For-Sale Mild C3AR1 54 34 COc1ccc2c(c1)CCC[C@H]2NCCCCC(C)C ZINC000147258393 CI For-Sale Anodyne GRIN2B 0 42 COc1ccc2c(c1)CCC[C@H]2NCCCCC(C)C ZINC000147258393 CI For-Sale Anodyne EBP 28 44 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc(Cn2cccn2)cc1 ZINC000147258396 FF On-Demand Anodyne AGTR1 23 41 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc(Cn2cccn2)cc1 ZINC000147258396 FF On-Demand Anodyne F10 15 43 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc(Cn2cccn2)cc1 ZINC000147258396 FF On-Demand Anodyne KIT 17 43 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc(Cn2cccn2)cc1 ZINC000147258396 FF On-Demand Anodyne PLA2G7 36 41 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc(Cn2cccn2)cc1 ZINC000147258396 FF On-Demand Anodyne FLT1 20 43 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc(Cn2cccn2)cc1 ZINC000147258396 FF On-Demand Anodyne BRAF 27 43 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc(Cn2cccn2)cc1 ZINC000147258396 FF On-Demand Anodyne NOD2 40 34 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCCC3)c2)CC1 ZINC000147258415 FE On-Demand Mild CACNA1B 28 43 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCCC3)c2)CC1 ZINC000147258415 FE On-Demand Mild PREP 25 46 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCCC3)c2)CC1 ZINC000147258415 FE On-Demand Mild EPHX2 15 49 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCCC3)c2)CC1 ZINC000147258415 FE On-Demand Mild AKR1C3 67 46 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCCC3)c2)CC1 ZINC000147258415 FE On-Demand Mild L3MBTL3 84 47 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147258454 DD On-Demand Anodyne CA2 27 46 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147258454 DD On-Demand Anodyne CA1 35 44 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147258454 DD On-Demand Anodyne CA4 35 53 CC(=O)Nc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147258454 DD On-Demand Anodyne IDO1 40 45 CN(Cc1ccc(C(=O)NC2CC2)cc1)C(=O)c1cc(F)ccc1NS(C)(=O)=O ZINC000147258456 HE On-Demand Anodyne MAPK14 34 42 CN(Cc1ccc(C(=O)NC2CC2)cc1)C(=O)c1cc(F)ccc1NS(C)(=O)=O ZINC000147258456 HE On-Demand Anodyne TRPV1 40 39 CN(Cc1ccc(C(=O)NC2CC2)cc1)C(=O)c1cc(F)ccc1NS(C)(=O)=O ZINC000147258456 HE On-Demand Anodyne MCHR1 16 42 CN(Cc1ccc(C(=O)NC2CC2)cc1)C(=O)c1cc(F)ccc1NS(C)(=O)=O ZINC000147258456 HE On-Demand Anodyne LIMK2 21 41 O=C(O)C1(NCc2cccc(C(F)(F)F)c2)CCC1 ZINC000147258483 CF On-Demand Anodyne PHES 0 42 NC(=O)c1c(N)ccc2ccccc12 ZINC000147258509 AD For-Sale Anodyne CYP73A1 0 48 BrC1C[C@@H]2CC[C@@H](C1)N2Cc1ccc2ncccc2c1 ZINC000147258530 EI For-Sale Reactive CCR3 26 41 BrC1C[C@@H]2CC[C@@H](C1)N2Cc1ccc2ncccc2c1 ZINC000147258530 EI For-Sale Reactive MET 0 45 CCCCCCCCNC(=O)N[C@H](CCC(N)=O)C(=O)O ZINC000147258548 DD For-Sale Mild FOLH1 78 51 CCCCCCCCNC(=O)N[C@H](CCC(N)=O)C(=O)O ZINC000147258548 DD For-Sale Mild CPT1A 27 47 CCCCCCCCNC(=O)N[C@H](CCC(N)=O)C(=O)O ZINC000147258548 DD For-Sale Mild C3AR1 59 36 CCCCCCCCNC(=O)N[C@H](CCC(N)=O)C(=O)O ZINC000147258548 DD For-Sale Mild NAALAD2 64 44 CCCCCCCCNC(=O)N[C@H](CCC(N)=O)C(=O)O ZINC000147258548 DD For-Sale Mild EPHX2 57 50 CCCCCCCCNC(=O)N[C@H](CCC(N)=O)C(=O)O ZINC000147258548 DD For-Sale Mild ASAH1 86 35 CCCCCCCCNC(=O)N[C@H](CCC(N)=O)C(=O)O ZINC000147258548 DD For-Sale Mild NOD1 120 55 CCCCCCCCNC(=O)N[C@H](CCC(N)=O)C(=O)O ZINC000147258548 DD For-Sale Mild CQSS 51 32 CCCC[C@H](NC(N)=O)C(=O)N1Cc2ccccc2[C@H](c2ccccc2)C1 ZINC000147258560 FG On-Demand Anodyne GHRHR 57 36 CCCC[C@H](NC(N)=O)C(=O)N1Cc2ccccc2[C@H](c2ccccc2)C1 ZINC000147258560 FG On-Demand Anodyne P2RY12 172 35 COc1ccc2c(c1)CCC[C@@H]2NCCCCC(C)C ZINC000147258597 CI For-Sale Anodyne GRIN2B 0 42 COc1ccc2c(c1)CCC[C@@H]2NCCCCC(C)C ZINC000147258597 CI For-Sale Anodyne EBP 28 44 CCCC[C@@H](NC(N)=O)C(=O)N1Cc2ccccc2[C@H](c2ccccc2)C1 ZINC000147258771 FG On-Demand Anodyne GHRHR 57 36 CCCC[C@@H](NC(N)=O)C(=O)N1Cc2ccccc2[C@H](c2ccccc2)C1 ZINC000147258771 FG On-Demand Anodyne P2RY12 172 35 CCCCCCCCNC(=O)N1CCC(CC(=O)O)CC1 ZINC000147258774 CG For-Sale Mild ASAH1 98 42 CCCCCCCNCCCCC(C)C ZINC000147258789 BI For-Sale Mild ADH1A 0 47 CCCCCCCNCCCCC(C)C ZINC000147258789 BI For-Sale Mild ADH7 0 44 CCCCCCCNCCCCC(C)C ZINC000147258789 BI For-Sale Mild S1PR3 21 50 CCCCCCCNCCCCC(C)C ZINC000147258789 BI For-Sale Mild S1PR2 47 50 CCCCCCCNCCCCC(C)C ZINC000147258789 BI For-Sale Mild ADH1B 0 47 CCCCCCCNCCCCC(C)C ZINC000147258789 BI For-Sale Mild ADH1C 0 47 CCCCCCCNCCCCC(C)C ZINC000147258789 BI For-Sale Mild Q8WS26_TRYCR 41 42 CCCCCCCNCCCCC(C)C ZINC000147258789 BI For-Sale Mild FPPS 0 42 CCCCCCCNCCCCC(C)C ZINC000147258789 BI For-Sale Mild SPPS 0 42 Cc1ccc(C(=O)Nc2ccccc2N2CCCCCC2)cc1[N+](=O)[O-] ZINC000147258812 FJ On-Demand Bother KCNQ2 91 44 Cc1ccc(C(=O)Nc2ccccc2N2CCCCCC2)cc1[N+](=O)[O-] ZINC000147258812 FJ On-Demand Bother HDAC1 17 45 Cc1ccc(C(=O)Nc2ccccc2N2CCCCCC2)cc1[N+](=O)[O-] ZINC000147258812 FJ On-Demand Bother CSF1R 22 57 Cc1ccc(C(=O)Nc2ccccc2N2CCCCCC2)cc1[N+](=O)[O-] ZINC000147258812 FJ On-Demand Bother TAAR1 46 55 Cc1ccc(C(=O)Nc2ccccc2N2CCCCCC2)cc1[N+](=O)[O-] ZINC000147258812 FJ On-Demand Bother WDR5 37 48 CCc1nc(CN(C)C(=O)N[C@@H](c2ccccc2)c2ccc(Cl)cc2)cs1 ZINC000147258814 GK On-Demand Anodyne UTS2 43 34 N#Cc1cccc(CNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)c1 ZINC000147258862 GF On-Demand Mild SCN3A 0 44 N#Cc1cccc(CNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)c1 ZINC000147258862 GF On-Demand Mild MAP1 40 34 N#Cc1cccc(CNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)c1 ZINC000147258862 GF On-Demand Mild SCN9A 0 46 N#Cc1cccc(CNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)c1 ZINC000147258862 GF On-Demand Mild PFK 0 45 CCCC[C@H](NC(N)=O)C(=O)N1Cc2ccccc2[C@@H](c2ccccc2)C1 ZINC000147258912 FG On-Demand Anodyne GHRHR 57 36 CCCC[C@H](NC(N)=O)C(=O)N1Cc2ccccc2[C@@H](c2ccccc2)C1 ZINC000147258912 FG On-Demand Anodyne P2RY12 172 35 CCCCCCCCNC(=O)N1[C@H](C)SC[C@@H]1C(=O)O ZINC000147258922 DF For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N1[C@H](C)SC[C@@H]1C(=O)O ZINC000147258922 DF For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N1[C@H](C)SC[C@@H]1C(=O)O ZINC000147258922 DF For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N1[C@H](C)SC[C@@H]1C(=O)O ZINC000147258922 DF For-Sale Mild ASAH1 96 39 CC[C@@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@@H]1N ZINC000147258950 CC On-Demand Anodyne SLC9A1 41 37 CC[C@@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@@H]1N ZINC000147258950 CC On-Demand Anodyne L3MBTL1 0 47 CC[C@@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@@H]1N ZINC000147258950 CC On-Demand Anodyne L3MBTL3 67 47 CC[C@@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@@H]1N ZINC000147258950 CC On-Demand Anodyne MBTD1 0 41 CC[C@@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@@H]1N ZINC000147258950 CC On-Demand Anodyne MVFR 0 43 Cc1ccc(NS(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147258958 GG On-Demand Mild LIMK2 39 43 Cc1ccc(NS(=O)(=O)c2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147258958 GG On-Demand Mild L3MBTL3 75 41 O=C(O)C1(NCCOc2ccc(F)cc2)CCC1 ZINC000147258992 CD For-Sale Anodyne DRD4 18 44 CN(C(=O)c1cccc(F)c1Cl)C(C)(C)C(=O)O ZINC000147259029 CE On-Demand Anodyne E3UJZ5_SPOLI 37 41 CCc1nc(CN(C)C(=O)N[C@H](c2ccccc2)c2ccc(Cl)cc2)cs1 ZINC000147259073 GK On-Demand Anodyne UTS2 43 34 CCCCCCCCNC(=O)N1[C@@H](C(=O)O)CS[C@@H]1C ZINC000147259119 DF For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N1[C@@H](C(=O)O)CS[C@@H]1C ZINC000147259119 DF For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N1[C@@H](C(=O)O)CS[C@@H]1C ZINC000147259119 DF For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N1[C@@H](C(=O)O)CS[C@@H]1C ZINC000147259119 DF For-Sale Mild ASAH1 96 39 CCCC[C@@H](NC(N)=O)C(=O)N1Cc2ccccc2[C@@H](c2ccccc2)C1 ZINC000147259145 FG On-Demand Anodyne GHRHR 57 36 CCCC[C@@H](NC(N)=O)C(=O)N1Cc2ccccc2[C@@H](c2ccccc2)C1 ZINC000147259145 FG On-Demand Anodyne P2RY12 172 35 CC[C@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@@H]1N ZINC000147259147 CC On-Demand Anodyne SLC9A1 41 37 CC[C@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@@H]1N ZINC000147259147 CC On-Demand Anodyne L3MBTL1 0 47 CC[C@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@@H]1N ZINC000147259147 CC On-Demand Anodyne L3MBTL3 67 47 CC[C@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@@H]1N ZINC000147259147 CC On-Demand Anodyne MBTD1 0 41 CC[C@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@@H]1N ZINC000147259147 CC On-Demand Anodyne MVFR 0 43 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)Nc3ccccc3)cc2)CC1 ZINC000147259160 FF On-Demand Mild SFRP1 83 41 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)Nc3ccccc3)cc2)CC1 ZINC000147259160 FF On-Demand Mild LIMK2 56 51 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)Nc3ccccc3)cc2)CC1 ZINC000147259160 FF On-Demand Mild WNT3 65 36 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)Nc3ccccc3)cc2)CC1 ZINC000147259160 FF On-Demand Mild L3MBTL3 77 40 COc1ccc(OCCNC2(C(=O)O)CCC2)cc1 ZINC000147259177 CD For-Sale Anodyne MMP13 19 40 COc1ccc(OCCNC2(C(=O)O)CCC2)cc1 ZINC000147259177 CD For-Sale Anodyne PLA2G4B 46 31 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2Cc2cccc(F)c2)cc1 ZINC000147259186 FF On-Demand Anodyne COLA 135 48 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2Cc2cccc(F)c2)cc1 ZINC000147259186 FF On-Demand Anodyne CPT1A 115 44 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2Cc2cccc(F)c2)cc1 ZINC000147259186 FF On-Demand Anodyne CPT2 47 36 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2Cc2cccc(F)c2)cc1 ZINC000147259186 FF On-Demand Anodyne CHRNA10 47 39 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2Cc2cccc(F)c2)cc1 ZINC000147259186 FF On-Demand Anodyne ACKR3 58 36 CN(C)C1(CNC(=O)c2cn[nH]c2N)CCCC1 ZINC000147259200 CC For-Sale Anodyne HCN1 49 30 CN(C)C1(CNC(=O)c2cn[nH]c2N)CCCC1 ZINC000147259200 CC For-Sale Anodyne HCN4 46 30 COc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1F ZINC000147259221 DD On-Demand Anodyne LEF 47 38 NNc1cc(N[C@@H]2CN3CCC2CC3)nc(C2CC2)n1 ZINC000147259294 CD For-Sale Anodyne HTR3A 17 40 NNc1cc(N[C@@H]2CN3CCC2CC3)nc(C2CC2)n1 ZINC000147259294 CD For-Sale Anodyne CHRNA7 16 40 CCCCCCCCNC(=O)N1[C@H](C)SC[C@H]1C(=O)O ZINC000147259326 DF For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N1[C@H](C)SC[C@H]1C(=O)O ZINC000147259326 DF For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N1[C@H](C)SC[C@H]1C(=O)O ZINC000147259326 DF For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N1[C@H](C)SC[C@H]1C(=O)O ZINC000147259326 DF For-Sale Mild ASAH1 96 39 CC[C@@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@H]1N ZINC000147259348 CC On-Demand Anodyne SLC9A1 41 37 CC[C@@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@H]1N ZINC000147259348 CC On-Demand Anodyne L3MBTL1 0 47 CC[C@@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@H]1N ZINC000147259348 CC On-Demand Anodyne L3MBTL3 67 47 CC[C@@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@H]1N ZINC000147259348 CC On-Demand Anodyne MBTD1 0 41 CC[C@@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@H]1N ZINC000147259348 CC On-Demand Anodyne MVFR 0 43 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2Cc2cccc(F)c2)cc1 ZINC000147259366 FF On-Demand Anodyne COLA 135 48 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2Cc2cccc(F)c2)cc1 ZINC000147259366 FF On-Demand Anodyne CPT1A 115 44 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2Cc2cccc(F)c2)cc1 ZINC000147259366 FF On-Demand Anodyne CPT2 47 36 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2Cc2cccc(F)c2)cc1 ZINC000147259366 FF On-Demand Anodyne CHRNA10 47 39 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2Cc2cccc(F)c2)cc1 ZINC000147259366 FF On-Demand Anodyne ACKR3 58 36 COc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1F ZINC000147259369 DD On-Demand Anodyne LEF 47 38 CN(C(=O)[C@@H]1C[C@@H]1c1ccccc1)C(C)(C)C(=O)O ZINC000147259404 CE For-Sale Anodyne FFAR1 0 45 CN(C(=O)[C@@H]1C[C@@H]1c1ccccc1)C(C)(C)C(=O)O ZINC000147259404 CE For-Sale Anodyne GPR88 0 50 CCOC[C@H](C)NC(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1C ZINC000147259415 FH On-Demand Anodyne LPL 42 34 CCOC[C@H](C)NC(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1C ZINC000147259415 FH On-Demand Anodyne CPT1A 43 30 CCOC[C@H](C)NC(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1C ZINC000147259415 FH On-Demand Anodyne PYGL 19 41 CCOC[C@H](C)NC(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1C ZINC000147259415 FH On-Demand Anodyne KCNK3 82 38 CCOC[C@H](C)NC(=O)Nc1cc(C(=O)Nc2ccccc2)ccc1C ZINC000147259415 FH On-Demand Anodyne KCNK9 68 38 NNc1cc(N[C@H]2CN3CCC2CC3)nc(C2CC2)n1 ZINC000147259459 CD For-Sale Anodyne HTR3A 17 40 NNc1cc(N[C@H]2CN3CCC2CC3)nc(C2CC2)n1 ZINC000147259459 CD For-Sale Anodyne CHRNA7 16 40 CC(C)NC(=O)CCOc1ccc(F)cc1S(N)(=O)=O ZINC000147259490 DC For-Sale Anodyne SDH1 0 42 CSc1nc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2s1 ZINC000147259494 FF On-Demand Anodyne PRMT3 46 34 CC(=O)Nc1ccc(-c2nc3ccncc3[nH]2)cc1 ZINC000147259513 CF On-Demand Anodyne GYRB 0 50 CC(=O)Nc1ccc(-c2nc3ccncc3[nH]2)cc1 ZINC000147259513 CF On-Demand Anodyne SCD1 29 42 CC(=O)Nc1ccc(-c2nc3ccncc3[nH]2)cc1 ZINC000147259513 CF On-Demand Anodyne SCD 0 42 O=C(CCCOc1ccc(Cl)c(F)c1)c1ccc(F)cc1 ZINC000147259519 DJ For-Sale Anodyne DRD4 0 40 O=C(CCCOc1ccc(Cl)c(F)c1)c1ccc(F)cc1 ZINC000147259519 DJ For-Sale Anodyne ERG2 18 40 CCCCCCCCNC(=O)N1[C@@H](C)SC[C@H]1C(=O)O ZINC000147259548 DF For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N1[C@@H](C)SC[C@H]1C(=O)O ZINC000147259548 DF For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N1[C@@H](C)SC[C@H]1C(=O)O ZINC000147259548 DF For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N1[C@@H](C)SC[C@H]1C(=O)O ZINC000147259548 DF For-Sale Mild ASAH1 96 39 CC[C@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@H]1N ZINC000147259552 CC On-Demand Anodyne SLC9A1 41 37 CC[C@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@H]1N ZINC000147259552 CC On-Demand Anodyne L3MBTL1 0 47 CC[C@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@H]1N ZINC000147259552 CC On-Demand Anodyne L3MBTL3 67 47 CC[C@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@H]1N ZINC000147259552 CC On-Demand Anodyne MBTD1 0 41 CC[C@H]1CN(C(=O)c2cccc(C(N)=O)c2)CC[C@H]1N ZINC000147259552 CC On-Demand Anodyne MVFR 0 43 CN(CCCOc1ccccc1)C(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147259560 GG On-Demand Anodyne LTA4H 27 42 CN(CCCOc1ccccc1)C(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147259560 GG On-Demand Anodyne PTGER3 22 42 CN(CCCOc1ccccc1)C(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147259560 GG On-Demand Anodyne CRTM 15 43 C[C@H](CNS(=O)(=O)c1cccc(C#N)c1)CC(=O)O ZINC000147259574 CC On-Demand Mild ITGA4 51 30 O=C1CC[C@@H](C(=O)Nc2c(Cl)cccc2C(F)(F)F)CN1 ZINC000147259583 DF For-Sale Anodyne SRD5A1 30 42 CC(C)(C)OC(=O)N1CCCN(C(=O)c2ccc(Br)c(C#N)c2)CC1 ZINC000147259590 HG For-Sale Anodyne HRH3 25 40 CC(C)(C)OC(=O)N1CCCN(C(=O)c2ccc(Br)c(C#N)c2)CC1 ZINC000147259590 HG For-Sale Anodyne GPR119 31 41 CSc1nc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2s1 ZINC000147259607 FF On-Demand Anodyne PRMT3 46 34 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147259644 GJ On-Demand Anodyne MAPK14 36 41 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147259644 GJ On-Demand Anodyne EPHX2 24 48 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147259644 GJ On-Demand Anodyne TAAR1 17 40 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147259644 GJ On-Demand Anodyne KDM1A 29 43 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147259644 GJ On-Demand Anodyne KCNK3 93 39 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147259644 GJ On-Demand Anodyne KCNK9 46 39 CN(C(=O)[C@H]1C[C@@H]1c1ccccc1)C(C)(C)C(=O)O ZINC000147259657 CE For-Sale Anodyne FFAR1 0 45 CN(C(=O)[C@H]1C[C@@H]1c1ccccc1)C(C)(C)C(=O)O ZINC000147259657 CE For-Sale Anodyne GPR88 0 50 CC(C)(C)c1nc(NN)cc(N[C@@H]2CN3CCC2CC3)n1 ZINC000147259696 CD For-Sale Anodyne HTR3A 17 40 CC(C)(C)c1nc(NN)cc(N[C@@H]2CN3CCC2CC3)n1 ZINC000147259696 CD For-Sale Anodyne CHRNA7 15 40 O=C1CC[C@H](C(=O)Nc2c(Cl)cccc2C(F)(F)F)CN1 ZINC000147259740 DF For-Sale Anodyne SRD5A1 30 42 CCCCCCCCNC(=O)N(CC(=O)O)C1CCCC1 ZINC000147259742 CG For-Sale Mild ACE 57 40 CCCCCCCCNC(=O)N(CC(=O)O)C1CCCC1 ZINC000147259742 CG For-Sale Mild EPHX2 29 41 CCCCCCCCNC(=O)N(CC(=O)O)C1CCCC1 ZINC000147259742 CG For-Sale Mild ASAH1 59 33 CC[C@@H]1CN(C(=O)c2ccc(C(C)(C)C)cc2)CC[C@@H]1N ZINC000147259783 CG On-Demand Anodyne L3MBTL1 0 42 CC[C@@H]1CN(C(=O)c2ccc(C(C)(C)C)cc2)CC[C@@H]1N ZINC000147259783 CG On-Demand Anodyne L3MBTL3 74 42 C[C@@H](CNS(=O)(=O)c1cccc(C#N)c1)CC(=O)O ZINC000147259789 CC On-Demand Mild ITGA4 51 30 N#CC1CCN(C(=O)Cc2ccc(-c3ccccc3)cc2)CC1 ZINC000147259800 DH On-Demand Mild DPP4 21 40 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147259821 GJ On-Demand Anodyne MAPK14 36 41 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147259821 GJ On-Demand Anodyne EPHX2 24 48 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147259821 GJ On-Demand Anodyne TAAR1 17 40 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147259821 GJ On-Demand Anodyne KDM1A 29 43 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147259821 GJ On-Demand Anodyne KCNK3 93 39 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147259821 GJ On-Demand Anodyne KCNK9 46 39 CCc1cc(S(=O)(=O)O)ccc1O ZINC000147259857 BD For-Sale Anodyne PTP1 0 44 CN(C(=O)[C@@H]1C[C@H]1c1ccccc1)C(C)(C)C(=O)O ZINC000147259863 CE For-Sale Anodyne FFAR1 0 45 CN(C(=O)[C@@H]1C[C@H]1c1ccccc1)C(C)(C)C(=O)O ZINC000147259863 CE For-Sale Anodyne GPR88 0 50 CC(C)(C)c1nc(NN)cc(N[C@H]2CN3CCC2CC3)n1 ZINC000147259929 CD For-Sale Anodyne HTR3A 17 40 CC(C)(C)c1nc(NN)cc(N[C@H]2CN3CCC2CC3)n1 ZINC000147259929 CD For-Sale Anodyne CHRNA7 15 40 CCCCCCCCNC(=O)N[C@H](C(=O)O)C(C)(C)C ZINC000147259974 CG For-Sale Mild PDF 50 40 CCCCCCCCNC(=O)N[C@H](C(=O)O)C(C)(C)C ZINC000147259974 CG For-Sale Mild CPT1A 44 51 CCCCCCCCNC(=O)N[C@H](C(=O)O)C(C)(C)C ZINC000147259974 CG For-Sale Mild EPHX2 54 48 CCCCCCCCNC(=O)N[C@H](C(=O)O)C(C)(C)C ZINC000147259974 CG For-Sale Mild ASAH1 82 35 CCCCCCCCNC(=O)N[C@H](C(=O)O)C(C)(C)C ZINC000147259974 CG For-Sale Mild NOD1 64 38 CCCCCCCCNC(=O)N[C@H](C(=O)O)C(C)(C)C ZINC000147259974 CG For-Sale Mild CQSS 49 30 COc1cc(Br)c(CNCCCCC(C)C)cc1OC ZINC000147259981 EI For-Sale Anodyne GPM3 0 43 CC[C@H]1CN(C(=O)c2ccc(C(C)(C)C)cc2)CC[C@@H]1N ZINC000147259997 CG On-Demand Anodyne L3MBTL1 0 42 CC[C@H]1CN(C(=O)c2ccc(C(C)(C)C)cc2)CC[C@@H]1N ZINC000147259997 CG On-Demand Anodyne L3MBTL3 74 42 O=C(COc1ccc(Cl)c(F)c1)c1ccc(Cl)c(Cl)c1 ZINC000147259998 EK For-Sale Anodyne KMO 0 46 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147260012 GJ On-Demand Anodyne MAPK14 36 41 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147260012 GJ On-Demand Anodyne EPHX2 24 48 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147260012 GJ On-Demand Anodyne TAAR1 17 40 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147260012 GJ On-Demand Anodyne KDM1A 29 43 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147260012 GJ On-Demand Anodyne KCNK3 93 39 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147260012 GJ On-Demand Anodyne KCNK9 46 39 CN(C(=O)[C@H]1C[C@H]1c1ccccc1)C(C)(C)C(=O)O ZINC000147260086 CE For-Sale Anodyne FFAR1 0 45 CN(C(=O)[C@H]1C[C@H]1c1ccccc1)C(C)(C)C(=O)O ZINC000147260086 CE For-Sale Anodyne GPR88 0 50 CN(Cc1cscn1)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147260118 FJ On-Demand Anodyne CYP3A4 18 44 CN(Cc1cscn1)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147260118 FJ On-Demand Anodyne UTS2 43 35 CN(C)NC(=O)c1cc(N)c2ccccc2n1 ZINC000147260162 BD For-Sale Reactive TACR3 44 38 CCCCCCCCNC(=O)N(C)C[C@@H](C)C(=O)O ZINC000147260177 CF On-Demand Mild EPHX2 29 49 CCCCCCCCNC(=O)N(C)C[C@@H](C)C(=O)O ZINC000147260177 CF On-Demand Mild ASAH1 74 32 CCCCCCCCNC(=O)N(C)C[C@@H](C)C(=O)O ZINC000147260177 CF On-Demand Mild NOD1 76 40 CC[C@@H]1CN(C(=O)c2ccc(C(C)(C)C)cc2)CC[C@H]1N ZINC000147260179 CG On-Demand Anodyne L3MBTL1 0 42 CC[C@@H]1CN(C(=O)c2ccc(C(C)(C)C)cc2)CC[C@H]1N ZINC000147260179 CG On-Demand Anodyne L3MBTL3 74 42 O=C(COc1ccc(Cl)c(F)c1)Cc1ccccc1 ZINC000147260220 CH On-Demand Anodyne PLA2G4B 69 40 O=C(COc1ccc(Cl)c(F)c1)Cc1ccccc1 ZINC000147260220 CH On-Demand Anodyne PDS 63 34 O=C(COc1ccc(Cl)c(F)c1)Cc1ccccc1 ZINC000147260220 CH On-Demand Anodyne GPR183 0 46 N[C@@H](c1sccc1Br)C1(N2CCCCC2)CCCC1 ZINC000147260267 EI For-Sale Anodyne CHRNA1 16 40 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147260274 GJ On-Demand Anodyne MAPK14 36 41 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147260274 GJ On-Demand Anodyne EPHX2 24 48 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147260274 GJ On-Demand Anodyne TAAR1 17 40 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147260274 GJ On-Demand Anodyne KDM1A 29 43 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147260274 GJ On-Demand Anodyne KCNK3 93 39 Cc1ccc(C(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147260274 GJ On-Demand Anodyne KCNK9 46 39 CN(Cc1cscn1)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147260328 FJ On-Demand Anodyne CYP3A4 18 44 CN(Cc1cscn1)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147260328 FJ On-Demand Anodyne UTS2 43 35 CCCCCCCCNC(=O)N(C)C[C@H](C)C(=O)O ZINC000147260376 CF On-Demand Mild EPHX2 29 49 CCCCCCCCNC(=O)N(C)C[C@H](C)C(=O)O ZINC000147260376 CF On-Demand Mild ASAH1 74 32 CCCCCCCCNC(=O)N(C)C[C@H](C)C(=O)O ZINC000147260376 CF On-Demand Mild NOD1 76 40 CC[C@H]1CN(C(=O)c2ccc(C(C)(C)C)cc2)CC[C@H]1N ZINC000147260391 CG On-Demand Anodyne L3MBTL1 0 42 CC[C@H]1CN(C(=O)c2ccc(C(C)(C)C)cc2)CC[C@H]1N ZINC000147260391 CG On-Demand Anodyne L3MBTL3 74 42 CC[C@@H](C)NCC(=O)NN(C)C ZINC000147260439 AB For-Sale Reactive KDM7A 0 41 NC(=O)c1cccc(CNC2(C(=O)O)CCC2)c1 ZINC000147260493 BC On-Demand Anodyne PARP15 0 43 NC(=O)c1cccc(CNC2(C(=O)O)CCC2)c1 ZINC000147260493 BC On-Demand Anodyne PARP10 0 43 N[C@H](c1sccc1Br)C1(N2CCCCC2)CCCC1 ZINC000147260513 EI For-Sale Anodyne CHRNA1 16 40 CCCCCCCCNC(=O)NC(C)(C)CC(=O)O ZINC000147260580 CF For-Sale Mild CPT1A 42 50 CCCCCCCCNC(=O)NC(C)(C)CC(=O)O ZINC000147260580 CF For-Sale Mild EPHX2 52 50 CCCCCCCCNC(=O)NC(C)(C)CC(=O)O ZINC000147260580 CF For-Sale Mild ASAH1 81 34 CCCCCCCCNC(=O)NC(C)(C)CC(=O)O ZINC000147260580 CF For-Sale Mild ACAT 0 42 COc1ccc(Cl)cc1CC1(O)CCN(C(=O)OC(C)(C)C)CC1 ZINC000147260599 FH For-Sale Anodyne COLA 38 40 CC[C@H](C)NCC(=O)NN(C)C ZINC000147260643 AB For-Sale Reactive KDM7A 0 41 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260661 CD On-Demand Anodyne DRD4 49 37 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260661 CD On-Demand Anodyne OPRD1 0 40 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260661 CD On-Demand Anodyne GRM3 18 41 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260661 CD On-Demand Anodyne CCR3 23 40 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260661 CD On-Demand Anodyne SLC18A3 24 44 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260661 CD On-Demand Anodyne MTNR1B 31 41 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260661 CD On-Demand Anodyne SCN5A 25 40 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260661 CD On-Demand Anodyne L3MBTL1 0 44 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260661 CD On-Demand Anodyne L3MBTL3 35 40 Cc1ccc(NS(C)(=O)=O)c(C(=O)N(C)CCCCc2ccccc2)c1 ZINC000147260664 FG On-Demand Anodyne LIMK2 39 40 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)N(C)CC(=O)N2CCCC2)cc1 ZINC000147260676 HD On-Demand Anodyne NAMPT 48 39 Cc1nc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2s1 ZINC000147260678 EE On-Demand Anodyne LDHA 39 42 Cc1nc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2s1 ZINC000147260678 EE On-Demand Anodyne FYN 17 40 Cc1nc2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2s1 ZINC000147260678 EE On-Demand Anodyne PRMT3 48 35 CC[C@@H](c1cccc(C)n1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147260722 KK Annotated Anodyne TP53 45 70 CC[C@@H](c1cccc(C)n1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147260722 KK Annotated Anodyne MDM2 254 70 CCCCCCCCNC(=O)N[C@@H](CC)C(=O)O ZINC000147260723 CF For-Sale Mild FOLH1 61 50 CCCCCCCCNC(=O)N[C@@H](CC)C(=O)O ZINC000147260723 CF For-Sale Mild CPT1A 43 54 CCCCCCCCNC(=O)N[C@@H](CC)C(=O)O ZINC000147260723 CF For-Sale Mild EPHX2 26 53 CCCCCCCCNC(=O)N[C@@H](CC)C(=O)O ZINC000147260723 CF For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N[C@@H](CC)C(=O)O ZINC000147260723 CF For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N[C@@H](CC)C(=O)O ZINC000147260723 CF For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N[C@@H](CC)C(=O)O ZINC000147260723 CF For-Sale Mild ASAH1 88 36 CCCCCCCCNC(=O)N[C@@H](CC)C(=O)O ZINC000147260723 CF For-Sale Mild NOD1 96 46 CCCCCCCCNC(=O)N[C@@H](CC)C(=O)O ZINC000147260723 CF For-Sale Mild CQSS 55 34 CCCCO[C@@H](C)C(=O)N(C)Cc1nc2ccccc2[nH]1 ZINC000147260759 CF On-Demand Anodyne CACNA1G 31 43 CCCCCCCCCCSC(C)(C)C ZINC000147260760 BK For-Sale Mild EST1_PIG 51 38 O=C(Cc1ccc(F)cc1)NNC(=O)Nc1nc(CN2CCCCC2)cs1 ZINC000147260821 GF On-Demand Reactive CCR3 60 41 Cc1nc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2s1 ZINC000147260874 EE On-Demand Anodyne LDHA 39 42 Cc1nc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2s1 ZINC000147260874 EE On-Demand Anodyne FYN 17 40 Cc1nc2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2s1 ZINC000147260874 EE On-Demand Anodyne PRMT3 48 35 COc1cccc(Nc2nc(-c3ccc4cn[nH]c4c3)cn3ccnc23)c1 ZINC000147260875 FI For-Sale Anodyne SYK 15 76 COc1cccc(Nc2nc(-c3ccc4cn[nH]c4c3)cn3ccnc23)c1 ZINC000147260875 FI For-Sale Anodyne ROCK2 20 40 COc1cccc(Nc2nc(-c3ccc4cn[nH]c4c3)cn3ccnc23)c1 ZINC000147260875 FI For-Sale Anodyne EPHB4 51 40 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260885 CD On-Demand Anodyne DRD4 49 37 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260885 CD On-Demand Anodyne OPRD1 0 40 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260885 CD On-Demand Anodyne GRM3 18 41 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260885 CD On-Demand Anodyne CCR3 23 40 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260885 CD On-Demand Anodyne SLC18A3 24 44 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260885 CD On-Demand Anodyne MTNR1B 31 41 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260885 CD On-Demand Anodyne SCN5A 25 40 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260885 CD On-Demand Anodyne L3MBTL1 0 44 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@@H]1N ZINC000147260885 CD On-Demand Anodyne L3MBTL3 35 40 NC(=O)c1ccsc1NC(=O)c1cccc2c1OCCN2 ZINC000147260906 DD For-Sale Anodyne MAPK8 23 50 CCCCCCCCNC(=O)N[C@H](CC)C(=O)O ZINC000147260922 CF For-Sale Mild FOLH1 61 50 CCCCCCCCNC(=O)N[C@H](CC)C(=O)O ZINC000147260922 CF For-Sale Mild CPT1A 43 54 CCCCCCCCNC(=O)N[C@H](CC)C(=O)O ZINC000147260922 CF For-Sale Mild EPHX2 26 53 CCCCCCCCNC(=O)N[C@H](CC)C(=O)O ZINC000147260922 CF For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)N[C@H](CC)C(=O)O ZINC000147260922 CF For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)N[C@H](CC)C(=O)O ZINC000147260922 CF For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)N[C@H](CC)C(=O)O ZINC000147260922 CF For-Sale Mild ASAH1 88 36 CCCCCCCCNC(=O)N[C@H](CC)C(=O)O ZINC000147260922 CF For-Sale Mild NOD1 96 46 CCCCCCCCNC(=O)N[C@H](CC)C(=O)O ZINC000147260922 CF For-Sale Mild CQSS 55 34 O=C(COc1ccc(Cl)cc1)N1CCC[C@H](CCBr)C1 ZINC000147260947 FH For-Sale Reactive COLA 42 45 O=C(COc1ccc(Cl)cc1)N1CCC[C@H](CCBr)C1 ZINC000147260947 FH For-Sale Reactive CPT1A 39 41 O=C(COc1ccc(Cl)cc1)N1CCC[C@H](CCBr)C1 ZINC000147260947 FH For-Sale Reactive CPT2 39 41 O=C(COc1ccc(Cl)cc1)N1CCC[C@H](CCBr)C1 ZINC000147260947 FH For-Sale Reactive GPR183 0 48 CCOC(=O)c1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147260955 EF On-Demand Anodyne KCNA5 27 42 CCOC(=O)c1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147260955 EF On-Demand Anodyne F2RL3 18 41 CCCCO[C@H](C)C(=O)N(C)Cc1nc2ccccc2[nH]1 ZINC000147260965 CF On-Demand Anodyne CACNA1G 31 43 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261074 CD On-Demand Anodyne DRD4 49 37 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261074 CD On-Demand Anodyne OPRD1 0 40 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261074 CD On-Demand Anodyne GRM3 18 41 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261074 CD On-Demand Anodyne CCR3 23 40 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261074 CD On-Demand Anodyne SLC18A3 24 44 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261074 CD On-Demand Anodyne MTNR1B 31 41 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261074 CD On-Demand Anodyne SCN5A 25 40 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261074 CD On-Demand Anodyne L3MBTL1 0 44 CC[C@@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261074 CD On-Demand Anodyne L3MBTL3 35 40 CC(C)c1nc(NN)cc(NCCN2CCOCC2)n1 ZINC000147261106 CC For-Sale Anodyne TLR9 0 41 O=C(COc1ccc(Cl)c(F)c1)c1cccc(Cl)c1 ZINC000147261136 CI For-Sale Anodyne MAOB 24 40 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147261162 FH For-Sale Reactive COLA 42 45 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147261162 FH For-Sale Reactive CPT1A 39 41 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147261162 FH For-Sale Reactive CPT2 39 41 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147261162 FH For-Sale Reactive GPR183 0 48 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCOCC1 ZINC000147261171 EC For-Sale Anodyne COLA 43 41 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCOCC1 ZINC000147261171 EC For-Sale Anodyne CPT1A 40 41 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCOCC1 ZINC000147261171 EC For-Sale Anodyne PTGDR2 32 45 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCOCC1 ZINC000147261171 EC For-Sale Anodyne AKR1C3 23 42 CCCCCCCCNC(=O)N[C@@H](CCO)C(=O)O ZINC000147261176 CD For-Sale Mild FOLH1 68 53 CCCCCCCCNC(=O)N[C@@H](CCO)C(=O)O ZINC000147261176 CD For-Sale Mild CPT1A 41 50 CCCCCCCCNC(=O)N[C@@H](CCO)C(=O)O ZINC000147261176 CD For-Sale Mild NAALAD2 48 39 CCCCCCCCNC(=O)N[C@@H](CCO)C(=O)O ZINC000147261176 CD For-Sale Mild EPHX2 59 50 CCCCCCCCNC(=O)N[C@@H](CCO)C(=O)O ZINC000147261176 CD For-Sale Mild ASAH1 75 35 CCCCCCCCNC(=O)N[C@@H](CCO)C(=O)O ZINC000147261176 CD For-Sale Mild NOD1 104 49 CCOC(=O)c1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147261195 EF On-Demand Anodyne KCNA5 30 42 CCOC(=O)c1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147261195 EF On-Demand Anodyne F2RL3 18 41 Cc1nn(C)c(Cl)c1C(=O)NCCn1c(C)nc2ccccc21 ZINC000147261210 EE On-Demand Anodyne PDE6D 15 40 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261280 CD On-Demand Anodyne DRD4 49 37 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261280 CD On-Demand Anodyne OPRD1 0 40 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261280 CD On-Demand Anodyne GRM3 18 41 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261280 CD On-Demand Anodyne CCR3 23 40 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261280 CD On-Demand Anodyne SLC18A3 24 44 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261280 CD On-Demand Anodyne MTNR1B 31 41 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261280 CD On-Demand Anodyne SCN5A 25 40 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261280 CD On-Demand Anodyne L3MBTL1 0 44 CC[C@H]1CN(C(=O)c2cccc(OC)c2)CC[C@H]1N ZINC000147261280 CD On-Demand Anodyne L3MBTL3 35 40 Cc1cc(C(=O)Nc2ccc(N3CCCC3)cc2C)cc([N+](=O)[O-])c1 ZINC000147261295 EI On-Demand Bother WDR5 34 41 NNc1cc(NCCN2CCOCC2)nc(C2CC2)n1 ZINC000147261322 CC For-Sale Anodyne TLR9 0 42 CO[C@H](C(=O)N1CCCC[C@@H]1c1ccccc1)c1ccccc1 ZINC000147261362 DI On-Demand Anodyne FKBP1A 54 40 CO[C@H](C(=O)N1CCCC[C@@H]1c1ccccc1)c1ccccc1 ZINC000147261362 DI On-Demand Anodyne SLC6A3 20 44 CO[C@H](C(=O)N1CCCC[C@@H]1c1ccccc1)c1ccccc1 ZINC000147261362 DI On-Demand Anodyne ADAM17 18 45 CO[C@H](C(=O)N1CCCC[C@@H]1c1ccccc1)c1ccccc1 ZINC000147261362 DI On-Demand Anodyne CPT1A 92 35 O=C(Nc1cccnc1)c1ccc2cc3n(c2n1)CCCNC3=O ZINC000147261381 DD Annotated Anodyne MAPKAPK2 15 72 O=C(Nc1cccnc1)c1ccc2cc3n(c2n1)CCCNC3=O ZINC000147261381 DD Annotated Anodyne RPS6KA3 105 72 CCCCCCCCNC(=O)N[C@H](CCO)C(=O)O ZINC000147261383 CD For-Sale Mild FOLH1 68 53 CCCCCCCCNC(=O)N[C@H](CCO)C(=O)O ZINC000147261383 CD For-Sale Mild CPT1A 41 50 CCCCCCCCNC(=O)N[C@H](CCO)C(=O)O ZINC000147261383 CD For-Sale Mild NAALAD2 48 39 CCCCCCCCNC(=O)N[C@H](CCO)C(=O)O ZINC000147261383 CD For-Sale Mild EPHX2 59 50 CCCCCCCCNC(=O)N[C@H](CCO)C(=O)O ZINC000147261383 CD For-Sale Mild ASAH1 75 35 CCCCCCCCNC(=O)N[C@H](CCO)C(=O)O ZINC000147261383 CD For-Sale Mild NOD1 104 49 CCOC(=O)c1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147261396 EF On-Demand Anodyne KCNA5 27 42 CCOC(=O)c1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147261396 EF On-Demand Anodyne F2RL3 18 41 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne CHRM2 20 47 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne CHRM1 17 42 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne DRD2 25 55 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne CNR1 17 43 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne DRD4 68 57 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne ACHE 37 57 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne DRD3 20 47 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne KCNH2 17 42 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne HTR4 18 44 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne CHRM3 34 42 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne LTA4H 20 41 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne SIGMAR1 55 60 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne SSTR5 50 42 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne CCR1 24 47 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne CCR3 35 45 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne APP 15 44 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne UTS2R 19 40 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne MLNR 26 40 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne SLC6A5 26 43 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne AKT1 15 41 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne PDK1 43 41 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne CXCR3 41 43 O=C(NC1CCN(Cc2ccc(Cl)cc2)CC1)c1sccc1-c1ccccc1 ZINC000147261405 HK On-Demand Anodyne MCHR1 63 55 CCN(CC)C(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147261409 DD For-Sale Anodyne PTGDR2 46 42 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccc(Cl)cc3Cl)c(F)c2)CC1 ZINC000147261472 KJ Annotated Clean MC4R 44 34 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccc(Cl)cc3Cl)c(F)c2)CC1 ZINC000147261472 KJ Annotated Clean MC5R 41 33 CC(=O)Nc1ccc(F)c(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147261493 ED On-Demand Anodyne ENV 40 33 C[C@H](Oc1cccc(Cl)c1)C(=O)N1CCC[C@H](CCBr)C1 ZINC000147261523 FI For-Sale Reactive GHSR 23 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ncn(Cc3ccccc3)n1)C2 ZINC000147261540 FF On-Demand Anodyne ROCK2 33 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ncn(Cc3ccccc3)n1)C2 ZINC000147261540 FF On-Demand Anodyne FAAH 17 46 CO[C@H](C(=O)N1CCCC[C@H]1c1ccccc1)c1ccccc1 ZINC000147261563 DI On-Demand Anodyne FKBP1A 54 40 CO[C@H](C(=O)N1CCCC[C@H]1c1ccccc1)c1ccccc1 ZINC000147261563 DI On-Demand Anodyne SLC6A3 20 44 CO[C@H](C(=O)N1CCCC[C@H]1c1ccccc1)c1ccccc1 ZINC000147261563 DI On-Demand Anodyne AGTR2 68 35 CO[C@H](C(=O)N1CCCC[C@H]1c1ccccc1)c1ccccc1 ZINC000147261563 DI On-Demand Anodyne ADAM17 45 47 CO[C@H](C(=O)N1CCCC[C@H]1c1ccccc1)c1ccccc1 ZINC000147261563 DI On-Demand Anodyne COLA 91 35 CO[C@H](C(=O)N1CCCC[C@H]1c1ccccc1)c1ccccc1 ZINC000147261563 DI On-Demand Anodyne CPT1A 92 35 CC(C)(C)c1nc(NN)cc(NCCN2CCOCC2)n1 ZINC000147261566 CC For-Sale Anodyne TLR9 0 42 Cc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)c(C)c1 ZINC000147261619 DG On-Demand Anodyne EPHX2 20 40 N#CC1CCN(C(=O)Cc2cccc(C(F)(F)F)c2)CC1 ZINC000147261625 CG On-Demand Mild CACNA1B 58 39 N#CC1CCN(C(=O)Cc2cccc(C(F)(F)F)c2)CC1 ZINC000147261625 CG On-Demand Mild CCR2 47 38 N#CC1CCN(C(=O)Cc2cccc(C(F)(F)F)c2)CC1 ZINC000147261625 CG On-Demand Mild SCD1 16 45 N#CC1CCN(C(=O)Cc2cccc(C(F)(F)F)c2)CC1 ZINC000147261625 CG On-Demand Mild LIPG 51 34 CCCCCCCCNC(=O)N[C@@H]1CCC[C@@H]1C(=O)O ZINC000147261635 CF For-Sale Mild EPHX2 31 60 CCCCCCCCNC(=O)N[C@@H]1CCC[C@@H]1C(=O)O ZINC000147261635 CF For-Sale Mild GNAI1 0 42 CCCCCCCCNC(=O)N[C@@H]1CCC[C@@H]1C(=O)O ZINC000147261635 CF For-Sale Mild GNAI3 0 42 CCCCCCCCNC(=O)N[C@@H]1CCC[C@@H]1C(=O)O ZINC000147261635 CF For-Sale Mild GNAO1 0 42 CCCCCCCCNC(=O)N[C@@H]1CCC[C@@H]1C(=O)O ZINC000147261635 CF For-Sale Mild ASAH1 56 33 O=C(O)CCNCc1ccc2nc(-c3ccccc3F)oc2c1 ZINC000147261664 DG For-Sale Anodyne S1PR1 15 48 O=C(O)CCNCc1ccc2nc(-c3ccccc3F)oc2c1 ZINC000147261664 DG For-Sale Anodyne HPSE 56 38 C[C@H](CNS(=O)(=O)c1cccc(C(F)(F)F)c1)CC(=O)O ZINC000147261699 EE On-Demand Anodyne CACNA1B 48 34 C[C@H](CNS(=O)(=O)c1cccc(C(F)(F)F)c1)CC(=O)O ZINC000147261699 EE On-Demand Anodyne COLA 17 44 C[C@H](CNS(=O)(=O)c1cccc(C(F)(F)F)c1)CC(=O)O ZINC000147261699 EE On-Demand Anodyne MTNN 29 40 C[C@H](CNS(=O)(=O)c1cccc(C(F)(F)F)c1)CC(=O)O ZINC000147261699 EE On-Demand Anodyne SFRP1 66 34 CC(=O)Nc1ccc(F)c(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147261717 ED On-Demand Anodyne ENV 40 33 C[C@@H](Oc1cccc(Cl)c1)C(=O)N1CCC[C@H](CCBr)C1 ZINC000147261721 FI For-Sale Reactive GHSR 23 42 CC(=O)N1CCN(c2ccc(CN(C3COC3)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147261754 IE Annotated Clean RORC 22 51 O=C(CCCOc1ccc(Cl)c(F)c1)c1ccc(Br)cc1 ZINC000147261762 FK For-Sale Anodyne SHC 41 44 O=C(CCCOc1ccc(Cl)c(F)c1)c1ccc(Br)cc1 ZINC000147261762 FK For-Sale Anodyne LSS 32 43 COc1ccc(CNCCCCC(C)C)c2ccccc12 ZINC000147261808 CJ For-Sale Anodyne SLC2A1 25 79 COc1ccc(CNCCCCC(C)C)c2ccccc12 ZINC000147261808 CJ For-Sale Anodyne HT1 22 79 COc1ccc(CNCCCCC(C)C)c2ccccc12 ZINC000147261808 CJ For-Sale Anodyne LMGT2 28 79 Cc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)c(C)c1 ZINC000147261839 DG On-Demand Anodyne EPHX2 20 40 CCCCCCCCNC(=O)N[C@H]1CCC[C@@H]1C(=O)O ZINC000147261870 CF For-Sale Mild EPHX2 31 60 CCCCCCCCNC(=O)N[C@H]1CCC[C@@H]1C(=O)O ZINC000147261870 CF For-Sale Mild GNAI1 0 42 CCCCCCCCNC(=O)N[C@H]1CCC[C@@H]1C(=O)O ZINC000147261870 CF For-Sale Mild GNAI3 0 42 CCCCCCCCNC(=O)N[C@H]1CCC[C@@H]1C(=O)O ZINC000147261870 CF For-Sale Mild GNAO1 0 42 CCCCCCCCNC(=O)N[C@H]1CCC[C@@H]1C(=O)O ZINC000147261870 CF For-Sale Mild ASAH1 56 33 N#Cc1cccc(COc2ccc(Cl)cc2S(N)(=O)=O)c1 ZINC000147261875 DE For-Sale Mild MAOB 24 44 C[C@@H](CNS(=O)(=O)c1cccc(C(F)(F)F)c1)CC(=O)O ZINC000147261891 EE On-Demand Anodyne CACNA1B 48 34 C[C@@H](CNS(=O)(=O)c1cccc(C(F)(F)F)c1)CC(=O)O ZINC000147261891 EE On-Demand Anodyne COLA 17 44 C[C@@H](CNS(=O)(=O)c1cccc(C(F)(F)F)c1)CC(=O)O ZINC000147261891 EE On-Demand Anodyne MTNN 29 40 C[C@@H](CNS(=O)(=O)c1cccc(C(F)(F)F)c1)CC(=O)O ZINC000147261891 EE On-Demand Anodyne SFRP1 66 34 O=C(NCCn1ccnc1)c1cccc2c1OCCN2 ZINC000147261913 CD For-Sale Anodyne TBXAS1 41 42 O=C(NCCn1ccnc1)c1cccc2c1OCCN2 ZINC000147261913 CD For-Sale Anodyne POLR1A 25 47 C[C@H](Oc1cccc(Cl)c1)C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147261919 FI For-Sale Reactive GHSR 23 42 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1F ZINC000147261940 DD On-Demand Anodyne ENV 44 36 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1F ZINC000147261940 DD On-Demand Anodyne QRFPR 42 36 COc1ccc(CNC2(C(=O)O)CCC2)cc1F ZINC000147261942 CD On-Demand Anodyne DRTS_TRYCR 44 31 COc1cc(/C=C/C(=O)N2CCC(C#N)CC2)cc(OC)c1OC ZINC000147261970 EE On-Demand Mild CCR2 69 43 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147262020 IG Annotated Clean ITGA4 42 37 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147262020 IG Annotated Clean RORC 24 52 Cn1ncc(C(=O)OCc2ccc(-n3cccn3)cc2)c1C1CC1 ZINC000147262026 DF On-Demand Anodyne AMP1_PLAFQ 49 31 Cc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)c(C)c1 ZINC000147262063 DG On-Demand Anodyne EPHX2 20 40 NC(=O)/C=C(/C(N)=O)c1ccccc1 ZINC000147262076 AC For-Sale Anodyne PA 15 42 CCCCCCCCNC(=O)N[C@@H]1CCC[C@H]1C(=O)O ZINC000147262084 CF For-Sale Mild EPHX2 31 60 CCCCCCCCNC(=O)N[C@@H]1CCC[C@H]1C(=O)O ZINC000147262084 CF For-Sale Mild GNAI1 0 42 CCCCCCCCNC(=O)N[C@@H]1CCC[C@H]1C(=O)O ZINC000147262084 CF For-Sale Mild GNAI3 0 42 CCCCCCCCNC(=O)N[C@@H]1CCC[C@H]1C(=O)O ZINC000147262084 CF For-Sale Mild GNAO1 0 42 CCCCCCCCNC(=O)N[C@@H]1CCC[C@H]1C(=O)O ZINC000147262084 CF For-Sale Mild ASAH1 56 33 C[C@@H](Oc1cccc(Cl)c1)C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147262106 FI For-Sale Reactive GHSR 23 42 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1F ZINC000147262131 DD On-Demand Anodyne ENV 44 36 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1F ZINC000147262131 DD On-Demand Anodyne QRFPR 42 36 CC(C)n1ncc2cc(NC(=O)c3ccc4cc5n(c4n3)CC(C)(C)CNC5=O)cnc21 ZINC000147262136 IG Annotated Anodyne RPS6KA3 44 58 C[C@H](CN)CC(=O)NN(C)C ZINC000147262149 AB For-Sale Reactive KDM7A 0 42 CC(=O)N1CCN(c2ccc(CN(C)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147262248 HE Annotated Clean RORC 30 57 O=C(C[C@@H]1CNc2ccccc21)N1CCCCCC1 ZINC000147262250 CF For-Sale Anodyne PREP 55 37 CCCCCCCCNC(=O)N[C@H]1CCC[C@H]1C(=O)O ZINC000147262302 CF For-Sale Mild EPHX2 31 60 CCCCCCCCNC(=O)N[C@H]1CCC[C@H]1C(=O)O ZINC000147262302 CF For-Sale Mild GNAI1 0 42 CCCCCCCCNC(=O)N[C@H]1CCC[C@H]1C(=O)O ZINC000147262302 CF For-Sale Mild GNAI3 0 42 CCCCCCCCNC(=O)N[C@H]1CCC[C@H]1C(=O)O ZINC000147262302 CF For-Sale Mild GNAO1 0 42 CCCCCCCCNC(=O)N[C@H]1CCC[C@H]1C(=O)O ZINC000147262302 CF For-Sale Mild ASAH1 56 33 C[C@@H](CN)CC(=O)NN(C)C ZINC000147262352 AB For-Sale Reactive KDM7A 0 42 COc1cc(C(=O)N2CCC[C@H](CCBr)C2)ccc1C ZINC000147262370 EH For-Sale Reactive GRM3 22 48 COc1cc(C(=O)N2CCC[C@H](CCBr)C2)ccc1C ZINC000147262370 EH For-Sale Reactive L3MBTL3 42 34 COc1cc(C(=O)N2CCC[C@H](CCBr)C2)ccc1C ZINC000147262370 EH For-Sale Reactive ACKR3 65 34 C[C@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccc(Br)cc1 ZINC000147262409 FE For-Sale Anodyne SDH1 0 48 C[C@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccc(Br)cc1 ZINC000147262409 FE For-Sale Anodyne ACACA 41 35 C[C@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccc(Br)cc1 ZINC000147262409 FE For-Sale Anodyne F7 15 44 O=C(C[C@H]1CNc2ccccc21)N1CCCCCC1 ZINC000147262470 CF For-Sale Anodyne PREP 55 37 CC(=O)N1CCN(c2ccc(CN(C3CC3)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147262493 IF Annotated Clean ITGA4 40 36 CC(=O)N1CCN(c2ccc(CN(C3CC3)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147262493 IF Annotated Clean RORC 24 53 C[C@@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccc(Br)cc1 ZINC000147262529 FE For-Sale Anodyne SDH1 0 48 C[C@@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccc(Br)cc1 ZINC000147262529 FE For-Sale Anodyne ACACA 41 35 C[C@@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccc(Br)cc1 ZINC000147262529 FE For-Sale Anodyne F7 15 44 COc1cc(C(=O)N2CCC[C@@H](CCBr)C2)ccc1C ZINC000147262567 EH For-Sale Reactive GRM3 22 48 COc1cc(C(=O)N2CCC[C@@H](CCBr)C2)ccc1C ZINC000147262567 EH For-Sale Reactive L3MBTL3 42 34 COc1cc(C(=O)N2CCC[C@@H](CCBr)C2)ccc1C ZINC000147262567 EH For-Sale Reactive ACKR3 65 34 CCOC(=O)c1cccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)c1 ZINC000147262596 HG On-Demand Anodyne ROCK2 23 42 CCOC(=O)c1cccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)c1 ZINC000147262596 HG On-Demand Anodyne EPHX2 18 43 CCOC(=O)c1cccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)c1 ZINC000147262596 HG On-Demand Anodyne HIF1A 15 40 CCCCCCCCNC(=O)N[C@@H]1CCCC[C@@H]1C(=O)O ZINC000147262639 CG For-Sale Mild EPHX2 31 64 CCCCCCCCNC(=O)N[C@@H]1CCCC[C@@H]1C(=O)O ZINC000147262639 CG For-Sale Mild ASAH1 56 33 Cc1ccccc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147262646 CD On-Demand Anodyne ITGAV 44 48 Cc1ccccc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147262646 CD On-Demand Anodyne ITGA2 0 42 Cc1ccccc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147262646 CD On-Demand Anodyne CTSA 42 32 CCN(Cc1ccc(N2CCN(C(C)=O)CC2)cc1)S(=O)(=O)Cc1ccccc1 ZINC000147262674 HF Annotated Clean RORC 36 61 CCOC(=O)c1cccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)c1 ZINC000147262786 HG On-Demand Anodyne ROCK2 23 42 CCOC(=O)c1cccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)c1 ZINC000147262786 HG On-Demand Anodyne EPHX2 18 43 CCOC(=O)c1cccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)c1 ZINC000147262786 HG On-Demand Anodyne HIF1A 15 40 CCCCCCCCNC(=O)N[C@H]1CCCC[C@@H]1C(=O)O ZINC000147262791 CG For-Sale Mild EPHX2 31 64 CCCCCCCCNC(=O)N[C@H]1CCCC[C@@H]1C(=O)O ZINC000147262791 CG For-Sale Mild ASAH1 56 33 Cc1ccccc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147262794 CD On-Demand Anodyne ITGAV 44 48 Cc1ccccc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147262794 CD On-Demand Anodyne ITGA2 0 42 Cc1ccccc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147262794 CD On-Demand Anodyne CTSA 42 32 O=C(c1cc2ccccc2o1)N1CCC[C@H](CCBr)C1 ZINC000147262864 EI For-Sale Reactive AKR1C3 0 48 CC[C@@H](C)NC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147262880 ED For-Sale Anodyne CA2 27 43 CC[C@@H](C)NC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147262880 ED For-Sale Anodyne CA1 16 43 CC[C@@H](C)NC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147262880 ED For-Sale Anodyne COLA 40 32 CC[C@@H](C)NC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147262880 ED For-Sale Anodyne CA4 20 43 CC[C@@H](C)NC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147262880 ED For-Sale Anodyne PTGDR2 26 40 C[C@](NC(=O)C1[C@H]2CCCC[C@H]12)(C(=O)O)c1ccccc1 ZINC000147262889 CF On-Demand Anodyne AMY2 49 33 Nc1cc(Cl)cc(-c2nc(-c3ccccc3Cl)no2)c1 ZINC000147262915 DI For-Sale Anodyne LUCI_PHOPE 34 40 C[C@H]1CN(S(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)C[C@@H](C)O1 ZINC000147262933 GD On-Demand Mild AKR1C3 63 45 CCCCCCCCNC(=O)N[C@@H]1CCCC[C@H]1C(=O)O ZINC000147262967 CG For-Sale Mild EPHX2 31 64 CCCCCCCCNC(=O)N[C@@H]1CCCC[C@H]1C(=O)O ZINC000147262967 CG For-Sale Mild ASAH1 56 33 CC[C@@H](C)[C@H](N)C(=O)NN(C)C ZINC000147262983 AB For-Sale Reactive SLC15A2 0 40 C[C@@H](CCc1ccccc1)S(=O)(=O)c1ccccc1 ZINC000147262986 CG On-Demand Anodyne MMP3 22 43 C[C@@H](CCc1ccccc1)S(=O)(=O)c1ccccc1 ZINC000147262986 CG On-Demand Anodyne LAP3 50 47 Cc1ccc(Cl)cc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147263010 DE On-Demand Anodyne TBXA2R 41 33 Cc1ccc(Cl)cc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147263010 DE On-Demand Anodyne PTGDR2 25 44 Cc1ccc(Cl)cc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147263010 DE On-Demand Anodyne OXER1 42 36 O=C(c1cc2ccccc2o1)N1CCC[C@@H](CCBr)C1 ZINC000147263022 EI For-Sale Reactive AKR1C3 0 48 CCOC(=O)CN(C(=O)Cc1ccccc1)c1ccc(F)cc1 ZINC000147263075 DF On-Demand Anodyne TDP1 0 61 CC[C@H](C)NC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147263094 ED For-Sale Anodyne CA2 27 43 CC[C@H](C)NC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147263094 ED For-Sale Anodyne COLA 40 32 CC[C@H](C)NC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147263094 ED For-Sale Anodyne PTGDR2 26 40 Cc1nn(C(F)F)c(C)c1CC(=O)NNc1ccccc1C(F)(F)F ZINC000147263151 FH On-Demand Reactive P2RX7 40 43 C[C@H]1CN(S(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)C[C@H](C)O1 ZINC000147263159 GD On-Demand Mild AKR1C3 63 45 CCCCCCCCNC(=O)N[C@H]1CCCC[C@H]1C(=O)O ZINC000147263183 CG For-Sale Mild EPHX2 31 64 CCCCCCCCNC(=O)N[C@H]1CCCC[C@H]1C(=O)O ZINC000147263183 CG For-Sale Mild ASAH1 56 33 CC[C@H](C)[C@H](N)C(=O)NN(C)C ZINC000147263218 AB For-Sale Reactive SLC15A2 0 40 C[C@H](CCc1ccccc1)S(=O)(=O)c1ccccc1 ZINC000147263223 CG On-Demand Anodyne MMP3 22 43 C[C@H](CCc1ccccc1)S(=O)(=O)c1ccccc1 ZINC000147263223 CG On-Demand Anodyne LAP3 50 47 Cc1ccc(Cl)cc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147263254 DE On-Demand Anodyne TBXA2R 41 33 Cc1ccc(Cl)cc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147263254 DE On-Demand Anodyne PTGDR2 25 44 Cc1ccc(Cl)cc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147263254 DE On-Demand Anodyne OXER1 42 36 CC(C)(C)c1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147263287 FJ For-Sale Reactive GRM3 15 47 CC(C)(C)c1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147263287 FJ For-Sale Reactive MLYCD 18 40 CC(C)(C)c1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147263287 FJ For-Sale Reactive L3MBTL1 0 40 CC(C)(C)c1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147263287 FJ For-Sale Reactive L3MBTL3 65 40 CC[C@@H](C)NC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147263293 ED For-Sale Anodyne CA2 27 43 CC[C@@H](C)NC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147263293 ED For-Sale Anodyne COLA 40 32 CC[C@@H](C)NC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147263293 ED For-Sale Anodyne PTGDR2 26 40 CCCC[C@H](CC)C(=O)N1CC[C@H](N)[C@H](CC)C1 ZINC000147263324 CF On-Demand Anodyne SLC22A20 0 41 CN(C)CCC(=O)c1cc(Cl)cc(Cl)c1 ZINC000147263325 BG Annotated Anodyne UTS2 43 35 C[C@](NC(=O)C1[C@H]2CCCC[C@@H]12)(C(=O)O)c1ccccc1 ZINC000147263326 CF For-Sale Anodyne AMY2 49 33 C[C@@H]1CN(S(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)C[C@@H](C)O1 ZINC000147263355 GD On-Demand Mild AKR1C3 63 45 CC(C)Oc1cccc(CC(=O)Nc2nnc(-c3ccco3)s2)c1 ZINC000147263361 EH On-Demand Anodyne CSNK1D 31 46 CCCCCCCCNC(=O)NCc1nc(C(=O)O)cs1 ZINC000147263410 DG For-Sale Mild EPHX2 50 41 CCCCCCCCNC(=O)NCc1nc(C(=O)O)cs1 ZINC000147263410 DG For-Sale Mild ASAH1 83 38 CCOC(=O)c1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147263470 GH On-Demand Anodyne NOS2 48 34 CCOC(=O)c1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147263470 GH On-Demand Anodyne ROCK2 36 41 CCOC(=O)c1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147263470 GH On-Demand Anodyne NAMPT 30 40 COc1ccc(C(=O)N(C)C)cc1NC(=O)c1cnn(-c2ccccc2Cl)c1 ZINC000147263476 GG On-Demand Anodyne CPT1A 47 33 COc1ccc(C(=O)N(C)C)cc1NC(=O)c1cnn(-c2ccccc2Cl)c1 ZINC000147263476 GG On-Demand Anodyne RBP4 22 43 COc1ccc(C(=O)N(C)C)cc1NC(=O)c1cnn(-c2ccccc2Cl)c1 ZINC000147263476 GG On-Demand Anodyne EPHB3 49 39 Cc1ccc(-c2noc(CNC3(C(=O)O)CCC3)n2)cc1 ZINC000147263482 CE For-Sale Anodyne NPPA 21 42 CC(C)(C)c1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147263490 FJ For-Sale Reactive GRM3 15 47 CC(C)(C)c1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147263490 FJ For-Sale Reactive MLYCD 18 40 CC(C)(C)c1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147263490 FJ For-Sale Reactive L3MBTL1 0 40 CC(C)(C)c1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147263490 FJ For-Sale Reactive L3MBTL3 65 40 O=C(CCCOc1ccc(Cl)c(F)c1)c1ccccc1 ZINC000147263495 CJ For-Sale Anodyne PLA2G4B 45 36 CC[C@H](C)NC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147263525 ED For-Sale Anodyne CA2 27 43 CC[C@H](C)NC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147263525 ED For-Sale Anodyne COLA 40 32 CC[C@H](C)NC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147263525 ED For-Sale Anodyne PTGDR2 26 40 C[C@@](NC(=O)C1[C@H]2CCCC[C@@H]12)(C(=O)O)c1ccccc1 ZINC000147263537 CF For-Sale Anodyne AMY2 49 33 O=C(C[C@@H]1CNc2ccccc21)Nc1cccnc1 ZINC000147263544 CF For-Sale Anodyne NAMPT 21 41 Cc1ccc(CNc2cc(NN)nc(C(C)C)n2)cc1 ZINC000147263546 CF For-Sale Anodyne PETD 0 43 CNc1cn2ccnc2c(Oc2ccccc2C(C)C)n1 ZINC000147263594 CH For-Sale Anodyne HIVRT 0 42 CCCCCCCCNC(=O)NC[C@](C)(O)C(=O)O ZINC000147263614 CD For-Sale Mild CPT1A 22 43 CCCCCCCCNC(=O)NC[C@](C)(O)C(=O)O ZINC000147263614 CD For-Sale Mild CES2 42 38 CCCCCCCCNC(=O)NC[C@](C)(O)C(=O)O ZINC000147263614 CD For-Sale Mild EST1_PIG 47 38 CCCCCCCCNC(=O)NC[C@](C)(O)C(=O)O ZINC000147263614 CD For-Sale Mild EPHX2 53 50 CCCCCCCCNC(=O)NC[C@](C)(O)C(=O)O ZINC000147263614 CD For-Sale Mild CES2C 47 38 CCCCCCCCNC(=O)NC[C@](C)(O)C(=O)O ZINC000147263614 CD For-Sale Mild ASAH1 81 34 COc1ccccc1CNC1(C(=O)O)CCC1 ZINC000147263677 BD On-Demand Anodyne TACR1 22 51 COc1ccccc1CNC1(C(=O)O)CCC1 ZINC000147263677 BD On-Demand Anodyne GPM3 0 45 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCCCC3)c2)CC1 ZINC000147263692 GF On-Demand Mild CACNA1B 28 43 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCCCC3)c2)CC1 ZINC000147263692 GF On-Demand Mild PREP 25 46 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCCCC3)c2)CC1 ZINC000147263692 GF On-Demand Mild EPHX2 20 49 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCCCC3)c2)CC1 ZINC000147263692 GF On-Demand Mild AKR1C3 67 46 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCCCC3)c2)CC1 ZINC000147263692 GF On-Demand Mild AKR1C1 23 42 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCCCC3)c2)CC1 ZINC000147263692 GF On-Demand Mild L3MBTL3 84 47 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cc(C(=O)N(C)C)ccc1OC)C2 ZINC000147263708 GF On-Demand Anodyne ROCK2 37 51 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cc(C(=O)N(C)C)ccc1OC)C2 ZINC000147263708 GF On-Demand Anodyne MT-ND4 49 30 Cc1nccc(-c2cccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)c2)n1 ZINC000147263714 FE On-Demand Anodyne PRKD1 57 32 O=C1CCN(C(=O)COc2ccc(Cl)c(F)c2)CC1 ZINC000147263732 CE On-Demand Anodyne GPR183 0 46 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCCC1 ZINC000147263738 DD For-Sale Anodyne HTR2A 23 43 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCCC1 ZINC000147263738 DD For-Sale Anodyne HTR2C 15 43 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCCC1 ZINC000147263738 DD For-Sale Anodyne LTA4H 36 47 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCCC1 ZINC000147263738 DD For-Sale Anodyne HRH3 38 46 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCCC1 ZINC000147263738 DD For-Sale Anodyne SIGMAR1 15 46 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCCC1 ZINC000147263738 DD For-Sale Anodyne HNMT 38 40 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCCC1 ZINC000147263738 DD For-Sale Anodyne MCHR1 0 40 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCCC1 ZINC000147263738 DD For-Sale Anodyne PSMB2 39 40 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCCC1 ZINC000147263738 DD For-Sale Anodyne PSMB1 43 40 CCCC[C@H](CC)C(=O)N1CC[C@@H](N)[C@H](CC)C1 ZINC000147263745 CF On-Demand Anodyne SLC22A20 0 41 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne ACE 41 48 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne OPRM1 16 43 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne OPRD1 20 43 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CELA1 26 47 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne ELANE 47 71 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne MME 54 43 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne TACR1 17 44 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CTSD 16 48 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne HRAS 59 41 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CASP3 37 57 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne BMP1 74 46 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CASP8 18 57 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne KLK3 92 42 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CTSB 87 67 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne PAPA1_CARPA 94 51 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CYSP_TRYCR 61 43 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CTSK 56 67 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CTSL 56 67 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne PGA 40 56 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CAPNS1 76 44 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne MMP8 40 38 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne MMP14 40 38 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne HLA-DRB1 60 38 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne LGMN 18 44 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne MMP11 54 33 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CTSS 26 57 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CAPN1 104 63 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CASP1 51 57 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CTRC 16 45 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CAPN2 153 56 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CASP6 40 57 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CASP9 53 57 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CYP3A4 31 42 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne NPR 89 46 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne XIAP 17 46 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne CASP10 39 41 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne PSMB5 49 41 CC(C)[C@@H](NC(=O)OCc1ccccc1)C(=O)N(C)CC(=O)O ZINC000147263746 DD For-Sale Anodyne Q6PRC7_IXORI 52 45 O=C(C[C@H]1CNc2ccccc21)Nc1cccnc1 ZINC000147263761 CF For-Sale Anodyne NAMPT 21 41 O=[N+]([O-])c1ccc2[nH]c(N3CCC(CBr)CC3)nc2c1 ZINC000147263793 EG For-Sale Reactive NPY5R 15 52 CCNc1ncc(Cl)c(Oc2ccccc2C(C)C)n1 ZINC000147263809 CI For-Sale Anodyne P2RX2 62 33 CCNc1ncc(Cl)c(Oc2ccccc2C(C)C)n1 ZINC000147263809 CI For-Sale Anodyne P2RX3 43 33 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EGFR 138 59 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne DRD2 19 41 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne ERBB2 95 55 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne PDGFRB 94 51 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne IGF1R 15 41 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne KIT 26 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne LCK 18 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MAPK14 26 56 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne FGFR2 40 38 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MAP2K5 27 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne SRC 85 56 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne AURKB 65 70 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne CSK 17 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne FLT1 34 59 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne KDR 48 62 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MAP2K2 22 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne SLC9A1 59 36 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne HDAC1 23 40 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne ABL2 20 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MST1R 32 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MAP2K1 35 47 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MET 70 48 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHB2 30 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne BLK 23 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHX2 19 43 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne FLT4 54 57 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne LYN 17 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne PDGFRA 35 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne FLT3 33 44 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne ERBB4 76 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne CSF1R 41 41 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne TEK 30 57 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MAPK12 21 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne IRAK1 21 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne ZAK 24 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne AURKA 66 67 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne GAK 16 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne RIPK2 25 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne STK10 35 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHA2 57 45 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHA3 22 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHA8 32 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne FRK 30 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne BMX 21 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHA5 35 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHB1 26 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHA4 28 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHA7 22 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne NEK9 16 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne SLK 25 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MKNK2 16 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHA6 42 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne TNIK 18 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MAP4K5 25 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne ULK3 26 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne FES 15 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne RET 16 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne BTK 37 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne FGR 15 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne AXL 49 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne TEC 24 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne TXK 17 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MKNK1 34 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne TIE1 23 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne DDR1 19 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MAP4K2 24 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne CDK11A 21 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne DDR2 18 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MYO3B 16 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne CDK8 23 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MAP4K1 17 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne CDK11B 15 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHA1 15 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne STK33 16 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne LTK 16 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne SRMS 30 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EIF2AK3 25 46 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EHMT2 76 37 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne EPHB6 20 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne ERBB3 38 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne SIK3 25 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne MAP3K19 17 53 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne HIPK4 32 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne PIP4K2C 15 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne CDK13 16 50 COc1cc2ncnc(Nc3ccc(C(=O)Nc4cc(F)ccc4N)cc3)c2cc1OCCCN1CCOCC1 ZINC000147263812 KI Annotated Anodyne DSTYK 17 50 CCCCCCCCNC(=O)NC[C@@](C)(O)C(=O)O ZINC000147263839 CD For-Sale Mild CPT1A 22 43 CCCCCCCCNC(=O)NC[C@@](C)(O)C(=O)O ZINC000147263839 CD For-Sale Mild CES2 42 38 CCCCCCCCNC(=O)NC[C@@](C)(O)C(=O)O ZINC000147263839 CD For-Sale Mild EST1_PIG 47 38 CCCCCCCCNC(=O)NC[C@@](C)(O)C(=O)O ZINC000147263839 CD For-Sale Mild EPHX2 53 50 CCCCCCCCNC(=O)NC[C@@](C)(O)C(=O)O ZINC000147263839 CD For-Sale Mild CES2C 47 38 CCCCCCCCNC(=O)NC[C@@](C)(O)C(=O)O ZINC000147263839 CD For-Sale Mild ASAH1 81 34 CCCCCCCCNC(=O)NC[C@@](C)(O)C(=O)O ZINC000147263839 CD For-Sale Mild FPPS 0 40 C[C@H](CNS(=O)(=O)c1cccnc1)CC(=O)O ZINC000147263915 CC On-Demand Anodyne TBXAS1 51 41 C[C@H](CNS(=O)(=O)c1cccnc1)CC(=O)O ZINC000147263915 CC On-Demand Anodyne KCNA5 45 38 C[C@H](CNS(=O)(=O)c1cccnc1)CC(=O)O ZINC000147263915 CC On-Demand Anodyne NAMPT 37 43 C[C@H]1C[C@@H](C)CN(S(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)C1 ZINC000147263919 GF On-Demand Mild CNR1 0 45 C[C@H]1C[C@@H](C)CN(S(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)C1 ZINC000147263919 GF On-Demand Mild ST14 48 34 C[C@H]1C[C@@H](C)CN(S(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)C1 ZINC000147263919 GF On-Demand Mild AKR1C3 64 43 Cc1nccc(-c2cccc(NC(=O)C(=O)NC[C@H]3CCCCO3)c2)n1 ZINC000147263948 FE On-Demand Anodyne PRKD1 57 32 N/C(CS)=N/[C@@H](Cc1ccccc1)c1ccccc1 ZINC000147263962 CG Annotated Mild ANPEP 15 43 Cc1cc(CN2[C@@H]3CC[C@@H]2CC(Br)C3)c2ccccc2n1 ZINC000147264022 EI For-Sale Reactive ADAM17 57 36 Cc1ccc(CNc2cc(NN)nc(C(C)(C)C)n2)cc1 ZINC000147264035 CF For-Sale Anodyne PETD 0 43 C#CCN(CC(=O)O)C(=O)NCCCCCCCC ZINC000147264063 CE For-Sale Mild EPHX2 0 41 C#CCN(CC(=O)O)C(=O)NCCCCCCCC ZINC000147264063 CE For-Sale Mild ASAH1 49 30 CN(C)NC(=O)[C@H](N)CCC(=O)O ZINC000147264095 AA For-Sale Reactive GSTM1 52 29 CN(C)NC(=O)[C@H](N)CCC(=O)O ZINC000147264095 AA For-Sale Reactive GRM8 27 52 CN(C)NC(=O)[C@H](N)CCC(=O)O ZINC000147264095 AA For-Sale Reactive GRIK3 32 52 CN(C)NC(=O)[C@H](N)CCC(=O)O ZINC000147264095 AA For-Sale Reactive GRIK5 15 52 CN(C)NC(=O)[C@H](N)CCC(=O)O ZINC000147264095 AA For-Sale Reactive GRIK2 16 52 CN(C)NC(=O)[C@H](N)CCC(=O)O ZINC000147264095 AA For-Sale Reactive GRIK1 15 52 CN(C)NC(=O)[C@H](N)CCC(=O)O ZINC000147264095 AA For-Sale Reactive KDM2A 40 31 CN(C)NC(=O)[C@H](N)CCC(=O)O ZINC000147264095 AA For-Sale Reactive PHF8 0 48 CN(C)NC(=O)[C@H](N)CCC(=O)O ZINC000147264095 AA For-Sale Reactive KDM7A 0 48 C[C@@H](CNS(=O)(=O)c1cccnc1)CC(=O)O ZINC000147264110 CC On-Demand Anodyne TBXAS1 51 41 C[C@@H](CNS(=O)(=O)c1cccnc1)CC(=O)O ZINC000147264110 CC On-Demand Anodyne KCNA5 45 38 C[C@@H](CNS(=O)(=O)c1cccnc1)CC(=O)O ZINC000147264110 CC On-Demand Anodyne NAMPT 37 43 C[C@@H]1C[C@@H](C)CN(S(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)C1 ZINC000147264144 GF On-Demand Mild CNR1 0 45 C[C@@H]1C[C@@H](C)CN(S(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)C1 ZINC000147264144 GF On-Demand Mild ST14 48 34 C[C@@H]1C[C@@H](C)CN(S(=O)(=O)c2cccc(C(=O)N3CCC(C#N)CC3)c2)C1 ZINC000147264144 GF On-Demand Mild AKR1C3 64 43 N/C(CS)=N/[C@H](Cc1ccccc1)c1ccccc1 ZINC000147264174 CG Annotated Mild ANPEP 15 43 CCc1ncc(C(=O)Nc2ccc(N3CCCC3)cc2C)s1 ZINC000147264218 DH On-Demand Anodyne MAPK14 15 41 CCc1ncc(C(=O)Nc2ccc(N3CCCC3)cc2C)s1 ZINC000147264218 DH On-Demand Anodyne HRH3 15 42 Cc1cc(CN2[C@H]3CC[C@@H]2CC(Br)C3)c2ccccc2n1 ZINC000147264226 EI For-Sale Reactive ADAM17 57 36 CCCCCCCCNC(=O)NCC1(C(=O)O)CCC1 ZINC000147264284 CF For-Sale Mild CPT1A 0 40 CCCCCCCCNC(=O)NCC1(C(=O)O)CCC1 ZINC000147264284 CF For-Sale Mild EPHX2 27 47 CCCCCCCCNC(=O)NCC1(C(=O)O)CCC1 ZINC000147264284 CF For-Sale Mild ASAH1 84 33 CCCCCCCCNC(=O)NCC1(C(=O)O)CCC1 ZINC000147264284 CF For-Sale Mild ACAT 0 41 CN(C)NC(=O)[C@@H](N)CCC(=O)O ZINC000147264314 AA For-Sale Reactive GSTM1 52 29 CN(C)NC(=O)[C@@H](N)CCC(=O)O ZINC000147264314 AA For-Sale Reactive GRM8 27 52 CN(C)NC(=O)[C@@H](N)CCC(=O)O ZINC000147264314 AA For-Sale Reactive GRIK3 32 52 CN(C)NC(=O)[C@@H](N)CCC(=O)O ZINC000147264314 AA For-Sale Reactive GRIK5 15 52 CN(C)NC(=O)[C@@H](N)CCC(=O)O ZINC000147264314 AA For-Sale Reactive GRIK2 16 52 CN(C)NC(=O)[C@@H](N)CCC(=O)O ZINC000147264314 AA For-Sale Reactive GRIK1 15 52 CN(C)NC(=O)[C@@H](N)CCC(=O)O ZINC000147264314 AA For-Sale Reactive KDM2A 40 31 CN(C)NC(=O)[C@@H](N)CCC(=O)O ZINC000147264314 AA For-Sale Reactive PHF8 0 48 CN(C)NC(=O)[C@@H](N)CCC(=O)O ZINC000147264314 AA For-Sale Reactive KDM7A 0 48 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCc4ccccc43)c2)CC1 ZINC000147264361 HG On-Demand Mild CYP11B2 28 41 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCc4ccccc43)c2)CC1 ZINC000147264361 HG On-Demand Mild AKR1C3 63 45 N#CC1CCN(C(=O)c2cccc(S(=O)(=O)N3CCCc4ccccc43)c2)CC1 ZINC000147264361 HG On-Demand Mild SFRP1 40 36 C[C@H](Oc1ccc(Cl)c(F)c1)C(=O)c1ccc(Br)cc1 ZINC000147264400 FJ For-Sale Anodyne GPR35 45 32 Cc1cc(CN2[C@H]3CC[C@H]2CC(Br)C3)c2ccccc2n1 ZINC000147264409 EI For-Sale Reactive ADAM17 57 36 CC(C)(C)c1nc(NN)cc(NCc2ccncc2)n1 ZINC000147264458 CE For-Sale Anodyne GPR39 0 43 CCNc1ncc(C)c(Oc2ccccc2C(C)C)n1 ZINC000147264473 CI For-Sale Anodyne P2RX2 51 32 Cc1ccc(F)c(C(=O)CCC(C)C)c1F ZINC000147264477 BH For-Sale Anodyne LEF 40 32 CCCCCCCCNC(=O)NCC1(C(=O)O)CC1 ZINC000147264485 CF For-Sale Mild CPT1A 25 41 CCCCCCCCNC(=O)NCC1(C(=O)O)CC1 ZINC000147264485 CF For-Sale Mild EPHX2 32 48 CCCCCCCCNC(=O)NCC1(C(=O)O)CC1 ZINC000147264485 CF For-Sale Mild ASAH1 88 35 C[C@@H](Oc1ccc(Cl)c(F)c1)C(=O)c1ccc(Br)cc1 ZINC000147264588 FJ For-Sale Anodyne GPR35 45 32 NC(=O)c1ccc(N2CCCCC2)c(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147264589 GI On-Demand Anodyne KCNQ2 56 42 NC(=O)c1ccc(N2CCCCC2)c(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147264589 GI On-Demand Anodyne CXCR3 17 40 NC(=O)c1ccc(N2CCCCC2)c(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147264589 GI On-Demand Anodyne TAAR1 27 45 CN1CCN(CCOc2ccc(Cl)cc2S(N)(=O)=O)CC1 ZINC000147264597 EC For-Sale Anodyne HTR2C 15 45 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(OC(F)F)c1 ZINC000147264601 ED On-Demand Anodyne TAAR1 21 43 O=C(NC1Cc2ccccc2C1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147264661 GF On-Demand Anodyne CA7 16 43 O=C(NC1Cc2ccccc2C1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147264661 GF On-Demand Anodyne MAP1 70 34 O=C(NC1Cc2ccccc2C1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147264661 GF On-Demand Anodyne GCK 19 40 CCCCCCCCNC(=O)N1CCCC[C@@H]1C(=O)O ZINC000147264664 CF For-Sale Mild ACE 48 49 CCCCCCCCNC(=O)N1CCCC[C@@H]1C(=O)O ZINC000147264664 CF For-Sale Mild FKBP1A 34 40 CCCCCCCCNC(=O)N1CCCC[C@@H]1C(=O)O ZINC000147264664 CF For-Sale Mild TPP2 54 50 CCCCCCCCNC(=O)N1CCCC[C@@H]1C(=O)O ZINC000147264664 CF For-Sale Mild GNAI1 0 43 CCCCCCCCNC(=O)N1CCCC[C@@H]1C(=O)O ZINC000147264664 CF For-Sale Mild GNAI3 0 43 CCCCCCCCNC(=O)N1CCCC[C@@H]1C(=O)O ZINC000147264664 CF For-Sale Mild GNAO1 0 43 CCCCCCCCNC(=O)N1CCCC[C@@H]1C(=O)O ZINC000147264664 CF For-Sale Mild ASAH1 104 44 CCCCCCCCNC(=O)N1CCCC[C@@H]1C(=O)O ZINC000147264664 CF For-Sale Mild DAPE 0 40 CCCNc1ncc(Cl)c(Oc2ccccc2C(C)C)n1 ZINC000147264693 DJ For-Sale Anodyne P2RX2 63 36 CCCNc1ncc(Cl)c(Oc2ccccc2C(C)C)n1 ZINC000147264693 DJ For-Sale Anodyne P2RX3 44 36 C[C@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264705 EB On-Demand Anodyne CA2 77 42 C[C@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264705 EB On-Demand Anodyne CA1 57 39 C[C@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264705 EB On-Demand Anodyne CA7 43 37 C[C@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264705 EB On-Demand Anodyne CA5B 44 37 C[C@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264705 EB On-Demand Anodyne CA4 81 42 C[C@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264705 EB On-Demand Anodyne CA5A 50 37 C[C@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264705 EB On-Demand Anodyne CA12 25 40 C[C@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264705 EB On-Demand Anodyne CA9 28 42 C[C@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264705 EB On-Demand Anodyne Q5TU56_ANOGA 0 45 CC(C)(C)c1nc(NN)cc(NCc2cccnc2)n1 ZINC000147264716 CE For-Sale Anodyne CLK4 15 40 Cc1ccc(NC(=O)C2CCN(C(=O)c3ccn(-c4cccc(F)c4)n3)CC2)nc1 ZINC000147264733 HG On-Demand Anodyne NPY5R 15 46 COc1ccc2c(c1Cl)CCNC2 ZINC000147264781 AD For-Sale Anodyne PNMT 39 43 NC(=O)c1ccc(N2CCCCC2)c(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147264787 GI On-Demand Anodyne KCNQ2 56 42 NC(=O)c1ccc(N2CCCCC2)c(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147264787 GI On-Demand Anodyne CXCR3 17 40 NC(=O)c1ccc(N2CCCCC2)c(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147264787 GI On-Demand Anodyne TAAR1 27 45 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(OC(F)F)c1 ZINC000147264821 ED On-Demand Anodyne TAAR1 21 43 Cc1ncoc1C(=O)N[C@@H](CCC(=O)O)c1ccccc1 ZINC000147264846 CE On-Demand Anodyne P2RY12 47 33 Cc1ncoc1C(=O)N[C@@H](CCC(=O)O)c1ccccc1 ZINC000147264846 CE On-Demand Anodyne PTGER3 52 35 Cc1ncoc1C(=O)N[C@@H](CCC(=O)O)c1ccccc1 ZINC000147264846 CE On-Demand Anodyne TACR3 41 35 Cc1ncoc1C(=O)N[C@@H](CCC(=O)O)c1ccccc1 ZINC000147264846 CE On-Demand Anodyne NAALAD2 27 40 Cc1ncoc1C(=O)N[C@@H](CCC(=O)O)c1ccccc1 ZINC000147264846 CE On-Demand Anodyne UTS2 59 40 CCCCCCCCNC(=O)N1CCCC[C@H]1C(=O)O ZINC000147264878 CF For-Sale Mild ACE 48 49 CCCCCCCCNC(=O)N1CCCC[C@H]1C(=O)O ZINC000147264878 CF For-Sale Mild FKBP1A 34 40 CCCCCCCCNC(=O)N1CCCC[C@H]1C(=O)O ZINC000147264878 CF For-Sale Mild TPP2 54 50 CCCCCCCCNC(=O)N1CCCC[C@H]1C(=O)O ZINC000147264878 CF For-Sale Mild GNAI1 0 43 CCCCCCCCNC(=O)N1CCCC[C@H]1C(=O)O ZINC000147264878 CF For-Sale Mild GNAI3 0 43 CCCCCCCCNC(=O)N1CCCC[C@H]1C(=O)O ZINC000147264878 CF For-Sale Mild GNAO1 0 43 CCCCCCCCNC(=O)N1CCCC[C@H]1C(=O)O ZINC000147264878 CF For-Sale Mild ASAH1 104 44 CCCCCCCCNC(=O)N1CCCC[C@H]1C(=O)O ZINC000147264878 CF For-Sale Mild DAPE 0 40 C[C@@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264894 EB On-Demand Anodyne CA2 77 42 C[C@@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264894 EB On-Demand Anodyne CA1 57 39 C[C@@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264894 EB On-Demand Anodyne CA7 43 37 C[C@@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264894 EB On-Demand Anodyne CA5B 44 37 C[C@@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264894 EB On-Demand Anodyne CA4 81 42 C[C@@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264894 EB On-Demand Anodyne CA5A 50 37 C[C@@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264894 EB On-Demand Anodyne CA12 25 40 C[C@@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264894 EB On-Demand Anodyne CA9 28 42 C[C@@H](CNS(=O)(=O)c1cccc(S(N)(=O)=O)c1)CC(=O)O ZINC000147264894 EB On-Demand Anodyne Q5TU56_ANOGA 0 45 NC(=O)c1ccc(N2CCCCC2)c(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147264977 GI On-Demand Anodyne KCNQ2 56 42 NC(=O)c1ccc(N2CCCCC2)c(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147264977 GI On-Demand Anodyne CXCR3 17 40 NC(=O)c1ccc(N2CCCCC2)c(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147264977 GI On-Demand Anodyne TAAR1 27 45 Cc1oc(-c2cccs2)nc1CNC1(C(=O)O)CCC1 ZINC000147265015 CF For-Sale Anodyne PPARG 24 43 Cc1oc(-c2cccs2)nc1CNC1(C(=O)O)CCC1 ZINC000147265015 CF For-Sale Anodyne PPARA 62 44 Cc1oc(-c2cccs2)nc1CNC1(C(=O)O)CCC1 ZINC000147265015 CF For-Sale Anodyne PDE8B 57 37 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147265023 HG On-Demand Mild AVPR1A 19 43 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147265023 HG On-Demand Mild MMP13 45 44 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147265023 HG On-Demand Mild ADAM17 37 40 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147265023 HG On-Demand Mild MMP1 24 40 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147265023 HG On-Demand Mild LIMK2 28 43 CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)N3CCC(C#N)CC3)cc2)cc1 ZINC000147265023 HG On-Demand Mild L3MBTL3 62 38 Cc1ncoc1C(=O)N[C@H](CCC(=O)O)c1ccccc1 ZINC000147265051 CE On-Demand Anodyne P2RY12 47 33 Cc1ncoc1C(=O)N[C@H](CCC(=O)O)c1ccccc1 ZINC000147265051 CE On-Demand Anodyne PTGER3 52 35 Cc1ncoc1C(=O)N[C@H](CCC(=O)O)c1ccccc1 ZINC000147265051 CE On-Demand Anodyne TACR3 41 35 Cc1ncoc1C(=O)N[C@H](CCC(=O)O)c1ccccc1 ZINC000147265051 CE On-Demand Anodyne NAALAD2 27 40 Cc1ncoc1C(=O)N[C@H](CCC(=O)O)c1ccccc1 ZINC000147265051 CE On-Demand Anodyne UTS2 59 40 CCCCCCCCNC(=O)N(CC(=O)O)CC(=O)O ZINC000147265082 CD For-Sale Mild FABP2 0 42 CCCCCCCCNC(=O)N(CC(=O)O)CC(=O)O ZINC000147265082 CD For-Sale Mild CPT1A 38 42 CCCCCCCCNC(=O)N(CC(=O)O)CC(=O)O ZINC000147265082 CD For-Sale Mild FAAH 0 42 CCCCCCCCNC(=O)N(CC(=O)O)CC(=O)O ZINC000147265082 CD For-Sale Mild S1PR2 45 38 CCCCCCCCNC(=O)N(CC(=O)O)CC(=O)O ZINC000147265082 CD For-Sale Mild EPHX2 33 48 CCCCCCCCNC(=O)N(CC(=O)O)CC(=O)O ZINC000147265082 CD For-Sale Mild ASAH1 87 35 CCCCCCCCNC(=O)N(CC(=O)O)CC(=O)O ZINC000147265082 CD For-Sale Mild SLC22A20 0 42 CCCCCCCCNC(=O)N(CC(=O)O)CC(=O)O ZINC000147265082 CD For-Sale Mild CQSS 48 30 CCN(C[C@@H]1CCCO1)C(=O)c1cccc2c1OCCN2 ZINC000147265131 CE For-Sale Anodyne OXTR 29 45 CCN(C[C@@H]1CCCO1)C(=O)c1cccc2c1OCCN2 ZINC000147265131 CE For-Sale Anodyne AVPR1A 0 45 NNc1cc(NCc2cccc(F)c2)nc(C2CC2)n1 ZINC000147265144 CE For-Sale Anodyne VCP 31 45 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccc(Cl)cc3)c(F)c2)CC1 ZINC000147265248 JH Annotated Clean SSTR3 49 37 Cn1cc(COC(=O)Cc2csc(-c3ccc(Cl)cc3Cl)n2)cn1 ZINC000147265266 GI On-Demand Anodyne DPP8 92 36 Cn1cc(COC(=O)Cc2csc(-c3ccc(Cl)cc3Cl)n2)cn1 ZINC000147265266 GI On-Demand Anodyne DPP9 87 35 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)NC1CC1 ZINC000147265292 DC For-Sale Anodyne CA2 15 40 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)NC1CC1 ZINC000147265292 DC For-Sale Anodyne CA1 16 40 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)NC1CC1 ZINC000147265292 DC For-Sale Anodyne CA7 18 40 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)NC1CC1 ZINC000147265292 DC For-Sale Anodyne NPY2R 0 41 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)NC1CC1 ZINC000147265292 DC For-Sale Anodyne PTGDR2 39 41 CCCCCCCCNC(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147265298 CF On-Demand Mild SLC6A1 103 38 CCCCCCCCNC(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147265298 CF On-Demand Mild F2R 0 42 CCCCCCCCNC(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147265298 CF On-Demand Mild EPHX2 15 46 CCCCCCCCNC(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147265298 CF On-Demand Mild TPP2 21 41 CCCCCCCCNC(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147265298 CF On-Demand Mild GNAI1 0 43 CCCCCCCCNC(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147265298 CF On-Demand Mild GNAI3 0 43 CCCCCCCCNC(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147265298 CF On-Demand Mild GNAO1 0 43 CCCCCCCCNC(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147265298 CF On-Demand Mild ASAH1 102 40 CCN(C[C@H]1CCCO1)C(=O)c1cccc2c1OCCN2 ZINC000147265302 CE For-Sale Anodyne OXTR 29 45 CCN(C[C@H]1CCCO1)C(=O)c1cccc2c1OCCN2 ZINC000147265302 CE For-Sale Anodyne AVPR1A 0 45 O=C(Nc1ccc(-n2ccnc2)c(F)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147265389 GI On-Demand Anodyne NPY2R 42 34 O=C(Nc1ccc(-n2ccnc2)c(F)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147265389 GI On-Demand Anodyne GRM4 60 45 O=C(Nc1ccc(-n2ccnc2)c(F)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147265389 GI On-Demand Anodyne MAPK10 16 42 CCc1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147265399 DG On-Demand Anodyne KCNA5 32 51 CC(C)CCCCNCc1ccc(F)c(-c2cccs2)c1 ZINC000147265408 DK For-Sale Anodyne LEF 82 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(F)c1 ZINC000147265423 DE On-Demand Anodyne ENV 62 50 O=C(O)C1(NCc2ccccc2OC(F)F)CCC1 ZINC000147265425 CE For-Sale Anodyne PHES 0 41 CC(C)(CCC(=O)O)NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147265454 CF For-Sale Anodyne NAMPT 22 40 CC(C)(CCC(=O)O)NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147265454 CF For-Sale Anodyne GPR88 0 41 COc1ccccc1NS(=O)(=O)c1cc(C(=O)N2CCC(C#N)CC2)ccc1C ZINC000147265487 HG On-Demand Mild CCR8 73 36 CC(C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147265497 DC For-Sale Anodyne CA2 36 41 CC(C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147265497 DC For-Sale Anodyne CA1 29 41 CC(C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147265497 DC For-Sale Anodyne CA4 30 41 CC(C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147265497 DC For-Sale Anodyne ALPL 18 41 CC(C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147265497 DC For-Sale Anodyne PTGDR2 43 41 C[C@@H](NC(=O)c1cc(F)ccc1NS(C)(=O)=O)c1ccc(OC(F)F)cc1 ZINC000147265533 HG On-Demand Anodyne TRPV1 54 34 C=C[C@@H]1CN2CC[C@H]1C[C@H]2[C@@H](NC(=S)Nc1cc(C(F)(F)F)cc(C(F)(F)F)c1)c1ccnc2ccc(OC)cc12 ZINC000147265546 KK For-Sale Mild SLC22A1 18 67 CCCCCCCCNC(=O)N[C@H](CC(N)=O)C(=O)O ZINC000147265555 CC For-Sale Mild FOLH1 46 40 CCCCCCCCNC(=O)N[C@H](CC(N)=O)C(=O)O ZINC000147265555 CC For-Sale Mild GRIA1 69 35 CCCCCCCCNC(=O)N[C@H](CC(N)=O)C(=O)O ZINC000147265555 CC For-Sale Mild EPHX2 20 55 CCCCCCCCNC(=O)N[C@H](CC(N)=O)C(=O)O ZINC000147265555 CC For-Sale Mild ASAH1 67 33 CCCCCCCCNC(=O)N[C@H](CC(N)=O)C(=O)O ZINC000147265555 CC For-Sale Mild NOD1 96 45 C[C@H](CNS(=O)(=O)c1c(Cl)cccc1Cl)CC(=O)O ZINC000147265592 EE On-Demand Anodyne ITGAV 17 45 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(-n3ccnc3)c(F)c1)C2 ZINC000147265602 FG On-Demand Anodyne ROCK2 33 49 C[C@H](N)CCCC(=O)NN(C)C ZINC000147265610 AC For-Sale Reactive NOD1 50 33 C[C@H](N)CCCC(=O)NN(C)C ZINC000147265610 AC For-Sale Reactive KDM7A 0 48 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(F)c1 ZINC000147265622 DE On-Demand Anodyne ENV 62 50 CCc1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147265624 DG On-Demand Anodyne KCNA5 32 51 CC[C@@H]1CN(C(=O)c2ccncc2)CC[C@@H]1N ZINC000147265630 BD On-Demand Anodyne L3MBTL1 0 40 CC[C@@H]1CN(C(=O)c2ccncc2)CC[C@@H]1N ZINC000147265630 BD On-Demand Anodyne L3MBTL3 69 40 CC(C)(CCC(=O)O)NC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147265670 CF For-Sale Anodyne NAMPT 22 40 CC(C)(CCC(=O)O)NC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147265670 CF For-Sale Anodyne GPR88 0 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne ACE 25 46 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne MME 48 46 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne LTA4H 21 45 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne ANPEP 45 32 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne NPR1 41 33 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne KLK3 64 39 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne CTSK 38 44 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne NPFFR2 53 36 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne TIMP3 65 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne C3AR1 56 33 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne HDAC8 27 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne HDAC10 47 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne MMP2 27 54 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne MMP3 53 54 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne HLA-DRB1 33 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne HDAC1 22 45 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne HDAC2 32 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne HDAC3 31 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne HDAC6 32 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne PCSK5 41 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne FURIN 75 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne CCKBR 18 44 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne ACE2 58 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne HDAC11 62 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne MMP1 15 52 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne POLG_WNV 68 33 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne QRFPR 46 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne NPFFR1 69 36 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265739 EH On-Demand Anodyne NOD1 67 35 CCCCCCCCNC(=O)NC1CCC(C(=O)O)CC1 ZINC000147265742 CG On-Demand Mild EPHX2 42 70 CCCCCCCCNC(=O)NC1CCC(C(=O)O)CC1 ZINC000147265742 CG On-Demand Mild ASAH1 57 33 CCCCCCCCNC(=O)NC1CCC(C(=O)O)CC1 ZINC000147265742 CG On-Demand Mild LASR 44 31 CC(C)(C)c1nc(NN)cc(NC2CCCCCC2)n1 ZINC000147265750 CG For-Sale Anodyne HRH4 17 40 CC(C)(C)c1nc(NN)cc(NC2CCCCCC2)n1 ZINC000147265750 CG For-Sale Anodyne PRKD1 55 33 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)N3CCCCCC3)cc2)CC1 ZINC000147265788 GF On-Demand Mild EPHX2 22 45 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)N3CCCCCC3)cc2)CC1 ZINC000147265788 GF On-Demand Mild TGM2 46 39 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)N3CCCCCC3)cc2)CC1 ZINC000147265788 GF On-Demand Mild F13A1 44 40 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)N3CCCCCC3)cc2)CC1 ZINC000147265788 GF On-Demand Mild L3MBTL3 100 64 N#CC1CCN(C(=O)c2ccc(S(=O)(=O)N3CCCCCC3)cc2)CC1 ZINC000147265788 GF On-Demand Mild NAMPT 24 43 Cc1nc(NC(=O)c2ccc(F)cc2)sc1-c1nc2ccccc2n1C(F)F ZINC000147265803 HK On-Demand Anodyne PIK3CG 16 42 C[C@@H](CNS(=O)(=O)c1c(Cl)cccc1Cl)CC(=O)O ZINC000147265809 EE On-Demand Anodyne ITGAV 17 45 COCC[n+]1cccc(C)c1 ZINC000147265811 AC For-Sale Anodyne Q0GKD7_LEIDO 25 46 CCc1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147265832 DG On-Demand Anodyne KCNA5 32 51 C[C@@H](N)CCCC(=O)NN(C)C ZINC000147265838 AC For-Sale Reactive NOD1 50 33 C[C@@H](N)CCCC(=O)NN(C)C ZINC000147265838 AC For-Sale Reactive KDM7A 0 48 CC[C@H]1CN(C(=O)c2ccncc2)CC[C@@H]1N ZINC000147265847 BD On-Demand Anodyne L3MBTL1 0 40 CC[C@H]1CN(C(=O)c2ccncc2)CC[C@@H]1N ZINC000147265847 BD On-Demand Anodyne L3MBTL3 69 40 CC(C)(CCC(=O)O)NC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147265869 CF For-Sale Anodyne NAMPT 22 40 CC(C)(CCC(=O)O)NC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147265869 CF For-Sale Anodyne GPR88 0 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne ACE 25 46 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne MME 48 46 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne LTA4H 21 45 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne ANPEP 45 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne NPR1 41 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne KLK3 64 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne CTSK 38 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne NPFFR2 53 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne TIMP3 65 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne C3AR1 56 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne HDAC8 27 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne HDAC10 47 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne MMP2 27 54 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne MMP3 53 54 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne HLA-DRB1 33 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne HDAC1 22 45 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne HDAC2 32 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne HDAC3 31 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne HDAC6 32 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne PCSK5 41 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne FURIN 75 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne CCKBR 18 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne ACE2 58 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne HDAC11 62 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne MMP1 15 52 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne POLG_WNV 68 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne QRFPR 46 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne NPFFR1 69 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(Nc2ccccc2)cc1 ZINC000147265947 EH On-Demand Anodyne NOD1 67 35 CC(C)S(=O)(=O)c1ccc(-c2cnc(N)c(C(=O)NN)n2)cc1 ZINC000147265959 EC For-Sale Reactive GSK3B 19 46 CC(C)S(=O)(=O)c1ccc(-c2cnc(N)c(C(=O)NN)n2)cc1 ZINC000147265959 EC For-Sale Reactive PIK3CG 17 47 CC(C)S(=O)(=O)c1ccc(-c2cnc(N)c(C(=O)NN)n2)cc1 ZINC000147265959 EC For-Sale Reactive ATR 78 75 CC(C)S(=O)(=O)c1ccc(-c2cnc(N)c(C(=O)NN)n2)cc1 ZINC000147265959 EC For-Sale Reactive TYRO3 44 38 CCCCCCCCNC(=O)N(CC)CC(=O)O ZINC000147265968 CE For-Sale Mild CPT1A 23 40 CCCCCCCCNC(=O)N(CC)CC(=O)O ZINC000147265968 CE For-Sale Mild S1PR2 43 36 CCCCCCCCNC(=O)N(CC)CC(=O)O ZINC000147265968 CE For-Sale Mild EPHX2 29 46 CCCCCCCCNC(=O)N(CC)CC(=O)O ZINC000147265968 CE For-Sale Mild ASAH1 80 33 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc(Cn2cccn2)cc1 ZINC000147266016 GG On-Demand Anodyne AGTR1 25 42 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc(Cn2cccn2)cc1 ZINC000147266016 GG On-Demand Anodyne FLT1 18 42 CCOc1ccc(C(=O)N2CCC(C#N)CC2)cc1OCC ZINC000147266030 DF On-Demand Mild HRH3 27 41 CCOc1ccc(C(=O)N2CCC(C#N)CC2)cc1OCC ZINC000147266030 DF On-Demand Mild SSTR5 43 34 CCOc1ccc(C(=O)N2CCC(C#N)CC2)cc1OCC ZINC000147266030 DF On-Demand Mild L3MBTL3 69 39 CC(C)CCCCNCc1ccc2c(c1)CCCN2C ZINC000147266047 CH For-Sale Clean LEF 54 34 CC[C@@H]1CN(C(=O)c2ccncc2)CC[C@H]1N ZINC000147266076 BD On-Demand Anodyne L3MBTL1 0 40 CC[C@@H]1CN(C(=O)c2ccncc2)CC[C@H]1N ZINC000147266076 BD On-Demand Anodyne L3MBTL3 69 40 CC(C)(CCC(=O)O)NC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147266099 CF For-Sale Anodyne NAMPT 22 40 CC(C)(CCC(=O)O)NC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147266099 CF For-Sale Anodyne GPR88 0 41 C#CCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266114 DC For-Sale Mild CA2 37 42 C#CCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266114 DC For-Sale Mild CA14 17 42 C#CCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266114 DC For-Sale Mild CA12 21 42 C#CCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266114 DC For-Sale Mild PTGDR2 42 39 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C(C)(C)C ZINC000147266178 CG For-Sale Mild PDF 50 40 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C(C)(C)C ZINC000147266178 CG For-Sale Mild CPT1A 44 51 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C(C)(C)C ZINC000147266178 CG For-Sale Mild EPHX2 54 48 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C(C)(C)C ZINC000147266178 CG For-Sale Mild ASAH1 82 35 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C(C)(C)C ZINC000147266178 CG For-Sale Mild NOD1 64 38 CCCCCCCCNC(=O)N[C@@H](C(=O)O)C(C)(C)C ZINC000147266178 CG For-Sale Mild CQSS 49 30 C[C@@H]1Cc2ccccc2N1S(=O)(=O)c1cccc(C(=O)N2CCC(C#N)CC2)c1 ZINC000147266258 HG On-Demand Mild AKR1C3 55 47 CC[C@H]1CN(C(=O)c2ccncc2)CC[C@H]1N ZINC000147266282 BD On-Demand Anodyne L3MBTL1 0 40 CC[C@H]1CN(C(=O)c2ccncc2)CC[C@H]1N ZINC000147266282 BD On-Demand Anodyne L3MBTL3 69 40 CC[C@@H](C)C(=O)c1c(F)ccc(C)c1F ZINC000147266335 BH For-Sale Anodyne LEF 59 32 CCCCCCCCNC(=O)N[C@@](C)(CCC)C(=O)O ZINC000147266408 CG For-Sale Mild CPT1A 0 41 CCCCCCCCNC(=O)N[C@@](C)(CCC)C(=O)O ZINC000147266408 CG For-Sale Mild EPHX2 44 44 CCCCCCCCNC(=O)N[C@@](C)(CCC)C(=O)O ZINC000147266408 CG For-Sale Mild ASAH1 71 32 CCOC(=O)CN(C(=O)Cc1cccc(C(F)(F)F)c1)C1CCC1 ZINC000147266440 EG On-Demand Anodyne ACE 25 42 CCOC(=O)CN(C(=O)Cc1cccc(C(F)(F)F)c1)C1CCC1 ZINC000147266440 EG On-Demand Anodyne TACR1 34 40 CCOC(=O)CN(C(=O)Cc1cccc(C(F)(F)F)c1)C1CCC1 ZINC000147266440 EG On-Demand Anodyne CACNA1B 48 34 CCOC(=O)CN(C(=O)Cc1cccc(C(F)(F)F)c1)C1CCC1 ZINC000147266440 EG On-Demand Anodyne AMY2 43 30 CCOC(=O)CN(C(=O)Cc1cccc(C(F)(F)F)c1)C1CCC1 ZINC000147266440 EG On-Demand Anodyne PTGDR2 21 42 CCOC(=O)CN(C(=O)Cc1cccc(C(F)(F)F)c1)C1CCC1 ZINC000147266440 EG On-Demand Anodyne SCD1 30 40 CCOC(=O)CN(C(=O)Cc1cccc(C(F)(F)F)c1)C1CCC1 ZINC000147266440 EG On-Demand Anodyne PDS 43 34 CC[C@@H]1CN(C(=O)c2ccc(F)cc2)CC[C@@H]1N ZINC000147266488 CE On-Demand Anodyne HSD11B1 0 51 CC[C@@H]1CN(C(=O)c2ccc(F)cc2)CC[C@@H]1N ZINC000147266488 CE On-Demand Anodyne SLC18A3 29 45 CC[C@@H]1CN(C(=O)c2ccc(F)cc2)CC[C@@H]1N ZINC000147266488 CE On-Demand Anodyne SLC9A1 41 38 CC[C@@H]1CN(C(=O)c2ccc(F)cc2)CC[C@@H]1N ZINC000147266488 CE On-Demand Anodyne L3MBTL1 0 43 CC[C@@H]1CN(C(=O)c2ccc(F)cc2)CC[C@@H]1N ZINC000147266488 CE On-Demand Anodyne L3MBTL3 78 43 C[C@H](CNS(=O)(=O)c1cccc(F)c1)CC(=O)O ZINC000147266500 CD On-Demand Anodyne LIMK2 23 40 CC[C@H](C)C(=O)c1c(F)ccc(C)c1F ZINC000147266520 BH For-Sale Anodyne LEF 59 32 C#CCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266532 DC For-Sale Mild CA2 32 40 C#CCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266532 DC For-Sale Mild CA1 23 40 C#CCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266532 DC For-Sale Mild CA4 27 40 C#CCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266532 DC For-Sale Mild CA14 15 40 CCCNc1ncc(Br)c(Oc2ccccc2C(C)C)n1 ZINC000147266549 FJ For-Sale Anodyne P2RX2 64 37 CCCNc1ncc(Br)c(Oc2ccccc2C(C)C)n1 ZINC000147266549 FJ For-Sale Anodyne P2RX3 44 37 Nc1cc(Cl)cc(-c2nc(-c3ccccc3F)no2)c1 ZINC000147266584 CH For-Sale Anodyne LUCI_PHOPE 36 44 CC(C)CCO[C@@H](C)C(=O)Nc1ccccc1OC(F)(F)F ZINC000147266591 DH On-Demand Anodyne P2RY1 45 39 CC(C)CCO[C@@H](C)C(=O)Nc1ccccc1OC(F)(F)F ZINC000147266591 DH On-Demand Anodyne KCNK3 19 40 CC(C)CCO[C@@H](C)C(=O)Nc1ccccc1OC(F)(F)F ZINC000147266591 DH On-Demand Anodyne KCNK9 25 40 O=C(O)C1(NCc2ccc([N+](=O)[O-])cc2)CCC1 ZINC000147266606 CD On-Demand Bother SLC27A4 42 32 O=C(O)C1(NCc2ccc([N+](=O)[O-])cc2)CCC1 ZINC000147266606 CD On-Demand Bother LUXR 16 40 CCCCCCCCNC(=O)N[C@](C)(CCC)C(=O)O ZINC000147266629 CG For-Sale Mild CPT1A 0 41 CCCCCCCCNC(=O)N[C@](C)(CCC)C(=O)O ZINC000147266629 CG For-Sale Mild EPHX2 44 44 CCCCCCCCNC(=O)N[C@](C)(CCC)C(=O)O ZINC000147266629 CG For-Sale Mild ASAH1 71 32 CCNc1cccc(N[C@@H](C)CCCN(CC)CC)n1 ZINC000147266633 CG For-Sale Anodyne CACNA2D1 28 54 CCNc1cccc(N[C@@H](C)CCCN(CC)CC)n1 ZINC000147266633 CG For-Sale Anodyne RBP_CHICK 0 42 CC[C@H](Oc1ccc(Cl)c(F)c1)C(=O)c1ccccc1 ZINC000147266638 CJ For-Sale Anodyne PPARA 23 41 CC[C@H](Oc1ccc(Cl)c(F)c1)C(=O)c1ccccc1 ZINC000147266638 CJ For-Sale Anodyne PDS 64 40 CC[C@H]1CN(C(=O)c2ccc(F)cc2)CC[C@@H]1N ZINC000147266668 CE On-Demand Anodyne HSD11B1 0 51 CC[C@H]1CN(C(=O)c2ccc(F)cc2)CC[C@@H]1N ZINC000147266668 CE On-Demand Anodyne SLC18A3 29 45 CC[C@H]1CN(C(=O)c2ccc(F)cc2)CC[C@@H]1N ZINC000147266668 CE On-Demand Anodyne SLC9A1 41 38 CC[C@H]1CN(C(=O)c2ccc(F)cc2)CC[C@@H]1N ZINC000147266668 CE On-Demand Anodyne L3MBTL1 0 43 CC[C@H]1CN(C(=O)c2ccc(F)cc2)CC[C@@H]1N ZINC000147266668 CE On-Demand Anodyne L3MBTL3 78 43 C#CCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266721 DC For-Sale Mild CA2 32 40 C#CCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266721 DC For-Sale Mild CA1 23 40 C#CCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266721 DC For-Sale Mild CA4 27 40 C#CCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266721 DC For-Sale Mild CA14 15 40 C[C@@H](CNS(=O)(=O)c1cccc(F)c1)CC(=O)O ZINC000147266729 CD On-Demand Anodyne LIMK2 23 40 O=C(Nc1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1)NC1CC1 ZINC000147266767 GH On-Demand Anodyne EPHX2 47 41 Nc1cc(Br)cc(-c2nc(-c3ccccc3F)no2)c1 ZINC000147266781 EH For-Sale Anodyne LUCI_PHOPE 37 45 CC(C)CCO[C@H](C)C(=O)Nc1ccccc1OC(F)(F)F ZINC000147266801 DH On-Demand Anodyne P2RY1 45 39 CC(C)CCO[C@H](C)C(=O)Nc1ccccc1OC(F)(F)F ZINC000147266801 DH On-Demand Anodyne KCNK3 19 40 CC(C)CCO[C@H](C)C(=O)Nc1ccccc1OC(F)(F)F ZINC000147266801 DH On-Demand Anodyne KCNK9 25 40 CCNc1cccc(N[C@H](C)CCCN(CC)CC)n1 ZINC000147266841 CG For-Sale Anodyne CACNA2D1 28 54 CCNc1cccc(N[C@H](C)CCCN(CC)CC)n1 ZINC000147266841 CG For-Sale Anodyne RBP_CHICK 0 42 CCCCCCCCNC(=O)N1CCO[C@H](C(=O)O)C1 ZINC000147266846 CD On-Demand Mild ASAH1 101 42 CC[C@@H](Oc1ccc(Cl)c(F)c1)C(=O)c1ccccc1 ZINC000147266852 CJ For-Sale Anodyne PPARA 23 41 CC[C@@H](Oc1ccc(Cl)c(F)c1)C(=O)c1ccccc1 ZINC000147266852 CJ For-Sale Anodyne PDS 64 40 CC[C@@H]1CN(C(=O)c2ccc(F)cc2)CC[C@H]1N ZINC000147266881 CE On-Demand Anodyne HSD11B1 0 51 CC[C@@H]1CN(C(=O)c2ccc(F)cc2)CC[C@H]1N ZINC000147266881 CE On-Demand Anodyne SLC18A3 29 45 CC[C@@H]1CN(C(=O)c2ccc(F)cc2)CC[C@H]1N ZINC000147266881 CE On-Demand Anodyne SLC9A1 41 38 CC[C@@H]1CN(C(=O)c2ccc(F)cc2)CC[C@H]1N ZINC000147266881 CE On-Demand Anodyne L3MBTL1 0 43 CC[C@@H]1CN(C(=O)c2ccc(F)cc2)CC[C@H]1N ZINC000147266881 CE On-Demand Anodyne L3MBTL3 78 43 O=c1cnc(-c2ccccc2)cn1Cc1ccc(Cl)cc1 ZINC000147266889 CH On-Demand Anodyne CYP11B1 21 50 O=c1cnc(-c2ccccc2)cn1Cc1ccc(Cl)cc1 ZINC000147266889 CH On-Demand Anodyne CYP11B2 22 50 CCC(CC)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266933 ED For-Sale Anodyne CA2 35 43 CCC(CC)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266933 ED For-Sale Anodyne CA1 27 43 CCC(CC)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266933 ED For-Sale Anodyne CA4 28 43 CCC(CC)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147266933 ED For-Sale Anodyne PTGDR2 42 40 CCCCCCCCNC(=O)N1CCO[C@@H](C(=O)O)C1 ZINC000147267001 CD On-Demand Mild ASAH1 101 42 C[C@H](CNS(=O)(=O)c1cccc(Cl)c1)CC(=O)O ZINC000147267021 CD On-Demand Anodyne TBXA2R 43 35 C[C@H](CNS(=O)(=O)c1cccc(Cl)c1)CC(=O)O ZINC000147267021 CD On-Demand Anodyne FBP1 33 43 C[C@H](CNS(=O)(=O)c1cccc(Cl)c1)CC(=O)O ZINC000147267021 CD On-Demand Anodyne OXER1 40 34 CCOc1ccccc1C(=O)COc1ccc(Cl)c(F)c1 ZINC000147267066 DI For-Sale Anodyne HCN1 48 32 CCOc1ccccc1C(=O)COc1ccc(Cl)c(F)c1 ZINC000147267066 DI For-Sale Anodyne HCN4 40 31 CCOc1ccccc1C(=O)COc1ccc(Cl)c(F)c1 ZINC000147267066 DI For-Sale Anodyne KCNK3 27 41 CCOc1ccccc1C(=O)COc1ccc(Cl)c(F)c1 ZINC000147267066 DI For-Sale Anodyne KCNK9 16 41 CC[C@H]1CN(C(=O)c2ccc(F)cc2)CC[C@H]1N ZINC000147267084 CE On-Demand Anodyne HSD11B1 0 51 CC[C@H]1CN(C(=O)c2ccc(F)cc2)CC[C@H]1N ZINC000147267084 CE On-Demand Anodyne SLC18A3 29 45 CC[C@H]1CN(C(=O)c2ccc(F)cc2)CC[C@H]1N ZINC000147267084 CE On-Demand Anodyne SLC9A1 41 38 CC[C@H]1CN(C(=O)c2ccc(F)cc2)CC[C@H]1N ZINC000147267084 CE On-Demand Anodyne L3MBTL1 0 43 CC[C@H]1CN(C(=O)c2ccc(F)cc2)CC[C@H]1N ZINC000147267084 CE On-Demand Anodyne L3MBTL3 78 43 CS(=O)(=O)NC(=O)C1(c2ccc(F)cc2)CCOCC1 ZINC000147267115 DC On-Demand Anodyne MMP13 16 41 CN(C)NC(=O)CN ZINC000147267171 AA For-Sale Reactive KDM7A 0 52 CCN(C)C(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147267192 DC For-Sale Anodyne PTGDR2 41 41 CCCCCCCCNC(=O)Cc1nc(CCl)cs1 ZINC000147267215 DH For-Sale Reactive ASAH1 90 38 C[C@@H](CNS(=O)(=O)c1cccc(Cl)c1)CC(=O)O ZINC000147267225 CD On-Demand Anodyne TBXA2R 43 35 C[C@@H](CNS(=O)(=O)c1cccc(Cl)c1)CC(=O)O ZINC000147267225 CD On-Demand Anodyne FBP1 33 43 C[C@@H](CNS(=O)(=O)c1cccc(Cl)c1)CC(=O)O ZINC000147267225 CD On-Demand Anodyne OXER1 40 34 CN(C)C1(CNC(=O)C(=O)O)CCCC1 ZINC000147267227 BC On-Demand Anodyne SLC6A5 15 42 CN(Cc1cccc(Cl)c1)C(=O)CNC1(C(=O)O)CCC1 ZINC000147267241 DD For-Sale Anodyne TACR3 36 40 CC[C@@H]1CN(C(=O)c2ccccn2)CC[C@@H]1N ZINC000147267299 BD On-Demand Anodyne CCR8 15 40 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267300 EE On-Demand Anodyne KIT 19 46 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267300 EE On-Demand Anodyne PLA2G7 46 42 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267300 EE On-Demand Anodyne BDKRB1 0 41 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267300 EE On-Demand Anodyne GRM4 59 42 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267300 EE On-Demand Anodyne NR1H4 23 40 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267300 EE On-Demand Anodyne BRAF 29 46 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267300 EE On-Demand Anodyne NR2E3 68 38 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267300 EE On-Demand Anodyne SHH 35 41 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267300 EE On-Demand Anodyne KCNK3 61 38 CS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267300 EE On-Demand Anodyne KCNK9 62 37 O=CNc1ccc(-n2ccnc2)cc1 ZINC000147267333 AD For-Sale Anodyne CYP2C19 18 44 CN(C)NC(=O)C[C@H](N)c1ccccc1 ZINC000147267389 BC For-Sale Reactive ANPEP 19 44 CCCCCCCCn1cnc2c(C(=O)O)cccc21 ZINC000147267427 CI For-Sale Mild CNR1 26 44 CCCCCCCCn1cnc2c(C(=O)O)cccc21 ZINC000147267427 CI For-Sale Mild CNR2 40 44 CCCCCCCCn1cnc2c(C(=O)O)cccc21 ZINC000147267427 CI For-Sale Mild PLA2G4B 79 36 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147267444 GF On-Demand Anodyne MAPK14 15 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147267444 GF On-Demand Anodyne PRNP 25 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147267444 GF On-Demand Anodyne KCNK3 121 54 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147267444 GF On-Demand Anodyne KCNK9 66 44 CC[C@H]1CN(C(=O)c2ccccn2)CC[C@@H]1N ZINC000147267487 BD On-Demand Anodyne CCR8 15 40 COc1ccc(OC)c(CNCC(F)F)c1 ZINC000147267519 BE On-Demand Anodyne DRTS_TOXGO 16 46 COc1ccc(OC)c(CNCC(F)F)c1 ZINC000147267519 BE On-Demand Anodyne DYR_PNECA 15 41 COc1ccc(OC)c(CNCC(F)F)c1 ZINC000147267519 BE On-Demand Anodyne MT-ND1 17 43 COc1ccc(OC)c(CNCC(F)F)c1 ZINC000147267519 BE On-Demand Anodyne PHES 0 40 CS(=O)(=O)Nc1ccc(F)cc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267532 FE On-Demand Anodyne PLA2G7 39 42 CS(=O)(=O)Nc1ccc(F)cc1C(=O)Nc1ccc2nccnc2c1 ZINC000147267532 FE On-Demand Anodyne GRM4 33 42 C[C@@H](CN1CCCC1)NC(=O)c1cccc2c1OCCN2 ZINC000147267580 CD For-Sale Anodyne PLD1 47 36 Cc1cc(C(=O)NCC(=O)Nc2c(C)cc(C)cc2C)cc([N+](=O)[O-])c1 ZINC000147267614 FG On-Demand Bother METC 0 59 CC(C)CCO[C@@H](C)C(=O)NCc1ccc(C(F)(F)F)cc1 ZINC000147267628 DH On-Demand Anodyne PPARA 23 43 CC(C)CCO[C@@H](C)C(=O)NCc1ccc(C(F)(F)F)cc1 ZINC000147267628 DH On-Demand Anodyne TRPV1 26 47 CC(C)CCO[C@@H](C)C(=O)NCc1ccc(C(F)(F)F)cc1 ZINC000147267628 DH On-Demand Anodyne PPARD 29 40 CC(C)CCO[C@@H](C)C(=O)NCc1ccc(C(F)(F)F)cc1 ZINC000147267628 DH On-Demand Anodyne AMP1_PLAFQ 20 42 CN(C)NC(=O)C[C@@H](N)c1ccccc1 ZINC000147267629 BC For-Sale Reactive ANPEP 19 44 CCCCCCCCn1c(C)nc2c(C(=O)O)cccc21 ZINC000147267647 CI For-Sale Mild CNR1 26 48 CCCCCCCCn1c(C)nc2c(C(=O)O)cccc21 ZINC000147267647 CI For-Sale Mild AGTR1 46 38 CCCCCCCCn1c(C)nc2c(C(=O)O)cccc21 ZINC000147267647 CI For-Sale Mild CNR2 36 48 CCCCCCCCn1c(C)nc2c(C(=O)O)cccc21 ZINC000147267647 CI For-Sale Mild AGTR1B 37 40 CCCCCCCCn1c(C)nc2c(C(=O)O)cccc21 ZINC000147267647 CI For-Sale Mild PLA2G4B 52 36 CCCCCCCCn1c(C)nc2c(C(=O)O)cccc21 ZINC000147267647 CI For-Sale Mild TLR8 0 50 CCCCCCCCn1c(C)nc2c(C(=O)O)cccc21 ZINC000147267647 CI For-Sale Mild OXER1 63 36 COc1cccc(COc2ccc(Cl)cc2S(N)(=O)=O)n1 ZINC000147267648 ED For-Sale Anodyne CPT1A 43 30 CN(C)C1(CNC(=O)c2ccc(C(=O)O)o2)CCCC1 ZINC000147267653 CD For-Sale Anodyne SLC6A5 16 48 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147267660 GF On-Demand Anodyne MAPK14 15 43 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147267660 GF On-Demand Anodyne PRNP 25 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147267660 GF On-Demand Anodyne KCNK3 121 54 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147267660 GF On-Demand Anodyne KCNK9 66 44 CC[C@@H]1CN(C(=O)c2ccccn2)CC[C@H]1N ZINC000147267674 BD On-Demand Anodyne CCR8 15 40 O=C(COc1ccc(Cl)c(F)c1)c1cccc(F)c1 ZINC000147267712 CH For-Sale Anodyne KMO 0 43 O=C(COc1ccc(Cl)c(F)c1)c1cccc(F)c1 ZINC000147267712 CH For-Sale Anodyne SENP1 0 45 CC(C)c1ccccc1Oc1ccnc(N)n1 ZINC000147267749 BF For-Sale Anodyne P2RX2 48 39 NC(=O)[C@H]1CCCN1C(=O)/C=C/Sc1ccccc1 ZINC000147267770 CD On-Demand Anodyne PREP 71 38 NC(=O)[C@H]1CCCN1C(=O)/C=C/Sc1ccccc1 ZINC000147267770 CD On-Demand Anodyne PEPD 0 42 CCCC[C@H](NC(N)=O)C(=O)NNc1nc2ccccc2c(=O)n1CC ZINC000147267776 FD On-Demand Reactive CCKBR 24 41 NC(=O)NCCCCC(=O)Nc1ccc2nccnc2c1 ZINC000147267780 CD On-Demand Anodyne HDAC1 22 43 NC(=O)NCCCCC(=O)Nc1ccc2nccnc2c1 ZINC000147267780 CD On-Demand Anodyne HDAC2 26 43 NC(=O)NCCCCC(=O)Nc1ccc2nccnc2c1 ZINC000147267780 CD On-Demand Anodyne HDAC3 45 37 NC(=O)NCCCCC(=O)Nc1ccc2nccnc2c1 ZINC000147267780 CD On-Demand Anodyne HDAC6 42 37 C[C@H](CN1CCCC1)NC(=O)c1cccc2c1OCCN2 ZINC000147267783 CD For-Sale Anodyne PLD1 47 36 CCC(=O)N1CCN2CCC1CC2 ZINC000147267784 AC On-Demand Anodyne CHRNA4 15 43 CCCCCCCCn1c(C)nc2cc(C(=O)O)ccc21 ZINC000147267833 CI For-Sale Mild CNR2 22 44 CCCCCCCCn1c(C)nc2cc(C(=O)O)ccc21 ZINC000147267833 CI For-Sale Mild RARB 22 42 CCCCCCCCn1c(C)nc2cc(C(=O)O)ccc21 ZINC000147267833 CI For-Sale Mild PLA2G4A 33 42 CCCCCCCCn1c(C)nc2cc(C(=O)O)ccc21 ZINC000147267833 CI For-Sale Mild PLA2G4B 56 39 CCCCCCCCn1c(C)nc2cc(C(=O)O)ccc21 ZINC000147267833 CI For-Sale Mild OXER1 60 32 CC(C)CCO[C@H](C)C(=O)NCc1ccc(C(F)(F)F)cc1 ZINC000147267841 DH On-Demand Anodyne PPARA 23 43 CC(C)CCO[C@H](C)C(=O)NCc1ccc(C(F)(F)F)cc1 ZINC000147267841 DH On-Demand Anodyne TRPV1 26 47 CC(C)CCO[C@H](C)C(=O)NCc1ccc(C(F)(F)F)cc1 ZINC000147267841 DH On-Demand Anodyne PPARD 29 40 CC(C)CCO[C@H](C)C(=O)NCc1ccc(C(F)(F)F)cc1 ZINC000147267841 DH On-Demand Anodyne AMP1_PLAFQ 20 42 O=C(CNC1(C(=O)O)CCC1)N1CCC[C@@H]2CCCC[C@H]21 ZINC000147267882 CD For-Sale Anodyne DPP4 19 41 CC[C@H]1CN(C(=O)c2ccccn2)CC[C@H]1N ZINC000147267885 BD On-Demand Anodyne CCR8 15 40 CCCN(CC(=O)O)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147267892 CE For-Sale Anodyne GPR88 0 47 CC(C)c1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147267894 CE On-Demand Anodyne TBXA2R 42 33 CNCc1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147267945 CH For-Sale Anodyne SLC6A4 16 62 CCCC[C@@H](NC(N)=O)C(=O)NNc1nc2ccccc2c(=O)n1CC ZINC000147267971 FD On-Demand Reactive CCKBR 24 41 COc1ccc([N+](=O)[O-])c(C(=O)N2CCC[C@@H](C(=O)Nc3ccc(C)cn3)C2)c1 ZINC000147267973 GF On-Demand Bother LUCI_LUCLA 16 42 COc1ccc([N+](=O)[O-])c(C(=O)N2CCC[C@@H](C(=O)Nc3ccc(C)cn3)C2)c1 ZINC000147267973 GF On-Demand Bother MAP3K12 17 40 Cc1ccc(NS(C)(=O)=O)c(C(=O)Nc2ccc3nccnc3c2)c1 ZINC000147267987 FF On-Demand Anodyne PLA2G7 35 41 Cc1ccc(NS(C)(=O)=O)c(C(=O)Nc2ccc3nccnc3c2)c1 ZINC000147267987 FF On-Demand Anodyne KCNK3 69 36 Cc1ccc(NS(C)(=O)=O)c(C(=O)Nc2ccc3nccnc3c2)c1 ZINC000147267987 FF On-Demand Anodyne KCNK9 54 35 NS(=O)(=O)c1ccccc1NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147267991 CB For-Sale Anodyne CA2 16 46 NS(=O)(=O)c1ccccc1NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147267991 CB For-Sale Anodyne CA4 19 46 NS(=O)(=O)c1ccccc1NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147267991 CB For-Sale Anodyne CYNT 15 42 CCCN(CC(=O)O)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147268061 CE For-Sale Anodyne GPR88 0 47 O=C(CNC1(C(=O)O)CCC1)N1CCC[C@@H]2CCCC[C@@H]21 ZINC000147268067 CD For-Sale Anodyne DPP4 19 41 CC(C)c1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147268071 CE On-Demand Anodyne TBXA2R 42 33 NS(=O)(=O)c1cc(Cl)ccc1OCc1ccncc1Cl ZINC000147268115 EF For-Sale Anodyne CA14 29 46 CN(C)C1(CNC(=O)c2cccc(C(=O)O)n2)CCCC1 ZINC000147268122 CD For-Sale Anodyne SLC6A5 16 47 CN(C)C1(CNC(=O)c2cccc(C(=O)O)n2)CCCC1 ZINC000147268122 CD For-Sale Anodyne HCN1 69 36 CN(C)C1(CNC(=O)c2cccc(C(=O)O)n2)CCCC1 ZINC000147268122 CD For-Sale Anodyne HCN4 51 34 Cc1cc(NC(=O)C(F)F)ccc1F ZINC000147268161 BE On-Demand Anodyne LEF 95 44 CNCc1ccc(Oc2ccc(Cl)c(F)c2)c(F)c1 ZINC000147268164 CI For-Sale Anodyne SLC6A4 20 57 COc1ccc([N+](=O)[O-])c(C(=O)N2CCC[C@H](C(=O)Nc3ccc(C)cn3)C2)c1 ZINC000147268175 GF On-Demand Bother LUCI_LUCLA 16 42 COc1ccc([N+](=O)[O-])c(C(=O)N2CCC[C@H](C(=O)Nc3ccc(C)cn3)C2)c1 ZINC000147268175 GF On-Demand Bother MAP3K12 17 40 O=C(CNC1(C(=O)O)CCC1)N1CCC[C@H]2CCCC[C@H]21 ZINC000147268219 CD For-Sale Anodyne DPP4 19 41 CC(C)c1ccccc1Oc1nc(N)nc2ccccc12 ZINC000147268256 CI For-Sale Anodyne DHFR 19 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147268258 GD On-Demand Anodyne KCNK3 93 50 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147268258 GD On-Demand Anodyne KCNK9 46 38 CCCN(CC(=O)O)C(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147268275 CE For-Sale Anodyne GPR88 0 47 CCCCCCCCC(=O)N1CC[C@H](N)[C@H](CC)C1 ZINC000147268304 CG On-Demand Mild CQSS 54 33 CNC(=O)c1ccc2ccn(Cc3c[nH]cn3)c2c1 ZINC000147268329 CD For-Sale Anodyne CYP17A1 25 47 CCCCCNC(=O)C[C@@H]1CNc2ccccc21 ZINC000147268373 BF For-Sale Anodyne ASAH1 76 36 NS(=O)(=O)c1ccccc1NC(=O)[C@H]1CCC(=O)NC1 ZINC000147268379 CB For-Sale Anodyne CA2 16 46 NS(=O)(=O)c1ccccc1NC(=O)[C@H]1CCC(=O)NC1 ZINC000147268379 CB For-Sale Anodyne CA4 19 46 NS(=O)(=O)c1ccccc1NC(=O)[C@H]1CCC(=O)NC1 ZINC000147268379 CB For-Sale Anodyne CYNT 15 42 COCc1nc(C(=O)Nc2ccc(S(=O)(=O)NC(C)C)cc2)cs1 ZINC000147268384 FE On-Demand Anodyne MMP13 37 45 COCc1nc(C(=O)Nc2ccc(S(=O)(=O)NC(C)C)cc2)cs1 ZINC000147268384 FE On-Demand Anodyne GRM4 29 41 COCc1nc(C(=O)Nc2ccc(S(=O)(=O)NC(C)C)cc2)cs1 ZINC000147268384 FE On-Demand Anodyne MMP2 27 45 O=C(CNC1(C(=O)O)CCC1)N1CCC[C@H]2CCCC[C@@H]21 ZINC000147268443 CD For-Sale Anodyne DPP4 19 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147268454 GD On-Demand Anodyne KCNK3 93 50 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147268454 GD On-Demand Anodyne KCNK9 46 38 CN1CCC(Oc2cccc(Br)c2)CC1 ZINC000147268471 CF For-Sale Anodyne HRH3 25 49 CN1CCC(Oc2cccc(Br)c2)CC1 ZINC000147268471 CF For-Sale Anodyne CHRNA10 49 35 CCCN(CC(=O)O)C(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147268482 CE For-Sale Anodyne GPR88 0 47 CCCCCNC(=O)C[C@H]1CNc2ccccc21 ZINC000147268497 BF For-Sale Anodyne ASAH1 76 36 CCCCCCCCC(=O)N1CC[C@@H](N)[C@H](CC)C1 ZINC000147268509 CG On-Demand Mild CQSS 54 33 CN(C)C1(CNC(=O)c2ccc(C(=O)O)cc2)CCCC1 ZINC000147268527 CD On-Demand Anodyne RARA 44 36 CN(C)C1(CNC(=O)c2ccc(C(=O)O)cc2)CCCC1 ZINC000147268527 CD On-Demand Anodyne RXRG 60 33 CN(C)C1(CNC(=O)c2ccc(C(=O)O)cc2)CCCC1 ZINC000147268527 CD On-Demand Anodyne RXRA 41 33 CN(C)C1(CNC(=O)c2ccc(C(=O)O)cc2)CCCC1 ZINC000147268527 CD On-Demand Anodyne RXRB 59 35 CN(C)C1(CNC(=O)c2ccc(C(=O)O)cc2)CCCC1 ZINC000147268527 CD On-Demand Anodyne SLC6A5 19 54 CN(C)C1(CNC(=O)c2ccc(C(=O)O)cc2)CCCC1 ZINC000147268527 CD On-Demand Anodyne HCN1 51 33 CN(C)C1(CNC(=O)c2ccc(C(=O)O)cc2)CCCC1 ZINC000147268527 CD On-Demand Anodyne HCN4 49 33 O=C1CC[C@@H](C(=O)Nc2cccc(O)c2)CN1 ZINC000147268612 BC On-Demand Anodyne PARP10 0 53 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147268613 BB For-Sale Reactive OPRM1 82 69 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147268613 BB For-Sale Reactive OPRD1 79 53 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147268613 BB For-Sale Reactive OPRK1 24 45 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147268613 BB For-Sale Reactive MME 38 44 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147268613 BB For-Sale Reactive SLC15A1 0 44 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147268613 BB For-Sale Reactive PDYN 0 41 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147268613 BB For-Sale Reactive GRIA1 59 41 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147268613 BB For-Sale Reactive YARS 104 52 CN(C)NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147268613 BB For-Sale Reactive SLC15A2 0 60 CC[C@@H](c1ccccn1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147268639 KK Annotated Anodyne TP53 45 70 CC[C@@H](c1ccccn1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147268639 KK Annotated Anodyne MDM2 256 70 C[C@H](CNS(=O)(=O)c1ccc(F)cc1[N+](=O)[O-])CC(=O)O ZINC000147268654 DD For-Sale Bother COLA 67 36 CCCCCCCCC(=O)N1CC[C@H](N)[C@@H](CC)C1 ZINC000147268694 CG On-Demand Mild CQSS 54 33 CC(C)[C@@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147268726 ED For-Sale Anodyne CA2 30 40 CC(C)[C@@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147268726 ED For-Sale Anodyne CA1 24 40 CS(=O)(=O)c1cccc(-c2ccc(-n3cc(C(F)(F)F)nc3-c3ccccc3Cl)cc2)c1 ZINC000147268744 JK Annotated Anodyne PTGS2 71 77 CS(=O)(=O)c1cccc(-c2ccc(-n3cc(C(F)(F)F)nc3-c3ccccc3Cl)cc2)c1 ZINC000147268744 JK Annotated Anodyne NR1H3 71 39 CS(=O)(=O)c1cccc(-c2ccc(-n3cc(C(F)(F)F)nc3-c3ccccc3Cl)cc2)c1 ZINC000147268744 JK Annotated Anodyne NR1H2 42 40 N#Cc1ccc(CSc2ccccc2C(=O)Nc2ccc3nccnc3c2)cc1 ZINC000147268784 GK On-Demand Mild NR2E3 61 34 O=C1CC[C@H](C(=O)Nc2cccc(O)c2)CN1 ZINC000147268797 BC On-Demand Anodyne PARP10 0 53 CNCc1ccc(Br)cc1Oc1ccc(Cl)c(F)c1 ZINC000147268808 EJ For-Sale Anodyne SLC6A4 24 79 Cc1ccc(C(=O)N2C[C@@]3(C)C[C@H]2CC(C)(C)C3)c(F)c1 ZINC000147268819 CI On-Demand Anodyne AVPR2 23 55 Cc1ccc(C(=O)N2C[C@@]3(C)C[C@H]2CC(C)(C)C3)c(F)c1 ZINC000147268819 CI On-Demand Anodyne AVPR1A 43 53 C[C@@H](CNS(=O)(=O)c1ccc(F)cc1[N+](=O)[O-])CC(=O)O ZINC000147268828 DD For-Sale Bother COLA 67 36 CCCCCCCCC(=O)N1CC[C@@H](N)[C@@H](CC)C1 ZINC000147268846 CG On-Demand Mild CQSS 54 33 CCCNCC(=O)NN(C)C ZINC000147268866 AB For-Sale Reactive KDM7A 0 43 CC1(c2ccc(Cl)cc2)CCCCC1 ZINC000147268867 BJ For-Sale Anodyne HSD11B1 15 41 CCCCCCCCn1c(C)cnc1SCC(=O)O ZINC000147268876 CH For-Sale Mild PLA2G4B 43 32 CC(C)[C@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147268908 ED For-Sale Anodyne CA2 30 40 CC(C)[C@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147268908 ED For-Sale Anodyne CA1 24 40 CC(C)[C@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147268908 ED For-Sale Anodyne CA4 25 40 CC[C@@H]1CN(C(=O)c2ccc3ccccc3n2)CC[C@@H]1N ZINC000147268986 CE On-Demand Anodyne SMO 46 36 Cc1ccc(C(=O)NCC2(N(C)C)CCCC2)c(F)c1 ZINC000147268988 CF On-Demand Anodyne HCN1 51 34 Cc1ccc(C(=O)NCC2(N(C)C)CCCC2)c(F)c1 ZINC000147268988 CF On-Demand Anodyne HCN4 48 34 C[C@H](CNS(=O)(=O)N1CCc2ccccc2C1)CC(=O)O ZINC000147269007 DC On-Demand Anodyne AKR1C3 62 44 CCN1CCN(c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)c(C)c2)CC1 ZINC000147269099 GH On-Demand Bother PRNP 35 42 CCN1CCN(c2ccc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)c(C)c2)CC1 ZINC000147269099 GH On-Demand Bother WDR5 34 40 COc1ccc(CC(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147269124 EG For-Sale Reactive OPRK1 0 43 COc1ccc(CC(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147269124 EG For-Sale Reactive GRM3 15 47 COc1ccc(CC(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147269124 EG For-Sale Reactive MMP13 31 44 COc1ccc(CC(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147269124 EG For-Sale Reactive MMP1 35 44 COc1ccc(CC(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147269124 EG For-Sale Reactive RORC 27 40 COc1ccc(CC(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147269124 EG For-Sale Reactive GPR183 0 43 CCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147269131 DC For-Sale Anodyne CA2 38 42 CCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147269131 DC For-Sale Anodyne CA1 36 42 CCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147269131 DC For-Sale Anodyne CA12 21 42 CCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147269131 DC For-Sale Anodyne PTGDR2 48 40 CCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147269131 DC For-Sale Anodyne PSBA 0 42 O=C(NCc1c(F)cccc1Cl)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147269139 IH On-Demand Anodyne MAP1 54 36 O=C(NCc1c(F)cccc1Cl)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147269139 IH On-Demand Anodyne GRM4 19 45 O=C(NCc1c(F)cccc1Cl)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147269139 IH On-Demand Anodyne PDE7A 16 53 COC(=O)[C@@H]1COc2ccc(Br)cc21 ZINC000147269175 CE In-Stock Anodyne HCRTR2 27 44 C[C@@H](CNS(=O)(=O)N1CCc2ccccc2C1)CC(=O)O ZINC000147269184 DC On-Demand Anodyne AKR1C3 62 44 CC[C@H]1CN(C(=O)c2ccc3ccccc3n2)CC[C@@H]1N ZINC000147269188 CE On-Demand Anodyne SMO 46 36 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269197 HI On-Demand Anodyne CA2 18 48 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269197 HI On-Demand Anodyne CA1 19 40 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269197 HI On-Demand Anodyne MMP13 33 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269197 HI On-Demand Anodyne CA4 18 48 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269197 HI On-Demand Anodyne MMP2 35 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269197 HI On-Demand Anodyne MMP9 15 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269197 HI On-Demand Anodyne CA12 15 42 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269197 HI On-Demand Anodyne CA9 17 42 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269197 HI On-Demand Anodyne IDO1 48 54 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269197 HI On-Demand Anodyne KDM1A 43 38 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269197 HI On-Demand Anodyne NAMPT 35 40 O=C(NC1C2CC3CC(C2)CC1C3)C1CCN(S(=O)(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147269228 JI On-Demand Anodyne HSD11B1 54 35 O=C(NC1C2CC3CC(C2)CC1C3)C1CCN(S(=O)(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147269228 JI On-Demand Anodyne EPHX2 54 54 O=C(NC1C2CC3CC(C2)CC1C3)C1CCN(S(=O)(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147269228 JI On-Demand Anodyne RBP4 72 33 O=C(NC1C2CC3CC(C2)CC1C3)C1CCN(S(=O)(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147269228 JI On-Demand Anodyne SFRP1 120 41 O=C(NC1C2CC3CC(C2)CC1C3)C1CCN(S(=O)(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147269228 JI On-Demand Anodyne WNT3 77 32 CCNc1nc(Cl)nc(Oc2ccccc2C(C)C)n1 ZINC000147269246 CH For-Sale Anodyne Q31945_CHEAL 0 44 CCNc1nc(Cl)nc(Oc2ccccc2C(C)C)n1 ZINC000147269246 CH For-Sale Anodyne PPX1 0 45 CN(C)C1(CNC(=O)c2cccc(C(=O)O)c2)CCCC1 ZINC000147269255 CD On-Demand Anodyne DRD4 41 31 CN(C)C1(CNC(=O)c2cccc(C(=O)O)c2)CCCC1 ZINC000147269255 CD On-Demand Anodyne SLC6A5 19 56 CN(C)C1(CNC(=O)c2cccc(C(=O)O)c2)CCCC1 ZINC000147269255 CD On-Demand Anodyne ACAT 0 43 CN(C)C1(CNC(=O)c2cccc(C(=O)O)c2)CCCC1 ZINC000147269255 CD On-Demand Anodyne HCN1 52 33 CN(C)C1(CNC(=O)c2cccc(C(=O)O)c2)CCCC1 ZINC000147269255 CD On-Demand Anodyne HCN4 49 33 CN(C)C1(CNC(=O)c2cccc(C(=O)O)c2)CCCC1 ZINC000147269255 CD On-Demand Anodyne KCNK3 61 34 COc1ccc(CC(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147269296 EG For-Sale Reactive OPRK1 0 43 COc1ccc(CC(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147269296 EG For-Sale Reactive GRM3 15 47 COc1ccc(CC(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147269296 EG For-Sale Reactive MMP13 31 44 COc1ccc(CC(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147269296 EG For-Sale Reactive MMP1 35 44 COc1ccc(CC(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147269296 EG For-Sale Reactive RORC 27 40 COc1ccc(CC(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147269296 EG For-Sale Reactive GPR183 0 43 CCCCCCCCn1cc(C)nc1SCC(=O)O ZINC000147269310 CH For-Sale Mild CSNK2A2 15 40 Nc1cc(Cl)cc(-c2nc(-c3ccc(F)cc3Cl)no2)c1 ZINC000147269333 DI For-Sale Anodyne DPP7 0 41 CC[C@@H]1CN(C(=O)c2ccc3ccccc3n2)CC[C@H]1N ZINC000147269365 CE On-Demand Anodyne SMO 46 36 Cn1c(-c2ccc(-c3ccccc3)cc2)ccc(O)c1=O ZINC000147269390 CG For-Sale Anodyne COMT 70 43 Cn1c(-c2ccc(-c3ccccc3)cc2)ccc(O)c1=O ZINC000147269390 CG For-Sale Anodyne HDAC8 15 40 Cn1c(-c2ccc(-c3ccccc3)cc2)ccc(O)c1=O ZINC000147269390 CG For-Sale Anodyne HDAC2 22 40 Cn1c(-c2ccc(-c3ccccc3)cc2)ccc(O)c1=O ZINC000147269390 CG For-Sale Anodyne GRM7 79 40 COC(=O)[C@H]1COc2ccc(Br)cc21 ZINC000147269396 CE In-Stock Anodyne HCRTR2 27 44 C[C@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccc(F)cc1 ZINC000147269400 CD For-Sale Anodyne ACACA 41 35 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269418 HI On-Demand Anodyne CA2 18 48 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269418 HI On-Demand Anodyne CA1 19 40 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269418 HI On-Demand Anodyne MMP13 33 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269418 HI On-Demand Anodyne CA4 18 48 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269418 HI On-Demand Anodyne MMP2 35 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269418 HI On-Demand Anodyne MMP9 15 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269418 HI On-Demand Anodyne CA12 15 42 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269418 HI On-Demand Anodyne CA9 17 42 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269418 HI On-Demand Anodyne IDO1 48 54 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269418 HI On-Demand Anodyne KDM1A 43 38 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@@H]3c3ccccc3)cc2)cc1 ZINC000147269418 HI On-Demand Anodyne NAMPT 35 40 C[C@H](CNS(=O)(=O)c1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147269437 EC On-Demand Anodyne PTGS2 15 40 C[C@H](CNS(=O)(=O)c1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147269437 EC On-Demand Anodyne TBXA2R 36 41 C[C@H](CNS(=O)(=O)c1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147269437 EC On-Demand Anodyne MMP10 15 40 C[C@H](CNS(=O)(=O)c1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147269437 EC On-Demand Anodyne O49150_SOLTU 41 34 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147269447 ED On-Demand Anodyne KCNK3 23 49 CCNCc1ccccc1Oc1ccc(Cl)c(F)c1 ZINC000147269459 CI For-Sale Anodyne SLC6A4 19 60 NNc1cc(-n2cnc3ccccc32)nc(C2CC2)n1 ZINC000147269509 CD For-Sale Anodyne LCK 17 45 O=C(c1cc2ccccc2s1)N1CCC[C@H](CCBr)C1 ZINC000147269523 FJ For-Sale Reactive AKR1C3 0 48 Nc1cc(Br)cc(-c2nc(-c3ccc(F)cc3Cl)no2)c1 ZINC000147269534 FJ For-Sale Anodyne DPP7 22 40 Cc1cc(C(=O)Nc2cccc(-n3cnnn3)c2)cc([N+](=O)[O-])c1 ZINC000147269555 DE On-Demand Bother KCNK3 80 36 Cc1cc(C(=O)Nc2cccc(-n3cnnn3)c2)cc([N+](=O)[O-])c1 ZINC000147269555 DE On-Demand Bother KCNK9 50 41 CC[C@H]1CN(C(=O)c2ccc3ccccc3n2)CC[C@H]1N ZINC000147269576 CE On-Demand Anodyne SMO 46 36 C[C@@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccc(F)cc1 ZINC000147269596 CD For-Sale Anodyne ACACA 41 35 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269614 HI On-Demand Anodyne CA2 18 48 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269614 HI On-Demand Anodyne CA1 19 40 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269614 HI On-Demand Anodyne MMP13 33 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269614 HI On-Demand Anodyne CA4 18 48 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269614 HI On-Demand Anodyne MMP2 35 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269614 HI On-Demand Anodyne MMP9 15 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269614 HI On-Demand Anodyne CA12 15 42 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269614 HI On-Demand Anodyne CA9 17 42 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269614 HI On-Demand Anodyne IDO1 48 54 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269614 HI On-Demand Anodyne KDM1A 43 38 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269614 HI On-Demand Anodyne NAMPT 35 40 C[C@@H](CNS(=O)(=O)c1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147269615 EC On-Demand Anodyne PTGS2 15 40 C[C@@H](CNS(=O)(=O)c1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147269615 EC On-Demand Anodyne TBXA2R 36 41 C[C@@H](CNS(=O)(=O)c1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147269615 EC On-Demand Anodyne MMP10 15 40 C[C@@H](CNS(=O)(=O)c1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147269615 EC On-Demand Anodyne O49150_SOLTU 41 34 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147269625 ED On-Demand Anodyne KCNK3 23 49 CC(C)c1nc(NN)cc(-n2cnc3ccccc32)n1 ZINC000147269708 CE For-Sale Anodyne PDGFRB 0 41 CC(C)c1nc(NN)cc(-n2cnc3ccccc32)n1 ZINC000147269708 CE For-Sale Anodyne LCK 19 46 O=C(c1cc2ccccc2s1)N1CCC[C@@H](CCBr)C1 ZINC000147269718 FJ For-Sale Reactive AKR1C3 0 48 CCCCCCCCNC(=O)C(=O)N1CCNCC1 ZINC000147269720 CC On-Demand Mild GNAI1 0 51 CCCCCCCCNC(=O)C(=O)N1CCNCC1 ZINC000147269720 CC On-Demand Mild GNAI3 0 51 CCCCCCCCNC(=O)C(=O)N1CCNCC1 ZINC000147269720 CC On-Demand Mild GNAO1 0 51 CCCCCCCCNC(=O)C(=O)N1CCNCC1 ZINC000147269720 CC On-Demand Mild ASAH1 86 38 Cc1nn(C(F)F)c(C)c1CC(=O)N[C@@H]1CCS(=O)(=O)c2ccccc21 ZINC000147269725 GE On-Demand Anodyne P2RX7 20 41 NC(=O)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147269786 DB For-Sale Anodyne CPT1A 43 30 CCCN(CC(=O)O)C(=O)C1[C@H]2CCCC[C@H]12 ZINC000147269798 BD On-Demand Anodyne ACE 24 47 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269804 HI On-Demand Anodyne CA2 18 48 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269804 HI On-Demand Anodyne CA1 19 40 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269804 HI On-Demand Anodyne MMP13 33 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269804 HI On-Demand Anodyne CA4 18 48 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269804 HI On-Demand Anodyne MMP2 35 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269804 HI On-Demand Anodyne MMP9 15 45 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269804 HI On-Demand Anodyne CA12 15 42 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269804 HI On-Demand Anodyne CA9 17 42 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269804 HI On-Demand Anodyne IDO1 48 54 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269804 HI On-Demand Anodyne KDM1A 43 38 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)N[C@H]3C[C@H]3c3ccccc3)cc2)cc1 ZINC000147269804 HI On-Demand Anodyne NAMPT 35 40 Oc1ccc(CNCC(F)F)cc1O ZINC000147269843 BD For-Sale Clean ALOX15 30 44 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne LTA4H 18 42 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne S1PR4 15 41 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne LPAR2 71 59 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne S1PR3 27 59 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne SLC2A1 28 46 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne PLA2G4B 57 35 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne S1PR2 77 59 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne S1PR1 17 59 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne SLC6A13 0 41 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne LEF 73 39 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne HT1 0 46 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne GPM3 0 50 CCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147269848 CJ For-Sale Anodyne LMGT2 0 46 CCOC(=O)[C@@H](C)NC(=O)c1cccc2c1OCCN2 ZINC000147269887 CD For-Sale Anodyne CCR3 0 48 Cc1nn(C(F)F)c(C)c1CC(=O)N[C@H]1CCS(=O)(=O)c2ccccc21 ZINC000147269908 GE On-Demand Anodyne P2RX7 20 41 CCCCCCCCNC(=O)C(=O)N1CCCNCC1 ZINC000147269926 CD On-Demand Mild GNAI1 0 47 CCCCCCCCNC(=O)C(=O)N1CCCNCC1 ZINC000147269926 CD On-Demand Mild GNAI3 0 47 CCCCCCCCNC(=O)C(=O)N1CCCNCC1 ZINC000147269926 CD On-Demand Mild GNAO1 0 47 CCCCCCCCNC(=O)C(=O)N1CCCNCC1 ZINC000147269926 CD On-Demand Mild ASAH1 74 35 CC(C)(C)c1nc(NN)cc(-n2cnc3ccccc32)n1 ZINC000147269964 CE For-Sale Anodyne PDGFRB 0 41 CC(C)(C)c1nc(NN)cc(-n2cnc3ccccc32)n1 ZINC000147269964 CE For-Sale Anodyne LCK 18 43 O=C1CCCN1c1ccc(S(=O)(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147269988 FF On-Demand Anodyne AKR1C3 26 48 COCc1nc(C(=O)Nc2nc(-c3ccc(C)cc3C)cs2)cs1 ZINC000147269991 FI On-Demand Anodyne MPL 52 39 CSc1ccc(NC(=O)CSc2nccn2-c2cccc(C)c2)cc1 ZINC000147270033 FJ On-Demand Anodyne ENPP1 57 34 CC(=O)Nc1ccc2c(c1)c(Cc1c[nH]cn1)cn2C ZINC000147270034 CE For-Sale Anodyne CYSLTR1 25 44 CC(=O)Nc1ccc2c(c1)c(Cc1c[nH]cn1)cn2C ZINC000147270034 CE For-Sale Anodyne HRH3 31 44 CCn1ccc(CNCCCCC(C)C)c1 ZINC000147270035 BG For-Sale Anodyne LEF 45 31 C=CCCOCC(=O)Nc1cccc(COc2cccc(F)c2)c1 ZINC000147270061 EH On-Demand Mild MAOB 15 40 CCOC(=O)[C@H](C)NC(=O)c1cccc2c1OCCN2 ZINC000147270109 CD For-Sale Anodyne CCR3 0 48 CCCCCCCCn1c(C)c(CC(=O)O)c(C)nc1=O ZINC000147270137 CF For-Sale Mild PLA2G4A 35 43 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne CA2 25 55 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne LPL 56 40 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne MAPK14 18 48 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne CA1 74 48 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne P2RY1 91 44 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne RAF1 39 49 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne KDR 35 44 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne EPHX2 53 41 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne ACR 48 36 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne CA12 43 55 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne PDGFRA 49 43 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne FLT3 42 41 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne TEK 28 41 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne CA9 40 55 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne NCE103 44 55 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne LIPG 20 40 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne MTCA1 40 38 CC(C)(C)Oc1ccc(NC(=O)Nc2ccccc2)cc1 ZINC000147270144 CJ On-Demand Anodyne P96878_MYCTU 51 48 COCCNCc1ccccc1Oc1ccc(Cl)c(F)c1 ZINC000147270146 DI For-Sale Anodyne SLC6A4 15 55 CC(C)c1ccccc1Oc1nc(N)ncc1Br ZINC000147270155 DH For-Sale Anodyne P2RX2 69 46 CC(C)c1ccccc1Oc1nc(N)ncc1Br ZINC000147270155 DH For-Sale Anodyne P2RX3 45 46 CN(C)NC(=O)[C@H](N)CC(=O)O ZINC000147270158 AA For-Sale Reactive SLC15A2 0 42 CN(C)NC(=O)[C@H](N)CC(=O)O ZINC000147270158 AA For-Sale Reactive KDM7A 0 42 CN(Cc1cscn1)C(=O)N[C@@H](Cc1ccccc1)c1ccccc1 ZINC000147270161 FI On-Demand Anodyne BMP1 58 39 CN(Cc1cscn1)C(=O)N[C@@H](Cc1ccccc1)c1ccccc1 ZINC000147270161 FI On-Demand Anodyne SOAT1 26 45 CN(Cc1cscn1)C(=O)N[C@@H](Cc1ccccc1)c1ccccc1 ZINC000147270161 FI On-Demand Anodyne CYP3A4 29 52 CN(Cc1cscn1)C(=O)N[C@@H](Cc1ccccc1)c1ccccc1 ZINC000147270161 FI On-Demand Anodyne GPR142 43 41 O=C1CCCN1c1ccc(S(=O)(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147270216 FF On-Demand Anodyne AKR1C3 26 48 C=C(C)COc1ccc(CCC(=O)O)cc1 ZINC000147270221 BF For-Sale Mild PLA2G4A 53 40 C=C(C)COc1ccc(CCC(=O)O)cc1 ZINC000147270221 BF For-Sale Mild PLA2G4B 82 40 C=C(C)COc1ccc(CCC(=O)O)cc1 ZINC000147270221 BF For-Sale Mild S1PR5 15 44 C=C(C)COc1ccc(CCC(=O)O)cc1 ZINC000147270221 BF For-Sale Mild TAAR1 16 43 C=C(C)COc1ccc(CCC(=O)O)cc1 ZINC000147270221 BF For-Sale Mild FFAR1 111 58 C=C(C)COc1ccc(CCC(=O)O)cc1 ZINC000147270221 BF For-Sale Mild PPO2 34 50 C=C(C)COc1ccc(CCC(=O)O)cc1 ZINC000147270221 BF For-Sale Mild FFAR4 70 49 CCCN(CC(=O)O)C(=O)C1[C@@H]2CCCC[C@@H]12 ZINC000147270267 BD On-Demand Anodyne ACE 24 47 O=C(N[C@H](CC(F)(F)F)c1ccccc1)c1ccc2c(c1)COC2 ZINC000147270334 EI On-Demand Anodyne UTS2 50 34 CN(C)NC(=O)[C@@H](N)CC(=O)O ZINC000147270359 AA For-Sale Reactive SLC15A2 0 42 CN(C)NC(=O)[C@@H](N)CC(=O)O ZINC000147270359 AA For-Sale Reactive KDM7A 0 42 CCCCCCCCn1c(C)cc(C(=O)CCl)c1C ZINC000147270361 CJ For-Sale Reactive THRB 45 31 CCNCc1cccc(Oc2ccc(Cl)c(F)c2)c1 ZINC000147270365 CI For-Sale Anodyne CRTM 56 38 CCNCc1cccc(Oc2ccc(Cl)c(F)c2)c1 ZINC000147270365 CI For-Sale Anodyne PDS 45 35 CN(Cc1cscn1)C(=O)N[C@H](Cc1ccccc1)c1ccccc1 ZINC000147270378 FI On-Demand Anodyne BMP1 58 39 CN(Cc1cscn1)C(=O)N[C@H](Cc1ccccc1)c1ccccc1 ZINC000147270378 FI On-Demand Anodyne SOAT1 26 45 CN(Cc1cscn1)C(=O)N[C@H](Cc1ccccc1)c1ccccc1 ZINC000147270378 FI On-Demand Anodyne CYP3A4 29 52 CN(Cc1cscn1)C(=O)N[C@H](Cc1ccccc1)c1ccccc1 ZINC000147270378 FI On-Demand Anodyne GPR142 43 41 O=C1CCCN1c1ccc(S(=O)(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147270445 FF On-Demand Anodyne AKR1C3 26 48 CCN(CC(=O)O)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147270490 BD For-Sale Anodyne GPR88 0 46 O=C(N[C@@H](CC(F)(F)F)c1ccccc1)c1ccc2c(c1)COC2 ZINC000147270521 EI On-Demand Anodyne UTS2 50 34 CN(C)NC(=O)CC1CNC1 ZINC000147270536 AB For-Sale Reactive KDM7A 0 41 CCNc1ncc(F)c(Oc2ccccc2C(C)C)n1 ZINC000147270595 CH For-Sale Anodyne P2RX2 44 31 COc1ccc(-c2cccnc2)c([N+](=O)[O-])c1 ZINC000147270663 BF For-Sale Bother CYP19A1 15 52 COc1ccc(-c2cccnc2)c([N+](=O)[O-])c1 ZINC000147270663 BF For-Sale Bother CYP11B1 47 49 COc1ccc(-c2cccnc2)c([N+](=O)[O-])c1 ZINC000147270663 BF For-Sale Bother PTAFR 15 40 COc1ccc(-c2cccnc2)c([N+](=O)[O-])c1 ZINC000147270663 BF For-Sale Bother DAPK3 22 40 COc1ccc(-c2cccnc2)c([N+](=O)[O-])c1 ZINC000147270663 BF For-Sale Bother CYP11B2 70 55 COc1ccc(-c2cccnc2)c([N+](=O)[O-])c1 ZINC000147270663 BF For-Sale Bother CYP17A1 16 55 COc1ccc(-c2cccnc2)c([N+](=O)[O-])c1 ZINC000147270663 BF For-Sale Bother TPPP 0 51 CCN(CC(=O)O)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147270702 BD For-Sale Anodyne GPR88 0 46 C=C(Cn1cncn1)c1ccc(Cl)cc1 ZINC000147270727 BF For-Sale Mild HIS3 44 37 O=C(O)C1(NCc2ccc3ccccc3n2)CCC1 ZINC000147270731 CE For-Sale Anodyne CYSLTR1 42 39 O=C(O)C1(NCc2ccc3ccccc3n2)CCC1 ZINC000147270731 CE For-Sale Anodyne ALOX5AP 35 42 Nc1ccc(C(=O)N2CCOCC2)cc1O ZINC000147270767 BC For-Sale Anodyne AKR1C3 32 50 Nc1ccc(C(=O)N2CCOCC2)cc1O ZINC000147270767 BC For-Sale Anodyne L3MBTL1 0 44 Nc1ccc(C(=O)N2CCOCC2)cc1O ZINC000147270767 BC For-Sale Anodyne L3MBTL3 56 41 Cc1cccc(N(CCO)Cc2ccccc2)c1 ZINC000147270862 BF On-Demand Anodyne CETP 0 46 CCN(CC(=O)O)C(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147270893 BD For-Sale Anodyne GPR88 0 46 CCCCCCCCNC(=O)NC(=O)[C@@H](C)Cl ZINC000147270914 CF For-Sale Reactive CPT1A 22 43 CCCCCCCCNC(=O)NC(=O)[C@@H](C)Cl ZINC000147270914 CF For-Sale Reactive EPHX2 60 43 CCCCCCCCNC(=O)NC(=O)[C@@H](C)Cl ZINC000147270914 CF For-Sale Reactive ASAH1 94 38 CCCCCCCCNC(=O)NC(=O)[C@@H](C)Cl ZINC000147270914 CF For-Sale Reactive CQSS 54 35 COc1ccc(N2CCOCC2)c2sc(NC(=O)CCc3ccccc3)nc12 ZINC000147270928 GH For-Sale Clean DRD2 15 44 COc1ccc(N2CCOCC2)c2sc(NC(=O)CCc3ccccc3)nc12 ZINC000147270928 GH For-Sale Clean ADRA1D 19 40 COc1ccc(N2CCOCC2)c2sc(NC(=O)CCc3ccccc3)nc12 ZINC000147270928 GH For-Sale Clean ADRA1A 15 40 COc1ccc(N2CCOCC2)c2sc(NC(=O)CCc3ccccc3)nc12 ZINC000147270928 GH For-Sale Clean ADRA1B 18 40 COc1ccc(N2CCOCC2)c2sc(NC(=O)CCc3ccccc3)nc12 ZINC000147270928 GH For-Sale Clean ADORA2B 17 44 COc1ccc(N2CCOCC2)c2sc(NC(=O)CCc3ccccc3)nc12 ZINC000147270928 GH For-Sale Clean CASR 28 47 COc1ccc(N2CCOCC2)c2sc(NC(=O)CCc3ccccc3)nc12 ZINC000147270928 GH For-Sale Clean PRKDC 49 35 C[C@@H](CCN(C)C)NC(=O)c1cccc2c1OCCN2 ZINC000147270956 CD For-Sale Anodyne UTS2 65 35 C[C@@H]1C[C@H]1C(=O)Nc1ccc(F)cc1C(=O)Nc1ccc2nccnc2c1 ZINC000147270969 FH On-Demand Anodyne TYK2 36 42 COc1cc(CCC(=O)O)c(Br)cc1O ZINC000147271009 CE For-Sale Anodyne TRPV1 20 52 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccnc1 ZINC000147271045 CE On-Demand Anodyne BMP1 46 33 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccnc1 ZINC000147271045 CE On-Demand Anodyne KCNA5 44 42 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccnc1 ZINC000147271045 CE On-Demand Anodyne CYP3A4 21 47 O=C1CC[C@@H](C(=O)Nc2cccc(CO)c2)CN1 ZINC000147271103 BC On-Demand Anodyne INHA 20 44 O=C1CC[C@@H](C(=O)Nc2cccc(CO)c2)CN1 ZINC000147271103 BC On-Demand Anodyne PARP10 0 47 CCN(CC(=O)O)C(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147271108 BD For-Sale Anodyne GPR88 0 46 CCCCCCCCNC(=O)NC(=O)[C@H](C)Cl ZINC000147271129 CF For-Sale Reactive CPT1A 22 43 CCCCCCCCNC(=O)NC(=O)[C@H](C)Cl ZINC000147271129 CF For-Sale Reactive EPHX2 60 43 CCCCCCCCNC(=O)NC(=O)[C@H](C)Cl ZINC000147271129 CF For-Sale Reactive ASAH1 94 38 CCCCCCCCNC(=O)NC(=O)[C@H](C)Cl ZINC000147271129 CF For-Sale Reactive CQSS 54 35 C[C@H](CCN(C)C)NC(=O)c1cccc2c1OCCN2 ZINC000147271177 CD For-Sale Anodyne UTS2 65 35 Cc1ccc(CNCC(F)F)cc1F ZINC000147271212 BE On-Demand Anodyne LEF 60 36 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C1CCCCC1 ZINC000147271250 FH On-Demand Anodyne HDAC10 41 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C1CCCCC1 ZINC000147271250 FH On-Demand Anodyne HDAC11 41 33 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccnc1 ZINC000147271256 CE On-Demand Anodyne BMP1 46 33 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccnc1 ZINC000147271256 CE On-Demand Anodyne KCNA5 44 42 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccnc1 ZINC000147271256 CE On-Demand Anodyne CYP3A4 21 47 O=C1CC[C@H](C(=O)Nc2cccc(CO)c2)CN1 ZINC000147271323 BC On-Demand Anodyne INHA 20 44 O=C1CC[C@H](C(=O)Nc2cccc(CO)c2)CN1 ZINC000147271323 BC On-Demand Anodyne PARP10 0 47 N#CCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147271327 DC For-Sale Mild CPT1A 43 30 N#CCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147271327 DC For-Sale Mild PTGDR2 48 38 CCN(CC(=O)O)C(=O)c1ccc(C)c(Br)c1 ZINC000147271329 DE On-Demand Anodyne OPRM1 0 40 CCCCCCCCNC(=O)NC(=O)CCCl ZINC000147271361 CF For-Sale Reactive CPT1A 0 40 CCCCCCCCNC(=O)NC(=O)CCCl ZINC000147271361 CF For-Sale Reactive FAAH 0 57 CCCCCCCCNC(=O)NC(=O)CCCl ZINC000147271361 CF For-Sale Reactive EPHX2 61 46 CCCCCCCCNC(=O)NC(=O)CCCl ZINC000147271361 CF For-Sale Reactive ASAH1 81 35 CCCCCCCCNC(=O)NC(=O)CCCl ZINC000147271361 CF For-Sale Reactive CQSS 51 32 O=C(NCCN1CCCCC1)c1cccc2c1OCCN2 ZINC000147271369 CD For-Sale Anodyne HTR1A 16 43 O=C(NCCN1CCCCC1)c1cccc2c1OCCN2 ZINC000147271369 CD For-Sale Anodyne DRD2 15 44 O=C(NCCN1CCCCC1)c1cccc2c1OCCN2 ZINC000147271369 CD For-Sale Anodyne DRD4 43 33 O=C(NCCN1CCCCC1)c1cccc2c1OCCN2 ZINC000147271369 CD For-Sale Anodyne HTR4 19 50 O=C(NCCN1CCCCC1)c1cccc2c1OCCN2 ZINC000147271369 CD For-Sale Anodyne CHRNA7 20 40 O=C(NCCN1CCCCC1)c1cccc2c1OCCN2 ZINC000147271369 CD For-Sale Anodyne PLD2 70 35 O=C(NCCN1CCCCC1)c1cccc2c1OCCN2 ZINC000147271369 CD For-Sale Anodyne POLR1A 15 43 C[C@@H](CCc1ccc(O)cc1)NCC(F)F ZINC000147271413 BF On-Demand Anodyne ADRB3 15 54 Cc1ccccc1[C@@H](C)NC(=O)CNC1(C(=O)O)CCC1 ZINC000147271438 CD For-Sale Anodyne CTSA 49 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C1CCCCC1 ZINC000147271444 FH On-Demand Anodyne HDAC10 41 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C1CCCCC1 ZINC000147271444 FH On-Demand Anodyne HDAC11 41 33 CCCNc1ncc(C)c(Oc2ccccc2C(C)C)n1 ZINC000147271474 CJ For-Sale Anodyne P2RX2 47 35 CC(C)NC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147271520 DD For-Sale Anodyne PTGDR2 17 40 C[C@H](CCc1ccc(O)cc1)NCC(F)F ZINC000147271579 BF On-Demand Anodyne ADRB3 15 54 C[C@H](CNS(=O)(=O)c1cc([N+](=O)[O-])ccc1F)CC(=O)O ZINC000147271583 DD For-Sale Bother COLA 56 39 C[C@H](CNS(=O)(=O)c1cc([N+](=O)[O-])ccc1F)CC(=O)O ZINC000147271583 DD For-Sale Bother MMP2 15 41 CCCCCCCCNc1cc(Cl)nc(C)n1 ZINC000147271586 CI In-Stock Mild ASAH1 46 34 COC[C@H](C)NS(=O)(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147271643 HE On-Demand Bother MMP13 25 41 COC[C@H](C)NS(=O)(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147271643 HE On-Demand Bother MMP2 22 52 Cc1ccccc1[C@H](C)NC(=O)CNC1(C(=O)O)CCC1 ZINC000147271653 CD For-Sale Anodyne CTSA 49 33 Cc1cnc(N)nc1Oc1ccccc1C(C)C ZINC000147271686 BG For-Sale Anodyne P2RX2 58 44 Cc1cnc(N)nc1Oc1ccccc1C(C)C ZINC000147271686 BG For-Sale Anodyne P2RX3 34 44 Oc1ccc(O)c2occc12 ZINC000147271708 AD For-Sale Anodyne KCNA2 42 32 CC(C)NC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147271745 DD For-Sale Anodyne PTGDR2 17 40 CCN(CC(=O)O)C(=O)C1[C@H]2CCCC[C@H]12 ZINC000147271773 BD On-Demand Anodyne ACE 28 45 Cc1ccc(CNCC(F)F)cc1C ZINC000147271775 AF On-Demand Anodyne LEF 46 35 Cc1cnc(NC(=O)C[C@@H]2CNc3ccccc32)s1 ZINC000147271778 CF For-Sale Anodyne CDK5 50 41 C[C@@H](CNS(=O)(=O)c1cc([N+](=O)[O-])ccc1F)CC(=O)O ZINC000147271792 DD For-Sale Bother COLA 56 39 C[C@@H](CNS(=O)(=O)c1cc([N+](=O)[O-])ccc1F)CC(=O)O ZINC000147271792 DD For-Sale Bother MMP2 15 41 CC(C)NCc1cc(F)ccc1Oc1ccc(Cl)c(F)c1 ZINC000147271835 DJ For-Sale Anodyne SLC6A4 22 62 COC[C@@H](C)NS(=O)(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147271855 HE On-Demand Bother MMP13 25 41 COC[C@@H](C)NS(=O)(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147271855 HE On-Demand Bother MMP2 22 52 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccc(OC(F)(F)F)cc3)c(F)c2)CC1 ZINC000147271883 KI Annotated Clean AVPR1B 18 41 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccc(OC(F)(F)F)cc3)c(F)c2)CC1 ZINC000147271883 KI Annotated Clean RORC 16 44 O=C(O)C1(NCCCc2ccccc2)CCC1 ZINC000147271893 BE For-Sale Anodyne SDH1 0 44 O=C(O)C1(NCCCc2ccccc2)CCC1 ZINC000147271893 BE For-Sale Anodyne SIGMAR1 21 46 O=C(O)C1(NCCCc2ccccc2)CCC1 ZINC000147271893 BE For-Sale Anodyne CES1 44 40 O=C(O)C1(NCCCc2ccccc2)CCC1 ZINC000147271893 BE For-Sale Anodyne AMP1_PLAFQ 23 40 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCOCC1 ZINC000147271973 DC For-Sale Anodyne HTR2A 20 46 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCOCC1 ZINC000147271973 DC For-Sale Anodyne THRB 0 43 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCOCC1 ZINC000147271973 DC For-Sale Anodyne FLT3 17 44 CC(C)(C)OC(=O)N1CCc2ccc(Cl)c(N)c2CC1 ZINC000147271975 CG For-Sale Anodyne GPR119 34 42 Cc1cnc(NC(=O)C[C@H]2CNc3ccccc32)s1 ZINC000147271999 CF For-Sale Anodyne CDK5 50 41 CCCC[C@H](NC(N)=O)C(=O)N(CC)CC(=O)NCc1ccc(F)cc1 ZINC000147272110 FD On-Demand Anodyne FURIN 45 34 CC(C)c1ccccc1Oc1nc(N)ncc1F ZINC000147272154 BG For-Sale Anodyne P2RX2 56 43 CC(C)c1ccccc1Oc1nc(N)ncc1F ZINC000147272154 BG For-Sale Anodyne P2RX3 33 40 NS(=O)(=O)c1cc(Cl)ccc1OCCCN1CCCC1 ZINC000147272171 DD For-Sale Anodyne DRD5 18 40 NS(=O)(=O)c1cc(Cl)ccc1OCCCN1CCCC1 ZINC000147272171 DD For-Sale Anodyne LTA4H 20 41 NS(=O)(=O)c1cc(Cl)ccc1OCCCN1CCCC1 ZINC000147272171 DD For-Sale Anodyne HRP1_PLAFA 73 34 NS(=O)(=O)c1cc(Cl)ccc1OCCCN1CCCC1 ZINC000147272171 DD For-Sale Anodyne HRH3 70 53 NS(=O)(=O)c1cc(Cl)ccc1OCCCN1CCCC1 ZINC000147272171 DD For-Sale Anodyne SIGMAR1 22 46 NS(=O)(=O)c1cc(Cl)ccc1OCCCN1CCCC1 ZINC000147272171 DD For-Sale Anodyne HNMT 67 42 CCN(CC(=O)O)C(=O)C1[C@@H]2CCCC[C@@H]12 ZINC000147272203 BD On-Demand Anodyne ACE 28 45 CN(C)C1(CNC(=O)c2cccn2CC(=O)O)CCCC1 ZINC000147272233 CD For-Sale Anodyne SLC6A5 15 44 CC(C)CCCCNCc1ccc(-c2ccccc2)s1 ZINC000147272277 CK For-Sale Anodyne CYP2E1 21 44 CNCc1ccc(Oc2ccc(Cl)c(F)c2)c(C)c1 ZINC000147272334 CI For-Sale Anodyne SLC6A4 20 54 CCCC[C@@H](NC(N)=O)C(=O)N(CC)CC(=O)NCc1ccc(F)cc1 ZINC000147272344 FD On-Demand Anodyne FURIN 45 34 Cc1cc([N+](=O)[O-])ccc1NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147272352 CD For-Sale Bother SLC27A4 42 31 CCCNCc1ccc(Oc2ccc(Cl)c(F)c2)c(C)c1 ZINC000147272509 DK For-Sale Anodyne LEF 56 40 CC[C@@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@@H]1N ZINC000147272523 CD On-Demand Anodyne L3MBTL1 0 41 CC[C@@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@@H]1N ZINC000147272523 CD On-Demand Anodyne L3MBTL3 71 41 CC[C@@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@@H]1N ZINC000147272523 CD On-Demand Anodyne GPR183 0 40 Cc1cc([N+](=O)[O-])ccc1NC(=O)[C@H]1CCC(=O)NC1 ZINC000147272534 CD For-Sale Bother SLC27A4 42 31 Cc1cccc(OCCNC2(C(=O)O)CCC2)c1 ZINC000147272685 BD For-Sale Anodyne DRD4 19 54 COc1ccc(S(=O)(=O)N(CCBr)C2CCCC2)cc1 ZINC000147272693 FG For-Sale Reactive AVPR1B 30 49 COc1ccc(S(=O)(=O)N(CCBr)C2CCCC2)cc1 ZINC000147272693 FG For-Sale Reactive CASR 0 40 COc1ccc(S(=O)(=O)N(CCBr)C2CCCC2)cc1 ZINC000147272693 FG For-Sale Reactive BMP1 71 46 COc1ccc(S(=O)(=O)N(CCBr)C2CCCC2)cc1 ZINC000147272693 FG For-Sale Reactive MMP13 46 45 COc1ccc(S(=O)(=O)N(CCBr)C2CCCC2)cc1 ZINC000147272693 FG For-Sale Reactive ADAM17 15 40 COc1ccc(S(=O)(=O)N(CCBr)C2CCCC2)cc1 ZINC000147272693 FG For-Sale Reactive MMP16 0 40 COc1ccc(S(=O)(=O)N(CCBr)C2CCCC2)cc1 ZINC000147272693 FG For-Sale Reactive MMP3 41 46 COc1ccc(S(=O)(=O)N(CCBr)C2CCCC2)cc1 ZINC000147272693 FG For-Sale Reactive MMP9 41 45 COc1ccc(S(=O)(=O)N(CCBr)C2CCCC2)cc1 ZINC000147272693 FG For-Sale Reactive MMP12 27 40 COc1ccc(S(=O)(=O)N(CCBr)C2CCCC2)cc1 ZINC000147272693 FG For-Sale Reactive MMP1 41 45 CC[C@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@@H]1N ZINC000147272709 CD On-Demand Anodyne L3MBTL1 0 41 CC[C@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@@H]1N ZINC000147272709 CD On-Demand Anodyne L3MBTL3 71 41 CC[C@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@@H]1N ZINC000147272709 CD On-Demand Anodyne GPR183 0 40 CCCCCCCNCC(F)F ZINC000147272719 AF For-Sale Mild S1PR2 33 41 CCCCCCCNCC(F)F ZINC000147272719 AF For-Sale Mild Q8WS26_TRYCR 45 52 CSc1ccc(-c2nc3cc(C(F)(F)F)ccc3[nH]2)cc1 ZINC000147272766 DJ For-Sale Anodyne CHEK2 58 48 CSc1ccc(-c2nc3cc(C(F)(F)F)ccc3[nH]2)cc1 ZINC000147272766 DJ For-Sale Anodyne NR2E3 54 35 CSc1ccc(-c2nc3cc(C(F)(F)F)ccc3[nH]2)cc1 ZINC000147272766 DJ For-Sale Anodyne SCD1 24 49 CSc1ccc(-c2nc3cc(C(F)(F)F)ccc3[nH]2)cc1 ZINC000147272766 DJ For-Sale Anodyne SCD 0 43 CSc1ccc(-c2nc3cc(C(F)(F)F)ccc3[nH]2)cc1 ZINC000147272766 DJ For-Sale Anodyne DGAT1 15 42 CCCC[C@H](NC(N)=O)C(=O)N(CCOC)Cc1ccccc1 ZINC000147272800 DD On-Demand Anodyne P2RY12 91 35 CCCC[C@H](NC(N)=O)C(=O)N(CCOC)Cc1ccccc1 ZINC000147272800 DD On-Demand Anodyne KLK3 42 35 CCCC[C@H](NC(N)=O)C(=O)N(CCOC)Cc1ccccc1 ZINC000147272800 DD On-Demand Anodyne CCKAR 15 42 CCCC[C@H](NC(N)=O)C(=O)N(CCOC)Cc1ccccc1 ZINC000147272800 DD On-Demand Anodyne CTSK 32 40 CCCC[C@H](NC(N)=O)C(=O)N(CCOC)Cc1ccccc1 ZINC000147272800 DD On-Demand Anodyne MMP3 20 40 CCCC[C@H](NC(N)=O)C(=O)N(CCOC)Cc1ccccc1 ZINC000147272800 DD On-Demand Anodyne CAPN1 23 40 CCCC[C@H](NC(N)=O)C(=O)N(CCOC)Cc1ccccc1 ZINC000147272800 DD On-Demand Anodyne CTRB_BOVIN 47 34 CCCC[C@H](NC(N)=O)C(=O)N(CCOC)Cc1ccccc1 ZINC000147272800 DD On-Demand Anodyne NPR 47 36 CCCC[C@H](NC(N)=O)C(=O)N(CCOC)Cc1ccccc1 ZINC000147272800 DD On-Demand Anodyne POLG_WNV 49 30 CCCC[C@H](NC(N)=O)C(=O)N(CCOC)Cc1ccccc1 ZINC000147272800 DD On-Demand Anodyne NOD1 40 30 CC(C)N(CCC(=O)O)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147272824 CF For-Sale Anodyne GPR88 0 49 CN(C)NC(=O)/C=C/c1cccc(N)c1 ZINC000147272861 BC For-Sale Reactive HDAC8 53 39 CN(C)NC(=O)/C=C/c1cccc(N)c1 ZINC000147272861 BC For-Sale Reactive MMP2 20 42 CN(C)NC(=O)/C=C/c1cccc(N)c1 ZINC000147272861 BC For-Sale Reactive HDAC6 33 41 CN(C)NC(=O)/C=C/c1cccc(N)c1 ZINC000147272861 BC For-Sale Reactive MMP9 18 42 CN(C)NC(=O)/C=C/c1cccc(N)c1 ZINC000147272861 BC For-Sale Reactive MMP1 22 42 CC[C@@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@H]1N ZINC000147272949 CD On-Demand Anodyne L3MBTL1 0 41 CC[C@@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@H]1N ZINC000147272949 CD On-Demand Anodyne L3MBTL3 71 41 CC[C@@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@H]1N ZINC000147272949 CD On-Demand Anodyne GPR183 0 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000147272981 EG On-Demand Clean DRD4 43 33 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000147272981 EG On-Demand Clean TAAR1 50 63 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000147272981 EG On-Demand Clean AKR1C3 26 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000147272981 EG On-Demand Clean AKR1C2 56 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000147272981 EG On-Demand Clean KCNK3 49 39 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(N3CCCC3)c2)c1 ZINC000147272981 EG On-Demand Clean KCNK9 50 39 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147272992 FG On-Demand Anodyne KIT 20 40 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147272992 FG On-Demand Anodyne GRM4 54 38 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147272992 FG On-Demand Anodyne BRAF 26 40 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147272992 FG On-Demand Anodyne NR2E3 64 35 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147272992 FG On-Demand Anodyne KCNK3 68 37 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147272992 FG On-Demand Anodyne KCNK9 60 37 CCc1ncc(C(=O)Nc2ccc(S(=O)(=O)N(C)C(C)C)cc2)s1 ZINC000147273005 FF On-Demand Anodyne USP47 42 33 CC(C)N(CCC(=O)O)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147273106 CF For-Sale Anodyne GPR88 0 49 CC[C@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@H]1N ZINC000147273161 CD On-Demand Anodyne L3MBTL1 0 41 CC[C@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@H]1N ZINC000147273161 CD On-Demand Anodyne L3MBTL3 71 41 CC[C@H]1CN(C(=O)c2ccc(N(C)C)cc2)CC[C@H]1N ZINC000147273161 CD On-Demand Anodyne GPR183 0 40 CC(C)CNCc1ccccc1Oc1ccc(Cl)c(F)c1 ZINC000147273162 DK For-Sale Anodyne SLC6A4 17 59 CC(C)CNCc1ccccc1Oc1ccc(Cl)c(F)c1 ZINC000147273162 DK For-Sale Anodyne PHES 0 42 CN(C)CCOc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147273183 EF On-Demand Anodyne NR2E3 61 35 CN(C)CCOc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147273183 EF On-Demand Anodyne KCNK3 63 46 CN(C)CCOc1ccccc1C(=O)Nc1ccc2nccnc2c1 ZINC000147273183 EF On-Demand Anodyne KCNK9 73 46 CCCN(Cc1ccc(N2CCN(C(C)=O)CC2)cc1)S(=O)(=O)Cc1ccccc1 ZINC000147273185 IG Annotated Clean RORC 38 60 COCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273210 DC For-Sale Anodyne CA2 35 43 COCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273210 DC For-Sale Anodyne CA1 29 43 COCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273210 DC For-Sale Anodyne COLA 64 36 COCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273210 DC For-Sale Anodyne CPT1A 60 36 COCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273210 DC For-Sale Anodyne CPT2 42 32 COCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273210 DC For-Sale Anodyne CA12 15 43 COCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273210 DC For-Sale Anodyne CPT1B 57 35 COCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273210 DC For-Sale Anodyne ALPL 35 44 COCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273210 DC For-Sale Anodyne PTGDR2 47 45 COCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273210 DC For-Sale Anodyne CAN2 0 46 CCCC[C@H](NC(N)=O)C(=O)N(CC)CC(=O)Nc1cccc(OC)c1 ZINC000147273232 FD On-Demand Anodyne MTNR1A 21 45 CCCC[C@H](NC(N)=O)C(=O)N(CC)CC(=O)Nc1cccc(OC)c1 ZINC000147273232 FD On-Demand Anodyne MTNR1B 28 45 CC(C)N(CCC(=O)O)C(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147273294 CF For-Sale Anodyne GPR88 0 49 CCCCCCCCNc1nnc(Cl)c2ccccc12 ZINC000147273308 CK For-Sale Mild UTS2R 18 48 CCCCCCCCNc1nnc(Cl)c2ccccc12 ZINC000147273308 CK For-Sale Mild SLC2A1 15 42 CCCCCCCCNc1nnc(Cl)c2ccccc12 ZINC000147273308 CK For-Sale Mild HT1 15 42 CCCCCCCCNc1nnc(Cl)c2ccccc12 ZINC000147273308 CK For-Sale Mild LMGT2 15 42 CNCc1cccc(Oc2ccc(Cl)c(F)c2)c1 ZINC000147273375 CH For-Sale Anodyne CRTM 49 37 CC[C@@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273409 DD For-Sale Anodyne CA2 32 44 CC[C@@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273409 DD For-Sale Anodyne CA1 23 44 CC[C@@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273409 DD For-Sale Anodyne CA4 25 44 CC[C@@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273409 DD For-Sale Anodyne PTGDR2 40 39 CCCC[C@@H](NC(N)=O)C(=O)N(CC)CC(=O)Nc1cccc(OC)c1 ZINC000147273428 FD On-Demand Anodyne MTNR1A 21 45 CCCC[C@@H](NC(N)=O)C(=O)N(CC)CC(=O)Nc1cccc(OC)c1 ZINC000147273428 FD On-Demand Anodyne MTNR1B 28 45 CN(C)NC(=O)c1cccc(F)c1N ZINC000147273480 AC For-Sale Reactive ECR 28 41 CN(C)NC(=O)c1cccc(F)c1N ZINC000147273480 AC For-Sale Reactive E3UJZ5_SPOLI 23 41 CCNc1ncc(Br)c(Oc2ccccc2C(C)C)n1 ZINC000147273504 EJ For-Sale Anodyne P2RX2 65 34 CCNc1ncc(Br)c(Oc2ccccc2C(C)C)n1 ZINC000147273504 EJ For-Sale Anodyne P2RX3 44 34 CC(C)N(CCC(=O)O)C(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147273505 CF For-Sale Anodyne GPR88 0 49 COCCN(Cc1ccc(N2CCN(C(C)=O)CC2)cc1)S(=O)(=O)Cc1ccccc1 ZINC000147273611 IE Annotated Clean RORC 31 57 CC[C@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273626 DD For-Sale Anodyne CA2 32 44 CC[C@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273626 DD For-Sale Anodyne CA1 23 44 CC[C@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273626 DD For-Sale Anodyne CA4 25 44 CC[C@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273626 DD For-Sale Anodyne PTGDR2 40 39 CN(C)C(=O)NCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147273630 CC On-Demand Anodyne E3UJZ5_SPOLI 45 36 NC(=O)c1ccc(OCC(=O)Nc2ccc3nccnc3c2)cc1 ZINC000147273646 DD On-Demand Anodyne ADORA2B 41 43 NC(=O)c1ccc(OCC(=O)Nc2ccc3nccnc3c2)cc1 ZINC000147273646 DD On-Demand Anodyne CETP 27 40 NC(=O)c1ccc(OCC(=O)Nc2ccc3nccnc3c2)cc1 ZINC000147273646 DD On-Demand Anodyne ACR 50 32 NC(=O)c1ccc(OCC(=O)Nc2ccc3nccnc3c2)cc1 ZINC000147273646 DD On-Demand Anodyne MCHR1 16 43 NC(=O)c1ccc(OCC(=O)Nc2ccc3nccnc3c2)cc1 ZINC000147273646 DD On-Demand Anodyne MCHR2 38 40 NC(=O)c1ccc(OCC(=O)Nc2ccc3nccnc3c2)cc1 ZINC000147273646 DD On-Demand Anodyne HIF1A 28 45 NC(=O)c1ccc(OCC(=O)Nc2ccc3nccnc3c2)cc1 ZINC000147273646 DD On-Demand Anodyne ENPP1 40 32 C=CCNCC(=O)NN(C)C ZINC000147273699 AB For-Sale Reactive KDM7A 0 41 COc1ccccc1N1CCC(NCc2csc(-c3ccco3)n2)CC1 ZINC000147273703 FI On-Demand Anodyne HTR1A 71 41 COc1ccccc1N1CCC(NCc2csc(-c3ccco3)n2)CC1 ZINC000147273703 FI On-Demand Anodyne DRD2 50 48 COc1ccccc1N1CCC(NCc2csc(-c3ccco3)n2)CC1 ZINC000147273703 FI On-Demand Anodyne DRD4 31 48 COc1ccccc1N1CCC(NCc2csc(-c3ccco3)n2)CC1 ZINC000147273703 FI On-Demand Anodyne ADRA1D 51 37 COc1ccccc1N1CCC(NCc2csc(-c3ccco3)n2)CC1 ZINC000147273703 FI On-Demand Anodyne ADRA1A 46 37 COc1ccccc1N1CCC(NCc2csc(-c3ccco3)n2)CC1 ZINC000147273703 FI On-Demand Anodyne ADRA1B 40 37 COc1ccccc1N1CCC(NCc2csc(-c3ccco3)n2)CC1 ZINC000147273703 FI On-Demand Anodyne DRD3 53 48 COc1ccccc1N1CCC(NCc2csc(-c3ccco3)n2)CC1 ZINC000147273703 FI On-Demand Anodyne HTR7 46 36 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(Sc3nc(C)cs3)cc2)c1 ZINC000147273713 HJ On-Demand Bother GSTM2 52 36 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(Sc3nc(C)cs3)cc2)c1 ZINC000147273713 HJ On-Demand Bother USP7 31 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(Sc3nc(C)cs3)cc2)c1 ZINC000147273713 HJ On-Demand Bother USP47 38 46 CCCCCCCCNc1nc(Cl)nc(N(CC)CC)n1 ZINC000147273729 DI For-Sale Mild AT1 0 43 CCCCCCCCNc1nc(Cl)nc(N(CC)CC)n1 ZINC000147273729 DI For-Sale Mild PPX1 0 41 NC(=O)c1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1Cl ZINC000147273754 ED On-Demand Anodyne ENV 44 35 COc1ccc(CNc2cccc3cc[nH]c23)cc1 ZINC000147273771 CH On-Demand Anodyne PTGDR 17 42 CC(=O)N1CCN(c2ccc(CN(C(C)C)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147273825 IG Annotated Clean SSTR3 42 33 CC(=O)N1CCN(c2ccc(CN(C(C)C)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147273825 IG Annotated Clean RORC 38 61 COCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273835 EC For-Sale Anodyne CA2 29 42 COCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273835 EC For-Sale Anodyne CA1 23 41 COCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273835 EC For-Sale Anodyne COLA 49 33 COCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273835 EC For-Sale Anodyne CPT1A 47 33 COCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273835 EC For-Sale Anodyne CA4 22 42 COCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273835 EC For-Sale Anodyne CA12 15 41 COCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273835 EC For-Sale Anodyne CPT1B 47 32 COCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273835 EC For-Sale Anodyne CA9 15 41 COCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147273835 EC For-Sale Anodyne PTGDR2 43 41 CCN(CC)S(=O)(=O)c1ccc2c(c1)CCN2C(=O)[C@H](C)Cc1cccc(F)c1 ZINC000147273891 HH On-Demand Anodyne TRY2_BOVIN 51 34 O=C(NC1CCN(C(=O)Nc2ccc(N3CCOCC3)nc2)CC1)c1ccoc1 ZINC000147273917 GD On-Demand Anodyne MTOR 41 38 O=C(NC1CCN(C(=O)Nc2ccc(N3CCOCC3)nc2)CC1)c1ccoc1 ZINC000147273917 GD On-Demand Anodyne DGAT1 47 44 O=C(NC1CCN(C(=O)Nc2ccc(N3CCOCC3)nc2)CC1)c1ccoc1 ZINC000147273917 GD On-Demand Anodyne HPGDS 35 55 NC(=O)c1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1Cl ZINC000147273990 ED On-Demand Anodyne ENV 44 35 O=C(O)C[C@H](NC(=O)C1CCC(F)(F)CC1)c1ccccc1 ZINC000147274084 DG On-Demand Anodyne CCR5 22 53 O=C(O)C[C@H](NC(=O)C1CCC(F)(F)CC1)c1ccccc1 ZINC000147274084 DG On-Demand Anodyne F11 48 42 O=C(O)C[C@H](NC(=O)C1CCC(F)(F)CC1)c1ccccc1 ZINC000147274084 DG On-Demand Anodyne CTSA 43 39 O=C(/C=C\c1cccnc1)N[C@H]1c2ccccc2C[C@H]1O ZINC000147274123 CD On-Demand Anodyne POL 0 42 O=C(/C=C\c1cccnc1)N[C@H]1c2ccccc2C[C@H]1O ZINC000147274123 CD On-Demand Anodyne PLM1_PLAFA 43 44 O=C(/C=C\c1cccnc1)N[C@H]1c2ccccc2C[C@H]1O ZINC000147274123 CD On-Demand Anodyne PLM2_PLAFA 31 44 O=C(/C=C\c1cccnc1)N[C@H]1c2ccccc2C[C@H]1O ZINC000147274123 CD On-Demand Anodyne Q8IM16_PLAF7 0 41 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1ccc2nccnc2c1 ZINC000147274143 DE On-Demand Anodyne FOLH1 40 32 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1ccc2nccnc2c1 ZINC000147274143 DE On-Demand Anodyne ANPEP 33 43 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1ccc2nccnc2c1 ZINC000147274143 DE On-Demand Anodyne CAPNS1 47 33 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1ccc2nccnc2c1 ZINC000147274143 DE On-Demand Anodyne CAPN1 59 37 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1ccc2nccnc2c1 ZINC000147274143 DE On-Demand Anodyne CAPN2 79 34 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1ccc2nccnc2c1 ZINC000147274143 DE On-Demand Anodyne FPR1 47 34 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne ESR1 43 36 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne HTR1A 21 56 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne DRD2 30 56 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne DRD4 21 50 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne HTR2A 25 59 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne SLC6A4 33 47 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne HRH1 38 50 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne SLC6A3 59 47 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne KCNH2 26 43 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne GRIN2B 54 44 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne LTA4H 84 57 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne HTR7 27 56 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne HRH3 48 48 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne SIGMAR1 61 56 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne NPY1R 42 35 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne CCR3 113 46 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne HTR5A 15 42 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne CYP2D6 17 48 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne CHRNA10 43 36 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne GRIN2C 19 41 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne CACNA1G 28 48 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne PSMB2 41 42 Fc1ccc(C[C@@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274175 CH On-Demand Anodyne PSMB1 45 42 Cc1nccn1-c1ccc(CNC(=O)Nc2ccc(N3CCOCC3)nc2)cc1F ZINC000147274190 HF On-Demand Anodyne MTOR 41 38 Cc1nccn1-c1ccc(CNC(=O)Nc2ccc(N3CCOCC3)nc2)cc1F ZINC000147274190 HF On-Demand Anodyne STAT6 43 32 Cc1nccn1-c1ccc(CNC(=O)Nc2ccc(N3CCOCC3)nc2)cc1F ZINC000147274190 HF On-Demand Anodyne DGAT1 39 43 Cc1nccn1-c1ccc(CNC(=O)Nc2ccc(N3CCOCC3)nc2)cc1F ZINC000147274190 HF On-Demand Anodyne NAMPT 35 40 CCCNc1ncc(F)c(Oc2ccccc2C(C)C)n1 ZINC000147274195 CI For-Sale Anodyne P2RX2 46 34 COc1ccccc1NC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147274216 HF On-Demand Anodyne OXTR 20 41 CCNCc1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147274262 CI For-Sale Anodyne LEF 41 39 CCNCC(=O)NN(C)C ZINC000147274334 AB For-Sale Reactive KDM7A 0 46 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274381 GG On-Demand Anodyne PIK3CA 48 42 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274381 GG On-Demand Anodyne MTOR 107 42 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274381 GG On-Demand Anodyne PIK3CG 39 40 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274381 GG On-Demand Anodyne STAT6 53 35 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274381 GG On-Demand Anodyne DGAT1 65 53 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274381 GG On-Demand Anodyne HPGDS 15 41 CN(C)C(=O)NCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147274402 CC On-Demand Anodyne DRD4 47 36 CN(C)C(=O)NCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147274402 CC On-Demand Anodyne AKR1C3 42 40 CN(C)C(=O)NCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147274402 CC On-Demand Anodyne KDM4E 28 47 CN(C)C(=O)NCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147274402 CC On-Demand Anodyne KCNK3 43 34 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne ESR1 43 36 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne HTR1A 21 56 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne DRD2 30 56 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne DRD4 21 50 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne HTR2A 25 59 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne SLC6A4 33 47 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne HRH1 38 50 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne SLC6A3 59 47 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne KCNH2 26 43 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne GRIN2B 54 44 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne LTA4H 84 57 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne HTR7 27 56 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne HRH3 48 48 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne SIGMAR1 61 56 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne NPY1R 42 35 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne CCR3 113 46 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne HTR5A 15 42 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne CYP2D6 17 48 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne CHRNA10 43 36 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne GRIN2C 19 41 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne CACNA1G 28 48 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne PSMB2 41 42 Fc1ccc(C[C@H]2CCN(CCOc3ccccc3)C2)cc1 ZINC000147274403 CH On-Demand Anodyne PSMB1 45 42 COc1ccccc1NC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147274424 HF On-Demand Anodyne OXTR 20 41 CNCc1ccccc1Oc1ccc(Cl)c(F)c1 ZINC000147274486 CH For-Sale Anodyne SLC6A2 19 63 CNCc1ccccc1Oc1ccc(Cl)c(F)c1 ZINC000147274486 CH For-Sale Anodyne HTR2A 0 78 CNCc1ccccc1Oc1ccc(Cl)c(F)c1 ZINC000147274486 CH For-Sale Anodyne SLC6A4 32 78 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274579 GG On-Demand Anodyne PIK3CA 48 42 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274579 GG On-Demand Anodyne MTOR 107 42 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274579 GG On-Demand Anodyne PIK3CG 39 40 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274579 GG On-Demand Anodyne STAT6 53 35 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274579 GG On-Demand Anodyne DGAT1 65 53 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274579 GG On-Demand Anodyne HPGDS 15 41 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)NCC1CC1 ZINC000147274608 DC For-Sale Anodyne PTGDR2 35 40 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)NCC1CC1 ZINC000147274608 DC For-Sale Anodyne CACNA1I 55 36 CC(=O)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147274723 FJ On-Demand Anodyne MAOB 19 40 CC(=O)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147274723 FJ On-Demand Anodyne CPT1A 45 39 CC(=O)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147274723 FJ On-Demand Anodyne PRNP 39 51 CC(=O)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147274723 FJ On-Demand Anodyne CSF1R 18 41 CC(=O)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147274723 FJ On-Demand Anodyne TAAR1 27 53 CC(=O)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147274723 FJ On-Demand Anodyne AKR1C3 19 40 CC(=O)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147274723 FJ On-Demand Anodyne AKR1C2 15 40 CC(=O)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147274723 FJ On-Demand Anodyne SMO 21 42 CC(=O)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147274723 FJ On-Demand Anodyne SENP1 0 40 CC(=O)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147274723 FJ On-Demand Anodyne KCNK3 71 40 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274794 GG On-Demand Anodyne PIK3CA 48 42 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274794 GG On-Demand Anodyne MTOR 107 42 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274794 GG On-Demand Anodyne PIK3CG 39 40 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274794 GG On-Demand Anodyne STAT6 53 35 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274794 GG On-Demand Anodyne DGAT1 65 53 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274794 GG On-Demand Anodyne HPGDS 15 41 CN(Cc1cscn1)C(=O)NCc1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147274804 HD On-Demand Anodyne NAMPT 65 48 NS(=O)(=O)c1cc(Cl)ccc1OCCn1ccnc1 ZINC000147274831 DD For-Sale Anodyne CYP19A1 16 44 NS(=O)(=O)c1cc(Cl)ccc1OCCn1ccnc1 ZINC000147274831 DD For-Sale Anodyne CYP11B1 25 45 NS(=O)(=O)c1cc(Cl)ccc1OCCn1ccnc1 ZINC000147274831 DD For-Sale Anodyne TBXAS1 48 46 NS(=O)(=O)c1cc(Cl)ccc1OCCn1ccnc1 ZINC000147274831 DD For-Sale Anodyne CYP11B2 27 40 NS(=O)(=O)c1cc(Cl)ccc1OCCn1ccnc1 ZINC000147274831 DD For-Sale Anodyne CYP17A1 24 43 NS(=O)(=O)c1cc(Cl)ccc1OCCn1ccnc1 ZINC000147274831 DD For-Sale Anodyne HMOX2 45 37 CCCCCCCCNc1cc(Cl)nc(SC)n1 ZINC000147274850 CJ For-Sale Mild PTGES 20 42 CC(C)CCCCNCc1ccc(O)cc1 ZINC000147274852 BG For-Sale Anodyne OPRM1 0 44 CC(C)CCCCNCc1ccc(O)cc1 ZINC000147274852 BG For-Sale Anodyne FDFT1 0 41 CC(C)CCCCNCc1ccc(O)cc1 ZINC000147274852 BG For-Sale Anodyne GRIA1 60 37 CC(C)CCCCNCc1ccc(O)cc1 ZINC000147274852 BG For-Sale Anodyne S1PR2 45 44 CC(C)CCCCNCc1ccc(O)cc1 ZINC000147274852 BG For-Sale Anodyne SLC6A13 0 43 CC(C)CCCCNCc1ccc(O)cc1 ZINC000147274852 BG For-Sale Anodyne LEF 94 39 CC(C)CCCCNCc1ccc(O)cc1 ZINC000147274852 BG For-Sale Anodyne GPM3 0 49 COc1ccc(CNc2cc(CN)ccn2)cc1 ZINC000147274856 BE For-Sale Anodyne PTGDR 31 45 COc1ccc(CNc2cc(CN)ccn2)cc1 ZINC000147274856 BE For-Sale Anodyne PROKR1 54 33 CO[C@H](C)C(=O)c1c(F)ccc(C)c1F ZINC000147274901 BE For-Sale Anodyne LEF 54 34 CNCc1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147274942 DJ For-Sale Anodyne SLC6A4 23 60 COc1ccc(S(=O)(=O)N(Cc2ccc(N3CCN(C(C)=O)CC3)cc2F)C2CCC2)cc1 ZINC000147274978 JG Annotated Clean AVPR1B 27 46 COc1ccc(S(=O)(=O)N(Cc2ccc(N3CCN(C(C)=O)CC3)cc2F)C2CCC2)cc1 ZINC000147274978 JG Annotated Clean BMP1 80 42 COc1ccc(S(=O)(=O)N(Cc2ccc(N3CCN(C(C)=O)CC3)cc2F)C2CCC2)cc1 ZINC000147274978 JG Annotated Clean MMP13 42 40 COc1ccc(S(=O)(=O)N(Cc2ccc(N3CCN(C(C)=O)CC3)cc2F)C2CCC2)cc1 ZINC000147274978 JG Annotated Clean MMP2 21 40 COc1ccc(S(=O)(=O)N(Cc2ccc(N3CCN(C(C)=O)CC3)cc2F)C2CCC2)cc1 ZINC000147274978 JG Annotated Clean MMP3 39 40 COc1ccc(S(=O)(=O)N(Cc2ccc(N3CCN(C(C)=O)CC3)cc2F)C2CCC2)cc1 ZINC000147274978 JG Annotated Clean MMP8 32 40 COc1ccc(S(=O)(=O)N(Cc2ccc(N3CCN(C(C)=O)CC3)cc2F)C2CCC2)cc1 ZINC000147274978 JG Annotated Clean MMP1 38 40 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274989 GG On-Demand Anodyne PIK3CA 48 42 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274989 GG On-Demand Anodyne MTOR 107 42 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274989 GG On-Demand Anodyne PIK3CG 39 40 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274989 GG On-Demand Anodyne STAT6 53 35 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274989 GG On-Demand Anodyne DGAT1 65 53 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(N2CCOCC2)nc1 ZINC000147274989 GG On-Demand Anodyne HPGDS 15 41 CC(C)(C)[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147275007 CE For-Sale Anodyne FFAR1 0 40 CC(C)(C)[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147275007 CE For-Sale Anodyne GPR88 0 48 CC[C@@H](CNC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147275034 DG On-Demand Anodyne BMP1 51 36 CO[C@@H](C)C(=O)c1c(F)ccc(C)c1F ZINC000147275066 BE For-Sale Anodyne LEF 54 34 O=c1cc(I)oc2ccccc12 ZINC000147275206 CE For-Sale Anodyne NQO1 44 36 O=c1cc(I)oc2ccccc12 ZINC000147275206 CE For-Sale Anodyne TNKS 54 56 O=c1cc(I)oc2ccccc12 ZINC000147275206 CE For-Sale Anodyne TNKS2 17 56 CC(C)(C)[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147275217 CE For-Sale Anodyne FFAR1 0 40 CC(C)(C)[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147275217 CE For-Sale Anodyne GPR88 0 48 O=C(Nc1ccc2nccnc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147275220 FG On-Demand Anodyne OPRL1 15 40 O=C(Nc1ccc2nccnc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147275220 FG On-Demand Anodyne FLT1 24 40 O=C(Nc1ccc2nccnc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147275220 FG On-Demand Anodyne KDR 21 40 O=C(Nc1ccc2nccnc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147275220 FG On-Demand Anodyne GRM4 53 38 O=C(Nc1ccc2nccnc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147275220 FG On-Demand Anodyne MET 24 50 O=C(Nc1ccc2nccnc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147275220 FG On-Demand Anodyne NR1I2 42 34 O=C(Nc1ccc2nccnc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147275220 FG On-Demand Anodyne NR2E3 67 39 O=C(Nc1ccc2nccnc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147275220 FG On-Demand Anodyne SHH 23 40 O=C(Nc1ccc2nccnc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147275220 FG On-Demand Anodyne KCNK3 64 38 O=C(Nc1ccc2nccnc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147275220 FG On-Demand Anodyne KCNK9 51 32 CC[C@H](CNC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147275259 DG On-Demand Anodyne BMP1 51 36 NS(=O)(=O)c1cc(Cl)ccc1OCCCn1ccnc1 ZINC000147275270 DD For-Sale Anodyne CYP19A1 15 45 NS(=O)(=O)c1cc(Cl)ccc1OCCCn1ccnc1 ZINC000147275270 DD For-Sale Anodyne CYP11B1 18 40 NS(=O)(=O)c1cc(Cl)ccc1OCCCn1ccnc1 ZINC000147275270 DD For-Sale Anodyne TBXAS1 50 47 NS(=O)(=O)c1cc(Cl)ccc1OCCCn1ccnc1 ZINC000147275270 DD For-Sale Anodyne CYP11B2 0 40 NS(=O)(=O)c1cc(Cl)ccc1OCCCn1ccnc1 ZINC000147275270 DD For-Sale Anodyne HMOX1 19 42 NS(=O)(=O)c1cc(Cl)ccc1OCCCn1ccnc1 ZINC000147275270 DD For-Sale Anodyne CYP17A1 24 47 NS(=O)(=O)c1cc(Cl)ccc1OCCCn1ccnc1 ZINC000147275270 DD For-Sale Anodyne HMOX2 57 41 NS(=O)(=O)c1cc(Cl)ccc1OCCCn1ccnc1 ZINC000147275270 DD For-Sale Anodyne QPCT 36 40 Cc1cc(C)c(C(=O)CSc2nnc(CCC(N)=O)n2Cc2ccco2)cc1C ZINC000147275310 HG On-Demand Anodyne HCRTR2 15 46 CC(C)(C)[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147275390 CE For-Sale Anodyne FFAR1 0 40 CC(C)(C)[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147275390 CE For-Sale Anodyne GPR88 0 48 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)Nc2ccc(N(C)C)nc2)cc1 ZINC000147275436 HE On-Demand Anodyne PRMT3 18 41 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)Nc2ccc(N(C)C)nc2)cc1 ZINC000147275436 HE On-Demand Anodyne NAMPT 71 46 CC(C)(C)[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147275496 CE For-Sale Anodyne FFAR1 0 40 CC(C)(C)[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147275496 CE For-Sale Anodyne GPR88 0 48 CCN(CC)C(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147275567 ED For-Sale Anodyne PTGDR2 24 41 CC[C@H](C(=O)N1CCC[C@H](CCBr)C1)c1ccccc1 ZINC000147275666 EI For-Sale Reactive KCNQ2 44 40 CC[C@H](C(=O)N1CCC[C@H](CCBr)C1)c1ccccc1 ZINC000147275666 EI For-Sale Reactive KCNQ4 0 40 CC(C)c1ccccc1Oc1nc(N)ncc1Cl ZINC000147275700 CH For-Sale Anodyne P2RX2 60 46 CC(C)c1ccccc1Oc1nc(N)ncc1Cl ZINC000147275700 CH For-Sale Anodyne P2RX3 36 46 Cc1ccc(C(=O)N[C@H](C(=O)O)C(C)(C)C)cc1Br ZINC000147275728 EF On-Demand Anodyne DERP1 0 41 Cc1c(F)cccc1NC(=O)c1cccc2c1OCCN2 ZINC000147275731 CG For-Sale Anodyne G2YM83_BOTF4 64 33 CCN(CC)C(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147275766 ED For-Sale Anodyne PTGDR2 24 41 O=C(Nc1ccc2nccnc2c1)c1csc(-c2ccccc2F)n1 ZINC000147275865 FI On-Demand Anodyne MPL 40 38 O=C(Nc1ccc2nccnc2c1)c1csc(-c2ccccc2F)n1 ZINC000147275865 FI On-Demand Anodyne GRM4 76 45 O=C(Nc1ccc2nccnc2c1)c1csc(-c2ccccc2F)n1 ZINC000147275865 FI On-Demand Anodyne NR2E3 52 37 O=C(Nc1ccc2nccnc2c1)c1csc(-c2ccccc2F)n1 ZINC000147275865 FI On-Demand Anodyne KCNK3 29 41 CC[C@@H](C(=O)N1CCC[C@H](CCBr)C1)c1ccccc1 ZINC000147275877 EI For-Sale Reactive KCNQ2 44 40 CC[C@@H](C(=O)N1CCC[C@H](CCBr)C1)c1ccccc1 ZINC000147275877 EI For-Sale Reactive KCNQ4 0 40 Brc1ccc(Cc2ccncc2)cc1 ZINC000147275928 BG For-Sale Anodyne CYP11B1 18 54 Brc1ccc(Cc2ccncc2)cc1 ZINC000147275928 BG For-Sale Anodyne CYP11B2 21 54 Brc1ccc(Cc2ccncc2)cc1 ZINC000147275928 BG For-Sale Anodyne CYP17A1 17 54 O=C(C[C@@H]1CNCCO1)c1ccccc1 ZINC000147276062 BD For-Sale Anodyne MGLL 0 40 CCNCc1ccc(Oc2ccc(Cl)c(F)c2)c(C)c1 ZINC000147276069 CJ For-Sale Anodyne LEF 47 39 CN(C)c1cccc(NC(=O)c2nc(-c3cccnc3)cnc2N)c1 ZINC000147276080 EE For-Sale Anodyne ABL1 19 45 CN(C)c1cccc(NC(=O)c2nc(-c3cccnc3)cnc2N)c1 ZINC000147276080 EE For-Sale Anodyne GSK3B 20 51 CN(C)c1cccc(NC(=O)c2nc(-c3cccnc3)cnc2N)c1 ZINC000147276080 EE For-Sale Anodyne MAPK9 20 42 CN(C)c1cccc(NC(=O)c2nc(-c3cccnc3)cnc2N)c1 ZINC000147276080 EE For-Sale Anodyne MAPK10 18 42 CN(C)c1cccc(NC(=O)c2nc(-c3cccnc3)cnc2N)c1 ZINC000147276080 EE For-Sale Anodyne PIK3CG 17 46 CN(C)c1cccc(NC(=O)c2nc(-c3cccnc3)cnc2N)c1 ZINC000147276080 EE For-Sale Anodyne CSF1R 15 48 CN(C)c1cccc(NC(=O)c2nc(-c3cccnc3)cnc2N)c1 ZINC000147276080 EE For-Sale Anodyne ATR 81 71 CN(C)c1cccc(NC(=O)c2nc(-c3cccnc3)cnc2N)c1 ZINC000147276080 EE For-Sale Anodyne BTK 17 42 CN(C)c1cccc(NC(=O)c2nc(-c3cccnc3)cnc2N)c1 ZINC000147276080 EE For-Sale Anodyne BRAF 23 44 CN(C)c1cccc(NC(=O)c2nc(-c3cccnc3)cnc2N)c1 ZINC000147276080 EE For-Sale Anodyne TYRO3 47 41 CC[C@H](C(=O)N1CCC[C@@H](CCBr)C1)c1ccccc1 ZINC000147276098 EI For-Sale Reactive KCNQ2 44 40 CC[C@H](C(=O)N1CCC[C@@H](CCBr)C1)c1ccccc1 ZINC000147276098 EI For-Sale Reactive KCNQ4 0 40 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3cc(F)cc(F)c3)c(F)c2)CC1 ZINC000147276156 JH Annotated Clean SSTR3 48 37 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C)c(NC(C)=O)c1C)C2 ZINC000147276192 FG On-Demand Anodyne MTNR1A 20 45 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C)c(NC(C)=O)c1C)C2 ZINC000147276192 FG On-Demand Anodyne ROCK2 33 49 CC[C@@H](Oc1cccc(Cn2c(C)c(C(=O)c3ccc(OC)cc3)c3ccc(OC(F)(F)F)cc32)c1)C(=O)O ZINC000147276193 KK For-Sale Anodyne PPARG 55 86 CC[C@@H](Oc1cccc(Cn2c(C)c(C(=O)c3ccc(OC)cc3)c3ccc(OC(F)(F)F)cc32)c1)C(=O)O ZINC000147276193 KK For-Sale Anodyne PPARA 29 86 CC[C@@H](Oc1cccc(Cn2c(C)c(C(=O)c3ccc(OC)cc3)c3ccc(OC(F)(F)F)cc32)c1)C(=O)O ZINC000147276193 KK For-Sale Anodyne PLA2G2A 45 41 CC[C@@H](Oc1cccc(Cn2c(C)c(C(=O)c3ccc(OC)cc3)c3ccc(OC(F)(F)F)cc32)c1)C(=O)O ZINC000147276193 KK For-Sale Anodyne PTGDS 27 44 O=C(C[C@H]1CNCCO1)c1ccccc1 ZINC000147276253 BD For-Sale Anodyne MGLL 0 40 C=C(C)[C@H]1CCc2ccc(O)cc2[C@]1(C)CCC(=O)O ZINC000147276266 CH Annotated Mild NR1H3 27 44 COCCNCc1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147276274 DI For-Sale Anodyne LEF 49 39 COc1cc(CNCC(F)F)ccc1O ZINC000147276279 BD For-Sale Anodyne PNLIP 0 40 COc1cc(CNCC(F)F)ccc1O ZINC000147276279 BD For-Sale Anodyne TRPV1 28 49 COc1cc(CNCC(F)F)ccc1O ZINC000147276279 BD For-Sale Anodyne SLC6A13 0 45 COc1cc(CNCC(F)F)ccc1O ZINC000147276279 BD For-Sale Anodyne TTR 0 54 COc1cc(CNCC(F)F)ccc1O ZINC000147276279 BD For-Sale Anodyne N1L 0 44 COc1cc(CNCC(F)F)ccc1O ZINC000147276279 BD For-Sale Anodyne CAN2 0 54 COc1cc(CNCC(F)F)ccc1O ZINC000147276279 BD For-Sale Anodyne SLC22A3 0 43 CC[C@@H](C(=O)N1CCC[C@@H](CCBr)C1)c1ccccc1 ZINC000147276314 EI For-Sale Reactive KCNQ2 44 40 CC[C@@H](C(=O)N1CCC[C@@H](CCBr)C1)c1ccccc1 ZINC000147276314 EI For-Sale Reactive KCNQ4 0 40 Cc1cc(C(=O)Nc2cccc3cccnc23)cc([N+](=O)[O-])c1 ZINC000147276329 DH On-Demand Bother PDE4A 0 42 Cc1cc(C(=O)Nc2cccc3cccnc23)cc([N+](=O)[O-])c1 ZINC000147276329 DH On-Demand Bother PDE4D 16 40 Cc1cc(C(=O)Nc2cccc3cccnc23)cc([N+](=O)[O-])c1 ZINC000147276329 DH On-Demand Bother PDE4C 18 42 Cc1cc(C(=O)Nc2cccc3cccnc23)cc([N+](=O)[O-])c1 ZINC000147276329 DH On-Demand Bother NFKBIA 0 53 Cc1cc(C(=O)Nc2cccc3cccnc23)cc([N+](=O)[O-])c1 ZINC000147276329 DH On-Demand Bother WNT3 17 42 Cc1cc(C(=O)Nc2cccc3cccnc23)cc([N+](=O)[O-])c1 ZINC000147276329 DH On-Demand Bother TNKS 21 43 CNCCCC(=O)NN(C)C ZINC000147276367 AB For-Sale Reactive KDM7A 0 54 CC(C)(C)OC(=O)N1CCC[C@H]1c1nc2c([nH]1)COc1cc(Br)ccc1-2 ZINC000147276412 HJ For-Sale Anodyne PRCP 40 33 C[C@H](CNS(=O)(=O)c1ccc(F)c(Cl)c1)CC(=O)O ZINC000147276484 DD On-Demand Anodyne TBXA2R 48 39 Cc1cc(C(=O)Nc2ccc3nc(-c4cc(F)ccc4F)[nH]c3c2)no1 ZINC000147276489 FI On-Demand Anodyne NR2E3 66 38 Cc1cc(C(=O)Nc2ccc3nc(-c4cc(F)ccc4F)[nH]c3c2)no1 ZINC000147276489 FI On-Demand Anodyne SHH 27 48 C=C(C)[C@H]1CCc2ccc(O)cc2[C@]1(C)CCC(=O)OC ZINC000147276506 CH Annotated Mild NR1H3 27 43 CCCCCCCCCC(=O)N1CCC[C@H](CCBr)C1 ZINC000147276601 EK For-Sale Reactive GNAI1 0 50 CCCCCCCCCC(=O)N1CCC[C@H](CCBr)C1 ZINC000147276601 EK For-Sale Reactive GNAI3 0 52 CCCCCCCCCC(=O)N1CCC[C@H](CCBr)C1 ZINC000147276601 EK For-Sale Reactive GNAO1 0 50 CCCNCc1cccc(Oc2ccc(Cl)c(F)c2)c1 ZINC000147276682 CJ For-Sale Anodyne CRTM 55 39 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@@H]1CCCc2ccccc21 ZINC000147276694 DF On-Demand Anodyne CTSK 32 49 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@@H]1CCCc2ccccc21 ZINC000147276694 DF On-Demand Anodyne CTSV 16 49 C[C@@H](CNS(=O)(=O)c1ccc(F)c(Cl)c1)CC(=O)O ZINC000147276705 DD On-Demand Anodyne TBXA2R 48 39 CCCCCCCCCC(=O)N1CCC[C@@H](CCBr)C1 ZINC000147276817 EK For-Sale Reactive GNAI1 0 50 CCCCCCCCCC(=O)N1CCC[C@@H](CCBr)C1 ZINC000147276817 EK For-Sale Reactive GNAI3 0 52 CCCCCCCCCC(=O)N1CCC[C@@H](CCBr)C1 ZINC000147276817 EK For-Sale Reactive GNAO1 0 50 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@H](C)CC)C(=O)O ZINC000147276839 IB For-Sale Anodyne OPRM1 15 40 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@H](C)CC)C(=O)O ZINC000147276839 IB For-Sale Anodyne OPRD1 24 41 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@H](C)CC)C(=O)O ZINC000147276839 IB For-Sale Anodyne CPB2 21 41 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@H](C)CC)C(=O)O ZINC000147276839 IB For-Sale Anodyne ADRBK1 15 48 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@H](C)CC)C(=O)O ZINC000147276839 IB For-Sale Anodyne HLA-A 64 52 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@H](C)CC)C(=O)O ZINC000147276839 IB For-Sale Anodyne GRPR 24 40 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@H](C)CC)C(=O)O ZINC000147276839 IB For-Sale Anodyne ENPEP 61 35 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@H](C)CC)C(=O)O ZINC000147276839 IB For-Sale Anodyne SIRT1 15 40 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@H](C)CC)C(=O)O ZINC000147276839 IB For-Sale Anodyne F2RL1 68 38 CC(=O)Nc1ccc(Cl)c(NC(=O)c2cnn(-c3ccccc3Cl)c2)c1 ZINC000147276841 GI On-Demand Anodyne MAOB 17 41 CC(=O)Nc1ccc(Cl)c(NC(=O)c2cnn(-c3ccccc3Cl)c2)c1 ZINC000147276841 GI On-Demand Anodyne GRM4 52 38 CC(=O)Nc1ccc(Cl)c(NC(=O)c2cnn(-c3ccccc3Cl)c2)c1 ZINC000147276841 GI On-Demand Anodyne MAPK10 21 44 CC(=O)Nc1ccc(Cl)c(NC(=O)c2cnn(-c3ccccc3Cl)c2)c1 ZINC000147276841 GI On-Demand Anodyne EPHB3 60 38 CC(=O)Nc1ccc(Cl)c(NC(=O)c2cnn(-c3ccccc3Cl)c2)c1 ZINC000147276841 GI On-Demand Anodyne SHH 46 39 CC(=O)Nc1ccc(Cl)c(NC(=O)c2cnn(-c3ccccc3Cl)c2)c1 ZINC000147276841 GI On-Demand Anodyne SMO 24 41 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@@H]1CCCc2ccccc21 ZINC000147276876 DF On-Demand Anodyne CTSK 32 49 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@@H]1CCCc2ccccc21 ZINC000147276876 DF On-Demand Anodyne CTSV 16 49 CCCCCCCCNc1nc(Cl)nc(-n2cncn2)n1 ZINC000147276958 DF For-Sale Mild PDE4A 0 43 C#Cc1c(N)c(=O)oc2ccccc12 ZINC000147277006 AD For-Sale Mild NQO1 24 40 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@@H](C)CC)C(=O)O ZINC000147277025 IB For-Sale Anodyne OPRM1 15 40 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@@H](C)CC)C(=O)O ZINC000147277025 IB For-Sale Anodyne OPRD1 24 41 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@@H](C)CC)C(=O)O ZINC000147277025 IB For-Sale Anodyne CPB2 21 41 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@@H](C)CC)C(=O)O ZINC000147277025 IB For-Sale Anodyne ADRBK1 15 48 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@@H](C)CC)C(=O)O ZINC000147277025 IB For-Sale Anodyne HLA-A 64 52 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@@H](C)CC)C(=O)O ZINC000147277025 IB For-Sale Anodyne GRPR 24 40 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@@H](C)CC)C(=O)O ZINC000147277025 IB For-Sale Anodyne ENPEP 61 35 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@@H](C)CC)C(=O)O ZINC000147277025 IB For-Sale Anodyne SIRT1 15 40 CC[C@H](C)[C@H](NC(=O)CNC(=O)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)[C@@H](C)CC)C(=O)O ZINC000147277025 IB For-Sale Anodyne F2RL1 68 38 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@H]1CCCc2ccccc21 ZINC000147277049 DF On-Demand Anodyne CTSK 32 49 CCCC[C@H](NC(N)=O)C(=O)N(C)[C@H]1CCCc2ccccc21 ZINC000147277049 DF On-Demand Anodyne CTSV 16 49 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCC1 ZINC000147277169 DD For-Sale Anodyne HTR2A 24 42 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCC1 ZINC000147277169 DD For-Sale Anodyne HTR2C 16 42 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCC1 ZINC000147277169 DD For-Sale Anodyne LTA4H 36 48 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCC1 ZINC000147277169 DD For-Sale Anodyne HRH3 29 45 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCC1 ZINC000147277169 DD For-Sale Anodyne MCHR1 0 41 NS(=O)(=O)c1cc(Cl)ccc1OCCN1CCCC1 ZINC000147277169 DD For-Sale Anodyne PSMB1 41 38 CC(=O)NOCc1cccc2ccccc12 ZINC000147277175 BE On-Demand Anodyne NQO2 33 40 CC(=O)NOCc1cccc2ccccc12 ZINC000147277175 BE On-Demand Anodyne MTNR1A 22 40 CC(=O)NOCc1cccc2ccccc12 ZINC000147277175 BE On-Demand Anodyne MTNR1B 25 43 CC(=O)NOCc1cccc2ccccc12 ZINC000147277175 BE On-Demand Anodyne KCNJ2 0 42 C[C@@H](C(=O)O)N(C)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147277182 BD For-Sale Anodyne GPR88 0 48 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@H]1CCCc2ccccc21 ZINC000147277229 DF On-Demand Anodyne CTSK 32 49 CCCC[C@@H](NC(N)=O)C(=O)N(C)[C@H]1CCCc2ccccc21 ZINC000147277229 DF On-Demand Anodyne CTSV 16 49 CN1CCC(CNC(=O)c2cccc3c2OCCN3)CC1 ZINC000147277264 CD For-Sale Anodyne HTR4 75 47 CN1CCC(CNC(=O)c2cccc3c2OCCN3)CC1 ZINC000147277264 CD For-Sale Anodyne CACNA1I 63 37 C[C@H](CNS(=O)(=O)c1ccc(F)c([N+](=O)[O-])c1)CC(=O)O ZINC000147277265 DD For-Sale Bother COLA 83 35 C[C@H](CNS(=O)(=O)c1ccc(F)c([N+](=O)[O-])c1)CC(=O)O ZINC000147277265 DD For-Sale Bother LEF 56 35 C[C@H](C(=O)O)N(C)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147277317 BD For-Sale Anodyne GPR88 0 48 CN(C)C(=O)NCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147277360 CB On-Demand Anodyne EPHX2 16 40 COCC[C@@H](N)C(=O)NN(C)C ZINC000147277385 AA For-Sale Reactive CHRNA4 46 36 CC(C)c1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147277419 EI For-Sale Reactive L3MBTL3 59 39 C[C@@H](CNS(=O)(=O)c1ccc(F)c([N+](=O)[O-])c1)CC(=O)O ZINC000147277465 DD For-Sale Bother COLA 83 35 C[C@@H](CNS(=O)(=O)c1ccc(F)c([N+](=O)[O-])c1)CC(=O)O ZINC000147277465 DD For-Sale Bother LEF 56 35 C[C@@H](C(=O)O)N(C)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147277481 BD For-Sale Anodyne GPR88 0 48 CN1CCC[C@H](CNC(=O)c2cccc3c2OCCN3)C1 ZINC000147277511 CD For-Sale Anodyne HTR4 62 42 CN1CCC[C@H](CNC(=O)c2cccc3c2OCCN3)C1 ZINC000147277511 CD For-Sale Anodyne CACNA1I 40 32 COCC[C@H](N)C(=O)NN(C)C ZINC000147277521 AA For-Sale Reactive CHRNA4 46 36 Cc1cc(N)cc(S(=O)(=O)NCCCCC(C)C)c1F ZINC000147277550 DF For-Sale Anodyne LEF 50 38 O=C(Nc1ccc2c(c1)OCCO2)c1cc(O)c(O)c(O)c1 ZINC000147277560 DD For-Sale Clean PLAU 17 50 O=C(Nc1ccc2c(c1)OCCO2)c1cc(O)c(O)c(O)c1 ZINC000147277560 DD For-Sale Clean KCNK3 53 33 CC(C)c1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147277568 EI For-Sale Reactive L3MBTL3 59 39 CC[C@@H](C)c1ccccc1Oc1nc(N)nc(OC)n1 ZINC000147277589 CF For-Sale Anodyne AO-ACHE 0 41 C[C@H](C(=O)O)N(C)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147277597 BD For-Sale Anodyne GPR88 0 48 C=C1CC[C@H]2C(C)(C)CCC[C@]2(C)[C@H]1Cc1coccc1=O ZINC000147277641 DJ Annotated Mild ICL1 0 43 CC[C@@H]([C@H](C)OC)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147277652 JK Annotated Anodyne TP53 60 83 CC[C@@H]([C@H](C)OC)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147277652 JK Annotated Anodyne MDM2 261 83 O=C(Nc1cc(Cl)ccc1Br)c1cc(Cl)ccc1F ZINC000147277658 FK On-Demand Anodyne KCNMA1 30 55 O=C(Nc1cc(Cl)ccc1Br)c1cc(Cl)ccc1F ZINC000147277658 FK On-Demand Anodyne Q25615_ONCVO 43 34 O=C(Nc1cc(Cl)ccc1Br)c1cc(Cl)ccc1F ZINC000147277658 FK On-Demand Anodyne TMPRSS4 0 44 CN1CCC[C@@H](CNC(=O)c2cccc3c2OCCN3)C1 ZINC000147277683 CD For-Sale Anodyne HTR4 62 42 CN1CCC[C@@H](CNC(=O)c2cccc3c2OCCN3)C1 ZINC000147277683 CD For-Sale Anodyne CACNA1I 40 32 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1-c1ccccc1 ZINC000147277690 EF On-Demand Anodyne OXTR 25 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1-c1ccccc1 ZINC000147277690 EF On-Demand Anodyne AVPR1A 16 41 CN(C)NC(=O)C[C@@H]1CCCNC1 ZINC000147277730 AB For-Sale Reactive CPN1 0 42 CCCC[C@H](NC(N)=O)C(=O)NCCCN1C(=O)NC2(CCCC2)C1=O ZINC000147277745 FC On-Demand Anodyne PCSK5 50 32 CC[C@H](C)c1ccccc1Oc1nc(N)nc(OC)n1 ZINC000147277755 CF For-Sale Anodyne AO-ACHE 0 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccccc1-c1ccccc1 ZINC000147277802 EF On-Demand Anodyne OXTR 25 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccccc1-c1ccccc1 ZINC000147277802 EF On-Demand Anodyne AVPR1A 16 41 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147277828 CF On-Demand Anodyne GHRHR 43 34 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147277828 CF On-Demand Anodyne GRIN2B 29 41 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147277828 CF On-Demand Anodyne SIGMAR1 22 45 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147277828 CF On-Demand Anodyne PREP 64 48 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147277828 CF On-Demand Anodyne FAAH 25 42 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147277828 CF On-Demand Anodyne MGLL 0 42 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147277828 CF On-Demand Anodyne CYP2J2 40 37 O=C(O)C1(NCc2ccccc2C(F)(F)F)CCC1 ZINC000147277839 CF For-Sale Anodyne RBP4 67 37 COc1ccc(C[C@H](NC(=O)N(C)Cc2cscn2)c2ccc(OC)cc2)cc1 ZINC000147277841 HI On-Demand Anodyne BMP1 63 34 COc1ccc(C[C@H](NC(=O)N(C)Cc2cscn2)c2ccc(OC)cc2)cc1 ZINC000147277841 HI On-Demand Anodyne CYP3A4 20 44 CCCNCc1ccccc1Oc1ccc(Cl)c(F)c1 ZINC000147277844 CJ For-Sale Anodyne SLC6A4 15 55 C[C@H](Oc1ccc(Cl)cc1S(N)(=O)=O)C(=O)NC(N)=O ZINC000147277868 DB For-Sale Anodyne CPT1A 47 33 C[C@H](Oc1ccc(Cl)cc1S(N)(=O)=O)C(=O)NC(N)=O ZINC000147277868 DB For-Sale Anodyne CPT2 42 32 CN(C)NC(=O)C[C@H]1CCCNC1 ZINC000147277886 AB For-Sale Reactive CPN1 0 42 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1C(=O)NC2(CCCC2)C1=O ZINC000147277891 FC On-Demand Anodyne PCSK5 50 32 CN1CCCC[C@@H]1CNC(=O)c1cccc2c1OCCN2 ZINC000147277943 CD For-Sale Anodyne DRD2 28 43 CN1CCCC[C@@H]1CNC(=O)c1cccc2c1OCCN2 ZINC000147277943 CD For-Sale Anodyne CHRNA10 44 33 CN1CCCC[C@@H]1CNC(=O)c1cccc2c1OCCN2 ZINC000147277943 CD For-Sale Anodyne HCRTR2 28 40 CN1CCCC[C@@H]1CNC(=O)c1cccc2c1OCCN2 ZINC000147277943 CD For-Sale Anodyne ACKR3 51 35 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cc(NC(C)=O)ccc1Cl)C2 ZINC000147277948 FG On-Demand Anodyne MTNR1A 17 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cc(NC(C)=O)ccc1Cl)C2 ZINC000147277948 FG On-Demand Anodyne ROCK2 35 49 CCCNc1cc(Oc2ccccc2[C@@H](C)CC)ncn1 ZINC000147277968 CJ For-Sale Anodyne AO-ACHE 0 40 COc1ccc(C[C@@H](NC(=O)N(C)Cc2cscn2)c2ccc(OC)cc2)cc1 ZINC000147277999 HI On-Demand Anodyne BMP1 63 34 COc1ccc(C[C@@H](NC(=O)N(C)Cc2cscn2)c2ccc(OC)cc2)cc1 ZINC000147277999 HI On-Demand Anodyne SOAT1 18 46 COc1ccc(C[C@@H](NC(=O)N(C)Cc2cscn2)c2ccc(OC)cc2)cc1 ZINC000147277999 HI On-Demand Anodyne CYP3A4 20 44 C[C@@H](Oc1ccc(Cl)cc1S(N)(=O)=O)C(=O)NC(N)=O ZINC000147278004 DB For-Sale Anodyne CPT1A 47 33 C[C@@H](Oc1ccc(Cl)cc1S(N)(=O)=O)C(=O)NC(N)=O ZINC000147278004 DB For-Sale Anodyne CPT2 42 32 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147278007 CF On-Demand Anodyne GHRHR 43 34 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147278007 CF On-Demand Anodyne GRIN2B 29 41 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147278007 CF On-Demand Anodyne SIGMAR1 22 45 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147278007 CF On-Demand Anodyne PREP 64 48 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147278007 CF On-Demand Anodyne FAAH 25 42 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147278007 CF On-Demand Anodyne MGLL 0 42 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@@H]1N ZINC000147278007 CF On-Demand Anodyne CYP2J2 40 37 Fc1cc(Oc2ccccc2CNC2CC2)ccc1Cl ZINC000147278048 CJ For-Sale Anodyne SLC6A4 18 55 CN1CCCC[C@H]1CNC(=O)c1cccc2c1OCCN2 ZINC000147278082 CD For-Sale Anodyne DRD2 28 43 CN1CCCC[C@H]1CNC(=O)c1cccc2c1OCCN2 ZINC000147278082 CD For-Sale Anodyne CHRNA10 44 33 CN1CCCC[C@H]1CNC(=O)c1cccc2c1OCCN2 ZINC000147278082 CD For-Sale Anodyne HCRTR2 28 40 CN1CCCC[C@H]1CNC(=O)c1cccc2c1OCCN2 ZINC000147278082 CD For-Sale Anodyne ACKR3 51 35 CCCNc1cc(Oc2ccccc2[C@H](C)CC)ncn1 ZINC000147278091 CJ For-Sale Anodyne AO-ACHE 0 40 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278100 CF On-Demand Anodyne GHRHR 43 34 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278100 CF On-Demand Anodyne GRIN2B 29 41 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278100 CF On-Demand Anodyne SIGMAR1 22 45 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278100 CF On-Demand Anodyne PREP 64 48 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278100 CF On-Demand Anodyne FAAH 25 42 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278100 CF On-Demand Anodyne MGLL 0 42 CC[C@@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278100 CF On-Demand Anodyne CYP2J2 40 37 CN(C)NC(=O)CC[C@@H](CCN)C(C)(C)C ZINC000147278110 BD For-Sale Reactive KDM7A 0 43 N#Cc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147278136 CD On-Demand Mild CCR3 16 41 Cc1ccc(CNCC(=O)NCCc2ccccc2F)cc1 ZINC000147278209 DF For-Sale Anodyne SLC6A5 21 42 Cc1ccc(CNCC(=O)NCCc2ccccc2F)cc1 ZINC000147278209 DF For-Sale Anodyne LEF 58 36 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne OPRM1 19 42 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne OPRD1 23 42 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne MME 36 41 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne KLK3 64 38 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne PAPA1_CARPA 45 38 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne CTSK 43 41 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne CTSL 25 40 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne NPFFR2 40 35 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne C3AR1 59 32 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne MMP3 36 40 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne HLA-DRB1 62 38 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne PCSK5 56 39 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne FURIN 51 39 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne CCKBR 17 40 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne CTSH 26 40 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne CAPN2 58 37 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne ACE2 49 37 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne NPR 55 38 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne AMP1_PLAFQ 22 45 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne POLG_WNV 65 33 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne QRFPR 45 40 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne NPFFR1 55 35 CCCC[C@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278211 DF On-Demand Anodyne NOD1 74 33 COc1ccc(NC(=O)[C@@H]2CCC(=O)NC2)cc1O ZINC000147278241 CC For-Sale Anodyne STK17B 40 36 CCCNCc1ccc(Oc2ccc(Cl)c(F)c2)c(F)c1 ZINC000147278252 DJ For-Sale Anodyne LPAR2 24 44 CCCNCc1ccc(Oc2ccc(Cl)c(F)c2)c(F)c1 ZINC000147278252 DJ For-Sale Anodyne S1PR2 23 44 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278262 CF On-Demand Anodyne GHRHR 43 34 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278262 CF On-Demand Anodyne GRIN2B 29 41 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278262 CF On-Demand Anodyne SIGMAR1 22 45 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278262 CF On-Demand Anodyne PREP 64 48 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278262 CF On-Demand Anodyne FAAH 25 42 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278262 CF On-Demand Anodyne MGLL 0 42 CC[C@H]1CN(C(=O)CCCc2ccccc2)CC[C@H]1N ZINC000147278262 CF On-Demand Anodyne CYP2J2 40 37 CN(C)NC(=O)CC[C@H](CCN)C(C)(C)C ZINC000147278267 BD For-Sale Reactive KDM7A 0 43 N#Cc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147278279 CD On-Demand Mild CCR3 16 41 CCNc1cc(Oc2ccccc2[C@H](C)CC)nc(N)n1 ZINC000147278310 CH For-Sale Anodyne AO-ACHE 0 40 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne OPRM1 19 42 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne OPRD1 23 42 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne MME 36 41 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne KLK3 64 38 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne PAPA1_CARPA 45 38 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne CTSK 43 41 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne CTSL 25 40 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne NPFFR2 40 35 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne C3AR1 59 32 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne MMP3 36 40 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne HLA-DRB1 62 38 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne PCSK5 56 39 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne FURIN 51 39 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne CCKBR 17 40 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne CTSH 26 40 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne CAPN2 58 37 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne ACE2 49 37 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne NPR 55 38 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne AMP1_PLAFQ 22 45 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne POLG_WNV 65 33 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne QRFPR 45 40 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne NPFFR1 55 35 CCCC[C@@H](NC(N)=O)C(=O)N(Cc1ccccc1)C(C)C ZINC000147278347 DF On-Demand Anodyne NOD1 74 33 CCCCCCCCNc1nc(Cl)ccc1[N+](=O)[O-] ZINC000147278399 CI For-Sale Mild PRKCQ 0 43 COc1ccc(NC(=O)[C@H]2CCC(=O)NC2)cc1O ZINC000147278413 CC For-Sale Anodyne STK17B 40 36 CCNc1cc(Oc2ccccc2[C@@H](C)CC)nc(N)n1 ZINC000147278423 CH For-Sale Anodyne AO-ACHE 0 40 COc1cccc(CC(=O)N2CCC[C@H](CCBr)C2)c1 ZINC000147278446 EG For-Sale Reactive DRD4 40 31 COc1cccc(CC(=O)N2CCC[C@H](CCBr)C2)c1 ZINC000147278446 EG For-Sale Reactive SIGMAR1 15 53 COc1cccc(CC(=O)N2CCC[C@H](CCBr)C2)c1 ZINC000147278446 EG For-Sale Reactive CCR3 17 45 COc1ccc(Cl)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147278450 FI On-Demand Anodyne HTR1A 87 51 COc1ccc(Cl)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147278450 FI On-Demand Anodyne DRD2 76 51 COc1ccc(Cl)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147278450 FI On-Demand Anodyne DRD1 20 44 COc1ccc(Cl)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147278450 FI On-Demand Anodyne DRD4 51 51 COc1ccc(Cl)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147278450 FI On-Demand Anodyne ADRA1D 89 48 COc1ccc(Cl)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147278450 FI On-Demand Anodyne HTR2A 23 44 COc1ccc(Cl)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147278450 FI On-Demand Anodyne ADRA1A 74 48 COc1ccc(Cl)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147278450 FI On-Demand Anodyne ADRA1B 72 48 COc1ccc(Cl)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147278450 FI On-Demand Anodyne DRD3 68 51 COc1ccc(Cl)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147278450 FI On-Demand Anodyne HTR7 53 51 COc1ccc(Cl)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147278450 FI On-Demand Anodyne RBP4 15 43 O=C(O)C1(NCc2ccc(-c3ccccc3)cc2)CCC1 ZINC000147278470 CG For-Sale Anodyne MME 48 41 O=C(O)C1(NCc2ccc(-c3ccccc3)cc2)CCC1 ZINC000147278470 CG For-Sale Anodyne ECE1 36 43 O=C(O)C1(NCc2ccc(-c3ccccc3)cc2)CCC1 ZINC000147278470 CG For-Sale Anodyne NPPA 42 31 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278474 DD For-Sale Anodyne CCR3 0 49 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278474 DD For-Sale Anodyne SLC9A1 20 50 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278474 DD For-Sale Anodyne ST14 40 32 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278474 DD For-Sale Anodyne AKR1C3 40 35 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278474 DD For-Sale Anodyne L3MBTL1 0 43 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278474 DD For-Sale Anodyne L3MBTL3 41 40 CC(C)CCO[C@H](C)C(=O)N[C@@H](C)C(N)=O ZINC000147278479 BC On-Demand Anodyne WDR5 30 40 Cc1ccc(F)c(C(=O)CCN(C)C)c1F ZINC000147278511 BE For-Sale Anodyne THRA 49 43 Cc1ccc(F)c(C(=O)CCN(C)C)c1F ZINC000147278511 BE For-Sale Anodyne THRB 36 43 CC(C)CCO[C@@H](C)C(=O)N[C@H](C)C(N)=O ZINC000147278568 BC On-Demand Anodyne WDR5 30 40 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278572 DD For-Sale Anodyne CCR3 0 49 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278572 DD For-Sale Anodyne SLC9A1 20 50 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278572 DD For-Sale Anodyne ST14 40 32 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278572 DD For-Sale Anodyne AKR1C3 40 35 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278572 DD For-Sale Anodyne L3MBTL1 0 43 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@@H]1N ZINC000147278572 DD For-Sale Anodyne L3MBTL3 41 40 COc1cccc(CC(=O)N2CCC[C@@H](CCBr)C2)c1 ZINC000147278580 EG For-Sale Reactive DRD4 40 31 COc1cccc(CC(=O)N2CCC[C@@H](CCBr)C2)c1 ZINC000147278580 EG For-Sale Reactive SIGMAR1 15 53 COc1cccc(CC(=O)N2CCC[C@@H](CCBr)C2)c1 ZINC000147278580 EG For-Sale Reactive CCR3 17 45 CS(=O)(=O)c1ccc2c(c1)CCCO2 ZINC000147278602 BD For-Sale Anodyne PTGS2 15 44 CS(=O)(=O)c1ccc2c(c1)CCCO2 ZINC000147278602 BD For-Sale Anodyne PKM 25 43 CN(C)NC(=O)c1cn(CCN)nn1 ZINC000147278663 AA For-Sale Reactive THYX_PBCV1 49 30 CC(C)CCO[C@H](C)C(=O)N[C@H](C)C(N)=O ZINC000147278701 BC On-Demand Anodyne WDR5 30 40 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278705 DD For-Sale Anodyne CCR3 0 49 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278705 DD For-Sale Anodyne SLC9A1 20 50 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278705 DD For-Sale Anodyne ST14 40 32 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278705 DD For-Sale Anodyne AKR1C3 40 35 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278705 DD For-Sale Anodyne L3MBTL1 0 43 CC[C@@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278705 DD For-Sale Anodyne L3MBTL3 41 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000147278761 FF On-Demand Anodyne TMK 26 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000147278761 FF On-Demand Anodyne ENV 46 37 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000147278761 FF On-Demand Anodyne Q8MMZ8_EIMTE 40 42 COc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1Br ZINC000147278772 FD On-Demand Anodyne MMP7 15 41 CNC(=O)CCCOc1ccc(Cl)cc1S(N)(=O)=O ZINC000147278864 DC For-Sale Anodyne CPT1A 44 31 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278900 DD For-Sale Anodyne CCR3 0 49 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278900 DD For-Sale Anodyne SLC9A1 20 50 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278900 DD For-Sale Anodyne ST14 40 32 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278900 DD For-Sale Anodyne AKR1C3 40 35 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278900 DD For-Sale Anodyne L3MBTL1 0 43 CC[C@H]1CN(C(=O)c2cccc(S(C)(=O)=O)c2)CC[C@H]1N ZINC000147278900 DD For-Sale Anodyne L3MBTL3 41 40 CC(C)CCCCN[C@@H](C)c1cccc(C(F)(F)F)c1 ZINC000147278926 CK For-Sale Anodyne CASR 18 47 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000147278948 FF On-Demand Anodyne TMK 26 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000147278948 FF On-Demand Anodyne ENV 46 37 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(C(F)(F)F)c1 ZINC000147278948 FF On-Demand Anodyne Q8MMZ8_EIMTE 40 42 NS(=O)(=O)c1ccc(NC(=O)[C@@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279016 GC For-Sale Anodyne CA2 36 52 NS(=O)(=O)c1ccc(NC(=O)[C@@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279016 GC For-Sale Anodyne CA1 38 49 NS(=O)(=O)c1ccc(NC(=O)[C@@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279016 GC For-Sale Anodyne CA7 35 45 NS(=O)(=O)c1ccc(NC(=O)[C@@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279016 GC For-Sale Anodyne CA5B 31 45 NS(=O)(=O)c1ccc(NC(=O)[C@@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279016 GC For-Sale Anodyne CA4 44 52 NS(=O)(=O)c1ccc(NC(=O)[C@@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279016 GC For-Sale Anodyne CA5A 35 45 NS(=O)(=O)c1ccc(NC(=O)[C@@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279016 GC For-Sale Anodyne CA12 20 46 NS(=O)(=O)c1ccc(NC(=O)[C@@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279016 GC For-Sale Anodyne CA9 19 45 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OCCCC#N ZINC000147279027 HI On-Demand Mild HTR1A 71 39 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OCCCC#N ZINC000147279027 HI On-Demand Mild DRD2 64 48 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OCCCC#N ZINC000147279027 HI On-Demand Mild DRD1 33 47 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OCCCC#N ZINC000147279027 HI On-Demand Mild ADRA1D 58 38 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OCCCC#N ZINC000147279027 HI On-Demand Mild ADRA1A 50 37 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OCCCC#N ZINC000147279027 HI On-Demand Mild ADRA1B 51 38 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OCCCC#N ZINC000147279027 HI On-Demand Mild DRD3 63 43 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OCCCC#N ZINC000147279027 HI On-Demand Mild HTR7 47 39 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OCCCC#N ZINC000147279027 HI On-Demand Mild SSTR5 45 39 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OCCCC#N ZINC000147279027 HI On-Demand Mild EHMT2 71 35 CC(C)(C)NCc1ccccc1Oc1ccc(Cl)c(F)c1 ZINC000147279087 DK For-Sale Anodyne SLC6A4 16 58 CC(C)CCCCN[C@H](C)c1cccc(C(F)(F)F)c1 ZINC000147279123 CK For-Sale Anodyne CASR 18 47 COc1cc(CC(=O)O)cc(I)c1O ZINC000147279141 DD For-Sale Anodyne THRA 20 45 COc1cc(CC(=O)O)cc(I)c1O ZINC000147279141 DD For-Sale Anodyne THRB 20 45 COc1cc(CC(=O)O)cc(I)c1O ZINC000147279141 DD For-Sale Anodyne TRPV1 24 57 COc1cc(CC(=O)O)cc(I)c1O ZINC000147279141 DD For-Sale Anodyne SLCO1C1 0 45 CC(C)C1CCN(Cc2ccnc(N)c2)CC1 ZINC000147279171 BF On-Demand Anodyne SSTR5 47 38 NS(=O)(=O)c1ccc(NC(=O)[C@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279214 GC For-Sale Anodyne CA2 36 52 NS(=O)(=O)c1ccc(NC(=O)[C@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279214 GC For-Sale Anodyne CA1 38 49 NS(=O)(=O)c1ccc(NC(=O)[C@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279214 GC For-Sale Anodyne CA7 35 45 NS(=O)(=O)c1ccc(NC(=O)[C@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279214 GC For-Sale Anodyne CA5B 31 45 NS(=O)(=O)c1ccc(NC(=O)[C@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279214 GC For-Sale Anodyne CA4 44 52 NS(=O)(=O)c1ccc(NC(=O)[C@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279214 GC For-Sale Anodyne CA5A 35 45 NS(=O)(=O)c1ccc(NC(=O)[C@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279214 GC For-Sale Anodyne CA12 20 46 NS(=O)(=O)c1ccc(NC(=O)[C@H]2CCC(=O)NC2)c(Br)c1 ZINC000147279214 GC For-Sale Anodyne CA9 19 45 CCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147279258 DC For-Sale Anodyne CA2 33 40 CCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147279258 DC For-Sale Anodyne CA1 24 40 CCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147279258 DC For-Sale Anodyne CA4 27 40 O=C(CNC1(C(=O)O)CCC1)NCCc1cccs1 ZINC000147279280 CD For-Sale Anodyne ADAM17 0 42 O=C(CNC1(C(=O)O)CCC1)NCCc1cccs1 ZINC000147279280 CD For-Sale Anodyne CA5B 27 40 C=C(C)COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC ZINC000147279286 GI On-Demand Mild HTR1A 74 40 C=C(C)COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC ZINC000147279286 GI On-Demand Mild DRD2 63 45 C=C(C)COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC ZINC000147279286 GI On-Demand Mild DRD1 31 44 C=C(C)COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC ZINC000147279286 GI On-Demand Mild ADRA1D 64 38 C=C(C)COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC ZINC000147279286 GI On-Demand Mild ADRA1A 54 38 C=C(C)COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC ZINC000147279286 GI On-Demand Mild ADRA1B 51 38 C=C(C)COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC ZINC000147279286 GI On-Demand Mild DRD3 62 40 C=C(C)COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC ZINC000147279286 GI On-Demand Mild HTR7 45 37 C=C(C)COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC ZINC000147279286 GI On-Demand Mild SSTR5 50 39 CNC(=O)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1Cl ZINC000147279295 FF On-Demand Anodyne Q8MMZ8_EIMTE 15 40 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCc3ccccc3)nc12 ZINC000147279297 GG For-Sale Clean HTR1A 27 41 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCc3ccccc3)nc12 ZINC000147279297 GG For-Sale Clean DRD2 22 41 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCc3ccccc3)nc12 ZINC000147279297 GG For-Sale Clean ADRA1D 25 40 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCc3ccccc3)nc12 ZINC000147279297 GG For-Sale Clean ADRA1A 21 40 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCc3ccccc3)nc12 ZINC000147279297 GG For-Sale Clean ADORA2B 17 45 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCc3ccccc3)nc12 ZINC000147279297 GG For-Sale Clean CASR 31 47 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCc3ccccc3)nc12 ZINC000147279297 GG For-Sale Clean MTOR 40 39 CCCCCCCCNc1nc(Cl)nc2ccccc12 ZINC000147279362 CK For-Sale Mild ACHE 34 40 CCCCCCCCNc1nc(Cl)nc2ccccc12 ZINC000147279362 CK For-Sale Mild BCHE 41 40 CCCCCCCCNc1nc(Cl)nc2ccccc12 ZINC000147279362 CK For-Sale Mild UTS2R 16 46 CCCCCCCCNc1nc(Cl)nc2ccccc12 ZINC000147279362 CK For-Sale Mild METG 58 34 CCCCCCCCNc1nc(Cl)nc2ccccc12 ZINC000147279362 CK For-Sale Mild TLR7 25 49 CN(C)NC(=O)CC1(CN)CCC1 ZINC000147279375 AC For-Sale Reactive CACNA2D1 30 48 NS(=O)(=O)c1ccc(Cl)c(NC(=O)[C@@H]2CCC(=O)NC2)c1 ZINC000147279421 EC For-Sale Anodyne CA2 33 42 NS(=O)(=O)c1ccc(Cl)c(NC(=O)[C@@H]2CCC(=O)NC2)c1 ZINC000147279421 EC For-Sale Anodyne CA4 31 42 NS(=O)(=O)c1ccc(Cl)c(NC(=O)[C@@H]2CCC(=O)NC2)c1 ZINC000147279421 EC For-Sale Anodyne CA9 19 42 CCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147279435 DC For-Sale Anodyne CA2 33 40 CCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147279435 DC For-Sale Anodyne CA1 24 40 CCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147279435 DC For-Sale Anodyne CA4 27 40 CC(C)Oc1cccc(CC(=O)N[C@@H](C)C(N)=O)c1 ZINC000147279451 CD On-Demand Anodyne PRSS1 17 44 Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147279504 DD On-Demand Bother TBXA2R 32 41 CC(C)CN(Cc1ccc(N2CCC(O)CC2)cc1)S(=O)(=O)Cc1ccccc1 ZINC000147279517 HH Annotated Clean RORC 54 75 O=C(O)C1(NCc2ncc(-c3cccc(Cl)c3)o2)CCC1 ZINC000147279518 DG For-Sale Anodyne NPPA 37 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000147279547 ED On-Demand Bother ENV 42 34 CC[C@@H]1CN(C(=O)c2cc(C)ccc2F)CC[C@@H]1N ZINC000147279550 CE On-Demand Anodyne PARP1 50 38 CC[C@@H]1CN(C(=O)c2cc(C)ccc2F)CC[C@@H]1N ZINC000147279550 CE On-Demand Anodyne HCRTR2 29 41 O=C(c1cccc2cccnc12)N1CCC[C@H](CCBr)C1 ZINC000147279559 EH For-Sale Reactive HCRTR1 27 40 O=C(c1cccc2cccnc12)N1CCC[C@H](CCBr)C1 ZINC000147279559 EH For-Sale Reactive HCRTR2 24 40 Cc1nn(C)c2ncc(NC(=O)NCc3ccc(Oc4cccnc4)c(F)c3)cc12 ZINC000147279566 HH On-Demand Anodyne MET 51 41 Cc1nn(C)c2ncc(NC(=O)NCc3ccc(Oc4cccnc4)c(F)c3)cc12 ZINC000147279566 HH On-Demand Anodyne NAMPT 47 40 CN(C)NC(=O)c1csc(N)n1 ZINC000147279567 AB For-Sale Reactive SHV5 0 40 COC(=O)COc1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)c(C)c1 ZINC000147279580 GF On-Demand Anodyne ROCK2 40 50 NS(=O)(=O)c1ccc(Cl)c(NC(=O)[C@H]2CCC(=O)NC2)c1 ZINC000147279589 EC For-Sale Anodyne CA2 33 42 NS(=O)(=O)c1ccc(Cl)c(NC(=O)[C@H]2CCC(=O)NC2)c1 ZINC000147279589 EC For-Sale Anodyne CA4 31 42 NS(=O)(=O)c1ccc(Cl)c(NC(=O)[C@H]2CCC(=O)NC2)c1 ZINC000147279589 EC For-Sale Anodyne CA9 19 42 CC(C)(C)[C@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147279598 CE For-Sale Anodyne FFAR1 0 40 CC(C)(C)[C@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147279598 CE For-Sale Anodyne GPR88 0 48 Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147279644 DD On-Demand Bother TBXA2R 32 41 COc1ccc(C=O)cc1NC(N)=S ZINC000147279712 BD For-Sale Anodyne TUBB1 58 35 CC(=O)N1CCN(c2ccc(CN(CC#N)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147279724 IE Annotated Clean SLC12A5 41 33 CC(=O)N1CCN(c2ccc(CN(CC#N)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147279724 IE Annotated Clean RORC 31 57 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(Cl)c([N+](=O)[O-])c1 ZINC000147279726 ED On-Demand Bother ENV 42 34 O=C(O)C1(NCc2ccc(Br)cc2F)CCC1 ZINC000147279731 DF On-Demand Anodyne AKR1B1 22 41 O=C(c1cccc2cccnc12)N1CCC[C@@H](CCBr)C1 ZINC000147279732 EH For-Sale Reactive HCRTR1 27 40 O=C(c1cccc2cccnc12)N1CCC[C@@H](CCBr)C1 ZINC000147279732 EH For-Sale Reactive HCRTR2 24 40 CC[C@H]1CN(C(=O)c2cc(C)ccc2F)CC[C@@H]1N ZINC000147279736 CE On-Demand Anodyne PARP1 50 38 CC[C@H]1CN(C(=O)c2cc(C)ccc2F)CC[C@@H]1N ZINC000147279736 CE On-Demand Anodyne HCRTR2 29 41 CC(C)(C)[C@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147279745 CE For-Sale Anodyne FFAR1 0 40 CC(C)(C)[C@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147279745 CE For-Sale Anodyne GPR88 0 48 Cc1cc(F)c(S(=O)(=O)NCCCCC(C)C)cc1N ZINC000147279834 DF For-Sale Anodyne LEF 43 39 CCNc1ncc(Cl)c(Oc2ccccc2[C@H](C)CC)n1 ZINC000147279838 DJ For-Sale Anodyne AO-ACHE 0 40 CC[C@@H]1CN(C(=O)c2cc(C)ccc2F)CC[C@H]1N ZINC000147279893 CE On-Demand Anodyne PARP1 50 38 CC[C@@H]1CN(C(=O)c2cc(C)ccc2F)CC[C@H]1N ZINC000147279893 CE On-Demand Anodyne HCRTR2 29 41 COC(=O)/C=C(\O)C(=O)OC ZINC000147279894 AB In-Stock Anodyne HCAR2 15 44 COc1cccc(CC/C=C(/C)CCC=C(C)C)c1 ZINC000147279956 CK For-Sale Anodyne GGPS1 42 41 COc1cccc(CC/C=C(/C)CCC=C(C)C)c1 ZINC000147279956 CK For-Sale Anodyne FDFT1 26 50 COc1cccc(CC/C=C(/C)CCC=C(C)C)c1 ZINC000147279956 CK For-Sale Anodyne MTNR1A 24 46 COc1cccc(CC/C=C(/C)CCC=C(C)C)c1 ZINC000147279956 CK For-Sale Anodyne MTNR1B 26 46 COc1cccc(CC/C=C(/C)CCC=C(C)C)c1 ZINC000147279956 CK For-Sale Anodyne TRPA1 26 47 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive ACE 56 42 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive OPRM1 84 50 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive OPRD1 83 50 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive OPRK1 16 43 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive CACNA2D1 16 58 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive MME 156 61 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive LTA4H 26 46 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive ANPEP 112 43 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive TACR1 17 57 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive FCER2 71 35 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive RNPEP 45 43 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive CTSB 48 39 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive PAPA1_CARPA 56 38 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive CYSP_TRYCR 54 35 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive CTSK 19 41 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive CTSL 40 41 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive CPA1 69 40 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive SLC15A1 0 61 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive TPH1 75 38 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive CTRB1 35 48 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive CAPNS1 62 39 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive PDYN 0 40 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive MMP3 25 45 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive MMP8 21 42 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive PAM 0 43 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive YARS 81 47 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive SLC1A1 24 45 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive DNPEP 0 48 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive CAPN1 75 47 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive MMP9 21 41 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive CAPN2 56 36 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive ACE2 70 38 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive LAP3 71 44 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive CTSC 49 38 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive GNPAT 0 40 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive MMP1 28 42 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive FPR1 51 40 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive POL 0 45 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive NPR 66 38 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive AMP1_PLAFQ 84 44 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive SLC15A2 0 59 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive NPFFR1 45 32 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive BLAIMP-1 0 43 CN(C)NC(=O)[C@H](N)Cc1ccccc1 ZINC000147279973 BC For-Sale Reactive VM1B1_BOTAS 0 51 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147279974 ED On-Demand Anodyne PDE5A 15 44 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147279974 ED On-Demand Anodyne GRM4 15 42 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147279974 ED On-Demand Anodyne ENV 42 34 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147279974 ED On-Demand Anodyne QRFPR 43 38 O=C(Cc1csc(-c2ccc(Cl)cc2Cl)n1)OCCc1cnccn1 ZINC000147279981 GI On-Demand Anodyne DPP8 51 33 O=C(Cc1csc(-c2ccc(Cl)cc2Cl)n1)OCCc1cnccn1 ZINC000147279981 GI On-Demand Anodyne DPP9 40 33 CNCc1c(Cl)cccc1Oc1ccc(Cl)c(F)c1 ZINC000147279985 DJ For-Sale Anodyne SLC6A4 19 57 CCNc1ncc(Cl)c(Oc2ccccc2[C@@H](C)CC)n1 ZINC000147279996 DJ For-Sale Anodyne AO-ACHE 0 40 CC[C@H]1CN(C(=O)c2cc(C)ccc2F)CC[C@H]1N ZINC000147280028 CE On-Demand Anodyne PARP1 50 38 CC[C@H]1CN(C(=O)c2cc(C)ccc2F)CC[C@H]1N ZINC000147280028 CE On-Demand Anodyne HCRTR2 29 41 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147280142 ED On-Demand Anodyne PDE5A 15 44 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147280142 ED On-Demand Anodyne GRM4 15 42 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147280142 ED On-Demand Anodyne ENV 42 34 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147280142 ED On-Demand Anodyne QRFPR 43 38 CCCCCCCCNC(=O)c1ccc(/C(N)=N/O)cc1 ZINC000147280199 CF For-Sale Mild FOLH1 31 51 CCCCCCCCNC(=O)c1ccc(/C(N)=N/O)cc1 ZINC000147280199 CF For-Sale Mild KCNQ1 0 47 CCCCCCCCNC(=O)c1ccc(/C(N)=N/O)cc1 ZINC000147280199 CF For-Sale Mild S1PR2 42 37 CCCCCCCCNC(=O)c1ccc(/C(N)=N/O)cc1 ZINC000147280199 CF For-Sale Mild HDA106 0 43 CCCCCCCCNC(=O)c1ccc(/C(N)=N/O)cc1 ZINC000147280199 CF For-Sale Mild ASAH1 94 38 CCCCCCCCNC(=O)c1ccc(/C(N)=N/O)cc1 ZINC000147280199 CF For-Sale Mild ACAT 0 43 O=C(NCC(F)(F)F)Nc1cccc(-c2cnc3cc(-c4ccncc4)ccn23)c1 ZINC000147280269 HJ Annotated Anodyne BRAF 48 47 O=C(NCC(F)(F)F)Nc1cccc(-c2cnc3cc(-c4ccncc4)ccn23)c1 ZINC000147280269 HJ Annotated Anodyne RIPK1 44 31 COc1cccc(S(=O)(=O)N(Cc2ccc(N3CCN(C(C)=O)CC3)cc2F)C2CCC2)c1 ZINC000147280285 JG Annotated Clean AVPR1B 16 40 CNCCC(=O)NN(C)C ZINC000147280287 AB For-Sale Reactive PHF8 0 58 CNCCC(=O)NN(C)C ZINC000147280287 AB For-Sale Reactive KDM7A 0 58 CCOc1ccccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147280362 DD On-Demand Anodyne HCN1 42 33 CCOc1ccccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147280362 DD On-Demand Anodyne HCN4 43 34 CCNCc1cc(F)ccc1Oc1ccc(Cl)c(F)c1 ZINC000147280403 CJ For-Sale Anodyne SLC6A4 25 63 CCNCc1cc(F)ccc1Oc1ccc(Cl)c(F)c1 ZINC000147280403 CJ For-Sale Anodyne TSPO 40 33 COc1cc(OC)cc(C(=O)N2CCC[C@H](CCBr)C2)c1 ZINC000147280438 FG For-Sale Reactive GRM3 17 52 NCC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147280560 AD For-Sale Anodyne KDM1A 42 36 NCC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147280560 AD For-Sale Anodyne GPR88 0 45 CCOc1ccccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147280573 DD On-Demand Anodyne HCN1 42 33 CCOc1ccccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147280573 DD On-Demand Anodyne HCN4 43 34 CC[C@@H]1CN(C(=O)c2cncc(C)c2)CC[C@@H]1N ZINC000147280574 BD On-Demand Anodyne L3MBTL1 0 45 Fc1ccc(Oc2ccc(Cl)c(F)c2)c(CNC2CC2)c1 ZINC000147280599 DJ For-Sale Anodyne SLC6A4 24 58 COc1cc(OC)cc(C(=O)N2CCC[C@@H](CCBr)C2)c1 ZINC000147280617 FG For-Sale Reactive GRM3 17 52 CCCCCCCCNC(=O)C1(/C(N)=N/O)CC(C)C1 ZINC000147280637 CF For-Sale Mild EPHX2 40 41 COC(=O)N1CCN(c2ccc(CN(CC(C)C)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147280649 JH Annotated Clean RORC 50 63 CCC[C@H]1CC(=O)N(CCCCC(=O)O)C1 ZINC000147280651 BD For-Sale Anodyne PTGER3 17 42 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)N[C@H](C)C(N)=O ZINC000147280664 EE On-Demand Anodyne CHRM4 21 40 CN(C)NC(=O)CCNC1CC1 ZINC000147280703 AB For-Sale Reactive KDM7A 0 48 COc1ccccc1N1CCC(NCc2ccc(C#N)cc2)CC1 ZINC000147280716 DG On-Demand Mild DRD2 58 42 COc1ccccc1N1CCC(NCc2ccc(C#N)cc2)CC1 ZINC000147280716 DG On-Demand Mild DRD1 25 42 COc1ccccc1N1CCC(NCc2ccc(C#N)cc2)CC1 ZINC000147280716 DG On-Demand Mild ADRA1D 60 38 COc1ccccc1N1CCC(NCc2ccc(C#N)cc2)CC1 ZINC000147280716 DG On-Demand Mild HTR2A 27 42 COc1ccccc1N1CCC(NCc2ccc(C#N)cc2)CC1 ZINC000147280716 DG On-Demand Mild ADRA1A 45 39 COc1ccccc1N1CCC(NCc2ccc(C#N)cc2)CC1 ZINC000147280716 DG On-Demand Mild ADRA1B 53 38 COc1ccccc1N1CCC(NCc2ccc(C#N)cc2)CC1 ZINC000147280716 DG On-Demand Mild DRD3 44 42 COc1ccccc1N1CCC(NCc2ccc(C#N)cc2)CC1 ZINC000147280716 DG On-Demand Mild HTR7 42 38 CC[C@H]1CN(C(=O)c2cncc(C)c2)CC[C@@H]1N ZINC000147280798 BD On-Demand Anodyne L3MBTL1 0 45 CCCCCCCCNC(=O)[C@@H](C)/C(N)=N/O ZINC000147280822 BD For-Sale Mild DPP7 0 49 CCCCCCCCNC(=O)[C@@H](C)/C(N)=N/O ZINC000147280822 BD For-Sale Mild ASAH1 72 33 CCCCCCCCNC(=O)[C@@H](C)/C(N)=N/O ZINC000147280822 BD For-Sale Mild NOD1 77 42 CCCCCCCCNC(=O)[C@@H](C)/C(N)=N/O ZINC000147280822 BD For-Sale Mild CQSS 53 36 CCC[C@@H]1CC(=O)N(CCCCC(=O)O)C1 ZINC000147280824 BD For-Sale Anodyne PTGER3 17 42 CC(C)NCC(=O)NN(C)C ZINC000147280907 AB For-Sale Reactive KDM7A 0 45 COc1ccc(Cl)cc1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147280915 FH For-Sale Reactive DRD2 33 40 COc1ccc(Cl)cc1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147280915 FH For-Sale Reactive RBP4 27 45 COc1ccc(Cl)cc1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147280915 FH For-Sale Reactive ACKR3 43 30 CC(C)COc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147280963 GG On-Demand Bother TAAR1 38 46 CC(C)COc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147280963 GG On-Demand Bother KCNK3 71 35 CC(C)COc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147280963 GG On-Demand Bother KCNK9 56 32 CCC[C@@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147280995 ED For-Sale Anodyne CA2 32 41 CCC[C@@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147280995 ED For-Sale Anodyne CA1 23 41 CCC[C@@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147280995 ED For-Sale Anodyne CA4 28 41 CCC[C@@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147280995 ED For-Sale Anodyne PTGDR2 42 41 COc1ccc2c(c1)nc(S)n2CCNC(=O)N(C)C ZINC000147281008 CD For-Sale Anodyne MTNR1A 52 37 COc1ccc2c(c1)nc(S)n2CCNC(=O)N(C)C ZINC000147281008 CD For-Sale Anodyne MTNR1B 41 37 CC[C@@H]1CN(C(=O)c2cncc(C)c2)CC[C@H]1N ZINC000147281027 BD On-Demand Anodyne L3MBTL1 0 45 CCCCCCCCNC(=O)[C@H](C)/C(N)=N/O ZINC000147281029 BD For-Sale Mild DPP7 0 49 CCCCCCCCNC(=O)[C@H](C)/C(N)=N/O ZINC000147281029 BD For-Sale Mild ASAH1 72 33 CCCCCCCCNC(=O)[C@H](C)/C(N)=N/O ZINC000147281029 BD For-Sale Mild NOD1 77 42 CCCCCCCCNC(=O)[C@H](C)/C(N)=N/O ZINC000147281029 BD For-Sale Mild CQSS 53 36 FC(F)CNCc1ccc2ncccc2c1 ZINC000147281049 BF On-Demand Anodyne MET 0 41 CN(C)NC(=O)CNC(=O)CN ZINC000147281125 AA For-Sale Reactive UREB 0 56 CN(C)NC(=O)CNC(=O)CN ZINC000147281125 AA For-Sale Reactive KDM7A 0 43 COc1ccc(Cl)cc1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147281134 FH For-Sale Reactive DRD2 33 40 COc1ccc(Cl)cc1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147281134 FH For-Sale Reactive RBP4 27 45 COc1ccc(Cl)cc1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147281134 FH For-Sale Reactive ACKR3 43 30 CCNc1ncc(C)c(Oc2ccccc2[C@H](C)CC)n1 ZINC000147281154 CJ For-Sale Anodyne AO-ACHE 0 40 COCCNC(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147281181 HF On-Demand Bother TAAR1 26 47 COCCNC(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147281181 HF On-Demand Bother AKR1C2 44 38 COCCNC(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147281181 HF On-Demand Bother USP7 28 41 COCCNC(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147281181 HF On-Demand Bother USP47 35 41 CC[C@H]1CN(C(=O)CSCCOc2ccc(S(N)(=O)=O)cc2)CCO1 ZINC000147281196 GD On-Demand Anodyne CA2 23 43 CC[C@H]1CN(C(=O)CSCCOc2ccc(S(N)(=O)=O)cc2)CCO1 ZINC000147281196 GD On-Demand Anodyne CA1 16 43 CC[C@H]1CN(C(=O)CSCCOc2ccc(S(N)(=O)=O)cc2)CCO1 ZINC000147281196 GD On-Demand Anodyne CA7 23 42 CC[C@H]1CN(C(=O)CSCCOc2ccc(S(N)(=O)=O)cc2)CCO1 ZINC000147281196 GD On-Demand Anodyne CA12 28 42 CC[C@H]1CN(C(=O)CSCCOc2ccc(S(N)(=O)=O)cc2)CCO1 ZINC000147281196 GD On-Demand Anodyne CA9 19 42 CCC[C@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281212 ED For-Sale Anodyne CA2 32 41 CCC[C@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281212 ED For-Sale Anodyne CA1 23 41 CCC[C@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281212 ED For-Sale Anodyne CA4 28 41 CCC[C@H](C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281212 ED For-Sale Anodyne PTGDR2 42 41 CC[C@H]1CN(C(=O)c2cncc(C)c2)CC[C@H]1N ZINC000147281224 BD On-Demand Anodyne L3MBTL1 0 45 CCCCCCCCNC(=O)C(C)(C)/C(N)=N/O ZINC000147281247 CE For-Sale Mild ASAH1 72 33 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne ACE 31 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne OPRM1 0 44 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne OPRD1 43 44 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne MME 65 39 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne ANPEP 63 36 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne FCER2 51 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne CTSL 31 45 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne HLA-DRB1 72 37 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne CTSS 22 45 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne CAPN1 29 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne ACE2 73 39 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne PIN1 32 42 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne FPR1 37 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne LEF 32 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne BLA1_STEMA 41 32 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](C)C(N)=O ZINC000147281253 CC On-Demand Anodyne NPFFR1 49 34 CNCc1ccc(Oc2ccc(Cl)c(F)c2)cc1C ZINC000147281271 CI For-Sale Anodyne SLC6A4 18 61 O=C(O)c1ccc(CNCC(F)F)cc1 ZINC000147281282 BD On-Demand Anodyne SRD5A2 27 40 COc1ccccc1N1CCC(NCc2csc(Br)c2)CC1 ZINC000147281356 GI On-Demand Anodyne HTR1A 77 41 COc1ccccc1N1CCC(NCc2csc(Br)c2)CC1 ZINC000147281356 GI On-Demand Anodyne DRD2 65 44 COc1ccccc1N1CCC(NCc2csc(Br)c2)CC1 ZINC000147281356 GI On-Demand Anodyne DRD1 16 40 COc1ccccc1N1CCC(NCc2csc(Br)c2)CC1 ZINC000147281356 GI On-Demand Anodyne DRD4 36 44 COc1ccccc1N1CCC(NCc2csc(Br)c2)CC1 ZINC000147281356 GI On-Demand Anodyne ADRA1D 71 44 COc1ccccc1N1CCC(NCc2csc(Br)c2)CC1 ZINC000147281356 GI On-Demand Anodyne HTR2A 16 40 COc1ccccc1N1CCC(NCc2csc(Br)c2)CC1 ZINC000147281356 GI On-Demand Anodyne ADRA1A 60 40 COc1ccccc1N1CCC(NCc2csc(Br)c2)CC1 ZINC000147281356 GI On-Demand Anodyne ADRA1B 56 44 COc1ccccc1N1CCC(NCc2csc(Br)c2)CC1 ZINC000147281356 GI On-Demand Anodyne DRD3 64 44 COc1ccccc1N1CCC(NCc2csc(Br)c2)CC1 ZINC000147281356 GI On-Demand Anodyne HTR7 45 40 COC(=O)c1ccc(F)c(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)c1 ZINC000147281361 HG On-Demand Anodyne CHRM3 18 43 COC(=O)c1ccc(F)c(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)c1 ZINC000147281361 HG On-Demand Anodyne CCR3 28 41 COCCNC(=O)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1Cl ZINC000147281369 HG On-Demand Anodyne GRM4 39 41 CCNc1ncc(C)c(Oc2ccccc2[C@@H](C)CC)n1 ZINC000147281372 CJ For-Sale Anodyne AO-ACHE 0 40 CCCCCCCCNC(=O)[C@@H](CC)/C(N)=N/O ZINC000147281449 CE For-Sale Mild ASAH1 74 32 CCCCCCCCNC(=O)[C@@H](CC)/C(N)=N/O ZINC000147281449 CE For-Sale Mild NOD1 45 38 CCCCCCCCNC(=O)[C@@H](CC)/C(N)=N/O ZINC000147281449 CE For-Sale Mild CQSS 54 38 COCCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281463 EC For-Sale Anodyne CA2 25 40 COCCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281463 EC For-Sale Anodyne CA1 17 40 COCCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281463 EC For-Sale Anodyne COLA 73 34 COCCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281463 EC For-Sale Anodyne CPT1A 68 34 COCCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281463 EC For-Sale Anodyne CPT2 43 32 COCCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281463 EC For-Sale Anodyne CPT1B 66 33 COCCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281463 EC For-Sale Anodyne ALPL 16 40 CC[C@@H]1CN(C(=O)c2ccc(OC)c(F)c2)CC[C@@H]1N ZINC000147281467 CE On-Demand Anodyne L3MBTL3 50 34 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne ACE 31 40 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne OPRM1 0 44 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne OPRD1 43 44 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne MME 65 39 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne ANPEP 63 36 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne FCER2 51 40 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne CTSL 31 45 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne HLA-DRB1 72 37 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne CTSS 22 45 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne CAPN1 29 40 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne ACE2 73 39 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne PIN1 32 42 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne FPR1 37 40 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne LEF 32 40 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne BLA1_STEMA 41 32 C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)C(N)=O ZINC000147281472 CC On-Demand Anodyne NPFFR1 49 34 NCc1cccc(Oc2ccc(Cl)c(F)c2)c1 ZINC000147281502 CH For-Sale Anodyne CRTM 41 37 O=C(N[C@H]1CC=CCC1)c1nccc2ccccc12 ZINC000147281514 CG On-Demand Anodyne CASP1 24 49 COC(=O)c1ccc(F)c(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)c1 ZINC000147281564 HG On-Demand Anodyne CHRM3 18 43 COC(=O)c1ccc(F)c(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)c1 ZINC000147281564 HG On-Demand Anodyne CCR3 28 41 COc1ccccc1N1CCC(NCc2ccccc2OCc2cccnc2)CC1 ZINC000147281609 HI On-Demand Anodyne HTR1A 68 41 COc1ccccc1N1CCC(NCc2ccccc2OCc2cccnc2)CC1 ZINC000147281609 HI On-Demand Anodyne DRD2 50 45 COc1ccccc1N1CCC(NCc2ccccc2OCc2cccnc2)CC1 ZINC000147281609 HI On-Demand Anodyne DRD4 30 45 COc1ccccc1N1CCC(NCc2ccccc2OCc2cccnc2)CC1 ZINC000147281609 HI On-Demand Anodyne ADRA1D 53 38 COc1ccccc1N1CCC(NCc2ccccc2OCc2cccnc2)CC1 ZINC000147281609 HI On-Demand Anodyne ADRA1A 46 38 COc1ccccc1N1CCC(NCc2ccccc2OCc2cccnc2)CC1 ZINC000147281609 HI On-Demand Anodyne ADRA1B 41 38 COc1ccccc1N1CCC(NCc2ccccc2OCc2cccnc2)CC1 ZINC000147281609 HI On-Demand Anodyne DRD3 49 45 COc1ccccc1N1CCC(NCc2ccccc2OCc2cccnc2)CC1 ZINC000147281609 HI On-Demand Anodyne HTR7 44 43 CC(C)[C@@H](N)C(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147281616 EG On-Demand Anodyne PIK3CA 21 45 CCCNc1cncc(Oc2ccccc2[C@@H](C)CC)n1 ZINC000147281619 CJ For-Sale Anodyne AO-ACHE 0 40 CC(C)N(C(=O)COc1ccc(I)cc1)C(C)C ZINC000147281625 FG On-Demand Anodyne SRD5A2 15 63 CC(C)N(C(=O)COc1ccc(I)cc1)C(C)C ZINC000147281625 FG On-Demand Anodyne PLA2G4B 40 32 CC(C)N(C(=O)COc1ccc(I)cc1)C(C)C ZINC000147281625 FG On-Demand Anodyne TRAR 16 42 CCCCCCCCNC(=O)[C@H](CC)/C(N)=N/O ZINC000147281648 CE For-Sale Mild ASAH1 74 32 CCCCCCCCNC(=O)[C@H](CC)/C(N)=N/O ZINC000147281648 CE For-Sale Mild NOD1 45 38 CCCCCCCCNC(=O)[C@H](CC)/C(N)=N/O ZINC000147281648 CE For-Sale Mild CQSS 54 38 CCc1ncc(C(=O)N[C@@H](C)c2cccc(C(F)(F)F)c2)s1 ZINC000147281654 EI On-Demand Anodyne CCR2 26 40 CCc1ncc(C(=O)N[C@@H](C)c2cccc(C(F)(F)F)c2)s1 ZINC000147281654 EI On-Demand Anodyne PDS 47 35 CC[C@H]1CN(C(=O)c2ccc(OC)c(F)c2)CC[C@@H]1N ZINC000147281676 CE On-Demand Anodyne L3MBTL3 50 34 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne ACE 31 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne OPRM1 21 44 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne OPRD1 43 44 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne MME 65 39 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne ANPEP 63 36 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne FCER2 51 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne CTSL 31 45 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne HLA-DRB1 72 37 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne CTSS 22 45 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne CAPN1 29 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne ACE2 73 39 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne PIN1 32 42 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne FPR1 37 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne LEF 32 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne BLA1_STEMA 41 32 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](C)C(N)=O ZINC000147281677 CC On-Demand Anodyne NPFFR1 49 34 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCCC1 ZINC000147281695 HG On-Demand Anodyne KCNQ2 45 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCCC1 ZINC000147281695 HG On-Demand Anodyne TEK 21 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCCC1 ZINC000147281695 HG On-Demand Anodyne LIPG 50 35 COCCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281701 EC For-Sale Anodyne CA2 25 40 COCCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281701 EC For-Sale Anodyne CA1 17 40 COCCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281701 EC For-Sale Anodyne COLA 73 34 COCCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281701 EC For-Sale Anodyne CPT1A 68 34 COCCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281701 EC For-Sale Anodyne CPT2 43 32 COCCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281701 EC For-Sale Anodyne CPT1B 66 33 COCCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147281701 EC For-Sale Anodyne ALPL 16 40 O=C(N[C@@H]1CC=CCC1)c1nccc2ccccc12 ZINC000147281713 CG On-Demand Anodyne CASP1 24 49 Fc1cc(Oc2cccc(CNC3CC3)c2)ccc1Cl ZINC000147281737 CJ For-Sale Anodyne GRIN2B 0 40 CCCNc1cncc(Oc2ccccc2[C@H](C)CC)n1 ZINC000147281792 CJ For-Sale Anodyne AO-ACHE 0 40 COc1ccc(CC/C=C(/C)CCC=C(C)C)cc1 ZINC000147281810 CK For-Sale Anodyne GGPS1 44 39 COc1ccc(CC/C=C(/C)CCC=C(C)C)cc1 ZINC000147281810 CK For-Sale Anodyne FDFT1 24 48 COc1ccc(CC/C=C(/C)CCC=C(C)C)cc1 ZINC000147281810 CK For-Sale Anodyne TRPA1 30 61 CC(=O)NC1CCN(c2ccc(CN(CC(C)C)S(=O)(=O)Cc3ccccc3)cc2)CC1 ZINC000147281835 JH Annotated Clean RORC 52 59 CCCCCCCCNC(=O)[C@@](C)(CC)/C(N)=N/O ZINC000147281856 CF For-Sale Mild ASAH1 60 31 CCc1ncc(C(=O)N[C@H](C)c2cccc(C(F)(F)F)c2)s1 ZINC000147281883 EI On-Demand Anodyne CCR2 26 40 CCc1ncc(C(=O)N[C@H](C)c2cccc(C(F)(F)F)c2)s1 ZINC000147281883 EI On-Demand Anodyne PDS 47 35 CC[C@@H]1CN(C(=O)c2ccc(OC)c(F)c2)CC[C@H]1N ZINC000147281887 CE On-Demand Anodyne L3MBTL3 50 34 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCCC1 ZINC000147281904 HG On-Demand Anodyne KCNQ2 45 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCCC1 ZINC000147281904 HG On-Demand Anodyne TEK 21 43 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCCCC1 ZINC000147281904 HG On-Demand Anodyne LIPG 50 35 COc1cccc(-c2noc(CSc3nnc(NCCc4cccs4)s3)n2)c1 ZINC000147281926 IJ Annotated Anodyne WNT3A 20 42 COc1cccc(-c2noc(CSc3nnc(NCCc4cccs4)s3)n2)c1 ZINC000147281926 IJ Annotated Anodyne TNKS2 15 42 O=C(C#Cc1ccccc1)c1ccsc1 ZINC000147281929 BF For-Sale Mild LOX1.1 48 37 O=C(C#Cc1ccccc1)c1ccsc1 ZINC000147281929 BF For-Sale Mild O49150_SOLTU 53 37 C[C@H](Oc1ccc(Cl)cc1S(N)(=O)=O)C(=O)N1CCCC1 ZINC000147281932 ED For-Sale Anodyne COLA 41 37 C[C@H](Oc1ccc(Cl)cc1S(N)(=O)=O)C(=O)N1CCCC1 ZINC000147281932 ED For-Sale Anodyne CPT2 43 33 C[C@H](Oc1ccc(Cl)cc1S(N)(=O)=O)C(=O)N1CCCC1 ZINC000147281932 ED For-Sale Anodyne DPP7 42 38 CCCNCc1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147281952 EK For-Sale Anodyne LPAR2 24 44 CCCNCc1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147281952 EK For-Sale Anodyne S1PR2 24 44 Cn1cc(-c2noc(-c3cc(N)cc(Cl)c3)n2)cn1 ZINC000147282004 CE For-Sale Anodyne ALOX5AP 33 40 CN(C)NC(=O)[C@](C)(N)c1ccccc1 ZINC000147282006 BC For-Sale Reactive AMY2 55 36 CCCCCCCCNC(=O)[C@](C)(CC)/C(N)=N/O ZINC000147282033 CF For-Sale Mild ASAH1 60 31 CC(C)CCCCNCc1ccccc1Br ZINC000147282036 CI For-Sale Anodyne LEF 57 39 COc1cc([N+](=O)[O-])ccc1NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147282052 CD For-Sale Bother KCNMA1 23 51 CCc1ncc(C(=O)N2CCN(Cc3ccc(Cl)cc3)CC2)s1 ZINC000147282076 EG On-Demand Anodyne SIGMAR1 23 43 CCc1ncc(C(=O)N2CCN(Cc3ccc(Cl)cc3)CC2)s1 ZINC000147282076 EG On-Demand Anodyne LSS 21 50 CCc1ncc(C(=O)N2CCN(Cc3ccc(Cl)cc3)CC2)s1 ZINC000147282076 EG On-Demand Anodyne FAAH 24 44 CC[C@H]1CN(C(=O)c2ccc(OC)c(F)c2)CC[C@H]1N ZINC000147282085 CE On-Demand Anodyne L3MBTL3 50 34 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive ESR1 25 57 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive NR3C2 15 45 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive ESR2 19 57 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive ESRRA 15 57 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive SHBG 32 60 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive ESRRB 25 57 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive STS 121 51 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive HSD17B1 70 60 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive AOX1 27 57 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive HSD17B2 15 52 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive CYP2B6 15 55 C[C@]12CC[C@@H]3c4ccc(O)cc4CC[C@H]3[C@@H]1CC=C2C#N ZINC000147282103 CI For-Sale Reactive AKR1C3 28 53 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCOCC1 ZINC000147282107 HE On-Demand Anodyne TEK 16 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCOCC1 ZINC000147282107 HE On-Demand Anodyne LIPG 48 38 CCOC(=O)NCC(=O)N[C@@H](C)C(c1ccccc1)c1ccccc1 ZINC000147282109 EG On-Demand Anodyne CAPN2 69 36 CCOC(=O)NCC(=O)N[C@@H](C)C(c1ccccc1)c1ccccc1 ZINC000147282109 EG On-Demand Anodyne NPR 53 32 CCOC(=O)NCC(=O)N[C@@H](C)C(c1ccccc1)c1ccccc1 ZINC000147282109 EG On-Demand Anodyne ACER2 0 42 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1nnc2ccc(C(F)(F)F)cn12 ZINC000147282146 GG On-Demand Anodyne CARM1 51 35 C[C@@H](Oc1ccc(Cl)cc1S(N)(=O)=O)C(=O)N1CCCC1 ZINC000147282173 ED For-Sale Anodyne COLA 41 37 C[C@@H](Oc1ccc(Cl)cc1S(N)(=O)=O)C(=O)N1CCCC1 ZINC000147282173 ED For-Sale Anodyne CPT2 43 33 C[C@@H](Oc1ccc(Cl)cc1S(N)(=O)=O)C(=O)N1CCCC1 ZINC000147282173 ED For-Sale Anodyne DPP7 42 38 COc1cc([N+](=O)[O-])ccc1NC(=O)[C@H]1CCC(=O)NC1 ZINC000147282235 CD For-Sale Bother KCNMA1 23 51 CN(C)NC(=O)[C@@](C)(N)c1ccccc1 ZINC000147282237 BC For-Sale Reactive AMY2 55 36 CCCCCCCCNC(=O)C1(/C(N)=N/O)CCC1 ZINC000147282245 CE For-Sale Mild ASAH1 58 30 CCOC(=O)NCC(=O)N[C@H](C)C(c1ccccc1)c1ccccc1 ZINC000147282304 EG On-Demand Anodyne CAPN2 69 36 CCOC(=O)NCC(=O)N[C@H](C)C(c1ccccc1)c1ccccc1 ZINC000147282304 EG On-Demand Anodyne NPR 53 32 CCOC(=O)NCC(=O)N[C@H](C)C(c1ccccc1)c1ccccc1 ZINC000147282304 EG On-Demand Anodyne ACER2 0 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCOCC1 ZINC000147282310 HE On-Demand Anodyne TEK 16 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cc(C(F)(F)F)ccc1N1CCOCC1 ZINC000147282310 HE On-Demand Anodyne LIPG 48 38 COc1ccccc1N1CCC(NCc2cccc(OCc3ccccn3)c2)CC1 ZINC000147282349 HI On-Demand Anodyne HTR1A 75 48 COc1ccccc1N1CCC(NCc2cccc(OCc3ccccn3)c2)CC1 ZINC000147282349 HI On-Demand Anodyne DRD2 58 46 COc1ccccc1N1CCC(NCc2cccc(OCc3ccccn3)c2)CC1 ZINC000147282349 HI On-Demand Anodyne DRD4 36 40 COc1ccccc1N1CCC(NCc2cccc(OCc3ccccn3)c2)CC1 ZINC000147282349 HI On-Demand Anodyne ADRA1D 51 42 COc1ccccc1N1CCC(NCc2cccc(OCc3ccccn3)c2)CC1 ZINC000147282349 HI On-Demand Anodyne ADRA1A 46 42 COc1ccccc1N1CCC(NCc2cccc(OCc3ccccn3)c2)CC1 ZINC000147282349 HI On-Demand Anodyne ADRA1B 40 42 COc1ccccc1N1CCC(NCc2cccc(OCc3ccccn3)c2)CC1 ZINC000147282349 HI On-Demand Anodyne DRD3 55 46 COc1ccccc1N1CCC(NCc2cccc(OCc3ccccn3)c2)CC1 ZINC000147282349 HI On-Demand Anodyne HTR7 47 49 Cc1c([N+](=O)[O-])cccc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147282410 DD On-Demand Bother COLA 92 38 CCCCCCCCNC(=O)c1ccc(/C(N)=N/O)cn1 ZINC000147282433 CE For-Sale Mild FOLH1 16 40 CCCCCCCCNC(=O)c1ccc(/C(N)=N/O)cn1 ZINC000147282433 CE For-Sale Mild ASAH1 72 33 CNc1cccc(NCCc2ccccc2)n1 ZINC000147282439 BF For-Sale Anodyne PETD 0 42 CC[C@@H](C)c1ccccc1Oc1nc(NC)nc(OC)n1 ZINC000147282455 CG For-Sale Anodyne AO-ACHE 0 45 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccc(C(F)(F)F)cc3)c(F)c2)CC1 ZINC000147282476 KI Annotated Clean TRPV1 39 40 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccc(C(F)(F)F)cc3)c(F)c2)CC1 ZINC000147282476 KI Annotated Clean CACNA1B 40 35 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccc(C(F)(F)F)cc3)c(F)c2)CC1 ZINC000147282476 KI Annotated Clean SLC6A9 26 45 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccc(C(F)(F)F)cc3)c(F)c2)CC1 ZINC000147282476 KI Annotated Clean RORC 17 47 COC(=O)c1ccc(F)c(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000147282494 GF On-Demand Anodyne ADRB1 46 40 CN(C)CCCCNC(=O)c1cccc2c1OCCN2 ZINC000147282515 CD For-Sale Anodyne POLR1A 32 42 Cc1c([N+](=O)[O-])cccc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147282619 DD On-Demand Bother COLA 92 38 CC(C)(C)C(=O)C(=O)N1CCN(c2ccccc2)CC1 ZINC000147282622 CD On-Demand Anodyne HTR1A 16 41 CC(=O)NCc1ccc(-c2csc(NC(=O)[C@@H](C)Cc3cccc(F)c3)n2)o1 ZINC000147282643 HH On-Demand Anodyne ROCK1 19 46 CCOC(=O)c1ccc(Sc2ccc(CO)cc2)cc1 ZINC000147282681 CH For-Sale Anodyne GSTM2 18 46 CCOC(=O)c1ccc(Sc2ccc(CO)cc2)cc1 ZINC000147282681 CH For-Sale Anodyne F2RL3 18 40 CC[C@H](C)c1ccccc1Oc1nc(NC)nc(OC)n1 ZINC000147282694 CG For-Sale Anodyne AO-ACHE 0 45 COC(=O)c1ccc(F)c(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000147282714 GF On-Demand Anodyne ADRB1 46 40 COc1ccc2nc(S)n(CCNC(=O)N(C)C)c2n1 ZINC000147282765 CC For-Sale Anodyne PDE10A 31 41 CC(C)N(C)C(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147282822 DD For-Sale Anodyne PTGDR2 46 45 COc1ccccc1N1CCC(NCc2ccc(OCc3ccccn3)cc2)CC1 ZINC000147282833 HI On-Demand Anodyne HTR1A 74 44 COc1ccccc1N1CCC(NCc2ccc(OCc3ccccn3)cc2)CC1 ZINC000147282833 HI On-Demand Anodyne DRD2 57 44 COc1ccccc1N1CCC(NCc2ccc(OCc3ccccn3)cc2)CC1 ZINC000147282833 HI On-Demand Anodyne DRD4 35 41 COc1ccccc1N1CCC(NCc2ccc(OCc3ccccn3)cc2)CC1 ZINC000147282833 HI On-Demand Anodyne ADRA1D 52 38 COc1ccccc1N1CCC(NCc2ccc(OCc3ccccn3)cc2)CC1 ZINC000147282833 HI On-Demand Anodyne ADRA1A 48 42 COc1ccccc1N1CCC(NCc2ccc(OCc3ccccn3)cc2)CC1 ZINC000147282833 HI On-Demand Anodyne ADRA1B 41 38 COc1ccccc1N1CCC(NCc2ccc(OCc3ccccn3)cc2)CC1 ZINC000147282833 HI On-Demand Anodyne DRD3 57 44 COc1ccccc1N1CCC(NCc2ccc(OCc3ccccn3)cc2)CC1 ZINC000147282833 HI On-Demand Anodyne HTR7 49 40 CC(=O)NCc1ccc(-c2csc(NC(=O)[C@H](C)Cc3cccc(F)c3)n2)o1 ZINC000147282877 HH On-Demand Anodyne ROCK1 19 46 CCCCCCCCNC(=O)[C@@H](CCC)/C(N)=N/O ZINC000147282905 CF For-Sale Mild S1PR2 17 41 CCCCCCCCNC(=O)[C@@H](CCC)/C(N)=N/O ZINC000147282905 CF For-Sale Mild ASAH1 70 31 CCCCCCCCNC(=O)[C@@H](CCC)/C(N)=N/O ZINC000147282905 CF For-Sale Mild NOD1 59 40 CCCCCCCCNC(=O)[C@@H](CCC)/C(N)=N/O ZINC000147282905 CF For-Sale Mild CQSS 52 34 CC[C@@H](c1ncccn1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147282933 KK Annotated Anodyne TP53 47 73 CC[C@@H](c1ncccn1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147282933 KK Annotated Anodyne MDM2 264 73 CCCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147283031 DD For-Sale Anodyne PTGDR2 32 42 CCCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147283031 DD For-Sale Anodyne PSBA 0 41 CCCNc1cccc(NCCc2ccccc2)n1 ZINC000147283045 CH For-Sale Anodyne PETD 0 42 CCCCCCCCNC(=O)[C@H](CCC)/C(N)=N/O ZINC000147283122 CF For-Sale Mild S1PR2 17 41 CCCCCCCCNC(=O)[C@H](CCC)/C(N)=N/O ZINC000147283122 CF For-Sale Mild ASAH1 70 31 CCCCCCCCNC(=O)[C@H](CCC)/C(N)=N/O ZINC000147283122 CF For-Sale Mild NOD1 59 40 CCCCCCCCNC(=O)[C@H](CCC)/C(N)=N/O ZINC000147283122 CF For-Sale Mild CQSS 52 34 CCn1c2ccccc2c2cc(CNCC(F)F)ccc21 ZINC000147283126 CI For-Sale Anodyne MCHR2 44 40 CCCNCc1cc(F)ccc1Oc1ccc(Cl)c(F)c1 ZINC000147283130 DJ For-Sale Anodyne SLC6A4 21 60 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283133 DF On-Demand Anodyne NPY2R 22 42 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283133 DF On-Demand Anodyne CACNA1B 60 40 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283133 DF On-Demand Anodyne SLC9A1 45 41 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283133 DF On-Demand Anodyne CCR2 68 43 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283133 DF On-Demand Anodyne LIPG 43 34 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283133 DF On-Demand Anodyne RHOA 0 45 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283133 DF On-Demand Anodyne L3MBTL1 0 43 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283133 DF On-Demand Anodyne L3MBTL3 34 40 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283133 DF On-Demand Anodyne MAP3K12 28 40 CCCCCC[C@@H](C)NCCCCC(C)C ZINC000147283151 BJ For-Sale Anodyne ADH1A 0 47 CCCCCC[C@@H](C)NCCCCC(C)C ZINC000147283151 BJ For-Sale Anodyne ADH1B 0 47 CCCCCC[C@@H](C)NCCCCC(C)C ZINC000147283151 BJ For-Sale Anodyne ADH1C 0 47 CCCCCC[C@@H](C)NCCCCC(C)C ZINC000147283151 BJ For-Sale Anodyne FPPS 0 44 COC(=O)c1ccc(F)c(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c1 ZINC000147283156 EG On-Demand Anodyne EPHX2 26 41 CCCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147283240 DD For-Sale Anodyne PTGDR2 32 42 CCCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147283240 DD For-Sale Anodyne PSBA 0 41 NC(=O)c1ccc(OCC(=O)Nc2ccccc2OC2CCCC2)cc1 ZINC000147283252 FG On-Demand Anodyne CPT1A 20 42 NC(=O)c1ccc(OCC(=O)Nc2ccccc2OC2CCCC2)cc1 ZINC000147283252 FG On-Demand Anodyne HIF1A 22 41 Cc1cc(Cl)ccc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147283273 DE On-Demand Anodyne OXER1 42 36 N#C[C@H](N)C(=O)c1ccccc1 ZINC000147283287 AC For-Sale Mild PLAUR 16 48 CCCCCCCCNC(=O)[C@H](/C(N)=N/O)C(C)C ZINC000147283296 CE For-Sale Mild ASAH1 70 32 CCCCCCCCNC(=O)[C@H](/C(N)=N/O)C(C)C ZINC000147283296 CE For-Sale Mild NOD1 59 40 CCCCCCCCNC(=O)[C@H](/C(N)=N/O)C(C)C ZINC000147283296 CE For-Sale Mild CQSS 41 34 COc1ccccc1N1CCC(NCc2ccccc2Br)CC1 ZINC000147283323 GI On-Demand Anodyne HTR1A 86 46 COc1ccccc1N1CCC(NCc2ccccc2Br)CC1 ZINC000147283323 GI On-Demand Anodyne DRD2 70 46 COc1ccccc1N1CCC(NCc2ccccc2Br)CC1 ZINC000147283323 GI On-Demand Anodyne DRD1 15 43 COc1ccccc1N1CCC(NCc2ccccc2Br)CC1 ZINC000147283323 GI On-Demand Anodyne DRD4 39 43 COc1ccccc1N1CCC(NCc2ccccc2Br)CC1 ZINC000147283323 GI On-Demand Anodyne ADRA1D 78 43 COc1ccccc1N1CCC(NCc2ccccc2Br)CC1 ZINC000147283323 GI On-Demand Anodyne HTR2A 19 43 COc1ccccc1N1CCC(NCc2ccccc2Br)CC1 ZINC000147283323 GI On-Demand Anodyne ADRA1A 66 41 COc1ccccc1N1CCC(NCc2ccccc2Br)CC1 ZINC000147283323 GI On-Demand Anodyne ADRA1B 62 43 COc1ccccc1N1CCC(NCc2ccccc2Br)CC1 ZINC000147283323 GI On-Demand Anodyne DRD3 67 46 COc1ccccc1N1CCC(NCc2ccccc2Br)CC1 ZINC000147283323 GI On-Demand Anodyne TACR1 15 42 COc1ccccc1N1CCC(NCc2ccccc2Br)CC1 ZINC000147283323 GI On-Demand Anodyne HTR7 52 45 CN(C)NC(=O)CNCC(F)(F)F ZINC000147283324 AB For-Sale Reactive KDM7A 0 45 COC(=O)c1ccc(F)c(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147283349 EG On-Demand Anodyne EPHX2 26 41 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283350 DF On-Demand Anodyne NPY2R 22 42 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283350 DF On-Demand Anodyne CACNA1B 60 40 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283350 DF On-Demand Anodyne SLC9A1 45 41 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283350 DF On-Demand Anodyne CCR2 68 43 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283350 DF On-Demand Anodyne LIPG 43 34 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283350 DF On-Demand Anodyne RHOA 0 45 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283350 DF On-Demand Anodyne L3MBTL1 0 43 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283350 DF On-Demand Anodyne L3MBTL3 34 40 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@@H]1N ZINC000147283350 DF On-Demand Anodyne MAP3K12 28 40 CCCCCC[C@H](C)NCCCCC(C)C ZINC000147283361 BJ For-Sale Anodyne ADH1A 0 47 CCCCCC[C@H](C)NCCCCC(C)C ZINC000147283361 BJ For-Sale Anodyne ADH1B 0 47 CCCCCC[C@H](C)NCCCCC(C)C ZINC000147283361 BJ For-Sale Anodyne ADH1C 0 47 CCCCCC[C@H](C)NCCCCC(C)C ZINC000147283361 BJ For-Sale Anodyne FPPS 0 44 CC[C@@H](C)c1ccccc1Oc1cc(N)ncn1 ZINC000147283364 BG For-Sale Anodyne AO-ACHE 0 41 CN(Cc1cscn1)C(=O)NCc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147283411 HF On-Demand Anodyne NAMPT 72 51 Cc1cc(Cl)ccc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147283499 DE On-Demand Anodyne OXER1 42 36 CC(C)c1ccc(O)c(S(=O)(=O)O)c1 ZINC000147283502 BD For-Sale Anodyne PPO2 17 47 COc1ccc2nc(S)n(CCNC(=O)N(C)C)c2c1 ZINC000147283509 CD For-Sale Anodyne DRD4 41 31 COc1ccc2nc(S)n(CCNC(=O)N(C)C)c2c1 ZINC000147283509 CD For-Sale Anodyne MTNR1A 50 37 COc1ccc2nc(S)n(CCNC(=O)N(C)C)c2c1 ZINC000147283509 CD For-Sale Anodyne SCD 17 40 CCCCCCCCNC(=O)[C@@H](/C(N)=N/O)C(C)C ZINC000147283513 CE For-Sale Mild ASAH1 70 32 CCCCCCCCNC(=O)[C@@H](/C(N)=N/O)C(C)C ZINC000147283513 CE For-Sale Mild NOD1 59 40 CCCCCCCCNC(=O)[C@@H](/C(N)=N/O)C(C)C ZINC000147283513 CE For-Sale Mild CQSS 41 34 N#C[C@@H](N)C(=O)c1ccccc1 ZINC000147283516 AC For-Sale Mild PLAUR 16 48 COC(=O)c1ccc(F)c(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000147283553 EG On-Demand Anodyne EPHX2 26 41 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283564 DF On-Demand Anodyne NPY2R 22 42 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283564 DF On-Demand Anodyne CACNA1B 60 40 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283564 DF On-Demand Anodyne SLC9A1 45 41 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283564 DF On-Demand Anodyne CCR2 68 43 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283564 DF On-Demand Anodyne LIPG 43 34 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283564 DF On-Demand Anodyne RHOA 0 45 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283564 DF On-Demand Anodyne L3MBTL1 0 43 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283564 DF On-Demand Anodyne L3MBTL3 34 40 CC[C@@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283564 DF On-Demand Anodyne MAP3K12 28 40 CN(C)NC(=O)CCOC1CCNCC1 ZINC000147283575 BB For-Sale Reactive KDM7A 0 41 CCOC(=O)[C@H](C#N)Cc1ccc(F)cc1Cl ZINC000147283599 CF For-Sale Mild P2RX7 60 42 CC[C@H](C)c1ccccc1Oc1cc(N)ncn1 ZINC000147283617 BG For-Sale Anodyne AO-ACHE 0 41 CCN(C(=O)COc1ccc(Cl)cc1S(N)(=O)=O)C1CC1 ZINC000147283639 ED For-Sale Anodyne PTGDR2 40 39 CN(CC(=O)Nc1cccc(Cl)c1)C(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147283641 HG On-Demand Anodyne CACNA1H 15 43 CN(CC(=O)Nc1cccc(Cl)c1)C(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147283641 HG On-Demand Anodyne DRTS_PLAFK 23 48 CN(CC(=O)Nc1cccc(Cl)c1)C(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147283641 HG On-Demand Anodyne PTGER3 35 51 O=C(O)COc1ccc([C@@H]2[C@@H](CCSc3ccc(F)cc3)C(=O)N2c2ccc(F)cc2)cc1 ZINC000147283657 JK For-Sale Anodyne NPC1L1 23 49 CC(C)COC1CCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147283658 EI On-Demand Anodyne MC4R 47 39 CC(C)COC1CCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147283658 EI On-Demand Anodyne EPHX2 15 44 CC(C)COC1CCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147283658 EI On-Demand Anodyne MDM2 116 34 CC(C)COC1CCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147283658 EI On-Demand Anodyne GPR88 0 42 CCCCCCCCNC(=O)C1(/C(N)=N/O)CC1 ZINC000147283677 CD For-Sale Mild ASAH1 70 31 CCCc1ccc(S(=O)(=O)N(CCBr)C2CCCC2)cc1 ZINC000147283719 FH For-Sale Reactive AVPR1B 24 42 COC(=O)c1ccc(F)c(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c1 ZINC000147283768 EG On-Demand Anodyne EPHX2 26 41 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283780 DF On-Demand Anodyne NPY2R 22 42 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283780 DF On-Demand Anodyne CACNA1B 60 40 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283780 DF On-Demand Anodyne SLC9A1 45 41 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283780 DF On-Demand Anodyne CCR2 68 43 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283780 DF On-Demand Anodyne LIPG 43 34 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283780 DF On-Demand Anodyne RHOA 0 45 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283780 DF On-Demand Anodyne L3MBTL1 0 43 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283780 DF On-Demand Anodyne L3MBTL3 34 40 CC[C@H]1CN(C(=O)c2cccc(C(F)(F)F)c2)CC[C@H]1N ZINC000147283780 DF On-Demand Anodyne MAP3K12 28 40 CCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OCc2ccncc2)c(OC)c1 ZINC000147283783 HF On-Demand Anodyne CTSB 30 44 CCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OCc2ccncc2)c(OC)c1 ZINC000147283783 HF On-Demand Anodyne CAPN1 45 44 CCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OCc2ccncc2)c(OC)c1 ZINC000147283783 HF On-Demand Anodyne CAPN2 89 44 CCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OCc2ccncc2)c(OC)c1 ZINC000147283783 HF On-Demand Anodyne ENPP1 44 30 CCOC(=O)[C@@H](C#N)Cc1ccc(F)cc1Cl ZINC000147283796 CF For-Sale Mild P2RX7 60 42 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne CA2 88 58 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne CA1 67 48 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne CA7 36 45 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne CA5B 58 34 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne CA4 82 58 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne CA5A 62 34 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne CA14 24 45 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne CCR2 27 40 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne CA12 29 45 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne CA9 45 42 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne CYNT 20 50 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne KCNK3 79 43 CCOc1ccc(C(=O)NCC(=O)Nc2cccc(S(N)(=O)=O)c2)cc1OCC ZINC000147283811 HD On-Demand Anodyne KCNK9 70 43 CCOC(=O)NCC(=O)N(C)CC(=O)Nc1cccc(Cl)c1 ZINC000147283817 ED On-Demand Anodyne CACNA1H 15 45 CC(C)COC1CCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147283826 EI On-Demand Anodyne MC4R 47 39 CC(C)COC1CCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147283826 EI On-Demand Anodyne EPHX2 15 44 CC(C)COC1CCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147283826 EI On-Demand Anodyne MDM2 116 34 CC(C)COC1CCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CC1 ZINC000147283826 EI On-Demand Anodyne GPR88 0 42 CC[C@H](CCN)CCC(=O)NN(C)C ZINC000147283827 BC For-Sale Reactive KDM7A 0 44 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@H](C)C2 ZINC000147283859 GH On-Demand Anodyne HTR1A 66 44 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@H](C)C2 ZINC000147283859 GH On-Demand Anodyne DRD2 52 44 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@H](C)C2 ZINC000147283859 GH On-Demand Anodyne DRD4 29 44 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@H](C)C2 ZINC000147283859 GH On-Demand Anodyne ADRA1D 58 39 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@H](C)C2 ZINC000147283859 GH On-Demand Anodyne ADRA1A 50 39 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@H](C)C2 ZINC000147283859 GH On-Demand Anodyne ADRA1B 47 37 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@H](C)C2 ZINC000147283859 GH On-Demand Anodyne DRD3 49 44 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@H](C)C2 ZINC000147283859 GH On-Demand Anodyne HTR7 46 44 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@H](C)C2 ZINC000147283859 GH On-Demand Anodyne NPY1R 18 40 O=C(O)COc1ccc([C@H]2[C@@H](CCSc3ccc(F)cc3)C(=O)N2c2ccc(F)cc2)cc1 ZINC000147283868 JK For-Sale Anodyne NPC1L1 23 49 COC(=O)c1ccc(Cn2c(C(=O)O)cc3ccccc32)cc1 ZINC000147283883 DG For-Sale Anodyne FABI 61 46 COC(=O)c1ccc(Cn2c(C(=O)O)cc3ccccc32)cc1 ZINC000147283883 DG For-Sale Anodyne AGTR1 68 38 COC(=O)c1ccc(Cn2c(C(=O)O)cc3ccccc32)cc1 ZINC000147283883 DG For-Sale Anodyne F10 17 53 COC(=O)c1ccc(Cn2c(C(=O)O)cc3ccccc32)cc1 ZINC000147283883 DG For-Sale Anodyne PLA2G2A 81 37 COC(=O)c1ccc(Cn2c(C(=O)O)cc3ccccc32)cc1 ZINC000147283883 DG For-Sale Anodyne CCR2 17 65 COC(=O)c1ccc(Cn2c(C(=O)O)cc3ccccc32)cc1 ZINC000147283883 DG For-Sale Anodyne MAPK8 25 46 COC(=O)c1ccc(Cn2c(C(=O)O)cc3ccccc32)cc1 ZINC000147283883 DG For-Sale Anodyne PLA2G2F 52 32 COC(=O)c1ccc(Cn2c(C(=O)O)cc3ccccc32)cc1 ZINC000147283883 DG For-Sale Anodyne PLA2G2D 54 35 COC(=O)c1ccc(Cn2c(C(=O)O)cc3ccccc32)cc1 ZINC000147283883 DG For-Sale Anodyne PTGDR2 17 42 COC(=O)c1ccc(Cn2c(C(=O)O)cc3ccccc32)cc1 ZINC000147283883 DG For-Sale Anodyne NPFFR1 21 42 C[C@H](NC(=O)N(C)Cc1cscn1)c1nc2ccccc2[nH]1 ZINC000147283889 DF On-Demand Anodyne BMP1 50 33 C[C@H](NC(=O)N(C)Cc1cscn1)c1nc2ccccc2[nH]1 ZINC000147283889 DF On-Demand Anodyne CYP3A4 18 41 CCCCCCCCNC(=O)c1cccc(/C(N)=N/O)c1 ZINC000147283896 CF For-Sale Mild DRD4 40 31 CCCCCCCCNC(=O)c1cccc(/C(N)=N/O)c1 ZINC000147283896 CF For-Sale Mild FOLH1 21 42 CCCCCCCCNC(=O)c1cccc(/C(N)=N/O)c1 ZINC000147283896 CF For-Sale Mild FAAH 15 43 CCCCCCCCNC(=O)c1cccc(/C(N)=N/O)c1 ZINC000147283896 CF For-Sale Mild EPHX2 0 41 CCCCCCCCNC(=O)c1cccc(/C(N)=N/O)c1 ZINC000147283896 CF For-Sale Mild PA2A1_NAJMO 0 41 CCCCCCCCNC(=O)c1cccc(/C(N)=N/O)c1 ZINC000147283896 CF For-Sale Mild ASAH1 89 35 CCCCCCCCNC(=O)c1cccc(/C(N)=N/O)c1 ZINC000147283896 CF For-Sale Mild ACAT 0 45 O=C(O)C1(NC[C@H]2Cc3ccccc3O2)CCC1 ZINC000147283902 BD For-Sale Anodyne HTR1D 0 42 COC(=O)c1ccc(F)c(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147284003 FD On-Demand Anodyne EPHX2 38 42 CC[C@@H](CCN)CCC(=O)NN(C)C ZINC000147284005 BC For-Sale Reactive KDM7A 0 44 CCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OCc2ccncc2)c(OC)c1 ZINC000147284018 HF On-Demand Anodyne CTSB 30 44 CCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OCc2ccncc2)c(OC)c1 ZINC000147284018 HF On-Demand Anodyne CAPN1 45 44 CCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OCc2ccncc2)c(OC)c1 ZINC000147284018 HF On-Demand Anodyne CAPN2 89 44 CCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OCc2ccncc2)c(OC)c1 ZINC000147284018 HF On-Demand Anodyne ENPP1 44 30 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@@H](C)C2 ZINC000147284033 GH On-Demand Anodyne HTR1A 66 44 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@@H](C)C2 ZINC000147284033 GH On-Demand Anodyne DRD2 52 44 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@@H](C)C2 ZINC000147284033 GH On-Demand Anodyne DRD4 29 44 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@@H](C)C2 ZINC000147284033 GH On-Demand Anodyne ADRA1D 58 39 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@@H](C)C2 ZINC000147284033 GH On-Demand Anodyne ADRA1A 50 39 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@@H](C)C2 ZINC000147284033 GH On-Demand Anodyne ADRA1B 47 37 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@@H](C)C2 ZINC000147284033 GH On-Demand Anodyne DRD3 49 44 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@@H](C)C2 ZINC000147284033 GH On-Demand Anodyne HTR7 46 44 COc1cc2c(cc1CNC1CCN(c3ccccc3OC)CC1)O[C@@H](C)C2 ZINC000147284033 GH On-Demand Anodyne NPY1R 18 40 CC(C)COC1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147284040 EI On-Demand Anodyne MC4R 47 39 CC(C)COC1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147284040 EI On-Demand Anodyne EPHX2 15 44 CC(C)COC1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147284040 EI On-Demand Anodyne MDM2 116 34 CC(C)COC1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147284040 EI On-Demand Anodyne GPR88 0 42 O=C(O)C1(NC[C@@H]2Cc3ccccc3O2)CCC1 ZINC000147284058 BD For-Sale Anodyne HTR1D 0 42 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284069 CD On-Demand Anodyne OPRK1 0 45 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284069 CD On-Demand Anodyne MMP13 49 42 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284069 CD On-Demand Anodyne MLNR 21 40 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284069 CD On-Demand Anodyne MMP3 49 42 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284069 CD On-Demand Anodyne MMP8 34 41 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284069 CD On-Demand Anodyne MMP9 51 42 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284069 CD On-Demand Anodyne MMP7 45 42 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284069 CD On-Demand Anodyne MMP1 52 46 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284069 CD On-Demand Anodyne GPR183 0 45 CC(C)=CCC/C(C)=C\CCc1ccccc1 ZINC000147284075 BK For-Sale Anodyne GGPS1 51 42 CC(C)=CCC/C(C)=C\CCc1ccccc1 ZINC000147284075 BK For-Sale Anodyne FDFT1 29 69 CC(C)=CCC/C(C)=C\CCc1ccccc1 ZINC000147284075 BK For-Sale Anodyne TRPA1 31 63 O=C(O)COc1ccc([C@@H]2[C@H](CCSc3ccc(F)cc3)C(=O)N2c2ccc(F)cc2)cc1 ZINC000147284089 JK For-Sale Anodyne NPC1L1 23 49 CCCCCCCCNC(=O)C(CC)(CC)/C(N)=N/O ZINC000147284099 CG For-Sale Mild ASAH1 68 32 C[C@@H](NC(=O)N(C)Cc1cscn1)c1nc2ccccc2[nH]1 ZINC000147284108 DF On-Demand Anodyne BMP1 50 33 C[C@@H](NC(=O)N(C)Cc1cscn1)c1nc2ccccc2[nH]1 ZINC000147284108 DF On-Demand Anodyne CYP3A4 18 41 NS(=O)(=O)c1cc(Cl)ccc1OCc1ncccn1 ZINC000147284121 CD For-Sale Anodyne PTGER1 52 39 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3ccccc3F)c(F)c2)CC1 ZINC000147284133 JG Annotated Clean SSTR1 35 40 BrC1C[C@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147284170 CH For-Sale Reactive SLC6A3 18 51 BrC1C[C@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147284170 CH For-Sale Reactive SLC18A2 41 35 BrC1C[C@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147284170 CH For-Sale Reactive KCNH2 25 45 BrC1C[C@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147284170 CH For-Sale Reactive LTA4H 15 46 BrC1C[C@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147284170 CH For-Sale Reactive SIGMAR1 34 59 BrC1C[C@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147284170 CH For-Sale Reactive ACHP_LYMST 24 51 BrC1C[C@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147284170 CH For-Sale Reactive ARG1 31 43 BrC1C[C@H]2CC[C@H](C1)N2Cc1ccccc1 ZINC000147284170 CH For-Sale Reactive ARG2 31 43 COC(=O)c1ccc(F)c(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147284213 FD On-Demand Anodyne EPHX2 38 42 CC(C)COC1CCN(C(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147284236 EI On-Demand Anodyne MC4R 47 39 CC(C)COC1CCN(C(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147284236 EI On-Demand Anodyne EPHX2 15 44 CC(C)COC1CCN(C(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147284236 EI On-Demand Anodyne MDM2 116 34 CC(C)COC1CCN(C(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147284236 EI On-Demand Anodyne GPR88 0 42 O=C(O)COc1ccc([C@H]2[C@H](CCSc3ccc(F)cc3)C(=O)N2c2ccc(F)cc2)cc1 ZINC000147284288 JK For-Sale Anodyne NPC1L1 23 49 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284315 CD On-Demand Anodyne OPRK1 0 45 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284315 CD On-Demand Anodyne MMP13 49 42 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284315 CD On-Demand Anodyne MLNR 21 40 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284315 CD On-Demand Anodyne MMP3 49 42 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284315 CD On-Demand Anodyne MMP8 34 41 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284315 CD On-Demand Anodyne MMP9 51 42 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284315 CD On-Demand Anodyne MMP7 45 42 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284315 CD On-Demand Anodyne MMP1 52 46 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@@H]1N ZINC000147284315 CD On-Demand Anodyne GPR183 0 45 COc1ccccc1N1CCC(NCc2ccc(Br)s2)CC1 ZINC000147284318 GI On-Demand Anodyne HTR1A 82 44 COc1ccccc1N1CCC(NCc2ccc(Br)s2)CC1 ZINC000147284318 GI On-Demand Anodyne DRD2 64 44 COc1ccccc1N1CCC(NCc2ccc(Br)s2)CC1 ZINC000147284318 GI On-Demand Anodyne DRD4 32 41 COc1ccccc1N1CCC(NCc2ccc(Br)s2)CC1 ZINC000147284318 GI On-Demand Anodyne ADRA1D 84 63 COc1ccccc1N1CCC(NCc2ccc(Br)s2)CC1 ZINC000147284318 GI On-Demand Anodyne ADRA1A 71 45 COc1ccccc1N1CCC(NCc2ccc(Br)s2)CC1 ZINC000147284318 GI On-Demand Anodyne ADRA1B 68 63 COc1ccccc1N1CCC(NCc2ccc(Br)s2)CC1 ZINC000147284318 GI On-Demand Anodyne DRD3 57 44 COc1ccccc1N1CCC(NCc2ccc(Br)s2)CC1 ZINC000147284318 GI On-Demand Anodyne HTR7 48 42 CC1(C)Oc2ncnc(N)c2C=C1c1ccc([C@@H]2CC[C@@H](CC(=O)O)CC2)cc1 ZINC000147284347 GJ Annotated Anodyne DGAT1 62 60 BrC1C[C@@H]2CC[C@@H](C1)N2Cc1ccccc1 ZINC000147284394 CH For-Sale Reactive SLC6A3 18 51 BrC1C[C@@H]2CC[C@@H](C1)N2Cc1ccccc1 ZINC000147284394 CH For-Sale Reactive SLC18A2 41 35 BrC1C[C@@H]2CC[C@@H](C1)N2Cc1ccccc1 ZINC000147284394 CH For-Sale Reactive KCNH2 25 45 BrC1C[C@@H]2CC[C@@H](C1)N2Cc1ccccc1 ZINC000147284394 CH For-Sale Reactive LTA4H 15 46 BrC1C[C@@H]2CC[C@@H](C1)N2Cc1ccccc1 ZINC000147284394 CH For-Sale Reactive SIGMAR1 34 59 BrC1C[C@@H]2CC[C@@H](C1)N2Cc1ccccc1 ZINC000147284394 CH For-Sale Reactive ACHP_LYMST 24 51 BrC1C[C@@H]2CC[C@@H](C1)N2Cc1ccccc1 ZINC000147284394 CH For-Sale Reactive ARG1 31 43 BrC1C[C@@H]2CC[C@@H](C1)N2Cc1ccccc1 ZINC000147284394 CH For-Sale Reactive ARG2 31 43 CCCCCCCCn1c(C)c(C)c2c(N)ncnc21 ZINC000147284521 CH For-Sale Mild ADA 52 45 CCCCCCCCn1c(C)c(C)c2c(N)ncnc21 ZINC000147284521 CH For-Sale Mild SRC 0 44 CCCCCCCCn1c(C)c(C)c2c(N)ncnc21 ZINC000147284521 CH For-Sale Mild HSP90B1 45 39 FCCc1cccc(Br)c1 ZINC000147284525 BF For-Sale Anodyne TAAR1 15 69 Cc1cccc(N(C)C(=O)c2cccc3c2OCCN3)c1 ZINC000147284528 CG For-Sale Anodyne HSD17B2 25 45 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284558 CD On-Demand Anodyne OPRK1 0 45 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284558 CD On-Demand Anodyne MMP13 49 42 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284558 CD On-Demand Anodyne MLNR 21 40 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284558 CD On-Demand Anodyne MMP3 49 42 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284558 CD On-Demand Anodyne MMP8 34 41 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284558 CD On-Demand Anodyne MMP9 51 42 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284558 CD On-Demand Anodyne MMP7 45 42 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284558 CD On-Demand Anodyne MMP1 52 46 CC[C@@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284558 CD On-Demand Anodyne GPR183 0 45 C[C@H](CNS(=O)(=O)Cc1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147284596 DD On-Demand Bother MMP1 33 42 CCCNc1nccc(Oc2ccccc2[C@@H](C)CC)n1 ZINC000147284707 CJ For-Sale Anodyne AO-ACHE 0 40 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284751 CD On-Demand Anodyne OPRK1 0 45 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284751 CD On-Demand Anodyne MMP13 57 46 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284751 CD On-Demand Anodyne MLNR 21 40 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284751 CD On-Demand Anodyne MMP3 59 42 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284751 CD On-Demand Anodyne MMP8 34 41 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284751 CD On-Demand Anodyne MMP9 53 46 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284751 CD On-Demand Anodyne MMP7 45 42 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284751 CD On-Demand Anodyne MMP1 61 46 CC[C@H]1CN(C(=O)Cc2ccc(OC)cc2)CC[C@H]1N ZINC000147284751 CD On-Demand Anodyne GPR183 0 45 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCCC1 ZINC000147284769 DC For-Sale Anodyne COLA 41 48 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCCC1 ZINC000147284769 DC For-Sale Anodyne CPT1A 37 48 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCCC1 ZINC000147284769 DC For-Sale Anodyne CPT2 45 36 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCCC1 ZINC000147284769 DC For-Sale Anodyne PTGDR2 37 42 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCCC1 ZINC000147284769 DC For-Sale Anodyne GPR183 0 41 COC(=O)c1ccc(F)c(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)c1 ZINC000147284771 HI On-Demand Anodyne ROCK2 36 43 COC(=O)c1ccc(F)c(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)c1 ZINC000147284771 HI On-Demand Anodyne NAMPT 38 40 C[C@@H](CNS(=O)(=O)Cc1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147284808 DD On-Demand Bother MMP1 33 42 CCCNc1nccc(Oc2ccccc2[C@H](C)CC)n1 ZINC000147284888 CJ For-Sale Anodyne AO-ACHE 0 40 CCN(C(=O)C[C@@H]1CNc2ccccc21)C1CC1 ZINC000147284927 BF For-Sale Anodyne MBTPS1 49 34 CCCCCCCCNC(=O)c1cn[nH]c1N ZINC000147284932 BE For-Sale Mild ASAH1 94 37 CCCNCc1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147284975 CJ For-Sale Anodyne LEF 54 40 CC[C@@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@@H]1N ZINC000147284985 CD On-Demand Anodyne CCR3 0 48 CC[C@@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@@H]1N ZINC000147284985 CD On-Demand Anodyne L3MBTL3 65 35 CC[C@@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@@H]1N ZINC000147284985 CD On-Demand Anodyne HPGD 45 37 CCS(=O)(=O)N[C@H]1CCOC1=O ZINC000147285011 AB On-Demand Anodyne LUXR 71 45 CCS(=O)(=O)N[C@H]1CCOC1=O ZINC000147285011 AB On-Demand Anodyne TRAR 86 45 CCS(=O)(=O)N[C@H]1CCOC1=O ZINC000147285011 AB On-Demand Anodyne LASR 69 45 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCCCC1 ZINC000147285015 ED For-Sale Anodyne COLA 34 47 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCCCC1 ZINC000147285015 ED For-Sale Anodyne CPT1A 30 47 NS(=O)(=O)c1cc(Cl)ccc1OCC(=O)N1CCCCC1 ZINC000147285015 ED For-Sale Anodyne PTGDR2 35 42 O=C(c1cc2cc(Br)ccc2[nH]1)N1CCNCC1 ZINC000147285055 DD On-Demand Anodyne GRIN2B 27 45 O=C(c1cc2cc(Br)ccc2[nH]1)N1CCNCC1 ZINC000147285055 DD On-Demand Anodyne HRH4 43 68 O=C(c1cc2cc(Br)ccc2[nH]1)N1CCNCC1 ZINC000147285055 DD On-Demand Anodyne FPR2 27 47 O=C(c1cc2cc(Br)ccc2[nH]1)N1CCNCC1 ZINC000147285055 DD On-Demand Anodyne AKR1C3 20 45 O=C(c1cc2cc(Br)ccc2[nH]1)N1CCNCC1 ZINC000147285055 DD On-Demand Anodyne PYK 54 41 CCc1c(N)ncnc1Oc1ccccc1[C@@H](C)CC ZINC000147285113 CH For-Sale Anodyne AO-ACHE 0 42 CCCCCCCCNC(=O)c1c(C)n[nH]c1N ZINC000147285126 CE For-Sale Mild ASAH1 78 34 CCN(C(=O)C[C@H]1CNc2ccccc21)C1CC1 ZINC000147285149 BF For-Sale Anodyne MBTPS1 49 34 CC[C@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@@H]1N ZINC000147285188 CD On-Demand Anodyne CCR3 0 48 CC[C@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@@H]1N ZINC000147285188 CD On-Demand Anodyne L3MBTL3 65 35 CC[C@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@@H]1N ZINC000147285188 CD On-Demand Anodyne HPGD 45 37 CC(C)NCc1ccccc1Oc1ccc(Cl)c(F)c1 ZINC000147285216 CJ For-Sale Anodyne SLC6A4 18 60 COc1cc(CNCCCCC(C)C)ccc1OC(C)C ZINC000147285240 CI For-Sale Anodyne LPAR2 44 34 COc1cc(CNCCCCC(C)C)ccc1OC(C)C ZINC000147285240 CI For-Sale Anodyne S1PR2 46 34 COc1cc(CNCCCCC(C)C)ccc1OC(C)C ZINC000147285240 CI For-Sale Anodyne LEF 76 38 COc1cc(CNCCCCC(C)C)ccc1OC(C)C ZINC000147285240 CI For-Sale Anodyne LMGT2 0 45 CC(C)CNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147285246 DD For-Sale Anodyne ALPL 16 40 CC(C)COC1CCN(C(=O)c2ccc3c(c2)COC3)CC1 ZINC000147285256 DF On-Demand Anodyne HRH3 18 45 CCc1c(N)ncnc1Oc1ccccc1[C@H](C)CC ZINC000147285318 CH For-Sale Anodyne AO-ACHE 0 42 CCCCCCCCNC(=O)c1cnn(C)c1N ZINC000147285346 CE On-Demand Mild ASAH1 98 42 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild ACE 48 41 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CNR1 0 45 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild OPRM1 98 67 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild OPRD1 99 66 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild OPRK1 32 48 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CACNA2D1 0 56 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild MME 140 59 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild LTA4H 19 42 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild ANPEP 106 39 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild TACR1 15 56 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild MC4R 38 43 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild FCER2 79 35 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild TACR2 38 41 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild RNPEP 46 44 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild PTPN2 22 42 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CTSB 56 42 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild PAPA1_CARPA 73 50 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CYSP_TRYCR 48 38 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CCKAR 40 39 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CTSK 22 40 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CTSL 54 41 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CPA1 55 37 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CCR3 0 42 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild SCN2A 32 43 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild F2R 0 40 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild BRS3 27 42 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild NPFFR2 60 39 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild TIMP3 74 35 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild C3AR1 46 45 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild S1PR4 36 40 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild TPH1 83 38 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CTRB1 33 43 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild S1PR3 35 49 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild TACR3 28 49 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild MC3R 55 35 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild MC5R 56 35 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CAPNS1 64 38 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild MMP2 24 49 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild MMP3 37 49 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild MMP8 29 48 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild GRIA1 104 45 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild HLA-DRB1 65 42 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild SOAT1 52 44 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild REN 26 41 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild FAAH 25 44 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild PCSK5 42 37 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild FURIN 59 37 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild PTPRA 46 42 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild SCN5A 0 42 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild YARS 70 43 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild PTPN1 18 44 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CCKBR 29 43 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CTSS 25 41 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild GHSR 21 40 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild SLC1A1 18 40 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild S1PR2 70 49 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CTSH 32 40 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CAPN1 78 50 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild MMP9 29 41 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild S1PR1 19 49 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CAPN2 94 46 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild EPHX2 18 42 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild ACE2 58 40 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild MC1R 79 43 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild S1PR5 25 40 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild LAP3 66 47 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CTSC 38 40 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild MMP7 20 45 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild TPP2 22 42 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild MMP1 31 45 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild FPR1 54 50 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild CTRB_BOVIN 52 41 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild NPR 62 45 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild AMP1_PLAFQ 71 49 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild KIF11 29 40 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild KISS1R 58 31 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild POLG_WNV 47 32 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild ASAH1 100 41 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild ERAP2 45 33 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild QRFPR 54 44 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild NPFFR1 78 39 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild NOD1 64 44 CCCCCCCCNC(=O)[C@@H](N)Cc1ccccc1 ZINC000147285383 CG For-Sale Mild TMPRSS6 43 35 CC[C@@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@H]1N ZINC000147285399 CD On-Demand Anodyne CCR3 0 48 CC[C@@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@H]1N ZINC000147285399 CD On-Demand Anodyne L3MBTL3 65 35 CC[C@@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@H]1N ZINC000147285399 CD On-Demand Anodyne HPGD 45 37 O=C(NCc1c(Cl)cccc1Cl)c1ccccc1Cl ZINC000147285403 DJ On-Demand Anodyne DRD3 20 45 O=C(NCc1c(Cl)cccc1Cl)c1ccccc1Cl ZINC000147285403 DJ On-Demand Anodyne P2RX7 33 50 O=C(NCc1c(Cl)cccc1Cl)c1ccccc1Cl ZINC000147285403 DJ On-Demand Anodyne ECR 64 47 O=C(NCc1c(Cl)cccc1Cl)c1ccccc1Cl ZINC000147285403 DJ On-Demand Anodyne SMO 19 46 O=C(NCc1c(Cl)cccc1Cl)c1ccccc1Cl ZINC000147285403 DJ On-Demand Anodyne E3UJZ5_SPOLI 42 40 O=C(NCc1c(Cl)cccc1Cl)c1ccccc1Cl ZINC000147285403 DJ On-Demand Anodyne KCNK3 19 41 CS(=O)(=O)Nc1ccc(F)cc1C(=O)NC[C@@H]1CCCc2ccccc21 ZINC000147285415 GG On-Demand Anodyne HTR6 48 46 CCNC(=O)c1cccc(NC(=O)c2csc(COC)n2)c1 ZINC000147285440 DE On-Demand Anodyne KCNK3 82 39 CCNC(=O)c1cccc(NC(=O)c2csc(COC)n2)c1 ZINC000147285440 DE On-Demand Anodyne KCNK9 71 37 NC(=O)c1ccc(OCC(=O)NCCN2CCN(c3ncccn3)CC2)cc1 ZINC000147285454 GB On-Demand Anodyne HTR1A 50 50 NC(=O)c1ccc(OCC(=O)NCCN2CCN(c3ncccn3)CC2)cc1 ZINC000147285454 GB On-Demand Anodyne DRD2 42 48 NC(=O)c1ccc(OCC(=O)NCCN2CCN(c3ncccn3)CC2)cc1 ZINC000147285454 GB On-Demand Anodyne DRD1 15 46 NC(=O)c1ccc(OCC(=O)NCCN2CCN(c3ncccn3)CC2)cc1 ZINC000147285454 GB On-Demand Anodyne DRD4 48 36 NC(=O)c1ccc(OCC(=O)NCCN2CCN(c3ncccn3)CC2)cc1 ZINC000147285454 GB On-Demand Anodyne HTR2A 20 46 NC(=O)c1ccc(OCC(=O)NCCN2CCN(c3ncccn3)CC2)cc1 ZINC000147285454 GB On-Demand Anodyne DRD3 49 46 CC(=O)N1CCN(c2ccc(CN(C3CCC3)S(=O)(=O)c3cccc(C#N)c3)c(F)c2)CC1 ZINC000147285467 JG Annotated Mild SSTR3 42 34 Cc1cc(C)c(S(=O)(=O)NC[C@@H](C)CC(=O)O)c(C)c1 ZINC000147285468 CE On-Demand Anodyne NR3C1 16 43 Cc1cc(C)c(S(=O)(=O)NC[C@@H](C)CC(=O)O)c(C)c1 ZINC000147285468 CE On-Demand Anodyne NR3C2 31 40 Cc1cc(C)c(S(=O)(=O)NC[C@@H](C)CC(=O)O)c(C)c1 ZINC000147285468 CE On-Demand Anodyne ITGAV 41 43 COc1ccccc1N1CCC(NCc2cn[nH]c2-c2ccc(C)o2)CC1 ZINC000147285478 FH On-Demand Anodyne HTR1A 61 39 COc1ccccc1N1CCC(NCc2cn[nH]c2-c2ccc(C)o2)CC1 ZINC000147285478 FH On-Demand Anodyne DRD2 50 39 COc1ccccc1N1CCC(NCc2cn[nH]c2-c2ccc(C)o2)CC1 ZINC000147285478 FH On-Demand Anodyne ADRA1D 53 35 COc1ccccc1N1CCC(NCc2cn[nH]c2-c2ccc(C)o2)CC1 ZINC000147285478 FH On-Demand Anodyne ADRA1A 42 36 COc1ccccc1N1CCC(NCc2cn[nH]c2-c2ccc(C)o2)CC1 ZINC000147285478 FH On-Demand Anodyne ADRA1B 44 36 COc1ccccc1N1CCC(NCc2cn[nH]c2-c2ccc(C)o2)CC1 ZINC000147285478 FH On-Demand Anodyne DRD3 43 37 COc1ccccc1N1CCC(NCc2cn[nH]c2-c2ccc(C)o2)CC1 ZINC000147285478 FH On-Demand Anodyne HTR7 45 37 COC(=O)Cn1cc(NC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)cn1 ZINC000147285509 GF On-Demand Anodyne PANC 45 33 COC(=O)Cn1cc(NC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)cn1 ZINC000147285509 GF On-Demand Anodyne NAMPT 25 43 CCCCCCCCn1c(N)cc2ccccc2c1=O ZINC000147285578 CH For-Sale Mild CNR1 31 42 CCCCCCCCn1c(N)cc2ccccc2c1=O ZINC000147285578 CH For-Sale Mild CNR2 39 43 CC[C@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@H]1N ZINC000147285607 CD On-Demand Anodyne CCR3 0 48 CC[C@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@H]1N ZINC000147285607 CD On-Demand Anodyne L3MBTL3 65 35 CC[C@H]1CN(C(=O)c2ccc3nccnc3c2)CC[C@H]1N ZINC000147285607 CD On-Demand Anodyne HPGD 45 37 O=C(NCCN1CCN(c2ncccn2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147285674 GD On-Demand Anodyne HTR1A 50 51 O=C(NCCN1CCN(c2ncccn2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147285674 GD On-Demand Anodyne DRD2 44 49 O=C(NCCN1CCN(c2ncccn2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147285674 GD On-Demand Anodyne DRD4 46 35 O=C(NCCN1CCN(c2ncccn2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147285674 GD On-Demand Anodyne DRD3 50 46 O=C(NCCN1CCN(c2ncccn2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147285674 GD On-Demand Anodyne PLD2 43 33 Cc1cc(C)c(S(=O)(=O)NC[C@H](C)CC(=O)O)c(C)c1 ZINC000147285685 CE On-Demand Anodyne NR3C1 16 43 Cc1cc(C)c(S(=O)(=O)NC[C@H](C)CC(=O)O)c(C)c1 ZINC000147285685 CE On-Demand Anodyne NR3C2 31 40 Cc1cc(C)c(S(=O)(=O)NC[C@H](C)CC(=O)O)c(C)c1 ZINC000147285685 CE On-Demand Anodyne ITGAV 41 43 C=CC(=O)NCC(=O)OCc1ccccc1 ZINC000147285698 BD For-Sale Anodyne PPIA 42 33 C=CC(=O)NCC(=O)OCc1ccccc1 ZINC000147285698 BD For-Sale Anodyne PAPA1_CARPA 48 32 C=CC(=O)NCC(=O)OCc1ccccc1 ZINC000147285698 BD For-Sale Anodyne CAPN2 58 33 C=CC(=O)NCC(=O)OCc1ccccc1 ZINC000147285698 BD For-Sale Anodyne TGM2 58 46 C=CC(=O)NCC(=O)OCc1ccccc1 ZINC000147285698 BD For-Sale Anodyne 17HSDCL 0 43 C=CC(=O)NCC(=O)OCc1ccccc1 ZINC000147285698 BD For-Sale Anodyne RHODESAIN 0 44 C=CC(=O)NCC(=O)OCc1ccccc1 ZINC000147285698 BD For-Sale Anodyne F13A1 60 43 COC(=O)Cn1cc(NC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)cn1 ZINC000147285712 GF On-Demand Anodyne PANC 45 33 COC(=O)Cn1cc(NC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)cn1 ZINC000147285712 GF On-Demand Anodyne NAMPT 25 43 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild CA2 102 71 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild DRD4 40 31 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild CA1 77 48 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild CA7 58 47 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild CA13 25 47 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild CA5B 52 36 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild CA4 79 48 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild CA5A 54 36 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild CA14 39 47 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild GRIA1 43 35 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild FBP1 21 43 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild EPHX2 0 40 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild CA12 39 44 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild CA9 46 47 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild PA2A1_NAJMO 0 41 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild TTK 32 44 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild AKR1C3 16 40 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild CYNT 24 42 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild NCE103 55 35 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild ASAH1 89 35 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild MTCA1 40 37 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild P96878_MYCTU 40 42 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild ACAT 0 45 CCCCCCCCNC(=O)c1cccc(S(N)(=O)=O)c1 ZINC000147285817 DE For-Sale Mild Q5TU56_ANOGA 0 41 COC(=O)Cn1cc(NC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)cn1 ZINC000147285886 GF On-Demand Anodyne PANC 45 33 COC(=O)Cn1cc(NC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)cn1 ZINC000147285886 GF On-Demand Anodyne NAMPT 25 43 CCCCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147285897 ED For-Sale Anodyne PPARG 25 40 CCCCNC(=O)[C@@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147285897 ED For-Sale Anodyne PTGDR2 32 40 C[C@H](CNS(=O)(=O)c1cc(Cl)ccc1Cl)CC(=O)O ZINC000147285914 EE On-Demand Anodyne OXER1 42 37 Cc1cccc(CCC(=O)N2CCC[C@H](CCBr)C2)c1 ZINC000147285985 EH For-Sale Reactive C3AR1 33 41 COc1ccccc1N1CCC(NCc2cccc(C#N)c2)CC1 ZINC000147285988 DG On-Demand Mild HTR1A 27 41 COc1ccccc1N1CCC(NCc2cccc(C#N)c2)CC1 ZINC000147285988 DG On-Demand Mild DRD2 63 42 COc1ccccc1N1CCC(NCc2cccc(C#N)c2)CC1 ZINC000147285988 DG On-Demand Mild DRD1 26 42 COc1ccccc1N1CCC(NCc2cccc(C#N)c2)CC1 ZINC000147285988 DG On-Demand Mild HTR2A 27 42 COc1ccccc1N1CCC(NCc2cccc(C#N)c2)CC1 ZINC000147285988 DG On-Demand Mild ADRA1A 47 41 COc1ccccc1N1CCC(NCc2cccc(C#N)c2)CC1 ZINC000147285988 DG On-Demand Mild DRD3 45 42 COc1ccccc1N1CCC(NCc2cccc(C#N)c2)CC1 ZINC000147285988 DG On-Demand Mild GRIN2B 0 46 COc1ccccc1N1CCC(NCc2cccc(C#N)c2)CC1 ZINC000147285988 DG On-Demand Mild HTR7 41 39 COc1ccccc1N1CCC(NCc2cccc(C#N)c2)CC1 ZINC000147285988 DG On-Demand Mild NPY1R 24 40 CCCCCCCCNS(=O)(=O)c1c[nH]ccc1=O ZINC000147286006 CE For-Sale Mild ALOX15 20 40 CCCCCCCCNS(=O)(=O)c1c[nH]ccc1=O ZINC000147286006 CE For-Sale Mild ASAH1 56 34 CCCCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147286119 ED For-Sale Anodyne PPARG 25 40 CCCCNC(=O)[C@H](C)Oc1ccc(Cl)cc1S(N)(=O)=O ZINC000147286119 ED For-Sale Anodyne PTGDR2 32 40 C[C@@H](CNS(=O)(=O)c1cc(Cl)ccc1Cl)CC(=O)O ZINC000147286131 EE On-Demand Anodyne OXER1 42 37 Cc1cccc(CCC(=O)N2CCC[C@@H](CCBr)C2)c1 ZINC000147286178 EH For-Sale Reactive C3AR1 33 41 COC(=O)Cn1cc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cn1 ZINC000147286222 EE On-Demand Anodyne MDM2 57 34 COC(=O)Cn1cc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cn1 ZINC000147286222 EE On-Demand Anodyne PANC 50 34 COC(=O)Cn1cc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cn1 ZINC000147286222 EE On-Demand Anodyne NAMPT 26 43 Cc1cccc(NC(=O)CCCNC2(C(=O)O)CCC2)c1 ZINC000147286252 CE For-Sale Anodyne CCKAR 24 41 Cc1cccc(NC(=O)CCCNC2(C(=O)O)CCC2)c1 ZINC000147286252 CE For-Sale Anodyne HDAC3 37 40 Cc1cccc(NC(=O)CCCNC2(C(=O)O)CCC2)c1 ZINC000147286252 CE For-Sale Anodyne HDAC6 26 41 Cc1cccc(NC(=O)CCCNC2(C(=O)O)CCC2)c1 ZINC000147286252 CE For-Sale Anodyne KCNK3 57 38 Cc1cccc(NC(=O)CCCNC2(C(=O)O)CCC2)c1 ZINC000147286252 CE For-Sale Anodyne KCNK9 43 38 Cc1cccc(NC(=O)CCCNC2(C(=O)O)CCC2)c1 ZINC000147286252 CE For-Sale Anodyne PARP10 0 42 CCCCCCCCNS(=O)(=O)c1sc(=O)[nH]c1C ZINC000147286410 DE For-Sale Mild ASAH1 49 30 COC(=O)Cn1cc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cn1 ZINC000147286445 EE On-Demand Anodyne MDM2 57 34 COC(=O)Cn1cc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cn1 ZINC000147286445 EE On-Demand Anodyne PANC 50 34 COC(=O)Cn1cc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cn1 ZINC000147286445 EE On-Demand Anodyne NAMPT 26 43 COc1ccc(CNCC(F)F)cc1C ZINC000147286494 BE On-Demand Clean MT-ND1 15 40 N#Cc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147286539 CD On-Demand Mild DHODH 68 46 CCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147286619 DD For-Sale Anodyne CA2 35 40 CCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147286619 DD For-Sale Anodyne CA1 33 40 CCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147286619 DD For-Sale Anodyne CA12 19 40 CCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147286619 DD For-Sale Anodyne PTGDR 23 40 CCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147286619 DD For-Sale Anodyne CA9 18 40 CCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147286619 DD For-Sale Anodyne PTGDR2 48 40 CCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147286619 DD For-Sale Anodyne CAN2 0 43 CCCCNC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147286619 DD For-Sale Anodyne PSBA 0 41 COC(=O)Cn1cc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cn1 ZINC000147286644 EE On-Demand Anodyne MDM2 57 34 COC(=O)Cn1cc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cn1 ZINC000147286644 EE On-Demand Anodyne PANC 50 34 COC(=O)Cn1cc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cn1 ZINC000147286644 EE On-Demand Anodyne NAMPT 26 43 O=c1nc(-c2c[nH]c3ccccc23)[nH]c2ccccc12 ZINC000147286736 CG In-Stock Anodyne PRKCE 0 50 O=c1nc(-c2c[nH]c3ccccc23)[nH]c2ccccc12 ZINC000147286736 CG In-Stock Anodyne PRKCB 28 50 CCNCCCOc1ccc(Cl)c(F)c1 ZINC000147286843 BF For-Sale Anodyne DRD4 22 51 CCCCCCCCNS(=O)(=O)c1c[nH]cn1 ZINC000147286864 CE On-Demand Mild HRH3 19 49 CCCCCCCCNS(=O)(=O)c1c[nH]cn1 ZINC000147286864 CE On-Demand Mild ASAH1 44 30 COc1ccccc1/C=C/c1ccc[nH]1 ZINC000147286903 AG For-Sale Anodyne CYP1B1 52 51 COc1ccccc1/C=C/c1ccc[nH]1 ZINC000147286903 AG For-Sale Anodyne CYP1A2 15 51 COC(=O)Cn1cc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cn1 ZINC000147286928 ED On-Demand Anodyne ROCK2 37 50 COC(=O)Cn1cc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cn1 ZINC000147286928 ED On-Demand Anodyne PANC 41 32 COc1ccc(C)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147286938 EH On-Demand Anodyne HTR1A 88 44 COc1ccc(C)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147286938 EH On-Demand Anodyne DRD2 72 46 COc1ccc(C)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147286938 EH On-Demand Anodyne DRD1 17 44 COc1ccc(C)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147286938 EH On-Demand Anodyne DRD4 42 44 COc1ccc(C)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147286938 EH On-Demand Anodyne ADRA1D 87 46 COc1ccc(C)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147286938 EH On-Demand Anodyne HTR2A 22 44 COc1ccc(C)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147286938 EH On-Demand Anodyne ADRA1A 74 46 COc1ccc(C)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147286938 EH On-Demand Anodyne ADRA1B 70 46 COc1ccc(C)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147286938 EH On-Demand Anodyne DRD3 66 44 COc1ccc(C)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147286938 EH On-Demand Anodyne HTR7 53 43 COc1ccc(C)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147286938 EH On-Demand Anodyne NPY1R 17 41 CC[C@@H](C)c1ccccc1Oc1ccnc(N)n1 ZINC000147286949 BG For-Sale Anodyne AO-ACHE 0 41 CCCCCCCCNS(=O)(=O)c1cnc(C)[nH]1 ZINC000147287084 CE For-Sale Mild ASAH1 43 30 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147287126 GH On-Demand Anodyne LCK 21 40 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147287126 GH On-Demand Anodyne CSNK1D 44 49 CN(C(=O)COc1ccc(Cl)cc1S(N)(=O)=O)C1CC1 ZINC000147287152 DC For-Sale Anodyne PTGDR2 41 39 COc1ccccc1N1CCC(NCc2cc3ccccc3o2)CC1 ZINC000147287168 EI On-Demand Anodyne HTR1A 85 48 COc1ccccc1N1CCC(NCc2cc3ccccc3o2)CC1 ZINC000147287168 EI On-Demand Anodyne DRD2 69 49 COc1ccccc1N1CCC(NCc2cc3ccccc3o2)CC1 ZINC000147287168 EI On-Demand Anodyne DRD1 16 47 COc1ccccc1N1CCC(NCc2cc3ccccc3o2)CC1 ZINC000147287168 EI On-Demand Anodyne DRD4 41 48 COc1ccccc1N1CCC(NCc2cc3ccccc3o2)CC1 ZINC000147287168 EI On-Demand Anodyne ADRA1D 74 41 COc1ccccc1N1CCC(NCc2cc3ccccc3o2)CC1 ZINC000147287168 EI On-Demand Anodyne HTR2A 19 42 COc1ccccc1N1CCC(NCc2cc3ccccc3o2)CC1 ZINC000147287168 EI On-Demand Anodyne ADRA1A 64 48 COc1ccccc1N1CCC(NCc2cc3ccccc3o2)CC1 ZINC000147287168 EI On-Demand Anodyne ADRA1B 60 41 COc1ccccc1N1CCC(NCc2cc3ccccc3o2)CC1 ZINC000147287168 EI On-Demand Anodyne DRD3 67 49 COc1ccccc1N1CCC(NCc2cc3ccccc3o2)CC1 ZINC000147287168 EI On-Demand Anodyne HTR2B 17 50 COc1ccccc1N1CCC(NCc2cc3ccccc3o2)CC1 ZINC000147287168 EI On-Demand Anodyne HTR7 51 43 CC[C@H](C)c1ccccc1Oc1ccnc(N)n1 ZINC000147287173 BG For-Sale Anodyne AO-ACHE 0 41 CCCN(C(=O)C[C@@H]1CNc2ccccc21)C1CC1 ZINC000147287213 CF For-Sale Anodyne MBTPS1 68 33 CN(C)C1(CNC(=O)c2ccc3cn[nH]c3c2)CCCC1 ZINC000147287323 CE For-Sale Anodyne SLC6A5 16 47 CCCNC[C@@H](C)COc1ccc(Cl)c(F)c1 ZINC000147287329 CG For-Sale Anodyne GRIN1 25 43 C[C@@H]1CCCN(C(=O)c2cccc3c2OCCN3)[C@@H]1C ZINC000147287331 CF For-Sale Anodyne TRPC6 51 37 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147287335 GH On-Demand Anodyne LCK 21 40 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147287335 GH On-Demand Anodyne CSNK1D 44 49 COc1ccccc1N1CCC(NCc2c(C)nn(Cc3ccccc3)c2C)CC1 ZINC000147287356 HI On-Demand Anodyne HTR1A 73 40 COc1ccccc1N1CCC(NCc2c(C)nn(Cc3ccccc3)c2C)CC1 ZINC000147287356 HI On-Demand Anodyne DRD2 56 41 COc1ccccc1N1CCC(NCc2c(C)nn(Cc3ccccc3)c2C)CC1 ZINC000147287356 HI On-Demand Anodyne DRD4 39 41 COc1ccccc1N1CCC(NCc2c(C)nn(Cc3ccccc3)c2C)CC1 ZINC000147287356 HI On-Demand Anodyne ADRA1D 55 38 COc1ccccc1N1CCC(NCc2c(C)nn(Cc3ccccc3)c2C)CC1 ZINC000147287356 HI On-Demand Anodyne ADRA1A 48 38 COc1ccccc1N1CCC(NCc2c(C)nn(Cc3ccccc3)c2C)CC1 ZINC000147287356 HI On-Demand Anodyne ADRA1B 45 38 COc1ccccc1N1CCC(NCc2c(C)nn(Cc3ccccc3)c2C)CC1 ZINC000147287356 HI On-Demand Anodyne DRD3 52 40 COc1ccccc1N1CCC(NCc2c(C)nn(Cc3ccccc3)c2C)CC1 ZINC000147287356 HI On-Demand Anodyne HTR7 43 40 Cc1cccc(C(=O)Nc2ccccc2C(=O)N2CCO[C@@H](c3ccc(F)cc3)C2)c1 ZINC000147287408 HJ On-Demand Anodyne KCNK3 65 39 Cc1cccc(C(=O)Nc2ccccc2C(=O)N2CCO[C@@H](c3ccc(F)cc3)C2)c1 ZINC000147287408 HJ On-Demand Anodyne KCNK9 46 39 CCCN(C(=O)C[C@H]1CNc2ccccc21)C1CC1 ZINC000147287422 CF For-Sale Anodyne MBTPS1 68 33 CCCCCCCCNS(=O)(=O)c1cn[nH]c1 ZINC000147287444 CE For-Sale Mild ALOX15 50 44 CCCNC[C@H](C)COc1ccc(Cl)c(F)c1 ZINC000147287535 CG For-Sale Anodyne GRIN1 25 43 C[C@H]1CCCN(C(=O)c2cccc3c2OCCN3)[C@@H]1C ZINC000147287541 CF For-Sale Anodyne TRPC6 51 37 O=C(O)c1ccc(CNc2cc(Cl)ccc2Br)cc1 ZINC000147287544 EI For-Sale Anodyne SRD5A2 24 41 O=C(O)c1ccc(CNc2cc(Cl)ccc2Br)cc1 ZINC000147287544 EI For-Sale Anodyne UL80 23 42 O=C(O)c1ccc(CNc2cc(Cl)ccc2Br)cc1 ZINC000147287544 EI For-Sale Anodyne RPA1 43 35 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147287550 GH On-Demand Anodyne LCK 21 40 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147287550 GH On-Demand Anodyne CSNK1D 44 49 COc1ccccc1N1CCC(NCc2cc(Br)cs2)CC1 ZINC000147287616 GI On-Demand Anodyne HTR1A 79 45 COc1ccccc1N1CCC(NCc2cc(Br)cs2)CC1 ZINC000147287616 GI On-Demand Anodyne DRD2 65 45 COc1ccccc1N1CCC(NCc2cc(Br)cs2)CC1 ZINC000147287616 GI On-Demand Anodyne DRD1 15 40 COc1ccccc1N1CCC(NCc2cc(Br)cs2)CC1 ZINC000147287616 GI On-Demand Anodyne DRD4 36 45 COc1ccccc1N1CCC(NCc2cc(Br)cs2)CC1 ZINC000147287616 GI On-Demand Anodyne ADRA1D 77 45 COc1ccccc1N1CCC(NCc2cc(Br)cs2)CC1 ZINC000147287616 GI On-Demand Anodyne HTR2A 16 40 COc1ccccc1N1CCC(NCc2cc(Br)cs2)CC1 ZINC000147287616 GI On-Demand Anodyne ADRA1A 66 41 COc1ccccc1N1CCC(NCc2cc(Br)cs2)CC1 ZINC000147287616 GI On-Demand Anodyne ADRA1B 62 45 COc1ccccc1N1CCC(NCc2cc(Br)cs2)CC1 ZINC000147287616 GI On-Demand Anodyne DRD3 62 45 COc1ccccc1N1CCC(NCc2cc(Br)cs2)CC1 ZINC000147287616 GI On-Demand Anodyne HTR7 47 43 CCCCCCCCNS(=O)(=O)c1c[nH]c(=O)c(Cl)c1 ZINC000147287644 DF For-Sale Mild ALOX15 38 43 CCCCCCCCNS(=O)(=O)c1c[nH]c(=O)c(Cl)c1 ZINC000147287644 DF For-Sale Mild ASAH1 52 32 COc1cccc(N(C)C(=O)[C@@H]2CCC(=O)NC2)c1 ZINC000147287676 CD For-Sale Anodyne MTNR1A 15 46 COc1cccc(N(C)C(=O)[C@@H]2CCC(=O)NC2)c1 ZINC000147287676 CD For-Sale Anodyne MTNR1B 20 46 COc1cccc(N(C)C(=O)[C@@H]2CCC(=O)NC2)c1 ZINC000147287676 CD For-Sale Anodyne HSD17B2 24 44 CN(C)NC(=O)C1CCC(CN)CC1 ZINC000147287744 AC For-Sale Reactive F11 45 35 C[C@H]1[C@H](C)CCCN1C(=O)c1cccc2c1OCCN2 ZINC000147287780 CF For-Sale Anodyne TRPC6 51 37 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne HTR1A 81 51 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne DRD2 72 51 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne DRD1 15 51 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne DRD4 55 51 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne ADRA1D 65 41 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne HTR2A 15 40 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne ADRA1A 56 41 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne ADRA1B 52 41 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne DRD3 71 51 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne HTR7 48 41 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne SIGMAR1 18 44 COc1ccccc1N1CCC(NCc2cnn(Cc3ccccc3)c2)CC1 ZINC000147287831 GH On-Demand Anodyne PANC 49 39 CC[C@@H](C)c1ccccc1Oc1nc(NC)ncc1F ZINC000147287844 CH For-Sale Anodyne AO-ACHE 0 46 COC(=O)c1cc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)ccc1Cl ZINC000147287876 HG On-Demand Anodyne ADRB2 22 40 COC(=O)c1cc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)ccc1Cl ZINC000147287876 HG On-Demand Anodyne ADRB1 48 36 CCCCCCCCNS(=O)(=O)c1ccc(=O)[nH]c1 ZINC000147287880 CE For-Sale Mild ALOX15 59 51 CCCCCCCCNS(=O)(=O)c1ccc(=O)[nH]c1 ZINC000147287880 CE For-Sale Mild ASAH1 53 35 COc1cccc(N(C)C(=O)[C@H]2CCC(=O)NC2)c1 ZINC000147287895 CD For-Sale Anodyne MTNR1A 15 46 COc1cccc(N(C)C(=O)[C@H]2CCC(=O)NC2)c1 ZINC000147287895 CD For-Sale Anodyne MTNR1B 20 46 COc1cccc(N(C)C(=O)[C@H]2CCC(=O)NC2)c1 ZINC000147287895 CD For-Sale Anodyne HSD17B2 24 44 C[C@H]1CCCN(C(=O)c2cccc3c2OCCN3)[C@H]1C ZINC000147287991 CF For-Sale Anodyne TRPC6 51 37 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne PPIA 16 41 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne F10 32 47 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne TRPV1 25 53 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne ECR 43 43 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne COLA 64 39 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne CPT1A 71 39 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne CPT2 45 38 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne PRNP 68 49 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne NR1H4 17 43 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne CPT1B 47 38 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne MAP3K5 63 48 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne TAAR1 17 41 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne TRPA1 16 45 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne SMO 15 45 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne UTS2 41 33 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne IMDH_CRYPV 15 41 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne NOD1 28 44 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne NOD2 41 34 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne NAMPT 16 54 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne Q25615_ONCVO 32 45 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne E3UJZ5_SPOLI 38 43 CC(C)(C)Nc1ccc(NC(=O)c2ccc(Cl)cc2)cc1 ZINC000147288024 DJ For-Sale Anodyne KCNK3 63 49 CC[C@H](C)c1ccccc1Oc1nc(NC)ncc1F ZINC000147288056 CH For-Sale Anodyne AO-ACHE 0 46 COC(=O)c1cc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)ccc1Cl ZINC000147288068 HG On-Demand Anodyne ADRB2 22 40 COC(=O)c1cc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)ccc1Cl ZINC000147288068 HG On-Demand Anodyne ADRB1 48 36 CCCCCCCCNC(=O)CCc1ccccc1N ZINC000147288072 CH For-Sale Mild CNR1 0 43 CCCCCCCCNC(=O)CCc1ccccc1N ZINC000147288072 CH For-Sale Mild TRPV1 0 42 CCCCCCCCNC(=O)CCc1ccccc1N ZINC000147288072 CH For-Sale Mild MTNR1A 42 43 CCCCCCCCNC(=O)CCc1ccccc1N ZINC000147288072 CH For-Sale Mild MTNR1B 36 42 CCCCCCCCNC(=O)CCc1ccccc1N ZINC000147288072 CH For-Sale Mild GRIA1 64 45 CCCCCCCCNC(=O)CCc1ccccc1N ZINC000147288072 CH For-Sale Mild FAAH 17 42 CCCCCCCCNC(=O)CCc1ccccc1N ZINC000147288072 CH For-Sale Mild FURIN 51 34 CCCCCCCCNC(=O)CCc1ccccc1N ZINC000147288072 CH For-Sale Mild EPHX2 27 43 CCCCCCCCNC(=O)CCc1ccccc1N ZINC000147288072 CH For-Sale Mild ASAH1 97 37 C[C@H](CNS(=O)(=O)c1ccc(F)c(F)c1)CC(=O)O ZINC000147288196 CD On-Demand Anodyne TBXA2R 50 36 C[C@H](CNS(=O)(=O)c1ccc(F)c(F)c1)CC(=O)O ZINC000147288196 CD On-Demand Anodyne LEF 61 39 CCCCCC(=O)N1CC[C@@](C)(c2cccc(O)c2)[C@H](C)C1 ZINC000147288230 DI For-Sale Anodyne OPRM1 60 70 CCCCCC(=O)N1CC[C@@](C)(c2cccc(O)c2)[C@H](C)C1 ZINC000147288230 DI For-Sale Anodyne OPRD1 51 55 CCCCCC(=O)N1CC[C@@](C)(c2cccc(O)c2)[C@H](C)C1 ZINC000147288230 DI For-Sale Anodyne OPRK1 63 70 CC(C)(C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147288234 DD For-Sale Anodyne CPT1A 43 30 CC(C)(C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147288234 DD For-Sale Anodyne PTGDR2 44 42 CC(C)CCCCNCc1cc(Br)ccc1OC(F)F ZINC000147288244 FJ For-Sale Anodyne LEF 57 34 CCCCCCCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147288293 CF For-Sale Mild THRA 41 32 CCCCCCCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147288293 CF For-Sale Mild FOLH1 29 46 CCCCCCCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147288293 CF For-Sale Mild RARB 21 42 CCCCCCCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147288293 CF For-Sale Mild THRB 22 50 CCCCCCCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147288293 CF For-Sale Mild KCNQ1 0 45 CCCCCCCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147288293 CF For-Sale Mild PLA2G4B 58 38 CCCCCCCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147288293 CF For-Sale Mild P4HTM 0 53 CCCCCCCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147288293 CF For-Sale Mild EPHX2 38 40 CCCCCCCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147288293 CF For-Sale Mild P4HA1 0 50 CCCCCCCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147288293 CF For-Sale Mild ASAH1 91 37 CCCCCCCCNC(=O)c1ccc(C(=O)O)nc1 ZINC000147288293 CF For-Sale Mild ACAT 0 44 COc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147288294 CD For-Sale Anodyne PDGFRB 21 41 COc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147288294 CD For-Sale Anodyne MTNR1A 46 49 COc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147288294 CD For-Sale Anodyne MTNR1B 48 54 COc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147288294 CD For-Sale Anodyne EPHX2 17 45 COc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147288294 CD For-Sale Anodyne FLT4 20 40 COc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147288294 CD For-Sale Anodyne TAAR1 39 43 COc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147288294 CD For-Sale Anodyne AKR1C3 20 42 COc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147288294 CD For-Sale Anodyne AKR1C2 41 37 COc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147288294 CD For-Sale Anodyne ACAT 0 53 COc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147288294 CD For-Sale Anodyne KCNK3 46 45 CC[C@@H](C)[C@@H](N)C(=O)Nc1ccc(Cl)cc1Br ZINC000147288303 DG For-Sale Anodyne ACPS 0 40 CC[C@@H](C)c1ccccc1Oc1nc(C)nc(N)c1C ZINC000147288329 CH For-Sale Anodyne AO-ACHE 0 41 COc1ccccc1N1CCC(NCc2c(C)nn(-c3ccccc3)c2C)CC1 ZINC000147288341 GI On-Demand Anodyne HTR1A 74 40 COc1ccccc1N1CCC(NCc2c(C)nn(-c3ccccc3)c2C)CC1 ZINC000147288341 GI On-Demand Anodyne DRD2 52 40 COc1ccccc1N1CCC(NCc2c(C)nn(-c3ccccc3)c2C)CC1 ZINC000147288341 GI On-Demand Anodyne DRD4 29 40 COc1ccccc1N1CCC(NCc2c(C)nn(-c3ccccc3)c2C)CC1 ZINC000147288341 GI On-Demand Anodyne ADRA1D 60 38 COc1ccccc1N1CCC(NCc2c(C)nn(-c3ccccc3)c2C)CC1 ZINC000147288341 GI On-Demand Anodyne HTR2A 17 40 COc1ccccc1N1CCC(NCc2c(C)nn(-c3ccccc3)c2C)CC1 ZINC000147288341 GI On-Demand Anodyne ADRA1A 52 39 COc1ccccc1N1CCC(NCc2c(C)nn(-c3ccccc3)c2C)CC1 ZINC000147288341 GI On-Demand Anodyne ADRA1B 48 38 COc1ccccc1N1CCC(NCc2c(C)nn(-c3ccccc3)c2C)CC1 ZINC000147288341 GI On-Demand Anodyne DRD3 49 40 COc1ccccc1N1CCC(NCc2c(C)nn(-c3ccccc3)c2C)CC1 ZINC000147288341 GI On-Demand Anodyne HTR7 48 38 COc1ccccc1N1CCC(NCc2c(C)nn(-c3ccccc3)c2C)CC1 ZINC000147288341 GI On-Demand Anodyne NPY1R 23 42 C[C@@H](CNS(=O)(=O)c1ccc(F)c(F)c1)CC(=O)O ZINC000147288367 CD On-Demand Anodyne TBXA2R 50 36 C[C@@H](CNS(=O)(=O)c1ccc(F)c(F)c1)CC(=O)O ZINC000147288367 CD On-Demand Anodyne LEF 61 39 CC(C)NC[C@@H](C)COc1ccc(Cl)c(F)c1 ZINC000147288380 CG For-Sale Anodyne GRIN1 0 40 CC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147288491 DD On-Demand Anodyne CASR 18 42 CC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147288491 DD On-Demand Anodyne CCR3 19 41 CC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147288491 DD On-Demand Anodyne AKR1C3 15 43 CC(=O)c1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147288491 DD On-Demand Anodyne KCNK3 47 37 CC[C@H](C)[C@@H](N)C(=O)Nc1ccc(Cl)cc1Br ZINC000147288499 DG For-Sale Anodyne ACPS 0 40 CC[C@H](C)c1ccccc1Oc1nc(C)nc(N)c1C ZINC000147288522 CH For-Sale Anodyne AO-ACHE 0 41 CCCCCCCCNC(=O)C1(C(=O)O)CC1 ZINC000147288532 BE For-Sale Mild EPHX2 65 46 CCCCCCCCNC(=O)C1(C(=O)O)CC1 ZINC000147288532 BE For-Sale Mild CPT1 0 43 CCCCCCCCNC(=O)C1(C(=O)O)CC1 ZINC000147288532 BE For-Sale Mild GNAI1 0 45 CCCCCCCCNC(=O)C1(C(=O)O)CC1 ZINC000147288532 BE For-Sale Mild GNAI3 0 45 CCCCCCCCNC(=O)C1(C(=O)O)CC1 ZINC000147288532 BE For-Sale Mild GNAO1 0 45 CCCCCCCCNC(=O)C1(C(=O)O)CC1 ZINC000147288532 BE For-Sale Mild ASAH1 86 34 Cc1cccc(C)c1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147288550 CD For-Sale Anodyne ACAT 0 47 COC(=O)c1cc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)ccc1Cl ZINC000147288554 EH On-Demand Anodyne EPHX2 40 41 CNC(=O)c1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147288570 DC On-Demand Anodyne CA2 29 48 CNC(=O)c1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147288570 DC On-Demand Anodyne TBXA2R 41 32 CNC(=O)c1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147288570 DC On-Demand Anodyne CA1 16 43 CC(C)NC[C@H](C)COc1ccc(Cl)c(F)c1 ZINC000147288572 CG For-Sale Anodyne GRIN1 0 40 CC[C@@H]1CN(C(=O)CCC2CCCC2)CC[C@@H]1N ZINC000147288592 CF On-Demand Anodyne F2R 22 40 CC[C@@H]1CN(C(=O)CCC2CCCC2)CC[C@@H]1N ZINC000147288592 CF On-Demand Anodyne GNAI3 0 40 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne DHODH 31 40 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne JUN 24 42 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne APOB 0 47 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne TRPV1 21 52 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne ATF1 61 48 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne NR1H4 15 40 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne F12 0 41 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne MTTP 61 47 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne NFKB1 56 48 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne EPHX2 25 49 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne MCHR1 0 43 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne BTK 22 41 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne PTPA 0 44 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne TRPM8 33 54 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne SMO 31 41 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne PSBA 0 47 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne KCNK3 83 44 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne KCNK9 74 36 Cc1ccc(Br)c(C(=O)Nc2ccc(C(F)(F)F)cc2)c1 ZINC000147288619 FK On-Demand Anodyne TMPRSS4 0 40 CN(C)C(=O)NCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147288692 CD On-Demand Anodyne CCKAR 38 61 CN(C)C(=O)NCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147288692 CD On-Demand Anodyne PYGL 89 54 CN(C)C(=O)NCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147288692 CD On-Demand Anodyne PYGM 29 41 CN(C)C(=O)NCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147288692 CD On-Demand Anodyne PLCG2 0 40 CN(C)C(=O)NCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147288692 CD On-Demand Anodyne PLD2 33 46 CN(C)C(=O)NCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147288692 CD On-Demand Anodyne FLT3 0 50 CN(C)C(=O)NCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147288692 CD On-Demand Anodyne AKR1C3 0 40 CN(C)C(=O)NCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147288692 CD On-Demand Anodyne PYK 47 41 O=C(O)[C@H]1CCC[C@H]1NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147288712 CE For-Sale Anodyne EPHX2 21 42 O=C(O)[C@H]1CCC[C@H]1NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147288712 CE For-Sale Anodyne GPR88 0 42 CCNc1nc(C)cc(Oc2ccccc2[C@H](C)CC)n1 ZINC000147288733 CJ For-Sale Anodyne AO-ACHE 0 40 CC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147288734 DD On-Demand Anodyne CASR 18 42 CC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147288734 DD On-Demand Anodyne CCR3 19 41 CC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147288734 DD On-Demand Anodyne AKR1C3 15 43 CC(=O)c1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147288734 DD On-Demand Anodyne KCNK3 47 37 CCCCCCCCNC(=O)c1ccc(C(=O)O)o1 ZINC000147288746 CG For-Sale Mild INHA 41 32 CCCCCCCCNC(=O)c1ccc(C(=O)O)o1 ZINC000147288746 CG For-Sale Mild PLA2G2A 49 39 CCCCCCCCNC(=O)c1ccc(C(=O)O)o1 ZINC000147288746 CG For-Sale Mild LPAR2 43 37 CCCCCCCCNC(=O)c1ccc(C(=O)O)o1 ZINC000147288746 CG For-Sale Mild S1PR3 43 38 CCCCCCCCNC(=O)c1ccc(C(=O)O)o1 ZINC000147288746 CG For-Sale Mild GRIA1 47 36 CCCCCCCCNC(=O)c1ccc(C(=O)O)o1 ZINC000147288746 CG For-Sale Mild PLA2G4B 51 34 CCCCCCCCNC(=O)c1ccc(C(=O)O)o1 ZINC000147288746 CG For-Sale Mild FAAH 21 43 CCCCCCCCNC(=O)c1ccc(C(=O)O)o1 ZINC000147288746 CG For-Sale Mild S1PR2 82 41 CCCCCCCCNC(=O)c1ccc(C(=O)O)o1 ZINC000147288746 CG For-Sale Mild S1PR1 19 40 CCCCCCCCNC(=O)c1ccc(C(=O)O)o1 ZINC000147288746 CG For-Sale Mild ASAH1 104 40 C#CCNCC(=O)NN(C)C ZINC000147288770 AA For-Sale Reactive KDM7A 0 42 CNC(=O)c1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147288780 DC On-Demand Anodyne CA2 29 48 CNC(=O)c1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147288780 DC On-Demand Anodyne TBXA2R 41 32 CNC(=O)c1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147288780 DC On-Demand Anodyne CA1 16 43 COC(=O)c1cc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)ccc1Cl ZINC000147288797 EH On-Demand Anodyne EPHX2 40 41 O=C(CNC1(C(=O)O)CCC1)Nc1cccc(Br)c1 ZINC000147288800 ED For-Sale Anodyne EGFR 31 42 CC[C@H]1CN(C(=O)CCC2CCCC2)CC[C@@H]1N ZINC000147288812 CF On-Demand Anodyne F2R 22 40 CC[C@H]1CN(C(=O)CCC2CCCC2)CC[C@@H]1N ZINC000147288812 CF On-Demand Anodyne GNAI3 0 40 Cc1ccc(C(=O)N[C@@H]2CCC[C@@H]2C(=O)O)cc1Br ZINC000147288922 EF On-Demand Anodyne MAPK14 41 39 Cc1ccc(C(=O)N[C@@H]2CCC[C@@H]2C(=O)O)cc1Br ZINC000147288922 EF On-Demand Anodyne ADAM17 23 44 Cc1ccc(C(=O)N[C@@H]2CCC[C@@H]2C(=O)O)cc1Br ZINC000147288922 EF On-Demand Anodyne MAPK13 41 38 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild HTR1A 15 44 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild THRA 46 38 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild DRD2 20 43 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild CNR1 16 41 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild DRD4 47 36 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild ACHE 19 41 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild DRD3 44 43 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild FOLH1 43 46 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild CNR2 17 44 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild RARB 19 42 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild THRB 26 50 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild CCKAR 0 42 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild CTSG 17 40 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild LTB4R 22 45 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild PLA2G4A 28 40 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild HDAC8 15 48 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild CTRB1 23 40 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild PLA2G4B 86 48 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild CELA2A 15 40 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild HDAC6 17 48 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild FAAH 25 48 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild S1PR2 57 35 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild EPHX2 36 43 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild HDAC9 22 42 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild AKR1C3 44 40 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild ASAH1 102 41 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild KDM4E 28 47 CCCCCCCCNC(=O)c1cccc(C(=O)O)c1 ZINC000147288937 CG For-Sale Mild KCNK3 49 34 Cc1cccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)c1 ZINC000147288957 CD On-Demand Anodyne FBP1 29 47 CCNc1nc(C)cc(Oc2ccccc2[C@@H](C)CC)n1 ZINC000147288965 CJ For-Sale Anodyne AO-ACHE 0 40 COC(=O)c1cc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)ccc1Cl ZINC000147288988 EH On-Demand Anodyne EPHX2 40 41 CC[C@@H]1CN(C(=O)CCC2CCCC2)CC[C@H]1N ZINC000147288989 CF On-Demand Anodyne F2R 22 40 CC[C@@H]1CN(C(=O)CCC2CCCC2)CC[C@H]1N ZINC000147288989 CF On-Demand Anodyne GNAI3 0 40 CC1(C)C[C@H]2C3=CC[C@@H]4[C@@]5(C)CC[C@@H](O)C(C)(C)[C@@H]5CC[C@@]4(C)[C@]3(C)CC[C@@]2(CO)[C@@H](O)[C@@H]1O ZINC000147289081 JK Annotated Anodyne PTPN2 58 58 CC1(C)C[C@H]2C3=CC[C@@H]4[C@@]5(C)CC[C@@H](O)C(C)(C)[C@@H]5CC[C@@]4(C)[C@]3(C)CC[C@@]2(CO)[C@@H](O)[C@@H]1O ZINC000147289081 JK Annotated Anodyne IKBKB 0 56 CC1(C)C[C@H]2C3=CC[C@@H]4[C@@]5(C)CC[C@@H](O)C(C)(C)[C@@H]5CC[C@@]4(C)[C@]3(C)CC[C@@]2(CO)[C@@H](O)[C@@H]1O ZINC000147289081 JK Annotated Anodyne HSD11B2 27 42 CC1(C)C[C@H]2C3=CC[C@@H]4[C@@]5(C)CC[C@@H](O)C(C)(C)[C@@H]5CC[C@@]4(C)[C@]3(C)CC[C@@]2(CO)[C@@H](O)[C@@H]1O ZINC000147289081 JK Annotated Anodyne PTPN1 42 58 CC1(C)C[C@H]2C3=CC[C@@H]4[C@@]5(C)CC[C@@H](O)C(C)(C)[C@@H]5CC[C@@]4(C)[C@]3(C)CC[C@@]2(CO)[C@@H](O)[C@@H]1O ZINC000147289081 JK Annotated Anodyne PTPN6 19 43 CC1(C)C[C@H]2C3=CC[C@@H]4[C@@]5(C)CC[C@@H](O)C(C)(C)[C@@H]5CC[C@@]4(C)[C@]3(C)CC[C@@]2(CO)[C@@H](O)[C@@H]1O ZINC000147289081 JK Annotated Anodyne PA2B1_NAJME 0 56 CC1(C)C[C@H]2C3=CC[C@@H]4[C@@]5(C)CC[C@@H](O)C(C)(C)[C@@H]5CC[C@@]4(C)[C@]3(C)CC[C@@]2(CO)[C@@H](O)[C@@H]1O ZINC000147289081 JK Annotated Anodyne PA2BA_PROFL 0 56 CC1(C)C[C@H]2C3=CC[C@@H]4[C@@]5(C)CC[C@@H](O)C(C)(C)[C@@H]5CC[C@@]4(C)[C@]3(C)CC[C@@]2(CO)[C@@H](O)[C@@H]1O ZINC000147289081 JK Annotated Anodyne PA2A1_ECHCA 0 56 CC1(C)C[C@H]2C3=CC[C@@H]4[C@@]5(C)CC[C@@H](O)C(C)(C)[C@@H]5CC[C@@]4(C)[C@]3(C)CC[C@@]2(CO)[C@@H](O)[C@@H]1O ZINC000147289081 JK Annotated Anodyne CD81 0 58 CCCCCCCCNC(=O)c1ccc(C(=O)O)c(C)n1 ZINC000147289138 CG For-Sale Mild ASAH1 90 36 Cc1ccc(C(=O)N[C@H]2CCC[C@@H]2C(=O)O)cc1Br ZINC000147289144 EF For-Sale Anodyne MAPK14 41 39 Cc1ccc(C(=O)N[C@H]2CCC[C@@H]2C(=O)O)cc1Br ZINC000147289144 EF For-Sale Anodyne ADAM17 23 44 Cc1ccc(C(=O)N[C@H]2CCC[C@@H]2C(=O)O)cc1Br ZINC000147289144 EF For-Sale Anodyne MAPK13 41 38 CN(C)C(=O)NCCNC(=O)c1cccc2[nH]ccc12 ZINC000147289147 CD On-Demand Anodyne HPGDS 20 40 Cc1cccc(S(=O)(=O)NC[C@H](C)CC(=O)O)c1 ZINC000147289182 CD On-Demand Anodyne FBP1 29 47 CC[C@H]1CN(C(=O)CCC2CCCC2)CC[C@H]1N ZINC000147289199 CF On-Demand Anodyne F2R 22 40 CC[C@H]1CN(C(=O)CCC2CCCC2)CC[C@H]1N ZINC000147289199 CF On-Demand Anodyne GNAI3 0 40 COC(=O)c1cc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)ccc1Cl ZINC000147289221 EH On-Demand Anodyne EPHX2 40 41 CCNc1nc(Cl)nc(Oc2ccccc2[C@H](C)CC)n1 ZINC000147289223 DI For-Sale Anodyne Q31945_CHEAL 0 43 CCNc1nc(Cl)nc(Oc2ccccc2[C@H](C)CC)n1 ZINC000147289223 DI For-Sale Anodyne AO-ACHE 0 40 CCNc1nc(Cl)nc(Oc2ccccc2[C@H](C)CC)n1 ZINC000147289223 DI For-Sale Anodyne PPX1 0 43 CS(=O)(=O)c1cc(C(=O)N2CCC[C@@H]2CCc2ccccc2)cc([N+](=O)[O-])c1 ZINC000147289267 HG On-Demand Bother PREP 61 34 CS(=O)(=O)c1cc(C(=O)N2CCC[C@@H]2CCc2ccccc2)cc([N+](=O)[O-])c1 ZINC000147289267 HG On-Demand Bother WNT3 40 31 CC(C)CCCCNCc1ccccc1OC(F)(F)F ZINC000147289271 CJ For-Sale Anodyne PHES 0 41 CC(C)CCCCNCc1ccccc1OC(F)(F)F ZINC000147289271 CJ For-Sale Anodyne LEF 57 37 CC(C)CCCCNCc1ccccc1OC(F)(F)F ZINC000147289271 CJ For-Sale Anodyne GPM3 0 51 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild THRA 42 32 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild DRD3 35 41 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild FOLH1 23 44 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild RARB 24 45 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild THRB 22 47 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild KCNQ1 0 45 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild PLA2G4A 26 41 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild PLA2G4B 61 41 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild P4HTM 0 50 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild EPHX2 15 41 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild P4HA1 0 50 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild ASAH1 92 37 CCCCCCCCNC(=O)c1ccc(C(=O)O)cn1 ZINC000147289307 CF For-Sale Mild ACAT 0 41 COc1ccccc1N1CCC(NCc2cc(OC)c(OC)c(OC)c2)CC1 ZINC000147289317 GG On-Demand Anodyne HTR1A 97 46 COc1ccccc1N1CCC(NCc2cc(OC)c(OC)c(OC)c2)CC1 ZINC000147289317 GG On-Demand Anodyne DRD2 82 46 COc1ccccc1N1CCC(NCc2cc(OC)c(OC)c(OC)c2)CC1 ZINC000147289317 GG On-Demand Anodyne DRD1 22 43 COc1ccccc1N1CCC(NCc2cc(OC)c(OC)c(OC)c2)CC1 ZINC000147289317 GG On-Demand Anodyne DRD4 47 43 COc1ccccc1N1CCC(NCc2cc(OC)c(OC)c(OC)c2)CC1 ZINC000147289317 GG On-Demand Anodyne ADRA1D 94 43 COc1ccccc1N1CCC(NCc2cc(OC)c(OC)c(OC)c2)CC1 ZINC000147289317 GG On-Demand Anodyne HTR2A 23 43 COc1ccccc1N1CCC(NCc2cc(OC)c(OC)c(OC)c2)CC1 ZINC000147289317 GG On-Demand Anodyne ADRA1A 81 43 COc1ccccc1N1CCC(NCc2cc(OC)c(OC)c(OC)c2)CC1 ZINC000147289317 GG On-Demand Anodyne ADRA1B 77 43 COc1ccccc1N1CCC(NCc2cc(OC)c(OC)c(OC)c2)CC1 ZINC000147289317 GG On-Demand Anodyne DRD3 75 46 COc1ccccc1N1CCC(NCc2cc(OC)c(OC)c(OC)c2)CC1 ZINC000147289317 GG On-Demand Anodyne HTR7 54 45 Cc1csc(CNC(=O)[C@@H]2CCC(=O)N(Cc3ccccc3)[C@@H]2c2ccccc2)n1 ZINC000147289329 HI On-Demand Anodyne P2RX7 27 44 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne ACE 15 41 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne ACHE 28 41 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne MME 20 40 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne TACR1 0 42 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne TPR 17 64 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne MC4R 41 44 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne TACR2 22 40 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne CCKAR 64 46 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne BRS3 24 46 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne NMBR 47 31 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne MMP2 22 40 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne MMP8 32 40 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne GRIA1 25 54 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne MMP14 64 38 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne GRPR 54 32 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne ECE1 46 39 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne SSTR3 22 41 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne MMP11 45 31 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne CCKBR 53 40 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne GHSR 40 38 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne MMP9 19 43 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne MC1R 49 38 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne MMP1 21 42 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne NPR 29 40 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne SLC15A2 0 44 CN(C)C(=O)NCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147289362 CD On-Demand Anodyne KISS1R 59 33 Cc1ccc(C(=O)N[C@@H]2CCC[C@H]2C(=O)O)cc1Br ZINC000147289382 EF For-Sale Anodyne MAPK14 41 39 Cc1ccc(C(=O)N[C@@H]2CCC[C@H]2C(=O)O)cc1Br ZINC000147289382 EF For-Sale Anodyne ADAM17 23 44 Cc1ccc(C(=O)N[C@@H]2CCC[C@H]2C(=O)O)cc1Br ZINC000147289382 EF For-Sale Anodyne MAPK13 41 38 C[C@H](CNS(=O)(=O)c1ccc(Cl)cc1[N+](=O)[O-])CC(=O)O ZINC000147289423 ED On-Demand Bother COLA 66 39 Cc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1Br ZINC000147289425 FE On-Demand Anodyne DHODH 19 47 Cc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1Br ZINC000147289425 FE On-Demand Anodyne TNK2 16 41 CCNc1nc(Cl)nc(Oc2ccccc2[C@@H](C)CC)n1 ZINC000147289432 DI For-Sale Anodyne Q31945_CHEAL 0 43 CCNc1nc(Cl)nc(Oc2ccccc2[C@@H](C)CC)n1 ZINC000147289432 DI For-Sale Anodyne AO-ACHE 0 40 CCNc1nc(Cl)nc(Oc2ccccc2[C@@H](C)CC)n1 ZINC000147289432 DI For-Sale Anodyne PPX1 0 43 c1ccc2c(c1)CCCCCNC2 ZINC000147289442 AF For-Sale Anodyne PNMT 33 41 CS(=O)(=O)c1cc(C(=O)N2CCC[C@H]2CCc2ccccc2)cc([N+](=O)[O-])c1 ZINC000147289455 HG On-Demand Bother PREP 61 34 CS(=O)(=O)c1cc(C(=O)N2CCC[C@H]2CCc2ccccc2)cc([N+](=O)[O-])c1 ZINC000147289455 HG On-Demand Bother WNT3 40 31 CCCCCCCCNC(=O)[C@@H]1CCC[C@H](C(=O)O)C1 ZINC000147289488 CG For-Sale Mild EPHX2 52 41 CCCCCCCCNC(=O)[C@@H]1CCC[C@H](C(=O)O)C1 ZINC000147289488 CG For-Sale Mild TPP2 31 42 CCCCCCCCNC(=O)[C@@H]1CCC[C@H](C(=O)O)C1 ZINC000147289488 CG For-Sale Mild ASAH1 57 33 CC(C)c1ccccc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147289502 CE For-Sale Anodyne SOAT1 24 40 CC(C)c1ccccc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147289502 CE For-Sale Anodyne ACAT 0 50 COC(=O)c1cc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)ccc1Cl ZINC000147289533 HH On-Demand Anodyne NOS2 51 32 COC(=O)c1cc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)ccc1Cl ZINC000147289533 HH On-Demand Anodyne ROCK2 17 42 Cc1csc(CNC(=O)[C@H]2CCC(=O)N(Cc3ccccc3)[C@@H]2c2ccccc2)n1 ZINC000147289551 HI On-Demand Anodyne P2RX7 27 44 CCC(C)(C)NC(=O)COc1ccc(Cl)cc1S(N)(=O)=O ZINC000147289589 ED For-Sale Anodyne PTGDR2 39 40 Cc1ccc(C(=O)N[C@H]2CCC[C@H]2C(=O)O)cc1Br ZINC000147289595 EF On-Demand Anodyne MAPK14 40 39 Cc1ccc(C(=O)N[C@H]2CCC[C@H]2C(=O)O)cc1Br ZINC000147289595 EF On-Demand Anodyne MAPK13 41 38 Cc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1Br ZINC000147289617 FE On-Demand Anodyne DHODH 19 47 Cc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1Br ZINC000147289617 FE On-Demand Anodyne TNK2 17 41 C[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1[N+](=O)[O-])CC(=O)O ZINC000147289619 ED On-Demand Bother COLA 66 39 O=C(O)/C=C/c1cc(F)ccc1Oc1ccc(Cl)c(F)c1 ZINC000147289653 DJ For-Sale Anodyne PTGER3 27 42 CCCCCCCCNC(=O)[C@H]1CCC[C@H](C(=O)O)C1 ZINC000147289680 CG For-Sale Mild EPHX2 52 41 CCCCCCCCNC(=O)[C@H]1CCC[C@H](C(=O)O)C1 ZINC000147289680 CG For-Sale Mild TPP2 31 42 CCCCCCCCNC(=O)[C@H]1CCC[C@H](C(=O)O)C1 ZINC000147289680 CG For-Sale Mild ASAH1 57 33 CC[C@@H](C)c1ccccc1Oc1cc(NC)nc(SC)n1 ZINC000147289686 DJ For-Sale Anodyne AO-ACHE 0 42 COc1ccc(Cl)cc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147289760 DD For-Sale Anodyne CYSP_TRYCR 0 41 COc1ccc(Cl)cc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147289760 DD For-Sale Anodyne NTSR2 22 41 COc1ccc(Cl)cc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147289760 DD For-Sale Anodyne COLA 62 36 COc1ccc(Cl)cc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147289760 DD For-Sale Anodyne CPT1A 60 33 COc1ccc(Cl)cc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147289760 DD For-Sale Anodyne CPT2 42 31 COc1ccc(Cl)cc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147289760 DD For-Sale Anodyne CPT1B 46 31 COc1ccc(Cl)cc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147289760 DD For-Sale Anodyne RBP4 19 44 Cc1csc(CNC(=O)[C@@H]2CCC(=O)N(Cc3ccccc3)[C@H]2c2ccccc2)n1 ZINC000147289761 HI On-Demand Anodyne P2RX7 27 44 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne HTR1A 102 50 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne DRD2 88 45 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne TSHR 67 36 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne DRD4 50 44 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne ADRA1D 90 42 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne HTR1D 20 50 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne HTR1B 26 50 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne HTR2A 24 40 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne ADRA1A 80 42 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne ADRA1B 72 42 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne DRD3 80 45 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne TACR1 15 44 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne HTR7 59 45 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne NPY1R 23 45 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne NPY2R 33 40 COc1ccccc1N1CCC(NCc2ccc(NC(C)=O)cc2)CC1 ZINC000147289779 FG On-Demand Anodyne MCHR1 15 41 C[C@H](CNS(=O)(=O)c1ccc(C(N)=O)cc1)CC(=O)O ZINC000147289807 DC On-Demand Anodyne CA2 32 43 C[C@H](CNS(=O)(=O)c1ccc(C(N)=O)cc1)CC(=O)O ZINC000147289807 DC On-Demand Anodyne CA1 16 41 C[C@H](CNS(=O)(=O)c1ccc(C(N)=O)cc1)CC(=O)O ZINC000147289807 DC On-Demand Anodyne CA4 23 40 C[C@H](CNS(=O)(=O)c1ccc(C(N)=O)cc1)CC(=O)O ZINC000147289807 DC On-Demand Anodyne LIMK2 45 40 CCCCCCCCNC(=O)[C@@H]1CCC[C@@H](C(=O)O)C1 ZINC000147289864 CG For-Sale Mild EPHX2 52 41 CCCCCCCCNC(=O)[C@@H]1CCC[C@@H](C(=O)O)C1 ZINC000147289864 CG For-Sale Mild TPP2 31 42 CCCCCCCCNC(=O)[C@@H]1CCC[C@@H](C(=O)O)C1 ZINC000147289864 CG For-Sale Mild ASAH1 57 33 CC[C@H](C)c1ccccc1Oc1cc(NC)nc(SC)n1 ZINC000147289865 DJ For-Sale Anodyne AO-ACHE 0 42 Cc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1[N+](=O)[O-] ZINC000147289866 FH For-Sale Reactive L3MBTL1 0 44 N[C@@H](Cc1cn(N=O)c2ccccc12)C(=O)O ZINC000147289891 BD For-Sale Anodyne CACNA2D1 35 45 O=C(O)C1(NCc2ccccc2[N+](=O)[O-])CCC1 ZINC000147289981 CD For-Sale Bother COLA 116 37 O=C(O)C1(NCc2ccccc2[N+](=O)[O-])CCC1 ZINC000147289981 CD For-Sale Bother PQSD 0 46 Cc1csc(CNC(=O)[C@H]2CCC(=O)N(Cc3ccccc3)[C@H]2c2ccccc2)n1 ZINC000147289983 HI On-Demand Anodyne P2RX7 27 44 C[C@@H](CNS(=O)(=O)c1ccc(C(N)=O)cc1)CC(=O)O ZINC000147290013 DC On-Demand Anodyne CA2 32 43 C[C@@H](CNS(=O)(=O)c1ccc(C(N)=O)cc1)CC(=O)O ZINC000147290013 DC On-Demand Anodyne CA1 16 41 C[C@@H](CNS(=O)(=O)c1ccc(C(N)=O)cc1)CC(=O)O ZINC000147290013 DC On-Demand Anodyne CA4 23 40 C[C@@H](CNS(=O)(=O)c1ccc(C(N)=O)cc1)CC(=O)O ZINC000147290013 DC On-Demand Anodyne LIMK2 45 40 Cc1cc(C(=O)N2CCN(Cc3ccc(Cl)cc3)CC2)cc([N+](=O)[O-])c1 ZINC000147290032 FH On-Demand Bother LSS 22 54 Cc1cc(C(=O)N2CCN(Cc3ccc(Cl)cc3)CC2)cc([N+](=O)[O-])c1 ZINC000147290032 FH On-Demand Bother FAAH 17 43 Cc1cc(C(=O)N2CCN(Cc3ccc(Cl)cc3)CC2)cc([N+](=O)[O-])c1 ZINC000147290032 FH On-Demand Bother KCNJ1 25 41 COc1ccccc1N1CCC(NCc2ccc(Br)cc2)CC1 ZINC000147290034 GI On-Demand Anodyne HTR1A 89 49 COc1ccccc1N1CCC(NCc2ccc(Br)cc2)CC1 ZINC000147290034 GI On-Demand Anodyne DRD2 73 46 COc1ccccc1N1CCC(NCc2ccc(Br)cc2)CC1 ZINC000147290034 GI On-Demand Anodyne DRD1 17 41 COc1ccccc1N1CCC(NCc2ccc(Br)cc2)CC1 ZINC000147290034 GI On-Demand Anodyne DRD4 43 43 COc1ccccc1N1CCC(NCc2ccc(Br)cc2)CC1 ZINC000147290034 GI On-Demand Anodyne ADRA1D 78 43 COc1ccccc1N1CCC(NCc2ccc(Br)cc2)CC1 ZINC000147290034 GI On-Demand Anodyne HTR2A 19 41 COc1ccccc1N1CCC(NCc2ccc(Br)cc2)CC1 ZINC000147290034 GI On-Demand Anodyne ADRA1A 68 42 COc1ccccc1N1CCC(NCc2ccc(Br)cc2)CC1 ZINC000147290034 GI On-Demand Anodyne ADRA1B 62 43 COc1ccccc1N1CCC(NCc2ccc(Br)cc2)CC1 ZINC000147290034 GI On-Demand Anodyne DRD3 69 46 COc1ccccc1N1CCC(NCc2ccc(Br)cc2)CC1 ZINC000147290034 GI On-Demand Anodyne HTR7 51 45 CCCCCCCCNC(=O)[C@H]1CCC[C@@H](C(=O)O)C1 ZINC000147290068 CG For-Sale Mild EPHX2 52 41 CCCCCCCCNC(=O)[C@H]1CCC[C@@H](C(=O)O)C1 ZINC000147290068 CG For-Sale Mild TPP2 31 42 CCCCCCCCNC(=O)[C@H]1CCC[C@@H](C(=O)O)C1 ZINC000147290068 CG For-Sale Mild ASAH1 57 33 Cc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1[N+](=O)[O-] ZINC000147290096 FH For-Sale Reactive L3MBTL1 0 44 N[C@H](Cc1cn(N=O)c2ccccc12)C(=O)O ZINC000147290105 BD For-Sale Anodyne CACNA2D1 35 45 N[C@H](Cc1cn(N=O)c2ccccc12)C(=O)O ZINC000147290105 BD For-Sale Anodyne GRIK1 27 41 c1ccc(CNc2nc(Nc3ccccc3)nc(N3CCNCC3)n2)cc1 ZINC000147290178 FF In-Stock Anodyne DNAB 0 46 c1ccc(CNc2nc(Nc3ccccc3)nc(N3CCNCC3)n2)cc1 ZINC000147290178 FF In-Stock Anodyne KHK 0 48 COCc1nc(C(=O)N2CCN(Cc3ccc(Cl)cc3)CC2)cs1 ZINC000147290284 FF On-Demand Anodyne LSS 20 47 COCc1nc(C(=O)N2CCN(Cc3ccc(Cl)cc3)CC2)cs1 ZINC000147290284 FF On-Demand Anodyne FAAH 16 40 COCc1nc(C(=O)N2CCN(Cc3ccc(Cl)cc3)CC2)cs1 ZINC000147290284 FF On-Demand Anodyne TRPC6 52 43 COCc1nc(C(=O)N2CCN(Cc3ccc(Cl)cc3)CC2)cs1 ZINC000147290284 FF On-Demand Anodyne TRPC3 24 43 COc1ccccc1N1CCC(NCc2cccc(Br)c2)CC1 ZINC000147290288 GI On-Demand Anodyne HTR1A 88 45 COc1ccccc1N1CCC(NCc2cccc(Br)c2)CC1 ZINC000147290288 GI On-Demand Anodyne DRD2 76 46 COc1ccccc1N1CCC(NCc2cccc(Br)c2)CC1 ZINC000147290288 GI On-Demand Anodyne DRD1 17 41 COc1ccccc1N1CCC(NCc2cccc(Br)c2)CC1 ZINC000147290288 GI On-Demand Anodyne DRD4 48 46 COc1ccccc1N1CCC(NCc2cccc(Br)c2)CC1 ZINC000147290288 GI On-Demand Anodyne ADRA1D 78 43 COc1ccccc1N1CCC(NCc2cccc(Br)c2)CC1 ZINC000147290288 GI On-Demand Anodyne HTR2A 20 41 COc1ccccc1N1CCC(NCc2cccc(Br)c2)CC1 ZINC000147290288 GI On-Demand Anodyne ADRA1A 67 43 COc1ccccc1N1CCC(NCc2cccc(Br)c2)CC1 ZINC000147290288 GI On-Demand Anodyne ADRA1B 63 43 COc1ccccc1N1CCC(NCc2cccc(Br)c2)CC1 ZINC000147290288 GI On-Demand Anodyne DRD3 72 46 COc1ccccc1N1CCC(NCc2cccc(Br)c2)CC1 ZINC000147290288 GI On-Demand Anodyne HTR7 51 43 COc1ccccc1N1CCC(NCc2cccc(Br)c2)CC1 ZINC000147290288 GI On-Demand Anodyne NPY1R 17 41 CCCCCCCCNC(=O)Cn1cc(C(=O)O)nn1 ZINC000147290298 CD For-Sale Mild ASAH1 102 38 O=C(O)/C=C/c1ccc(Br)cc1Oc1ccc(Cl)c(F)c1 ZINC000147290346 FK For-Sale Anodyne PTGER3 16 41 CN(C)NC(=O)c1ccnc(CN)c1 ZINC000147290386 AB For-Sale Reactive KDM4E 31 41 COc1ccccc1N1CCC(NCc2cccc(OC)c2OC)CC1 ZINC000147290505 FG On-Demand Anodyne HTR1A 97 46 COc1ccccc1N1CCC(NCc2cccc(OC)c2OC)CC1 ZINC000147290505 FG On-Demand Anodyne DRD2 76 46 COc1ccccc1N1CCC(NCc2cccc(OC)c2OC)CC1 ZINC000147290505 FG On-Demand Anodyne DRD1 16 43 COc1ccccc1N1CCC(NCc2cccc(OC)c2OC)CC1 ZINC000147290505 FG On-Demand Anodyne DRD4 44 43 COc1ccccc1N1CCC(NCc2cccc(OC)c2OC)CC1 ZINC000147290505 FG On-Demand Anodyne ADRA1D 89 43 COc1ccccc1N1CCC(NCc2cccc(OC)c2OC)CC1 ZINC000147290505 FG On-Demand Anodyne HTR2A 22 46 COc1ccccc1N1CCC(NCc2cccc(OC)c2OC)CC1 ZINC000147290505 FG On-Demand Anodyne ADRA1A 77 43 COc1ccccc1N1CCC(NCc2cccc(OC)c2OC)CC1 ZINC000147290505 FG On-Demand Anodyne ADRA1B 74 43 COc1ccccc1N1CCC(NCc2cccc(OC)c2OC)CC1 ZINC000147290505 FG On-Demand Anodyne DRD3 68 46 COc1ccccc1N1CCC(NCc2cccc(OC)c2OC)CC1 ZINC000147290505 FG On-Demand Anodyne TACR1 22 43 COc1ccccc1N1CCC(NCc2cccc(OC)c2OC)CC1 ZINC000147290505 FG On-Demand Anodyne HTR7 56 46 Cc1ccc(C(=O)Nc2ccc(NC(C)(C)C)cc2)cc1 ZINC000147290518 CI For-Sale Anodyne TRPV1 26 54 Cc1ccc(C(=O)Nc2ccc(NC(C)(C)C)cc2)cc1 ZINC000147290518 CI For-Sale Anodyne ECR 32 42 Cc1ccc(C(=O)Nc2ccc(NC(C)(C)C)cc2)cc1 ZINC000147290518 CI For-Sale Anodyne PRNP 76 49 Cc1ccc(C(=O)Nc2ccc(NC(C)(C)C)cc2)cc1 ZINC000147290518 CI For-Sale Anodyne NR1H4 16 43 Cc1ccc(C(=O)Nc2ccc(NC(C)(C)C)cc2)cc1 ZINC000147290518 CI For-Sale Anodyne ACR 19 40 Cc1ccc(C(=O)Nc2ccc(NC(C)(C)C)cc2)cc1 ZINC000147290518 CI For-Sale Anodyne MCHR1 16 46 Cc1ccc(C(=O)Nc2ccc(NC(C)(C)C)cc2)cc1 ZINC000147290518 CI For-Sale Anodyne MAP3K5 64 43 Cc1ccc(C(=O)Nc2ccc(NC(C)(C)C)cc2)cc1 ZINC000147290518 CI For-Sale Anodyne NAMPT 16 47 Cc1ccc(C(=O)Nc2ccc(NC(C)(C)C)cc2)cc1 ZINC000147290518 CI For-Sale Anodyne KCNK3 96 47 Cc1ccc(C(=O)Nc2ccc(NC(C)(C)C)cc2)cc1 ZINC000147290518 CI For-Sale Anodyne KCNK9 53 40 CCCCCCCCNC(=O)c1ccc(C(=O)O)s1 ZINC000147290519 CH For-Sale Mild S1PR2 41 35 CCCCCCCCNC(=O)c1ccc(C(=O)O)s1 ZINC000147290519 CH For-Sale Mild EPHX2 33 40 CCCCCCCCNC(=O)c1ccc(C(=O)O)s1 ZINC000147290519 CH For-Sale Mild ASAH1 106 42 O=C(O)/C=C/c1c(Cl)cccc1Oc1ccc(Cl)c(F)c1 ZINC000147290568 EK For-Sale Anodyne PTGER3 25 44 CN(C)C(=O)NCCNC(=O)c1c[nH]c2ccccc12 ZINC000147290569 CD For-Sale Anodyne GABRA1 15 46 CN(C)C(=O)NCCNC(=O)c1c[nH]c2ccccc12 ZINC000147290569 CD For-Sale Anodyne TPR 17 43 CN(C)C(=O)NCCNC(=O)c1c[nH]c2ccccc12 ZINC000147290569 CD For-Sale Anodyne CCKAR 15 43 CN(C)C(=O)NCCNC(=O)c1c[nH]c2ccccc12 ZINC000147290569 CD For-Sale Anodyne CFTR 37 43 CN(C)NC(=O)CNC(C)(C)C ZINC000147290628 AB For-Sale Reactive KDM7A 0 45 CC(C)(C)c1ccc(CNC2(C(=O)O)CCC2)cc1 ZINC000147290631 CG For-Sale Anodyne TRPV1 27 43 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1c(F)cccc1F ZINC000147290662 CD On-Demand Anodyne TNK2 23 41 O=C(O)c1cnn2c1N[C@H](c1ccccc1)CC21CCCCC1 ZINC000147290695 DH For-Sale Anodyne CASR 67 50 CCCCCCCCNC(=O)c1cccn1CC(=O)O ZINC000147290741 CF For-Sale Mild ASAH1 105 43 CCCCCCCCNC(=O)c1cccn1CC(=O)O ZINC000147290741 CF For-Sale Mild ACAT 0 46 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne RARA 15 40 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne TRPV1 22 63 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne PRNP 66 45 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne NR1H4 15 41 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne ACR 57 47 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne SCN10A 36 43 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne CA9 15 42 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne MAP3K5 53 38 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne SHH 57 39 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne NOD1 15 40 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne NOD2 43 40 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne KCNK3 87 43 Cc1ccc(C(=O)Nc2ccc(OC(C)(C)C)cc2)cc1 ZINC000147290743 CI On-Demand Anodyne KCNK9 51 38 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne HTR1A 91 49 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne DRD2 75 49 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne DRD1 19 44 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne DRD4 44 47 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne ADRA1D 81 49 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne HTR2A 24 44 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne ADRA1A 69 49 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne ADRA1B 65 49 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne DRD3 70 44 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne AVPR1B 15 42 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne TACR1 19 48 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne HTR7 56 45 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)c(OC)c1 ZINC000147290752 FG On-Demand Anodyne EBP 25 40 CCc1cccc(C)c1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147290829 CE For-Sale Anodyne ACAT 0 42 CC(C)NCCC(=O)NN(C)C ZINC000147290859 AB For-Sale Reactive KDM7A 0 52 O=C(NC[C@H]1CCCCO1)C(=O)Nc1c(F)cccc1F ZINC000147290877 CD On-Demand Anodyne TNK2 23 41 O=C(NCc1cccc(NC(=O)[C@@H]2CCCO2)c1)Nc1ccc(-n2cccn2)nc1 ZINC000147290898 HF On-Demand Anodyne NAMPT 42 38 O=C(O)c1cnn2c1N[C@@H](c1ccccc1)CC21CCCCC1 ZINC000147290902 DH For-Sale Anodyne CASR 67 50 CCCCCCCCNC(=O)c1cccc(C(=O)O)n1 ZINC000147290928 CF For-Sale Mild HTR2A 19 41 CCCCCCCCNC(=O)c1cccc(C(=O)O)n1 ZINC000147290928 CF For-Sale Mild HTR2C 21 41 CCCCCCCCNC(=O)c1cccc(C(=O)O)n1 ZINC000147290928 CF For-Sale Mild DRD3 31 42 CCCCCCCCNC(=O)c1cccc(C(=O)O)n1 ZINC000147290928 CF For-Sale Mild P2RY12 37 43 CCCCCCCCNC(=O)c1cccc(C(=O)O)n1 ZINC000147290928 CF For-Sale Mild TBXA2R 0 41 CCCCCCCCNC(=O)c1cccc(C(=O)O)n1 ZINC000147290928 CF For-Sale Mild FAAH 28 47 CCCCCCCCNC(=O)c1cccc(C(=O)O)n1 ZINC000147290928 CF For-Sale Mild PA2A1_NAJMO 0 44 CCCCCCCCNC(=O)c1cccc(C(=O)O)n1 ZINC000147290928 CF For-Sale Mild ASAH1 99 38 CCCCCCCCNC(=O)c1cccc(C(=O)O)n1 ZINC000147290928 CF For-Sale Mild ACAT 0 49 CCCCCCCCNC(=O)c1cccc(C(=O)O)n1 ZINC000147290928 CF For-Sale Mild PSBA 0 40 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne HTR1A 97 51 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne DRD2 81 49 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne DRD1 20 44 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne DRD4 47 47 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne ADRA1D 86 49 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne HTR2A 26 44 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne ADRA1A 74 49 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne ADRA1B 68 49 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne DRD3 72 44 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne TACR1 34 50 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne HTR7 57 45 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne SIGMAR1 17 53 COc1ccc(OC)c(CNC2CCN(c3ccccc3OC)CC2)c1 ZINC000147290967 FG On-Demand Anodyne EBP 31 40 O=C(O)/C=C/c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147290984 EK For-Sale Anodyne NR0B2 0 40 CC[C@@H](C)c1ccccc1Oc1nc(Cl)nc(NC)n1 ZINC000147291006 CH For-Sale Anodyne AO-ACHE 0 44 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne OPRM1 28 45 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne OPRD1 32 41 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CACNA2D1 23 51 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne MME 56 43 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne LTA4H 19 44 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne ANPEP 84 51 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne RNPEP 48 57 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne KLK3 71 34 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CTSB 39 43 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CYSP_TRYCR 41 38 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CTSK 33 44 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CTSL 27 44 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne SLC15A1 0 48 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CAPNS1 62 37 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne MMP2 28 46 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne MMP3 54 42 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne MMP8 19 51 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne HLA-DRB1 44 35 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne FAAH 64 41 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne PAM 0 42 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne S1PR2 20 40 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne DNPEP 0 40 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CAPN1 79 45 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne MMP9 15 46 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CASP1 23 44 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CES1 64 40 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CAPN2 106 41 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne DPP7 15 40 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne LAP3 78 48 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CTSC 19 41 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne PROTEASE 0 43 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne MMP1 24 46 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne FPR1 56 41 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne NPR 90 39 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne AMP1_PLAFQ 58 51 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne AMPX_VIBPR 0 44 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne KIF11 32 42 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne DAGLA 22 41 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne VM1B1_BOTAS 0 46 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne CES1D 44 31 CC(C)C[C@@H](N)C(=O)CCCc1ccccc1 ZINC000147291043 BF For-Sale Anodyne GPR88 0 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(F)c(F)c1 ZINC000147291123 CD On-Demand Anodyne ENV 46 38 CCCCCCCCNC(=O)C1CCC(C(=O)O)CC1 ZINC000147291133 CG For-Sale Mild EPHX2 53 42 CCCCCCCCNC(=O)C1CCC(C(=O)O)CC1 ZINC000147291133 CG For-Sale Mild TPP2 31 42 CCCCCCCCNC(=O)C1CCC(C(=O)O)CC1 ZINC000147291133 CG For-Sale Mild ASAH1 85 36 O=C(NCc1cccc(NC(=O)[C@H]2CCCO2)c1)Nc1ccc(-n2cccn2)nc1 ZINC000147291137 HF On-Demand Anodyne NAMPT 42 38 CC[C@H](C)c1ccccc1Oc1nc(Cl)nc(NC)n1 ZINC000147291196 CH For-Sale Anodyne AO-ACHE 0 44 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne OPRM1 28 45 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne OPRD1 32 41 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CACNA2D1 23 51 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne MME 56 43 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne LTA4H 19 44 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne ANPEP 84 51 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne RNPEP 48 57 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne KLK3 71 34 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CTSB 39 43 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CYSP_TRYCR 41 38 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CTSK 33 44 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CTSL 27 44 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne SLC15A1 0 48 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CAPNS1 62 37 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne MMP2 28 46 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne MMP3 54 42 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne MMP8 19 51 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne HLA-DRB1 44 35 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne FAAH 64 41 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne PAM 0 42 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne S1PR2 20 40 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne DNPEP 0 40 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CAPN1 79 45 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne MMP9 15 46 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CASP1 23 44 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CES1 64 40 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CAPN2 106 41 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne DPP7 15 40 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne LAP3 78 48 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CTSC 19 41 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne PROTEASE 0 43 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne MMP1 24 46 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne FPR1 56 41 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne NPR 90 39 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne AMP1_PLAFQ 58 51 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne AMPX_VIBPR 0 44 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne KIF11 32 42 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne DAGLA 22 41 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne VM1B1_BOTAS 0 46 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne CES1D 44 31 CC(C)C[C@H](N)C(=O)CCCc1ccccc1 ZINC000147291261 BF For-Sale Anodyne GPR88 0 40 O=C(O)C1(NCCOc2ccc(Cl)cc2Cl)CCC1 ZINC000147291286 DF For-Sale Anodyne S1PR4 34 45 CN(C)C(=O)NCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147291297 ED On-Demand Reactive CA2 23 44 CN(C)C(=O)NCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147291297 ED On-Demand Reactive TBXA2R 50 38 CN(C)C(=O)NCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147291297 ED On-Demand Reactive CA1 22 44 CN(C)C(=O)NCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147291297 ED On-Demand Reactive CA4 16 41 CN(C)C(=O)NCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147291297 ED On-Demand Reactive ALOX15 46 34 CN(C)C(=O)NCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147291297 ED On-Demand Reactive CYNT 18 41 CN(C)C(=O)NCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147291297 ED On-Demand Reactive A6YCJ1_9METZ 22 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(F)c(F)c1 ZINC000147291333 CD On-Demand Anodyne ENV 46 38 CCCCCCCCNC(=O)C1(C(=O)O)CCC1 ZINC000147291342 CF For-Sale Mild EPHX2 57 44 CCCCCCCCNC(=O)C1(C(=O)O)CCC1 ZINC000147291342 CF For-Sale Mild CPT1 0 41 CCCCCCCCNC(=O)C1(C(=O)O)CCC1 ZINC000147291342 CF For-Sale Mild GNAI1 0 43 CCCCCCCCNC(=O)C1(C(=O)O)CCC1 ZINC000147291342 CF For-Sale Mild GNAI3 0 43 CCCCCCCCNC(=O)C1(C(=O)O)CCC1 ZINC000147291342 CF For-Sale Mild GNAO1 0 43 CCCCCCCCNC(=O)C1(C(=O)O)CCC1 ZINC000147291342 CF For-Sale Mild ASAH1 83 33 O=C(NC[C@@H]1CCCOC1)c1ccc2c(c1)COC2 ZINC000147291354 CD On-Demand Anodyne CACNA1I 42 33 Cc1csc(CNC(=O)Cc2c(C)nn(C(F)F)c2C)n1 ZINC000147291417 DF On-Demand Anodyne P2RX7 52 47 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne HTR1A 100 46 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne DRD2 83 49 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne DRD1 20 43 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne DRD4 49 43 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne ADRA1D 98 44 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne HTR1B 15 45 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne HTR2A 23 43 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne ADRA1A 84 43 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne ADRA1B 80 44 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne DRD3 74 46 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne HTR7 53 45 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne SSTR5 40 44 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne UTS2R 16 40 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147291446 FG On-Demand Anodyne EHMT2 43 37 CC(C)(CC(=O)O)NC(=O)c1cccc(F)c1Cl ZINC000147291480 CE On-Demand Anodyne ECR 40 39 Cc1cn([C@@H]2C[C@@H]3OC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)OC(C)(C)C)[C@@H]3O2)c(=O)[nH]c1=O ZINC000147291495 KD Annotated Anodyne TK 43 34 Cc1cn([C@@H]2C[C@@H]3OC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)OC(C)(C)C)[C@@H]3O2)c(=O)[nH]c1=O ZINC000147291495 KD Annotated Anodyne PGC 63 37 Cc1cn([C@@H]2C[C@@H]3OC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)OC(C)(C)C)[C@@H]3O2)c(=O)[nH]c1=O ZINC000147291495 KD Annotated Anodyne PAPA1_CARPA 43 42 Cc1cn([C@@H]2C[C@@H]3OC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)OC(C)(C)C)[C@@H]3O2)c(=O)[nH]c1=O ZINC000147291495 KD Annotated Anodyne CCKAR 52 46 Cc1cn([C@@H]2C[C@@H]3OC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)OC(C)(C)C)[C@@H]3O2)c(=O)[nH]c1=O ZINC000147291495 KD Annotated Anodyne CTSL 27 42 Cc1cn([C@@H]2C[C@@H]3OC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)OC(C)(C)C)[C@@H]3O2)c(=O)[nH]c1=O ZINC000147291495 KD Annotated Anodyne REN 77 42 Cc1cn([C@@H]2C[C@@H]3OC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)OC(C)(C)C)[C@@H]3O2)c(=O)[nH]c1=O ZINC000147291495 KD Annotated Anodyne CTSE 41 37 Cc1cn([C@@H]2C[C@@H]3OC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)OC(C)(C)C)[C@@H]3O2)c(=O)[nH]c1=O ZINC000147291495 KD Annotated Anodyne FPR1 52 40 Cc1cn([C@@H]2C[C@@H]3OC[C@H](NC(=O)[C@H](Cc4ccccc4)NC(=O)OC(C)(C)C)[C@@H]3O2)c(=O)[nH]c1=O ZINC000147291495 KD Annotated Anodyne TK2 63 38 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1OC ZINC000147291540 DD On-Demand Anodyne QRFPR 44 37 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1OC ZINC000147291540 DD On-Demand Anodyne ENPP1 58 34 CN(C)C(=O)NCCNS(=O)(=O)c1ccc(CBr)cc1 ZINC000147291556 FD For-Sale Reactive CA2 15 40 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild THRA 50 36 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild DRD3 32 40 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild FOLH1 36 57 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild PTAFR 16 41 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild RARB 32 53 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild THRB 27 63 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild CTSG 22 41 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild PLA2G4A 28 48 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild CTRB1 23 41 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild PLA2G4B 72 48 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild CELA2A 20 41 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild HDAC6 19 49 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild FAAH 17 48 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild S1PR2 56 38 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild EPHX2 24 44 CCCCCCCCNC(=O)c1ccc(C(=O)O)cc1 ZINC000147291579 CG For-Sale Mild ASAH1 108 42 O=C(NC[C@H]1CCCOC1)c1ccc2c(c1)COC2 ZINC000147291590 CD On-Demand Anodyne CACNA1I 42 33 O=C(c1cccc2c1OCCN2)N1CCC[C@@H]1CCCO ZINC000147291671 CD For-Sale Anodyne HCRTR1 18 43 O=C(c1cccc2c1OCCN2)N1CCC[C@@H]1CCCO ZINC000147291671 CD For-Sale Anodyne HCRTR2 0 43 CC(C)(CC(=O)O)NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147291698 CE For-Sale Anodyne FFAR1 0 40 CC(C)(CC(=O)O)NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147291698 CE For-Sale Anodyne GPR88 0 43 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1OC ZINC000147291763 DD On-Demand Anodyne QRFPR 44 37 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1OC ZINC000147291763 DD On-Demand Anodyne ENPP1 58 34 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1C(=O)N1CCC(C)CC1)C2 ZINC000147291804 HH On-Demand Anodyne CHRM2 31 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1C(=O)N1CCC(C)CC1)C2 ZINC000147291804 HH On-Demand Anodyne ROCK2 31 44 CCCCCCCCNC(=O)c1cn(CC(=O)O)nn1 ZINC000147291810 CD For-Sale Mild LGALS3 15 41 CCCCCCCCNC(=O)c1cn(CC(=O)O)nn1 ZINC000147291810 CD For-Sale Mild ASAH1 97 38 CCCCCCCCNC(=O)c1cn(CC(=O)O)nn1 ZINC000147291810 CD For-Sale Mild LGALS7B 0 41 CC[C@@H](C)c1ccccc1Oc1nc(N)ccc1[N+](=O)[O-] ZINC000147291866 CH For-Sale Bother AO-ACHE 0 40 CC(C)(CC(=O)O)NC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147291882 CE For-Sale Anodyne FFAR1 0 40 CC(C)(CC(=O)O)NC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147291882 CE For-Sale Anodyne GPR88 0 43 O=C(c1cccc2c1OCCN2)N1CCC[C@H]1CCCO ZINC000147291889 CD For-Sale Anodyne HCRTR1 18 43 O=C(c1cccc2c1OCCN2)N1CCC[C@H]1CCCO ZINC000147291889 CD For-Sale Anodyne HCRTR2 0 43 COc1ccccc1N1CCC(NCc2ccc(OC)c(OC)c2OC)CC1 ZINC000147291895 GG On-Demand Anodyne HTR1A 86 45 COc1ccccc1N1CCC(NCc2ccc(OC)c(OC)c2OC)CC1 ZINC000147291895 GG On-Demand Anodyne DRD2 70 45 COc1ccccc1N1CCC(NCc2ccc(OC)c(OC)c2OC)CC1 ZINC000147291895 GG On-Demand Anodyne DRD1 17 43 COc1ccccc1N1CCC(NCc2ccc(OC)c(OC)c2OC)CC1 ZINC000147291895 GG On-Demand Anodyne DRD4 37 42 COc1ccccc1N1CCC(NCc2ccc(OC)c(OC)c2OC)CC1 ZINC000147291895 GG On-Demand Anodyne ADRA1D 85 40 COc1ccccc1N1CCC(NCc2ccc(OC)c(OC)c2OC)CC1 ZINC000147291895 GG On-Demand Anodyne HTR2A 20 43 COc1ccccc1N1CCC(NCc2ccc(OC)c(OC)c2OC)CC1 ZINC000147291895 GG On-Demand Anodyne ADRA1A 72 41 COc1ccccc1N1CCC(NCc2ccc(OC)c(OC)c2OC)CC1 ZINC000147291895 GG On-Demand Anodyne ADRA1B 70 40 COc1ccccc1N1CCC(NCc2ccc(OC)c(OC)c2OC)CC1 ZINC000147291895 GG On-Demand Anodyne DRD3 64 45 COc1ccccc1N1CCC(NCc2ccc(OC)c(OC)c2OC)CC1 ZINC000147291895 GG On-Demand Anodyne HTR7 52 44 CC[C@@H]1CN(C(=O)Cc2ccccc2OC)CC[C@@H]1N ZINC000147291962 CD On-Demand Anodyne CHRM5 20 47 CC[C@@H]1CN(C(=O)Cc2ccccc2OC)CC[C@@H]1N ZINC000147291962 CD On-Demand Anodyne CCR3 15 53 CC[C@@H]1CN(C(=O)Cc2ccccc2OC)CC[C@@H]1N ZINC000147291962 CD On-Demand Anodyne MBTPS1 45 32 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(F)c(Cl)c1 ZINC000147291981 DE On-Demand Anodyne ERBB4 42 32 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(F)c(Cl)c1 ZINC000147291981 DE On-Demand Anodyne ENV 50 40 CCCCCCCCNC(=O)c1c(C)[nH]c(C(=O)O)c1C ZINC000147292015 CG For-Sale Mild ASAH1 90 37 CC[C@H](C)c1ccccc1Oc1nc(N)ccc1[N+](=O)[O-] ZINC000147292064 CH For-Sale Bother AO-ACHE 0 40 COCC[C@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147292138 CC For-Sale Anodyne NPPA 45 35 CCn1cc(NC(=O)c2ccccc2Nc2ccc(OC(F)F)cc2)ccc1=O ZINC000147292139 GI On-Demand Anodyne AKR1C2 35 40 CCn1cc(NC(=O)c2ccccc2Nc2ccc(OC(F)F)cc2)ccc1=O ZINC000147292139 GI On-Demand Anodyne KCNK3 40 33 COc1ccc(Br)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292146 HI On-Demand Anodyne HTR1A 80 45 COc1ccc(Br)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292146 HI On-Demand Anodyne DRD2 70 48 COc1ccc(Br)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292146 HI On-Demand Anodyne DRD1 17 44 COc1ccc(Br)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292146 HI On-Demand Anodyne DRD4 40 48 COc1ccc(Br)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292146 HI On-Demand Anodyne ADRA1D 78 46 COc1ccc(Br)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292146 HI On-Demand Anodyne HTR2A 19 44 COc1ccc(Br)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292146 HI On-Demand Anodyne ADRA1A 65 46 COc1ccc(Br)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292146 HI On-Demand Anodyne ADRA1B 63 46 COc1ccc(Br)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292146 HI On-Demand Anodyne DRD3 67 48 COc1ccc(Br)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292146 HI On-Demand Anodyne HTR7 51 42 CC(C)(CC(=O)O)NC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147292149 CE For-Sale Anodyne FFAR1 0 40 CC(C)(CC(=O)O)NC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147292149 CE For-Sale Anodyne GPR88 0 43 Cn1cc(I)c(=O)n(Cc2ccc(F)cc2Cl)c1=O ZINC000147292164 GD On-Demand Anodyne P2RX7 61 43 CC[C@H]1CN(C(=O)[C@@H]2CCCN(c3ccccn3)C2)CCO1 ZINC000147292173 DD On-Demand Anodyne GPBAR1 18 48 NC(=O)NCCn1c(SCC(=O)O)nc2cc(F)ccc21 ZINC000147292175 DD For-Sale Anodyne GNRHR 15 41 NC(=O)NCCn1c(SCC(=O)O)nc2cc(F)ccc21 ZINC000147292175 DD For-Sale Anodyne PTGDR2 15 44 CCOC(=O)[C@](C)(C#N)Cc1ccc(F)cc1Cl ZINC000147292187 CG For-Sale Mild P2RX7 55 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(F)c(Cl)c1 ZINC000147292192 DE On-Demand Anodyne ERBB4 42 32 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(F)c(Cl)c1 ZINC000147292192 DE On-Demand Anodyne ENV 50 40 CC[C@H]1CN(C(=O)Cc2ccccc2OC)CC[C@@H]1N ZINC000147292193 CD On-Demand Anodyne CHRM5 20 47 CC[C@H]1CN(C(=O)Cc2ccccc2OC)CC[C@@H]1N ZINC000147292193 CD On-Demand Anodyne CCR3 15 53 Cn1nnnc1SCC1=C(C(=O)O)N2C(=O)[C@@H](NC(=O)Cn3ccc4ccccc43)[C@H]2SC1 ZINC000147292200 JC Annotated Anodyne SLC22A6 64 68 Cn1nnnc1SCC1=C(C(=O)O)N2C(=O)[C@@H](NC(=O)Cn3ccc4ccccc43)[C@H]2SC1 ZINC000147292200 JC Annotated Anodyne SLC22A8 0 68 Cn1nnnc1SCC1=C(C(=O)O)N2C(=O)[C@@H](NC(=O)Cn3ccc4ccccc43)[C@H]2SC1 ZINC000147292200 JC Annotated Anodyne SLC22A11 0 68 CCCCCCCCNC(=O)Cn1cccc1C(=O)O ZINC000147292261 CF For-Sale Mild ASAH1 107 44 CCCCCCCCNC(=O)Cn1cccc1C(=O)O ZINC000147292261 CF For-Sale Mild ACAT 0 41 CC[C@@H](C)c1ccccc1Oc1cc(NC)nc(N)n1 ZINC000147292305 CG For-Sale Anodyne AO-ACHE 0 43 CC(C)(CC(=O)O)NC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147292351 CE For-Sale Anodyne FFAR1 0 40 CC(C)(CC(=O)O)NC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147292351 CE For-Sale Anodyne GPR88 0 43 COc1cc(OC)c(OC)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292356 GG On-Demand Anodyne HTR1A 95 47 COc1cc(OC)c(OC)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292356 GG On-Demand Anodyne DRD2 79 48 COc1cc(OC)c(OC)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292356 GG On-Demand Anodyne DRD1 18 47 COc1cc(OC)c(OC)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292356 GG On-Demand Anodyne DRD4 46 44 COc1cc(OC)c(OC)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292356 GG On-Demand Anodyne ADRA1D 89 44 COc1cc(OC)c(OC)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292356 GG On-Demand Anodyne HTR2A 23 48 COc1cc(OC)c(OC)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292356 GG On-Demand Anodyne ADRA1A 76 44 COc1cc(OC)c(OC)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292356 GG On-Demand Anodyne ADRA1B 72 44 COc1cc(OC)c(OC)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292356 GG On-Demand Anodyne DRD3 72 48 COc1cc(OC)c(OC)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292356 GG On-Demand Anodyne HTR7 55 46 COc1cc(OC)c(OC)cc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147292356 GG On-Demand Anodyne NPY1R 21 43 COCC[C@@H](NC(=O)c1cccc2c1OCCN2)C(=O)O ZINC000147292358 CC For-Sale Anodyne NPPA 45 35 CCn1cc(NC(=O)c2ccccc2Nc2ccc(C)cc2)ccc1=O ZINC000147292365 EI On-Demand Anodyne AKR1C3 21 51 CCn1cc(NC(=O)c2ccccc2Nc2ccc(C)cc2)ccc1=O ZINC000147292365 EI On-Demand Anodyne KCNK3 48 36 CCn1cc(NC(=O)c2ccccc2Nc2ccc(C)cc2)ccc1=O ZINC000147292365 EI On-Demand Anodyne KCNK9 50 36 CN(C)NC(=O)CCCN ZINC000147292370 AB For-Sale Reactive ABAT 42 34 CN(C)NC(=O)CCCN ZINC000147292370 AB For-Sale Reactive APHA 41 38 CN(C)NC(=O)CCCN ZINC000147292370 AB For-Sale Reactive KDM7A 0 56 CCOC(=O)[C@@](C)(C#N)Cc1ccc(F)cc1Cl ZINC000147292403 CG For-Sale Mild P2RX7 55 40 NC(=O)NCCn1c(SCC(=O)O)nc2cc(Br)ccc21 ZINC000147292406 FD For-Sale Anodyne PTGDR2 15 41 CC[C@@H]1CN(C(=O)Cc2ccccc2OC)CC[C@H]1N ZINC000147292408 CD On-Demand Anodyne CHRM5 20 47 CC[C@@H]1CN(C(=O)Cc2ccccc2OC)CC[C@H]1N ZINC000147292408 CD On-Demand Anodyne CCR3 15 53 CCCCCCCCNS(=O)(=O)c1ccc([C@@H](C)O)cc1 ZINC000147292460 DG For-Sale Mild TBXA2R 15 45 CCCCCCCCNS(=O)(=O)c1ccc([C@@H](C)O)cc1 ZINC000147292460 DG For-Sale Mild ALOX15 58 45 CCCCCCCCNS(=O)(=O)c1ccc([C@@H](C)O)cc1 ZINC000147292460 DG For-Sale Mild ASAH1 68 35 Cc1ccc(C#N)cc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147292480 CD On-Demand Mild TBXA2R 0 46 CC[C@H](C)c1ccccc1Oc1cc(NC)nc(N)n1 ZINC000147292558 CG For-Sale Anodyne AO-ACHE 0 43 CN(C)NC(=O)CCCCCN ZINC000147292581 AC For-Sale Reactive PAOX 18 41 CN(C)NC(=O)CCCCCN ZINC000147292581 AC For-Sale Reactive APHA 0 44 CN(C)NC(=O)CCCCCN ZINC000147292581 AC For-Sale Reactive KDM7A 0 52 CCCCCCCC(=O)Cc1ccc(F)c(F)c1 ZINC000147292582 CI For-Sale Mild RARB 16 43 CCCCCCCC(=O)Cc1ccc(F)c(F)c1 ZINC000147292582 CI For-Sale Mild PLA2G4B 75 37 CCCCCCCC(=O)Cc1ccc(F)c(F)c1 ZINC000147292582 CI For-Sale Mild CQSS 53 33 CC[C@H]1CN(C(=O)Cc2ccccc2OC)CC[C@H]1N ZINC000147292605 CD On-Demand Anodyne CHRM5 20 47 CC[C@H]1CN(C(=O)Cc2ccccc2OC)CC[C@H]1N ZINC000147292605 CD On-Demand Anodyne CCR3 15 53 CN(C)C1(CNC(=O)c2csc(C#CCO)c2)CCCC1 ZINC000147292651 DD For-Sale Mild SLC6A5 15 44 CCCCCCCCNS(=O)(=O)c1ccc([C@H](C)O)cc1 ZINC000147292680 DG For-Sale Mild TBXA2R 15 45 CCCCCCCCNS(=O)(=O)c1ccc([C@H](C)O)cc1 ZINC000147292680 DG For-Sale Mild ALOX15 58 45 CCCCCCCCNS(=O)(=O)c1ccc([C@H](C)O)cc1 ZINC000147292680 DG For-Sale Mild ASAH1 68 35 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1ccc(-n2cccn2)nc1 ZINC000147292701 HH On-Demand Anodyne ROCK2 18 44 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1ccc(-n2cccn2)nc1 ZINC000147292701 HH On-Demand Anodyne MET 50 46 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1ccc(-n2cccn2)nc1 ZINC000147292701 HH On-Demand Anodyne NAMPT 45 44 Cc1ccc(C#N)cc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147292729 CD On-Demand Mild TBXA2R 0 46 CCNc1ncc(Br)c(Oc2ccccc2[C@H](C)CC)n1 ZINC000147292788 FJ For-Sale Anodyne AO-ACHE 0 40 CCCCCCCCNS(=O)(=O)c1cccc([C@@H](C)O)c1 ZINC000147292880 DG For-Sale Mild FBP1 20 40 CCCCCCCCNS(=O)(=O)c1cccc([C@@H](C)O)c1 ZINC000147292880 DG For-Sale Mild ALOX15 46 40 CCCCCCCCC(=O)Cc1ccc(F)c(F)c1 ZINC000147292943 CJ For-Sale Mild THRA 41 40 CCCCCCCCC(=O)Cc1ccc(F)c(F)c1 ZINC000147292943 CJ For-Sale Mild RARB 16 43 CCCCCCCCC(=O)Cc1ccc(F)c(F)c1 ZINC000147292943 CJ For-Sale Mild THRB 24 40 CCCCCCCCC(=O)Cc1ccc(F)c(F)c1 ZINC000147292943 CJ For-Sale Mild PLA2G4B 60 37 CCCCCCCCC(=O)Cc1ccc(F)c(F)c1 ZINC000147292943 CJ For-Sale Mild CQSS 53 33 CCNc1ncc(Br)c(Oc2ccccc2[C@@H](C)CC)n1 ZINC000147292990 FJ For-Sale Anodyne AO-ACHE 0 40 C#CCOc1ccccc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147293017 FG On-Demand Mild HTR1A 63 41 C#CCOc1ccccc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147293017 FG On-Demand Mild DRD2 55 41 C#CCOc1ccccc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147293017 FG On-Demand Mild DRD1 30 40 C#CCOc1ccccc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147293017 FG On-Demand Mild ADRA1D 63 38 C#CCOc1ccccc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147293017 FG On-Demand Mild HTR2A 27 40 C#CCOc1ccccc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147293017 FG On-Demand Mild ADRA1A 50 40 C#CCOc1ccccc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147293017 FG On-Demand Mild ADRA1B 56 38 C#CCOc1ccccc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147293017 FG On-Demand Mild DRD3 40 39 C#CCOc1ccccc1CNC1CCN(c2ccccc2OC)CC1 ZINC000147293017 FG On-Demand Mild HTR7 45 42 CC1=C(C(=O)O)N2C(=O)[C@@H](NC(=O)Cn3ccc4ccccc43)[C@H]2SC1 ZINC000147293029 FD Annotated Anodyne SLC22A6 49 45 NS(=O)(=O)c1ccc(OCCN2CCCCC2)c(F)c1F ZINC000147293049 DD For-Sale Anodyne LTA4H 36 43 NS(=O)(=O)c1ccc(OCCN2CCCCC2)c(F)c1F ZINC000147293049 DD For-Sale Anodyne HRH3 29 47 NS(=O)(=O)c1ccc(OCCN2CCCCC2)c(F)c1F ZINC000147293049 DD For-Sale Anodyne PSMB2 40 40 NS(=O)(=O)c1ccc(OCCN2CCCCC2)c(F)c1F ZINC000147293049 DD For-Sale Anodyne PSMB1 44 41 CCCCCCCCNS(=O)(=O)c1cccc([C@H](C)O)c1 ZINC000147293061 DG For-Sale Mild FBP1 20 40 CCCCCCCCNS(=O)(=O)c1cccc([C@H](C)O)c1 ZINC000147293061 DG For-Sale Mild ALOX15 46 40 CC(C)CCCCN[C@@H](C)C(=O)O ZINC000147293144 AD On-Demand Anodyne DNPEP 49 31 CC(C)CCCCN[C@@H](C)C(=O)O ZINC000147293144 AD On-Demand Anodyne SIRT1 27 41 CC(C)CCCCN[C@@H](C)C(=O)O ZINC000147293144 AD On-Demand Anodyne BHMT2 44 28 CC(C)(C)Nc1ccc(NS(=O)(=O)c2ccccc2)cc1 ZINC000147293181 DH For-Sale Anodyne CA2 15 59 CC(C)(C)Nc1ccc(NS(=O)(=O)c2ccccc2)cc1 ZINC000147293181 DH For-Sale Anodyne CA1 15 42 CC(C)(C)Nc1ccc(NS(=O)(=O)c2ccccc2)cc1 ZINC000147293181 DH For-Sale Anodyne CA4 23 59 CC(C)(C)Nc1ccc(NS(=O)(=O)c2ccccc2)cc1 ZINC000147293181 DH For-Sale Anodyne PRTN3 52 33 CC(C)(C)Nc1ccc(NS(=O)(=O)c2ccccc2)cc1 ZINC000147293181 DH For-Sale Anodyne ALPL 15 56 CC(C)(C)Nc1ccc(NS(=O)(=O)c2ccccc2)cc1 ZINC000147293181 DH For-Sale Anodyne CYNT 19 50 CC(C)(C)Nc1ccc(NS(=O)(=O)c2ccccc2)cc1 ZINC000147293181 DH For-Sale Anodyne LIMK2 52 40 CCCCCCCCn1c(C)ccc1C ZINC000147293274 BI For-Sale Mild TLR8 0 45 CCCCCCCCn1c(C)ccc1C ZINC000147293274 BI For-Sale Mild CQSS 52 35 C[C@@H]1Cc2ccccc2N1C(=O)CNC1(C(=O)O)CCC1 ZINC000147293295 CD For-Sale Anodyne ACE 17 41 C[C@@H]1Cc2ccccc2N1C(=O)CNC1(C(=O)O)CCC1 ZINC000147293295 CD For-Sale Anodyne DRD4 30 48 C[C@@H]1Cc2ccccc2N1C(=O)CNC1(C(=O)O)CCC1 ZINC000147293295 CD For-Sale Anodyne TPP2 58 35 NC(=O)NCCn1c(SCC(=O)O)nc2cccc(Cl)c21 ZINC000147293298 ED For-Sale Anodyne PTGDR2 15 41 CC(C)CCCCN[C@H](C)C(=O)O ZINC000147293382 AD On-Demand Anodyne DNPEP 49 31 CC(C)CCCCN[C@H](C)C(=O)O ZINC000147293382 AD On-Demand Anodyne SIRT1 27 41 CC(C)CCCCN[C@H](C)C(=O)O ZINC000147293382 AD On-Demand Anodyne BHMT2 44 28 O=C(Nc1ccccc1)[C@H]1CCCN(C(=O)c2sccc2-c2ccccc2)C1 ZINC000147293417 GJ On-Demand Anodyne INHA 17 40 Cc1cc(C(=O)N2CCN(Cc3nc4ccccc4s3)CC2)cc([N+](=O)[O-])c1 ZINC000147293431 GG On-Demand Bother AKR1B1 19 43 Cc1cc(C(=O)N2CCN(Cc3nc4ccccc4s3)CC2)cc([N+](=O)[O-])c1 ZINC000147293431 GG On-Demand Bother MGLL 0 41 CCCCCCCC(=O)N1CC[C@H](N)[C@H](CC)C1 ZINC000147293442 CF On-Demand Mild GNAI1 0 56 CCCCCCCC(=O)N1CC[C@H](N)[C@H](CC)C1 ZINC000147293442 CF On-Demand Mild GNAI3 0 53 CCCCCCCC(=O)N1CC[C@H](N)[C@H](CC)C1 ZINC000147293442 CF On-Demand Mild GNAO1 0 53 CCCCCCCC(=O)N1CC[C@H](N)[C@H](CC)C1 ZINC000147293442 CF On-Demand Mild CQSS 54 33 C[C@H]1Cc2ccccc2N1C(=O)CNC1(C(=O)O)CCC1 ZINC000147293463 CD For-Sale Anodyne ACE 17 41 C[C@H]1Cc2ccccc2N1C(=O)CNC1(C(=O)O)CCC1 ZINC000147293463 CD For-Sale Anodyne DRD4 30 48 C[C@H]1Cc2ccccc2N1C(=O)CNC1(C(=O)O)CCC1 ZINC000147293463 CD For-Sale Anodyne TPP2 58 35 CCCCCCCCNC(=O)c1ccc2[nH]cnc2c1 ZINC000147293521 CH For-Sale Mild FOLH1 18 41 CCCCCCCCNC(=O)c1ccc2[nH]cnc2c1 ZINC000147293521 CH For-Sale Mild HDAC9 15 42 CCCCCCCCNC(=O)c1ccc2[nH]cnc2c1 ZINC000147293521 CH For-Sale Mild ASAH1 87 36 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)NN(C)c2ccccc2)cc1 ZINC000147293559 GF On-Demand Reactive COLA 44 34 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)NN(C)c2ccccc2)cc1 ZINC000147293559 GF On-Demand Reactive CA5B 16 40 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)NN(C)c2ccccc2)cc1 ZINC000147293559 GF On-Demand Reactive CA5A 18 40 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)NN(C)c2ccccc2)cc1 ZINC000147293559 GF On-Demand Reactive MMP9 17 43 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)NN(C)c2ccccc2)cc1 ZINC000147293559 GF On-Demand Reactive LIMK2 38 44 CC(C)N(C)S(=O)(=O)c1ccc(CNC(=O)NN(C)c2ccccc2)cc1 ZINC000147293559 GF On-Demand Reactive NAMPT 38 40 CCCCCCCC(=O)N1CC[C@@H](N)[C@H](CC)C1 ZINC000147293635 CF On-Demand Mild GNAI1 0 56 CCCCCCCC(=O)N1CC[C@@H](N)[C@H](CC)C1 ZINC000147293635 CF On-Demand Mild GNAI3 0 53 CCCCCCCC(=O)N1CC[C@@H](N)[C@H](CC)C1 ZINC000147293635 CF On-Demand Mild GNAO1 0 53 CCCCCCCC(=O)N1CC[C@@H](N)[C@H](CC)C1 ZINC000147293635 CF On-Demand Mild CQSS 54 33 O=C(Nc1ccccc1)[C@@H]1CCCN(C(=O)c2sccc2-c2ccccc2)C1 ZINC000147293636 GJ On-Demand Anodyne INHA 17 40 CCNc1cc(Oc2ccccc2[C@H](C)CC)nc(C)n1 ZINC000147293652 CJ For-Sale Anodyne AO-ACHE 0 40 O=C1COc2cc(I)ccc2N1Cc1ccc(F)cc1 ZINC000147293684 GG For-Sale Anodyne SLC5A2 63 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000147293685 EE On-Demand Anodyne DHODH 51 50 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000147293685 EE On-Demand Anodyne EPHX2 22 41 Cc1ccc2c(c1)nc(SCC(=O)O)n2CCNC(N)=O ZINC000147293708 DD For-Sale Anodyne PTGDR2 17 41 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild ACE 15 42 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild CNR1 15 42 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild ACHE 36 48 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild SSTR2 28 40 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MME 25 41 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild EDNRA 41 39 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild TACR1 27 43 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild CNR2 15 46 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild TPR 23 78 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MC4R 56 41 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild TSPO 30 60 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild CCKAR 108 50 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild BCHE 22 45 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MPO 44 41 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild BRS3 30 49 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild NMBR 73 33 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MC3R 84 39 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MC5R 86 40 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MTNR1A 27 41 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MMP2 30 56 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MMP8 36 56 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild GRIA1 70 60 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MMP14 19 41 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild GRPR 94 39 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild ECE1 52 39 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild HDAC1 17 45 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild SSTR3 24 40 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MMP11 54 38 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild CCKBR 92 48 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild GHSR 56 43 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild CFTR 34 45 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild S1PR2 42 32 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild ALOX15 30 51 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MMP9 26 56 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MC1R 107 42 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild ADAM9 39 40 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MMP7 19 56 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild MMP1 24 56 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild HDA106 0 43 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild SLC15A2 0 44 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild KISS1R 81 38 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild ASAH1 99 39 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild ERAP2 43 40 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild ERAP1 0 40 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild ACAT 0 44 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild LASB 0 41 CCCCCCCCNC(=O)Cc1c[nH]c2ccccc12 ZINC000147293742 CI On-Demand Mild CAN2 0 42 CCCCCCCC(=O)N1CC[C@H](N)[C@@H](CC)C1 ZINC000147293828 CF On-Demand Mild GNAI1 0 56 CCCCCCCC(=O)N1CC[C@H](N)[C@@H](CC)C1 ZINC000147293828 CF On-Demand Mild GNAI3 0 53 CCCCCCCC(=O)N1CC[C@H](N)[C@@H](CC)C1 ZINC000147293828 CF On-Demand Mild GNAO1 0 53 CCCCCCCC(=O)N1CC[C@H](N)[C@@H](CC)C1 ZINC000147293828 CF On-Demand Mild CQSS 54 33 C[C@H](N)CC(=O)NN(C)C ZINC000147293850 AB For-Sale Reactive KDM7A 0 45 CCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c2ccccc12 ZINC000147293852 HD On-Demand Anodyne CCR8 108 53 CCNc1cc(Oc2ccccc2[C@@H](C)CC)nc(C)n1 ZINC000147293866 CJ For-Sale Anodyne AO-ACHE 0 40 O=C(O)C1(NCc2ccc(Cl)c(Cl)c2)CCC1 ZINC000147293910 CG On-Demand Anodyne DNAE 42 35 NC(=O)NCCn1c(SCC(=O)O)nc2cc(Cl)ccc21 ZINC000147293917 ED For-Sale Anodyne TBXA2R 0 42 NC(=O)NCCn1c(SCC(=O)O)nc2cc(Cl)ccc21 ZINC000147293917 ED For-Sale Anodyne PTGDR2 15 43 CCCC[C@H](NC(N)=O)C(=O)N1CCN(Cc2csc(C)n2)CC1 ZINC000147293927 FD On-Demand Anodyne P2RY12 170 36 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000147293942 EE On-Demand Anodyne DHODH 51 50 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(F)(F)F)cc1 ZINC000147293942 EE On-Demand Anodyne EPHX2 22 41 CCCCCCCCNC(=O)c1cccc2cc[nH]c12 ZINC000147293946 CI For-Sale Mild PA2A1_NAJMO 0 41 CCCCCCCCNC(=O)c1cccc2cc[nH]c12 ZINC000147293946 CI For-Sale Mild ASAH1 91 37 CCCCCCCCNC(=O)c1cccc2cc[nH]c12 ZINC000147293946 CI For-Sale Mild ACAT 0 45 CCCCCCCCNC(=O)c1cccc2cc[nH]c12 ZINC000147293946 CI For-Sale Mild POLR1A 52 35 CCOc1c(Cl)cc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147294028 HJ On-Demand Anodyne HTR1A 71 40 CCOc1c(Cl)cc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147294028 HJ On-Demand Anodyne DRD2 64 40 CCOc1c(Cl)cc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147294028 HJ On-Demand Anodyne DRD4 47 40 CCOc1c(Cl)cc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147294028 HJ On-Demand Anodyne ADRA1D 62 38 CCOc1c(Cl)cc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147294028 HJ On-Demand Anodyne ADRA1A 54 38 CCOc1c(Cl)cc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147294028 HJ On-Demand Anodyne ADRA1B 49 39 CCOc1c(Cl)cc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147294028 HJ On-Demand Anodyne DRD3 62 40 CCOc1c(Cl)cc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147294028 HJ On-Demand Anodyne HTR7 52 40 CCOc1c(Cl)cc(CNC2CCN(c3ccccc3OC)CC2)cc1OC ZINC000147294028 HJ On-Demand Anodyne SSTR5 63 36 C[C@@H](N)CC(=O)NN(C)C ZINC000147294038 AB For-Sale Reactive KDM7A 0 45 CCCCCCCC(=O)N1CC[C@@H](N)[C@@H](CC)C1 ZINC000147294057 CF On-Demand Mild GNAI1 0 56 CCCCCCCC(=O)N1CC[C@@H](N)[C@@H](CC)C1 ZINC000147294057 CF On-Demand Mild GNAI3 0 53 CCCCCCCC(=O)N1CC[C@@H](N)[C@@H](CC)C1 ZINC000147294057 CF On-Demand Mild GNAO1 0 53 CCCCCCCC(=O)N1CC[C@@H](N)[C@@H](CC)C1 ZINC000147294057 CF On-Demand Mild CQSS 54 33 O=C(CSc1ccccc1C(=O)NCC1(c2ccccc2)CC1)NCC1CCCCC1 ZINC000147294113 IJ On-Demand Anodyne KCNA3 58 46 O=C(CSc1ccccc1C(=O)NCC1(c2ccccc2)CC1)NCC1CCCCC1 ZINC000147294113 IJ On-Demand Anodyne HCN1 70 36 O=C(CSc1ccccc1C(=O)NCC1(c2ccccc2)CC1)NCC1CCCCC1 ZINC000147294113 IJ On-Demand Anodyne HCN4 55 36 NC(=O)NCCn1c(SCC(=O)O)nc2ccccc21 ZINC000147294115 CC For-Sale Anodyne PTGDR2 21 51 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(Cc2csc(C)n2)CC1 ZINC000147294154 FD On-Demand Anodyne P2RY12 170 36 CCCCCCCCNC(=O)c1c(C)n[nH]c1C ZINC000147294157 CG For-Sale Mild ASAH1 84 35 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC(F)F ZINC000147294233 GI On-Demand Anodyne HTR1A 75 40 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC(F)F ZINC000147294233 GI On-Demand Anodyne DRD2 69 44 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC(F)F ZINC000147294233 GI On-Demand Anodyne ADRA1D 78 41 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC(F)F ZINC000147294233 GI On-Demand Anodyne ADRA1A 68 41 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC(F)F ZINC000147294233 GI On-Demand Anodyne ADRA1B 60 41 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC(F)F ZINC000147294233 GI On-Demand Anodyne DRD3 61 40 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1OC(F)F ZINC000147294233 GI On-Demand Anodyne HTR7 45 39 CC(C)(C)Nc1ccc(NS(=O)(=O)c2ccccc2)cn1 ZINC000147294272 DG For-Sale Anodyne PRTN3 43 32 CC(C)(C)Nc1ccc(NS(=O)(=O)c2ccccc2)cn1 ZINC000147294272 DG For-Sale Anodyne ALPL 28 43 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc2c(c1)CCCC2 ZINC000147294291 EH On-Demand Anodyne BMP1 47 34 Cc1ccc(C#CC(N)=O)cc1 ZINC000147294292 AC For-Sale Mild LOX1.1 45 33 Cc1ccc(C#CC(N)=O)cc1 ZINC000147294292 AC For-Sale Mild FFAR1 17 47 Cc1ccc(C#CC(N)=O)cc1 ZINC000147294292 AC For-Sale Mild O49150_SOLTU 49 34 Cc1cccc2nc(SCC(=O)O)n(CCNC(N)=O)c12 ZINC000147294326 DD For-Sale Anodyne PTGDR2 15 41 CCCCCCCCNC(=O)c1nc(C(C)(C)C)n[nH]1 ZINC000147294361 CG For-Sale Mild ASAH1 72 36 Cc1ccccc1-n1nc(C(=O)N[C@@H](C)c2nnc3n2CCCCC3)c2c1CCC2 ZINC000147294382 HG On-Demand Anodyne CNR1 55 35 CCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147294390 DD On-Demand Anodyne ACACA 0 40 CCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147294390 DD On-Demand Anodyne ADAM17 30 41 CCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147294390 DD On-Demand Anodyne MMP2 33 40 CCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147294390 DD On-Demand Anodyne MMP14 24 41 CCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147294390 DD On-Demand Anodyne MMP9 35 43 CCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147294390 DD On-Demand Anodyne ADAMTS4 64 38 CCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147294390 DD On-Demand Anodyne MMP1 25 47 CCCCCCCCCC(=O)Cc1ccc(F)c(F)c1 ZINC000147294415 CK For-Sale Mild RARB 16 43 CCCCCCCCCC(=O)Cc1ccc(F)c(F)c1 ZINC000147294415 CK For-Sale Mild PLA2G4B 75 37 CCCCCCCCCC(=O)Cc1ccc(F)c(F)c1 ZINC000147294415 CK For-Sale Mild CQSS 53 33 CCc1ccc(C(=O)N2CC[C@H](N)[C@H](CC)C2)cc1 ZINC000147294424 CE On-Demand Anodyne L3MBTL1 0 43 CCc1ccc(C(=O)N2CC[C@H](N)[C@H](CC)C2)cc1 ZINC000147294424 CE On-Demand Anodyne L3MBTL3 76 43 CCc1ccc(C(=O)N2CC[C@H](N)[C@H](CC)C2)cc1 ZINC000147294424 CE On-Demand Anodyne MBTD1 0 41 CN(C)NC(=O)CC[C@@H]1CCCCN1 ZINC000147294458 AC For-Sale Reactive KDM7A 0 41 CCOc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147294472 HI On-Demand Anodyne HTR1A 62 38 CCOc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147294472 HI On-Demand Anodyne DRD2 60 45 CCOc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147294472 HI On-Demand Anodyne DRD4 39 40 CCOc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147294472 HI On-Demand Anodyne ADRA1D 61 38 CCOc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147294472 HI On-Demand Anodyne ADRA1A 54 38 CCOc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147294472 HI On-Demand Anodyne ADRA1B 49 38 CCOc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147294472 HI On-Demand Anodyne DRD3 52 40 CCOc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147294472 HI On-Demand Anodyne HTR7 46 36 CCOc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147294472 HI On-Demand Anodyne SSTR5 75 42 CCCCCc1ccc2c(c1)OC(C)(C)[C@@H]1CCC(C)=C[C@@H]21 ZINC000147294480 CK For-Sale Anodyne CNR1 18 51 CCCCCc1ccc2c(c1)OC(C)(C)[C@@H]1CCC(C)=C[C@@H]21 ZINC000147294480 CK For-Sale Anodyne CNR2 16 67 CCNc1ncnc(Oc2ccccc2[C@H](C)CC)c1C ZINC000147294488 CJ For-Sale Anodyne AO-ACHE 0 41 C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc2c(c1)CCCC2 ZINC000147294512 EH On-Demand Anodyne BMP1 47 34 COC(=O)c1ccc(F)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147294545 GC On-Demand Anodyne SFRP1 88 36 COC(=O)c1ccc(F)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147294545 GC On-Demand Anodyne WNT3 60 32 CC[C@@H](C)[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147294555 CF On-Demand Anodyne CCR1 21 43 CC[C@@H](C)[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147294555 CF On-Demand Anodyne ACE2 46 34 CCCCC[C@@H](C)NCCP(=O)(OCC)OCC ZINC000147294564 CH For-Sale Anodyne FDPS 15 43 NC(=O)NCCn1c(SCC(=O)O)nc2ccc(Br)cc21 ZINC000147294565 FD For-Sale Anodyne PTGDR2 15 41 Cc1ccccc1-n1nc(C(=O)N[C@H](C)c2nnc3n2CCCCC3)c2c1CCC2 ZINC000147294590 HG On-Demand Anodyne CNR1 55 35 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild CNR1 16 43 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild DRD3 31 56 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild TSPO 25 49 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild CCKAR 27 62 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild PYGL 87 46 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild PLD1 32 40 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild PYGM 29 41 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild PLCG2 0 40 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild PLD2 34 47 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild PA2A1_NAJMO 0 40 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild AKR1C3 0 78 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild ASAH1 99 42 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild PYK 46 46 CCCCCCCCNC(=O)c1cc2ccccc2[nH]1 ZINC000147294596 CI For-Sale Mild ACAT 0 45 CCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147294604 DD On-Demand Anodyne ACACA 0 40 CCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147294604 DD On-Demand Anodyne ADAM17 30 41 CCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147294604 DD On-Demand Anodyne MMP2 33 40 CCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147294604 DD On-Demand Anodyne MMP14 24 41 CCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147294604 DD On-Demand Anodyne MMP9 35 43 CCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147294604 DD On-Demand Anodyne ADAMTS4 64 38 CCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147294604 DD On-Demand Anodyne MMP1 25 47 Cc1cc(NC(=O)c2cccc3c2OCCN3)ccc1F ZINC000147294614 CG For-Sale Anodyne MTTP 41 36 Cc1cc(NC(=O)c2cccc3c2OCCN3)ccc1F ZINC000147294614 CG For-Sale Anodyne KCNK3 72 38 Cc1cc(NC(=O)c2cccc3c2OCCN3)ccc1F ZINC000147294614 CG For-Sale Anodyne KCNK9 67 36 CC(C)[C@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294627 GE On-Demand Anodyne PRSS1 22 44 CC(C)[C@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294627 GE On-Demand Anodyne CASP1 16 42 CC(C)[C@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294627 GE On-Demand Anodyne PLAU 17 44 CC(C)[C@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294627 GE On-Demand Anodyne DGAT1 19 49 CC(C)[C@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294627 GE On-Demand Anodyne KCNK3 61 42 CC(C)[C@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294627 GE On-Demand Anodyne KCNK9 43 32 CCc1ccc(C(=O)N2CC[C@@H](N)[C@H](CC)C2)cc1 ZINC000147294650 CE On-Demand Anodyne L3MBTL1 0 43 CCc1ccc(C(=O)N2CC[C@@H](N)[C@H](CC)C2)cc1 ZINC000147294650 CE On-Demand Anodyne L3MBTL3 76 43 CCc1ccc(C(=O)N2CC[C@@H](N)[C@H](CC)C2)cc1 ZINC000147294650 CE On-Demand Anodyne MBTD1 0 41 Cc1nnc(SCC2=C(C(=O)O)N3C(=O)[C@@H](NC(=O)Cn4ccc5ccccc54)[C@H]3SC2)s1 ZINC000147294680 KE Annotated Anodyne SLC22A6 60 67 CN(C)NC(=O)CC[C@H]1CCCCN1 ZINC000147294683 AC For-Sale Reactive KDM7A 0 41 O=C1COc2cc(I)ccc2N1Cc1cc(F)ccc1F ZINC000147294684 HG For-Sale Anodyne SLC5A2 53 40 O=C1COc2cc(I)ccc2N1Cc1cc(F)ccc1F ZINC000147294684 HG For-Sale Anodyne Q9M629_MAIZE 50 39 CCNc1ncnc(Oc2ccccc2[C@@H](C)CC)c1C ZINC000147294699 CJ For-Sale Anodyne AO-ACHE 0 41 COC(=O)c1ccc(F)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147294763 GC On-Demand Anodyne SFRP1 88 36 COC(=O)c1ccc(F)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147294763 GC On-Demand Anodyne WNT3 60 32 CC[C@@H](C)[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147294781 CF On-Demand Anodyne CCR1 21 43 CC[C@@H](C)[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147294781 CF On-Demand Anodyne ACE2 46 34 CCCCCCCCNC(=O)[C@@H]1CCC(=O)NC1 ZINC000147294784 CD On-Demand Mild GNAI1 0 57 CCCCCCCCNC(=O)[C@@H]1CCC(=O)NC1 ZINC000147294784 CD On-Demand Mild GNAI3 0 57 CCCCCCCCNC(=O)[C@@H]1CCC(=O)NC1 ZINC000147294784 CD On-Demand Mild GNAO1 0 57 CCCCCCCCNC(=O)[C@@H]1CCC(=O)NC1 ZINC000147294784 CD On-Demand Mild ASAH1 90 36 CCCCCCCCNC(=O)[C@@H]1CCC(=O)NC1 ZINC000147294784 CD On-Demand Mild LASR 45 32 CCCCC[C@H](C)NCCP(=O)(OCC)OCC ZINC000147294804 CH For-Sale Anodyne FDPS 15 43 C#CCNC(=O)COc1ccc(S(N)(=O)=O)c(F)c1F ZINC000147294817 DB For-Sale Mild CA2 17 42 CCc1ccc(C(=O)N2CC[C@H](N)[C@@H](CC)C2)cc1 ZINC000147294840 CE On-Demand Anodyne L3MBTL1 0 43 CCc1ccc(C(=O)N2CC[C@H](N)[C@@H](CC)C2)cc1 ZINC000147294840 CE On-Demand Anodyne L3MBTL3 76 43 CCc1ccc(C(=O)N2CC[C@H](N)[C@@H](CC)C2)cc1 ZINC000147294840 CE On-Demand Anodyne MBTD1 0 41 CC(C)[C@@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294846 GE On-Demand Anodyne PRSS1 22 44 CC(C)[C@@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294846 GE On-Demand Anodyne CASP1 16 42 CC(C)[C@@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294846 GE On-Demand Anodyne PLAU 17 44 CC(C)[C@@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294846 GE On-Demand Anodyne DGAT1 19 49 CC(C)[C@@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294846 GE On-Demand Anodyne KCNK3 61 42 CC(C)[C@@H](NC(=O)c1ccc(F)cc1)C(=O)Nc1cccc(OCC(N)=O)c1 ZINC000147294846 GE On-Demand Anodyne KCNK9 43 32 C[C@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147294857 DE On-Demand Anodyne F2 21 46 C[C@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147294857 DE On-Demand Anodyne SERPINC1 0 40 C[C@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147294857 DE On-Demand Anodyne MMP13 28 50 C[C@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147294857 DE On-Demand Anodyne TRY2_BOVIN 63 42 C[C@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147294857 DE On-Demand Anodyne MMP2 29 50 C[C@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147294857 DE On-Demand Anodyne MMP3 15 44 C[C@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147294857 DE On-Demand Anodyne MMP12 31 43 C[C@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147294857 DE On-Demand Anodyne ADAMTS4 47 41 C[C@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147294857 DE On-Demand Anodyne AKR1C3 15 45 C[C@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147294857 DE On-Demand Anodyne Q9JN24_ECOLX 0 43 CCN[C@@H](C)CC(=O)NN(C)C ZINC000147294920 AB For-Sale Reactive KDM7A 0 41 CCOc1cccc(CNC2CCN(c3ccccc3OC)CC2)c1OC(F)F ZINC000147294955 HI On-Demand Anodyne HTR1A 70 40 CCOc1cccc(CNC2CCN(c3ccccc3OC)CC2)c1OC(F)F ZINC000147294955 HI On-Demand Anodyne DRD2 55 45 CCOc1cccc(CNC2CCN(c3ccccc3OC)CC2)c1OC(F)F ZINC000147294955 HI On-Demand Anodyne DRD4 30 45 CCOc1cccc(CNC2CCN(c3ccccc3OC)CC2)c1OC(F)F ZINC000147294955 HI On-Demand Anodyne ADRA1D 62 42 CCOc1cccc(CNC2CCN(c3ccccc3OC)CC2)c1OC(F)F ZINC000147294955 HI On-Demand Anodyne ADRA1A 53 42 CCOc1cccc(CNC2CCN(c3ccccc3OC)CC2)c1OC(F)F ZINC000147294955 HI On-Demand Anodyne ADRA1B 50 42 CCOc1cccc(CNC2CCN(c3ccccc3OC)CC2)c1OC(F)F ZINC000147294955 HI On-Demand Anodyne DRD3 47 45 CCOc1cccc(CNC2CCN(c3ccccc3OC)CC2)c1OC(F)F ZINC000147294955 HI On-Demand Anodyne HTR7 54 40 CCCCCCCCNC(=O)[C@H]1CCC(=O)NC1 ZINC000147294983 CD On-Demand Mild GNAI1 0 57 CCCCCCCCNC(=O)[C@H]1CCC(=O)NC1 ZINC000147294983 CD On-Demand Mild GNAI3 0 57 CCCCCCCCNC(=O)[C@H]1CCC(=O)NC1 ZINC000147294983 CD On-Demand Mild GNAO1 0 57 CCCCCCCCNC(=O)[C@H]1CCC(=O)NC1 ZINC000147294983 CD On-Demand Mild ASAH1 90 36 CCCCCCCCNC(=O)[C@H]1CCC(=O)NC1 ZINC000147294983 CD On-Demand Mild LASR 45 32 CC[C@H](C)[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147294992 CF On-Demand Anodyne CCR1 21 43 CC[C@H](C)[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147294992 CF On-Demand Anodyne ACE2 46 34 CCc1ccc(C(=O)N2CC[C@@H](N)[C@@H](CC)C2)cc1 ZINC000147295015 CE On-Demand Anodyne L3MBTL1 0 43 CCc1ccc(C(=O)N2CC[C@@H](N)[C@@H](CC)C2)cc1 ZINC000147295015 CE On-Demand Anodyne L3MBTL3 76 43 CCc1ccc(C(=O)N2CC[C@@H](N)[C@@H](CC)C2)cc1 ZINC000147295015 CE On-Demand Anodyne MBTD1 0 41 CCOc1nc(N)nc(Oc2ccccc2[C@H](C)CC)n1 ZINC000147295016 CG For-Sale Anodyne AO-ACHE 0 41 Cc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1F ZINC000147295038 CD On-Demand Anodyne ENV 47 39 C#CCNC(=O)[C@H](C)Oc1ccc(S(N)(=O)=O)c(F)c1F ZINC000147295041 DC For-Sale Mild CA2 19 40 C#CCNC(=O)[C@H](C)Oc1ccc(S(N)(=O)=O)c(F)c1F ZINC000147295041 DC For-Sale Mild CA14 16 40 CCOCCCCNC(=O)c1cc(OC)ccc1[N+](=O)[O-] ZINC000147295054 CE On-Demand Bother U38 0 40 C[C@@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147295077 DE On-Demand Anodyne F2 21 46 C[C@@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147295077 DE On-Demand Anodyne SERPINC1 0 40 C[C@@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147295077 DE On-Demand Anodyne MMP13 28 50 C[C@@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147295077 DE On-Demand Anodyne TRY2_BOVIN 63 42 C[C@@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147295077 DE On-Demand Anodyne MMP2 29 50 C[C@@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147295077 DE On-Demand Anodyne MMP3 15 44 C[C@@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147295077 DE On-Demand Anodyne MMP12 31 43 C[C@@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147295077 DE On-Demand Anodyne ADAMTS4 47 41 C[C@@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147295077 DE On-Demand Anodyne AKR1C3 15 45 C[C@@H](CNS(=O)(=O)c1ccc2ccccc2c1)CC(=O)O ZINC000147295077 DE On-Demand Anodyne Q9JN24_ECOLX 0 43 CCN[C@H](C)CC(=O)NN(C)C ZINC000147295160 AB For-Sale Reactive KDM7A 0 41 CCCCCCCCNC(=O)c1cn[nH]c1C ZINC000147295179 BF On-Demand Mild ASAH1 82 37 Cc1ccc2nc(SCC(=O)O)n(CCNC(N)=O)c2c1 ZINC000147295194 DD For-Sale Anodyne PTGDR2 16 41 CC[C@@H](C)[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147295203 CE For-Sale Anodyne ACE2 48 37 CC[C@@H](C)[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147295203 CE For-Sale Anodyne GPR88 0 50 Cc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1F ZINC000147295244 CD On-Demand Anodyne ENV 47 39 C#CCNC(=O)[C@@H](C)Oc1ccc(S(N)(=O)=O)c(F)c1F ZINC000147295248 DC For-Sale Mild CA2 19 40 C#CCNC(=O)[C@@H](C)Oc1ccc(S(N)(=O)=O)c(F)c1F ZINC000147295248 DC For-Sale Mild CA14 16 40 CCOc1nc(N)nc(Oc2ccccc2[C@@H](C)CC)n1 ZINC000147295265 CG For-Sale Anodyne AO-ACHE 0 41 CC[C@@H]1CN(C(=O)c2ccc(C)cc2C)CC[C@@H]1N ZINC000147295270 CF On-Demand Anodyne L3MBTL1 0 40 C[C@H](CNS(=O)(=O)c1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147295274 DC On-Demand Bother CACNA1D 62 35 C[C@H](CNS(=O)(=O)c1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147295274 DC On-Demand Bother COLA 53 34 Cc1ccc(OCCNC2(C(=O)O)CCC2)cc1 ZINC000147295284 BD For-Sale Anodyne DRD4 19 49 COCCN(C)C(=O)Nc1nc2c(OC)ccc(N3CCOCC3)c2s1 ZINC000147295322 GE For-Sale Clean ADORA2B 18 48 COCCN(C)C(=O)Nc1nc2c(OC)ccc(N3CCOCC3)c2s1 ZINC000147295322 GE For-Sale Clean CASR 32 49 CCCCCCCCNC(=O)c1ccc2[nH]ccc2c1 ZINC000147295387 CI For-Sale Mild FOLH1 19 43 CCCCCCCCNC(=O)c1ccc2[nH]ccc2c1 ZINC000147295387 CI For-Sale Mild KCNQ1 0 42 CCCCCCCCNC(=O)c1ccc2[nH]ccc2c1 ZINC000147295387 CI For-Sale Mild HDAC9 19 44 CCCCCCCCNC(=O)c1ccc2[nH]ccc2c1 ZINC000147295387 CI For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)c1ccc2[nH]ccc2c1 ZINC000147295387 CI For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)c1ccc2[nH]ccc2c1 ZINC000147295387 CI For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)c1ccc2[nH]ccc2c1 ZINC000147295387 CI For-Sale Mild ASAH1 90 38 NC(=O)NCCn1c(SCC(=O)O)nc2ccc(Cl)cc21 ZINC000147295410 ED For-Sale Anodyne PTGDR2 16 43 CC[C@@H](C)[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147295435 CE For-Sale Anodyne ACE2 48 37 CC[C@@H](C)[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147295435 CE For-Sale Anodyne GPR88 0 50 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147295448 HC On-Demand Anodyne HRH2 15 41 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147295448 HC On-Demand Anodyne OPRM1 16 40 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147295448 HC On-Demand Anodyne OPRD1 36 40 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147295448 HC On-Demand Anodyne SFRP1 58 33 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147295448 HC On-Demand Anodyne LIMK2 28 43 CC[C@H]1CN(C(=O)c2ccc(C)cc2C)CC[C@@H]1N ZINC000147295461 CF On-Demand Anodyne L3MBTL1 0 40 C[C@@H](CNS(=O)(=O)c1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147295465 DC On-Demand Bother CACNA1D 62 35 C[C@@H](CNS(=O)(=O)c1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147295465 DC On-Demand Bother COLA 53 34 CC(=O)Cc1ccccc1CC(=O)O ZINC000147295513 AD For-Sale Anodyne CXCL8 43 42 CC(=O)Cc1ccccc1CC(=O)O ZINC000147295513 AD For-Sale Anodyne CPA3 53 33 CCCCCCCCNC(=O)c1cccc2[nH]ccc12 ZINC000147295603 CI For-Sale Mild TPR 17 40 CCCCCCCCNC(=O)c1cccc2[nH]ccc12 ZINC000147295603 CI For-Sale Mild ASAH1 93 38 CCCCCCCCNC(=O)c1cccc2[nH]ccc12 ZINC000147295603 CI For-Sale Mild ACAT 0 47 CCCCCCCCNC(=O)c1cccc2[nH]ccc12 ZINC000147295603 CI For-Sale Mild HPGDS 21 46 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147295640 HC On-Demand Anodyne HRH2 15 41 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147295640 HC On-Demand Anodyne OPRM1 16 40 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147295640 HC On-Demand Anodyne OPRD1 36 40 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147295640 HC On-Demand Anodyne SFRP1 58 33 CCN(CC)C(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147295640 HC On-Demand Anodyne LIMK2 28 43 CC[C@H](C)[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147295665 CE For-Sale Anodyne ACE2 48 37 CC[C@H](C)[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147295665 CE For-Sale Anodyne GPR88 0 50 COc1ccccc1N1CCC(NCc2cc(Cl)c3c(c2)OCCO3)CC1 ZINC000147295669 GH On-Demand Anodyne HTR1A 68 45 COc1ccccc1N1CCC(NCc2cc(Cl)c3c(c2)OCCO3)CC1 ZINC000147295669 GH On-Demand Anodyne DRD2 56 45 COc1ccccc1N1CCC(NCc2cc(Cl)c3c(c2)OCCO3)CC1 ZINC000147295669 GH On-Demand Anodyne DRD4 36 45 COc1ccccc1N1CCC(NCc2cc(Cl)c3c(c2)OCCO3)CC1 ZINC000147295669 GH On-Demand Anodyne ADRA1D 55 42 COc1ccccc1N1CCC(NCc2cc(Cl)c3c(c2)OCCO3)CC1 ZINC000147295669 GH On-Demand Anodyne ADRA1A 47 42 COc1ccccc1N1CCC(NCc2cc(Cl)c3c(c2)OCCO3)CC1 ZINC000147295669 GH On-Demand Anodyne ADRA1B 42 42 COc1ccccc1N1CCC(NCc2cc(Cl)c3c(c2)OCCO3)CC1 ZINC000147295669 GH On-Demand Anodyne DRD3 51 45 COc1ccccc1N1CCC(NCc2cc(Cl)c3c(c2)OCCO3)CC1 ZINC000147295669 GH On-Demand Anodyne HTR7 41 45 CC[C@@H]1CN(C(=O)c2ccc(C)cc2C)CC[C@H]1N ZINC000147295682 CF On-Demand Anodyne L3MBTL1 0 40 NS(=O)(=O)c1ccc(OCc2ccncc2Cl)c(F)c1F ZINC000147295699 EE For-Sale Anodyne CA14 26 45 C[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295708 CD On-Demand Anodyne KCNA5 0 42 C[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295708 CD On-Demand Anodyne MMP13 24 49 C[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295708 CD On-Demand Anodyne CA4 17 43 C[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295708 CD On-Demand Anodyne MMP8 20 49 C[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295708 CD On-Demand Anodyne MMP9 22 52 C[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295708 CD On-Demand Anodyne MMP12 26 48 C[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295708 CD On-Demand Anodyne MMP10 17 52 C[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295708 CD On-Demand Anodyne ADAMTS4 46 38 C[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295708 CD On-Demand Anodyne LIMK2 43 38 C[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295708 CD On-Demand Anodyne Q9JN24_ECOLX 0 40 COc1ccc(C)cc1CNCC(F)F ZINC000147295776 BE On-Demand Anodyne PHES 0 48 COC(=O)c1cccc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1C ZINC000147295817 GF On-Demand Anodyne ADRB2 18 43 CCCCCCNCCP(=O)(OCC)OCC ZINC000147295822 CG For-Sale Anodyne FDPS 39 43 CCCCCCNCCP(=O)(OCC)OCC ZINC000147295822 CG For-Sale Anodyne S1PR4 21 59 CCCCCCNCCP(=O)(OCC)OCC ZINC000147295822 CG For-Sale Anodyne LPAR2 73 38 CCCCCCNCCP(=O)(OCC)OCC ZINC000147295822 CG For-Sale Anodyne S1PR3 46 59 CCCCCCNCCP(=O)(OCC)OCC ZINC000147295822 CG For-Sale Anodyne S1PR2 92 59 CCCCCCNCCP(=O)(OCC)OCC ZINC000147295822 CG For-Sale Anodyne S1PR1 18 59 CCCCCCNCCP(=O)(OCC)OCC ZINC000147295822 CG For-Sale Anodyne LPAR3 41 41 CCCCCCNCCP(=O)(OCC)OCC ZINC000147295822 CG For-Sale Anodyne Q8WS26_TRYCR 54 47 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(F)c(C(F)(F)F)c2)C1 ZINC000147295838 HD On-Demand Anodyne SFRP1 141 42 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(F)c(C(F)(F)F)c2)C1 ZINC000147295838 HD On-Demand Anodyne WNT3 94 38 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild GABRA1 15 47 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild CNR1 19 40 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild DRD3 15 53 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild TPR 21 53 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild TSPO 32 55 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild CCKAR 42 54 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild BCHE 25 48 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild MC3R 41 32 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild MC5R 50 32 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild MMP2 23 47 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild MMP8 28 47 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild GRIA1 46 45 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild CFTR 38 47 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild ALOX15 25 44 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild MC1R 53 40 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild MMP1 22 47 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild KISS1R 64 33 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild ASAH1 95 39 CCCCCCCCNC(=O)c1c[nH]c2ccccc12 ZINC000147295854 CI For-Sale Mild ACAT 0 45 CC[C@@H](C)[C@@H](NC(=O)c1ccc(C)c(Br)c1)C(=O)O ZINC000147295883 EF On-Demand Anodyne CA2 25 59 CC[C@@H](C)[C@@H](NC(=O)c1ccc(C)c(Br)c1)C(=O)O ZINC000147295883 EF On-Demand Anodyne CA4 15 59 CC[C@H]1CN(C(=O)c2ccc(C)cc2C)CC[C@H]1N ZINC000147295894 CF On-Demand Anodyne L3MBTL1 0 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(F)c(-c2nnc3n2CCCCC3)c1 ZINC000147295906 HF On-Demand Anodyne F2R 40 32 C[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295910 CD On-Demand Anodyne KCNA5 0 42 C[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295910 CD On-Demand Anodyne MMP13 24 49 C[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295910 CD On-Demand Anodyne CA4 17 43 C[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295910 CD On-Demand Anodyne MMP8 20 49 C[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295910 CD On-Demand Anodyne MMP9 22 52 C[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295910 CD On-Demand Anodyne MMP12 26 48 C[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295910 CD On-Demand Anodyne MMP10 17 52 C[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295910 CD On-Demand Anodyne ADAMTS4 46 38 C[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295910 CD On-Demand Anodyne LIMK2 43 38 C[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147295910 CD On-Demand Anodyne Q9JN24_ECOLX 0 40 COC(=O)c1cccc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1C ZINC000147296025 GF On-Demand Anodyne ADRB2 18 43 CC[C@H](C)[C@@H](NC(=O)c1ccc(C)c(Br)c1)C(=O)O ZINC000147296058 EF On-Demand Anodyne CA2 25 59 CC[C@H](C)[C@@H](NC(=O)c1ccc(C)c(Br)c1)C(=O)O ZINC000147296058 EF On-Demand Anodyne CA4 15 59 CCCCCCCCNC(=O)c1n[nH]c(CCC)n1 ZINC000147296090 CF For-Sale Mild ASAH1 75 35 CCCCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147296093 HD On-Demand Anodyne HRH2 18 48 CCCCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147296093 HD On-Demand Anodyne HRH3 22 48 CCCCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147296093 HD On-Demand Anodyne MMP13 36 43 CCCCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147296093 HD On-Demand Anodyne MMP2 17 43 CCCCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147296093 HD On-Demand Anodyne MMP3 23 43 CCCCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147296093 HD On-Demand Anodyne PLA2G4B 70 34 CCCCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147296093 HD On-Demand Anodyne MMP1 19 41 CC[C@@H]1CN(C(=O)c2ccc3c(c2)OCCO3)CC[C@@H]1N ZINC000147296105 CD On-Demand Anodyne L3MBTL3 61 35 C[C@H](CNS(=O)(=O)c1ccc(Cl)c(Cl)c1)CC(=O)O ZINC000147296133 EE On-Demand Anodyne TBXA2R 42 34 C[C@H](CNS(=O)(=O)c1ccc(Cl)c(Cl)c1)CC(=O)O ZINC000147296133 EE On-Demand Anodyne KMO 0 40 O=C(NC[C@@H]1CCCOC1)c1cnn(-c2ccccc2Cl)c1 ZINC000147296176 DF On-Demand Anodyne CACNA1I 43 34 CCCCCCCCNC(=O)c1n[nH]c(C(C)C)n1 ZINC000147296296 CG For-Sale Mild ASAH1 82 35 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cccc3cnccc23)C1 ZINC000147296308 FC On-Demand Anodyne P2RX7 39 42 CC[C@H]1CN(C(=O)c2ccc3c(c2)OCCO3)CC[C@@H]1N ZINC000147296310 CD On-Demand Anodyne L3MBTL3 61 35 C[C@@H](CNS(=O)(=O)c1ccc(Cl)c(Cl)c1)CC(=O)O ZINC000147296352 EE On-Demand Anodyne TBXA2R 42 34 C[C@@H](CNS(=O)(=O)c1ccc(Cl)c(Cl)c1)CC(=O)O ZINC000147296352 EE On-Demand Anodyne KMO 0 40 O=C(NC[C@H]1CCCOC1)c1cnn(-c2ccccc2Cl)c1 ZINC000147296376 DF On-Demand Anodyne CACNA1I 43 34 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1Br ZINC000147296389 HI On-Demand Anodyne HTR1A 84 42 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1Br ZINC000147296389 HI On-Demand Anodyne DRD2 74 43 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1Br ZINC000147296389 HI On-Demand Anodyne DRD1 17 41 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1Br ZINC000147296389 HI On-Demand Anodyne DRD4 41 43 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1Br ZINC000147296389 HI On-Demand Anodyne ADRA1D 79 41 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1Br ZINC000147296389 HI On-Demand Anodyne HTR2A 21 41 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1Br ZINC000147296389 HI On-Demand Anodyne ADRA1A 68 41 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1Br ZINC000147296389 HI On-Demand Anodyne ADRA1B 62 41 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1Br ZINC000147296389 HI On-Demand Anodyne DRD3 70 43 COc1ccc(CNC2CCN(c3ccccc3OC)CC2)cc1Br ZINC000147296389 HI On-Demand Anodyne HTR7 49 42 FC(F)(F)Oc1ccc(CN2[C@@H]3CC[C@@H]2CC(Br)C3)cc1 ZINC000147296400 FI For-Sale Reactive HCRTR1 25 40 FC(F)(F)Oc1ccc(CN2[C@@H]3CC[C@@H]2CC(Br)C3)cc1 ZINC000147296400 FI For-Sale Reactive HCRTR2 29 40 COC(=O)c1cccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c1C ZINC000147296465 DG On-Demand Anodyne EPHX2 25 46 CC[C@@H]1CN(C(=O)c2ccc3c(c2)OCCO3)CC[C@H]1N ZINC000147296487 CD On-Demand Anodyne L3MBTL3 61 35 CCCCCCCCNC(=O)C1=NNC(=O)CC1 ZINC000147296488 CD For-Sale Mild ASAH1 96 41 COc1nc(N)nc(Oc2ccc(Cl)cc2Br)n1 ZINC000147296509 EF For-Sale Anodyne AGPAT2 39 42 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2cccc3cnccc23)C1 ZINC000147296523 FC On-Demand Anodyne P2RX7 39 42 Cc1ccc(F)c(S(=O)(=O)NC[C@@H](C)CC(=O)O)c1 ZINC000147296575 CD On-Demand Anodyne LEF 46 36 COc1ccc2c(c1)OC[C@H](C(=O)NC[C@@H]1CCCOC1)C2 ZINC000147296612 DD On-Demand Anodyne MTR1B_CHICK 0 40 COc1ccc2c(c1)OC[C@H](C(=O)NC[C@@H]1CCCOC1)C2 ZINC000147296612 DD On-Demand Anodyne MTNR1A 33 42 COc1ccc2c(c1)OC[C@H](C(=O)NC[C@@H]1CCCOC1)C2 ZINC000147296612 DD On-Demand Anodyne ROCK2 23 41 CCN(CC)S(=O)(=O)c1ccc([C@@H](C)NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147296625 HG On-Demand Bother COLA 43 34 CCN(CC)S(=O)(=O)c1ccc([C@@H](C)NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147296625 HG On-Demand Bother MMP8 25 40 CCN(CC)S(=O)(=O)c1ccc([C@@H](C)NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147296625 HG On-Demand Bother MMP1 17 40 FC(F)(F)Oc1ccc(CN2[C@H]3CC[C@@H]2CC(Br)C3)cc1 ZINC000147296639 FI For-Sale Reactive HCRTR1 25 40 FC(F)(F)Oc1ccc(CN2[C@H]3CC[C@@H]2CC(Br)C3)cc1 ZINC000147296639 FI For-Sale Reactive HCRTR2 29 40 CCCCCCCCNC(=O)c1ccc2cc[nH]c2c1 ZINC000147296679 CI For-Sale Mild DRD2 17 41 CCCCCCCCNC(=O)c1ccc2cc[nH]c2c1 ZINC000147296679 CI For-Sale Mild DRD3 41 43 CCCCCCCCNC(=O)c1ccc2cc[nH]c2c1 ZINC000147296679 CI For-Sale Mild FOLH1 19 43 CCCCCCCCNC(=O)c1ccc2cc[nH]c2c1 ZINC000147296679 CI For-Sale Mild KCNQ1 0 44 CCCCCCCCNC(=O)c1ccc2cc[nH]c2c1 ZINC000147296679 CI For-Sale Mild HDAC9 20 46 CCCCCCCCNC(=O)c1ccc2cc[nH]c2c1 ZINC000147296679 CI For-Sale Mild GNAI1 0 40 CCCCCCCCNC(=O)c1ccc2cc[nH]c2c1 ZINC000147296679 CI For-Sale Mild GNAI3 0 40 CCCCCCCCNC(=O)c1ccc2cc[nH]c2c1 ZINC000147296679 CI For-Sale Mild GNAO1 0 40 CCCCCCCCNC(=O)c1ccc2cc[nH]c2c1 ZINC000147296679 CI For-Sale Mild ASAH1 94 38 CCCCCCCCNC(=O)c1ccc2cc[nH]c2c1 ZINC000147296679 CI For-Sale Mild ACAT 0 43 COC(=O)c1cccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1C ZINC000147296690 DG On-Demand Anodyne EPHX2 25 46 FC(F)CNCc1ccc(Cl)cc1Cl ZINC000147296694 BG On-Demand Anodyne P2RX7 27 41 CC[C@H]1CN(C(=O)c2ccc3c(c2)OCCO3)CC[C@H]1N ZINC000147296699 CD On-Demand Anodyne L3MBTL3 61 35 CCCCCCCCCCCCCCCC[C@@H](C)OC[C@H](O)CO ZINC000147296773 EK For-Sale Mild CQSS 41 33 Cc1ccc(F)c(S(=O)(=O)NC[C@H](C)CC(=O)O)c1 ZINC000147296797 CD On-Demand Anodyne LEF 46 36 COc1ccc2c(c1)OC[C@@H](C(=O)NC[C@@H]1CCCOC1)C2 ZINC000147296808 DD On-Demand Anodyne MTR1B_CHICK 0 40 COc1ccc2c(c1)OC[C@@H](C(=O)NC[C@@H]1CCCOC1)C2 ZINC000147296808 DD On-Demand Anodyne MTNR1A 33 42 COc1ccc2c(c1)OC[C@@H](C(=O)NC[C@@H]1CCCOC1)C2 ZINC000147296808 DD On-Demand Anodyne ROCK2 23 41 FC(F)(F)Oc1ccc(CN2[C@H]3CC[C@H]2CC(Br)C3)cc1 ZINC000147296853 FI For-Sale Reactive HCRTR1 25 40 FC(F)(F)Oc1ccc(CN2[C@H]3CC[C@H]2CC(Br)C3)cc1 ZINC000147296853 FI For-Sale Reactive HCRTR2 29 40 COc1ccccc1N1CCC(NCc2cc(Br)c3c(c2)OCO3)CC1 ZINC000147296867 HH On-Demand Anodyne HTR1A 59 43 COc1ccccc1N1CCC(NCc2cc(Br)c3c(c2)OCO3)CC1 ZINC000147296867 HH On-Demand Anodyne DRD2 47 43 COc1ccccc1N1CCC(NCc2cc(Br)c3c(c2)OCO3)CC1 ZINC000147296867 HH On-Demand Anodyne DRD4 26 41 COc1ccccc1N1CCC(NCc2cc(Br)c3c(c2)OCO3)CC1 ZINC000147296867 HH On-Demand Anodyne ADRA1D 48 48 COc1ccccc1N1CCC(NCc2cc(Br)c3c(c2)OCO3)CC1 ZINC000147296867 HH On-Demand Anodyne ADRA1A 42 48 COc1ccccc1N1CCC(NCc2cc(Br)c3c(c2)OCO3)CC1 ZINC000147296867 HH On-Demand Anodyne ADRA1B 38 48 COc1ccccc1N1CCC(NCc2cc(Br)c3c(c2)OCO3)CC1 ZINC000147296867 HH On-Demand Anodyne DRD3 43 41 COc1ccccc1N1CCC(NCc2cc(Br)c3c(c2)OCO3)CC1 ZINC000147296867 HH On-Demand Anodyne HTR7 37 41 CCN(CC)S(=O)(=O)c1ccc([C@H](C)NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147296878 HG On-Demand Bother COLA 43 34 CCN(CC)S(=O)(=O)c1ccc([C@H](C)NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147296878 HG On-Demand Bother MMP8 25 40 CCN(CC)S(=O)(=O)c1ccc([C@H](C)NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147296878 HG On-Demand Bother MMP1 17 40 CCCCCCCCNC(=O)c1n[nH]c(CC)n1 ZINC000147296888 CE For-Sale Mild EPHX2 28 41 CCCCCCCCNC(=O)c1n[nH]c(CC)n1 ZINC000147296888 CE For-Sale Mild ASAH1 86 38 COC(=O)c1cccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1C ZINC000147296928 DG On-Demand Anodyne EPHX2 25 46 c1ccc(Nc2ncc(-c3ccccc3)cn2)cc1 ZINC000147296945 BH For-Sale Anodyne PLK1 26 48 c1ccc(Nc2ncc(-c3ccccc3)cn2)cc1 ZINC000147296945 BH For-Sale Anodyne GSK3A 15 41 c1ccc(Nc2ncc(-c3ccccc3)cn2)cc1 ZINC000147296945 BH For-Sale Anodyne AURKA 17 50 C[C@H](NCC(F)F)c1cccc([N+](=O)[O-])c1 ZINC000147296946 BF On-Demand Bother CACNA1D 40 34 Fc1ccc(Cn2cc(Cl)c(I)n2)c(Cl)c1 ZINC000147296967 FH For-Sale Anodyne P2RX7 40 38 CCCCCCCCCCCCCCCC[C@H](C)OC[C@H](O)CO ZINC000147296975 EK For-Sale Mild CQSS 41 33 C[C@H](CNS(=O)(=O)c1ccc(F)c(C#N)c1)CC(=O)O ZINC000147296982 DD On-Demand Mild TBXA2R 43 36 C[C@H](CNS(=O)(=O)c1ccc(F)c(C#N)c1)CC(=O)O ZINC000147296982 DD On-Demand Mild LEF 55 35 COc1ccc2c(c1)OC[C@H](C(=O)NC[C@H]1CCCOC1)C2 ZINC000147297007 DD On-Demand Anodyne MTR1B_CHICK 0 40 COc1ccc2c(c1)OC[C@H](C(=O)NC[C@H]1CCCOC1)C2 ZINC000147297007 DD On-Demand Anodyne MTNR1A 33 42 COc1ccc2c(c1)OC[C@H](C(=O)NC[C@H]1CCCOC1)C2 ZINC000147297007 DD On-Demand Anodyne ROCK2 23 41 CN(C)C[C@@H]1CCCN1C(=O)c1cccc2c1OCCN2 ZINC000147297013 CD For-Sale Anodyne HCRTR1 0 41 CN(C)C[C@@H]1CCCN1C(=O)c1cccc2c1OCCN2 ZINC000147297013 CD For-Sale Anodyne HCRTR2 0 41 COc1ccccc1N1CCC(NCc2cc(Br)ccc2F)CC1 ZINC000147297112 GI On-Demand Anodyne HTR1A 74 44 COc1ccccc1N1CCC(NCc2cc(Br)ccc2F)CC1 ZINC000147297112 GI On-Demand Anodyne DRD2 65 44 COc1ccccc1N1CCC(NCc2cc(Br)ccc2F)CC1 ZINC000147297112 GI On-Demand Anodyne DRD1 16 42 COc1ccccc1N1CCC(NCc2cc(Br)ccc2F)CC1 ZINC000147297112 GI On-Demand Anodyne DRD4 41 44 COc1ccccc1N1CCC(NCc2cc(Br)ccc2F)CC1 ZINC000147297112 GI On-Demand Anodyne ADRA1D 76 43 COc1ccccc1N1CCC(NCc2cc(Br)ccc2F)CC1 ZINC000147297112 GI On-Demand Anodyne HTR2A 17 42 COc1ccccc1N1CCC(NCc2cc(Br)ccc2F)CC1 ZINC000147297112 GI On-Demand Anodyne ADRA1A 65 43 COc1ccccc1N1CCC(NCc2cc(Br)ccc2F)CC1 ZINC000147297112 GI On-Demand Anodyne ADRA1B 61 43 COc1ccccc1N1CCC(NCc2cc(Br)ccc2F)CC1 ZINC000147297112 GI On-Demand Anodyne DRD3 63 44 COc1ccccc1N1CCC(NCc2cc(Br)ccc2F)CC1 ZINC000147297112 GI On-Demand Anodyne HTR7 50 44 CCCCCCCCNC(=O)c1ccc2cn[nH]c2c1 ZINC000147297139 CH For-Sale Mild DRD3 36 41 CCCCCCCCNC(=O)c1ccc2cn[nH]c2c1 ZINC000147297139 CH For-Sale Mild FOLH1 25 44 CCCCCCCCNC(=O)c1ccc2cn[nH]c2c1 ZINC000147297139 CH For-Sale Mild CCKAR 0 40 CCCCCCCCNC(=O)c1ccc2cn[nH]c2c1 ZINC000147297139 CH For-Sale Mild HDAC9 20 45 CCCCCCCCNC(=O)c1ccc2cn[nH]c2c1 ZINC000147297139 CH For-Sale Mild ASAH1 88 38 CC(C)C[C@H](CN)CC(=O)NN(C)C ZINC000147297144 BC For-Sale Reactive CACNA2D1 0 56 COC(=O)c1cccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c1C ZINC000147297145 DG On-Demand Anodyne EPHX2 25 46 C[C@@H](NCC(F)F)c1cccc([N+](=O)[O-])c1 ZINC000147297163 BF On-Demand Bother CACNA1D 40 34 COc1ccc2c(c1)OC[C@@H](C(=O)NC[C@H]1CCCOC1)C2 ZINC000147297182 DD On-Demand Anodyne MTR1B_CHICK 0 40 COc1ccc2c(c1)OC[C@@H](C(=O)NC[C@H]1CCCOC1)C2 ZINC000147297182 DD On-Demand Anodyne MTNR1A 33 42 COc1ccc2c(c1)OC[C@@H](C(=O)NC[C@H]1CCCOC1)C2 ZINC000147297182 DD On-Demand Anodyne ROCK2 23 41 CCCCCCCCCCCCCCCC[C@@H](C)OC[C@@H](O)CO ZINC000147297183 EK For-Sale Mild CQSS 41 33 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297212 GC On-Demand Anodyne HTR1A 46 51 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297212 GC On-Demand Anodyne DRD2 42 44 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297212 GC On-Demand Anodyne DRD4 23 44 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297212 GC On-Demand Anodyne ADRA1D 26 40 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297212 GC On-Demand Anodyne HTR2A 39 44 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297212 GC On-Demand Anodyne HTR2C 34 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297212 GC On-Demand Anodyne ADRA1A 28 40 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297212 GC On-Demand Anodyne DRD3 55 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297212 GC On-Demand Anodyne FURIN 42 32 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297212 GC On-Demand Anodyne HPN 66 33 C[C@@H](CNS(=O)(=O)c1ccc(F)c(C#N)c1)CC(=O)O ZINC000147297217 DD On-Demand Mild TBXA2R 43 36 C[C@@H](CNS(=O)(=O)c1ccc(F)c(C#N)c1)CC(=O)O ZINC000147297217 DD On-Demand Mild LEF 55 35 CN(C)C[C@H]1CCCN1C(=O)c1cccc2c1OCCN2 ZINC000147297226 CD For-Sale Anodyne HCRTR1 0 41 CN(C)C[C@H]1CCCN1C(=O)c1cccc2c1OCCN2 ZINC000147297226 CD For-Sale Anodyne HCRTR2 0 41 Cc1ccc(S(C)(=O)=O)cc1S(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000147297235 HC On-Demand Anodyne SFRP1 125 36 Cc1ccc(S(C)(=O)=O)cc1S(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000147297235 HC On-Demand Anodyne WNT3 83 34 CCNc1ncnc(Oc2ccc(Cl)cc2Br)c1[N+](=O)[O-] ZINC000147297249 FI For-Sale Bother S1PR4 20 47 CN(Cc1cscn1)C(=O)NCc1ccccc1CN1CCOCC1 ZINC000147297296 FE On-Demand Anodyne SCN5A 40 35 COC(=O)c1cccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1C ZINC000147297351 FD On-Demand Anodyne LPL 43 33 COC(=O)c1cccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1C ZINC000147297351 FD On-Demand Anodyne EPHX2 33 42 COCCOc1ccc2c(c1)c(C#N)cn2-c1ccc(C(=O)O)cc1 ZINC000147297370 EG Annotated Anodyne PLA2G4A 45 42 COCCOc1ccc2c(c1)c(C#N)cn2-c1ccc(C(=O)O)cc1 ZINC000147297370 EG Annotated Anodyne PLA2G4B 41 34 COCCOc1ccc2c(c1)c(C#N)cn2-c1ccc(C(=O)O)cc1 ZINC000147297370 EG Annotated Anodyne PFKFB3 50 42 CCCCCCCCNC(=O)c1[nH]nc2ccccc12 ZINC000147297371 CH For-Sale Mild ACHE 41 38 CCCCCCCCNC(=O)c1[nH]nc2ccccc12 ZINC000147297371 CH For-Sale Mild DRD3 16 54 CCCCCCCCNC(=O)c1[nH]nc2ccccc12 ZINC000147297371 CH For-Sale Mild TSPO 23 47 CCCCCCCCNC(=O)c1[nH]nc2ccccc12 ZINC000147297371 CH For-Sale Mild BCHE 57 38 CCCCCCCCNC(=O)c1[nH]nc2ccccc12 ZINC000147297371 CH For-Sale Mild ASAH1 97 38 CCCCCCCCCCCCCCCC[C@H](C)OC[C@@H](O)CO ZINC000147297421 EK For-Sale Mild CQSS 41 33 Cc1ccc(S(C)(=O)=O)cc1S(=O)(=O)N[C@H]1CCCN(S(C)(=O)=O)C1 ZINC000147297439 HC On-Demand Anodyne SFRP1 125 36 Cc1ccc(S(C)(=O)=O)cc1S(=O)(=O)N[C@H]1CCCN(S(C)(=O)=O)C1 ZINC000147297439 HC On-Demand Anodyne WNT3 83 34 CC(C)n1cc(NC(=O)c2cccc3c2OCCN3)cn1 ZINC000147297444 CF For-Sale Anodyne ITK 46 32 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297460 GC On-Demand Anodyne HTR1A 46 51 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297460 GC On-Demand Anodyne DRD2 42 44 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297460 GC On-Demand Anodyne DRD4 23 44 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297460 GC On-Demand Anodyne ADRA1D 26 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297460 GC On-Demand Anodyne HTR2A 39 44 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297460 GC On-Demand Anodyne HTR2C 34 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297460 GC On-Demand Anodyne ADRA1A 28 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297460 GC On-Demand Anodyne DRD3 55 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297460 GC On-Demand Anodyne FURIN 42 32 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2ncccn2)CC1 ZINC000147297460 GC On-Demand Anodyne HPN 66 33 CNc1cccc(Oc2ccc(Cl)cc2Br)c1[N+](=O)[O-] ZINC000147297481 FJ For-Sale Bother ENR 0 45 O=C(O)c1ccc2c(c1)N(S(=O)(=O)c1ccccc1)CC2 ZINC000147297495 DE For-Sale Anodyne MMP26 0 41 O=C(O)c1ccc2c(c1)N(S(=O)(=O)c1ccccc1)CC2 ZINC000147297495 DE For-Sale Anodyne CYP11B2 34 46 O=C(O)c1ccc2c(c1)N(S(=O)(=O)c1ccccc1)CC2 ZINC000147297495 DE For-Sale Anodyne CPT1A 40 52 O=C(O)c1ccc2c(c1)N(S(=O)(=O)c1ccccc1)CC2 ZINC000147297495 DE For-Sale Anodyne MMP15 0 41 O=C(O)c1ccc2c(c1)N(S(=O)(=O)c1ccccc1)CC2 ZINC000147297495 DE For-Sale Anodyne MMP16 0 41 O=C(O)c1ccc2c(c1)N(S(=O)(=O)c1ccccc1)CC2 ZINC000147297495 DE For-Sale Anodyne CPT1B 26 47 O=C(O)c1ccc2c(c1)N(S(=O)(=O)c1ccccc1)CC2 ZINC000147297495 DE For-Sale Anodyne AKR1C3 31 45 O=C(O)c1ccc2c(c1)N(S(=O)(=O)c1ccccc1)CC2 ZINC000147297495 DE For-Sale Anodyne AKR1C1 31 43 COc1ccc(C(=O)c2c(C)n(-c3cccc(O)c3)c3cc(OC(F)(F)F)ccc23)cc1 ZINC000147297498 IK For-Sale Anodyne HPD 22 44 COc1ccc(C(=O)c2c(C)n(-c3cccc(O)c3)c3cc(OC(F)(F)F)ccc23)cc1 ZINC000147297498 IK For-Sale Anodyne PPARG 32 54 COc1ccc(C(=O)c2c(C)n(-c3cccc(O)c3)c3cc(OC(F)(F)F)ccc23)cc1 ZINC000147297498 IK For-Sale Anodyne PTGDS 27 41 O[C@@H]1C[C@@H](Cc2ccccc2)CN(Cc2ccccc2)C1 ZINC000147297539 CG For-Sale Anodyne DRD4 20 40 O[C@@H]1C[C@@H](Cc2ccccc2)CN(Cc2ccccc2)C1 ZINC000147297539 CG For-Sale Anodyne SIGMAR1 54 44 COC(=O)c1cccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1C ZINC000147297565 FD On-Demand Anodyne LPL 43 33 COC(=O)c1cccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1C ZINC000147297565 FD On-Demand Anodyne EPHX2 33 42 O=C(CCNC1(C(=O)O)CCC1)Nc1cccc(F)c1 ZINC000147297572 CD For-Sale Anodyne FUCA1 15 43 O=C(CCNC1(C(=O)O)CCC1)Nc1cccc(F)c1 ZINC000147297572 CD For-Sale Anodyne KCNK3 15 40 CCCCCCCCNC(=O)c1nc(C)n[nH]1 ZINC000147297577 BE For-Sale Mild ASAH1 86 38 Cc1ncoc1C(=O)N1CCc2ccccc2[C@@H]1C(=O)O ZINC000147297652 CD On-Demand Anodyne MTNR1B 0 40 O=C(Nc1cc(Br)ccc1Cl)c1cccc2c1OCCN2 ZINC000147297661 FI For-Sale Anodyne G2YM83_BOTF4 51 32 O[C@H]1C[C@@H](Cc2ccccc2)CN(Cc2ccccc2)C1 ZINC000147297749 CG For-Sale Anodyne DRD4 20 40 O[C@H]1C[C@@H](Cc2ccccc2)CN(Cc2ccccc2)C1 ZINC000147297749 CG For-Sale Anodyne SIGMAR1 54 44 Cc1ccc([C@@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147297787 CG For-Sale Anodyne DRD2 26 52 Cc1ccc([C@@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147297787 CG For-Sale Anodyne DRD4 67 52 Cc1ccc([C@@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147297787 CG For-Sale Anodyne ACHE 39 49 Cc1ccc([C@@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147297787 CG For-Sale Anodyne DRD3 35 47 Cc1ccc([C@@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147297787 CG For-Sale Anodyne SIGMAR1 66 43 Cc1ccc([C@@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147297787 CG For-Sale Anodyne CCR5 23 47 Cc1ccc([C@@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147297787 CG For-Sale Anodyne AKT2 55 34 Cc1ccc([C@@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147297787 CG For-Sale Anodyne SLC18A3 24 40 Cc1ccc([C@@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147297787 CG For-Sale Anodyne SCN5A 35 42 CCCCCCCCNC(=O)c1n[nH]c(C2CC2)n1 ZINC000147297790 CF For-Sale Mild GNAI1 0 42 CCCCCCCCNC(=O)c1n[nH]c(C2CC2)n1 ZINC000147297790 CF For-Sale Mild GNAI3 0 42 CCCCCCCCNC(=O)c1n[nH]c(C2CC2)n1 ZINC000147297790 CF For-Sale Mild GNAO1 0 42 CCCCCCCCNC(=O)c1n[nH]c(C2CC2)n1 ZINC000147297790 CF For-Sale Mild ASAH1 67 35 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2c(C)cc(C)cc2C)c1 ZINC000147297799 EH On-Demand Bother NQO2 45 37 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2c(C)cc(C)cc2C)c1 ZINC000147297799 EH On-Demand Bother MTNR1A 74 38 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2c(C)cc(C)cc2C)c1 ZINC000147297799 EH On-Demand Bother MTNR1B 66 38 CS(=O)(=O)NCCc1ccc(-c2ccc(CCNS(C)(=O)=O)cc2)cc1 ZINC000147297827 GD For-Sale Anodyne CA2 16 47 CS(=O)(=O)NCCc1ccc(-c2ccc(CCNS(C)(=O)=O)cc2)cc1 ZINC000147297827 GD For-Sale Anodyne CA1 17 47 CS(=O)(=O)NCCc1ccc(-c2ccc(CCNS(C)(=O)=O)cc2)cc1 ZINC000147297827 GD For-Sale Anodyne GRIA4 16 65 CS(=O)(=O)NCCc1ccc(-c2ccc(CCNS(C)(=O)=O)cc2)cc1 ZINC000147297827 GD For-Sale Anodyne CA9 15 47 CS(=O)(=O)NCCc1ccc(-c2ccc(CCNS(C)(=O)=O)cc2)cc1 ZINC000147297827 GD For-Sale Anodyne A6YCJ1_9METZ 15 41 Cc1ncoc1C(=O)N1CCc2ccccc2[C@H]1C(=O)O ZINC000147297849 CD On-Demand Anodyne MTNR1B 0 40 COc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1OC ZINC000147297873 DD On-Demand Anodyne IAP 0 41 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1OC ZINC000147297919 FG For-Sale Reactive GRM3 29 49 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1OC ZINC000147297919 FG For-Sale Reactive L3MBTL3 53 35 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1OC ZINC000147297919 FG For-Sale Reactive ACKR3 72 40 O[C@@H]1C[C@H](Cc2ccccc2)CN(Cc2ccccc2)C1 ZINC000147297943 CG For-Sale Anodyne DRD4 20 40 O[C@@H]1C[C@H](Cc2ccccc2)CN(Cc2ccccc2)C1 ZINC000147297943 CG For-Sale Anodyne SIGMAR1 54 44 COc1cccc(CCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1OC ZINC000147297990 HD On-Demand Bother NQO2 48 45 COc1cccc(CCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1OC ZINC000147297990 HD On-Demand Bother MTNR1A 43 45 COc1cccc(CCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1OC ZINC000147297990 HD On-Demand Bother MTNR1B 30 45 Cc1ccc([C@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147298006 CG For-Sale Anodyne DRD2 26 52 Cc1ccc([C@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147298006 CG For-Sale Anodyne DRD4 67 52 Cc1ccc([C@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147298006 CG For-Sale Anodyne ACHE 39 49 Cc1ccc([C@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147298006 CG For-Sale Anodyne DRD3 35 47 Cc1ccc([C@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147298006 CG For-Sale Anodyne SIGMAR1 66 43 Cc1ccc([C@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147298006 CG For-Sale Anodyne CCR5 23 47 Cc1ccc([C@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147298006 CG For-Sale Anodyne AKT2 55 34 Cc1ccc([C@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147298006 CG For-Sale Anodyne SLC18A3 24 40 Cc1ccc([C@H]2CCN(Cc3ccccc3)C2)nc1 ZINC000147298006 CG For-Sale Anodyne SCN5A 35 42 CCCCCCCCNS(=O)(=O)C[C@@H](C)CCl ZINC000147298018 CG For-Sale Reactive RELA 19 44 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1N1CCCCC1 ZINC000147298029 EE On-Demand Anodyne KCNQ2 92 47 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1N1CCCCC1 ZINC000147298029 EE On-Demand Anodyne CSF1R 20 47 O=C(N[C@H](C(=O)O)C1CC1)c1cccc(F)c1Cl ZINC000147298057 CE On-Demand Anodyne NTSR2 42 43 O=C(N[C@H](C(=O)O)C1CC1)c1cccc(F)c1Cl ZINC000147298057 CE On-Demand Anodyne PYGL 30 49 COc1ccccc1N1CCC(NCc2ccc(OCCN(C)C)cc2)CC1 ZINC000147298078 GG On-Demand Anodyne HTR1A 71 46 COc1ccccc1N1CCC(NCc2ccc(OCCN(C)C)cc2)CC1 ZINC000147298078 GG On-Demand Anodyne DRD2 58 49 COc1ccccc1N1CCC(NCc2ccc(OCCN(C)C)cc2)CC1 ZINC000147298078 GG On-Demand Anodyne ADRA1D 51 38 COc1ccccc1N1CCC(NCc2ccc(OCCN(C)C)cc2)CC1 ZINC000147298078 GG On-Demand Anodyne ADRA1A 46 38 COc1ccccc1N1CCC(NCc2ccc(OCCN(C)C)cc2)CC1 ZINC000147298078 GG On-Demand Anodyne DRD3 57 49 COc1ccccc1N1CCC(NCc2ccc(OCCN(C)C)cc2)CC1 ZINC000147298078 GG On-Demand Anodyne LTA4H 19 43 COc1ccccc1N1CCC(NCc2ccc(OCCN(C)C)cc2)CC1 ZINC000147298078 GG On-Demand Anodyne HTR7 49 42 COc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1OC ZINC000147298089 DD On-Demand Anodyne IAP 0 41 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1OC ZINC000147298117 FG For-Sale Reactive GRM3 29 49 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1OC ZINC000147298117 FG For-Sale Reactive L3MBTL3 53 35 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1OC ZINC000147298117 FG For-Sale Reactive ACKR3 72 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CA2 62 49 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne PTGS1 19 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne PTGS2 69 50 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CA6 20 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CA1 57 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CA7 57 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CA13 29 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CA4 37 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CA12 52 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CA9 57 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CAH_METTE 54 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CYNT 36 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne NCE103 31 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CA15 29 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne P96878_MYCTU 37 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne CA 0 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne A6YCJ1_9METZ 35 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)cc1 ZINC000147298163 DF For-Sale Anodyne Q5TU56_ANOGA 0 42 Cc1c(NCCCCC(C)C)cc(N)cc1S(N)(=O)=O ZINC000147298183 CE For-Sale Anodyne ILK 0 40 Cc1c(NCCCCC(C)C)cc(N)cc1S(N)(=O)=O ZINC000147298183 CE For-Sale Anodyne PHLPP1 0 40 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2cccc(OC)c2OC)c1 ZINC000147298215 FF On-Demand Bother NQO2 51 37 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2cccc(OC)c2OC)c1 ZINC000147298215 FF On-Demand Bother MTNR1A 83 48 COc1ccc([N+](=O)[O-])c(C(=O)NCCc2cccc(OC)c2OC)c1 ZINC000147298215 FF On-Demand Bother MTNR1B 64 40 C=CCNC(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147298223 HC On-Demand Mild SFRP1 74 35 CCCCCCCCNS(=O)(=O)C[C@H](C)CCl ZINC000147298228 CG For-Sale Reactive RELA 19 44 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccccc1N1CCCCC1 ZINC000147298240 EE On-Demand Anodyne KCNQ2 92 47 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccccc1N1CCCCC1 ZINC000147298240 EE On-Demand Anodyne CSF1R 20 47 COC(=O)c1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1C ZINC000147298252 GG On-Demand Anodyne NOS2 48 33 COC(=O)c1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1C ZINC000147298252 GG On-Demand Anodyne ROCK2 15 40 CC[C@H](NCC(F)F)c1ccc(F)cc1 ZINC000147298266 BG For-Sale Anodyne LEF 20 42 O=C(N[C@@H](C(=O)O)C1CC1)c1cccc(F)c1Cl ZINC000147298306 CE On-Demand Anodyne NTSR2 42 43 O=C(N[C@@H](C(=O)O)C1CC1)c1cccc(F)c1Cl ZINC000147298306 CE On-Demand Anodyne PYGL 30 49 COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147298373 GI On-Demand Anodyne HTR1A 76 40 COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147298373 GI On-Demand Anodyne DRD2 68 46 COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147298373 GI On-Demand Anodyne ADRA1D 78 41 COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147298373 GI On-Demand Anodyne ADRA1A 69 41 COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147298373 GI On-Demand Anodyne ADRA1B 61 41 COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147298373 GI On-Demand Anodyne DRD3 60 40 COc1cc(CNC2CCN(c3ccccc3OC)CC2)ccc1OC(F)F ZINC000147298373 GI On-Demand Anodyne HTR7 46 39 C/C=C\Cn1cc(C)c(=O)[nH]c1=O ZINC000147298374 AC For-Sale Anodyne TK1 41 56 C/C=C\Cn1cc(C)c(=O)[nH]c1=O ZINC000147298374 AC For-Sale Anodyne TMK 53 51 C/C=C\Cn1cc(C)c(=O)[nH]c1=O ZINC000147298374 AC For-Sale Anodyne TYMP 52 47 C/C=C\Cn1cc(C)c(=O)[nH]c1=O ZINC000147298374 AC For-Sale Anodyne TK2 37 56 C/C(N)=N/N=C/c1ccccc1 ZINC000147298401 AD For-Sale Mild AMD1 18 42 C/C(N)=N/N=C/c1ccccc1 ZINC000147298401 AD For-Sale Mild UREA_CANEN 37 43 CN(C)NC(=O)/C=C/c1ccc(N)cc1 ZINC000147298403 BC For-Sale Reactive HDAC8 28 40 CN(C)NC(=O)/C=C/c1ccc(N)cc1 ZINC000147298403 BC For-Sale Reactive MMP2 17 41 CN(C)NC(=O)/C=C/c1ccc(N)cc1 ZINC000147298403 BC For-Sale Reactive HDAC1 28 40 CN(C)NC(=O)/C=C/c1ccc(N)cc1 ZINC000147298403 BC For-Sale Reactive HDAC2 15 42 Cc1cc(Oc2ccc(Cl)c(F)c2)ccc1S(N)(=O)=O ZINC000147298404 DG For-Sale Anodyne PTGS2 15 43 OCCCCCCSc1nc2ccccc2s1 ZINC000147298422 CH On-Demand Anodyne HMOX1 16 57 OCCCCCCSc1nc2ccccc2s1 ZINC000147298422 CH On-Demand Anodyne HMOX2 43 57 C=CCNC(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147298436 HC On-Demand Mild SFRP1 74 35 COc1cccc(CCNC(=O)c2ccn(-c3cccc(F)c3)n2)c1OC ZINC000147298437 FG On-Demand Anodyne CARM1 31 40 CCCCCCCCNS(=O)(=O)c1ccc(CBr)cc1 ZINC000147298448 FI For-Sale Reactive ALOX15B 0 40 CCCCCCCCNS(=O)(=O)c1ccc(CBr)cc1 ZINC000147298448 FI For-Sale Reactive ALOX15 68 53 CCCCCCCCNS(=O)(=O)c1ccc(CBr)cc1 ZINC000147298448 FI For-Sale Reactive A6YCJ1_9METZ 15 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(OC(F)(F)F)c1 ZINC000147298472 EE On-Demand Anodyne TAAR1 27 45 CC[C@@H](NCC(F)F)c1ccc(F)cc1 ZINC000147298493 BG For-Sale Anodyne LEF 20 42 Cc1cc(C(=O)N2CCN(Cc3ccc(C#N)cc3)CC2)cc([N+](=O)[O-])c1 ZINC000147298520 FF On-Demand Mild KCNJ1 38 40 O=C(O)[C@@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C1CC1 ZINC000147298524 CD For-Sale Anodyne GPR88 0 52 C/C=C\Cn1ccc(=O)[nH]c1=O ZINC000147298584 AC For-Sale Anodyne DUT 54 42 C/C=C\Cn1ccc(=O)[nH]c1=O ZINC000147298584 AC For-Sale Anodyne Q8II92_PLAF7 63 53 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne CA2 32 51 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne PTGS2 43 43 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne CA1 31 42 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne CA13 15 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne CA4 27 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne CA12 22 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne CA9 24 43 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne CAH_METTE 42 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne CYNT 24 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne NCE103 23 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne CA15 22 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne CA 0 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne A6YCJ1_9METZ 19 45 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147298627 EH For-Sale Anodyne Q5TU56_ANOGA 0 41 CCCCCCCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147298669 EI For-Sale Reactive CA2 15 44 CCCCCCCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147298669 EI For-Sale Reactive TBXA2R 42 36 CCCCCCCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147298669 EI For-Sale Reactive ALOX15B 0 43 CCCCCCCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147298669 EI For-Sale Reactive S1PR2 31 40 CCCCCCCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147298669 EI For-Sale Reactive ALOX15 68 54 CCCCCCCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147298669 EI For-Sale Reactive TPSAB1 15 40 CCCCCCCCNS(=O)(=O)c1ccc(CCCl)cc1 ZINC000147298669 EI For-Sale Reactive A6YCJ1_9METZ 23 44 COc1cc(CNC2(C(=O)O)CCC2)ccc1OC(F)F ZINC000147298673 DE On-Demand Anodyne PDEC 0 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(OC(F)(F)F)c1 ZINC000147298682 EE On-Demand Anodyne TAAR1 27 45 COC(=O)c1cccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)c1C ZINC000147298709 HI On-Demand Anodyne TRPV1 16 42 COC(=O)c1cccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)c1C ZINC000147298709 HI On-Demand Anodyne ROCK2 26 42 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cccc(F)c2[N+](=O)[O-])C1 ZINC000147298714 GC On-Demand Bother SFRP1 63 32 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cccc(F)c2[N+](=O)[O-])C1 ZINC000147298714 GC On-Demand Bother WNT3 41 30 O=C(O)[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C1CC1 ZINC000147298744 CD For-Sale Anodyne GPR88 0 52 O=C(c1ccc2ccccc2c1)N1CCC[C@H](CCBr)C1 ZINC000147298770 EI For-Sale Reactive AKR1C3 0 52 O=C(c1ccc2ccccc2c1)N1CCC[C@H](CCBr)C1 ZINC000147298770 EI For-Sale Reactive L3MBTL1 0 44 O=C(c1ccc2ccccc2c1)N1CCC[C@H](CCBr)C1 ZINC000147298770 EI For-Sale Reactive L3MBTL3 56 44 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne CA2 27 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne PTGS2 36 41 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne CA1 24 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne CA4 24 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne CA12 18 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne CA9 20 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne CAH_METTE 41 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne CYNT 24 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne NCE103 15 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne CA15 19 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne CA 0 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne A6YCJ1_9METZ 15 40 NS(=O)(=O)c1ccc(Oc2ccc(Cl)c(F)c2)c(Br)c1 ZINC000147298836 GH For-Sale Anodyne Q5TU56_ANOGA 0 40 CCCCCCCCNC(=O)c1ccc(C#CCO)cc1 ZINC000147298843 CG For-Sale Mild FOLH1 25 46 CCCCCCCCNC(=O)c1ccc(C#CCO)cc1 ZINC000147298843 CG For-Sale Mild ASAH1 88 37 O=C(O)C1(NCCCOc2ccc(F)cc2)CCC1 ZINC000147298865 CE For-Sale Anodyne DRD4 19 47 O=C(O)C1(NCCCOc2ccc(F)cc2)CCC1 ZINC000147298865 CE For-Sale Anodyne PLA2G4B 40 31 O=C1COc2ccc(I)cc2N1Cc1ccc(F)cc1 ZINC000147298878 GG For-Sale Anodyne PIK3CG 20 44 O=C1COc2ccc(I)cc2N1Cc1ccc(F)cc1 ZINC000147298878 GG For-Sale Anodyne SLC5A2 66 45 O=C(O)[C@@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C1CC1 ZINC000147298926 CD For-Sale Anodyne GPR88 0 52 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2cccc(F)c2[N+](=O)[O-])C1 ZINC000147298943 GC On-Demand Bother SFRP1 63 32 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2cccc(F)c2[N+](=O)[O-])C1 ZINC000147298943 GC On-Demand Bother WNT3 41 30 O=C(c1ccc2ccccc2c1)N1CCC[C@@H](CCBr)C1 ZINC000147298953 EI For-Sale Reactive AKR1C3 0 52 O=C(c1ccc2ccccc2c1)N1CCC[C@@H](CCBr)C1 ZINC000147298953 EI For-Sale Reactive L3MBTL1 0 44 O=C(c1ccc2ccccc2c1)N1CCC[C@@H](CCBr)C1 ZINC000147298953 EI For-Sale Reactive L3MBTL3 56 44 COC(=O)c1cnc(NC(=O)Cc2cccc(OC(C)C)c2)s1 ZINC000147298991 EF On-Demand Anodyne ADRB1 18 40 COC(=O)c1cnc(NC(=O)Cc2cccc(OC(C)C)c2)s1 ZINC000147298991 EF On-Demand Anodyne ADRB3 17 40 COC(=O)c1cnc(NC(=O)Cc2cccc(OC(C)C)c2)s1 ZINC000147298991 EF On-Demand Anodyne CSNK1D 32 48 COC(=O)c1cnc(NC(=O)Cc2cccc(OC(C)C)c2)s1 ZINC000147298991 EF On-Demand Anodyne CDK5 34 49 CC(C)[C@H](N)CC(=O)NN(C)C ZINC000147299005 AB For-Sale Reactive KDM7A 0 42 CCCCCCCCNC(=O)c1ccncc1C#CCO ZINC000147299065 CF For-Sale Mild ASAH1 53 32 C/C=C/Cn1cc(F)c(=O)[nH]c1=O ZINC000147299074 AC For-Sale Anodyne TMK 40 36 C/C=C/Cn1cc(F)c(=O)[nH]c1=O ZINC000147299074 AC For-Sale Anodyne GRIA3 15 47 NS(=O)(=O)c1ccc(OCCCN2CCCC2)c(F)c1F ZINC000147299122 DD For-Sale Anodyne HRH3 60 54 O=C(O)[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C1CC1 ZINC000147299145 CD For-Sale Anodyne GPR88 0 52 O[C@@H]1CNC[C@@H](Cc2ccccc2)C1 ZINC000147299146 AD For-Sale Anodyne SLC18A2 23 41 COc1cccc(OC)c1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147299202 FG For-Sale Reactive ACKR3 61 31 CC(C)[C@@H](N)CC(=O)NN(C)C ZINC000147299232 AB For-Sale Reactive KDM7A 0 42 CCCCCCCCNC(=O)c1csc(C#CCO)c1 ZINC000147299249 CG For-Sale Mild ASAH1 71 32 CNc1cn2ccnc2c(Oc2ccc(Cl)cc2Br)n1 ZINC000147299261 FH For-Sale Anodyne HIVRT 0 52 C/C=C\Cn1cc(Cl)c(=O)[nH]c1=O ZINC000147299272 BC For-Sale Anodyne TMK 40 36 C/C=C\Cn1cc(Cl)c(=O)[nH]c1=O ZINC000147299272 BC For-Sale Anodyne GRIA3 15 47 C/C=C\Cn1cc(Cl)c(=O)[nH]c1=O ZINC000147299272 BC For-Sale Anodyne DNK 0 40 C/C=C\Cn1cc(Cl)c(=O)[nH]c1=O ZINC000147299272 BC For-Sale Anodyne GRIK5 25 47 O[C@H]1CNC[C@@H](Cc2ccccc2)C1 ZINC000147299301 AD For-Sale Anodyne SLC18A2 23 41 COC(=O)c1cnc(NC(=O)[C@@H](C)Cc2cccc(F)c2)s1 ZINC000147299343 DF On-Demand Anodyne SCD1 28 42 Cc1ccc(C(=O)N[C@H](C(=O)O)C2CC2)cc1Br ZINC000147299356 DE On-Demand Anodyne PYGL 29 40 CCCS(=O)(=O)Nc1ccccc1C(=O)N(C)Cc1cccc(C(F)(F)F)c1 ZINC000147299360 HI On-Demand Anodyne TACR1 24 48 O=C1CC[C@@H](C(=O)Nc2ccon2)CN1 ZINC000147299365 BC For-Sale Anodyne TYK2 44 35 CCCCCCCCNC(=O)c1ccc(C#CCCO)s1 ZINC000147299418 DH For-Sale Mild ASAH1 66 35 COc1cccc(OC)c1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147299440 FG For-Sale Reactive ACKR3 61 31 Cc1ccc(C(=O)N[C@@H](C(=O)O)C2CC2)cc1Br ZINC000147299488 DE On-Demand Anodyne PYGL 29 40 O[C@@H]1CNC[C@H](Cc2ccccc2)C1 ZINC000147299490 AD For-Sale Anodyne SLC18A2 23 41 COC(=O)c1cnc(NC(=O)[C@H](C)Cc2cccc(F)c2)s1 ZINC000147299498 DF On-Demand Anodyne SCD1 28 42 C/C=C\Cn1cc(Br)c(=O)[nH]c1=O ZINC000147299549 BC For-Sale Anodyne TMK 43 43 C/C=C\Cn1cc(Br)c(=O)[nH]c1=O ZINC000147299549 BC For-Sale Anodyne GRIA3 15 47 C/C=C\Cn1cc(Br)c(=O)[nH]c1=O ZINC000147299549 BC For-Sale Anodyne GRIK5 25 47 COc1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147299564 CD For-Sale Anodyne HTR1A 20 50 COc1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147299564 CD For-Sale Anodyne ADRA1D 29 50 COc1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147299564 CD For-Sale Anodyne ADRA1A 23 50 COc1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147299564 CD For-Sale Anodyne ADRA1B 27 50 COc1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147299564 CD For-Sale Anodyne KCNA3 41 36 Cc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1[N+](=O)[O-] ZINC000147299565 DD On-Demand Bother BDKRB1 0 40 Cc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1[N+](=O)[O-] ZINC000147299565 DD On-Demand Bother COLA 51 34 CCCCCCCCCCC/C=C(/C=O)CCCCCCCCCC ZINC000147299571 FK For-Sale Reactive DPEP1 19 40 CCCCCCCCCCC/C=C(/C=O)CCCCCCCCCC ZINC000147299571 FK For-Sale Reactive FAAH 21 50 CCCCCCCCCCC/C=C(/C=O)CCCCCCCCCC ZINC000147299571 FK For-Sale Reactive CES2 51 45 CCCCCCCCCCC/C=C(/C=O)CCCCCCCCCC ZINC000147299571 FK For-Sale Reactive CES1 28 45 CCCCCCCCCCC/C=C(/C=O)CCCCCCCCCC ZINC000147299571 FK For-Sale Reactive EST1_PIG 68 45 CCCCCCCCCCC/C=C(/C=O)CCCCCCCCCC ZINC000147299571 FK For-Sale Reactive CES2C 58 39 CCCCCCCCCCC/C=C(/C=O)CCCCCCCCCC ZINC000147299571 FK For-Sale Reactive FABP3 40 52 CCCCCCCCCCC/C=C(/C=O)CCCCCCCCCC ZINC000147299571 FK For-Sale Reactive FABP5 18 52 CCCCCCCCCCC/C=C(/C=O)CCCCCCCCCC ZINC000147299571 FK For-Sale Reactive FABP1 17 52 CCCCCCCCCCC/C=C(/C=O)CCCCCCCCCC ZINC000147299571 FK For-Sale Reactive CQSS 66 41 O=C1CC[C@H](C(=O)Nc2ccon2)CN1 ZINC000147299581 BC For-Sale Anodyne TYK2 44 35 CCCCCCCCNC(=O)c1sccc1C#CCCO ZINC000147299585 DH For-Sale Mild ASAH1 55 33 CC(=O)Nc1cccc2c1CCCN2C(=O)c1cnn(-c2ccccc2Cl)c1 ZINC000147299631 GI On-Demand Anodyne AVPR2 84 43 CC(=O)Nc1cccc2c1CCCN2C(=O)c1cnn(-c2ccccc2Cl)c1 ZINC000147299631 GI On-Demand Anodyne AVPR1A 28 41 CC(=O)Nc1cccc2c1CCCN2C(=O)c1cnn(-c2ccccc2Cl)c1 ZINC000147299631 GI On-Demand Anodyne KCNQ2 47 34 CC(=O)Nc1cccc2c1CCCN2C(=O)c1cnn(-c2ccccc2Cl)c1 ZINC000147299631 GI On-Demand Anodyne EPHB3 41 33 CCOC(=O)NCC(=O)Nc1cccc(COc2cccc(F)c2)c1 ZINC000147299636 EG On-Demand Anodyne MAOB 28 40 CCOC(=O)NCC(=O)Nc1cccc(COc2cccc(F)c2)c1 ZINC000147299636 EG On-Demand Anodyne PDS 59 44 CCCNc1cc(Oc2ccc(Cl)cc2Br)nc(N)n1 ZINC000147299647 FI For-Sale Anodyne AGPAT2 76 44 O[C@H]1CNC[C@H](Cc2ccccc2)C1 ZINC000147299697 AD For-Sale Anodyne SLC18A2 23 41 COC(=O)c1cnc(NC(=O)COc2ccc([N+](=O)[O-])c(OC)c2)s1 ZINC000147299705 FD On-Demand Bother PDGFRB 19 41 C[C@H](NCC(F)F)c1ccccc1[N+](=O)[O-] ZINC000147299738 BF On-Demand Bother COLA 89 35 C[C@H](NCC(F)F)c1ccccc1[N+](=O)[O-] ZINC000147299738 BF On-Demand Bother PQSD 0 43 CCCCCCCCNC(=O)c1cc(C)c(C#CCO)s1 ZINC000147299781 DG For-Sale Mild ASAH1 68 32 O=C1COc2ccc(I)cc2N1Cc1cc(F)ccc1F ZINC000147299790 HG For-Sale Anodyne SLC5A2 52 41 Cc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1[N+](=O)[O-] ZINC000147299795 DD On-Demand Bother BDKRB1 0 40 Cc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1[N+](=O)[O-] ZINC000147299795 DD On-Demand Bother COLA 51 34 C[C@@H](NCC(F)F)c1ccccc1[N+](=O)[O-] ZINC000147299880 BF On-Demand Bother COLA 89 35 C[C@@H](NCC(F)F)c1ccccc1[N+](=O)[O-] ZINC000147299880 BF On-Demand Bother PQSD 0 43 C[C@H](CCN)CCC(=O)NN(C)C ZINC000147299970 AC For-Sale Reactive KDM7A 0 48 CCCCCCCCNC(=O)c1cccc(C#CCO)c1 ZINC000147299998 CG For-Sale Mild DRD4 40 31 CCCCCCCCNC(=O)c1cccc(C#CCO)c1 ZINC000147299998 CG For-Sale Mild DRD3 23 42 CCCCCCCCNC(=O)c1cccc(C#CCO)c1 ZINC000147299998 CG For-Sale Mild PLA2G4B 41 37 CCCCCCCCNC(=O)c1cccc(C#CCO)c1 ZINC000147299998 CG For-Sale Mild ASAH1 73 34 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne NPY1R 27 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne KLK3 63 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne PAPA1_CARPA 42 32 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne CTSK 51 43 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne NPFFR2 41 39 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne C3AR1 59 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne MMP3 19 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne PCSK5 54 36 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne FURIN 61 34 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne CTSS 20 52 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne CAPN2 52 38 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne NPR 43 35 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne POLG_DEN26 0 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne POLG_WNV 80 33 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne NPFFR1 57 39 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300073 DD On-Demand Anodyne NOD1 62 32 CC(=O)Nc1cccc2c1CCCN2C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147300089 FI On-Demand Anodyne AVPR2 17 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1C(=O)N1CCOCC1 ZINC000147300092 GC On-Demand Anodyne BDKRB1 16 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1C(=O)N1CCOCC1 ZINC000147300092 GC On-Demand Anodyne TNK2 20 41 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)c(O)c1 ZINC000147300099 EG For-Sale Reactive GRM3 16 48 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)c(O)c1 ZINC000147300099 EG For-Sale Reactive RORC 42 40 Cc1cccc(CNCC(F)F)c1C ZINC000147300117 AF On-Demand Anodyne PHES 0 42 O=C(Nc1cccc(-c2cnc3cc(-c4ccc(F)cc4)ccn23)c1)NC1CC1 ZINC000147300134 GK Annotated Anodyne F10 0 41 O=C(Nc1cccc(-c2cnc3cc(-c4ccc(F)cc4)ccn23)c1)NC1CC1 ZINC000147300134 GK Annotated Anodyne CCR3 57 40 O=C(Nc1cccc(-c2cnc3cc(-c4ccc(F)cc4)ccn23)c1)NC1CC1 ZINC000147300134 GK Annotated Anodyne MAPK13 67 33 O=C(Nc1cccc(-c2cnc3cc(-c4ccc(F)cc4)ccn23)c1)NC1CC1 ZINC000147300134 GK Annotated Anodyne RIPK1 44 32 C[C@@H](CCN)CCC(=O)NN(C)C ZINC000147300143 AC For-Sale Reactive KDM7A 0 48 CN(C)C1(Cn2c(N)nc3cccc(Cl)c32)CCCC1 ZINC000147300152 CG For-Sale Anodyne Q581W1_TRYB2 0 50 CCCCCCCCNC(=O)c1ccc(C#CCO)s1 ZINC000147300236 CG For-Sale Mild ASAH1 81 36 CC(=O)Nc1cccc2c1CCCN2C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147300287 FI On-Demand Anodyne AVPR2 17 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne NPY1R 27 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne KLK3 63 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne PAPA1_CARPA 42 32 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne CTSK 51 43 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne NPFFR2 41 39 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne C3AR1 59 37 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne MMP3 19 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne PCSK5 54 36 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne FURIN 61 34 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne CTSS 20 52 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne CAPN2 52 38 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne NPR 43 35 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne POLG_DEN26 0 41 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne POLG_WNV 80 33 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne NPFFR1 57 39 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](OC)c1ccccc1 ZINC000147300290 DD On-Demand Anodyne NOD1 62 32 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccccc1C(=O)N1CCOCC1 ZINC000147300295 GC On-Demand Anodyne BDKRB1 16 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccccc1C(=O)N1CCOCC1 ZINC000147300295 GC On-Demand Anodyne TNK2 20 41 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)c(O)c1 ZINC000147300302 EG For-Sale Reactive GRM3 16 48 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)c(O)c1 ZINC000147300302 EG For-Sale Reactive RORC 42 40 O=C(O)[C@H]1CCN(C(=O)c2cccc3c2OCCN3)C1 ZINC000147300375 CD For-Sale Anodyne SLC6A1 71 33 OC[C@@H]1C[C@@H](Cc2ccccc2)CN1Cc1ccccc1 ZINC000147300435 CG For-Sale Anodyne CACNA1C 18 49 OC[C@@H]1C[C@@H](Cc2ccccc2)CN1Cc1ccccc1 ZINC000147300435 CG For-Sale Anodyne CACNA1B 26 49 CCCCCCCCNC(=O)c1csc(C#CCCO)c1 ZINC000147300439 DH For-Sale Mild ASAH1 53 31 CC[C@H](NCCCCC(C)C)c1ccc(OC)c(OC)c1 ZINC000147300490 CJ For-Sale Anodyne LEF 33 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne NPY1R 27 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne KLK3 63 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne PAPA1_CARPA 42 32 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne CTSK 51 43 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne NPFFR2 41 39 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne C3AR1 59 37 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne MMP3 19 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne PCSK5 54 36 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne FURIN 61 34 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne CTSS 20 52 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne CAPN2 52 38 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne NPR 43 35 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne POLG_DEN26 0 41 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne POLG_WNV 80 33 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne NPFFR1 57 39 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](OC)c1ccccc1 ZINC000147300494 DD On-Demand Anodyne NOD1 62 32 CC(=O)Nc1cccc2c1CCCN2C(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147300513 FI On-Demand Anodyne AVPR2 17 40 Cc1ncc(-c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)o1 ZINC000147300522 EE On-Demand Anodyne MTOR 40 33 CCCCCCCCCCC/C=C(\C=O)CCCCCCCCCC ZINC000147300561 FK For-Sale Reactive DPEP1 19 40 CCCCCCCCCCC/C=C(\C=O)CCCCCCCCCC ZINC000147300561 FK For-Sale Reactive FAAH 21 50 CCCCCCCCCCC/C=C(\C=O)CCCCCCCCCC ZINC000147300561 FK For-Sale Reactive CES2 51 45 CCCCCCCCCCC/C=C(\C=O)CCCCCCCCCC ZINC000147300561 FK For-Sale Reactive CES1 28 45 CCCCCCCCCCC/C=C(\C=O)CCCCCCCCCC ZINC000147300561 FK For-Sale Reactive EST1_PIG 68 45 CCCCCCCCCCC/C=C(\C=O)CCCCCCCCCC ZINC000147300561 FK For-Sale Reactive CES2C 58 39 CCCCCCCCCCC/C=C(\C=O)CCCCCCCCCC ZINC000147300561 FK For-Sale Reactive FABP3 40 52 CCCCCCCCCCC/C=C(\C=O)CCCCCCCCCC ZINC000147300561 FK For-Sale Reactive FABP5 18 52 CCCCCCCCCCC/C=C(\C=O)CCCCCCCCCC ZINC000147300561 FK For-Sale Reactive FABP1 17 52 CCCCCCCCCCC/C=C(\C=O)CCCCCCCCCC ZINC000147300561 FK For-Sale Reactive CQSS 66 41 O=C(O)[C@@H]1CCN(C(=O)c2cccc3c2OCCN3)C1 ZINC000147300582 CD For-Sale Anodyne SLC6A1 71 33 COCc1nc(C(=O)N2CCC[C@@H]2c2ccc3c(c2)OCCO3)cs1 ZINC000147300625 FG On-Demand Anodyne TRPC6 42 44 COCc1nc(C(=O)N2CCC[C@@H]2c2ccc3c(c2)OCCO3)cs1 ZINC000147300625 FG On-Demand Anodyne TRPC3 52 44 CC(C)(C)C[C@H]1N[C@@H](C(=O)NC2CN(CCO)C2)[C@H](c2cccc(Cl)c2F)[C@@]12C(=O)Nc1cc(Cl)ccc12 ZINC000147300638 KH Annotated Anodyne MDM2 105 73 OC[C@H]1C[C@@H](Cc2ccccc2)CN1Cc1ccccc1 ZINC000147300641 CG For-Sale Anodyne CACNA1C 18 49 OC[C@H]1C[C@@H](Cc2ccccc2)CN1Cc1ccccc1 ZINC000147300641 CG For-Sale Anodyne SIGMAR1 25 54 OC[C@H]1C[C@@H](Cc2ccccc2)CN1Cc1ccccc1 ZINC000147300641 CG For-Sale Anodyne CACNA1B 26 49 CC[C@@H](NCCCCC(C)C)c1ccc(OC)c(OC)c1 ZINC000147300675 CJ For-Sale Anodyne LEF 33 41 Cc1cc(=O)n2nc(CNC3(C(=O)O)CCC3)sc2n1 ZINC000147300682 CC For-Sale Anodyne XDH 19 49 CC(=O)Nc1cccc2c1CCCN2C(=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147300686 FI On-Demand Anodyne AVPR2 17 40 CCCCCCCCNC(=O)c1sccc1C#CCO ZINC000147300691 CG For-Sale Mild ASAH1 76 34 Cc1ncc(-c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)o1 ZINC000147300739 EE On-Demand Anodyne MTOR 40 33 CO[C@H](CNC(=O)Cc1c(C)nn(C(F)F)c1C)c1ccccc1 ZINC000147300758 EF On-Demand Anodyne P2RX7 44 44 O=C(c1cccc2c1OCCN2)N1CCn2ccnc2C1 ZINC000147300787 CD For-Sale Anodyne P2RX7 31 54 C[C@@](O)(COc1ccc(Cl)c(F)c1)c1ccccc1 ZINC000147300833 CH For-Sale Anodyne PDS 51 33 COCc1nc(C(=O)N2CCC[C@H]2c2ccc3c(c2)OCCO3)cs1 ZINC000147300852 FG On-Demand Anodyne TRPC6 42 44 COCc1nc(C(=O)N2CCC[C@H]2c2ccc3c(c2)OCCO3)cs1 ZINC000147300852 FG On-Demand Anodyne TRPC3 52 44 OC[C@@H]1C[C@H](Cc2ccccc2)CN1Cc1ccccc1 ZINC000147300875 CG For-Sale Anodyne CACNA1C 18 49 OC[C@@H]1C[C@H](Cc2ccccc2)CN1Cc1ccccc1 ZINC000147300875 CG For-Sale Anodyne SIGMAR1 25 54 OC[C@@H]1C[C@H](Cc2ccccc2)CN1Cc1ccccc1 ZINC000147300875 CG For-Sale Anodyne CACNA1B 26 49 CCC[C@@H](NC(=O)CCC(=O)O)C(=O)O ZINC000147300883 BC On-Demand Anodyne FOLH1 54 46 CCC[C@@H](NC(=O)CCC(=O)O)C(=O)O ZINC000147300883 BC On-Demand Anodyne NAALAD2 68 52 CCC[C@@H](NC(=O)CCC(=O)O)C(=O)O ZINC000147300883 BC On-Demand Anodyne NOD1 114 56 CCC[C@@H](NC(=O)CCC(=O)O)C(=O)O ZINC000147300883 BC On-Demand Anodyne KDM4E 23 40 CCC[C@@H](NC(=O)CCC(=O)O)C(=O)O ZINC000147300883 BC On-Demand Anodyne KDM2A 41 41 COc1cccc(CNC2(C(=O)O)CCC2)c1 ZINC000147300898 BD On-Demand Anodyne DRD4 40 31 COc1cccc(CNC2(C(=O)O)CCC2)c1 ZINC000147300898 BD On-Demand Anodyne ROCK1 37 43 COc1cccc(CNC2(C(=O)O)CCC2)c1 ZINC000147300898 BD On-Demand Anodyne MTNR1A 49 44 COc1cccc(CNC2(C(=O)O)CCC2)c1 ZINC000147300898 BD On-Demand Anodyne MTNR1B 39 42 COc1cccc(CNC2(C(=O)O)CCC2)c1 ZINC000147300898 BD On-Demand Anodyne ROCK2 42 39 COc1cccc(CNC2(C(=O)O)CCC2)c1 ZINC000147300898 BD On-Demand Anodyne AKR1C3 18 40 CCCCCCCCNC(=O)c1ccc(C#CCO)cn1 ZINC000147300918 CF For-Sale Mild GRM5 15 53 CCCCCCCCNC(=O)c1ccc(C#CCO)cn1 ZINC000147300918 CF For-Sale Mild ASAH1 65 33 CC(C)CCO[C@@H](C)C(=O)N(C)C1CCCC1 ZINC000147300926 BF On-Demand Anodyne CHRNA4 0 41 COc1cc(Cl)ccc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147300932 DD On-Demand Anodyne COLA 73 38 COc1cc(Cl)ccc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147300932 DD On-Demand Anodyne CPT1A 47 33 Cc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147301020 DE On-Demand Anodyne DHODH 24 47 NC[C@@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301029 ED On-Demand Anodyne CHRM1 15 40 NC[C@@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301029 ED On-Demand Anodyne KLK3 54 31 NC[C@@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301029 ED On-Demand Anodyne CTSB 46 37 NC[C@@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301029 ED On-Demand Anodyne PAPA1_CARPA 50 33 NC[C@@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301029 ED On-Demand Anodyne CTSK 24 40 NC[C@@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301029 ED On-Demand Anodyne CAPNS1 56 36 NC[C@@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301029 ED On-Demand Anodyne CTSS 16 40 NC[C@@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301029 ED On-Demand Anodyne CAPN1 74 39 NC[C@@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301029 ED On-Demand Anodyne CAPN2 96 38 NC[C@@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301029 ED On-Demand Anodyne NPR 67 40 C[C@](O)(COc1ccc(Cl)c(F)c1)c1ccccc1 ZINC000147301037 CH For-Sale Anodyne PDS 51 33 OC[C@H]1C[C@H](Cc2ccccc2)CN1Cc1ccccc1 ZINC000147301076 CG For-Sale Anodyne CACNA1C 18 49 OC[C@H]1C[C@H](Cc2ccccc2)CN1Cc1ccccc1 ZINC000147301076 CG For-Sale Anodyne SIGMAR1 25 54 OC[C@H]1C[C@H](Cc2ccccc2)CN1Cc1ccccc1 ZINC000147301076 CG For-Sale Anodyne CACNA1B 26 49 O=C(O)/C=C1\c2ccccc2CCc2cc(Cl)ccc21 ZINC000147301083 CH For-Sale Anodyne SRD5A2 15 51 Cc1cc(C(=O)N2CCC(C(=O)N3CCCCC3)CC2)cc([N+](=O)[O-])c1 ZINC000147301094 FF On-Demand Bother L3MBTL1 0 41 Cc1cc(C(=O)N2CCC(C(=O)N3CCCCC3)CC2)cc([N+](=O)[O-])c1 ZINC000147301094 FF On-Demand Bother L3MBTL3 59 37 COCCN1CCN(c2ccc(S(=O)(=O)N3CCCCC3)cc2[N+](=O)[O-])CC1 ZINC000147301126 HD On-Demand Bother CASP3 42 38 COCCN1CCN(c2ccc(S(=O)(=O)N3CCCCC3)cc2[N+](=O)[O-])CC1 ZINC000147301126 HD On-Demand Bother CASP7 53 38 COc1cc(Cl)ccc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147301132 DD On-Demand Anodyne COLA 73 38 COc1cc(Cl)ccc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147301132 DD On-Demand Anodyne CPT1A 47 33 CC(C)CCO[C@H](C)C(=O)N(C)C1CCCC1 ZINC000147301140 BF On-Demand Anodyne CHRNA4 0 41 C[C@@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301141 CD For-Sale Anodyne ACE 52 36 C[C@@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301141 CD For-Sale Anodyne MME 92 38 C[C@@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301141 CD For-Sale Anodyne ANPEP 47 35 C[C@@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301141 CD For-Sale Anodyne TIMP3 40 32 C[C@@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301141 CD For-Sale Anodyne F11 48 37 C[C@@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301141 CD For-Sale Anodyne CAPN1 47 37 C[C@@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301141 CD For-Sale Anodyne ACE2 54 35 CCCCCCCCNC(=O)c1ccccc1C#CCO ZINC000147301146 CG For-Sale Mild ASAH1 86 38 CC(C)(NC(=O)c1cccc(F)c1Cl)C(C)(C)C(=O)O ZINC000147301147 DG For-Sale Anodyne ECR 41 40 CC(C)(NC(=O)c1cccc(F)c1Cl)C(C)(C)C(=O)O ZINC000147301147 DG For-Sale Anodyne E3UJZ5_SPOLI 32 40 CC(C)NCCCC(=O)NN(C)C ZINC000147301148 AC For-Sale Reactive KDM7A 0 48 NC[C@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301228 ED On-Demand Anodyne CHRM1 15 40 NC[C@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301228 ED On-Demand Anodyne KLK3 54 31 NC[C@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301228 ED On-Demand Anodyne CTSB 46 37 NC[C@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301228 ED On-Demand Anodyne PAPA1_CARPA 50 33 NC[C@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301228 ED On-Demand Anodyne CTSK 24 40 NC[C@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301228 ED On-Demand Anodyne CAPNS1 56 36 NC[C@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301228 ED On-Demand Anodyne CTSS 16 40 NC[C@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301228 ED On-Demand Anodyne CAPN1 74 39 NC[C@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301228 ED On-Demand Anodyne CAPN2 96 38 NC[C@H](C(=O)NCCC(=O)OCc1ccccc1)c1ccccc1 ZINC000147301228 ED On-Demand Anodyne NPR 67 40 Cc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147301244 DE On-Demand Anodyne DHODH 24 47 Cc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147301244 DE On-Demand Anodyne NPY2R 35 42 Cc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147301244 DE On-Demand Anodyne ENV 44 37 CC[C@@H]1OC[C@@H](O)[C@@H]1NC(=O)OC(C)(C)C ZINC000147301302 BD For-Sale Anodyne CTSK 16 40 O=C(O)C[C@@H]1c2ccccc2CCc2cc(Cl)ccc21 ZINC000147301313 CI For-Sale Anodyne SIGMAR1 16 40 O=C(O)C[C@@H]1c2ccccc2CCc2cc(Cl)ccc21 ZINC000147301313 CI For-Sale Anodyne PYGL 18 41 O=C(O)C[C@@H]1c2ccccc2CCc2cc(Cl)ccc21 ZINC000147301313 CI For-Sale Anodyne PTGDR2 25 40 C[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301353 CD For-Sale Anodyne ACE 52 36 C[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301353 CD For-Sale Anodyne MME 92 38 C[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301353 CD For-Sale Anodyne ANPEP 47 35 C[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301353 CD For-Sale Anodyne TIMP3 40 32 C[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301353 CD For-Sale Anodyne F11 48 37 C[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301353 CD For-Sale Anodyne CAPN1 47 37 C[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCC(=O)NC1 ZINC000147301353 CD For-Sale Anodyne ACE2 54 35 CN(C)NC(=O)CNCC1CC1 ZINC000147301360 AB For-Sale Reactive KDM7A 0 41 CCCCCCCCNC(=O)c1cncc(C#CCO)c1 ZINC000147301406 CF For-Sale Mild KCNQ1 0 40 CCCCCCCCNC(=O)c1cncc(C#CCO)c1 ZINC000147301406 CF For-Sale Mild ASAH1 63 32 COc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1NC(C)=O ZINC000147301445 ED On-Demand Anodyne QRFPR 41 35 O=C(O)C[C@H]1c2ccccc2CCc2cc(Cl)ccc21 ZINC000147301505 CI For-Sale Anodyne SIGMAR1 16 40 O=C(O)C[C@H]1c2ccccc2CCc2cc(Cl)ccc21 ZINC000147301505 CI For-Sale Anodyne PYGL 18 41 O=C(O)C[C@H]1c2ccccc2CCc2cc(Cl)ccc21 ZINC000147301505 CI For-Sale Anodyne PTGDR2 25 40 NS(=O)(=O)c1ccc(OCCn2ccnc2)c(F)c1F ZINC000147301526 DC For-Sale Anodyne CYP19A1 15 44 NS(=O)(=O)c1ccc(OCCn2ccnc2)c(F)c1F ZINC000147301526 DC For-Sale Anodyne CYP11B1 26 46 NS(=O)(=O)c1ccc(OCCn2ccnc2)c(F)c1F ZINC000147301526 DC For-Sale Anodyne TBXAS1 39 47 CC[C@@H]1OC[C@H](O)[C@@H]1NC(=O)OC(C)(C)C ZINC000147301541 BD For-Sale Anodyne CTSK 16 40 Nc1ccc(Oc2ccc(Cl)c(F)c2)c(C(=O)O)c1 ZINC000147301557 CH For-Sale Anodyne PPXII 0 40 COc1ccc(CCn2cc(I)c(=O)[nH]c2=O)cc1 ZINC000147301614 FD For-Sale Anodyne GRIK5 17 42 C[C@@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301627 CD For-Sale Anodyne ACE 52 36 C[C@@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301627 CD For-Sale Anodyne MME 92 38 C[C@@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301627 CD For-Sale Anodyne ANPEP 47 35 C[C@@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301627 CD For-Sale Anodyne TIMP3 40 32 C[C@@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301627 CD For-Sale Anodyne F11 48 37 C[C@@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301627 CD For-Sale Anodyne CAPN1 47 37 C[C@@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301627 CD For-Sale Anodyne ACE2 54 35 COc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1NC(C)=O ZINC000147301635 ED On-Demand Anodyne QRFPR 41 35 CC[C@@H]1CN(C(=O)c2ccoc2)CC[C@@H]1N ZINC000147301645 BD On-Demand Anodyne L3MBTL3 51 36 COC(=O)[C@H]1[C@H](C(=O)OC)[C@@H](C(=O)OC)[C@@H]1C(=O)OC ZINC000147301649 CB In-Stock Anodyne Q8AWE3_CHICK 18 46 CCCCCCCCNC(=O)c1ccncc1C#CCN ZINC000147301662 CE For-Sale Mild ASAH1 57 32 COCc1nc(C(=O)Nc2nc(-c3ccc(SC)cc3)cs2)cs1 ZINC000147301686 GI On-Demand Anodyne MPL 50 40 COCc1nc(C(=O)Nc2nc(-c3ccc(SC)cc3)cs2)cs1 ZINC000147301686 GI On-Demand Anodyne ROCK1 20 40 O=C(Nc1cc(Cl)ccc1C#CCCO)c1ccccc1 ZINC000147301752 CG For-Sale Mild HDAC1 0 41 O=C(Nc1cc(Cl)ccc1C#CCCO)c1ccccc1 ZINC000147301752 CG For-Sale Mild KCNK3 49 43 CCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1C ZINC000147301767 DD For-Sale Anodyne PTGDR2 23 42 CCOc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1C ZINC000147301767 DD For-Sale Anodyne LEF 41 39 COc1ccc2c(c1)OC[C@H](C(=O)N1CCCc3c(NC(C)=O)cccc31)C2 ZINC000147301807 GG On-Demand Anodyne AVPR2 15 40 COc1ccc2c(c1)OC[C@H](C(=O)N1CCCc3c(NC(C)=O)cccc31)C2 ZINC000147301807 GG On-Demand Anodyne MTNR1A 29 40 COc1ccc2c(c1)OC[C@H](C(=O)N1CCCc3c(NC(C)=O)cccc31)C2 ZINC000147301807 GG On-Demand Anodyne ROCK2 25 40 C[C@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301814 CD For-Sale Anodyne ACE 52 36 C[C@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301814 CD For-Sale Anodyne MME 92 38 C[C@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301814 CD For-Sale Anodyne ANPEP 47 35 C[C@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301814 CD For-Sale Anodyne TIMP3 40 32 C[C@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301814 CD For-Sale Anodyne F11 48 37 C[C@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301814 CD For-Sale Anodyne CAPN1 47 37 C[C@H](Cc1ccccc1)NC(=O)[C@H]1CCC(=O)NC1 ZINC000147301814 CD For-Sale Anodyne ACE2 54 35 O=C(O)C1(NCc2cccc([N+](=O)[O-])c2)CCC1 ZINC000147301837 CD On-Demand Bother CACNA1C 56 42 O=C(O)C1(NCc2cccc([N+](=O)[O-])c2)CCC1 ZINC000147301837 CD On-Demand Bother CACNA1D 91 42 O=C(O)C1(NCc2cccc([N+](=O)[O-])c2)CCC1 ZINC000147301837 CD On-Demand Bother LUXR 17 45 O=C(O)C1(NCc2cccc([N+](=O)[O-])c2)CCC1 ZINC000147301837 CD On-Demand Bother TRPM8 25 43 COC(=O)c1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1Cl ZINC000147301844 FD On-Demand Anodyne ENV 42 38 CCCCCCCCNC(=O)c1ccc(C#CCN)cn1 ZINC000147301886 CE For-Sale Mild ASAH1 58 33 CC[C@H]1CN(C(=O)c2ccoc2)CC[C@@H]1N ZINC000147301890 BD On-Demand Anodyne L3MBTL3 51 36 CCn1nc(C)c2c1CCN([C@@H](C(=O)NC)c1ccccc1)[C@H]2CCc1ccc(Cl)cc1 ZINC000147301931 JJ Annotated Anodyne HCRTR1 47 88 Cc1[nH]c2cc(OC(F)(F)F)ccc2c1C(=O)c1ccc(Cl)cc1 ZINC000147301975 FK For-Sale Anodyne PPARG 23 47 COC[C@@H]1C[C@H](O)CC(=O)O1 ZINC000147301984 AB For-Sale Anodyne HMGCR 84 44 CCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1C ZINC000147301995 DD For-Sale Anodyne PTGDR2 23 42 CCOc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1C ZINC000147301995 DD For-Sale Anodyne LEF 41 39 NS(=O)(=O)c1ccc(OCCCn2ccnc2)c(F)c1F ZINC000147302004 DD For-Sale Anodyne CYP11B1 22 40 NS(=O)(=O)c1ccc(OCCCn2ccnc2)c(F)c1F ZINC000147302004 DD For-Sale Anodyne TBXAS1 41 45 NS(=O)(=O)c1ccc(OCCCn2ccnc2)c(F)c1F ZINC000147302004 DD For-Sale Anodyne CYP17A1 0 42 NS(=O)(=O)c1ccc(OCCCn2ccnc2)c(F)c1F ZINC000147302004 DD For-Sale Anodyne HMOX2 41 42 Nc1cc(C(=O)O)cnc1Oc1ccc(Cl)c(F)c1 ZINC000147302011 CF For-Sale Anodyne H9BT73_9POAL 0 45 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCCc3c(NC(C)=O)cccc31)C2 ZINC000147302034 GG On-Demand Anodyne AVPR2 15 40 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCCc3c(NC(C)=O)cccc31)C2 ZINC000147302034 GG On-Demand Anodyne MTNR1A 29 40 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCCc3c(NC(C)=O)cccc31)C2 ZINC000147302034 GG On-Demand Anodyne ROCK2 25 40 COC(=O)c1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1Cl ZINC000147302046 FD On-Demand Anodyne ENV 42 38 CCCCCCCCNC(=O)c1csc(C#CCN)c1 ZINC000147302059 CG For-Sale Mild ASAH1 74 32 CC[C@@H]1CN(C(=O)c2ccoc2)CC[C@H]1N ZINC000147302091 BD On-Demand Anodyne L3MBTL3 51 36 COc1ccc([N+](=O)[O-])c(C(=O)NCCCCOCCc2ccccc2)c1 ZINC000147302133 FG On-Demand Bother AKR1C2 25 42 COc1ccc(CC[C@H](C)NCCCCC(C)C)cc1 ZINC000147302135 CI For-Sale Anodyne SLC2A1 0 42 COc1ccc(CC[C@H](C)NCCCCC(C)C)cc1 ZINC000147302135 CI For-Sale Anodyne HT1 0 42 COc1ccc(CC[C@H](C)NCCCCC(C)C)cc1 ZINC000147302135 CI For-Sale Anodyne LMGT2 0 42 CCOc1cc([C@@H](CS(C)(=O)=O)N2C(=O)c3cccc(NC(=O)CC)c3C2=O)ccc1OC ZINC000147302168 JF For-Sale Anodyne TNF 25 52 CCOc1cc([C@@H](CS(C)(=O)=O)N2C(=O)c3cccc(NC(=O)CC)c3C2=O)ccc1OC ZINC000147302168 JF For-Sale Anodyne UTS2R 32 42 COC[C@H]1C[C@H](O)CC(=O)O1 ZINC000147302169 AB For-Sale Anodyne HMGCR 84 44 CC(C)Oc1cccc(CC(=O)N(C)C2CCCC2)c1 ZINC000147302173 CG On-Demand Anodyne OPRK1 25 40 O=C(/C=C/CBr)OCc1ccccc1 ZINC000147302295 CF For-Sale Reactive CAPNS1 52 32 O=C(/C=C/CBr)OCc1ccccc1 ZINC000147302295 CF For-Sale Reactive AKR1B10 28 43 CC[C@H]1CN(C(=O)c2ccoc2)CC[C@H]1N ZINC000147302296 BD On-Demand Anodyne L3MBTL3 51 36 CCCCCCCCNC(=O)c1cncc(C#CCN)c1 ZINC000147302309 CE For-Sale Mild ASAH1 53 31 COc1ccc(CC[C@@H](C)NCCCCC(C)C)cc1 ZINC000147302339 CI For-Sale Anodyne SLC2A1 0 42 COc1ccc(CC[C@@H](C)NCCCCC(C)C)cc1 ZINC000147302339 CI For-Sale Anodyne HT1 0 42 COc1ccc(CC[C@@H](C)NCCCCC(C)C)cc1 ZINC000147302339 CI For-Sale Anodyne LMGT2 0 42 COC[C@@H]1C[C@@H](O)CC(=O)O1 ZINC000147302353 AB For-Sale Anodyne HMGCR 84 44 CCOc1cc([C@H](CS(C)(=O)=O)N2C(=O)c3cccc(NC(=O)CC)c3C2=O)ccc1OC ZINC000147302385 JF For-Sale Anodyne TNF 25 52 CCOc1cc([C@H](CS(C)(=O)=O)N2C(=O)c3cccc(NC(=O)CC)c3C2=O)ccc1OC ZINC000147302385 JF For-Sale Anodyne UTS2R 32 42 Nc1ccc(Oc2ccc(Cl)c(F)c2)cc1C(=O)O ZINC000147302437 CH For-Sale Anodyne PYGL 26 40 Nc1ccc(Oc2ccc(Cl)c(F)c2)cc1C(=O)O ZINC000147302437 CH For-Sale Anodyne PYGM 24 40 Cn1ccnc1CN1CCC(NC(=O)OC(C)(C)C)CC1 ZINC000147302439 CD On-Demand Anodyne SSTR5 45 39 O=C1CC[C@@H](C(=O)N[C@H](CO)c2ccccc2)CN1 ZINC000147302468 CC On-Demand Anodyne F11 40 37 CCCCCCCCNC(=O)c1sccc1C#CCN ZINC000147302531 CG For-Sale Mild ASAH1 71 33 COC[C@H]1C[C@@H](O)CC(=O)O1 ZINC000147302561 AB For-Sale Anodyne HMGCR 84 44 COc1ccc(-c2sccc2Br)c(C(=O)O)c1 ZINC000147302589 DH For-Sale Anodyne AKR1C3 23 42 COc1ccc(-c2sccc2Br)c(C(=O)O)c1 ZINC000147302589 DH For-Sale Anodyne AKR1C2 57 42 CN(C)NC(=O)CC[C@H](N)c1ccccc1 ZINC000147302692 BD For-Sale Reactive CHRNA4 0 42 CN(C)NC(=O)CC[C@H](N)c1ccccc1 ZINC000147302692 BD For-Sale Reactive KDM7A 0 44 O=C1CC[C@@H](C(=O)N[C@@H](CO)c2ccccc2)CN1 ZINC000147302709 CC On-Demand Anodyne F11 40 37 CN(C)C(=O)NCCNC(=O)c1cccc(C#CCO)c1 ZINC000147302742 CC For-Sale Mild DRD4 40 31 CCCCCCCCNC(=O)c1cc(C)c(C#CCN)s1 ZINC000147302745 DG For-Sale Mild ASAH1 60 32 O=C1CC[C@H](C(=O)N[C@H](CO)c2ccccc2)CN1 ZINC000147302899 CC On-Demand Anodyne F11 40 37 COc1ccc(CNc2nnc(SCCC(=O)NC(N)=O)s2)cc1 ZINC000147302914 FD On-Demand Anodyne CA9 15 41 COc1ccc(CNc2nnc(SCCC(=O)NC(N)=O)s2)cc1 ZINC000147302914 FD On-Demand Anodyne PROKR1 44 31 CN(C)NC(=O)CC[C@@H](N)c1ccccc1 ZINC000147302933 BD For-Sale Reactive CHRNA4 0 42 CN(C)NC(=O)CC[C@@H](N)c1ccccc1 ZINC000147302933 BD For-Sale Reactive KDM7A 0 44 CC1CCC(CNC(=O)c2cccc3c2OCCN3)CC1 ZINC000147302935 CG For-Sale Anodyne HTR4 40 42 CN(C)C1(Cn2c(N)nc3c(F)cccc32)CCCC1 ZINC000147302949 CF For-Sale Anodyne TLR8 0 40 CCCCCCCCNC(=O)c1ccccc1C#CCN ZINC000147302985 CG For-Sale Mild ASAH1 87 35 O=C(O)C1(NCc2ccc(Cl)cc2Cl)CCC1 ZINC000147302987 CG On-Demand Anodyne P2RX7 33 42 O=C(O)C1(NCc2ccc(Cl)cc2Cl)CCC1 ZINC000147302987 CG On-Demand Anodyne EPHX2 17 49 NS(=O)(=O)c1ccc(OCCN2CCCC2)c(F)c1F ZINC000147303079 DD For-Sale Anodyne LTA4H 35 44 NS(=O)(=O)c1ccc(OCCN2CCCC2)c(F)c1F ZINC000147303079 DD For-Sale Anodyne HRH3 19 46 NS(=O)(=O)c1ccc(OCCN2CCCC2)c(F)c1F ZINC000147303079 DD For-Sale Anodyne PSMB2 47 38 NS(=O)(=O)c1ccc(OCCN2CCCC2)c(F)c1F ZINC000147303079 DD For-Sale Anodyne PSMB1 42 39 O=C1CC[C@H](C(=O)N[C@@H](CO)c2ccccc2)CN1 ZINC000147303090 CC On-Demand Anodyne F11 40 37 C[C@H](CNS(=O)(=O)c1ccc2c(c1)CCC2)CC(=O)O ZINC000147303103 CD On-Demand Anodyne CA7 17 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1C(F)(F)F ZINC000147303110 EE On-Demand Anodyne RBP4 42 35 CN(C)NC(=O)c1ccc(CCN)cc1 ZINC000147303168 BC For-Sale Reactive ECR 52 40 CN(C)NC(=O)c1ccc(CCN)cc1 ZINC000147303168 BC For-Sale Reactive TAAR1 23 42 CN(C)NC(=O)c1ccc(CCN)cc1 ZINC000147303168 BC For-Sale Reactive E3UJZ5_SPOLI 49 40 CN(C)NC(=O)c1ccc(CCN)cc1 ZINC000147303168 BC For-Sale Reactive H9TVJ1_CHISP 0 42 CCCCCCCCNC(=O)c1ccc(C#CCN)cc1 ZINC000147303175 CG For-Sale Mild FOLH1 24 45 CCCCCCCCNC(=O)c1ccc(C#CCN)cc1 ZINC000147303175 CG For-Sale Mild ASAH1 86 36 Cc1cc(C(=O)NCCn2ccnc2)cc([N+](=O)[O-])c1 ZINC000147303210 CD On-Demand Bother TBXAS1 31 45 Cc1cc(C(=O)NCCn2ccnc2)cc([N+](=O)[O-])c1 ZINC000147303210 CD On-Demand Bother QPCT 29 41 O=C(NCC(F)(F)F)Nc1cccc(-c2cnc3cc(-c4ccc(NC5CCOCC5)nn4)ccn23)c1 ZINC000147303216 KJ Annotated Anodyne MAPK1 53 34 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccccc1C(F)(F)F ZINC000147303305 EE On-Demand Anodyne RBP4 42 35 C[C@@H](CNS(=O)(=O)c1ccc2c(c1)CCC2)CC(=O)O ZINC000147303313 CD On-Demand Anodyne CA7 17 42 O=C1CC[C@@H](C(=O)N[C@H](CO)Cc2ccccc2)CN1 ZINC000147303324 CC On-Demand Anodyne F11 50 38 CCCCCCCCNC(=O)c1cccc(C#CCN)c1 ZINC000147303345 CG For-Sale Mild DRD3 19 46 CCCCCCCCNC(=O)c1cccc(C#CCN)c1 ZINC000147303345 CG For-Sale Mild PLA2G4B 40 36 CCCCCCCCNC(=O)c1cccc(C#CCN)c1 ZINC000147303345 CG For-Sale Mild ASAH1 75 34 N#Cc1c(C2CCCC2)[nH]c(SCc2cccc(F)c2F)nc1=O ZINC000147303347 EH Annotated Mild CXCR2 22 92 O=C1CC[C@@H](C(=O)N[C@@H](CO)Cc2ccccc2)CN1 ZINC000147303522 CC On-Demand Anodyne F11 50 38 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(F)(F)F)c1 ZINC000147303533 EE On-Demand Anodyne DHODH 19 47 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(C(F)(F)F)c1 ZINC000147303533 EE On-Demand Anodyne CCR2 40 39 COc1ccc(-c2[nH]c(SCc3cccc(F)c3F)nc(=O)c2C#N)cc1C ZINC000147303541 GI Annotated Mild CXCR2 15 69 CCCCCCCCNC(=O)c1ccc(C#CCN)s1 ZINC000147303553 CG For-Sale Mild ASAH1 77 36 O=C(NCCc1ccc2c(c1)OCO2)[C@H]1Cc2ccccc2CN1 ZINC000147303597 DD On-Demand Anodyne MC4R 31 40 O=C(NCCc1ccc2c(c1)OCO2)[C@H]1Cc2ccccc2CN1 ZINC000147303597 DD On-Demand Anodyne NOS2 91 42 CCNc1ccc([N+](=O)[O-])c(Oc2ccc(Cl)cc2Br)n1 ZINC000147303683 FJ For-Sale Bother S1PR4 0 47 C[C@@H](Cc1cccc(F)c1)C(=O)N(C)C1CCCC1 ZINC000147303719 CG On-Demand Anodyne PRSS1 15 41 CCCCCCCCNS(=O)(=O)c1cccc(Br)c1 ZINC000147303733 EI For-Sale Mild FBP1 23 41 CCCCCCCCNS(=O)(=O)c1cccc(Br)c1 ZINC000147303733 EI For-Sale Mild ALOX15 49 40 O=C1CC[C@H](C(=O)N[C@H](CO)Cc2ccccc2)CN1 ZINC000147303746 CC On-Demand Anodyne F11 50 38 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(C(F)(F)F)c1 ZINC000147303769 EE On-Demand Anodyne CCR2 40 39 N#Cc1c(C2CCC2)[nH]c(SCc2cccc(F)c2F)nc1=O ZINC000147303782 EG Annotated Mild CXCR2 22 92 O=C(NCCc1cccnc1)[C@@H]1CCC(=O)N(Cc2ccccc2)[C@@H]1c1ccccc1 ZINC000147303807 HH On-Demand Anodyne P2RX7 18 41 O=C(NCCc1cccnc1)[C@@H]1CCC(=O)N(Cc2ccccc2)[C@@H]1c1ccccc1 ZINC000147303807 HH On-Demand Anodyne NAMPT 43 39 Cc1ccnc(NCCCCC(C)C)c1N ZINC000147303812 BG For-Sale Anodyne UTS2R 0 41 CCc1ccc([C@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147303841 EI On-Demand Anodyne CYP3A4 17 44 O=Cc1c[nH]c2c(F)c(Cl)ccc12 ZINC000147303844 AF For-Sale Anodyne PIM3 15 44 C[C@H](Cc1cccc(F)c1)C(=O)N(C)C1CCCC1 ZINC000147303926 CG On-Demand Anodyne PRSS1 15 41 O=C1CC[C@H](C(=O)N[C@@H](CO)Cc2ccccc2)CN1 ZINC000147303961 CC On-Demand Anodyne F11 50 38 C[C@H](CNS(=O)(=O)c1cccc2cnccc12)CC(=O)O ZINC000147303966 DD On-Demand Anodyne KCNA5 0 51 C[C@H](CNS(=O)(=O)c1cccc2cnccc12)CC(=O)O ZINC000147303966 DD On-Demand Anodyne TRPV1 36 42 C[C@H](CNS(=O)(=O)c1cccc2cnccc12)CC(=O)O ZINC000147303966 DD On-Demand Anodyne P2RX7 36 52 C[C@H](CNS(=O)(=O)c1cccc2cnccc12)CC(=O)O ZINC000147303966 DD On-Demand Anodyne Q95J97_RABIT 0 59 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc2cnccc12 ZINC000147303997 DD On-Demand Anodyne TRPV1 52 48 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc2cnccc12 ZINC000147303997 DD On-Demand Anodyne CDK5 28 45 CCc1ccc([C@@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147304023 EI On-Demand Anodyne CYP3A4 17 44 CC(C)c1[nH]c(SCc2cccc(F)c2F)nc(=O)c1C#N ZINC000147304027 DG Annotated Mild CXCR2 29 41 CC(C)c1[nH]c(SCc2cccc(F)c2F)nc(=O)c1C#N ZINC000147304027 DG Annotated Mild NS5B 23 45 O=C(NCCc1cccnc1)[C@@H]1CCC(=O)N(Cc2ccccc2)[C@H]1c1ccccc1 ZINC000147304033 HH On-Demand Anodyne P2RX7 18 41 O=C(NCCc1cccnc1)[C@@H]1CCC(=O)N(Cc2ccccc2)[C@H]1c1ccccc1 ZINC000147304033 HH On-Demand Anodyne NAMPT 43 39 O=C(CNC1(C(=O)O)CCC1)NCc1ccccc1Cl ZINC000147304058 CD For-Sale Anodyne P2RX7 32 44 CC(C)S(=O)(=O)NC(=O)c1cccc(N)c1 ZINC000147304143 BC For-Sale Anodyne ABAT 22 44 COc1cccc(CNc2ccc([C@@H](C)CC(=O)O)cc2)c1 ZINC000147304170 CH On-Demand Anodyne ANPEP 16 47 COc1cccc(CNc2ccc([C@@H](C)CC(=O)O)cc2)c1 ZINC000147304170 CH On-Demand Anodyne CTSK 20 41 COc1cccc(CNc2ccc([C@@H](C)CC(=O)O)cc2)c1 ZINC000147304170 CH On-Demand Anodyne CTSL 21 41 COc1cccc(CNc2ccc([C@@H](C)CC(=O)O)cc2)c1 ZINC000147304170 CH On-Demand Anodyne ROCK1 39 40 COc1cccc(CNc2ccc([C@@H](C)CC(=O)O)cc2)c1 ZINC000147304170 CH On-Demand Anodyne MTNR1A 39 42 COc1cccc(CNc2ccc([C@@H](C)CC(=O)O)cc2)c1 ZINC000147304170 CH On-Demand Anodyne MTNR1B 42 43 COc1cccc(CNc2ccc([C@@H](C)CC(=O)O)cc2)c1 ZINC000147304170 CH On-Demand Anodyne ROCK2 44 44 COc1cccc(CNc2ccc([C@@H](C)CC(=O)O)cc2)c1 ZINC000147304170 CH On-Demand Anodyne PTPRB 17 42 COc1cccc(CNc2ccc([C@@H](C)CC(=O)O)cc2)c1 ZINC000147304170 CH On-Demand Anodyne FFAR1 46 50 COc1cccc(CNc2ccc([C@@H](C)CC(=O)O)cc2)c1 ZINC000147304170 CH On-Demand Anodyne AKR1C2 41 33 COc1cccc(CNc2ccc([C@@H](C)CC(=O)O)cc2)c1 ZINC000147304170 CH On-Demand Anodyne DRTS_TRYCR 43 32 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc2cnccc12 ZINC000147304186 DD On-Demand Anodyne TRPV1 52 48 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc2cnccc12 ZINC000147304186 DD On-Demand Anodyne CDK5 28 45 C[C@@H](CNS(=O)(=O)c1cccc2cnccc12)CC(=O)O ZINC000147304202 DD On-Demand Anodyne KCNA5 0 51 C[C@@H](CNS(=O)(=O)c1cccc2cnccc12)CC(=O)O ZINC000147304202 DD On-Demand Anodyne TRPV1 36 42 C[C@@H](CNS(=O)(=O)c1cccc2cnccc12)CC(=O)O ZINC000147304202 DD On-Demand Anodyne P2RX7 36 52 C[C@@H](CNS(=O)(=O)c1cccc2cnccc12)CC(=O)O ZINC000147304202 DD On-Demand Anodyne Q95J97_RABIT 0 59 CC(C)c1ccc([C@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147304235 EJ On-Demand Anodyne CYP3A4 18 43 O=C(NCCc1cccnc1)[C@H]1CCC(=O)N(Cc2ccccc2)[C@@H]1c1ccccc1 ZINC000147304246 HH On-Demand Anodyne P2RX7 18 41 O=C(NCCc1cccnc1)[C@H]1CCC(=O)N(Cc2ccccc2)[C@@H]1c1ccccc1 ZINC000147304246 HH On-Demand Anodyne NAMPT 43 39 O=C(Nc1cccc(Cn2cncn2)c1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147304284 FH On-Demand Anodyne CYP19A1 17 41 CC(C)CCCCN[C@@H](C)c1ccc(C(F)(F)F)cc1 ZINC000147304291 CK For-Sale Anodyne CASR 15 42 CCCCCCCCNS(=O)(=O)c1ccc(Br)c(C)c1 ZINC000147304350 FI For-Sale Mild TBXA2R 15 42 CCCCCCCCNS(=O)(=O)c1ccc(Br)c(C)c1 ZINC000147304350 FI For-Sale Mild ALOX15 53 42 CCCCCCCCNS(=O)(=O)c1ccc(Br)c(C)c1 ZINC000147304350 FI For-Sale Mild LEF 19 41 COc1cccc(CNc2ccc([C@H](C)CC(=O)O)cc2)c1 ZINC000147304402 CH On-Demand Anodyne ANPEP 16 47 COc1cccc(CNc2ccc([C@H](C)CC(=O)O)cc2)c1 ZINC000147304402 CH On-Demand Anodyne CTSK 20 41 COc1cccc(CNc2ccc([C@H](C)CC(=O)O)cc2)c1 ZINC000147304402 CH On-Demand Anodyne CTSL 21 41 COc1cccc(CNc2ccc([C@H](C)CC(=O)O)cc2)c1 ZINC000147304402 CH On-Demand Anodyne ROCK1 39 40 COc1cccc(CNc2ccc([C@H](C)CC(=O)O)cc2)c1 ZINC000147304402 CH On-Demand Anodyne MTNR1A 39 42 COc1cccc(CNc2ccc([C@H](C)CC(=O)O)cc2)c1 ZINC000147304402 CH On-Demand Anodyne MTNR1B 42 43 COc1cccc(CNc2ccc([C@H](C)CC(=O)O)cc2)c1 ZINC000147304402 CH On-Demand Anodyne ROCK2 44 44 COc1cccc(CNc2ccc([C@H](C)CC(=O)O)cc2)c1 ZINC000147304402 CH On-Demand Anodyne PTPRB 17 42 COc1cccc(CNc2ccc([C@H](C)CC(=O)O)cc2)c1 ZINC000147304402 CH On-Demand Anodyne FFAR1 46 50 COc1cccc(CNc2ccc([C@H](C)CC(=O)O)cc2)c1 ZINC000147304402 CH On-Demand Anodyne AKR1C2 41 33 COc1cccc(CNc2ccc([C@H](C)CC(=O)O)cc2)c1 ZINC000147304402 CH On-Demand Anodyne DRTS_TRYCR 43 32 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne HTR1A 143 60 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne DRD2 103 48 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne DRD1 31 45 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne DRD4 63 45 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne ADRA1D 56 57 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne HTR2A 96 53 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne HTR2C 57 50 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne SLC6A4 29 49 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne ADRA1A 80 57 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne ADRA1B 48 57 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne DRD3 129 53 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne DRD5 28 41 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne HTR7 147 45 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne SIGMAR1 17 43 Cc1cc(C)n([C@@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304405 GF On-Demand Anodyne HTR6 21 42 COc1ccc(Cl)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147304408 ED On-Demand Anodyne COLA 46 33 COc1ccc(Cl)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147304408 ED On-Demand Anodyne CPT1B 40 31 COc1ccc(Cl)cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147304408 ED On-Demand Anodyne RBP4 25 42 O=C(NCCc1cccnc1)[C@H]1CCC(=O)N(Cc2ccccc2)[C@H]1c1ccccc1 ZINC000147304454 HH On-Demand Anodyne P2RX7 18 41 O=C(NCCc1cccnc1)[C@H]1CCC(=O)N(Cc2ccccc2)[C@H]1c1ccccc1 ZINC000147304454 HH On-Demand Anodyne NAMPT 43 39 CC(C)c1ccc([C@@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147304455 EJ On-Demand Anodyne CYP3A4 18 43 CC(C)CCCCN[C@H](C)c1ccc(C(F)(F)F)cc1 ZINC000147304522 CK For-Sale Anodyne CASR 15 42 O=C(Nc1cccc(Cn2cncn2)c1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147304541 FH On-Demand Anodyne CYP19A1 17 41 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne HTR1A 143 60 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne DRD2 103 48 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne DRD1 31 45 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne DRD4 63 45 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne ADRA1D 56 57 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne HTR2A 96 53 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne HTR2C 57 50 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne SLC6A4 29 49 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne ADRA1A 80 57 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne ADRA1B 48 57 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne DRD3 129 53 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne DRD5 28 41 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne HTR7 147 45 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne SIGMAR1 17 43 Cc1cc(C)n([C@H](C)C(=O)NCCCCN2CCN(c3ccccc3)CC2)n1 ZINC000147304586 GF On-Demand Anodyne HTR6 21 42 COc1ccc(Cl)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147304601 ED On-Demand Anodyne CPT1B 40 31 COc1ccc(Cl)cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147304601 ED On-Demand Anodyne RBP4 25 42 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother CHRM2 20 40 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother DRD2 15 55 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother DRD4 43 57 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother ACHE 35 51 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother DRD3 32 50 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother CHRM3 26 40 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother TACR1 17 47 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother SIGMAR1 44 56 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother SSTR5 46 44 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother CCR3 33 46 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother UTS2R 21 44 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother CCR2 21 55 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother SLC6A5 26 43 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother BACE1 19 54 Cc1cc(C(=O)N[C@@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304668 EF On-Demand Bother MCHR1 38 54 CC(C)COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147304727 GD On-Demand Anodyne HRH2 16 41 O=C(Nc1cccc(Cn2cncn2)c1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147304761 FH On-Demand Anodyne CYP19A1 17 41 C[C@H](NC(=O)N(C)Cc1cscn1)c1cc2ccccc2o1 ZINC000147304779 DH On-Demand Anodyne CYP3A4 20 44 Cc1ccncc1NC(=O)c1cccc2c1OCCN2 ZINC000147304815 CE For-Sale Anodyne G2YM83_BOTF4 51 33 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother CHRM2 20 40 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother DRD2 15 55 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother DRD4 43 57 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother ACHE 35 51 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother DRD3 32 50 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother CHRM3 26 40 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother TACR1 17 47 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother SIGMAR1 44 56 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother SSTR5 46 44 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother CCR3 33 46 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother UTS2R 21 44 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother CCR2 21 55 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother SLC6A5 26 43 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother BACE1 19 54 Cc1cc(C(=O)N[C@H]2CCN(Cc3ccccc3)C2)cc([N+](=O)[O-])c1 ZINC000147304886 EF On-Demand Bother MCHR1 38 54 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne FABP4 17 74 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne PAOX 42 47 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne S1PR4 18 52 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne S1PR3 28 52 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne PLA2G4B 37 40 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne CES2 50 48 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne S1PR2 58 54 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne CES1 26 42 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne EST1_PIG 65 48 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne CES2C 58 48 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne FABP3 45 59 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne FABP5 25 74 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne Q8WS26_TRYCR 43 44 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne FABP1 19 59 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne ASAH1 81 35 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne LASR 46 33 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne NOD1 61 39 CCCCCCCCCNCCCCCCC(=O)O ZINC000147304910 CI For-Sale Anodyne CQSS 68 42 CC(C)COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147304911 GD On-Demand Anodyne HRH2 16 41 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cc2ccccc2o1 ZINC000147304962 DH On-Demand Anodyne CYP3A4 20 44 COc1cccc([C@H](O)CNC2(C(=O)O)CCC2)c1 ZINC000147304988 CD For-Sale Anodyne ADRB3 53 38 COc1cccc([C@H](O)CNC2(C(=O)O)CCC2)c1 ZINC000147304988 CD For-Sale Anodyne MTNR1A 37 40 COc1cccc([C@H](O)CNC2(C(=O)O)CCC2)c1 ZINC000147304988 CD For-Sale Anodyne MTNR1B 39 40 COc1cccc([C@H](O)CNC2(C(=O)O)CCC2)c1 ZINC000147304988 CD For-Sale Anodyne PHES 0 47 CCCOCC(=O)NCCc1cccnc1 ZINC000147305058 BD On-Demand Anodyne TBXAS1 36 42 CCCOCC(=O)NCCc1cccnc1 ZINC000147305058 BD On-Demand Anodyne PTAFR 37 43 CCCOCC(=O)NCCc1cccnc1 ZINC000147305058 BD On-Demand Anodyne NAMPT 31 40 CCCOCC(=O)NCCc1cccnc1 ZINC000147305058 BD On-Demand Anodyne ISPH 0 44 COc1ccc(Br)c(CNC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147305102 GE On-Demand Anodyne MTNR1A 62 42 COc1ccc(Br)c(CNC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147305102 GE On-Demand Anodyne MTNR1B 44 37 COc1ccc(Br)c(CNC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147305102 GE On-Demand Anodyne MT-ND1 15 40 CCOC(=O)C[C@H](NC(=O)c1cc(OC)ccc1[N+](=O)[O-])c1cccc(OC)c1 ZINC000147305161 HG On-Demand Bother TAAR1 22 41 COc1cccc([C@@H](O)CNC2(C(=O)O)CCC2)c1 ZINC000147305196 CD For-Sale Anodyne ADRB3 53 38 COc1cccc([C@@H](O)CNC2(C(=O)O)CCC2)c1 ZINC000147305196 CD For-Sale Anodyne MTNR1A 37 40 COc1cccc([C@@H](O)CNC2(C(=O)O)CCC2)c1 ZINC000147305196 CD For-Sale Anodyne MTNR1B 39 40 COc1cccc([C@@H](O)CNC2(C(=O)O)CCC2)c1 ZINC000147305196 CD For-Sale Anodyne PHES 0 47 Cc1oc2ccccc2c1[C@H](O)Cc1ccc(F)cc1Cl ZINC000147305214 DJ For-Sale Anodyne P2RX7 48 37 Cc1ccc(NC(=O)c2cccc3c2OCCN3)cc1Br ZINC000147305249 EH For-Sale Anodyne AVPR2 16 40 Cc1ccc(NC(=O)c2cccc3c2OCCN3)cc1Br ZINC000147305249 EH For-Sale Anodyne KCNK3 66 38 Cc1ccc(NC(=O)c2cccc3c2OCCN3)cc1Br ZINC000147305249 EH For-Sale Anodyne KCNK9 66 36 CNc1cc(Oc2ccc(Cl)cc2Br)cc([N+](=O)[O-])c1 ZINC000147305264 FJ For-Sale Bother ENR 0 48 CNc1cc(Oc2ccc(Cl)cc2Br)cc([N+](=O)[O-])c1 ZINC000147305264 FJ For-Sale Bother PPOX1 15 47 C[C@H](CNS(=O)(=O)CCc1ccncc1)CC(=O)O ZINC000147305266 CC For-Sale Anodyne MMP12 15 43 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc3c(c2)CCCC(=O)N3)C1 ZINC000147305268 HC On-Demand Anodyne PKM 34 45 CCCCO[C@@H](C)C(=O)NCCc1cccnc1 ZINC000147305321 CD On-Demand Anodyne TBXAS1 48 42 CCCCO[C@@H](C)C(=O)NCCc1cccnc1 ZINC000147305321 CD On-Demand Anodyne PTAFR 42 46 CCCCO[C@@H](C)C(=O)NCCc1cccnc1 ZINC000147305321 CD On-Demand Anodyne KCNA5 15 41 CCCCO[C@@H](C)C(=O)NCCc1cccnc1 ZINC000147305321 CD On-Demand Anodyne PLM2_PLAFA 24 41 CCCCO[C@@H](C)C(=O)NCCc1cccnc1 ZINC000147305321 CD On-Demand Anodyne NAMPT 25 41 CCOC(=O)C[C@@H](NC(=O)c1cc(OC)ccc1[N+](=O)[O-])c1cccc(OC)c1 ZINC000147305368 HG On-Demand Bother TAAR1 22 41 CC(C)CCCCNc1ccc(N)c(OCC(C)C)n1 ZINC000147305420 CH For-Sale Anodyne HRH4 0 41 Cc1oc2ccccc2c1[C@@H](O)Cc1ccc(F)cc1Cl ZINC000147305436 DJ For-Sale Anodyne P2RX7 48 37 NCC(=O)Nc1csc2ncccc12 ZINC000147305445 BD For-Sale Anodyne MAPK9 22 40 NCC(=O)Nc1csc2ncccc12 ZINC000147305445 BD For-Sale Anodyne MAPK10 24 40 C[C@@H](CNS(=O)(=O)CCc1ccncc1)CC(=O)O ZINC000147305452 CC For-Sale Anodyne MMP12 15 43 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc3c(c2)CCCC(=O)N3)C1 ZINC000147305466 HC On-Demand Anodyne PKM 34 45 CCCOc1nc(N)nc(Oc2ccc(Cl)cc2Br)n1 ZINC000147305490 FG For-Sale Anodyne S1PR4 23 40 CCCCO[C@H](C)C(=O)NCCc1cccnc1 ZINC000147305519 CD On-Demand Anodyne TBXAS1 48 42 CCCCO[C@H](C)C(=O)NCCc1cccnc1 ZINC000147305519 CD On-Demand Anodyne PTAFR 42 46 CCCCO[C@H](C)C(=O)NCCc1cccnc1 ZINC000147305519 CD On-Demand Anodyne KCNA5 15 41 CCCCO[C@H](C)C(=O)NCCc1cccnc1 ZINC000147305519 CD On-Demand Anodyne PLM2_PLAFA 24 41 CCCCO[C@H](C)C(=O)NCCc1cccnc1 ZINC000147305519 CD On-Demand Anodyne NAMPT 25 41 O=S(=O)(c1ccc(F)cc1)N(CCBr)C1CCCCC1 ZINC000147305577 FH For-Sale Reactive AVPR1B 18 40 CCOC(=O)C[C@H](NC(=O)c1ccn(-c2cccc(F)c2)n1)c1cccc(OC)c1 ZINC000147305584 HG On-Demand Anodyne CTSA 47 36 CC(C)c1cccc(C(C)C)c1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147305639 EH On-Demand Anodyne SOAT1 55 44 COc1cc([N+](=O)[O-])ccc1S(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000147305696 GC On-Demand Bother ADRA1B 19 44 CNc1ccc([N+](=O)[O-])c(Oc2ccc(Cl)cc2Br)n1 ZINC000147305718 FI For-Sale Bother S1PR4 17 46 C/C=C(/CC)c1ccc(C(=O)OC)c(C)c1 ZINC000147305744 BH For-Sale Anodyne CA7 16 44 CCOC(=O)C[C@@H](NC(=O)c1ccn(-c2cccc(F)c2)n1)c1cccc(OC)c1 ZINC000147305789 HG On-Demand Anodyne CTSA 47 36 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(Cn3cncn3)c1)C2 ZINC000147305797 FF On-Demand Anodyne ROCK2 31 44 CCCOc1ccc([C@@H](C)NCCCCC(C)C)cc1 ZINC000147305839 CJ For-Sale Anodyne ACACA 47 46 CCCOc1ccc([C@@H](C)NCCCCC(C)C)cc1 ZINC000147305839 CJ For-Sale Anodyne ACACB 26 46 CCCOc1ccc([C@@H](C)NCCCCC(C)C)cc1 ZINC000147305839 CJ For-Sale Anodyne SLC2A1 0 55 CCCOc1ccc([C@@H](C)NCCCCC(C)C)cc1 ZINC000147305839 CJ For-Sale Anodyne HT1 0 55 CCCOc1ccc([C@@H](C)NCCCCC(C)C)cc1 ZINC000147305839 CJ For-Sale Anodyne LMGT2 0 55 CC(C)c1cccc(C(C)C)c1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147305868 EH On-Demand Anodyne SOAT1 55 44 COc1cc([N+](=O)[O-])ccc1S(=O)(=O)N[C@H]1CCCN(S(C)(=O)=O)C1 ZINC000147305914 GC On-Demand Bother ADRA1B 19 44 CC(=O)OCc1ccc(OC2CCCCC2)cc1 ZINC000147305933 BG For-Sale Anodyne PRSS2 57 34 CC(=O)OCc1ccc(OC2CCCCC2)cc1 ZINC000147305933 BG For-Sale Anodyne HRH3 17 41 CC(=O)OCc1ccc(OC2CCCCC2)cc1 ZINC000147305933 BG For-Sale Anodyne EPHX2 20 46 CC(=O)OCc1ccc(OC2CCCCC2)cc1 ZINC000147305933 BG For-Sale Anodyne NAAA 26 57 CC(=O)OCc1ccc(OC2CCCCC2)cc1 ZINC000147305933 BG For-Sale Anodyne SLC12A5 42 35 Nc1ncc(Br)c(Oc2ccc(Cl)cc2Br)n1 ZINC000147305940 GI For-Sale Anodyne P2RX2 39 41 Nc1ncc(Br)c(Oc2ccc(Cl)cc2Br)n1 ZINC000147305940 GI For-Sale Anodyne P2RX3 25 41 Nc1ncc(Br)c(Oc2ccc(Cl)cc2Br)n1 ZINC000147305940 GI For-Sale Anodyne S1PR4 0 40 Nc1ncc(Br)c(Oc2ccc(Cl)cc2Br)n1 ZINC000147305940 GI For-Sale Anodyne AGPAT2 46 37 Nc1c(Oc2ccc(Cl)c(F)c2)cccc1C(=O)O ZINC000147306003 CH For-Sale Anodyne PYGL 23 42 Nc1c(Oc2ccc(Cl)c(F)c2)cccc1C(=O)O ZINC000147306003 CH For-Sale Anodyne PYGM 34 42 CN(C)C(=O)[C@H]1CCC(=O)N(Cc2ccccc2)[C@@H]1c1ccccc1 ZINC000147306014 EG On-Demand Anodyne P2RX7 20 44 CCCOc1ccc([C@H](C)NCCCCC(C)C)cc1 ZINC000147306042 CJ For-Sale Anodyne ACACA 47 46 CCCOc1ccc([C@H](C)NCCCCC(C)C)cc1 ZINC000147306042 CJ For-Sale Anodyne ACACB 26 46 CCCOc1ccc([C@H](C)NCCCCC(C)C)cc1 ZINC000147306042 CJ For-Sale Anodyne SLC2A1 0 55 CCCOc1ccc([C@H](C)NCCCCC(C)C)cc1 ZINC000147306042 CJ For-Sale Anodyne HT1 0 55 CCCOc1ccc([C@H](C)NCCCCC(C)C)cc1 ZINC000147306042 CJ For-Sale Anodyne LMGT2 0 55 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccccc1OC(C)C)C2 ZINC000147306053 FG On-Demand Anodyne MTNR1A 44 42 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccccc1OC(C)C)C2 ZINC000147306053 FG On-Demand Anodyne MTNR1B 32 42 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccccc1OC(C)C)C2 ZINC000147306053 FG On-Demand Anodyne ROCK2 25 40 CC(C)(C)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147306094 DF On-Demand Anodyne DHODH 71 41 C[C@H](CN)CCC(=O)NN(C)C ZINC000147306133 AB For-Sale Reactive KDM7A 0 50 CN(C)C(=O)[C@@H]1CCC(=O)N(Cc2ccccc2)[C@H]1c1ccccc1 ZINC000147306199 EG On-Demand Anodyne P2RX7 20 44 CCCCCCCCNS(=O)(=O)c1ccc(OC)c(Br)c1 ZINC000147306243 GI For-Sale Mild S1PR2 40 37 CCCCCCCCNS(=O)(=O)c1ccc(OC)c(Br)c1 ZINC000147306243 GI For-Sale Mild ALOX15 50 43 CCCCCCCCNS(=O)(=O)c1ccc(OC)c(Br)c1 ZINC000147306243 GI For-Sale Mild IAP 0 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccccc1OC(C)C)C2 ZINC000147306246 FG On-Demand Anodyne MTNR1A 44 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccccc1OC(C)C)C2 ZINC000147306246 FG On-Demand Anodyne MTNR1B 32 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccccc1OC(C)C)C2 ZINC000147306246 FG On-Demand Anodyne ROCK2 25 40 CCNc1cccc(Oc2ccc(Cl)cc2Br)c1[N+](=O)[O-] ZINC000147306294 FK For-Sale Bother ENR 0 42 CC(C)(C)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147306297 DF On-Demand Anodyne DHODH 71 41 C[C@@H](CN)CCC(=O)NN(C)C ZINC000147306322 AB For-Sale Reactive KDM7A 0 50 O=C(c1cccc(CNS(=O)(=O)c2cccc3ccccc23)c1)N1CCOCC1 ZINC000147306375 HF On-Demand Anodyne TRY2_BOVIN 79 44 O=C(c1cccc(CNS(=O)(=O)c2cccc3ccccc23)c1)N1CCOCC1 ZINC000147306375 HF On-Demand Anodyne NPY5R 22 48 O=C(c1cccc(CNS(=O)(=O)c2cccc3ccccc23)c1)N1CCOCC1 ZINC000147306375 HF On-Demand Anodyne PARP1 18 50 O=C(c1cccc(CNS(=O)(=O)c2cccc3ccccc23)c1)N1CCOCC1 ZINC000147306375 HF On-Demand Anodyne ST14 26 42 CN(C)C(=O)[C@H]1CCC(=O)N(Cc2ccccc2)[C@H]1c1ccccc1 ZINC000147306386 EG On-Demand Anodyne P2RX7 20 44 O=C(O)c1cccc(OP(=O)(O)O)c1 ZINC000147306421 BC In-Stock Anodyne SRD5A2 0 42 O=C(O)c1cccc(OP(=O)(O)O)c1 ZINC000147306421 BC In-Stock Anodyne PLA2G4B 16 41 O=C(O)c1cccc(OP(=O)(O)O)c1 ZINC000147306421 BC In-Stock Anodyne FABH 0 47 O=C(O)c1cccc(OP(=O)(O)O)c1 ZINC000147306421 BC In-Stock Anodyne AROA 0 67 O=C(O)c1cccc(OP(=O)(O)O)c1 ZINC000147306421 BC In-Stock Anodyne AKR1C3 43 59 O=C(O)c1cccc(OP(=O)(O)O)c1 ZINC000147306421 BC In-Stock Anodyne KCNK3 42 40 CC(C)CCCCNc1cc2c(cc1N)CCC(=O)N2 ZINC000147306438 CG For-Sale Anodyne PKM 37 42 NS(=O)(=O)c1ccc(OCCc2cccnc2)c(F)c1F ZINC000147306443 DD For-Sale Anodyne CA14 23 42 CC[C@H](NC(=O)c1ccc2c(c1)COC2)c1ccc2c(c1)OCCO2 ZINC000147306462 EG On-Demand Anodyne UTS2 54 32 CC(=O)Nc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147306495 DD On-Demand Anodyne KCNK3 57 38 CN(C)NC(=O)C[C@@H](N)C(C)(C)C ZINC000147306560 AC For-Sale Reactive KDM7A 0 41 COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1F ZINC000147306579 FC On-Demand Anodyne ADRA1D 26 42 COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1F ZINC000147306579 FC On-Demand Anodyne ADRA1A 19 41 COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1F ZINC000147306579 FC On-Demand Anodyne ADRA1B 34 42 Cc1cccc2nc(N)n(CC3(N(C)C)CCCC3)c12 ZINC000147306589 CF For-Sale Anodyne TLR8 0 52 C#CCNC(=O)CCNCc1ccc(-n2cccn2)cc1 ZINC000147306655 CD On-Demand Mild AMP1_PLAFQ 52 36 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H](c1ccc(F)cc1)[C@@H]1CCCO1)C2 ZINC000147306675 GG On-Demand Anodyne ROCK2 22 41 CC(=O)Nc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147306681 DD On-Demand Anodyne KCNK3 57 38 CN(C)NC(=O)C[C@H](N)C(C)(C)C ZINC000147306741 AC For-Sale Reactive KDM7A 0 41 COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1F ZINC000147306772 FC On-Demand Anodyne ADRA1D 26 42 COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1F ZINC000147306772 FC On-Demand Anodyne ADRA1A 19 41 COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1F ZINC000147306772 FC On-Demand Anodyne ADRA1B 34 42 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1ccccc1-n1cccn1 ZINC000147306785 HJ On-Demand Anodyne NAMPT 39 42 CCOc1ccc(Oc2cc(NN)nc(C(C)C)n2)cc1 ZINC000147306842 CG For-Sale Anodyne ACACB 17 40 COc1ccc(OC)c([C@H](C)NC(=O)N(C)Cc2cscn2)c1 ZINC000147306893 EG On-Demand Anodyne BMP1 42 33 COC(=O)c1cc(NCCCCC(C)C)cc(C)c1N ZINC000147306914 CH For-Sale Anodyne LEF 69 32 O=C(O)Cn1c(=O)ccc2cc(Cl)c(Cl)cc21 ZINC000147306940 CE For-Sale Anodyne PTGDR2 39 42 CN(C)NC(=O)CCCCN ZINC000147306968 AB For-Sale Reactive APHA 0 41 CN(C)NC(=O)CCCCN ZINC000147306968 AB For-Sale Reactive KDM7A 0 54 O[C@@H]1COC[C@@H]1N1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147306997 CD On-Demand Anodyne DRD4 35 40 O[C@@H]1COC[C@@H]1N1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147306997 CD On-Demand Anodyne SIGMAR1 25 50 COc1ccc2c(c1)OC[C@H](C(=O)N[C@H](c1ccc(F)cc1)[C@@H]1CCCO1)C2 ZINC000147307022 GG On-Demand Anodyne ROCK2 22 41 COc1ccc(OC)c([C@@H](C)NC(=O)N(C)Cc2cscn2)c1 ZINC000147307049 EG On-Demand Anodyne BMP1 42 33 COc1ccc(OC)c(C(=O)N2CCC[C@H](CCBr)C2)c1 ZINC000147307077 FG For-Sale Reactive GRM3 16 48 Cc1cc(NCc2cccc(F)c2)nc(-c2cccnc2)n1 ZINC000147307096 CH On-Demand Anodyne ROS1 59 38 Brc1ncccc1-c1nc2ccccc2s1 ZINC000147307166 CI For-Sale Anodyne LUCI_PHOPY 15 43 Brc1ncccc1-c1nc2ccccc2s1 ZINC000147307166 CI For-Sale Anodyne LUCI_PHOPE 17 43 CC[C@H](N)C(=O)NN(C)C ZINC000147307180 AB For-Sale Reactive DPP7 0 41 CC[C@H](N)C(=O)NN(C)C ZINC000147307180 AB For-Sale Reactive DPP8 0 41 CC[C@H](N)C(=O)NN(C)C ZINC000147307180 AB For-Sale Reactive DPP9 0 41 COc1ccc(OC)c(C(=O)N2CCC[C@@H](CCBr)C2)c1 ZINC000147307243 FG For-Sale Reactive GRM3 16 48 O[C@@H]1COC[C@H]1N1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147307275 CD On-Demand Anodyne DRD4 35 40 O[C@@H]1COC[C@H]1N1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147307275 CD On-Demand Anodyne SIGMAR1 25 50 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000147307313 FG On-Demand Anodyne LTA4H 44 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000147307313 FG On-Demand Anodyne F13A1 22 41 CCC[C@@H](C)CNCCCCC(C)C ZINC000147307318 AH For-Sale Anodyne SPPS 41 35 O=C(O)C1(NCc2cncn2C2CC2)CCC1 ZINC000147307325 BD For-Sale Anodyne CAMC 0 42 O[C@H]1COC[C@H]1N1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147307447 CD On-Demand Anodyne DRD4 35 40 O[C@H]1COC[C@H]1N1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147307447 CD On-Demand Anodyne SIGMAR1 25 50 CCC[C@H](C)CNCCCCC(C)C ZINC000147307469 AH For-Sale Anodyne SPPS 41 35 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000147307483 FG On-Demand Anodyne LTA4H 44 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(Oc2ccccc2)cc1 ZINC000147307483 FG On-Demand Anodyne F13A1 22 41 Cc1cnc(N)nc1Oc1ccc(Cl)cc1Br ZINC000147307642 DH For-Sale Anodyne AGPAT2 44 35 Cc1cnc(N)nc1Oc1ccc(Cl)cc1Br ZINC000147307642 DH For-Sale Anodyne MAP3K14 40 42 O=C(O)CC1(NC(=O)[C@H]2C[C@H]2c2ccccc2)CCC1 ZINC000147307651 CE For-Sale Anodyne GPR88 0 41 O=C(O)CC1(NC(=O)[C@H]2C[C@@H]2c2ccccc2)CCC1 ZINC000147307866 CE For-Sale Anodyne GPR88 0 41 CCOC(=O)c1cc(C)nc2c1c(C)nn2-c1ccccc1 ZINC000147307881 CG For-Sale Anodyne SLC5A1 19 40 CC(C)CCCCNCc1csc(-c2ccc(F)cc2)n1 ZINC000147307958 DJ For-Sale Anodyne AVPR1B 0 47 CC(C)CCCCNCc1csc(-c2ccc(F)cc2)n1 ZINC000147307958 DJ For-Sale Anodyne LEF 80 36 COc1cc(CNCC(F)F)cc(Cl)c1OCC(N)=O ZINC000147307974 DD On-Demand Anodyne LPAR2 27 44 COc1cc(CNCC(F)F)cc(Cl)c1OCC(N)=O ZINC000147307974 DD On-Demand Anodyne PDE6A 41 32 COc1cc(CNCC(F)F)cc(Cl)c1OCC(N)=O ZINC000147307974 DD On-Demand Anodyne S1PR2 26 44 COc1cc(CNCC(F)F)cc(Cl)c1OCC(N)=O ZINC000147307974 DD On-Demand Anodyne DRTS_TRYCR 44 32 CCCCCCCCNc1cc(C(=O)OC)c(N)cc1F ZINC000147308050 CH For-Sale Mild ASAH1 56 38 O=C(O)CC1(NC(=O)[C@@H]2C[C@H]2c2ccccc2)CCC1 ZINC000147308059 CE For-Sale Anodyne GPR88 0 41 COc1ccc(N(C)C(=O)[C@H](Cc2cccc(I)c2)NC(=O)OC(C)(C)C)cc1 ZINC000147308073 KI For-Sale Anodyne PAPA1_CARPA 56 46 COc1ccc(N(C)C(=O)[C@H](Cc2cccc(I)c2)NC(=O)OC(C)(C)C)cc1 ZINC000147308073 KI For-Sale Anodyne CTSL 24 46 COc1ccc(N(C)C(=O)[C@H](Cc2cccc(I)c2)NC(=O)OC(C)(C)C)cc1 ZINC000147308073 KI For-Sale Anodyne CACNA1B 15 40 COc1ccc(N(C)C(=O)[C@H](Cc2cccc(I)c2)NC(=O)OC(C)(C)C)cc1 ZINC000147308073 KI For-Sale Anodyne CTSS 19 46 COc1ccc(N(C)C(=O)[C@H](Cc2cccc(I)c2)NC(=O)OC(C)(C)C)cc1 ZINC000147308073 KI For-Sale Anodyne FPR1 53 42 CCNc1cc(Oc2ccc(Cl)cc2Br)cc([N+](=O)[O-])c1 ZINC000147308103 FK For-Sale Bother ENR 0 45 CCNc1cc(Oc2ccc(Cl)cc2Br)cc([N+](=O)[O-])c1 ZINC000147308103 FK For-Sale Bother PPOX1 15 44 C[C@@H]1CCCN(C(=O)c2cccc3c2OCCN3)CC1 ZINC000147308163 CF For-Sale Anodyne L3MBTL3 46 38 CC[C@@H](C)[C@@H](N)C(=O)NN(C)C ZINC000147308182 AB For-Sale Reactive SLC15A2 0 40 O=C(CNC1(C(=O)O)CCC1)Nc1ccc2c(c1)CCC2 ZINC000147308186 CD For-Sale Anodyne PTPRF 40 30 O=C(O)CC1(NC(=O)[C@@H]2C[C@@H]2c2ccccc2)CCC1 ZINC000147308206 CE For-Sale Anodyne GPR88 0 41 COc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)c(OC)c1 ZINC000147308222 DD On-Demand Anodyne MTNR1A 43 38 CCCCCCCCNc1nccc(C(=O)OC)c1N ZINC000147308244 CG For-Sale Mild UTS2R 16 45 COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c2cccnc12 ZINC000147308330 GC On-Demand Anodyne CCR8 76 37 CC[C@H](C)[C@@H](N)C(=O)NN(C)C ZINC000147308349 AB For-Sale Reactive SLC15A2 0 40 C[C@H]1CCCN(C(=O)c2cccc3c2OCCN3)CC1 ZINC000147308352 CF For-Sale Anodyne L3MBTL3 46 38 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308379 GD On-Demand Anodyne P2RY12 185 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308379 GD On-Demand Anodyne MC4R 89 39 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308379 GD On-Demand Anodyne TRY2_BOVIN 53 35 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308379 GD On-Demand Anodyne CCR1 46 47 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308379 GD On-Demand Anodyne CCKBR 22 43 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308379 GD On-Demand Anodyne DPP7 50 39 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308379 GD On-Demand Anodyne UTS2 44 34 CC[C@@H]1CN(C(=O)Cc2ccc(F)c(F)c2)CC[C@@H]1N ZINC000147308415 CE On-Demand Anodyne MLNR 34 44 CCCCCCCCNc1nccc(C(=O)O)c1N ZINC000147308459 CG For-Sale Mild UTS2R 18 47 CCCCCCCCCCCCCCCCCC(=O)OC[C@@H](O)COC(=O)CCC(=O)O ZINC000147308460 JK For-Sale Anodyne PRKCA 22 54 CCCCCCCCCCCCCCCCCC(=O)OC[C@@H](O)COC(=O)CCC(=O)O ZINC000147308460 JK For-Sale Anodyne LPAR3 41 66 CCCCCCCCCCCCCCCCCC(=O)OC[C@@H](O)COC(=O)CCC(=O)O ZINC000147308460 JK For-Sale Anodyne FABP3 45 43 CCCCCCCCCCCCCCCCCC(=O)OC[C@@H](O)COC(=O)CCC(=O)O ZINC000147308460 JK For-Sale Anodyne FABP5 17 52 CCCCCCCCCCCCCCCCCC(=O)OC[C@@H](O)COC(=O)CCC(=O)O ZINC000147308460 JK For-Sale Anodyne ENPP2 25 57 CCCCCCCCCCCCCCCCCC(=O)OC[C@@H](O)COC(=O)CCC(=O)O ZINC000147308460 JK For-Sale Anodyne NOD1 56 36 CCCCCCCCCCCCCCCCCC(=O)OC[C@@H](O)COC(=O)CCC(=O)O ZINC000147308460 JK For-Sale Anodyne CQSS 68 42 COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c2cccnc12 ZINC000147308550 GC On-Demand Anodyne CCR8 76 37 CNC(=O)c1cccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147308553 DF On-Demand Bother PYGL 22 42 CNC(=O)c1cccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147308553 DF On-Demand Bother DDX3X 0 42 CNC(=O)c1cccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147308553 DF On-Demand Bother SENP1 0 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000147308582 HC On-Demand Anodyne CASR 31 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000147308582 HC On-Demand Anodyne EPHX2 22 50 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000147308582 HC On-Demand Anodyne AKR1C3 57 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308585 GD On-Demand Anodyne P2RY12 185 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308585 GD On-Demand Anodyne MC4R 89 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308585 GD On-Demand Anodyne TRY2_BOVIN 53 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308585 GD On-Demand Anodyne CCR1 46 47 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308585 GD On-Demand Anodyne CCKBR 22 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308585 GD On-Demand Anodyne DPP7 50 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(Cl)cc2)CC1 ZINC000147308585 GD On-Demand Anodyne UTS2 44 34 CC[C@H]1CN(C(=O)Cc2ccc(F)c(F)c2)CC[C@@H]1N ZINC000147308591 CE On-Demand Anodyne MLNR 34 44 Cc1cc(S(=O)(=O)NC[C@@H](C)CC(=O)O)ccc1Br ZINC000147308618 FE On-Demand Anodyne LEF 59 37 CCCCCCCCCCCCCCCCCC(=O)OC[C@H](O)COC(=O)CCC(=O)O ZINC000147308649 JK For-Sale Anodyne PRKCA 22 54 CCCCCCCCCCCCCCCCCC(=O)OC[C@H](O)COC(=O)CCC(=O)O ZINC000147308649 JK For-Sale Anodyne LPAR3 41 66 CCCCCCCCCCCCCCCCCC(=O)OC[C@H](O)COC(=O)CCC(=O)O ZINC000147308649 JK For-Sale Anodyne FABP3 45 43 CCCCCCCCCCCCCCCCCC(=O)OC[C@H](O)COC(=O)CCC(=O)O ZINC000147308649 JK For-Sale Anodyne FABP5 17 52 CCCCCCCCCCCCCCCCCC(=O)OC[C@H](O)COC(=O)CCC(=O)O ZINC000147308649 JK For-Sale Anodyne ENPP2 25 57 CCCCCCCCCCCCCCCCCC(=O)OC[C@H](O)COC(=O)CCC(=O)O ZINC000147308649 JK For-Sale Anodyne NOD1 56 36 CCCCCCCCCCCCCCCCCC(=O)OC[C@H](O)COC(=O)CCC(=O)O ZINC000147308649 JK For-Sale Anodyne CQSS 68 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000147308785 HC On-Demand Anodyne CASR 31 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000147308785 HC On-Demand Anodyne EPHX2 22 50 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCOCC2)c1 ZINC000147308785 HC On-Demand Anodyne AKR1C3 57 43 CC[C@@H]1CN(C(=O)Cc2ccc(F)c(F)c2)CC[C@H]1N ZINC000147308801 CE On-Demand Anodyne MLNR 34 44 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne ALOX5 46 65 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne ACE 19 49 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne MAOB 46 53 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne PPARG 34 48 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne PTGER2 15 40 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne PPARA 46 49 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne MME 22 49 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne LTA4H 48 54 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne PTGER3 52 36 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne ACACA 18 45 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne CTSB 41 46 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne PAPA1_CARPA 49 32 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne CTSK 27 43 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne ACACB 21 45 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne ADAM17 20 41 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne PPARD 22 40 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne CAPNS1 53 34 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne PLA2G4B 61 34 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne FAAH 23 53 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne CAPN1 65 46 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne CAPN2 103 46 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne ACE2 54 49 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne ADAMTS4 34 45 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne NPR 59 35 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne TAAR1 29 45 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne FFAR1 87 52 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne FFAR4 45 38 CCOC(=O)[C@@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147308814 CH For-Sale Anodyne PDS 65 39 Cc1cc(S(=O)(=O)NC[C@H](C)CC(=O)O)ccc1Br ZINC000147308822 FE On-Demand Anodyne LEF 59 37 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1Br ZINC000147308856 HI For-Sale Reactive GRM3 15 48 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1Br ZINC000147308856 HI For-Sale Reactive L3MBTL3 41 38 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1Br ZINC000147308856 HI For-Sale Reactive ACKR3 63 34 CCCCCCCCNc1cccc(C(N)=O)c1N ZINC000147308895 CG For-Sale Mild PARP1 29 41 CCCCCCCCNc1cccc(C(N)=O)c1N ZINC000147308895 CG For-Sale Mild ASAH1 63 32 CC(C)CCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147308901 HD On-Demand Anodyne HRH2 17 45 CC(C)CCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147308901 HD On-Demand Anodyne HRH3 15 45 CC(C)CCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147308901 HD On-Demand Anodyne MMP13 26 41 CC(C)CCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147308901 HD On-Demand Anodyne ADAM17 20 41 CC(C)CCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147308901 HD On-Demand Anodyne MMP3 15 40 CC[C@H]1CN(C(=O)Cc2ccc(F)c(F)c2)CC[C@H]1N ZINC000147308974 CE On-Demand Anodyne MLNR 34 44 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147308975 HC On-Demand Anodyne EPHX2 21 48 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147308975 HC On-Demand Anodyne TGM2 75 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147308975 HC On-Demand Anodyne F13A1 93 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147308975 HC On-Demand Anodyne MERTK 34 46 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147308975 HC On-Demand Anodyne NAMPT 47 46 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne ALOX5 46 65 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne ACE 19 49 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne MAOB 46 53 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne PPARG 34 48 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne PTGER2 15 40 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne PPARA 46 49 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne MME 22 49 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne LTA4H 48 54 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne PTGER3 52 36 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne ACACA 18 45 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne CTSB 41 46 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne PAPA1_CARPA 49 32 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne CTSK 27 43 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne ACACB 21 45 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne ADAM17 20 41 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne PPARD 22 40 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne CAPNS1 53 34 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne PLA2G4B 61 34 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne FAAH 23 53 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne CAPN1 65 46 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne CAPN2 103 46 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne ACE2 54 49 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne ADAMTS4 34 45 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne NPR 59 35 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne TAAR1 29 45 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne FFAR1 87 52 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne FFAR4 45 38 CCOC(=O)[C@H](C)c1ccc(OCc2ccccc2)cc1 ZINC000147309009 CH For-Sale Anodyne PDS 65 39 C[C@H](CNS(=O)(=O)c1ccc(Cl)c([N+](=O)[O-])c1)CC(=O)O ZINC000147309032 ED For-Sale Bother COLA 81 37 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1Br ZINC000147309035 HI For-Sale Reactive GRM3 15 48 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1Br ZINC000147309035 HI For-Sale Reactive L3MBTL3 41 38 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1Br ZINC000147309035 HI For-Sale Reactive ACKR3 63 34 CCCCCCCCNc1ccc(N)c(C(N)=O)c1 ZINC000147309067 CG For-Sale Mild ASAH1 70 32 CC[C@H](NC(=O)[C@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309086 GG On-Demand Anodyne EDNRB 45 41 CC[C@H](NC(=O)[C@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309086 GG On-Demand Anodyne EDNRA 37 41 CC[C@H](NC(=O)[C@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309086 GG On-Demand Anodyne MTNR1A 15 40 CC[C@H](NC(=O)[C@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309086 GG On-Demand Anodyne ROCK2 24 41 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309157 HB On-Demand Anodyne HRH2 17 46 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309157 HB On-Demand Anodyne MMP13 48 42 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309157 HB On-Demand Anodyne ADAM17 32 42 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309157 HB On-Demand Anodyne MMP3 35 40 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309157 HB On-Demand Anodyne MMP9 26 40 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309157 HB On-Demand Anodyne MMP7 40 40 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309157 HB On-Demand Anodyne MMP1 38 40 COC(=O)COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309157 HB On-Demand Anodyne SFRP1 46 30 CC[C@@H]1CN(C(=O)Cn2nnc(-c3ccccc3)n2)CCO1 ZINC000147309162 DC On-Demand Anodyne SCARB1 44 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147309178 HC On-Demand Anodyne EPHX2 21 48 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147309178 HC On-Demand Anodyne TGM2 75 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147309178 HC On-Demand Anodyne F13A1 93 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147309178 HC On-Demand Anodyne MERTK 34 46 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCOCC2)cc1 ZINC000147309178 HC On-Demand Anodyne NAMPT 47 46 CCCNc1ncnc(Oc2ccc(Cl)cc2Br)c1CC ZINC000147309190 FK For-Sale Anodyne HTT 0 42 C[C@@H](CNS(=O)(=O)c1ccc(Cl)c([N+](=O)[O-])c1)CC(=O)O ZINC000147309224 ED For-Sale Bother COLA 81 37 CC[C@@H](NC(=O)[C@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309242 GG On-Demand Anodyne EDNRB 45 41 CC[C@@H](NC(=O)[C@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309242 GG On-Demand Anodyne EDNRA 37 41 CC[C@@H](NC(=O)[C@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309242 GG On-Demand Anodyne MTNR1A 15 40 CC[C@@H](NC(=O)[C@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309242 GG On-Demand Anodyne ROCK2 24 41 CCCCCCCCNc1ccc(N)c(C(=O)O)c1 ZINC000147309258 CH For-Sale Mild RARB 17 41 CCCCCCCCNc1ccc(N)c(C(=O)O)c1 ZINC000147309258 CH For-Sale Mild ASAH1 85 33 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@H](CCBr)C1 ZINC000147309279 FI For-Sale Reactive CACNA1B 55 35 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@H](CCBr)C1 ZINC000147309279 FI For-Sale Reactive CCR2 73 44 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@H](CCBr)C1 ZINC000147309279 FI For-Sale Reactive RHOA 0 47 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@H](CCBr)C1 ZINC000147309279 FI For-Sale Reactive HPGD 17 41 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@H](CCBr)C1 ZINC000147309279 FI For-Sale Reactive MAP3K12 31 43 O=C(O)Cc1ccccc1NC(=O)c1cccc(F)c1Cl ZINC000147309319 DG On-Demand Anodyne CXCL8 41 47 O=C(O)Cc1ccccc1NC(=O)c1cccc(F)c1Cl ZINC000147309319 DG On-Demand Anodyne NR1H4 0 41 O=C(O)Cc1ccccc1NC(=O)c1cccc(F)c1Cl ZINC000147309319 DG On-Demand Anodyne KCNMA1 18 43 O=C(O)Cc1ccccc1NC(=O)c1cccc(F)c1Cl ZINC000147309319 DG On-Demand Anodyne G2YM83_BOTF4 65 33 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309345 HB On-Demand Anodyne HRH2 17 46 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309345 HB On-Demand Anodyne MMP13 48 42 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309345 HB On-Demand Anodyne ADAM17 32 42 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309345 HB On-Demand Anodyne MMP3 35 40 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309345 HB On-Demand Anodyne MMP9 26 40 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309345 HB On-Demand Anodyne MMP7 40 40 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309345 HB On-Demand Anodyne MMP1 38 40 COC(=O)COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147309345 HB On-Demand Anodyne SFRP1 46 30 CC[C@H]1CN(C(=O)Cn2nnc(-c3ccccc3)n2)CCO1 ZINC000147309373 DC On-Demand Anodyne SCARB1 44 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(-c2ccccc2)cc1 ZINC000147309405 EF On-Demand Anodyne TNK2 51 39 Cc1cnccc1NC(=O)c1cccc2c1OCCN2 ZINC000147309424 CE For-Sale Anodyne G2YM83_BOTF4 58 33 CC[C@H](NC(=O)[C@@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309428 GG On-Demand Anodyne EDNRB 45 41 CC[C@H](NC(=O)[C@@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309428 GG On-Demand Anodyne EDNRA 37 41 CC[C@H](NC(=O)[C@@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309428 GG On-Demand Anodyne MTNR1A 15 40 CC[C@H](NC(=O)[C@@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309428 GG On-Demand Anodyne ROCK2 24 41 C[C@H](CNS(=O)(=O)c1ccccc1[N+](=O)[O-])CC(=O)O ZINC000147309444 DC On-Demand Bother COLA 101 45 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@@H](CCBr)C1 ZINC000147309476 FI For-Sale Reactive CACNA1B 55 35 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@@H](CCBr)C1 ZINC000147309476 FI For-Sale Reactive CCR2 73 44 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@@H](CCBr)C1 ZINC000147309476 FI For-Sale Reactive RHOA 0 47 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@@H](CCBr)C1 ZINC000147309476 FI For-Sale Reactive HPGD 17 41 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@@H](CCBr)C1 ZINC000147309476 FI For-Sale Reactive MAP3K12 31 43 CCCCCCCCCCNC1(C(=O)O)CCC1 ZINC000147309486 CH For-Sale Mild CES2 34 42 CCCCCCCCCCNC1(C(=O)O)CCC1 ZINC000147309486 CH For-Sale Mild EST1_PIG 50 35 CCCCCCCCCCNC1(C(=O)O)CCC1 ZINC000147309486 CH For-Sale Mild CES2C 40 42 CCCCCCCCNc1cc(C(N)=O)c(N)cc1F ZINC000147309498 CG For-Sale Mild ASAH1 60 34 Cc1ccc(C(=O)Nc2ccccc2CC(=O)O)cc1Br ZINC000147309511 EH On-Demand Anodyne CXCL8 28 44 Cc1ccc(C(=O)Nc2ccccc2CC(=O)O)cc1Br ZINC000147309511 EH On-Demand Anodyne NR1H4 23 43 Cc1ccc(C(=O)Nc2ccccc2CC(=O)O)cc1Br ZINC000147309511 EH On-Demand Anodyne CAPN2 42 33 Cc1ccc(C(=O)Nc2ccccc2CC(=O)O)cc1Br ZINC000147309511 EH On-Demand Anodyne FABH 0 44 Cc1ccc(C(=O)Nc2ccccc2CC(=O)O)cc1Br ZINC000147309511 EH On-Demand Anodyne KCNK3 59 37 Brc1nc(C2CCCCC2)n2c1cnc1[nH]ccc12 ZINC000147309531 DI For-Sale Anodyne JAK1 50 64 Brc1nc(C2CCCCC2)n2c1cnc1[nH]ccc12 ZINC000147309531 DI For-Sale Anodyne JAK2 15 62 COc1ccc2nc(N)n(CCNC(=O)N(C)C)c2n1 ZINC000147309556 CC For-Sale Anodyne PDE10A 32 41 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(C#N)cc2C(F)(F)F)C1 ZINC000147309574 HD On-Demand Mild SFRP1 134 47 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(C#N)cc2C(F)(F)F)C1 ZINC000147309574 HD On-Demand Mild WNT3 89 36 CC[C@@H](NC(=O)[C@@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309576 GG On-Demand Anodyne EDNRB 45 41 CC[C@@H](NC(=O)[C@@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309576 GG On-Demand Anodyne EDNRA 37 41 CC[C@@H](NC(=O)[C@@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309576 GG On-Demand Anodyne MTNR1A 15 40 CC[C@@H](NC(=O)[C@@H]1COc2cc(OC)ccc2C1)c1ccc2c(c1)OCCO2 ZINC000147309576 GG On-Demand Anodyne ROCK2 24 41 C[C@@H](CNS(=O)(=O)c1ccccc1[N+](=O)[O-])CC(=O)O ZINC000147309600 DC On-Demand Bother COLA 101 45 CN(C)NC(=O)CNc1ccccc1 ZINC000147309609 AC For-Sale Reactive KDM7A 0 42 CN(C)NC(=O)CNc1ccccc1 ZINC000147309609 AC For-Sale Reactive PSBA 0 44 CCCCCCCCNc1ccc(N)cc1C(=O)OCC ZINC000147309610 CI For-Sale Mild ACAT 0 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(-c2ccccc2)cc1 ZINC000147309629 EF On-Demand Anodyne TNK2 51 39 Cc1nc(C)c(C(=O)Nc2ccccc2CC(=O)O)o1 ZINC000147309696 CE On-Demand Anodyne LPL 41 30 Cc1nc(C)c(C(=O)Nc2ccccc2CC(=O)O)o1 ZINC000147309696 CE On-Demand Anodyne CXCL8 36 40 O=C(Cc1cncc(Cl)c1)c1ccc(Cl)cc1 ZINC000147309738 CH For-Sale Anodyne PLA2G7 20 41 O=C(Cc1cncc(Cl)c1)c1ccc(Cl)cc1 ZINC000147309738 CH For-Sale Anodyne SCN10A 48 39 Cc1ccc(C(=O)NCCNC(N)=O)cc1C#CCCO ZINC000147309739 CC For-Sale Mild DDR1 44 39 CC(=O)N1[C@H](C)SC(C)(C)[C@H]1C(=O)O ZINC000147309768 BD For-Sale Anodyne BLAB_BACCE 0 40 O=C(O)C1(NCc2nc3ccccc3c(=O)[nH]2)CCC1 ZINC000147309782 CD For-Sale Anodyne PARP1 25 45 O=C(O)C1(NCc2nc3ccccc3c(=O)[nH]2)CCC1 ZINC000147309782 CD For-Sale Anodyne PARP3 34 45 O=C(O)C1(NCc2nc3ccccc3c(=O)[nH]2)CCC1 ZINC000147309782 CD For-Sale Anodyne QTRT1 0 40 O=C(O)C1(NCc2nc3ccccc3c(=O)[nH]2)CCC1 ZINC000147309782 CD For-Sale Anodyne TNKS 17 41 CCCCCCCCNc1ccc(C(=O)OCC)cc1N ZINC000147309788 CI For-Sale Mild CNGA1 0 42 CCCCCCCCNc1ccc(C(=O)OCC)cc1N ZINC000147309788 CI For-Sale Mild ACAT 0 40 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc(C#N)cc2C(F)(F)F)C1 ZINC000147309790 HD On-Demand Mild SFRP1 134 47 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc(C#N)cc2C(F)(F)F)C1 ZINC000147309790 HD On-Demand Mild WNT3 89 36 CC[C@@H](N)C(=O)NN(C)C ZINC000147309838 AB For-Sale Reactive DPP7 0 41 CC[C@@H](N)C(=O)NN(C)C ZINC000147309838 AB For-Sale Reactive DPP8 0 41 CC[C@@H](N)C(=O)NN(C)C ZINC000147309838 AB For-Sale Reactive DPP9 0 41 CC(C)[C@H](NC(=O)N(C)Cc1cscn1)c1ccc2c(c1)OCCO2 ZINC000147309857 FG On-Demand Anodyne CYP3A4 17 41 O=C(O)Cc1ccccc1NC(=O)C1[C@H]2CCCC[C@H]12 ZINC000147309906 CF On-Demand Anodyne CXCL8 36 43 CC(C)CCCCN[C@@H]1CCOc2c(Cl)cc(Cl)cc21 ZINC000147309946 DK For-Sale Anodyne METG 28 52 CCCCCCCCNc1ccc(C(=O)O)cc1N ZINC000147309974 CH For-Sale Mild THRA 54 34 CCCCCCCCNc1ccc(C(=O)O)cc1N ZINC000147309974 CH For-Sale Mild RARB 21 43 CCCCCCCCNc1ccc(C(=O)O)cc1N ZINC000147309974 CH For-Sale Mild PLA2G4A 29 42 CCCCCCCCNc1ccc(C(=O)O)cc1N ZINC000147309974 CH For-Sale Mild PLA2G4B 69 42 CCCCCCCCNc1ccc(C(=O)O)cc1N ZINC000147309974 CH For-Sale Mild ASAH1 70 32 CCCCCCCCNc1ccc(C(=O)O)cc1N ZINC000147309974 CH For-Sale Mild NOD1 66 32 CC(C)[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc2c(c1)OCCO2 ZINC000147310093 FG On-Demand Anodyne CYP3A4 17 41 CNc1cc(Oc2ccc(Cl)cc2Br)nc(N)n1 ZINC000147310113 EG For-Sale Anodyne AGPAT2 76 42 CCOC(=O)c1cc2c(cn1)c(C(=O)c1ccc(F)cc1)cn2Cc1ccc(F)cc1 ZINC000147310116 HJ For-Sale Anodyne PTAFR 28 40 CCOC(=O)c1cc2c(cn1)c(C(=O)c1ccc(F)cc1)cn2Cc1ccc(F)cc1 ZINC000147310116 HJ For-Sale Anodyne F2RL3 18 42 CCOC(=O)c1cc2c(cn1)c(C(=O)c1ccc(F)cc1)cn2Cc1ccc(F)cc1 ZINC000147310116 HJ For-Sale Anodyne Q76353_9HIV1 0 41 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cc3c(cc2F)NC(=O)CC3)C1 ZINC000147310125 HC On-Demand Anodyne PKM 46 50 CC[C@@H]1CN(C(=O)C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)CCO1 ZINC000147310130 FE On-Demand Anodyne PSEN2 64 38 CC[C@@H]1CN(C(=O)C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)CCO1 ZINC000147310130 FE On-Demand Anodyne MMP13 29 43 CC[C@@H]1CN(C(=O)C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)CCO1 ZINC000147310130 FE On-Demand Anodyne APP 40 40 CC[C@@H]1CN(C(=O)C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)CCO1 ZINC000147310130 FE On-Demand Anodyne PSEN1 50 38 CC(C)CCCCN[C@H]1CCOc2c(Cl)cc(Cl)cc21 ZINC000147310136 DK For-Sale Anodyne METG 28 52 CCCCC1CCC(NC(=O)Nc2ccc(CC(=O)NCC(=O)OC)cc2)CC1 ZINC000147310197 HG On-Demand Anodyne EPHX2 48 41 CCCCCCCCNc1cccc(C(=O)OCC)c1N ZINC000147310216 CI For-Sale Mild ACAT 0 43 O=C(O)Cc1ccccc1NC(=O)C1[C@@H]2CCCC[C@@H]12 ZINC000147310311 CF On-Demand Anodyne CXCL8 36 43 CC[C@H]1CN(C(=O)C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)CCO1 ZINC000147310313 FE On-Demand Anodyne PSEN2 64 38 CC[C@H]1CN(C(=O)C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)CCO1 ZINC000147310313 FE On-Demand Anodyne MMP13 29 43 CC[C@H]1CN(C(=O)C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)CCO1 ZINC000147310313 FE On-Demand Anodyne APP 40 40 CC[C@H]1CN(C(=O)C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)CCO1 ZINC000147310313 FE On-Demand Anodyne PSEN1 50 38 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2cc3c(cc2F)NC(=O)CC3)C1 ZINC000147310358 HC On-Demand Anodyne PKM 46 50 Cc1cc(CNC(=O)Nc2ccc(CC(=O)N3CCOCC3)cc2)no1 ZINC000147310420 FD On-Demand Anodyne MTOR 75 39 Cc1cc(CNC(=O)Nc2ccc(CC(=O)N3CCOCC3)cc2)no1 ZINC000147310420 FD On-Demand Anodyne EPHX2 37 41 Cc1cc(CNC(=O)Nc2ccc(CC(=O)N3CCOCC3)cc2)no1 ZINC000147310420 FD On-Demand Anodyne NAMPT 46 49 CCCCCCCCNc1ccc(C(=O)OC)cc1N ZINC000147310427 CH For-Sale Mild THRA 43 33 CN(C)C(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147310570 GC On-Demand Anodyne AKR1C3 38 45 CN(C)C(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147310570 GC On-Demand Anodyne SFRP1 85 38 CN(C)C(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147310570 GC On-Demand Anodyne WNT3 60 35 CCCCCCCCNc1ccc(N)c(C(=O)OC)c1 ZINC000147310652 CH For-Sale Mild ASAH1 47 32 O=C(CNC1(C(=O)O)CCC1)N1CCCc2ccccc21 ZINC000147310653 CD For-Sale Anodyne AVPR2 47 46 O=C(CNC1(C(=O)O)CCC1)N1CCCc2ccccc21 ZINC000147310653 CD For-Sale Anodyne AVPR1A 15 42 CC(=O)c1cccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)c1 ZINC000147310753 CD On-Demand Anodyne CASP3 22 42 CC(=O)c1cccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)c1 ZINC000147310753 CD On-Demand Anodyne AKR1C3 22 45 O=C(N[C@@H]1CCCC[C@@H]1C(=O)O)c1cccc(F)c1Cl ZINC000147310762 CF For-Sale Anodyne SSTR3 31 40 CN(C)C(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147310785 GC On-Demand Anodyne AKR1C3 38 45 CN(C)C(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147310785 GC On-Demand Anodyne SFRP1 85 38 CN(C)C(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147310785 GC On-Demand Anodyne WNT3 60 35 CCc1ncc(C(=O)N2CCC[C@@H]2c2cccs2)s1 ZINC000147310829 CH On-Demand Anodyne CPT1A 52 38 CCc1ncc(C(=O)N2CCC[C@@H]2c2cccs2)s1 ZINC000147310829 CH On-Demand Anodyne PREP 72 38 NS(=O)(=O)c1ccc(OCCc2ccncc2)c(F)c1F ZINC000147310847 DD For-Sale Anodyne CA14 0 43 CCCCCCCCNc1cccc(C(=O)O)c1N ZINC000147310880 CH For-Sale Mild ASAH1 63 33 CCCCCCCCNc1cccc(C(=O)O)c1N ZINC000147310880 CH For-Sale Mild AKR1C2 63 38 CC(=O)CCC(=O)NCc1ccc(O)c(O)c1 ZINC000147310883 BD On-Demand Clean TRPV1 20 49 CC(=O)CCC(=O)NCc1ccc(O)c(O)c1 ZINC000147310883 BD On-Demand Clean NCE103 25 42 CC(=O)CCC(=O)NCc1ccc(O)c(O)c1 ZINC000147310883 BD On-Demand Clean P96878_MYCTU 16 42 COc1cccc(Oc2cc(NN)nc(C(C)C)n2)c1 ZINC000147310923 CF For-Sale Anodyne MTNR1B 15 40 CS(=O)(=O)c1cc(C(=O)Nc2ccc(Oc3ccccc3)nc2)cc([N+](=O)[O-])c1 ZINC000147310975 HG On-Demand Bother GCK 36 42 O=C(N[C@H]1CCCC[C@@H]1C(=O)O)c1cccc(F)c1Cl ZINC000147310980 CF For-Sale Anodyne SSTR3 31 40 CC(=O)c1cccc(S(=O)(=O)NC[C@H](C)CC(=O)O)c1 ZINC000147310982 CD On-Demand Anodyne CASP3 22 42 CC(=O)c1cccc(S(=O)(=O)NC[C@H](C)CC(=O)O)c1 ZINC000147310982 CD On-Demand Anodyne AKR1C3 22 45 Cc1nc(C)c(-c2cc[nH]c(=O)n2)s1 ZINC000147310999 BD For-Sale Anodyne CDK4 18 43 O=C(O)c1ccc(CNCC(F)F)o1 ZINC000147311002 BD For-Sale Anodyne MAP 0 41 CCc1ncc(C(=O)N2CCC[C@H]2c2cccs2)s1 ZINC000147311033 CH On-Demand Anodyne CPT1A 52 38 CCc1ncc(C(=O)N2CCC[C@H]2c2cccs2)s1 ZINC000147311033 CH On-Demand Anodyne PREP 72 38 O=C(C[C@@H]1CNc2ccccc21)N(CCO)C1CC1 ZINC000147311036 CD For-Sale Anodyne MBTPS1 49 30 CCCCCCCCNc1cc(N)ccc1C(=O)O ZINC000147311073 CH For-Sale Mild RARB 17 40 CCCCCCCCNc1cc(N)ccc1C(=O)O ZINC000147311073 CH For-Sale Mild ASAH1 63 32 CCCCCCCCNc1cc(N)ccc1C(=O)O ZINC000147311073 CH For-Sale Mild AKR1C2 49 35 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000147311088 HD On-Demand Anodyne LPL 46 38 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000147311088 HD On-Demand Anodyne EPHX2 28 45 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000147311088 HD On-Demand Anodyne TGM2 37 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000147311088 HD On-Demand Anodyne F13A1 47 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000147311088 HD On-Demand Anodyne AKR1C3 57 44 O=C(Nc1ccc(CC(=O)N2CCOCC2)cc1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147311101 GF On-Demand Anodyne EPHX2 65 50 O=C(Nc1ccc(CC(=O)N2CCOCC2)cc1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147311101 GF On-Demand Anodyne KDM1A 49 33 O=C(N[C@@H]1CCCC[C@H]1C(=O)O)c1cccc(F)c1Cl ZINC000147311169 CF For-Sale Anodyne SSTR3 31 40 O=C(C[C@H]1CNc2ccccc21)N(CCO)C1CC1 ZINC000147311250 CD For-Sale Anodyne MBTPS1 49 30 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000147311291 HD On-Demand Anodyne LPL 46 38 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000147311291 HD On-Demand Anodyne EPHX2 28 45 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000147311291 HD On-Demand Anodyne TGM2 37 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000147311291 HD On-Demand Anodyne F13A1 47 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(S(=O)(=O)N2CCCCC2)c1 ZINC000147311291 HD On-Demand Anodyne AKR1C3 57 44 O=C(Nc1ccc(CC(=O)N2CCOCC2)cc1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147311304 GF On-Demand Anodyne EPHX2 65 50 O=C(Nc1ccc(CC(=O)N2CCOCC2)cc1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147311304 GF On-Demand Anodyne KDM1A 49 33 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311309 ED On-Demand Anodyne CYP11B1 42 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311309 ED On-Demand Anodyne TBXAS1 41 38 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311309 ED On-Demand Anodyne AGTR2 15 45 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311309 ED On-Demand Anodyne NPY1R 22 40 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311309 ED On-Demand Anodyne F2R 40 33 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311309 ED On-Demand Anodyne CYP11B2 38 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311309 ED On-Demand Anodyne PCSK5 47 39 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311309 ED On-Demand Anodyne FURIN 63 39 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311309 ED On-Demand Anodyne CYP17A1 22 42 CCCCCCCCNc1ncc(C(=O)O)cc1N ZINC000147311310 CG For-Sale Mild PLA2G4B 42 35 CCCCCCCCNc1ncc(C(=O)O)cc1N ZINC000147311310 CG For-Sale Mild NOD1 40 31 COc1ccc2nc(N)n(CCNC(=O)N(C)C)c2c1 ZINC000147311332 CC For-Sale Anodyne DRD4 41 31 COc1ccc2nc(N)n(CCNC(=O)N(C)C)c2c1 ZINC000147311332 CC For-Sale Anodyne MTNR1A 50 37 COc1ccc2nc(N)n(CCNC(=O)N(C)C)c2c1 ZINC000147311332 CC For-Sale Anodyne MTNR1B 40 37 COc1ccc2nc(N)n(CCNC(=O)N(C)C)c2c1 ZINC000147311332 CC For-Sale Anodyne SCD 17 40 COc1ccc2nc(N)n(CCNC(=O)N(C)C)c2c1 ZINC000147311332 CC For-Sale Anodyne PROKR1 43 30 O=C(N[C@H]1CCCC[C@H]1C(=O)O)c1cccc(F)c1Cl ZINC000147311362 CF On-Demand Anodyne SSTR3 30 40 CCCNc1ncnc(Oc2ccc(Cl)cc2Br)c1C ZINC000147311363 FJ For-Sale Anodyne HTT 0 42 O=C(Nc1ccc(CC(=O)N2CCOCC2)cc1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147311470 GF On-Demand Anodyne EPHX2 65 50 O=C(Nc1ccc(CC(=O)N2CCOCC2)cc1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147311470 GF On-Demand Anodyne KDM1A 49 33 CCCCCCCCNc1cc(C(=O)O)c(N)cc1F ZINC000147311505 CH For-Sale Mild ASAH1 75 35 CCCCCCCCNc1cc(C(=O)O)c(N)cc1F ZINC000147311505 CH For-Sale Mild NOD1 49 31 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311539 ED On-Demand Anodyne CYP11B1 42 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311539 ED On-Demand Anodyne TBXAS1 41 38 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311539 ED On-Demand Anodyne AGTR2 15 45 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311539 ED On-Demand Anodyne NPY1R 22 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311539 ED On-Demand Anodyne F2R 40 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311539 ED On-Demand Anodyne CYP11B2 38 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311539 ED On-Demand Anodyne PCSK5 47 39 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311539 ED On-Demand Anodyne FURIN 63 39 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(Cn2ccnc2)cc1 ZINC000147311539 ED On-Demand Anodyne CYP17A1 22 42 O=C(NCC1CCOCC1)c1cccc2c1OCCN2 ZINC000147311541 CD For-Sale Anodyne HTR4 28 41 Cc1ccc(Nc2ccccc2C(=O)N2CCC(c3nnc4n3CCC4)CC2)cc1 ZINC000147311545 HI On-Demand Anodyne L3MBTL3 20 40 Cc1ccc(Nc2ccccc2C(=O)N2CCC(c3nnc4n3CCC4)CC2)cc1 ZINC000147311545 HI On-Demand Anodyne TRPC6 26 40 Cc1ccc(Nc2ccccc2C(=O)N2CCC(c3nnc4n3CCC4)CC2)cc1 ZINC000147311545 HI On-Demand Anodyne TRPC3 29 40 O=C(CNC1(C(=O)O)CCC1)Nc1cccc(F)c1 ZINC000147311580 CD For-Sale Anodyne KCNK3 33 42 Nc1ncc(Cl)c(Oc2ccc(Cl)cc2Br)n1 ZINC000147311584 EH For-Sale Anodyne P2RX2 38 40 Nc1ncc(Cl)c(Oc2ccc(Cl)cc2Br)n1 ZINC000147311584 EH For-Sale Anodyne P2RX3 23 40 Nc1ncc(Cl)c(Oc2ccc(Cl)cc2Br)n1 ZINC000147311584 EH For-Sale Anodyne S1PR4 0 41 Nc1ncc(Cl)c(Oc2ccc(Cl)cc2Br)n1 ZINC000147311584 EH For-Sale Anodyne AGPAT2 41 36 c1ccc2c(CO[C@H]3CNCC[C@@H]3c3ccoc3)cccc2c1 ZINC000147311604 DI For-Sale Anodyne REN 19 47 O=C(Nc1ccc(CC(=O)N2CCOCC2)cc1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147311652 GF On-Demand Anodyne EPHX2 65 50 O=C(Nc1ccc(CC(=O)N2CCOCC2)cc1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147311652 GF On-Demand Anodyne KDM1A 49 33 CCCCCCCCNc1nccc(C(=O)OCC)c1N ZINC000147311725 CH For-Sale Mild UTS2R 18 47 C#CCNC(=O)CCNCc1c(C)nn(-c2ccccc2)c1C ZINC000147311820 DD On-Demand Mild P2RX7 36 56 CCCCCCNC(=O)C[C@@H]1CNc2ccccc21 ZINC000147311827 CG For-Sale Anodyne ASAH1 87 38 CC(C)(C)c1ccc(CO[C@H]2CNCC[C@@H]2c2ccoc2)cc1 ZINC000147311832 DI For-Sale Anodyne REN 19 44 O=C1CC[C@@H](C(=O)Nc2ccc(O)c(F)c2)CN1 ZINC000147311859 CC For-Sale Anodyne MAPK1 29 43 CCO[C@@H]1CCCN(C(=O)Nc2ccc(CC(=O)N3CCOCC3)cc2)C1 ZINC000147311895 GE On-Demand Anodyne TIMP3 55 32 CCO[C@@H]1CCCN(C(=O)Nc2ccc(CC(=O)N3CCOCC3)cc2)C1 ZINC000147311895 GE On-Demand Anodyne MLNR 24 40 CCO[C@@H]1CCCN(C(=O)Nc2ccc(CC(=O)N3CCOCC3)cc2)C1 ZINC000147311895 GE On-Demand Anodyne EPHX2 36 46 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147311934 GD On-Demand Anodyne LPL 45 35 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147311934 GD On-Demand Anodyne EPHX2 24 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147311934 GD On-Demand Anodyne TGM2 79 45 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147311934 GD On-Demand Anodyne F13A1 98 47 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147311934 GD On-Demand Anodyne NAMPT 50 47 CN(C)NC(=O)c1ccccc1CCN ZINC000147311947 BC For-Sale Reactive ECR 42 38 CN(C)NC(=O)c1ccccc1CCN ZINC000147311947 BC For-Sale Reactive TAAR1 15 46 CCCCCCCCn1c(CCl)nc2ccccc2c1=O ZINC000147311950 DI For-Sale Reactive CNR1 22 42 CCCCCCCCn1c(CCl)nc2ccccc2c1=O ZINC000147311950 DI For-Sale Reactive AGTR1 55 49 CCCCCCCCn1c(CCl)nc2ccccc2c1=O ZINC000147311950 DI For-Sale Reactive CNR2 26 42 CCCCCCCCn1c(CCl)nc2ccccc2c1=O ZINC000147311950 DI For-Sale Reactive AGTR1B 40 37 CCCCCCCCn1c(CCl)nc2ccccc2c1=O ZINC000147311950 DI For-Sale Reactive TLR7 38 41 CCCCCCCCn1c(CCl)nc2ccccc2c1=O ZINC000147311950 DI For-Sale Reactive RORB 0 43 CN(C)C(=O)NCCn1c(N)nc2ccccc21 ZINC000147312003 BC For-Sale Anodyne CDPK1 0 40 COc1cccc(CNC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147312007 CC For-Sale Anodyne ROCK1 36 43 COc1cccc(CNC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147312007 CC For-Sale Anodyne MTNR1A 68 43 COc1cccc(CNC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147312007 CC For-Sale Anodyne MTNR1B 64 43 COc1cccc(CNC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147312007 CC For-Sale Anodyne ROCK2 40 47 COc1cccc(CNC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147312007 CC For-Sale Anodyne NPFFR1 15 42 COc1cccc(CNC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147312007 CC For-Sale Anodyne PDS 43 40 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(Cl)c(C#N)c2)C1 ZINC000147312017 GC On-Demand Mild CTSC 15 40 CCCCCCNC(=O)C[C@H]1CNc2ccccc21 ZINC000147312031 CG For-Sale Anodyne ASAH1 87 38 O=C1CC[C@H](C(=O)Nc2ccc(O)c(F)c2)CN1 ZINC000147312070 CC For-Sale Anodyne MAPK1 29 43 Brc1ccc(CO[C@H]2CNCC[C@@H]2c2ccoc2)cc1 ZINC000147312073 EH For-Sale Anodyne REN 24 59 CCO[C@H]1CCCN(C(=O)Nc2ccc(CC(=O)N3CCOCC3)cc2)C1 ZINC000147312102 GE On-Demand Anodyne TIMP3 55 32 CCO[C@H]1CCCN(C(=O)Nc2ccc(CC(=O)N3CCOCC3)cc2)C1 ZINC000147312102 GE On-Demand Anodyne MLNR 24 40 CCO[C@H]1CCCN(C(=O)Nc2ccc(CC(=O)N3CCOCC3)cc2)C1 ZINC000147312102 GE On-Demand Anodyne EPHX2 36 46 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147312119 GD On-Demand Anodyne LPL 45 35 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147312119 GD On-Demand Anodyne EPHX2 24 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147312119 GD On-Demand Anodyne TGM2 79 45 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147312119 GD On-Demand Anodyne F13A1 98 47 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCC2)cc1 ZINC000147312119 GD On-Demand Anodyne NAMPT 50 47 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild FOLH1 17 41 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild CA1 21 47 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild SCN2A 18 40 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild FAAH 20 40 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild S1PR2 42 35 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild EPHX2 32 60 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild CA9 15 47 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild PPO2 15 42 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild ASAH1 98 39 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild P96878_MYCTU 17 47 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild ACAT 0 55 CCCCCCCCNC(=O)Nc1ccc(C(C)=O)cc1 ZINC000147312127 CI For-Sale Mild PSBA 0 42 CNC(=O)c1cccc(NC(=O)c2csc(COC)n2)c1 ZINC000147312203 DD On-Demand Anodyne TAAR1 26 40 CNC(=O)c1cccc(NC(=O)c2csc(COC)n2)c1 ZINC000147312203 DD On-Demand Anodyne KCNK3 85 40 CNC(=O)c1cccc(NC(=O)c2csc(COC)n2)c1 ZINC000147312203 DD On-Demand Anodyne KCNK9 69 38 O=C(O)[C@H]1CCCC[C@H]1NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147312230 CF For-Sale Anodyne EPHX2 21 42 O=C(O)[C@H]1CCCC[C@H]1NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147312230 CF For-Sale Anodyne GPR88 0 42 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc(Cl)c(C#N)c2)C1 ZINC000147312246 GC On-Demand Mild CTSC 15 40 O=C(NCc1cccc(NC(=O)[C@@H]2CCCO2)c1)Nc1cccnc1N1CCCC1 ZINC000147312311 HG On-Demand Anodyne TRPV1 22 41 Cc1cccc(CO[C@H]2CNCC[C@@H]2c2ccoc2)c1 ZINC000147312314 CG For-Sale Anodyne REN 26 48 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312317 HD On-Demand Anodyne LPL 40 37 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312317 HD On-Demand Anodyne EPHX2 24 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312317 HD On-Demand Anodyne TGM2 78 44 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312317 HD On-Demand Anodyne F13A1 87 46 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312317 HD On-Demand Anodyne MERTK 26 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312317 HD On-Demand Anodyne NAMPT 49 48 Cc1cc(-c2ccncc2NC(=O)c2nc(-c3ccccc3F)ccc2N)nc(N)n1 ZINC000147312332 HG Annotated Anodyne PIM1 36 55 Cc1cc(-c2ccncc2NC(=O)c2nc(-c3ccccc3F)ccc2N)nc(N)n1 ZINC000147312332 HG Annotated Anodyne PIM2 18 55 Cc1cc(-c2ccncc2NC(=O)c2nc(-c3ccccc3F)ccc2N)nc(N)n1 ZINC000147312332 HG Annotated Anodyne PIM3 24 55 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild INHA 25 40 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild CA1 15 41 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild CCR3 43 51 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild GUAB 0 48 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild SOAT1 22 41 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild FAAH 16 42 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild EPHX2 34 64 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild PA2A1_NAJMO 0 42 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild AKR1C3 23 47 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild ASAH1 91 37 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild ACAT 0 58 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild IMDH_CRYPV 46 35 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild PARP15 0 40 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild PSBA 0 46 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild KCNK3 93 37 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild KCNK9 55 37 CCCCCCCCNC(=O)Nc1cccc(C(C)=O)c1 ZINC000147312337 CI For-Sale Mild PARP10 0 42 Cc1ccc(C(=O)N[C@@H]2CCCC[C@@H]2C(=O)O)cc1Br ZINC000147312475 EG On-Demand Anodyne MAPK14 40 39 Cc1ccc(C(=O)N[C@@H]2CCCC[C@@H]2C(=O)O)cc1Br ZINC000147312475 EG On-Demand Anodyne ADAM17 17 40 Cc1ccc(C(=O)N[C@@H]2CCCC[C@@H]2C(=O)O)cc1Br ZINC000147312475 EG On-Demand Anodyne MAPK13 40 36 O=C(NCc1cccc(NC(=O)[C@H]2CCCO2)c1)Nc1cccnc1N1CCCC1 ZINC000147312486 HG On-Demand Anodyne TRPV1 22 41 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)O)cc1 ZINC000147312488 CI For-Sale Mild SOAT1 31 42 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)O)cc1 ZINC000147312488 CI For-Sale Mild EPHX2 26 58 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)O)cc1 ZINC000147312488 CI For-Sale Mild ENPP2 32 47 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)O)cc1 ZINC000147312488 CI For-Sale Mild ASAH1 104 40 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)O)cc1 ZINC000147312488 CI For-Sale Mild P96878_MYCTU 16 41 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)O)cc1 ZINC000147312488 CI For-Sale Mild ACAT 0 52 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)O)cc1 ZINC000147312488 CI For-Sale Mild CQSS 41 33 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)O)cc1 ZINC000147312488 CI For-Sale Mild PSBA 0 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312495 HD On-Demand Anodyne LPL 40 37 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312495 HD On-Demand Anodyne EPHX2 24 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312495 HD On-Demand Anodyne TGM2 78 44 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312495 HD On-Demand Anodyne F13A1 87 46 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312495 HD On-Demand Anodyne MERTK 26 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147312495 HD On-Demand Anodyne NAMPT 49 48 C[C@H](CNS(=O)(=O)c1ccc(Cl)cc1F)CC(=O)O ZINC000147312535 DD On-Demand Anodyne OXER1 42 36 Oc1ccc2cc(-c3ccc(-c4ccccc4)[nH]3)ccc2c1 ZINC000147312548 CK For-Sale Anodyne ESR1 24 58 Oc1ccc2cc(-c3ccc(-c4ccccc4)[nH]3)ccc2c1 ZINC000147312548 CK For-Sale Anodyne ESR2 31 49 Oc1ccc2cc(-c3ccc(-c4ccccc4)[nH]3)ccc2c1 ZINC000147312548 CK For-Sale Anodyne HSD17B1 31 58 Oc1ccc2cc(-c3ccc(-c4ccccc4)[nH]3)ccc2c1 ZINC000147312548 CK For-Sale Anodyne HSD17B2 15 41 Cc1ccc(C(=O)N[C@H]2CCCC[C@@H]2C(=O)O)cc1Br ZINC000147312597 EG For-Sale Anodyne MAPK14 41 39 Cc1ccc(C(=O)N[C@H]2CCCC[C@@H]2C(=O)O)cc1Br ZINC000147312597 EG For-Sale Anodyne ADAM17 20 42 Cc1ccc(C(=O)N[C@H]2CCCC[C@@H]2C(=O)O)cc1Br ZINC000147312597 EG For-Sale Anodyne MAPK13 40 36 CCCCCCCCNC(=O)Nc1ccc([C@H](C)O)cc1 ZINC000147312629 CI For-Sale Mild SOAT1 31 42 CCCCCCCCNC(=O)Nc1ccc([C@H](C)O)cc1 ZINC000147312629 CI For-Sale Mild EPHX2 26 58 CCCCCCCCNC(=O)Nc1ccc([C@H](C)O)cc1 ZINC000147312629 CI For-Sale Mild ENPP2 32 47 CCCCCCCCNC(=O)Nc1ccc([C@H](C)O)cc1 ZINC000147312629 CI For-Sale Mild ASAH1 104 40 CCCCCCCCNC(=O)Nc1ccc([C@H](C)O)cc1 ZINC000147312629 CI For-Sale Mild P96878_MYCTU 16 41 CCCCCCCCNC(=O)Nc1ccc([C@H](C)O)cc1 ZINC000147312629 CI For-Sale Mild ACAT 0 52 CCCCCCCCNC(=O)Nc1ccc([C@H](C)O)cc1 ZINC000147312629 CI For-Sale Mild CQSS 41 33 CCCCCCCCNC(=O)Nc1ccc([C@H](C)O)cc1 ZINC000147312629 CI For-Sale Mild PSBA 0 40 C[C@@H](CCC[C@@H](C)N)C(=O)NN(C)C ZINC000147312634 BC For-Sale Reactive NOD1 50 32 C[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1F)CC(=O)O ZINC000147312676 DD On-Demand Anodyne OXER1 42 36 COc1ccc(NC(=O)c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)cc1 ZINC000147312696 HF On-Demand Anodyne F10 15 41 COc1ccc(NC(=O)c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)cc1 ZINC000147312696 HF On-Demand Anodyne PRNP 44 32 COc1ccc(NC(=O)c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)cc1 ZINC000147312696 HF On-Demand Anodyne NOD1 15 41 COc1ccc(NC(=O)c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2)cc1 ZINC000147312696 HF On-Demand Anodyne NOD2 32 41 C[C@@H](N)CCC[C@@H](C)C(=O)NN(C)C ZINC000147312782 BC For-Sale Reactive NOD1 50 32 Cc1ccc(C(=O)N[C@@H]2CCCC[C@H]2C(=O)O)cc1Br ZINC000147312809 EG For-Sale Anodyne MAPK14 41 39 Cc1ccc(C(=O)N[C@@H]2CCCC[C@H]2C(=O)O)cc1Br ZINC000147312809 EG For-Sale Anodyne ADAM17 20 42 Cc1ccc(C(=O)N[C@@H]2CCCC[C@H]2C(=O)O)cc1Br ZINC000147312809 EG For-Sale Anodyne MAPK13 40 36 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)O)c1 ZINC000147312816 CI For-Sale Mild SOAT1 60 49 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)O)c1 ZINC000147312816 CI For-Sale Mild EPHX2 25 64 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)O)c1 ZINC000147312816 CI For-Sale Mild PA2A1_NAJMO 0 40 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)O)c1 ZINC000147312816 CI For-Sale Mild ASAH1 98 40 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)O)c1 ZINC000147312816 CI For-Sale Mild ACAT 0 54 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)O)c1 ZINC000147312816 CI For-Sale Mild PSBA 0 43 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)O)c1 ZINC000147312816 CI For-Sale Mild ACER2 0 40 CC[C@@H]1CN(C(=O)c2cccc3ncccc23)CC[C@@H]1N ZINC000147312825 CE On-Demand Anodyne FAP 0 43 C[C@H](CNS(=O)(=O)c1ccccc1Cl)CC(=O)O ZINC000147312891 CD On-Demand Anodyne CXCL8 42 34 C[C@H](CNS(=O)(=O)c1ccccc1Cl)CC(=O)O ZINC000147312891 CD On-Demand Anodyne ITGAV 38 47 COc1ccc(NC(=O)c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)cc1 ZINC000147312911 HF On-Demand Anodyne F10 15 41 COc1ccc(NC(=O)c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)cc1 ZINC000147312911 HF On-Demand Anodyne PRNP 44 32 COc1ccc(NC(=O)c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)cc1 ZINC000147312911 HF On-Demand Anodyne NOD1 15 41 COc1ccc(NC(=O)c2ccc(NC(=O)C(=O)NC[C@H]3CCCCO3)cc2)cc1 ZINC000147312911 HF On-Demand Anodyne NOD2 32 41 Cc1ccc2c(CNC3(C(=O)O)CCC3)cc(=O)oc2c1 ZINC000147312913 CE For-Sale Anodyne HSD17B3 21 40 Cc1ccc(C(=O)N[C@H]2CCCC[C@H]2C(=O)O)cc1Br ZINC000147312928 EG For-Sale Anodyne MAPK14 41 39 Cc1ccc(C(=O)N[C@H]2CCCC[C@H]2C(=O)O)cc1Br ZINC000147312928 EG For-Sale Anodyne ADAM17 20 42 Cc1ccc(C(=O)N[C@H]2CCCC[C@H]2C(=O)O)cc1Br ZINC000147312928 EG For-Sale Anodyne MAPK13 40 36 C[C@H](N)CCC[C@H](C)C(=O)NN(C)C ZINC000147312944 BC For-Sale Reactive NOD1 50 32 CCCCCCCCNC(=O)Nc1cccc([C@H](C)O)c1 ZINC000147312950 CI For-Sale Mild SOAT1 60 49 CCCCCCCCNC(=O)Nc1cccc([C@H](C)O)c1 ZINC000147312950 CI For-Sale Mild EPHX2 25 64 CCCCCCCCNC(=O)Nc1cccc([C@H](C)O)c1 ZINC000147312950 CI For-Sale Mild PA2A1_NAJMO 0 40 CCCCCCCCNC(=O)Nc1cccc([C@H](C)O)c1 ZINC000147312950 CI For-Sale Mild ASAH1 98 40 CCCCCCCCNC(=O)Nc1cccc([C@H](C)O)c1 ZINC000147312950 CI For-Sale Mild ACAT 0 54 CCCCCCCCNC(=O)Nc1cccc([C@H](C)O)c1 ZINC000147312950 CI For-Sale Mild PSBA 0 43 CCCCCCCCNC(=O)Nc1cccc([C@H](C)O)c1 ZINC000147312950 CI For-Sale Mild ACER2 0 40 CC[C@H]1CN(C(=O)c2cccc3ncccc23)CC[C@@H]1N ZINC000147312972 CE On-Demand Anodyne FAP 0 43 C[C@@H](CNS(=O)(=O)c1ccccc1Cl)CC(=O)O ZINC000147313037 CD On-Demand Anodyne CXCL8 42 34 C[C@@H](CNS(=O)(=O)c1ccccc1Cl)CC(=O)O ZINC000147313037 CD On-Demand Anodyne ITGAV 38 47 C[C@H](N)CCC[C@@H](C)C(=O)NN(C)C ZINC000147313064 BC For-Sale Reactive NOD1 50 32 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)N)c1 ZINC000147313068 CI For-Sale Mild SOAT1 55 47 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)N)c1 ZINC000147313068 CI For-Sale Mild EPHX2 23 60 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)N)c1 ZINC000147313068 CI For-Sale Mild S1PR5 16 41 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)N)c1 ZINC000147313068 CI For-Sale Mild ASAH1 84 36 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)N)c1 ZINC000147313068 CI For-Sale Mild ACAT 0 53 CCCCCCCCNC(=O)Nc1cccc([C@@H](C)N)c1 ZINC000147313068 CI For-Sale Mild PSBA 0 43 Nc1cc(Cl)cc(-c2nc3cc(Cl)ccc3o2)c1 ZINC000147313070 CI For-Sale Anodyne AGPAT2 25 40 CC[C@@H]1CN(C(=O)c2cccc3ncccc23)CC[C@H]1N ZINC000147313071 CE On-Demand Anodyne FAP 0 43 Cc1ccc(C(=O)NCCNC(N)=O)cc1C#CCO ZINC000147313139 CB For-Sale Mild KIT 0 41 Cc1ccc(C(=O)NCCNC(N)=O)cc1C#CCO ZINC000147313139 CB For-Sale Mild DDR1 53 41 CC[C@H]1CN(C(=O)c2cccc3ncccc23)CC[C@H]1N ZINC000147313194 CE On-Demand Anodyne FAP 0 43 CCCCCCCCNC(=O)Nc1cccc([C@H](C)N)c1 ZINC000147313206 CI For-Sale Mild SOAT1 55 47 CCCCCCCCNC(=O)Nc1cccc([C@H](C)N)c1 ZINC000147313206 CI For-Sale Mild EPHX2 23 60 CCCCCCCCNC(=O)Nc1cccc([C@H](C)N)c1 ZINC000147313206 CI For-Sale Mild S1PR5 16 41 CCCCCCCCNC(=O)Nc1cccc([C@H](C)N)c1 ZINC000147313206 CI For-Sale Mild ASAH1 84 36 CCCCCCCCNC(=O)Nc1cccc([C@H](C)N)c1 ZINC000147313206 CI For-Sale Mild ACAT 0 53 CCCCCCCCNC(=O)Nc1cccc([C@H](C)N)c1 ZINC000147313206 CI For-Sale Mild PSBA 0 43 CC(C)C[C@@H](CN)CC(=O)NN(C)C ZINC000147313252 BC For-Sale Reactive CACNA2D1 0 56 Cc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1C ZINC000147313271 CD On-Demand Anodyne LEF 59 37 CCNc1cn2ccnc2c(Oc2ccc(Cl)cc2Br)n1 ZINC000147313291 FI For-Sale Anodyne HIVRT 0 49 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)N)cc1 ZINC000147313341 CI For-Sale Mild CA1 35 40 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)N)cc1 ZINC000147313341 CI For-Sale Mild SOAT1 30 41 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)N)cc1 ZINC000147313341 CI For-Sale Mild EPHX2 23 57 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)N)cc1 ZINC000147313341 CI For-Sale Mild CA12 19 40 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)N)cc1 ZINC000147313341 CI For-Sale Mild CA9 19 40 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)N)cc1 ZINC000147313341 CI For-Sale Mild ENPP2 30 43 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)N)cc1 ZINC000147313341 CI For-Sale Mild ASAH1 95 37 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)N)cc1 ZINC000147313341 CI For-Sale Mild P96878_MYCTU 20 43 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)N)cc1 ZINC000147313341 CI For-Sale Mild ACAT 0 51 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)N)cc1 ZINC000147313341 CI For-Sale Mild DOT1L 40 31 CCCCCCCCNC(=O)Nc1ccc([C@@H](C)N)cc1 ZINC000147313341 CI For-Sale Mild PSBA 0 40 CCN(CC)C(=O)[C@@]1(c2ccccc2)C[C@H]1CBr ZINC000147313381 DG For-Sale Reactive SLC6A2 19 75 Cc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1C ZINC000147313417 CD On-Demand Anodyne LEF 59 37 Cc1ccc2nc(-c3cc(N)cc(Cl)c3)oc2c1 ZINC000147313465 CI For-Sale Anodyne AGPAT2 15 42 CCCCCCCCNC(=O)Nc1ccc([C@H](C)N)cc1 ZINC000147313502 CI For-Sale Mild CA1 35 40 CCCCCCCCNC(=O)Nc1ccc([C@H](C)N)cc1 ZINC000147313502 CI For-Sale Mild SOAT1 30 41 CCCCCCCCNC(=O)Nc1ccc([C@H](C)N)cc1 ZINC000147313502 CI For-Sale Mild EPHX2 23 57 CCCCCCCCNC(=O)Nc1ccc([C@H](C)N)cc1 ZINC000147313502 CI For-Sale Mild CA12 19 40 CCCCCCCCNC(=O)Nc1ccc([C@H](C)N)cc1 ZINC000147313502 CI For-Sale Mild CA9 19 40 CCCCCCCCNC(=O)Nc1ccc([C@H](C)N)cc1 ZINC000147313502 CI For-Sale Mild ENPP2 30 43 CCCCCCCCNC(=O)Nc1ccc([C@H](C)N)cc1 ZINC000147313502 CI For-Sale Mild ASAH1 95 37 CCCCCCCCNC(=O)Nc1ccc([C@H](C)N)cc1 ZINC000147313502 CI For-Sale Mild P96878_MYCTU 20 43 CCCCCCCCNC(=O)Nc1ccc([C@H](C)N)cc1 ZINC000147313502 CI For-Sale Mild ACAT 0 51 CCCCCCCCNC(=O)Nc1ccc([C@H](C)N)cc1 ZINC000147313502 CI For-Sale Mild DOT1L 40 31 CCCCCCCCNC(=O)Nc1ccc([C@H](C)N)cc1 ZINC000147313502 CI For-Sale Mild PSBA 0 40 CSSc1ccc(C(=O)O)cn1 ZINC000147313503 BE For-Sale Reactive P4HTM 0 52 CSSc1ccc(C(=O)O)cn1 ZINC000147313503 BE For-Sale Reactive P4HA1 0 50 COc1nc(N)nc(Oc2ccccc2NC(C)=O)n1 ZINC000147313580 CD For-Sale Anodyne ALS 46 38 Cc1ccc(S(=O)(=O)n2ccc3c(N[C@@H]4CCN(C(=O)OC(C)(C)C)C4)ncnc32)cc1 ZINC000147313639 JG For-Sale Anodyne GPR119 58 55 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1cccnc1N1CCCC1 ZINC000147313710 HI On-Demand Anodyne TRPV1 15 40 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1cccnc1N1CCCC1 ZINC000147313710 HI On-Demand Anodyne P2RY1 44 34 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1cccnc1N1CCCC1 ZINC000147313710 HI On-Demand Anodyne SCN2A 17 42 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1cccnc1N1CCCC1 ZINC000147313710 HI On-Demand Anodyne SCN10A 18 42 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1cccnc1N1CCCC1 ZINC000147313710 HI On-Demand Anodyne NAMPT 52 41 CCNc1cccc(NCCN2CCOCC2)n1 ZINC000147313738 CD For-Sale Anodyne CASR 40 36 CCNc1cccc(NCCN2CCOCC2)n1 ZINC000147313738 CD For-Sale Anodyne TLR9 0 50 Cc1ccc(O[C@@H](C)C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1 ZINC000147313760 FI On-Demand Mild GRM5 20 42 CCCNc1cc(Oc2ccccc2NC(C)=O)ncn1 ZINC000147313772 CG For-Sale Anodyne INHA 19 43 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cccc(OC(F)(F)F)c2)C1 ZINC000147313836 HD On-Demand Anodyne ADRA1D 15 41 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cccc(OC(F)(F)F)c2)C1 ZINC000147313836 HD On-Demand Anodyne ADRA1B 20 41 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cccc(OC(F)(F)F)c2)C1 ZINC000147313836 HD On-Demand Anodyne SFRP1 123 36 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cccc(OC(F)(F)F)c2)C1 ZINC000147313836 HD On-Demand Anodyne WNT3 83 35 CCOC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147313854 ED On-Demand Anodyne ACR 48 34 Cc1ccc(O[C@H](C)C(=O)Nc2cccc(C#Cc3ccccn3)c2)cc1 ZINC000147313917 FI On-Demand Mild GRM5 20 42 CCCS(=O)(=O)Nc1ccccc1C(=O)N1CCC(c2nnc3n2CCC3)CC1 ZINC000147313968 HE On-Demand Anodyne CCR8 62 33 O=C(Nc1ccccc1Cn1cncn1)c1cnn(-c2ccccc2Cl)c1 ZINC000147313985 GG On-Demand Anodyne CNR1 26 42 O=C(Nc1ccccc1Cn1cncn1)c1cnn(-c2ccccc2Cl)c1 ZINC000147313985 GG On-Demand Anodyne EPHB3 51 35 CCOC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147314004 ED On-Demand Anodyne ACR 48 34 CC1(CNC(=O)c2cccc3c2OCCN3)CCCC1 ZINC000147314021 CF For-Sale Anodyne HCN1 55 36 CC1(CNC(=O)c2cccc3c2OCCN3)CCCC1 ZINC000147314021 CF For-Sale Anodyne HCN4 50 32 Cc1noc([C@@H]2CCCN(C(=O)c3cnn(-c4ccccc4Cl)c3)C2)n1 ZINC000147314264 FG On-Demand Anodyne GRM5 23 45 Cc1noc([C@@H]2CCCN(C(=O)c3cnn(-c4ccccc4Cl)c3)C2)n1 ZINC000147314264 FG On-Demand Anodyne MAP3K12 34 41 COc1ccc2c(c1)[C@H](NCCCCC(C)C)CCC2 ZINC000147314382 CI For-Sale Anodyne NQO2 36 44 COC(=O)c1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147314419 DC On-Demand Anodyne MMP2 23 43 COC(=O)c1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147314419 DC On-Demand Anodyne MMP10 15 42 COC(=O)c1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147314419 DC On-Demand Anodyne LIMK2 43 37 NCCc1ccccc1NO ZINC000147314435 AC For-Sale Anodyne TAAR1 29 56 Cc1ccc2oc(-c3cc(N)cc(Cl)c3)nc2c1 ZINC000147314436 CI For-Sale Anodyne AGPAT2 29 42 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2c[nH]c(C(=O)N3CCCC3)c2)C1 ZINC000147314437 HB On-Demand Anodyne SFRP1 73 34 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2c[nH]c(C(=O)N3CCCC3)c2)C1 ZINC000147314437 HB On-Demand Anodyne WNT3 47 30 CC[C@@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@@H]1N ZINC000147314472 DF On-Demand Anodyne SLC9A1 44 41 CC[C@@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@@H]1N ZINC000147314472 DF On-Demand Anodyne L3MBTL1 0 40 CC[C@@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@@H]1N ZINC000147314472 DF On-Demand Anodyne L3MBTL3 67 40 CCc1cccc(OCC(=O)Nc2ccccc2N2CCCCC2)c1 ZINC000147314484 EI On-Demand Anodyne HRH2 47 42 CCc1cccc(OCC(=O)Nc2ccccc2N2CCCCC2)c1 ZINC000147314484 EI On-Demand Anodyne ABCC8 20 40 CCc1cccc(OCC(=O)Nc2ccccc2N2CCCCC2)c1 ZINC000147314484 EI On-Demand Anodyne KCNQ2 101 57 CCc1cccc(OCC(=O)Nc2ccccc2N2CCCCC2)c1 ZINC000147314484 EI On-Demand Anodyne CPT1A 43 35 CCc1cccc(OCC(=O)Nc2ccccc2N2CCCCC2)c1 ZINC000147314484 EI On-Demand Anodyne CSF1R 16 45 CCc1cccc(OCC(=O)Nc2ccccc2N2CCCCC2)c1 ZINC000147314484 EI On-Demand Anodyne TAAR1 21 42 Cc1noc([C@@H]2CCCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)C2)n1 ZINC000147314490 EH On-Demand Anodyne GRM5 29 55 NC(=O)c1ccc(OCC(=O)N2CCC(c3nnc4n3CCC4)CC2)cc1 ZINC000147314510 FD On-Demand Anodyne CPT1A 67 41 CC(=O)CCCCCC#CCC(=O)O ZINC000147314551 AE For-Sale Anodyne PAOX 42 36 COc1ccc2c(c1)[C@@H](NCCCCC(C)C)CCC2 ZINC000147314561 CI For-Sale Anodyne NQO2 36 44 COC(=O)c1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147314589 DC On-Demand Anodyne MMP2 23 43 COC(=O)c1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147314589 DC On-Demand Anodyne MMP10 15 42 COC(=O)c1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147314589 DC On-Demand Anodyne LIMK2 43 37 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2c[nH]c(C(=O)N3CCCC3)c2)C1 ZINC000147314594 HB On-Demand Anodyne SFRP1 73 34 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2c[nH]c(C(=O)N3CCCC3)c2)C1 ZINC000147314594 HB On-Demand Anodyne WNT3 47 30 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne ALOX5 15 45 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne ACE 42 47 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne PTGS1 22 49 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne PPARG 35 47 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne PTGER2 27 43 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne PPARA 41 47 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne MME 110 47 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne LTA4H 21 41 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne PTGER4 32 45 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne ACACA 33 42 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne MMP13 17 45 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne CTSB 24 40 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne PAPA1_CARPA 40 36 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne CPA1 55 40 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne SLC15A1 0 45 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne ACACB 15 42 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne CAPNS1 57 34 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne MMP2 22 41 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne MMP3 17 40 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne SLC1A6 0 46 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne PTPN1 0 40 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne CAPN1 48 40 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne SLC1A7 0 46 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne CAPN2 70 36 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne ACE2 91 47 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne MMP12 15 42 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne SLC1A2 25 46 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne ADAMTS4 74 44 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne POL 0 50 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne NPR 70 33 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne NAAA 17 41 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne FFAR1 51 49 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne FFAR4 41 35 C[C@@H](OCc1ccc(-c2ccccc2)cc1)C(=O)O ZINC000147314628 CG For-Sale Anodyne BLAIMP-1 0 49 CC[C@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@@H]1N ZINC000147314640 DF On-Demand Anodyne SLC9A1 44 41 CC[C@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@@H]1N ZINC000147314640 DF On-Demand Anodyne L3MBTL1 0 40 CC[C@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@@H]1N ZINC000147314640 DF On-Demand Anodyne L3MBTL3 67 40 CC[C@@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@H]1N ZINC000147314802 DF On-Demand Anodyne SLC9A1 44 41 CC[C@@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@H]1N ZINC000147314802 DF On-Demand Anodyne L3MBTL1 0 40 CC[C@@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@H]1N ZINC000147314802 DF On-Demand Anodyne L3MBTL3 67 40 CS(=O)(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147314829 GB On-Demand Anodyne SFRP1 75 34 CS(=O)(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147314829 GB On-Demand Anodyne WNT3 47 32 NC1(CNC(=O)c2ccccc2)CCCCC1 ZINC000147314837 BE On-Demand Anodyne ECR 24 40 NC1(CNC(=O)c2ccccc2)CCCCC1 ZINC000147314837 BE On-Demand Anodyne CTRB1 22 42 NC1(CNC(=O)c2ccccc2)CCCCC1 ZINC000147314837 BE On-Demand Anodyne SLC6A9 17 47 NC1(CNC(=O)c2ccccc2)CCCCC1 ZINC000147314837 BE On-Demand Anodyne ACAT 0 43 NC1(CNC(=O)c2ccccc2)CCCCC1 ZINC000147314837 BE On-Demand Anodyne HCN1 55 34 NC1(CNC(=O)c2ccccc2)CCCCC1 ZINC000147314837 BE On-Demand Anodyne HCN4 53 34 NC1(CNC(=O)c2ccccc2)CCCCC1 ZINC000147314837 BE On-Demand Anodyne KCNK3 43 34 Cc1noc([C@@H]2CCCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)C2)n1 ZINC000147314843 EH On-Demand Anodyne GRM5 29 55 CN(Cc1cscn1)C(=O)NCCc1ccc2c(c1)OCO2 ZINC000147314903 DE On-Demand Anodyne BMP1 41 35 CN(Cc1cscn1)C(=O)NCCc1ccc2c(c1)OCO2 ZINC000147314903 DE On-Demand Anodyne NOS2 68 37 CC(C)(C)C1CCC2(CC1)N=C(c1cc(Cl)cc(Cl)c1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147314942 KK Annotated Anodyne GCGR 57 70 CC(C)(C)C1CCC2(CC1)N=C(c1cc(Cl)cc(Cl)c1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147314942 KK Annotated Anodyne GLP1R 18 52 CC(C)(C)C1CCC2(CC1)N=C(c1cc(Cl)cc(Cl)c1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147314942 KK Annotated Anodyne CACNA1I 48 33 CC(C)(C)C1CCC2(CC1)N=C(c1cc(Cl)cc(Cl)c1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147314942 KK Annotated Anodyne GIPR 93 42 CC[C@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@H]1N ZINC000147314963 DF On-Demand Anodyne SLC9A1 44 41 CC[C@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@H]1N ZINC000147314963 DF On-Demand Anodyne L3MBTL1 0 40 CC[C@H]1CN(C(=O)c2ccc(C(F)(F)F)cc2)CC[C@H]1N ZINC000147314963 DF On-Demand Anodyne L3MBTL3 67 40 CS(=O)(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147314989 GB On-Demand Anodyne SFRP1 75 34 CS(=O)(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147314989 GB On-Demand Anodyne WNT3 47 32 CNc1ncc(Cl)c(Oc2ccccc2NC(C)=O)n1 ZINC000147315028 CF For-Sale Anodyne MAPK9 46 36 CNc1ncc(Cl)c(Oc2ccccc2NC(C)=O)n1 ZINC000147315028 CF For-Sale Anodyne MAPK10 47 36 CNc1ncc(Cl)c(Oc2ccccc2NC(C)=O)n1 ZINC000147315028 CF For-Sale Anodyne LRRK2 15 45 Fc1cc(OCc2ccc(Br)cc2)ccc1Cl ZINC000147315062 DJ For-Sale Anodyne MAOA 19 45 Fc1cc(OCc2ccc(Br)cc2)ccc1Cl ZINC000147315062 DJ For-Sale Anodyne MAOB 49 51 Fc1cc(OCc2ccc(Br)cc2)ccc1Cl ZINC000147315062 DJ For-Sale Anodyne CCR5 21 41 Fc1cc(OCc2ccc(Br)cc2)ccc1Cl ZINC000147315062 DJ For-Sale Anodyne ACR 16 40 Cc1noc([C@@H]2CCCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Br)c3)C2)n1 ZINC000147315144 GH On-Demand Anodyne GRM5 16 49 CCc1nc(CN(C)C(=O)NCCc2ccc3c(c2)OCO3)cs1 ZINC000147315159 EF On-Demand Anodyne BMP1 40 37 CCc1nc(CN(C)C(=O)NCCc2ccc3c(c2)OCO3)cs1 ZINC000147315159 EF On-Demand Anodyne NOS2 62 41 C[C@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315213 ED On-Demand Anodyne MMP13 19 56 C[C@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315213 ED On-Demand Anodyne MMP2 22 51 C[C@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315213 ED On-Demand Anodyne MMP3 15 56 C[C@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315213 ED On-Demand Anodyne MMP14 21 51 C[C@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315213 ED On-Demand Anodyne MMP9 17 55 C[C@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315213 ED On-Demand Anodyne MMP10 15 43 C[C@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315213 ED On-Demand Anodyne MMP7 19 44 C[C@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315213 ED On-Demand Anodyne IDO1 23 42 Cc1cc(NCCCCC(C)C)ccc1N ZINC000147315258 BH For-Sale Anodyne LEF 58 32 CCN(CC)CCc1c[nH]c2cc(F)c(F)cc12 ZINC000147315259 CG For-Sale Anodyne HTR1D 48 61 CCN(CC)CCc1c[nH]c2cc(F)c(F)cc12 ZINC000147315259 CG For-Sale Anodyne HTR1B 20 48 CCN(CC)CCc1c[nH]c2cc(F)c(F)cc12 ZINC000147315259 CG For-Sale Anodyne MPO 97 49 CCN(CC)CCc1c[nH]c2cc(F)c(F)cc12 ZINC000147315259 CG For-Sale Anodyne HTR1E 16 41 CCN(CC)CCc1c[nH]c2cc(F)c(F)cc12 ZINC000147315259 CG For-Sale Anodyne HTR5A 21 40 CCCc1c(N)ncnc1Oc1ccccc1NC(C)=O ZINC000147315277 CF For-Sale Anodyne INHA 15 44 Fc1cc(OCc2cccc(Br)c2)ccc1Cl ZINC000147315294 DJ For-Sale Anodyne MAOA 18 51 Fc1cc(OCc2cccc(Br)c2)ccc1Cl ZINC000147315294 DJ For-Sale Anodyne MAOB 69 53 Fc1cc(OCc2cccc(Br)c2)ccc1Cl ZINC000147315294 DJ For-Sale Anodyne F9 0 42 Fc1cc(OCc2cccc(Br)c2)ccc1Cl ZINC000147315294 DJ For-Sale Anodyne FFAR1 28 40 C[C@@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315346 ED On-Demand Anodyne MMP13 19 56 C[C@@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315346 ED On-Demand Anodyne MMP2 22 51 C[C@@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315346 ED On-Demand Anodyne MMP3 15 56 C[C@@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315346 ED On-Demand Anodyne MMP14 21 51 C[C@@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315346 ED On-Demand Anodyne MMP9 17 55 C[C@@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315346 ED On-Demand Anodyne MMP10 15 43 C[C@@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315346 ED On-Demand Anodyne MMP7 19 44 C[C@@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147315346 ED On-Demand Anodyne IDO1 23 42 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne F2 15 48 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne ACE 57 58 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne OPRM1 31 45 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne OPRD1 36 45 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne FOLH1 49 42 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne ELANE 29 43 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne MME 102 47 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne ANPEP 73 35 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CCNA2 0 42 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CASP3 24 47 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne BMP1 34 45 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne RNPEP 41 40 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne NPY1R 30 41 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne KLK3 100 44 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CTSB 85 54 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PAPA1_CARPA 95 48 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CYSP_TRYCR 62 43 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CCKAR 34 45 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CTSK 68 52 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CTSL 67 50 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne SLC15A1 0 43 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PGA 21 42 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CHRNA4 0 52 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne NPFFR2 60 40 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne C3AR1 100 43 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CAPNS1 77 44 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CANX_CHICK 0 41 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne MMP2 25 54 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne MMP3 44 48 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne MMP8 38 40 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne GRIA1 59 37 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne MMP14 38 48 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne ECE1 18 40 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne HLA-DRB1 54 37 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne HDAC1 15 47 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne HDAC2 23 46 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne HDAC6 15 46 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne MMP11 42 34 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne FAAH 15 46 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PAM 0 45 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PCSK5 58 42 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne FURIN 95 47 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PCSK1 0 42 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CTSS 28 52 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne GHSR 20 41 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CAPN1 109 52 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne MMP9 15 51 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CASP1 35 51 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CAPN2 168 52 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne KYNU 0 43 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne ACE2 59 36 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CASP6 34 45 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne CASP9 38 45 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne TGM2 33 50 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PCSK6 0 42 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne LAP3 51 39 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PROTEASE 0 44 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne KLK5 23 47 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne TPSAB1 57 40 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne ST14 45 35 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne MMP1 15 51 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne FPR1 58 39 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne POL 0 57 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne NPR 112 52 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne AMP1_PLAFQ 43 39 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne RHODESAIN 0 44 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne NAAA 44 38 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne SIRT1 34 46 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PSMB5 48 45 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne SLC15A2 0 43 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne KISS1R 48 31 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne POLG_WNV 77 48 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne SSPA 0 41 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne QRFPR 53 47 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne NPFFR1 84 40 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PADI4 0 42 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne MCA2 0 52 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne TMPRSS11D 57 47 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne TMPRSS6 53 35 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PADI1 0 42 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PADI2 0 40 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PADI3 0 42 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne VM1B1_BOTAS 0 44 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne PDS 44 33 C[C@@H](CCCNC(=O)OCc1ccccc1)C(=O)O ZINC000147315358 CE For-Sale Anodyne Q8I6Z5_PLAF7 0 46 C=CCOC(=O)[C@@H]1CCCCN1C(=O)C(=O)C(C)(C)CO ZINC000147315364 CC For-Sale Anodyne FKBP1A 75 56 C=CCOC(=O)[C@@H]1CCCCN1C(=O)C(=O)C(C)(C)CO ZINC000147315364 CC For-Sale Anodyne MTOR 26 43 CC(C)(C)C1CCC2(CC1)N=C(c1ccccc1F)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147315366 KJ Annotated Anodyne GCGR 33 57 CC(C)(C)C1CCC2(CC1)N=C(c1ccccc1F)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147315366 KJ Annotated Anodyne GLP1R 15 40 CC(C)(C)C1CCC2(CC1)N=C(c1ccccc1F)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147315366 KJ Annotated Anodyne GIPR 77 41 C[C@@H](CC(=O)NN(C)C)[C@@H]1CCCNC1 ZINC000147315420 BC For-Sale Reactive CPN1 0 49 COc1ccc([N+](=O)[O-])c(C(=O)NCC(=O)Nc2ccc(Br)cc2)c1 ZINC000147315427 HF On-Demand Bother FPR2 19 40 COc1ccc([N+](=O)[O-])c(C(=O)NCC(=O)Nc2ccc(Br)cc2)c1 ZINC000147315427 HF On-Demand Bother TAAR1 22 43 COc1ccc([N+](=O)[O-])c(C(=O)NCC(=O)Nc2ccc(Br)cc2)c1 ZINC000147315427 HF On-Demand Bother AKR1C3 15 41 COc1ccc([N+](=O)[O-])c(C(=O)NCC(=O)Nc2ccc(Br)cc2)c1 ZINC000147315427 HF On-Demand Bother AKR1C2 41 41 COc1ccc(Cl)cc1CNC1(C(=O)O)CCC1 ZINC000147315438 CE On-Demand Anodyne NTSR2 23 43 COc1ccc(Cl)cc1CNC1(C(=O)O)CCC1 ZINC000147315438 CE On-Demand Anodyne COLA 70 41 COc1ccc(Cl)cc1CNC1(C(=O)O)CCC1 ZINC000147315438 CE On-Demand Anodyne CPT1A 67 41 COc1ccc(Cl)cc1CNC1(C(=O)O)CCC1 ZINC000147315438 CE On-Demand Anodyne CPT1B 65 36 COc1ccc(Cl)cc1CNC1(C(=O)O)CCC1 ZINC000147315438 CE On-Demand Anodyne QRFPR 40 39 CC(C)CCCCNc1cc(N)ccn1 ZINC000147315445 BF For-Sale Anodyne HRH4 0 44 Cc1noc([C@@H]2CCCN(C(=O)[C@H]3C[C@@H]3c3cccc(Br)c3)C2)n1 ZINC000147315462 GH On-Demand Anodyne GRM5 16 49 C[C@H](CC(=O)NN(C)C)[C@@H]1CCCNC1 ZINC000147315491 BC For-Sale Reactive CPN1 0 49 CC(C)(C)C1CCC2(CC1)N=C(c1cccc(Cl)c1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147315559 KK Annotated Anodyne GLP1R 16 45 CC(C)(C)C1CCC2(CC1)N=C(c1cccc(Cl)c1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147315559 KK Annotated Anodyne MDM2 42 32 CC(C)(C)C1CCC2(CC1)N=C(c1cccc(Cl)c1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147315559 KK Annotated Anodyne GIPR 85 40 COc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1C ZINC000147315571 DD On-Demand Anodyne LEF 52 38 COc1ccc2c(c1)nc(N)n2CCNC(=O)N(C)C ZINC000147315628 CC For-Sale Anodyne MTNR1A 52 37 COc1ccc2c(c1)nc(N)n2CCNC(=O)N(C)C ZINC000147315628 CC For-Sale Anodyne MTNR1B 42 37 COc1ccc2c(c1)nc(N)n2CCNC(=O)N(C)C ZINC000147315628 CC For-Sale Anodyne PROKR1 50 30 C[C@@H](CC(=O)NN(C)C)[C@H]1CCCNC1 ZINC000147315641 BC For-Sale Reactive CPN1 0 49 Cc1cc(Br)cc(S(N)(=O)=O)c1OCCN1CCCCC1 ZINC000147315671 GE For-Sale Anodyne HRH3 20 42 Cc1cc(Br)cc(S(N)(=O)=O)c1OCCN1CCCCC1 ZINC000147315671 GE For-Sale Anodyne PSMB2 46 38 Cc1cc(Br)cc(S(N)(=O)=O)c1OCCN1CCCCC1 ZINC000147315671 GE For-Sale Anodyne PSMB1 41 38 O=C(CNC1(C(=O)O)CCC1)Nc1ccc([N+](=O)[O-])cc1 ZINC000147315673 CD For-Sale Bother NMBR 47 33 CCCNc1nc(N)nc(-c2ccccc2)n1 ZINC000147315675 BD For-Sale Anodyne TPH1 57 49 CC[C@@H]1CN(C(=O)c2ccc(C)cc2)CC[C@@H]1N ZINC000147315680 BE On-Demand Anodyne L3MBTL1 0 43 CC[C@@H]1CN(C(=O)c2ccc(C)cc2)CC[C@@H]1N ZINC000147315680 BE On-Demand Anodyne L3MBTL3 77 43 CC[C@@H]1CN(C(=O)c2ccc(C)cc2)CC[C@@H]1N ZINC000147315680 BE On-Demand Anodyne MBTD1 0 40 CC[C@@H]1CN(C(=O)c2ccc(C)cc2)CC[C@@H]1N ZINC000147315680 BE On-Demand Anodyne SLC6A7 0 40 COC(=O)/C=C/c1ccc(Cl)c(N)c1 ZINC000147315690 BE In-Stock Anodyne PYGL 0 43 COC(=O)/C=C/c1ccc(Cl)c(N)c1 ZINC000147315690 BE In-Stock Anodyne MMP2 0 40 COC(=O)/C=C/c1ccc(Cl)c(N)c1 ZINC000147315690 BE In-Stock Anodyne NR1H4 50 42 COC(=O)/C=C/c1ccc(Cl)c(N)c1 ZINC000147315690 BE In-Stock Anodyne MMP9 0 40 COC(=O)/C=C/c1ccc(Cl)c(N)c1 ZINC000147315690 BE In-Stock Anodyne MMP12 0 40 COC(=O)/C=C/c1ccc(Cl)c(N)c1 ZINC000147315690 BE In-Stock Anodyne MMP1 0 40 C[C@H](NC(=O)c1cccc2c1OCCN2)c1ccccc1 ZINC000147315755 CF For-Sale Anodyne PTGER4 23 40 C[C@H](NC(=O)c1cccc2c1OCCN2)c1ccccc1 ZINC000147315755 CF For-Sale Anodyne KCNA5 0 44 CNc1cccc(NCCN2CCOCC2)n1 ZINC000147315757 BC For-Sale Anodyne CASR 40 36 CNc1cccc(NCCN2CCOCC2)n1 ZINC000147315757 BC For-Sale Anodyne TLR9 0 50 COc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1C ZINC000147315760 DD On-Demand Anodyne LEF 52 38 CC(C)(C)C1CCC2(CC1)N=C(c1ccc(C(F)(F)F)cc1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147315768 KK Annotated Anodyne GLP1R 20 43 CC(C)(C)C1CCC2(CC1)N=C(c1ccc(C(F)(F)F)cc1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147315768 KK Annotated Anodyne GIPR 106 48 C[C@H](CC(=O)NN(C)C)[C@H]1CCCNC1 ZINC000147315847 BC For-Sale Reactive CPN1 0 49 CC[C@H]1CN(C(=O)c2ccc(C)cc2)CC[C@@H]1N ZINC000147315873 BE On-Demand Anodyne L3MBTL1 0 43 CC[C@H]1CN(C(=O)c2ccc(C)cc2)CC[C@@H]1N ZINC000147315873 BE On-Demand Anodyne L3MBTL3 77 43 CC[C@H]1CN(C(=O)c2ccc(C)cc2)CC[C@@H]1N ZINC000147315873 BE On-Demand Anodyne MBTD1 0 40 CC[C@H]1CN(C(=O)c2ccc(C)cc2)CC[C@@H]1N ZINC000147315873 BE On-Demand Anodyne SLC6A7 0 40 COc1ccc([C@@H](O)c2c(C)oc3ccccc23)cc1 ZINC000147315958 CH For-Sale Anodyne NQO1 38 53 CC(C)(C)[C@@H](O)C(=O)c1ccc(Cl)cc1 ZINC000147315961 BF For-Sale Anodyne FABP1 15 46 C[C@@H](NC(=O)c1cccc2c1OCCN2)c1ccccc1 ZINC000147315964 CF For-Sale Anodyne PTGER4 23 40 C[C@@H](NC(=O)c1cccc2c1OCCN2)c1ccccc1 ZINC000147315964 CF For-Sale Anodyne KCNA5 0 44 C[C@@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147315990 KK Annotated Anodyne GCGR 59 90 C[C@@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147315990 KK Annotated Anodyne CCKBR 51 35 C[C@@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147315990 KK Annotated Anodyne GLP1R 25 68 C[C@@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147315990 KK Annotated Anodyne CACNA1I 40 32 C[C@@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147315990 KK Annotated Anodyne GIPR 71 46 O=C(O)C[C@H](NC(=O)c1ccccc1)C1CC1 ZINC000147316016 BD On-Demand Anodyne ECR 27 41 O=C(O)C[C@H](NC(=O)c1ccccc1)C1CC1 ZINC000147316016 BD On-Demand Anodyne KCNK3 44 35 Cc1cc(C(=O)N2CCN(Cc3cccc(Cl)c3)CC2)cc([N+](=O)[O-])c1 ZINC000147316029 FH On-Demand Bother DRD4 17 40 Cc1cc(C(=O)N2CCN(Cc3cccc(Cl)c3)CC2)cc([N+](=O)[O-])c1 ZINC000147316029 FH On-Demand Bother FAAH 24 49 Cc1cc(C(=O)N2CCN(Cc3cccc(Cl)c3)CC2)cc([N+](=O)[O-])c1 ZINC000147316029 FH On-Demand Bother CCR8 20 40 COc1ccc(C(=O)NN(C)C)c(N)c1 ZINC000147316045 BC For-Sale Reactive AKR1C3 21 40 COc1ccc(C(=O)NN(C)C)c(N)c1 ZINC000147316045 BC For-Sale Reactive AKR1C2 54 40 CC[C@@H]1CN(C(=O)c2ccc(C)cc2)CC[C@H]1N ZINC000147316064 BE On-Demand Anodyne L3MBTL1 0 43 CC[C@@H]1CN(C(=O)c2ccc(C)cc2)CC[C@H]1N ZINC000147316064 BE On-Demand Anodyne L3MBTL3 77 43 CC[C@@H]1CN(C(=O)c2ccc(C)cc2)CC[C@H]1N ZINC000147316064 BE On-Demand Anodyne MBTD1 0 40 CC[C@@H]1CN(C(=O)c2ccc(C)cc2)CC[C@H]1N ZINC000147316064 BE On-Demand Anodyne SLC6A7 0 40 COc1ccc([C@H](O)c2c(C)oc3ccccc23)cc1 ZINC000147316133 CH For-Sale Anodyne NQO1 38 53 CC(C)(C)[C@H](O)C(=O)c1ccc(Cl)cc1 ZINC000147316160 BF For-Sale Anodyne FABP1 15 46 CNc1nc(OC)nc(Oc2ccccc2NC(C)=O)n1 ZINC000147316192 CD For-Sale Anodyne ALS 47 37 O=C(O)C[C@@H](NC(=O)c1ccccc1)C1CC1 ZINC000147316205 BD On-Demand Anodyne ECR 27 41 O=C(O)C[C@@H](NC(=O)c1ccccc1)C1CC1 ZINC000147316205 BD On-Demand Anodyne KCNK3 44 35 CC(C)(C)C1CCC2(CC1)N=C(c1ccc(Cl)cc1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147316219 KK Annotated Anodyne GCGR 52 63 CC(C)(C)C1CCC2(CC1)N=C(c1ccc(Cl)cc1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147316219 KK Annotated Anodyne GLP1R 16 44 CC(C)(C)C1CCC2(CC1)N=C(c1ccc(Cl)cc1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147316219 KK Annotated Anodyne GIPR 89 40 Cc1cc(C(=O)N2CCN(Cc3ccccc3C)CC2)cc([N+](=O)[O-])c1 ZINC000147316269 FG On-Demand Bother MGLL 0 43 Cc1cc(C(=O)N2CCN(Cc3ccccc3C)CC2)cc([N+](=O)[O-])c1 ZINC000147316269 FG On-Demand Bother ABHD6 0 43 CC[C@H]1CN(C(=O)c2ccc(C)cc2)CC[C@H]1N ZINC000147316290 BE On-Demand Anodyne L3MBTL1 0 43 CC[C@H]1CN(C(=O)c2ccc(C)cc2)CC[C@H]1N ZINC000147316290 BE On-Demand Anodyne L3MBTL3 77 43 CC[C@H]1CN(C(=O)c2ccc(C)cc2)CC[C@H]1N ZINC000147316290 BE On-Demand Anodyne MBTD1 0 40 CC[C@H]1CN(C(=O)c2ccc(C)cc2)CC[C@H]1N ZINC000147316290 BE On-Demand Anodyne SLC6A7 0 40 CCCCOC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147316305 FE On-Demand Anodyne ACR 41 40 CCCNc1cccc(NCCN2CCOCC2)n1 ZINC000147316373 CD For-Sale Anodyne CASR 40 36 CCCNc1cccc(NCCN2CCOCC2)n1 ZINC000147316373 CD For-Sale Anodyne TLR9 0 50 Cc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c(Br)c1 ZINC000147316410 HD On-Demand Anodyne CTSC 16 40 Cn1ncnc1NC(=O)NCc1ccccc1 ZINC000147316434 BD On-Demand Anodyne ACAT 0 50 Cn1ncnc1NC(=O)NCc1ccccc1 ZINC000147316434 BD On-Demand Anodyne PDS 41 33 CC(C)(C)C1CCC2(CC1)N=C(c1ccc(Cl)c(Cl)c1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147316442 KK Annotated Anodyne GCGR 143 85 CC(C)(C)C1CCC2(CC1)N=C(c1ccc(Cl)c(Cl)c1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147316442 KK Annotated Anodyne GLP1R 16 44 CC(C)(C)C1CCC2(CC1)N=C(c1ccc(Cl)c(Cl)c1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147316442 KK Annotated Anodyne GIPR 91 41 COc1ccc(CCn2cc(I)c(C)cc2=O)cc1 ZINC000147316455 FG For-Sale Anodyne KCNA5 26 43 COc1ccc(CCn2cc(I)c(C)cc2=O)cc1 ZINC000147316455 FG For-Sale Anodyne IDH1 19 40 CCNc1cc(Oc2ccccc2NC(C)=O)ncn1 ZINC000147316458 CF For-Sale Anodyne INHA 18 42 C[C@H](CNS(=O)(=O)Cc1ccc(F)cc1)CC(=O)O ZINC000147316460 CD On-Demand Anodyne HMGCR 87 36 CCCCOC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147316475 FE On-Demand Anodyne ACR 41 40 Cc1noc([C@@H]2CCCN(C(=O)c3ccc4c(c3)COC4)C2)n1 ZINC000147316491 DE On-Demand Anodyne GRM5 19 48 Cc1noc([C@@H]2CCCN(C(=O)c3ccc4c(c3)COC4)C2)n1 ZINC000147316491 DE On-Demand Anodyne L3MBTL3 41 33 Cc1noc([C@@H]2CCCN(C(=O)c3ccc4c(c3)COC4)C2)n1 ZINC000147316491 DE On-Demand Anodyne ETHR 41 34 N#CC[C@H]1CCOc2cc(S(=O)(=O)c3ccccc3)ccc21 ZINC000147316600 DG For-Sale Mild HTR6 38 44 NC[C@@H](O)[C@@H](N)C(=O)O ZINC000147316606 AA For-Sale Anodyne SLC1A6 49 31 NC[C@@H](O)[C@@H](N)C(=O)O ZINC000147316606 AA For-Sale Anodyne SLC1A7 49 31 C[C@@H](CNS(=O)(=O)Cc1ccc(F)cc1)CC(=O)O ZINC000147316647 CD On-Demand Anodyne HMGCR 87 36 Cn1cc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1C(N)=O ZINC000147316691 FA On-Demand Anodyne SFRP1 49 31 CCOc1ccc(C(=O)N2CC[C@H](N)[C@H](CC)C2)cc1 ZINC000147316705 CE On-Demand Anodyne AVPR1A 23 49 CCOc1ccc(C(=O)N2CC[C@H](N)[C@H](CC)C2)cc1 ZINC000147316705 CE On-Demand Anodyne L3MBTL1 0 40 CCOc1ccc(C(=O)N2CC[C@H](N)[C@H](CC)C2)cc1 ZINC000147316705 CE On-Demand Anodyne L3MBTL3 66 40 Cc1ccc2nc(N)n(CCNC(=O)N(C)C)c2c1 ZINC000147316720 CD For-Sale Anodyne CDPK1 0 40 Cc1noc([C@H]2CCCN(C(=O)CCCc3ccc4c(c3)-c3ccccc3C4)C2)n1 ZINC000147316778 HJ On-Demand Anodyne PREP 50 38 Cc1noc([C@H]2CCCN(C(=O)CCCc3ccc4c(c3)-c3ccccc3C4)C2)n1 ZINC000147316778 HJ On-Demand Anodyne ETHR 56 39 N#CC[C@@H]1CCOc2cc(S(=O)(=O)c3ccccc3)ccc21 ZINC000147316803 DG For-Sale Mild HTR6 38 44 CC(C)(C)C1CCC2(CC1)N=C(c1ccc(OC(F)(F)F)cc1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147316827 KK Annotated Anodyne GCGR 161 83 CC(C)(C)C1CCC2(CC1)N=C(c1ccc(OC(F)(F)F)cc1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147316827 KK Annotated Anodyne GLP1R 17 53 CC(C)(C)C1CCC2(CC1)N=C(c1ccc(OC(F)(F)F)cc1)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147316827 KK Annotated Anodyne GIPR 117 53 NC[C@H](O)[C@@H](N)C(=O)O ZINC000147316837 AA For-Sale Anodyne SLC1A6 49 31 NC[C@H](O)[C@@H](N)C(=O)O ZINC000147316837 AA For-Sale Anodyne SLC1A7 49 31 C[C@H](CNS(=O)(=O)c1ccc2c(c1)CC(=O)N2)CC(=O)O ZINC000147316857 DC On-Demand Anodyne PKM 32 41 Cn1cc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1C(N)=O ZINC000147316884 FA On-Demand Anodyne SFRP1 49 31 CCOc1ccc(C(=O)N2CC[C@H](N)[C@@H](CC)C2)cc1 ZINC000147316964 CE On-Demand Anodyne AVPR1A 23 49 CCOc1ccc(C(=O)N2CC[C@H](N)[C@@H](CC)C2)cc1 ZINC000147316964 CE On-Demand Anodyne L3MBTL1 0 40 CCOc1ccc(C(=O)N2CC[C@H](N)[C@@H](CC)C2)cc1 ZINC000147316964 CE On-Demand Anodyne L3MBTL3 66 40 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147316995 EH On-Demand Anodyne PRCP 58 38 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147316995 EH On-Demand Anodyne GRM5 24 46 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147316995 EH On-Demand Anodyne SMO 51 39 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147316995 EH On-Demand Anodyne ETHR 60 36 CC[C@H](N)CC(=O)NN(C)C ZINC000147317008 AB For-Sale Reactive KDM7A 0 42 Nc1c(C(=O)Nc2ccc(Cl)cn2)oc2ccc([N+](=O)[O-])cc12 ZINC000147317025 EG For-Sale Bother F10 53 36 O=C1OC(c2ccc(OCCO)cc2)(c2ccc(OCCO)cc2)c2ccccc21 ZINC000147317054 HF For-Sale Anodyne AKR1C1 17 51 C[C@@H](CNS(=O)(=O)c1ccc2c(c1)CC(=O)N2)CC(=O)O ZINC000147317071 DC On-Demand Anodyne PKM 32 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147317079 EE On-Demand Anodyne CTSS 23 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147317079 EE On-Demand Anodyne EPHX2 57 50 CC(C)(C)C1CCC2(CC1)N=C(c1ccccc1Cl)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147317087 KK Annotated Anodyne GCGR 122 85 CC(C)(C)C1CCC2(CC1)N=C(c1ccccc1Cl)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147317087 KK Annotated Anodyne GLP1R 15 40 CC(C)(C)C1CCC2(CC1)N=C(c1ccccc1Cl)C(=O)N2Cc1ccc(C(=O)NCCC(=O)O)cc1 ZINC000147317087 KK Annotated Anodyne GIPR 60 40 Cc1cc(C)c2oc(-c3cc(N)cc(Cl)c3)nc2c1 ZINC000147317101 CI For-Sale Anodyne CETP 0 44 CC(C)(C)OC(=O)N1CCC(COC(=O)Nc2ccccc2C(N)=O)CC1 ZINC000147317133 GF For-Sale Anodyne CCR8 38 40 CC(C)(C)OC(=O)N1CCC(COC(=O)Nc2ccccc2C(N)=O)CC1 ZINC000147317133 GF For-Sale Anodyne GPR119 50 44 CCOc1ccc(C(=O)N2CC[C@@H](N)[C@H](CC)C2)cc1 ZINC000147317160 CE On-Demand Anodyne AVPR1A 23 49 CCOc1ccc(C(=O)N2CC[C@@H](N)[C@H](CC)C2)cc1 ZINC000147317160 CE On-Demand Anodyne L3MBTL1 0 40 CCOc1ccc(C(=O)N2CC[C@@H](N)[C@H](CC)C2)cc1 ZINC000147317160 CE On-Demand Anodyne L3MBTL3 66 40 Fc1cc(OCc2ccc(F)c(Br)c2)ccc1Cl ZINC000147317168 EJ For-Sale Anodyne MAOB 40 38 Fc1cc(OCc2ccc(F)c(Br)c2)ccc1Cl ZINC000147317168 EJ For-Sale Anodyne F9 0 40 Cc1noc(C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317183 EH On-Demand Anodyne PRCP 58 38 Cc1noc(C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317183 EH On-Demand Anodyne GRM5 24 46 Cc1noc(C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317183 EH On-Demand Anodyne SMO 51 39 Cc1noc(C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317183 EH On-Demand Anodyne ETHR 60 36 COc1cc(F)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1OC ZINC000147317193 GC On-Demand Anodyne SFRP1 41 31 CC[C@@H](N)CC(=O)NN(C)C ZINC000147317230 AB For-Sale Reactive KDM7A 0 42 O=S(=O)(NCc1ccccc1)Nc1ncnc(OCCO)c1-c1ccc(Br)cc1 ZINC000147317290 JF For-Sale Anodyne EDNRB 20 79 O=S(=O)(NCc1ccccc1)Nc1ncnc(OCCO)c1-c1ccc(Br)cc1 ZINC000147317290 JF For-Sale Anodyne EDNRA 36 79 N[C@@H]1C[C@H]1c1cc(F)c(F)cc1F ZINC000147317311 AD For-Sale Anodyne DPP4 45 51 N[C@@H]1C[C@H]1c1cc(F)c(F)cc1F ZINC000147317311 AD For-Sale Anodyne DPP7 0 46 N[C@@H]1C[C@H]1c1cc(F)c(F)cc1F ZINC000147317311 AD For-Sale Anodyne DPP8 0 51 N[C@@H]1C[C@H]1c1cc(F)c(F)cc1F ZINC000147317311 AD For-Sale Anodyne DPP9 0 51 Cc1cc(C)c2oc(-c3cc(N)cc(Br)c3)nc2c1 ZINC000147317317 DI For-Sale Anodyne CETP 0 44 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147317335 EE On-Demand Anodyne CTSS 23 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147317335 EE On-Demand Anodyne EPHX2 57 50 Fc1cc(OCCOc2cccc(Br)c2)ccc1Cl ZINC000147317355 EJ For-Sale Anodyne HMOX2 19 40 COc1cc(F)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1OC ZINC000147317371 GC On-Demand Anodyne SFRP1 41 31 CCOc1ccc(C(=O)N2CC[C@@H](N)[C@@H](CC)C2)cc1 ZINC000147317381 CE On-Demand Anodyne AVPR1A 23 49 CCOc1ccc(C(=O)N2CC[C@@H](N)[C@@H](CC)C2)cc1 ZINC000147317381 CE On-Demand Anodyne L3MBTL1 0 40 CCOc1ccc(C(=O)N2CC[C@@H](N)[C@@H](CC)C2)cc1 ZINC000147317381 CE On-Demand Anodyne L3MBTL3 66 40 O=C(C[C@@H]1CNc2ccccc21)Nc1ncc(Br)s1 ZINC000147317407 EG For-Sale Anodyne FBP1 29 42 O=C(C[C@@H]1CNc2ccccc21)Nc1ncc(Br)s1 ZINC000147317407 EG For-Sale Anodyne CDK5 49 40 CC[C@@H]1CN(C(=O)c2cc(=O)c3ccccc3[nH]2)CCO1 ZINC000147317413 CD On-Demand Anodyne GRIN2B 23 41 CC[C@@H]1CN(C(=O)c2cc(=O)c3ccccc3[nH]2)CCO1 ZINC000147317413 CD On-Demand Anodyne HRH4 23 41 CC[C@@H]1CN(C(=O)c2cc(=O)c3ccccc3[nH]2)CCO1 ZINC000147317413 CD On-Demand Anodyne AKR1C3 17 40 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317414 EH On-Demand Anodyne PRCP 58 38 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317414 EH On-Demand Anodyne GRM5 24 46 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317414 EH On-Demand Anodyne SMO 51 39 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317414 EH On-Demand Anodyne ETHR 60 36 COc1ccc(CCNC2(C(=O)O)CCC2)cc1 ZINC000147317471 BD For-Sale Anodyne MMP1 25 43 CC(C)c1nc(NN)cc(Oc2ccc(Cl)cc2Cl)n1 ZINC000147317474 DH For-Sale Anodyne S1PR4 23 40 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1cccnc1N1CCCC1 ZINC000147317534 GH On-Demand Anodyne KCNQ2 41 33 CCc1ccc2oc(-c3cc(N)cc(Cl)c3)nc2c1 ZINC000147317543 CI For-Sale Anodyne HPSE 44 39 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(C(F)(F)F)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147317563 KK Annotated Anodyne CCR2 43 34 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(C(F)(F)F)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147317563 KK Annotated Anodyne GLP1R 22 51 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(C(F)(F)F)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147317563 KK Annotated Anodyne GIPR 78 45 CC[C@@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@@H]1N ZINC000147317595 CD On-Demand Anodyne CCR5 15 40 CC[C@@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@@H]1N ZINC000147317595 CD On-Demand Anodyne DPP4 18 42 CC[C@@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@@H]1N ZINC000147317595 CD On-Demand Anodyne MLNR 45 47 O=C(C[C@H]1CNc2ccccc21)Nc1ncc(Br)s1 ZINC000147317627 EG For-Sale Anodyne FBP1 29 42 O=C(C[C@H]1CNc2ccccc21)Nc1ncc(Br)s1 ZINC000147317627 EG For-Sale Anodyne CDK5 49 40 CC[C@H]1CN(C(=O)c2cc(=O)c3ccccc3[nH]2)CCO1 ZINC000147317632 CD On-Demand Anodyne GRIN2B 23 41 CC[C@H]1CN(C(=O)c2cc(=O)c3ccccc3[nH]2)CCO1 ZINC000147317632 CD On-Demand Anodyne HRH4 23 41 CC[C@H]1CN(C(=O)c2cc(=O)c3ccccc3[nH]2)CCO1 ZINC000147317632 CD On-Demand Anodyne AKR1C3 17 40 Cc1noc(C2CCN(C(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317647 EH On-Demand Anodyne PRCP 58 38 Cc1noc(C2CCN(C(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317647 EH On-Demand Anodyne GRM5 24 46 Cc1noc(C2CCN(C(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317647 EH On-Demand Anodyne SMO 51 39 Cc1noc(C2CCN(C(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)CC2)n1 ZINC000147317647 EH On-Demand Anodyne ETHR 60 36 Ic1ccc(-c2cnn(CCCc3ccccc3)c2)cc1 ZINC000147317672 GJ For-Sale Anodyne SIGMAR1 21 41 CCCC(=O)Nc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147317687 HF On-Demand Bother TAAR1 24 45 CCCC(=O)Nc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147317687 HF On-Demand Bother KCNK3 98 36 CCCC(=O)Nc1cccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)c1 ZINC000147317687 HF On-Demand Bother KCNK9 59 36 Cc1cc(=O)c(C(=O)Nc2cccc(OCC(N)=O)c2)nn1-c1ccccc1F ZINC000147317692 GD On-Demand Anodyne CTSA 49 36 Cc1cc(=O)c(C(=O)Nc2cccc(OCC(N)=O)c2)nn1-c1ccccc1F ZINC000147317692 GD On-Demand Anodyne KCNK3 42 31 Cc1cc(=O)c(C(=O)Nc2cccc(OCC(N)=O)c2)nn1-c1ccccc1F ZINC000147317692 GD On-Demand Anodyne KCNK9 42 31 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1cccnc1N1CCCC1 ZINC000147317738 GH On-Demand Anodyne KCNQ2 41 33 Cc1cccc(COc2cc(Cn3oc(=O)[nH]c3=O)cc(OCc3cccc(C)c3)c2)c1 ZINC000147317747 IH For-Sale Anodyne MAOB 35 44 C[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@](C)(C(=O)O)C1CC1 ZINC000147317776 DD On-Demand Anodyne PGC 44 33 C[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@](C)(C(=O)O)C1CC1 ZINC000147317776 DD On-Demand Anodyne PAPA1_CARPA 48 38 C[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@](C)(C(=O)O)C1CC1 ZINC000147317776 DD On-Demand Anodyne CTSK 15 41 C[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@](C)(C(=O)O)C1CC1 ZINC000147317776 DD On-Demand Anodyne REN 42 40 C[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@](C)(C(=O)O)C1CC1 ZINC000147317776 DD On-Demand Anodyne FPR1 37 40 CC[C@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@@H]1N ZINC000147317813 CD On-Demand Anodyne CCR5 15 40 CC[C@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@@H]1N ZINC000147317813 CD On-Demand Anodyne DPP4 18 42 CC[C@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@@H]1N ZINC000147317813 CD On-Demand Anodyne MLNR 45 47 COc1ccc2c(c1)OC[C@H](C(=O)N1CCC(c3nc(C)no3)CC1)C2 ZINC000147317850 FE On-Demand Anodyne ETHR 43 41 COc1cccc(C(=O)N2CCC[C@H](CCBr)C2)c1OC ZINC000147317888 FG For-Sale Reactive DRD2 40 41 COc1cccc(C(=O)N2CCC[C@H](CCBr)C2)c1OC ZINC000147317888 FG For-Sale Reactive DRD3 0 40 COc1cccc(C(=O)N2CCC[C@H](CCBr)C2)c1OC ZINC000147317888 FG For-Sale Reactive ACKR3 47 32 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)Cc2ccccc2C)c1 ZINC000147317920 EG On-Demand Bother COLA 95 43 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)Cc2ccccc2C)c1 ZINC000147317920 EG On-Demand Bother AKR1C2 33 44 O=C(O)C1(NCCCOc2ccc(Cl)cc2)CCC1 ZINC000147317921 CF For-Sale Anodyne DRD4 19 51 O=C(O)C1(NCCCOc2ccc(Cl)cc2)CCC1 ZINC000147317921 CF For-Sale Anodyne PLA2G4B 40 31 O=C(O)C1(NCCCOc2ccc(Cl)cc2)CCC1 ZINC000147317921 CF For-Sale Anodyne CVIR 0 41 CCn1c2ccccc2c2cc(NC(=O)C(=O)NC[C@@H]3CCCCO3)ccc21 ZINC000147317936 GG On-Demand Anodyne NPY5R 15 51 Nc1cc(Cl)cc(-c2nc3cc(C(F)(F)F)ccc3o2)c1 ZINC000147317974 DJ For-Sale Anodyne AGPAT2 19 44 CC[C@@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@H]1N ZINC000147318007 CD On-Demand Anodyne CCR5 15 40 CC[C@@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@H]1N ZINC000147318007 CD On-Demand Anodyne DPP4 18 42 CC[C@@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@H]1N ZINC000147318007 CD On-Demand Anodyne MLNR 45 47 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cccnc1N1CCCC1 ZINC000147318019 GH On-Demand Anodyne KCNQ2 41 33 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC(c3nc(C)no3)CC1)C2 ZINC000147318028 FE On-Demand Anodyne ETHR 43 41 COCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147318068 GC On-Demand Anodyne HRH2 18 50 COCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147318068 GC On-Demand Anodyne HRH3 16 50 COCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147318068 GC On-Demand Anodyne MMP13 42 39 COCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147318068 GC On-Demand Anodyne ADAM17 25 40 COCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147318068 GC On-Demand Anodyne MMP7 38 41 COc1cccc(C(=O)N2CCC[C@@H](CCBr)C2)c1OC ZINC000147318109 FG For-Sale Reactive DRD2 40 41 COc1cccc(C(=O)N2CCC[C@@H](CCBr)C2)c1OC ZINC000147318109 FG For-Sale Reactive DRD3 0 40 COc1cccc(C(=O)N2CCC[C@@H](CCBr)C2)c1OC ZINC000147318109 FG For-Sale Reactive ACKR3 47 32 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)Cc2ccccc2C)c1 ZINC000147318130 EG On-Demand Bother COLA 95 43 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)Cc2ccccc2C)c1 ZINC000147318130 EG On-Demand Bother AKR1C2 33 44 CCn1c2ccccc2c2cc(NC(=O)C(=O)NC[C@H]3CCCCO3)ccc21 ZINC000147318133 GG On-Demand Anodyne NPY5R 15 51 C[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@](C)(C(=O)O)C1CC1 ZINC000147318154 DD On-Demand Anodyne PGC 44 33 C[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@](C)(C(=O)O)C1CC1 ZINC000147318154 DD On-Demand Anodyne PAPA1_CARPA 48 38 C[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@](C)(C(=O)O)C1CC1 ZINC000147318154 DD On-Demand Anodyne CTSK 15 41 C[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@](C)(C(=O)O)C1CC1 ZINC000147318154 DD On-Demand Anodyne REN 42 40 C[C@@H](NC(=O)OC(C)(C)C)C(=O)N[C@@](C)(C(=O)O)C1CC1 ZINC000147318154 DD On-Demand Anodyne FPR1 37 40 CC[C@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@H]1N ZINC000147318187 CD On-Demand Anodyne CCR5 15 40 CC[C@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@H]1N ZINC000147318187 CD On-Demand Anodyne DPP4 18 42 CC[C@H]1CN(C(=O)Cc2ccc(F)cc2)CC[C@H]1N ZINC000147318187 CD On-Demand Anodyne MLNR 45 47 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cccnc1N1CCCC1 ZINC000147318194 GH On-Demand Anodyne KCNQ2 41 33 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccccc2F)=NC12CCC(C(C)(C)C)CC2 ZINC000147318201 KK Annotated Anodyne GCGR 48 73 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccccc2F)=NC12CCC(C(C)(C)C)CC2 ZINC000147318201 KK Annotated Anodyne GLP1R 21 49 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccccc2F)=NC12CCC(C(C)(C)C)CC2 ZINC000147318201 KK Annotated Anodyne GIPR 55 39 CC(=O)Nc1ccccc1Oc1cc(N)cc([N+](=O)[O-])c1 ZINC000147318239 CF For-Sale Bother PYGL 31 46 CC(=O)Nc1ccccc1Oc1cc(N)cc([N+](=O)[O-])c1 ZINC000147318239 CF For-Sale Bother PYGM 20 46 CC(=O)Nc1ccccc1Oc1cc(N)cc([N+](=O)[O-])c1 ZINC000147318239 CF For-Sale Bother KCNMA1 18 40 CC[C@@H]1CN(C(=O)C2CCN(C(=O)c3ccc(OC)c4ccccc34)CC2)CCO1 ZINC000147318250 HG On-Demand Anodyne L3MBTL3 23 43 C=C(C(=O)O)C(=O)c1ccc(OCC)cc1 ZINC000147318271 BD Annotated Mild RARB 15 40 C=C(C(=O)O)C(=O)c1ccc(OCC)cc1 ZINC000147318271 BD Annotated Mild PLA2G4B 68 38 CN(C)NC(=O)[C@H]1NCCc2ccccc21 ZINC000147318273 BC For-Sale Reactive PRCP 0 43 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318293 GH On-Demand Anodyne PRCP 41 34 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318293 GH On-Demand Anodyne SMO 50 35 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318293 GH On-Demand Anodyne ETHR 60 36 COCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147318297 GC On-Demand Anodyne HRH2 18 50 COCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147318297 GC On-Demand Anodyne HRH3 16 50 COCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147318297 GC On-Demand Anodyne MMP13 42 39 COCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147318297 GC On-Demand Anodyne ADAM17 25 40 COCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147318297 GC On-Demand Anodyne MMP7 38 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(N2CCCCC2)cc1 ZINC000147318349 EE On-Demand Anodyne TNK2 30 45 O=C(c1ccc2c(c1)OCCO2)N1CCC[C@H](CCBr)C1 ZINC000147318404 FG For-Sale Reactive L3MBTL3 47 35 CC[C@H]1CN(C(=O)C2CCN(C(=O)c3ccc(OC)c4ccccc34)CC2)CCO1 ZINC000147318438 HG On-Demand Anodyne L3MBTL3 23 43 CN(C)NC(=O)[C@@H]1NCCc2ccccc21 ZINC000147318446 BC For-Sale Reactive PRCP 0 43 Cc1noc(C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318466 GH On-Demand Anodyne PRCP 41 34 Cc1noc(C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318466 GH On-Demand Anodyne SMO 50 35 Cc1noc(C2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318466 GH On-Demand Anodyne ETHR 60 36 O=C(c1ccc2c(c1)OCCO2)N1CCC[C@@H](CCBr)C1 ZINC000147318561 FG For-Sale Reactive L3MBTL3 47 35 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(N2CCCCC2)cc1 ZINC000147318572 EE On-Demand Anodyne TNK2 30 45 CN(C)C1(CNC(=O)c2csc(C#CCN)c2)CCCC1 ZINC000147318606 DD For-Sale Mild SLC6A5 16 47 CCCC[C@H](N)C(=O)NN1CCCCC1 ZINC000147318658 BD For-Sale Anodyne DPP7 42 43 CCCC[C@H](N)C(=O)NN1CCCCC1 ZINC000147318658 BD For-Sale Anodyne NOD1 55 34 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318689 GH On-Demand Anodyne PRCP 41 34 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318689 GH On-Demand Anodyne SMO 50 35 Cc1noc(C2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318689 GH On-Demand Anodyne ETHR 60 36 CCCC[C@H](NC(N)=O)C(=O)N(C)Cc1ccc(C(=O)NC2CC2)cc1 ZINC000147318850 FD On-Demand Anodyne PCSK5 40 32 CCCC[C@H](NC(N)=O)C(=O)N(C)Cc1ccc(C(=O)NC2CC2)cc1 ZINC000147318850 FD On-Demand Anodyne SLC6A5 33 41 CCCC[C@@H](N)C(=O)NN1CCCCC1 ZINC000147318882 BD For-Sale Anodyne DPP7 42 43 CCCC[C@@H](N)C(=O)NN1CCCCC1 ZINC000147318882 BD For-Sale Anodyne NOD1 55 34 FC(F)CN[C@@H]1CCCc2cccnc21 ZINC000147318945 BE For-Sale Anodyne CXCR4 72 37 Cc1noc(C2CCN(C(=O)[C@H]3C[C@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318952 GH On-Demand Anodyne PRCP 41 34 Cc1noc(C2CCN(C(=O)[C@H]3C[C@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318952 GH On-Demand Anodyne SMO 50 35 Cc1noc(C2CCN(C(=O)[C@H]3C[C@H]3c3cccc(Br)c3)CC2)n1 ZINC000147318952 GH On-Demand Anodyne ETHR 60 36 CC(=O)c1ccc(O)cc1C(C)C ZINC000147318996 AF For-Sale Anodyne CA7 17 49 Fc1ccc(Cn2cc(-c3ccc(I)cc3)cn2)cc1 ZINC000147318998 GI For-Sale Anodyne ADORA2B 15 43 Fc1ccc(Cn2cc(-c3ccc(I)cc3)cn2)cc1 ZINC000147318998 GI For-Sale Anodyne ALK 0 55 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(C(F)(F)F)cc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147319046 KK Annotated Anodyne MTTP 41 32 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(C(F)(F)F)cc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147319046 KK Annotated Anodyne GLP1R 23 52 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(C(F)(F)F)cc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147319046 KK Annotated Anodyne GIPR 89 46 CCCC[C@@H](NC(N)=O)C(=O)N(C)Cc1ccc(C(=O)NC2CC2)cc1 ZINC000147319063 FD On-Demand Anodyne PCSK5 40 32 CCCC[C@@H](NC(N)=O)C(=O)N(C)Cc1ccc(C(=O)NC2CC2)cc1 ZINC000147319063 FD On-Demand Anodyne SLC6A5 33 41 COc1ccc(Br)cc1COc1ccc(Cl)c(F)c1 ZINC000147319073 EJ For-Sale Anodyne CCR5 16 40 Cc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1C(N)=O ZINC000147319090 GB On-Demand Anodyne CCR8 54 33 Cc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1C(N)=O ZINC000147319090 GB On-Demand Anodyne SFRP1 55 31 Cc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1C(N)=O ZINC000147319090 GB On-Demand Anodyne WNT3 41 30 O=C(Cc1ccc(C(F)(F)F)cc1)Nc1cccc2[nH]c(=O)[nH]c12 ZINC000147319113 EG On-Demand Anodyne KCNQ2 19 40 Cc1noc(C2CCN(C(=O)c3ccc4c(c3)COC4)CC2)n1 ZINC000147319116 DE On-Demand Anodyne SMO 54 37 Cc1noc(C2CCN(C(=O)c3ccc4c(c3)COC4)CC2)n1 ZINC000147319116 DE On-Demand Anodyne L3MBTL3 56 38 Cc1noc(C2CCN(C(=O)c3ccc4c(c3)COC4)CC2)n1 ZINC000147319116 DE On-Demand Anodyne ETHR 59 39 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3cccnc3N3CCCC3)c2)CCO1 ZINC000147319146 HG On-Demand Anodyne TRPV1 20 41 FC(F)CN[C@H]1CCCc2cccnc21 ZINC000147319155 BE For-Sale Anodyne CXCR4 72 37 Cc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1C(N)=O ZINC000147319303 GB On-Demand Anodyne CCR8 54 33 Cc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1C(N)=O ZINC000147319303 GB On-Demand Anodyne SFRP1 55 31 Cc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1C(N)=O ZINC000147319303 GB On-Demand Anodyne WNT3 41 30 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne PPIA 24 40 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne LTA4H 22 40 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne CA1 23 51 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne CHEK2 19 40 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne RAF1 29 46 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne FAAH 23 45 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne CFTR 31 41 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne ACR 26 40 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne F13A1 34 51 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne TAAR1 38 44 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne SIRT2 28 41 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne CRTM 40 42 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne Q25615_ONCVO 29 46 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne KCNK3 53 40 NC(=O)Nc1cccc(Oc2ccc(Cl)cc2)c1 ZINC000147319334 CH In-Stock Anodyne KCNK9 43 35 CCCCCCCCNC(=O)c1ccc(/C=C/C(=O)O)s1 ZINC000147319341 DH For-Sale Mild ASAH1 99 40 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3cccnc3N3CCCC3)c2)CCO1 ZINC000147319355 HG On-Demand Anodyne TRPV1 20 41 CCCCCCCCNC(=O)c1csc(/C=C/C(=O)O)c1 ZINC000147319538 DH For-Sale Mild FOLH1 22 41 CCCCCCCCNC(=O)c1csc(/C=C/C(=O)O)c1 ZINC000147319538 DH For-Sale Mild ASAH1 95 36 Cc1cc(C(=O)N[C@@H](C)c2ccc3c(c2)OCCO3)cc([N+](=O)[O-])c1 ZINC000147319540 EG On-Demand Bother PLK1 15 41 CCNc1nc(Cl)nc(Oc2ccccc2NC(C)=O)n1 ZINC000147319648 DF For-Sale Anodyne PPX1 0 42 CC[C@@H](C)c1ccc([C@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147319656 FK On-Demand Anodyne CYP3A4 15 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cc(F)cc(Br)c1)C2 ZINC000147319666 GG On-Demand Anodyne MTNR1A 18 40 CC[C@@H](C)c1ccc(OCc2cccnc2)cc1 ZINC000147319720 BI On-Demand Anodyne CYP26A1 33 41 Cc1cc(C(=O)N[C@H](C)c2ccc3c(c2)OCCO3)cc([N+](=O)[O-])c1 ZINC000147319733 EG On-Demand Bother PLK1 15 41 CCCCCCCCNC(=O)c1sccc1/C=C/C(=O)O ZINC000147319748 DH For-Sale Mild ASAH1 77 36 CCCCCCCCn1cnc(CCN)c1 ZINC000147319782 BF For-Sale Mild CPB2 53 55 CCCCCCCCn1cnc(CCN)c1 ZINC000147319782 BF For-Sale Mild CPB1 42 52 CCCCCCCCn1cnc(CCN)c1 ZINC000147319782 BF For-Sale Mild Q43014_PRUAV 0 43 COc1ccc(CCC(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147319798 FH For-Sale Reactive GRM3 15 46 COc1ccc(CCC(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147319798 FH For-Sale Reactive MMP1 18 40 Cn1c(-c2ccc(C(=O)c3ccccc3)cc2)ccc(O)c1=O ZINC000147319821 DF For-Sale Anodyne SRD5A2 17 42 Cn1c(-c2ccc(C(=O)c3ccccc3)cc2)ccc(O)c1=O ZINC000147319821 DF For-Sale Anodyne GRM7 72 36 Cn1c([C@@H]2CCCCN2C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)nc2ccccc21 ZINC000147319843 GK On-Demand Anodyne GRM5 15 40 CC[C@H](C)c1ccc([C@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147319875 FK On-Demand Anodyne CYP3A4 15 42 CC(=O)c1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147319928 CD On-Demand Anodyne ADAMTS4 16 42 CC(=O)c1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1 ZINC000147319928 CD On-Demand Anodyne LIMK2 43 38 CC[C@H](C)c1ccc(OCc2cccnc2)cc1 ZINC000147319936 BI On-Demand Anodyne CYP26A1 33 41 CCCCCCCCN1CC[C@H](C)N[C@H](CC)CC1 ZINC000147319969 CI For-Sale Mild SIGMAR1 15 41 CCCCCCCCN1CC[C@H](C)N[C@H](CC)CC1 ZINC000147319969 CI For-Sale Mild GNAI1 0 43 CCCCCCCCN1CC[C@H](C)N[C@H](CC)CC1 ZINC000147319969 CI For-Sale Mild GNAI3 0 43 CCCCCCCCN1CC[C@H](C)N[C@H](CC)CC1 ZINC000147319969 CI For-Sale Mild GNAO1 0 51 CCCCCCCCN1CC[C@H](C)N[C@H](CC)CC1 ZINC000147319969 CI For-Sale Mild ZM.86993 0 41 COc1ccc(CCC(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147319981 FH For-Sale Reactive GRM3 15 46 COc1ccc(CCC(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147319981 FH For-Sale Reactive MMP1 18 40 Fc1cc(OCc2ccc(I)cc2)ccc1Cl ZINC000147320040 FJ For-Sale Anodyne MAOA 15 45 Fc1cc(OCc2ccc(I)cc2)ccc1Cl ZINC000147320040 FJ For-Sale Anodyne MAOB 40 45 Fc1cc(OCc2ccc(I)cc2)ccc1Cl ZINC000147320040 FJ For-Sale Anodyne ACR 19 40 COc1cc2nc(N)n(CCNC(N)=O)c2cc1OC ZINC000147320041 CC For-Sale Anodyne ENPP1 45 30 CC[C@@H](C)c1ccc([C@@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147320053 FK On-Demand Anodyne CYP3A4 15 42 Fc1ccc(F)c(Cn2cc(-c3ccc(I)cc3)cn2)c1 ZINC000147320070 GI For-Sale Anodyne ALK 15 59 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(F)cc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147320089 KK Annotated Anodyne GCGR 52 81 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(F)cc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147320089 KK Annotated Anodyne GLP1R 22 55 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(F)cc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147320089 KK Annotated Anodyne GIPR 77 40 O=C(NC1CCN(C(=O)Nc2cccnc2N2CCCC2)CC1)c1ccoc1 ZINC000147320093 GF On-Demand Anodyne HPGDS 32 40 CCNC(=O)c1ccc(N)c(NCCCCC(C)C)c1 ZINC000147320118 CG For-Sale Anodyne ERAP1 0 44 CCNc1nc2c(ncn2[C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]1 ZINC000147320120 CB For-Sale Anodyne ADA 25 44 CCNc1nc2c(ncn2[C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]1 ZINC000147320120 CB For-Sale Anodyne ADORA1 56 42 CCNc1nc2c(ncn2[C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]1 ZINC000147320120 CB For-Sale Anodyne SLC29A1 33 45 CCNc1nc2c(ncn2[C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]1 ZINC000147320120 CB For-Sale Anodyne TK 55 48 CCNc1nc2c(ncn2[C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]1 ZINC000147320120 CB For-Sale Anodyne TK1 59 48 CCNc1nc2c(ncn2[C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]1 ZINC000147320120 CB For-Sale Anodyne POLB 38 51 CCNc1nc2c(ncn2[C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]1 ZINC000147320120 CB For-Sale Anodyne ADCY5 21 46 CCNc1nc2c(ncn2[C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]1 ZINC000147320120 CB For-Sale Anodyne NS5B 42 50 CCNc1nc2c(ncn2[C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]1 ZINC000147320120 CB For-Sale Anodyne TK2 53 37 CCNc1nc2c(ncn2[C@@H]2C[C@H](O)[C@@H](CO)O2)c(=O)[nH]1 ZINC000147320120 CB For-Sale Anodyne Q4VQ11_PIG 60 36 CC(=O)c1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147320122 CD On-Demand Anodyne ADAMTS4 16 42 CC(=O)c1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1 ZINC000147320122 CD On-Demand Anodyne LIMK2 43 38 CCNc1ncc(F)c(Oc2ccccc2NC(C)=O)n1 ZINC000147320135 CF For-Sale Anodyne P2RY1 29 40 O=C(NC1CCN(Cc2ccncc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147320171 FF On-Demand Anodyne DRD4 22 44 O=C(NC1CCN(Cc2ccncc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147320171 FF On-Demand Anodyne SIGMAR1 25 43 O=C(NC1CCN(Cc2ccncc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147320171 FF On-Demand Anodyne SSTR5 49 39 O=C(NC1CCN(Cc2ccncc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147320171 FF On-Demand Anodyne MCHR1 43 39 CCCCCCCCN1CC[C@@H](C)N[C@H](CC)CC1 ZINC000147320215 CI For-Sale Mild SIGMAR1 15 41 CCCCCCCCN1CC[C@@H](C)N[C@H](CC)CC1 ZINC000147320215 CI For-Sale Mild GNAI1 0 43 CCCCCCCCN1CC[C@@H](C)N[C@H](CC)CC1 ZINC000147320215 CI For-Sale Mild GNAI3 0 43 CCCCCCCCN1CC[C@@H](C)N[C@H](CC)CC1 ZINC000147320215 CI For-Sale Mild GNAO1 0 51 CCCCCCCCN1CC[C@@H](C)N[C@H](CC)CC1 ZINC000147320215 CI For-Sale Mild ZM.86993 0 41 Cn1c([C@@H]2CCCCN2C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)nc2ccccc21 ZINC000147320226 GK On-Demand Anodyne GRM5 15 40 CC[C@H](C)c1ccc([C@@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147320232 FK On-Demand Anodyne CYP3A4 15 42 C[C@H](CNS(=O)(=O)c1ccccc1F)CC(=O)O ZINC000147320341 CD On-Demand Anodyne CTSA 52 33 COc1ccc(Cc2nc3ccccc3c3nc(N)nn23)c(OC)c1 ZINC000147320377 EE Annotated Anodyne DHFR 17 42 COc1ccc(Cc2nc3ccccc3c3nc(N)nn23)c(OC)c1 ZINC000147320377 EE Annotated Anodyne DRTS_TOXGO 35 43 COc1ccc(Cc2nc3ccccc3c3nc(N)nn23)c(OC)c1 ZINC000147320377 EE Annotated Anodyne DYR_PNECA 22 42 COc1ccc(Cc2nc3ccccc3c3nc(N)nn23)c(OC)c1 ZINC000147320377 EE Annotated Anodyne HSP90AB1 19 52 COc1ccc(Cc2nc3ccccc3c3nc(N)nn23)c(OC)c1 ZINC000147320377 EE Annotated Anodyne PDE10A 21 40 CCCCCCCCN1CCCN[C@H](C)CC1 ZINC000147320422 BG For-Sale Mild SIGMAR1 16 46 Cc1nc2ccccc2n1CCNC(=O)N(C)Cc1cscn1 ZINC000147320464 EF On-Demand Anodyne IMDH_CRYPV 27 41 CCOc1ncccc1NC(=O)NCc1cccc(CN2CCO[C@H](C)C2)c1 ZINC000147320478 GG On-Demand Anodyne CCR3 19 40 CCOC(=O)c1cc(O)c(O)cc1O ZINC000147320511 AC For-Sale Clean CA7 22 65 CCOC(=O)c1cc(O)c(O)cc1O ZINC000147320511 AC For-Sale Clean CA14 23 65 CCOC(=O)c1cc(O)c(O)cc1O ZINC000147320511 AC For-Sale Clean HISB 0 42 C[C@@H](CNS(=O)(=O)c1ccccc1F)CC(=O)O ZINC000147320550 CD On-Demand Anodyne CTSA 52 33 CCCCCCCCN1CCCN[C@@H](C)CC1 ZINC000147320620 BG For-Sale Mild SIGMAR1 16 46 COc1ccc2c(c1)OC[C@H](C(=O)N1CCCC[C@H]1c1nc3ccccc3n1C)C2 ZINC000147320645 HH On-Demand Anodyne CPT1A 72 37 COc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1F ZINC000147320673 DG On-Demand Anodyne BMP1 55 36 COc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1F ZINC000147320673 DG On-Demand Anodyne CYP3A4 15 43 O=C1CCc2cc(I)ccc2N1CCCc1ccccc1 ZINC000147320691 GI For-Sale Anodyne SIGMAR1 25 50 O=C1CCc2cc(I)ccc2N1CCCc1ccccc1 ZINC000147320691 GI For-Sale Anodyne ALDH1A1 32 43 CCOc1ncccc1NC(=O)NCc1cccc(CN2CCO[C@@H](C)C2)c1 ZINC000147320692 GG On-Demand Anodyne CCR3 19 40 O=C(NN1CCCCC1)[C@H]1Cc2ccccc2CN1 ZINC000147320778 CD For-Sale Anodyne MC4R 39 42 O=C(NN1CCCCC1)[C@H]1Cc2ccccc2CN1 ZINC000147320778 CD For-Sale Anodyne MC5R 36 40 CCC[C@@H](NC(N)=O)C(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000147320810 EC On-Demand Anodyne DRD4 23 40 CCC[C@@H](NC(N)=O)C(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000147320810 EC On-Demand Anodyne ACHE 17 41 CCC[C@@H](NC(N)=O)C(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000147320810 EC On-Demand Anodyne CHRM3 16 41 CCC[C@@H](NC(N)=O)C(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000147320810 EC On-Demand Anodyne SIGMAR1 28 44 CCC[C@@H](NC(N)=O)C(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000147320810 EC On-Demand Anodyne SSTR5 50 38 CCC[C@@H](NC(N)=O)C(=O)NC1CCN(Cc2ccncc2)CC1 ZINC000147320810 EC On-Demand Anodyne MCHR1 43 39 CCCCCCCCN1CC[C@H](C)NC[C@H](C)C1 ZINC000147320829 CH For-Sale Mild SIGMAR1 15 44 COc1ccc2c(c1)OC[C@H](C(=O)N1CCCC[C@@H]1c1nc3ccccc3n1C)C2 ZINC000147320831 HH On-Demand Anodyne CPT1A 72 37 COc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1F ZINC000147320856 DG On-Demand Anodyne BMP1 55 36 COc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1F ZINC000147320856 DG On-Demand Anodyne CYP3A4 15 43 Oc1c(C(F)(F)F)ccc2ccccc12 ZINC000147320983 BH For-Sale Anodyne KCNJ11 117 43 C#CCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147321026 CD On-Demand Mild CACNA1I 45 35 C#CCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147321026 CD On-Demand Mild HCAR1 0 41 CCCCCCCCN1CC[C@@H](C)NC[C@H](C)C1 ZINC000147321048 CH For-Sale Mild SIGMAR1 15 44 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCCC[C@H]1c1nc3ccccc3n1C)C2 ZINC000147321051 HH On-Demand Anodyne CPT1A 72 37 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)c3ccc(C)c(F)c3)CC2)c1 ZINC000147321095 HF On-Demand Bother SLC6A9 19 40 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)c3ccc(C)c(F)c3)CC2)c1 ZINC000147321095 HF On-Demand Bother TAAR1 23 40 COc1ccc([N+](=O)[O-])c(C(=O)N2CCN(C(=O)c3ccc(C)c(F)c3)CC2)c1 ZINC000147321095 HF On-Demand Bother AKR1C3 19 40 COc1ccccc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147321201 CD On-Demand Anodyne ITGAV 30 51 COc1ccccc1S(=O)(=O)NC[C@@H](C)CC(=O)O ZINC000147321201 CD On-Demand Anodyne GLMU 0 40 Cn1c([C@@H]2CCCCN2C(=O)c2ccc3c(c2)COC3)nc2ccccc21 ZINC000147321259 FH On-Demand Anodyne CPT1A 73 34 CCOC(=O)CCCNC(=O)CNC1(C(=O)O)CCC1 ZINC000147321274 CC For-Sale Anodyne EPHX2 0 40 COC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147321278 GC On-Demand Anodyne HRH2 16 45 COC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147321278 GC On-Demand Anodyne SFRP1 88 34 COC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147321278 GC On-Demand Anodyne WNT3 62 32 OCCCn1cc(CNCC(F)F)nn1 ZINC000147321287 BC For-Sale Anodyne GBA 17 43 CCCNc1cccc(NCCCN(C)C)n1 ZINC000147321304 BE For-Sale Anodyne TERT 15 43 CC[C@H]1CN(C(=O)c2ccccc2NS(=O)(=O)c2cc(F)ccc2F)CCO1 ZINC000147321316 HG On-Demand Anodyne CCR8 52 33 CCCCCCCCN1CC[C@H](CC)NC[C@H](C)C1 ZINC000147321331 CI For-Sale Mild SIGMAR1 15 41 CCCCCCCCN1CC[C@H](CC)NC[C@H](C)C1 ZINC000147321331 CI For-Sale Mild GNAO1 0 44 CCCCCCCCN1CC[C@H](CC)NC[C@H](C)C1 ZINC000147321331 CI For-Sale Mild ZM.86993 0 41 CCOC[C@H](C)NC(=O)Nc1cccnc1OCC ZINC000147321362 CE On-Demand Anodyne P2RY1 52 42 COc1ccccc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147321402 CD On-Demand Anodyne ITGAV 30 51 COc1ccccc1S(=O)(=O)NC[C@H](C)CC(=O)O ZINC000147321402 CD On-Demand Anodyne GLMU 0 40 CCC[C@H](N)C(=O)NN1CCCCC1 ZINC000147321433 AC For-Sale Anodyne DPP7 68 40 CCC[C@H](N)C(=O)NN1CCCCC1 ZINC000147321433 AC For-Sale Anodyne DPP8 0 40 CCC[C@H](N)C(=O)NN1CCCCC1 ZINC000147321433 AC For-Sale Anodyne DPP9 0 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H]1CCCc2ccccc21 ZINC000147321436 DE On-Demand Anodyne CTSK 19 46 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H]1CCCc2ccccc21 ZINC000147321436 DE On-Demand Anodyne HTR6 21 45 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H]1CCCc2ccccc21 ZINC000147321436 DE On-Demand Anodyne CTSV 15 46 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H]1CCCc2ccccc21 ZINC000147321436 DE On-Demand Anodyne NPFFR1 41 30 COC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147321476 GC On-Demand Anodyne HRH2 16 45 COC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147321476 GC On-Demand Anodyne SFRP1 88 34 COC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147321476 GC On-Demand Anodyne WNT3 62 32 CCCCCCCCN1CC[C@@H](CC)NC[C@H](C)C1 ZINC000147321505 CI For-Sale Mild SIGMAR1 15 41 CCCCCCCCN1CC[C@@H](CC)NC[C@H](C)C1 ZINC000147321505 CI For-Sale Mild GNAO1 0 44 CCCCCCCCN1CC[C@@H](CC)NC[C@H](C)C1 ZINC000147321505 CI For-Sale Mild ZM.86993 0 41 NC(=O)[C@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321586 CD For-Sale Anodyne F2 16 42 NC(=O)[C@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321586 CD For-Sale Anodyne ACE 21 41 NC(=O)[C@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321586 CD For-Sale Anodyne TRHR 58 38 NC(=O)[C@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321586 CD For-Sale Anodyne CPT2 43 34 NC(=O)[C@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321586 CD For-Sale Anodyne DPP4 15 50 NC(=O)[C@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321586 CD For-Sale Anodyne PREP 117 41 NC(=O)[C@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321586 CD For-Sale Anodyne PEPD 0 42 C[C@H](CNS(=O)(=O)c1cccc(Cl)c1Cl)CC(=O)O ZINC000147321617 EE On-Demand Anodyne CXCL8 40 31 CCC[C@@H](N)C(=O)NN1CCCCC1 ZINC000147321622 AC For-Sale Anodyne DPP7 68 40 CCC[C@@H](N)C(=O)NN1CCCCC1 ZINC000147321622 AC For-Sale Anodyne DPP8 0 40 CCC[C@@H](N)C(=O)NN1CCCCC1 ZINC000147321622 AC For-Sale Anodyne DPP9 0 40 Cc1ccc(-c2nc(CNC3(C(=O)O)CCC3)no2)cc1 ZINC000147321671 CE For-Sale Anodyne KCNQ1 0 42 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2ccccc2F)CC1 ZINC000147321692 FH On-Demand Anodyne ADRB1 19 47 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2ccccc2F)CC1 ZINC000147321692 FH On-Demand Anodyne HTR1A 29 74 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2ccccc2F)CC1 ZINC000147321692 FH On-Demand Anodyne SLC6A4 25 55 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2ccccc2F)CC1 ZINC000147321692 FH On-Demand Anodyne ADRB3 21 57 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2ccccc2F)CC1 ZINC000147321692 FH On-Demand Anodyne ABCB1 53 40 Cc1cc(Br)cc(S(N)(=O)=O)c1OCCCN1CCCC1 ZINC000147321747 GE For-Sale Anodyne HRH3 53 38 O=C(Nc1ccccc1O)c1cccc2c1OCCN2 ZINC000147321752 CE For-Sale Anodyne KCNMA1 27 40 O=C(Nc1ccccc1O)c1cccc2c1OCCN2 ZINC000147321752 CE For-Sale Anodyne G2YM83_BOTF4 60 34 NC(=O)[C@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147321784 CD For-Sale Anodyne F2 16 42 NC(=O)[C@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147321784 CD For-Sale Anodyne ACE 21 41 NC(=O)[C@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147321784 CD For-Sale Anodyne TRHR 58 38 NC(=O)[C@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147321784 CD For-Sale Anodyne CPT2 43 34 NC(=O)[C@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147321784 CD For-Sale Anodyne DPP4 15 50 NC(=O)[C@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147321784 CD For-Sale Anodyne PREP 117 41 NC(=O)[C@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147321784 CD For-Sale Anodyne PEPD 0 42 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cccc(C#N)c2)C1 ZINC000147321804 EC On-Demand Mild CTSC 17 48 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cccc(C#N)c2)C1 ZINC000147321804 EC On-Demand Mild SFRP1 34 46 CC(C)C[C@@H](N)C(=O)NN1CCCCC1 ZINC000147321843 BC For-Sale Anodyne DNPEP 0 44 CC(C)C[C@@H](N)C(=O)NN1CCCCC1 ZINC000147321843 BC For-Sale Anodyne AMPX_VIBPR 0 52 CC(C)C[C@@H](N)C(=O)NN1CCCCC1 ZINC000147321843 BC For-Sale Anodyne SLC15A2 0 41 COc1ccc(S(=O)(=O)N(CCBr)C2CCCCC2)cc1 ZINC000147321865 GG For-Sale Reactive CHRM2 26 40 COc1ccc(S(=O)(=O)N(CCBr)C2CCCCC2)cc1 ZINC000147321865 GG For-Sale Reactive AVPR1B 30 48 COc1ccc(S(=O)(=O)N(CCBr)C2CCCCC2)cc1 ZINC000147321865 GG For-Sale Reactive BMP1 62 47 COc1ccc(S(=O)(=O)N(CCBr)C2CCCCC2)cc1 ZINC000147321865 GG For-Sale Reactive MMP13 41 44 COc1ccc(S(=O)(=O)N(CCBr)C2CCCCC2)cc1 ZINC000147321865 GG For-Sale Reactive MMP2 26 40 COc1ccc(S(=O)(=O)N(CCBr)C2CCCCC2)cc1 ZINC000147321865 GG For-Sale Reactive MMP3 37 47 COc1ccc(S(=O)(=O)N(CCBr)C2CCCCC2)cc1 ZINC000147321865 GG For-Sale Reactive MMP8 29 41 COc1ccc(S(=O)(=O)N(CCBr)C2CCCCC2)cc1 ZINC000147321865 GG For-Sale Reactive MMP9 38 44 COc1ccc(S(=O)(=O)N(CCBr)C2CCCCC2)cc1 ZINC000147321865 GG For-Sale Reactive MMP12 26 40 COc1ccc(S(=O)(=O)N(CCBr)C2CCCCC2)cc1 ZINC000147321865 GG For-Sale Reactive MMP1 37 44 CN1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147321914 DE On-Demand Anodyne CACNA1H 42 37 CC[C@@H]1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)CCO1 ZINC000147321957 HG On-Demand Anodyne PRTN3 50 38 CC[C@@H]1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)CCO1 ZINC000147321957 HG On-Demand Anodyne CCR8 43 31 CC[C@@H]1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)CCO1 ZINC000147321957 HG On-Demand Anodyne SFRP1 44 33 CC[C@@H]1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)CCO1 ZINC000147321957 HG On-Demand Anodyne WNT3 56 33 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne HTR1A 34 48 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne DRD2 38 62 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne ADRA1D 42 47 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne HTR2A 38 43 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne SLC6A1 76 46 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne ADRA1A 47 47 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne ADRA1B 36 47 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne DRD3 54 62 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne HTR4 44 36 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne HRH3 25 44 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne SIGMAR1 35 46 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne CCR3 30 46 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne SCN2A 16 54 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne CCR5 56 42 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne CHRNA7 26 46 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne EPHX2 23 49 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne CACNA1G 46 42 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne CYP2J2 46 32 O=C(NCCCN1CCCC1)C1CCN(CC(c2ccccc2)c2ccccc2)CC1 ZINC000147321983 HI On-Demand Anodyne TBK1 59 34 NC(=O)[C@@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321991 CD For-Sale Anodyne F2 16 42 NC(=O)[C@@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321991 CD For-Sale Anodyne ACE 21 41 NC(=O)[C@@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321991 CD For-Sale Anodyne TRHR 58 38 NC(=O)[C@@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321991 CD For-Sale Anodyne CPT2 43 34 NC(=O)[C@@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321991 CD For-Sale Anodyne DPP4 15 50 NC(=O)[C@@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321991 CD For-Sale Anodyne PREP 117 41 NC(=O)[C@@H]1CCCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147321991 CD For-Sale Anodyne PEPD 0 42 NCC#Cc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147322004 CG For-Sale Mild MAOB 43 38 CC[C@@H]1CN(C(=O)c2c(F)cccc2F)CC[C@@H]1N ZINC000147322005 CE On-Demand Anodyne CCR5 0 40 CC(C)CNC(=O)c1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147322007 HF On-Demand Bother CA2 16 40 CC(C)CNC(=O)c1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147322007 HF On-Demand Bother F3 91 40 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2cccc(C#N)c2)C1 ZINC000147322020 EC On-Demand Mild CTSC 17 48 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2cccc(C#N)c2)C1 ZINC000147322020 EC On-Demand Mild SFRP1 34 46 CCOc1ncccc1NC(=O)NCc1ccc(S(=O)(=O)N(C)C(C)C)cc1 ZINC000147322040 HF On-Demand Anodyne P2RY1 42 37 CCOc1ncccc1NC(=O)NCc1ccc(S(=O)(=O)N(C)C(C)C)cc1 ZINC000147322040 HF On-Demand Anodyne NAMPT 66 44 CC(C)OC(=O)CCNC(=O)c1ccc(-c2ccc(F)cc2)s1 ZINC000147322155 EH On-Demand Anodyne MAPK11 15 42 CC(C)OC(=O)CCNC(=O)c1ccc(-c2ccc(F)cc2)s1 ZINC000147322155 EH On-Demand Anodyne HSD17B2 38 42 CCCCCCCCN1CC[C@H](C)N[C@H](C)CC1 ZINC000147322161 CH For-Sale Mild SIGMAR1 17 47 CC[C@H]1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)CCO1 ZINC000147322169 HG On-Demand Anodyne PRTN3 50 38 CC[C@H]1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)CCO1 ZINC000147322169 HG On-Demand Anodyne CCR8 43 31 CC[C@H]1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)CCO1 ZINC000147322169 HG On-Demand Anodyne SFRP1 44 33 CC[C@H]1CN(C(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)CCO1 ZINC000147322169 HG On-Demand Anodyne WNT3 56 33 CC[C@H]1CN(C(=O)c2c(F)cccc2F)CC[C@@H]1N ZINC000147322190 CE On-Demand Anodyne CCR5 0 40 CCOC(=O)c1cnc(-c2ccccc2C)nc1 ZINC000147322193 BF For-Sale Anodyne P2RY12 22 40 NC(=O)[C@@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147322194 CD For-Sale Anodyne F2 16 42 NC(=O)[C@@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147322194 CD For-Sale Anodyne ACE 21 41 NC(=O)[C@@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147322194 CD For-Sale Anodyne TRHR 58 38 NC(=O)[C@@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147322194 CD For-Sale Anodyne CPT2 43 34 NC(=O)[C@@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147322194 CD For-Sale Anodyne DPP4 15 50 NC(=O)[C@@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147322194 CD For-Sale Anodyne PREP 117 41 NC(=O)[C@@H]1CCCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147322194 CD For-Sale Anodyne PEPD 0 42 Cc1ccc(CCNCCCN)cc1 ZINC000147322245 AD For-Sale Anodyne GRIA1 53 42 Cc1ccc(CCNCCCN)cc1 ZINC000147322245 AD For-Sale Anodyne S1PR2 16 40 CCOc1ncccc1NC(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147322273 FE On-Demand Anodyne SSTR5 49 37 N[C@@H](C(=O)NN1CCCCC1)c1ccccc1 ZINC000147322284 BD For-Sale Anodyne KCNQ2 53 40 N[C@@H](C(=O)NN1CCCCC1)c1ccccc1 ZINC000147322284 BD For-Sale Anodyne DPP7 31 40 CCCCCCCCN1CC[C@@H](C)N[C@H](C)CC1 ZINC000147322341 CH For-Sale Mild SIGMAR1 17 47 CC[C@@H]1CN(C(=O)c2c(F)cccc2F)CC[C@H]1N ZINC000147322415 CE On-Demand Anodyne CCR5 0 40 CCOC(=O)c1cc(C)nc2c1cnn2-c1ccc(OC)cc1 ZINC000147322424 DF For-Sale Anodyne ADORA1 21 44 CCOC(=O)c1cc(C)nc2c1cnn2-c1ccc(OC)cc1 ZINC000147322424 DF For-Sale Anodyne NPBWR1 101 45 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ncccn2)CC1 ZINC000147322427 FD On-Demand Anodyne ADRB2 50 54 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ncccn2)CC1 ZINC000147322427 FD On-Demand Anodyne ADRB1 0 54 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ncccn2)CC1 ZINC000147322427 FD On-Demand Anodyne HTR1A 25 56 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ncccn2)CC1 ZINC000147322427 FD On-Demand Anodyne SLC6A4 22 46 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ncccn2)CC1 ZINC000147322427 FD On-Demand Anodyne ADRB3 50 54 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ncccn2)CC1 ZINC000147322427 FD On-Demand Anodyne ABCB1 60 43 CC[C@@H](C)Oc1cccc(NC(=O)c2c[nH]nc2C(C)(C)C)c1 ZINC000147322445 DI On-Demand Anodyne KCNK3 76 40 CC[C@@H](C)Oc1cccc(NC(=O)c2c[nH]nc2C(C)(C)C)c1 ZINC000147322445 DI On-Demand Anodyne KCNK9 65 40 O=C(O)C1(NCCOc2ccccc2)CCC1 ZINC000147322544 BD For-Sale Anodyne LTA4H 22 42 CCCCCCCCN1CC[C@H](C)N[C@@H](C)CC1 ZINC000147322578 CH For-Sale Mild SIGMAR1 17 47 NCC(=O)c1ccccc1C(=O)O ZINC000147322606 AC For-Sale Anodyne SLC1A6 44 28 NCC(=O)c1ccccc1C(=O)O ZINC000147322606 AC For-Sale Anodyne SLC1A7 44 28 NCC(=O)c1ccccc1C(=O)O ZINC000147322606 AC For-Sale Anodyne AKR1C2 42 41 CC(C)CCCCNCCCN ZINC000147322614 AD For-Sale Anodyne PAOX 19 45 CC(C)CCCCNCCCN ZINC000147322614 AD For-Sale Anodyne DHPS 44 38 CC(C)CCCCNCCCN ZINC000147322614 AD For-Sale Anodyne APHA 47 39 CC[C@H]1CN(C(=O)c2c(F)cccc2F)CC[C@H]1N ZINC000147322630 CE On-Demand Anodyne CCR5 0 40 CC[C@H](C)Oc1cccc(NC(=O)c2c[nH]nc2C(C)(C)C)c1 ZINC000147322656 DI On-Demand Anodyne F2R 15 40 CC[C@H](C)Oc1cccc(NC(=O)c2c[nH]nc2C(C)(C)C)c1 ZINC000147322656 DI On-Demand Anodyne KCNK3 76 40 CC[C@H](C)Oc1cccc(NC(=O)c2c[nH]nc2C(C)(C)C)c1 ZINC000147322656 DI On-Demand Anodyne KCNK9 65 40 O=C(CNC1CCCC1)NN1CCCCC1 ZINC000147322700 BD For-Sale Anodyne DPP7 19 45 O=C1c2ccccc2C(=O)N1CCNC1(C(=O)O)CCC1 ZINC000147322786 CC For-Sale Anodyne HEXB 0 42 O=C1c2ccccc2C(=O)N1CCNC1(C(=O)O)CCC1 ZINC000147322786 CC For-Sale Anodyne HEXA 0 42 COCc1nc(C(=O)N2CCN(Cc3ccccc3C)CC2)cs1 ZINC000147322824 EF On-Demand Anodyne TRPC6 62 35 CC[C@@H]1CN(C(=O)c2cc(C)ccc2C)CC[C@@H]1N ZINC000147322844 CF On-Demand Anodyne L3MBTL1 0 40 CC[C@@H]1CN(C(=O)c2cc(C)ccc2C)CC[C@@H]1N ZINC000147322844 CF On-Demand Anodyne L3MBTL3 15 40 CC[C@H]1CN(C(=O)CCNc2ccc(S(N)(=O)=O)cc2[N+](=O)[O-])CCO1 ZINC000147322881 GC On-Demand Bother BCL2L1 21 41 CC[C@H]1CN(C(=O)CCNc2ccc(S(N)(=O)=O)cc2[N+](=O)[O-])CCO1 ZINC000147322881 GC On-Demand Bother BCL2 20 41 CC[C@H]1CN(C(=O)CCNc2ccc(S(N)(=O)=O)cc2[N+](=O)[O-])CCO1 ZINC000147322881 GC On-Demand Bother CCR8 51 35 Cc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1F ZINC000147322886 CD On-Demand Anodyne TBXA2R 48 35 Cc1ccc(S(=O)(=O)NC[C@@H](C)CC(=O)O)cc1F ZINC000147322886 CD On-Demand Anodyne LEF 64 40 CCOc1nc(N)nc(Oc2ccccc2NC(C)=O)n1 ZINC000147322915 CD For-Sale Anodyne INHA 15 41 CCCCCCCCCCCCNC1(C(=O)O)CCC1 ZINC000147322961 CJ For-Sale Mild CES2 34 42 CCCCCCCCCCCCNC1(C(=O)O)CCC1 ZINC000147322961 CJ For-Sale Mild EST1_PIG 50 35 CCCCCCCCCCCCNC1(C(=O)O)CCC1 ZINC000147322961 CJ For-Sale Mild CES2C 40 42 CCCCCCCCCCCCNC1(C(=O)O)CCC1 ZINC000147322961 CJ For-Sale Mild JHE 0 42 COc1cc(OC)c(CNC(=O)c2cccc(I)c2)c(OC)c1 ZINC000147323016 IG On-Demand Anodyne DRD4 49 37 COc1cc(OC)c(CNC(=O)c2cccc(I)c2)c(OC)c1 ZINC000147323016 IG On-Demand Anodyne CYP1B1 15 42 COc1cc(OC)c(CNC(=O)c2cccc(I)c2)c(OC)c1 ZINC000147323016 IG On-Demand Anodyne ROCK2 15 42 COc1cc(OC)c(CNC(=O)c2cccc(I)c2)c(OC)c1 ZINC000147323016 IG On-Demand Anodyne MT-ND1 17 40 COc1cc(OC)c(CNC(=O)c2cccc(I)c2)c(OC)c1 ZINC000147323016 IG On-Demand Anodyne KCNK3 40 34 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)NC3CCCCC3)cc2C)c1 ZINC000147323026 HI On-Demand Bother MAPK11 31 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)NC3CCCCC3)cc2C)c1 ZINC000147323026 HI On-Demand Bother MAPK14 26 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)NC3CCCCC3)cc2C)c1 ZINC000147323026 HI On-Demand Bother TAAR1 24 42 c1nc(N[C@H]2CC[C@@H](N3CCOCC3)CC2)c2c3c(sc2n1)CCC3 ZINC000147323029 FG Annotated Anodyne IRAK4 20 63 COCc1nc(C(=O)N2CCN(Cc3cccc(Cl)c3)CC2)cs1 ZINC000147323037 FF On-Demand Anodyne TRPC6 48 37 CC(C)CCCCNc1cc2c(cc1N)NC(=O)CC2 ZINC000147323050 CG For-Sale Anodyne PKM 36 40 Cc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1F ZINC000147323060 CD On-Demand Anodyne TBXA2R 48 35 Cc1ccc(S(=O)(=O)NC[C@H](C)CC(=O)O)cc1F ZINC000147323060 CD On-Demand Anodyne LEF 64 40 CC[C@H]1CN(C(=O)c2cc(C)ccc2C)CC[C@@H]1N ZINC000147323062 CF On-Demand Anodyne L3MBTL1 0 40 CC[C@H]1CN(C(=O)c2cc(C)ccc2C)CC[C@@H]1N ZINC000147323062 CF On-Demand Anodyne L3MBTL3 15 40 O=C(c1cc2ccccc2nc1O)N1CC[C@H](c2ccc(Cl)cc2)C1 ZINC000147323169 FI On-Demand Anodyne CCR1 45 43 O=C(c1cc2ccccc2nc1O)N1CC[C@H](c2ccc(Cl)cc2)C1 ZINC000147323169 FI On-Demand Anodyne SMO 41 39 Cc1nc(-c2ccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)cc2)oc1C ZINC000147323178 GK On-Demand Anodyne PRNP 44 34 Cc1nc(-c2ccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)cc2)oc1C ZINC000147323178 GK On-Demand Anodyne MAPK10 17 40 Cc1nc(-c2ccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)cc2)oc1C ZINC000147323178 GK On-Demand Anodyne NR2E3 61 35 Cc1nc(-c2ccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)cc2)oc1C ZINC000147323178 GK On-Demand Anodyne SMO 19 52 O=C(CNC1(C(=O)O)CCC1)Nc1ccc(F)c(Cl)c1 ZINC000147323222 DE For-Sale Anodyne SLC1A1 34 43 O=C(CNC1(C(=O)O)CCC1)Nc1ccc(F)c(Cl)c1 ZINC000147323222 DE For-Sale Anodyne SLC1A2 39 43 O=C(CNC1(C(=O)O)CCC1)Nc1ccc(F)c(Cl)c1 ZINC000147323222 DE For-Sale Anodyne ERBB4 40 34 O=C(CNC1(C(=O)O)CCC1)Nc1ccc(F)c(Cl)c1 ZINC000147323222 DE For-Sale Anodyne ENV 44 36 O=C(CNC1(C(=O)O)CCC1)Nc1ccc(F)c(Cl)c1 ZINC000147323222 DE For-Sale Anodyne MCHR1 25 51 CCC(C)(C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147323237 CG On-Demand Anodyne HCAR1 0 40 CC[C@H]1CN(C(=O)c2ccccc2NS(=O)(=O)c2cccc([N+](=O)[O-])c2)CCO1 ZINC000147323273 HF On-Demand Bother PRTN3 44 34 CC[C@@H]1CN(C(=O)c2cc(C)ccc2C)CC[C@H]1N ZINC000147323291 CF On-Demand Anodyne L3MBTL1 0 40 CC[C@@H]1CN(C(=O)c2cc(C)ccc2C)CC[C@H]1N ZINC000147323291 CF On-Demand Anodyne L3MBTL3 15 40 CCOc1ncccc1NC(=O)NC[C@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147323347 GG On-Demand Anodyne TRPV1 17 40 CCOc1ncccc1NC(=O)NC[C@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147323347 GG On-Demand Anodyne P2RY1 58 53 CCOc1ncccc1NC(=O)NC[C@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147323347 GG On-Demand Anodyne PDS 69 44 O=C(c1cc2ccccc2nc1O)N1CC[C@@H](c2ccc(Cl)cc2)C1 ZINC000147323371 FI On-Demand Anodyne CCR1 45 43 O=C(c1cc2ccccc2nc1O)N1CC[C@@H](c2ccc(Cl)cc2)C1 ZINC000147323371 FI On-Demand Anodyne SMO 41 39 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(F)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147323385 KK Annotated Anodyne GCGR 52 81 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(F)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147323385 KK Annotated Anodyne GLP1R 21 52 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(F)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147323385 KK Annotated Anodyne GIPR 64 39 O=C(Nc1cc(Br)cc(C(=O)O)c1)Nc1nccs1 ZINC000147323445 EG For-Sale Anodyne MAP 0 41 O=C(Nc1cc(Br)cc(C(=O)O)c1)Nc1nccs1 ZINC000147323445 EG For-Sale Anodyne MAP1 97 37 CC[C@H]1CN(C(=O)c2cc(C)ccc2C)CC[C@H]1N ZINC000147323485 CF On-Demand Anodyne L3MBTL1 0 40 CC[C@H]1CN(C(=O)c2cc(C)ccc2C)CC[C@H]1N ZINC000147323485 CF On-Demand Anodyne L3MBTL3 15 40 CCOc1ncccc1NC(=O)NC[C@@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147323561 GG On-Demand Anodyne TRPV1 17 40 CCOc1ncccc1NC(=O)NC[C@@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147323561 GG On-Demand Anodyne P2RY1 58 53 CCOc1ncccc1NC(=O)NC[C@@H](O)COc1cccc(C(F)(F)F)c1 ZINC000147323561 GG On-Demand Anodyne PDS 69 44 CC(C)CCN(C(=O)C[C@@H]1CNc2ccccc21)C1CC1 ZINC000147323607 CH For-Sale Anodyne MBTPS1 47 30 O=C(Nc1cc(Cl)cc(C(=O)O)c1)Nc1nccs1 ZINC000147323622 CG For-Sale Anodyne PPIA 19 41 O=C(Nc1cc(Cl)cc(C(=O)O)c1)Nc1nccs1 ZINC000147323622 CG For-Sale Anodyne MAP 0 47 O=C(Nc1cc(Cl)cc(C(=O)O)c1)Nc1nccs1 ZINC000147323622 CG For-Sale Anodyne MAP1 107 37 CCCCCCCCN1C[C@@H](C)CNC[C@@H](C)C1 ZINC000147323644 CH For-Sale Mild SIGMAR1 16 56 CCCCCCCCN1C[C@@H](C)CNC[C@@H](C)C1 ZINC000147323644 CH For-Sale Mild Q2TU57_MAIZE 15 56 CC[C@@H]1CN(C(=O)c2cc(C)cc(C)c2)CC[C@@H]1N ZINC000147323675 CF On-Demand Anodyne L3MBTL3 52 35 C[C@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccccc1 ZINC000147323681 CD For-Sale Anodyne ACACA 44 38 C[C@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccccc1 ZINC000147323681 CD For-Sale Anodyne CTSK 29 43 C[C@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccccc1 ZINC000147323681 CD For-Sale Anodyne F7 17 43 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccccc2OC(F)(F)F)C1 ZINC000147323698 HD On-Demand Anodyne CCR8 54 35 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccccc2OC(F)(F)F)C1 ZINC000147323698 HD On-Demand Anodyne SFRP1 132 37 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccccc2OC(F)(F)F)C1 ZINC000147323698 HD On-Demand Anodyne WNT3 89 36 OCC#Cc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147323739 CG For-Sale Mild MAOB 52 41 OCC#Cc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147323739 CG For-Sale Mild GYS1 64 39 CC(C)CCN(C(=O)C[C@H]1CNc2ccccc21)C1CC1 ZINC000147323795 CH For-Sale Anodyne MBTPS1 47 30 CCCCCCCCN1C[C@@H](C)CNC[C@H](C)C1 ZINC000147323821 CH For-Sale Mild SIGMAR1 16 56 CCCCCCCCN1C[C@@H](C)CNC[C@H](C)C1 ZINC000147323821 CH For-Sale Mild Q2TU57_MAIZE 15 56 C[C@@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccccc1 ZINC000147323839 CD For-Sale Anodyne ACACA 44 38 C[C@@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccccc1 ZINC000147323839 CD For-Sale Anodyne CTSK 29 43 C[C@@H](NC(=O)CNC1(C(=O)O)CCC1)c1ccccc1 ZINC000147323839 CD For-Sale Anodyne F7 17 43 CC[C@H]1CN(C(=O)c2cc(C)cc(C)c2)CC[C@@H]1N ZINC000147323841 CF On-Demand Anodyne L3MBTL3 52 35 CCNc1cc(Oc2ccc(C)cc2OC)nc(N)n1 ZINC000147323855 CF For-Sale Anodyne AGPAT2 40 35 CC(C)CCCCNCc1ccc(N2CCCCC2)cc1 ZINC000147323862 CJ For-Sale Clean DPP7 47 39 CC(C)CCCCNCc1ccc(N2CCCCC2)cc1 ZINC000147323862 CJ For-Sale Clean LEF 58 34 CCOc1ncccc1NC(=O)NCc1ccc(-n2ccnc2C)c(F)c1 ZINC000147323907 FG On-Demand Anodyne P2RY1 46 44 COC(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147323951 GC On-Demand Anodyne HRH2 15 40 COC(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147323951 GC On-Demand Anodyne SFRP1 93 39 COC(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147323951 GC On-Demand Anodyne WNT3 71 33 CC1(C)CCC[C@@]2(C)[C@@H]1CC[C@@](C)(O)[C@H]2CO ZINC000147323970 BF Annotated Anodyne UGT2B7 73 40 Cc1cc(Br)cc(S(N)(=O)=O)c1OCCn1ccnc1 ZINC000147323993 FD For-Sale Anodyne TBXAS1 24 42 CC[C@@H]1CN(C(=O)c2cc(C)cc(C)c2)CC[C@H]1N ZINC000147324024 CF On-Demand Anodyne L3MBTL3 52 35 COc1cc2ncc(Br)c(Cl)c2cc1OC ZINC000147324042 DH For-Sale Anodyne EGFR 28 43 COc1cc2ncc(Br)c(Cl)c2cc1OC ZINC000147324042 DH For-Sale Anodyne SRC 34 47 COc1cc2ncc(Br)c(Cl)c2cc1OC ZINC000147324042 DH For-Sale Anodyne PDPK1 41 41 COc1cc2ncc(Br)c(Cl)c2cc1OC ZINC000147324042 DH For-Sale Anodyne CSF1R 32 42 CCCCCCCCN1C[C@H](C)CNC[C@@H](C)C1 ZINC000147324043 CH For-Sale Mild SIGMAR1 16 56 CCCCCCCCN1C[C@H](C)CNC[C@@H](C)C1 ZINC000147324043 CH For-Sale Mild Q2TU57_MAIZE 15 56 CC(C)(C)C[C@H]1N[C@@H](C(=O)NCCCN2CCN(C3CC3)CC2)[C@H](c2cccc(Cl)c2F)[C@@]12C(=O)Nc1cc(Cl)ccc12 ZINC000147324090 KK Annotated Anodyne MDM2 101 80 Cc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147324111 CD For-Sale Anodyne CCKAR 24 42 Cc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147324111 CD For-Sale Anodyne F12 0 41 Cc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147324111 CD For-Sale Anodyne ACAT 0 51 Cc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147324111 CD For-Sale Anodyne KCNK3 84 43 Cc1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147324111 CD For-Sale Anodyne KCNK9 51 43 COc1ccc(C)cc1[C@@H](C)NC(=O)N(C)Cc1cscn1 ZINC000147324119 DG On-Demand Anodyne BMP1 53 34 COC(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147324126 GC On-Demand Anodyne HRH2 15 40 COC(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147324126 GC On-Demand Anodyne SFRP1 93 39 COC(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147324126 GC On-Demand Anodyne WNT3 71 33 O=S(=O)(c1ccccc1Cl)N1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000147324184 ED On-Demand Anodyne CCR1 18 48 O=S(=O)(c1ccccc1Cl)N1CCN([C@H]2CCC[C@@H]2O)CC1 ZINC000147324184 ED On-Demand Anodyne SLC18A3 58 44 CCC[C@@H](NC(N)=O)C(=O)N1CCC(Oc2cccc3c2OC(C)(C)C3)CC1 ZINC000147324230 GF On-Demand Anodyne GHRHR 44 30 CCC[C@@H](NC(N)=O)C(=O)N1CCC(Oc2cccc3c2OC(C)(C)C3)CC1 ZINC000147324230 GF On-Demand Anodyne P2RY12 135 37 CCC[C@@H](NC(N)=O)C(=O)N1CCC(Oc2cccc3c2OC(C)(C)C3)CC1 ZINC000147324230 GF On-Demand Anodyne TRY2_BOVIN 40 34 CCC[C@@H](NC(N)=O)C(=O)N1CCC(Oc2cccc3c2OC(C)(C)C3)CC1 ZINC000147324230 GF On-Demand Anodyne ST14 47 33 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(-n3cncn3)c(F)c1)C2 ZINC000147324238 FF On-Demand Anodyne ROCK2 29 47 C[C@@H]1CCCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147324274 CG On-Demand Anodyne HRH3 0 40 C[C@@H]1CCCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147324274 CG On-Demand Anodyne CACNA1I 46 34 CC[C@H]1CN(C(=O)c2cc(C)cc(C)c2)CC[C@H]1N ZINC000147324283 CF On-Demand Anodyne L3MBTL3 52 35 CCCCCCCCn1c(C)c(C(=O)O)c(C)cc1=O ZINC000147324297 CH For-Sale Mild THRB 40 39 CCCCCCCCn1c(C)c(C(=O)O)c(C)cc1=O ZINC000147324297 CH For-Sale Mild POLC 49 34 COc1ccc(C)cc1[C@H](C)NC(=O)N(C)Cc1cscn1 ZINC000147324317 DG On-Demand Anodyne BMP1 53 34 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147324320 KK Annotated Anodyne CCKBR 43 38 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147324320 KK Annotated Anodyne GLP1R 23 60 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147324320 KK Annotated Anodyne MDM2 61 32 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147324320 KK Annotated Anodyne GIPR 72 43 C=CCCOCC(=O)Nc1ccc(NC(=O)c2cccnc2)c(OC)c1 ZINC000147324366 FF On-Demand Mild GRM4 18 41 C=CCCOCC(=O)Nc1ccc(NC(=O)c2cccnc2)c(OC)c1 ZINC000147324366 FF On-Demand Mild ENPP1 57 35 OCCC#Cc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147324369 DH For-Sale Mild MAOB 44 39 OCCC#Cc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147324369 DH For-Sale Mild GYS1 53 36 Cc1cc(Br)cc(S(N)(=O)=O)c1OCCCn1ccnc1 ZINC000147324397 FE For-Sale Anodyne TBXAS1 33 40 Cc1cc(Br)cc(S(N)(=O)=O)c1OCCCn1ccnc1 ZINC000147324397 FE For-Sale Anodyne HMOX2 19 43 C[C@H]1CCCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147324464 CG On-Demand Anodyne HRH3 0 40 C[C@H]1CCCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147324464 CG On-Demand Anodyne CACNA1I 46 34 NNc1cc(Oc2ccc(C(N)=O)cc2)nc(C2CC2)n1 ZINC000147324482 CD For-Sale Anodyne ST14 25 42 COc1cccc(-n2ccnc2SCC(=O)Nc2ccc(SC)cc2)c1 ZINC000147324505 GI On-Demand Anodyne MTNR1A 18 44 COc1cccc(-n2ccnc2SCC(=O)Nc2ccc(SC)cc2)c1 ZINC000147324505 GI On-Demand Anodyne MTNR1B 24 41 COc1cccc(-n2ccnc2SCC(=O)Nc2ccc(SC)cc2)c1 ZINC000147324505 GI On-Demand Anodyne ENPP1 76 40 COc1cccc(-n2ccnc2SCC(=O)Nc2ccc(SC)cc2)c1 ZINC000147324505 GI On-Demand Anodyne FAS 41 40 CCCN(CC(=O)N(C)C)C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147324548 DF On-Demand Anodyne MDM2 47 33 CNc1cn2ccnc2c(Oc2ccc(C)cc2OC)n1 ZINC000147324550 CF For-Sale Anodyne SYK 29 40 CNc1cn2ccnc2c(Oc2ccc(C)cc2OC)n1 ZINC000147324550 CF For-Sale Anodyne HIVRT 0 47 CCOc1ccccc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147324551 CD For-Sale Anodyne HCN1 52 35 CCOc1ccccc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147324551 CD For-Sale Anodyne HCN4 44 34 CCOc1ncccc1NC(=O)NC[C@@H]1CCCO[C@@H]1c1ccccc1 ZINC000147324557 FH On-Demand Anodyne P2RY1 42 36 FC(F)CNCc1c[nH]c2ccccc12 ZINC000147324576 BF For-Sale Anodyne MPO 79 47 FC(F)CNCc1c[nH]c2ccccc12 ZINC000147324576 BF For-Sale Anodyne SLC15A2 0 40 CC[C@H](CNS(=O)(=O)c1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147324579 DD On-Demand Bother MMP2 18 47 Cc1ccc2nc(NCC3(N(C)C)CCCC3)sc2c1 ZINC000147324610 CH For-Sale Anodyne CSNK1D 18 40 O=S(=O)(c1ccccc1Cl)N1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000147324665 ED On-Demand Anodyne CCR1 18 48 O=S(=O)(c1ccccc1Cl)N1CCN([C@@H]2CCC[C@H]2O)CC1 ZINC000147324665 ED On-Demand Anodyne SLC18A3 58 44 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2cccc(C)n2)CC1 ZINC000147324696 FD On-Demand Anodyne P2RY12 178 37 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2cccc(C)n2)CC1 ZINC000147324696 FD On-Demand Anodyne TRY2_BOVIN 52 36 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2cccc(C)n2)CC1 ZINC000147324696 FD On-Demand Anodyne ST14 73 34 CC(C)OCc1ccc(C(=O)NCc2ccccc2OC(F)(F)F)cc1 ZINC000147324705 FI On-Demand Anodyne PPARA 18 44 CC(C)OCc1ccc(C(=O)NCc2ccccc2OC(F)(F)F)cc1 ZINC000147324705 FI On-Demand Anodyne GRIN2B 19 47 CC(C)OCc1ccc(C(=O)NCc2ccccc2OC(F)(F)F)cc1 ZINC000147324705 FI On-Demand Anodyne PPARD 24 45 CC(C)OCc1ccc(C(=O)NCc2ccccc2OC(F)(F)F)cc1 ZINC000147324705 FI On-Demand Anodyne KCNK9 25 40 O=C(O)C1(NCC23CC4CC(CC(C4)C2)C3)CCC1 ZINC000147324753 CF For-Sale Anodyne P2RX7 0 43 CCOc1ncccc1NC(=O)NC[C@H]1CCCO[C@@H]1c1ccccc1 ZINC000147324757 FH On-Demand Anodyne P2RY1 42 36 CCCN(CC(=O)N(C)C)C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147324762 DF On-Demand Anodyne MDM2 47 33 CCNc1ncc(Cl)c(Oc2ccc(C)cc2OC)n1 ZINC000147324783 CH For-Sale Anodyne P2RX2 49 32 CC[C@@H](CNS(=O)(=O)c1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147324795 DD On-Demand Bother MMP2 18 47 COc1ccc2nc(NCC3(N(C)C)CCCC3)sc2c1 ZINC000147324860 DH For-Sale Anodyne CSNK1D 33 49 COc1ccc2nc(NCC3(N(C)C)CCCC3)sc2c1 ZINC000147324860 DH For-Sale Anodyne LUCI_PHOPE 31 40 COc1ccc2nc(NCC3(N(C)C)CCCC3)sc2c1 ZINC000147324860 DH For-Sale Anodyne ISPD 0 43 O=S(=O)(c1ccccc1Cl)N1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000147324877 ED On-Demand Anodyne CCR1 18 48 O=S(=O)(c1ccccc1Cl)N1CCN([C@H]2CCC[C@H]2O)CC1 ZINC000147324877 ED On-Demand Anodyne SLC18A3 58 44 CC(C)CCCCNc1cc(C(N)=O)ccc1N ZINC000147324917 BF For-Sale Anodyne ERAP1 0 40 O=C(NCc1nnc2ccc(C(F)(F)F)cn12)c1ccc(-n2cnc3ccccc32)cc1 ZINC000147324932 II On-Demand Anodyne F9 47 44 O=C(NCc1nnc2ccc(C(F)(F)F)cn12)c1ccc(-n2cnc3ccccc32)cc1 ZINC000147324932 II On-Demand Anodyne HPGD 23 40 O=C(NCc1ccco1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147324933 CF On-Demand Anodyne PPIA 16 42 CCCCCCCCn1cnc(C(=O)OCC)c1N ZINC000147324935 CG For-Sale Mild ADA 40 36 CCCN(CC(=O)N(C)C)C(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147324953 DF On-Demand Anodyne MDM2 47 33 CCOc1ncccc1NC(=O)NC[C@@H]1CCCO[C@H]1c1ccccc1 ZINC000147324957 FH On-Demand Anodyne P2RY1 42 36 COc1ccc(C(C)=O)cc1CNC1(C(=O)O)CCC1 ZINC000147324968 CD For-Sale Anodyne MT-ND1 15 40 COc1ccc(C(C)=O)cc1CNC1(C(=O)O)CCC1 ZINC000147324968 CD For-Sale Anodyne QRFPR 40 35 CCCNc1cc(Oc2ccc(C)cc2OC)nc(N)n1 ZINC000147325022 CF For-Sale Anodyne AGPAT2 46 36 O=S(=O)(c1ccccc1Cl)N1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000147325107 ED On-Demand Anodyne CCR1 18 48 O=S(=O)(c1ccccc1Cl)N1CCN([C@@H]2CCC[C@@H]2O)CC1 ZINC000147325107 ED On-Demand Anodyne SLC18A3 58 44 CC(C)CCCCNCc1ccccc1Cl ZINC000147325134 BI For-Sale Anodyne LEF 45 37 COc1ccc(C(=O)c2cc(NCCC(F)(F)F)c3ncc(-c4ccc(C(=O)NC5CC5)c(C)c4)n3n2)cc1F ZINC000147325154 KK Annotated Anodyne MAPK13 70 36 CCOc1ncccc1NC(=O)NC[C@H]1CCCO[C@H]1c1ccccc1 ZINC000147325162 FH On-Demand Anodyne P2RY1 42 36 CCCc1ccc([C@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147325181 EJ On-Demand Anodyne CYP3A4 16 43 CC[C@H]1CN(C(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)CCO1 ZINC000147325185 GI On-Demand Anodyne UGCG 39 46 CC[C@H]1CN(C(=O)c2cccnc2Oc2ccc(Cl)cc2Cl)CCO1 ZINC000147325185 GI On-Demand Anodyne GPBAR1 44 49 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2ccc(C)cn2)CC1 ZINC000147325191 FD On-Demand Anodyne P2RY12 104 34 N#C[C@@H](Cl)CC(=O)c1ccccc1 ZINC000147325280 AE For-Sale Reactive PLAUR 22 68 N#C[C@@H](Cl)CC(=O)c1ccccc1 ZINC000147325280 AE For-Sale Reactive KMO 0 40 CN1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147325345 CD On-Demand Anodyne CACNA1H 48 38 CN1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147325345 CD On-Demand Anodyne HTR1D 15 42 CN1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147325345 CD On-Demand Anodyne HRH4 26 41 CN1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147325345 CD On-Demand Anodyne CACNA1I 45 35 CN1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147325345 CD On-Demand Anodyne HCAR1 0 40 CCCc1ccc([C@@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147325366 EJ On-Demand Anodyne BMP1 48 34 CCCc1ccc([C@@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147325366 EJ On-Demand Anodyne CYP3A4 16 43 COc1cc(C(=O)CCCC2CCCC2)c(OC)cc1C ZINC000147325438 CJ For-Sale Anodyne HTR4 40 50 Cc1cc(Br)cc(S(N)(=O)=O)c1OCCN1CCCC1 ZINC000147325441 FD For-Sale Anodyne LTA4H 27 40 N#C[C@H](Cl)CC(=O)c1ccccc1 ZINC000147325487 AE For-Sale Reactive PLAUR 22 68 N#C[C@H](Cl)CC(=O)c1ccccc1 ZINC000147325487 AE For-Sale Reactive KMO 0 40 C=CCCOCC(=O)Nc1cccc(OCc2ccccn2)c1 ZINC000147325488 DG On-Demand Mild GRM4 15 41 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1)C(=O)C2 ZINC000147325550 GC On-Demand Anodyne CA5B 27 47 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1)C(=O)C2 ZINC000147325550 GC On-Demand Anodyne CA5A 30 47 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1)C(=O)C2 ZINC000147325550 GC On-Demand Anodyne CXCR3 15 46 COC(=O)c1cc2c(O)cccc2s1 ZINC000147325563 BE In-Stock Anodyne F9 57 33 COC(=O)c1cc2c(O)cccc2s1 ZINC000147325563 BE In-Stock Anodyne SELE 55 32 COC(=O)c1cc2c(O)cccc2s1 ZINC000147325563 BE In-Stock Anodyne ICAM1 42 32 COC(=O)c1cc2c(O)cccc2s1 ZINC000147325563 BE In-Stock Anodyne SLC9A1 17 42 COC(=O)c1cc2c(O)cccc2s1 ZINC000147325563 BE In-Stock Anodyne PLAU 32 42 CN(C)C1(CNc2nc3ccc(Cl)cc3s2)CCCC1 ZINC000147325569 DI For-Sale Anodyne CSNK1D 23 40 Nc1ccc(-c2ccncc2NC(=O)c2nc(-c3ccccc3F)ccc2N)cn1 ZINC000147325576 HH Annotated Anodyne PIM1 35 58 Nc1ccc(-c2ccncc2NC(=O)c2nc(-c3ccccc3F)ccc2N)cn1 ZINC000147325576 HH Annotated Anodyne ATR 46 40 Nc1ccc(-c2ccncc2NC(=O)c2nc(-c3ccccc3F)ccc2N)cn1 ZINC000147325576 HH Annotated Anodyne PIM2 26 58 Nc1ccc(-c2ccncc2NC(=O)c2nc(-c3ccccc3F)ccc2N)cn1 ZINC000147325576 HH Annotated Anodyne PIM3 25 58 Cc1ccc(Br)c(C(=O)Nc2cccc3ccccc23)c1 ZINC000147325601 EK On-Demand Anodyne KCNJ11 47 38 Cc1ccc(Br)c(C(=O)Nc2cccc3ccccc23)c1 ZINC000147325601 EK On-Demand Anodyne TRPV1 19 44 Cc1ccc(Br)c(C(=O)Nc2cccc3ccccc23)c1 ZINC000147325601 EK On-Demand Anodyne CCR8 47 34 Cc1ccc(Br)c(C(=O)Nc2cccc3ccccc23)c1 ZINC000147325601 EK On-Demand Anodyne KCNK3 63 36 Cc1ccc(Br)c(C(=O)Nc2cccc3ccccc23)c1 ZINC000147325601 EK On-Demand Anodyne KCNK9 56 36 CC[C@@H](S)C(=O)NC(C)C ZINC000147325662 AD For-Sale Mild ACE2 38 43 CCCNc1ncc(Cl)c(Oc2ccc(C)cc2OC)n1 ZINC000147325668 DI For-Sale Anodyne P2RX2 50 35 COc1ncc(-c2cccc(CCO)c2)c2c(OC(=O)c3ccccc3)cccc12 ZINC000147325764 GJ For-Sale Anodyne FFAR1 16 40 COCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147325781 CD On-Demand Anodyne CACNA1H 25 40 COCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147325781 CD On-Demand Anodyne CACNA1I 52 36 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cccc(S(N)(=O)=O)c2)C1 ZINC000147325783 GB On-Demand Anodyne SFRP1 60 32 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2cccc(S(N)(=O)=O)c2)C1 ZINC000147325783 GB On-Demand Anodyne WNT3 41 31 CCOc1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147325844 CE For-Sale Anodyne ADRA1D 15 50 CCOc1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147325844 CE For-Sale Anodyne ADRA1B 0 45 CCOc1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147325844 CE For-Sale Anodyne HCN1 55 38 CCOc1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147325844 CE For-Sale Anodyne HCN4 47 37 CC[C@H](S)C(=O)NC(C)C ZINC000147325869 AD For-Sale Mild ACE2 38 43 CCCc1ccc(S(=O)(=O)NC[C@@H](CC)CC(=O)O)cc1 ZINC000147325889 DE On-Demand Anodyne CA2 17 42 CCCc1ccc(S(=O)(=O)NC[C@@H](CC)CC(=O)O)cc1 ZINC000147325889 DE On-Demand Anodyne TBXA2R 47 35 COc1ccc(O)c([C@H](C)NCC(F)F)c1 ZINC000147325903 BE On-Demand Clean THRA 43 33 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2cccc(S(N)(=O)=O)c2)C1 ZINC000147325955 GB On-Demand Anodyne SFRP1 60 32 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2cccc(S(N)(=O)=O)c2)C1 ZINC000147325955 GB On-Demand Anodyne WNT3 41 31 O=C(O)CCC/C=C\c1cccnc1 ZINC000147325971 AE For-Sale Anodyne TBXA2R 56 40 O=C(O)CCC/C=C\c1cccnc1 ZINC000147325971 AE For-Sale Anodyne TBXAS1 142 55 CCCCCCCCn1ccc2c1CC(C)(C)C[C@@H]2O ZINC000147325979 CJ For-Sale Mild GBA2 45 34 CCCCCCCCCn1ccc(I)n1 ZINC000147326019 DI For-Sale Mild ADA 0 40 COc1ccc2c(c1)OC[C@H](C(=O)NCc1cccc(NC(=O)c3ccncc3)c1)C2 ZINC000147326051 HG On-Demand Anodyne ROCK1 27 40 COc1ccc2c(c1)OC[C@H](C(=O)NCc1cccc(NC(=O)c3ccncc3)c1)C2 ZINC000147326051 HG On-Demand Anodyne ROCK2 56 43 CCCc1ccc(S(=O)(=O)NC[C@H](CC)CC(=O)O)cc1 ZINC000147326089 DE On-Demand Anodyne TBXA2R 47 35 COc1ccc(O)c([C@@H](C)NCC(F)F)c1 ZINC000147326108 BE On-Demand Clean THRA 43 33 N#Cc1cc(-c2ccccn2)ccc1N ZINC000147326166 AE For-Sale Anodyne XDH 42 38 N#Cc1cc(-c2ccccn2)ccc1N ZINC000147326166 AE For-Sale Anodyne PLAUR 16 50 N#Cc1cc(-c2ccccn2)ccc1N ZINC000147326166 AE For-Sale Anodyne GRM5 19 43 CCCCCCCCn1ccc2c1CC(C)(C)C[C@H]2O ZINC000147326175 CJ For-Sale Mild GBA2 45 34 CCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326233 GD On-Demand Anodyne HRH2 18 47 CCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326233 GD On-Demand Anodyne HRH3 16 47 CCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326233 GD On-Demand Anodyne MMP13 36 42 CCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326233 GD On-Demand Anodyne MMP2 19 42 CCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326233 GD On-Demand Anodyne MMP3 21 42 CCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326233 GD On-Demand Anodyne MMP7 32 41 CCCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326233 GD On-Demand Anodyne MMP1 20 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(NC(=O)c3ccncc3)c1)C2 ZINC000147326274 HG On-Demand Anodyne ROCK1 27 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc(NC(=O)c3ccncc3)c1)C2 ZINC000147326274 HG On-Demand Anodyne ROCK2 56 43 CCCc1ccc([C@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147326284 GK On-Demand Anodyne CYP3A4 17 43 CCCCCCCCn1c(C)cc2c1CCC[C@@H]2O ZINC000147326401 CJ For-Sale Mild GBA2 44 31 CCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326410 GD On-Demand Anodyne HRH2 18 47 CCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326410 GD On-Demand Anodyne HRH3 16 47 CCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326410 GD On-Demand Anodyne MMP13 36 42 CCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326410 GD On-Demand Anodyne MMP2 19 42 CCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326410 GD On-Demand Anodyne MMP3 21 42 CCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326410 GD On-Demand Anodyne MMP7 32 41 CCCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147326410 GD On-Demand Anodyne MMP1 20 42 CC[C@@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147326430 CF On-Demand Anodyne HCAR1 0 40 CCCc1ccc([C@@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147326472 GK On-Demand Anodyne CYP3A4 17 43 Cc1cc(CNC(=O)Nc2ccc(NC(=O)c3ccccc3)cc2C(F)(F)F)no1 ZINC000147326473 HJ On-Demand Anodyne ABL1 44 35 Cc1cc(CNC(=O)Nc2ccc(NC(=O)c3ccccc3)cc2C(F)(F)F)no1 ZINC000147326473 HJ On-Demand Anodyne RAF1 46 37 Cc1cc(CNC(=O)Nc2ccc(NC(=O)c3ccccc3)cc2C(F)(F)F)no1 ZINC000147326473 HJ On-Demand Anodyne FLT1 26 42 Cc1cc(CNC(=O)Nc2ccc(NC(=O)c3ccccc3)cc2C(F)(F)F)no1 ZINC000147326473 HJ On-Demand Anodyne KDR 17 42 Cc1cc(CNC(=O)Nc2ccc(NC(=O)c3ccccc3)cc2C(F)(F)F)no1 ZINC000147326473 HJ On-Demand Anodyne FLT3 19 42 Cc1cc(CNC(=O)Nc2ccc(NC(=O)c3ccccc3)cc2C(F)(F)F)no1 ZINC000147326473 HJ On-Demand Anodyne KCNK3 89 43 Cc1cc(CNC(=O)Nc2ccc(NC(=O)c3ccccc3)cc2C(F)(F)F)no1 ZINC000147326473 HJ On-Demand Anodyne KCNK9 49 37 COc1cccc2oc(C(=O)CBr)cc12 ZINC000147326476 CG For-Sale Reactive NQO1 23 40 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(F)cc1 ZINC000147326478 DH On-Demand Mild AURKB 25 40 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(F)cc1 ZINC000147326478 DH On-Demand Mild PRNP 38 40 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(F)cc1 ZINC000147326478 DH On-Demand Mild GRM4 54 43 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(F)cc1 ZINC000147326478 DH On-Demand Mild GRM5 43 48 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(F)cc1 ZINC000147326478 DH On-Demand Mild TAAR1 45 37 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(F)cc1 ZINC000147326478 DH On-Demand Mild SHH 33 40 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(F)cc1 ZINC000147326478 DH On-Demand Mild SMO 26 42 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(F)cc1 ZINC000147326478 DH On-Demand Mild KCNK3 123 57 O=C(Nc1cccc(C#Cc2ccccn2)c1)c1ccc(F)cc1 ZINC000147326478 DH On-Demand Mild KCNK9 81 38 O=C(O)/C=C/c1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147326572 DI For-Sale Anodyne ESR1 15 40 O=C(O)/C=C/c1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147326572 DI For-Sale Anodyne MAOB 34 40 O=C(O)/C=C/c1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147326572 DI For-Sale Anodyne PTGER2 37 43 O=C(O)/C=C/c1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147326572 DI For-Sale Anodyne PTGER4 22 43 O=C(O)/C=C/c1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147326572 DI For-Sale Anodyne PTPN2 0 45 O=C(O)/C=C/c1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147326572 DI For-Sale Anodyne PTGER3 16 46 O=C(O)/C=C/c1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147326572 DI For-Sale Anodyne CDC25B 24 45 O=C(O)/C=C/c1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147326572 DI For-Sale Anodyne AKR1C3 33 46 CCCCCCCCn1c(C)cc2c1CCC[C@H]2O ZINC000147326588 CJ For-Sale Mild GBA2 44 31 CC[C@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147326617 CF On-Demand Anodyne HCAR1 0 40 BrC1C[C@H]2CC[C@H](C1)N2C[C@@H]1CCCc2ccccc21 ZINC000147326643 EI For-Sale Reactive ACHP_LYMST 28 41 Cc1ccc2nc(-c3ccc(NC(=O)C(=O)NC[C@@H]4CCCCO4)cc3)sc2c1 ZINC000147326651 HH On-Demand Anodyne APP 23 48 CC[C@H](CNS(=O)(=O)c1ccc(C#N)cc1)CC(=O)O ZINC000147326710 CD On-Demand Mild TBXA2R 16 41 O=C(c1cccc2c1OCCN2)N(CC1CC1)C1CC1 ZINC000147326715 CF For-Sale Anodyne TRPM8 0 40 CCCCCCCCn1ccc2c1CCC[C@@H]2O ZINC000147326742 BI For-Sale Mild GBA2 45 32 O=C(O)/C=C/c1ccsc1COc1ccc(Cl)c(F)c1 ZINC000147326764 DI For-Sale Anodyne CDC25B 0 40 O=C(N1CCCc2cc([N+](=O)[O-])ccc21)C(F)(F)F ZINC000147326769 CE For-Sale Bother AVPR2 15 44 O=C(Nc1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147326811 HI On-Demand Anodyne ROCK2 20 41 O=C(Nc1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147326811 HI On-Demand Anodyne TYK2 42 36 O=C(Nc1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147326811 HI On-Demand Anodyne NAMPT 28 40 O=C(Nc1cccc(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147326811 HI On-Demand Anodyne KCNK3 62 44 CN(C)CCNC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147326814 HE On-Demand Anodyne AVPR2 54 40 CN(C)CCNC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147326814 HE On-Demand Anodyne AVPR1A 29 40 CN(C)CCNC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147326814 HE On-Demand Anodyne NOD2 40 33 CN(C)CCNC(=O)c1ccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147326814 HE On-Demand Anodyne POLR1A 44 41 CC(C)CNC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147326833 DF For-Sale Anodyne F3 68 34 Cc1ccc(C(=O)NCCNC(N)=O)cc1C#CCN ZINC000147326847 CB For-Sale Mild KIT 0 42 Cc1ccc(C(=O)NCCNC(N)=O)cc1C#CCN ZINC000147326847 CB For-Sale Mild DDR1 53 41 BrC1C[C@@H]2CC[C@H](C1)N2C[C@H]1CCCc2ccccc21 ZINC000147326852 EI For-Sale Reactive ACHP_LYMST 28 41 Cc1ccc2nc(-c3ccc(NC(=O)C(=O)NC[C@H]4CCCCO4)cc3)sc2c1 ZINC000147326864 HH On-Demand Anodyne APP 23 48 CCOC[C@H](C)NC(=O)Nc1ccc(NC(=O)c2ccccc2)cc1C(F)(F)F ZINC000147326896 HJ On-Demand Anodyne MTTP 47 36 CCOC[C@H](C)NC(=O)Nc1ccc(NC(=O)c2ccccc2)cc1C(F)(F)F ZINC000147326896 HJ On-Demand Anodyne KCNK3 90 43 CCOC[C@H](C)NC(=O)Nc1ccc(NC(=O)c2ccccc2)cc1C(F)(F)F ZINC000147326896 HJ On-Demand Anodyne KCNK9 59 39 CC[C@@H](CNS(=O)(=O)c1ccc(C#N)cc1)CC(=O)O ZINC000147326917 CD On-Demand Mild TBXA2R 16 41 CCCCCCCCn1ccc2c1CCC[C@H]2O ZINC000147326949 BI For-Sale Mild GBA2 45 32 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne MAOB 67 41 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne PTGER2 40 46 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne PTGER4 22 46 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne PTGER3 16 46 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne LTB4R 22 42 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne CDC25B 24 44 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne NR1H4 53 39 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne GYS1 48 37 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne HCAR2 0 42 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne FFAR1 66 44 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne AKR1C3 35 47 O=C(O)/C=C/c1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147326965 DI For-Sale Anodyne ADCYAP1R1 44 40 CC(C)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147327001 CF On-Demand Anodyne F3 67 33 CC(C)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147327001 CF On-Demand Anodyne HCAR1 0 40 O=C(Nc1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327004 HI On-Demand Anodyne ROCK2 20 41 O=C(Nc1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327004 HI On-Demand Anodyne TYK2 42 36 O=C(Nc1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327004 HI On-Demand Anodyne NAMPT 28 40 O=C(Nc1cccc(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327004 HI On-Demand Anodyne KCNK3 62 44 FC(F)CNCc1cnc[nH]1 ZINC000147327035 AC For-Sale Anodyne GABRR2 0 40 BrC1C[C@@H]2CC[C@H](C1)N2C[C@@H]1CCCc2ccccc21 ZINC000147327070 EI For-Sale Reactive ACHP_LYMST 28 41 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccc(S(N)(=O)=O)c1 ZINC000147327081 FD On-Demand Anodyne CYP3A4 18 44 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccccc2Cl)=NC12CCC(C(C)(C)C)CC2 ZINC000147327082 KK Annotated Anodyne GCGR 49 72 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccccc2Cl)=NC12CCC(C(C)(C)C)CC2 ZINC000147327082 KK Annotated Anodyne GLP1R 21 53 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccccc2Cl)=NC12CCC(C(C)(C)C)CC2 ZINC000147327082 KK Annotated Anodyne GIPR 54 37 CC(C)Oc1ccccc1NC(=O)NCc1cccc(CN2CCO[C@H](C)C2)c1 ZINC000147327130 GI On-Demand Anodyne DRD4 21 42 CC(C)Oc1ccccc1NC(=O)NCc1cccc(CN2CCO[C@H](C)C2)c1 ZINC000147327130 GI On-Demand Anodyne HRH2 22 42 CCCCCCCCn1c(C)cc2c1CC(C)(C)C[C@@H]2O ZINC000147327149 CK For-Sale Mild GBA2 41 33 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccc(S(N)(=O)=O)c1 ZINC000147327213 FD On-Demand Anodyne BMP1 47 33 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccc(S(N)(=O)=O)c1 ZINC000147327213 FD On-Demand Anodyne CYP3A4 18 44 O=C(Nc1cccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327220 HI On-Demand Anodyne ROCK2 20 41 O=C(Nc1cccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327220 HI On-Demand Anodyne TYK2 42 36 O=C(Nc1cccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327220 HI On-Demand Anodyne NAMPT 28 40 O=C(Nc1cccc(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327220 HI On-Demand Anodyne KCNK3 62 44 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(Cl)c(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147327289 KK Annotated Anodyne GCGR 56 80 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(Cl)c(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147327289 KK Annotated Anodyne GLP1R 23 58 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(Cl)c(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147327289 KK Annotated Anodyne GIPR 73 41 CCOc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327336 DE For-Sale Anodyne CSNK1D 38 52 CCOc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327336 DE For-Sale Anodyne Q50565_METTH 0 47 CCOc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327336 DE For-Sale Anodyne ISPD 0 42 CC(C)Oc1ccccc1NC(=O)NCc1cccc(CN2CCO[C@@H](C)C2)c1 ZINC000147327337 GI On-Demand Anodyne DRD4 21 42 CC(C)Oc1ccccc1NC(=O)NCc1cccc(CN2CCO[C@@H](C)C2)c1 ZINC000147327337 GI On-Demand Anodyne HRH2 22 42 CCCCOC(=O)c1ncccc1Oc1nc(OC)cc(OC)n1 ZINC000147327350 EF For-Sale Anodyne INHA 40 46 CCCCOC(=O)c1ncccc1Oc1nc(OC)cc(OC)n1 ZINC000147327350 EF For-Sale Anodyne ALS 96 49 Cc1cc(C)c(C(=O)N2CCC[C@H](CCBr)C2)c(C)c1 ZINC000147327364 EI For-Sale Reactive AKR1C3 0 41 CCCCCCCCn1c(C)cc2c1CC(C)(C)C[C@H]2O ZINC000147327373 CK For-Sale Mild GBA2 41 33 CCCNc1ncc(Br)c(Oc2ccc(C)cc2OC)n1 ZINC000147327381 FI For-Sale Anodyne P2RX2 46 35 O=C(O)/C=C/c1ccccc1COc1ccc(Cl)c(F)c1 ZINC000147327401 DI For-Sale Anodyne PTGER2 59 53 O=C(O)/C=C/c1ccccc1COc1ccc(Cl)c(F)c1 ZINC000147327401 DI For-Sale Anodyne PTGER4 28 46 O=C(O)/C=C/c1ccccc1COc1ccc(Cl)c(F)c1 ZINC000147327401 DI For-Sale Anodyne PTGER3 29 56 O=C(O)/C=C/c1ccccc1COc1ccc(Cl)c(F)c1 ZINC000147327401 DI For-Sale Anodyne CDC25B 26 50 O=C(O)/C=C/c1ccccc1COc1ccc(Cl)c(F)c1 ZINC000147327401 DI For-Sale Anodyne GYS1 44 32 O=C(O)/C=C/c1ccccc1COc1ccc(Cl)c(F)c1 ZINC000147327401 DI For-Sale Anodyne PTGDR 0 56 O=C(Nc1cccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327425 HI On-Demand Anodyne ROCK2 20 41 O=C(Nc1cccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327425 HI On-Demand Anodyne TYK2 42 36 O=C(Nc1cccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327425 HI On-Demand Anodyne NAMPT 28 40 O=C(Nc1cccc(CNC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1)c1ccncc1 ZINC000147327425 HI On-Demand Anodyne KCNK3 62 44 CCC(CC)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147327469 CG On-Demand Anodyne HCAR1 0 40 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(OC(F)(F)F)cc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147327474 KK Annotated Anodyne GLP1R 23 51 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(OC(F)(F)F)cc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147327474 KK Annotated Anodyne GIPR 104 51 CC(C)CCCCN[C@@H](C)c1ccc(-n2ccnc2)cc1 ZINC000147327491 CI For-Sale Anodyne CYP2C19 17 44 Cc1cc(C(=O)NCCC(=O)N2CCN(c3ccc(F)cc3)CC2)no1 ZINC000147327542 FD On-Demand Anodyne CCR1 15 42 CN(CCCNC(=O)N(C)Cc1cscn1)Cc1ccccc1 ZINC000147327554 EF On-Demand Anodyne ACHE 0 41 CN(CCCNC(=O)N(C)Cc1cscn1)Cc1ccccc1 ZINC000147327554 EF On-Demand Anodyne BMP1 49 34 CC[C@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147327557 CD On-Demand Anodyne CAPN2 45 33 CC[C@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147327557 CD On-Demand Anodyne Q9JN24_ECOLX 0 42 Cc1cc(C)c(C(=O)N2CCC[C@@H](CCBr)C2)c(C)c1 ZINC000147327567 EI For-Sale Reactive AKR1C3 0 41 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne CA2 20 41 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne CSNK1D 52 58 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne NMT1 19 45 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne PIK3CA 19 53 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne MTNR1A 52 38 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne MTNR1B 44 38 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne PIK3CG 17 40 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne HSD17B2 15 41 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne LUCI_PHOPE 32 42 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne PROKR1 53 31 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne FABK 0 48 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne PORCN 0 44 COc1ccc2nc(NCCNC(=O)N(C)C)sc2c1 ZINC000147327589 CD For-Sale Anodyne ISPD 0 50 CC(=O)OCc1ccc2c(c1)ncn2-c1cccc(-c2ccccc2)c1 ZINC000147327639 EJ For-Sale Anodyne COMT 65 37 CC(=O)OCc1ccc2c(c1)ncn2-c1cccc(-c2ccccc2)c1 ZINC000147327639 EJ For-Sale Anodyne F9 40 38 CC(=O)OCc1ccc2c(c1)ncn2-c1cccc(-c2ccccc2)c1 ZINC000147327639 EJ For-Sale Anodyne PDGFRB 20 51 CC(=O)OCc1ccc2c(c1)ncn2-c1cccc(-c2ccccc2)c1 ZINC000147327639 EJ For-Sale Anodyne PLK1 55 38 CC(=O)OCc1ccc2c(c1)ncn2-c1cccc(-c2ccccc2)c1 ZINC000147327639 EJ For-Sale Anodyne HPGD 45 41 O=C(c1cc2ccccc2nc1O)N1CCC[C@@H]1c1cccc(Cl)c1 ZINC000147327655 FJ On-Demand Anodyne ADAM17 15 44 O=C(c1cc2ccccc2nc1O)N1CCC[C@@H]1c1cccc(Cl)c1 ZINC000147327655 FJ On-Demand Anodyne MMP14 0 42 O=C(c1cc2ccccc2nc1O)N1CCC[C@@H]1c1cccc(Cl)c1 ZINC000147327655 FJ On-Demand Anodyne GRM5 17 41 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000147327712 HC On-Demand Anodyne CPT1A 46 49 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000147327712 HC On-Demand Anodyne CPT2 45 34 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000147327712 HC On-Demand Anodyne CCR8 41 32 CC(C)CCCCN[C@H](C)c1ccc(-n2ccnc2)cc1 ZINC000147327715 CI For-Sale Anodyne CYP2C19 17 44 Cc1cc(C)n([C@@H](C)C(=O)NCCC(=O)N2CCN(c3ccc(F)cc3)CC2)n1 ZINC000147327742 HE On-Demand Anodyne CCR1 38 43 Cc1cc(C)n([C@@H](C)C(=O)NCCC(=O)N2CCN(c3ccc(F)cc3)CC2)n1 ZINC000147327742 HE On-Demand Anodyne SSTR1 30 41 CC[C@@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147327788 CD On-Demand Anodyne CAPN2 45 33 CC[C@@H](CNS(=O)(=O)Cc1ccccc1)CC(=O)O ZINC000147327788 CD On-Demand Anodyne Q9JN24_ECOLX 0 42 O=C(c1cc2ccccc2nc1O)N1CCC[C@H]1c1cccc(Cl)c1 ZINC000147327862 FJ On-Demand Anodyne ADAM17 15 44 O=C(c1cc2ccccc2nc1O)N1CCC[C@H]1c1cccc(Cl)c1 ZINC000147327862 FJ On-Demand Anodyne MMP14 0 42 O=C(c1cc2ccccc2nc1O)N1CCC[C@H]1c1cccc(Cl)c1 ZINC000147327862 FJ On-Demand Anodyne GRM5 17 41 CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147327879 BD On-Demand Anodyne HCAR1 0 47 CC[C@@H]1CN(C(=O)c2cc(F)ccc2F)CC[C@@H]1N ZINC000147327887 CE On-Demand Anodyne DPP4 27 45 CC[C@@H]1CN(C(=O)c2cc(F)ccc2F)CC[C@@H]1N ZINC000147327887 CE On-Demand Anodyne PARP1 48 39 COc1ccc([N+](=O)[O-])cc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147327926 ED On-Demand Bother KCNMA1 20 46 Cc1cc(C)n([C@H](C)C(=O)NCCC(=O)N2CCN(c3ccc(F)cc3)CC2)n1 ZINC000147327927 HE On-Demand Anodyne CCR1 18 43 Cc1cc(C)n([C@H](C)C(=O)NCCC(=O)N2CCN(c3ccc(F)cc3)CC2)n1 ZINC000147327927 HE On-Demand Anodyne SSTR1 30 41 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@H]1CCCN(S(C)(=O)=O)C1 ZINC000147327929 HC On-Demand Anodyne CPT1A 46 49 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@H]1CCCN(S(C)(=O)=O)C1 ZINC000147327929 HC On-Demand Anodyne CPT2 45 34 COc1ccc(NC(C)=O)cc1S(=O)(=O)N[C@H]1CCCN(S(C)(=O)=O)C1 ZINC000147327929 HC On-Demand Anodyne CCR8 41 32 CC(=O)NCC(=O)c1cccc(Cl)c1 ZINC000147327992 BD For-Sale Anodyne ABAT 22 47 CC(=O)NCC(=O)c1cccc(Cl)c1 ZINC000147327992 BD For-Sale Anodyne KMO 0 51 CC(=O)NCC(=O)c1cccc(Cl)c1 ZINC000147327992 BD For-Sale Anodyne CTSV 28 40 CC(=O)NCC(=O)c1cccc(Cl)c1 ZINC000147327992 BD For-Sale Anodyne FEN1 0 57 CCCCCCC(=O)N(C)CCCCCO ZINC000147328004 BF On-Demand Anodyne FABP2 0 42 CCCCCCC(=O)N(C)CCCCCO ZINC000147328004 BF On-Demand Anodyne DNM1 0 45 CCCCCCC(=O)N(C)CCCCCO ZINC000147328004 BF On-Demand Anodyne SLC22A20 0 42 CCCCCCC(=O)N(C)CCCCCO ZINC000147328004 BF On-Demand Anodyne KDM4A 0 46 CCCCCCC(=O)N(C)CCCCCO ZINC000147328004 BF On-Demand Anodyne CQSS 60 37 NC(=O)c1ccccc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147328005 CC For-Sale Anodyne PAGA 0 45 FC(F)CNCc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147328024 DI On-Demand Mild TACR1 16 46 FC(F)CNCc1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147328024 DI On-Demand Mild PHES 0 41 CC[C@H]1CN(C(=O)c2cc(F)ccc2F)CC[C@@H]1N ZINC000147328087 CE On-Demand Anodyne DPP4 27 45 CC[C@H]1CN(C(=O)c2cc(F)ccc2F)CC[C@@H]1N ZINC000147328087 CE On-Demand Anodyne PARP1 48 39 CCC[C@@H](NC(N)=O)C(=O)NCCC(=O)N1CCN(c2ccc(F)cc2)CC1 ZINC000147328167 GC On-Demand Anodyne SSTR1 25 41 COc1ccc([N+](=O)[O-])cc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147328200 ED On-Demand Bother KCNMA1 20 46 COc1ccc(C)cc1-n1ccc(C(=O)Nc2cccc(NS(C)(=O)=O)c2)n1 ZINC000147328271 HF On-Demand Anodyne PLA2G7 29 41 COc1ccc(C)cc1-n1ccc(C(=O)Nc2cccc(NS(C)(=O)=O)c2)n1 ZINC000147328271 HF On-Demand Anodyne CPT1A 45 32 COc1ccc(C)cc1-n1ccc(C(=O)Nc2cccc(NS(C)(=O)=O)c2)n1 ZINC000147328271 HF On-Demand Anodyne KCNK3 93 42 COc1ccc(C)cc1-n1ccc(C(=O)Nc2cccc(NS(C)(=O)=O)c2)n1 ZINC000147328271 HF On-Demand Anodyne KCNK9 79 42 CC[C@@H]1CN(C(=O)c2cc(F)ccc2F)CC[C@H]1N ZINC000147328302 CE On-Demand Anodyne DPP4 27 45 CC[C@@H]1CN(C(=O)c2cc(F)ccc2F)CC[C@H]1N ZINC000147328302 CE On-Demand Anodyne PARP1 48 39 CN(C)CCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147328312 CD For-Sale Anodyne CACNA1H 24 40 O=C(c1nccc2ccccc12)N1CCC[C@H](CCBr)C1 ZINC000147328335 EH For-Sale Reactive CASP1 0 40 CNC(=O)CNC(=O)c1cn(-c2ccccc2)nc1-c1ccc(-c2ccccc2)cc1 ZINC000147328355 HH On-Demand Anodyne CDK2 20 53 CC[C@H](CNS(=O)(=O)CCc1ccccc1)CC(=O)O ZINC000147328361 CD On-Demand Anodyne MMP12 25 50 Cc1ccc(OCCCNC2(C(=O)O)CCC2)cc1C ZINC000147328446 CF For-Sale Anodyne DRD4 19 52 Cc1ccc(OCCCNC2(C(=O)O)CCC2)cc1C ZINC000147328446 CF For-Sale Anodyne PPARA 21 44 Cc1ccc(OCCCNC2(C(=O)O)CCC2)cc1C ZINC000147328446 CF For-Sale Anodyne PPARD 17 47 Cc1ccc(OCCCNC2(C(=O)O)CCC2)cc1C ZINC000147328446 CF For-Sale Anodyne PLA2G4B 49 31 COc1ccc(-c2cnc3ccc(NCCCO)nn23)cc1 ZINC000147328484 CE Annotated Anodyne IKBKB 31 53 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cscc1C ZINC000147328504 CF On-Demand Anodyne FKBP1A 59 41 CCOC(=O)[C@@H]1CCCCN1C(=O)c1cscc1C ZINC000147328504 CF On-Demand Anodyne FKBP12.6 0 51 CC[C@H]1CN(C(=O)c2cc(F)ccc2F)CC[C@H]1N ZINC000147328511 CE On-Demand Anodyne DPP4 27 45 CC[C@H]1CN(C(=O)c2cc(F)ccc2F)CC[C@H]1N ZINC000147328511 CE On-Demand Anodyne PARP1 48 39 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccccc2F)C1 ZINC000147328527 EC On-Demand Anodyne ADRA1B 16 44 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccccc2F)C1 ZINC000147328527 EC On-Demand Anodyne CCR8 54 32 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccccc2F)C1 ZINC000147328527 EC On-Demand Anodyne SFRP1 96 34 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccccc2F)C1 ZINC000147328527 EC On-Demand Anodyne WNT3 72 33 COCCOc1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147328537 FG On-Demand Anodyne GRM4 23 40 COCCOc1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147328537 FG On-Demand Anodyne KCNK3 48 36 COCCOc1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147328537 FG On-Demand Anodyne KCNK9 49 36 CN(C(=O)Nc1cc(Br)cc(C(=O)O)c1)c1ccccc1 ZINC000147328541 EH For-Sale Anodyne PSBA 0 41 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive ANPEP 43 32 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CASP3 15 41 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive BMP1 18 42 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive KLK3 76 42 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CTSB 77 50 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive PAPA1_CARPA 70 49 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CYSP_TRYCR 63 42 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CTSK 52 51 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CTSL 48 49 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive PGA 24 48 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CAPNS1 67 44 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive MMP11 45 33 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CTSS 33 50 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CAPN1 92 47 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CASP1 23 40 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CAPN2 125 50 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CASP6 22 40 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CASP9 30 40 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CTSC 44 45 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive CTRB_BOVIN 58 34 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive NPR 65 42 CCC[C@@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328542 CD For-Sale Reactive PSMB5 49 38 CCCCCCCCCCCC(=O)OC[N+](CC)(CC)CC ZINC000147328545 DK For-Sale Mild LPAR3 39 44 CCCCCCCCCCCC(=O)OC[N+](CC)(CC)CC ZINC000147328545 DK For-Sale Mild FABP5 15 43 CCCCCCCCCCCC(=O)OC[N+](CC)(CC)CC ZINC000147328545 DK For-Sale Mild ENPP2 15 43 CCCCCCCCCCCC(=O)OC[N+](CC)(CC)CC ZINC000147328545 DK For-Sale Mild NOD1 41 33 CCCCCCCCCCCC(=O)OC[N+](CC)(CC)CC ZINC000147328545 DK For-Sale Mild CQSS 63 40 COc1cc(C)ccc1Oc1ccnc(N)n1 ZINC000147328553 BE For-Sale Anodyne P2RX2 40 35 CC[C@@H](CNS(=O)(=O)CCc1ccccc1)CC(=O)O ZINC000147328554 CD On-Demand Anodyne MMP8 17 52 CC[C@@H](CNS(=O)(=O)CCc1ccccc1)CC(=O)O ZINC000147328554 CD On-Demand Anodyne MMP12 25 50 O=C(c1nccc2ccccc12)N1CCC[C@@H](CCBr)C1 ZINC000147328565 EH For-Sale Reactive CASP1 0 40 CC(C)Oc1ccccc1NC(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147328573 FG On-Demand Anodyne ADRA1D 23 46 CC(C)Oc1ccccc1NC(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147328573 FG On-Demand Anodyne ADRA1B 23 46 CC(C)Oc1ccccc1NC(=O)N1CCC(NC(=O)c2ccoc2)CC1 ZINC000147328573 FG On-Demand Anodyne SMO 25 42 Cc1ccccc1-n1nc(C(=O)Nc2cccc(NS(C)(=O)=O)c2)c2c1CCC2 ZINC000147328676 HG On-Demand Anodyne KCNK3 95 38 Cc1ccccc1-n1nc(C(=O)Nc2cccc(NS(C)(=O)=O)c2)c2c1CCC2 ZINC000147328676 HG On-Demand Anodyne KCNK9 54 37 O[C@@H](COc1cccc2[nH]ccc12)CN1CC=C(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147328681 HI On-Demand Anodyne HTR1A 25 63 O[C@@H](COc1cccc2[nH]ccc12)CN1CC=C(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147328681 HI On-Demand Anodyne SLC6A4 39 53 CCOC(=O)[C@H]1CCCCN1C(=O)c1cscc1C ZINC000147328717 CF On-Demand Anodyne FKBP12.6 0 51 O=C(O)c1cc(Cl)ccc1COc1ccccc1Cl ZINC000147328719 CI For-Sale Anodyne PTGER1 102 55 O=C(O)c1cc(Cl)ccc1COc1ccccc1Cl ZINC000147328719 CI For-Sale Anodyne PTGER4 18 40 O=C(O)c1cc(Cl)ccc1COc1ccccc1Cl ZINC000147328719 CI For-Sale Anodyne CXCL8 25 44 O=C(O)c1cc(Cl)ccc1COc1ccccc1Cl ZINC000147328719 CI For-Sale Anodyne FABP4 21 48 O=C(O)c1cc(Cl)ccc1COc1ccccc1Cl ZINC000147328719 CI For-Sale Anodyne PTGER3 34 40 O=C(O)c1cc(Cl)ccc1COc1ccccc1Cl ZINC000147328719 CI For-Sale Anodyne FABP5 33 48 O=C(O)c1cc(Cl)ccc1COc1ccccc1Cl ZINC000147328719 CI For-Sale Anodyne PTGDR2 24 48 O=C(O)c1cc(Cl)ccc1COc1ccccc1Cl ZINC000147328719 CI For-Sale Anodyne MCL1 19 54 O=C(O)c1cc(Cl)ccc1COc1ccccc1Cl ZINC000147328719 CI For-Sale Anodyne FFAR4 24 43 O=C(O)c1cc(Cl)ccc1COc1ccccc1Cl ZINC000147328719 CI For-Sale Anodyne AKR1C2 61 39 O=C(O)c1cc(Cl)ccc1COc1ccccc1Cl ZINC000147328719 CI For-Sale Anodyne AKR1C1 60 39 CC[C@@H]1CN(C(=O)Cc2cccc(F)c2)CC[C@@H]1N ZINC000147328724 CD On-Demand Anodyne DPP4 17 42 CC[C@@H]1CN(C(=O)Cc2cccc(F)c2)CC[C@@H]1N ZINC000147328724 CD On-Demand Anodyne MLNR 31 42 O=Cc1ccc2c(c1)ncn2-c1cccc(-c2ccccc2)c1 ZINC000147328726 CJ For-Sale Anodyne COMT 69 41 O=Cc1ccc2c(c1)ncn2-c1cccc(-c2ccccc2)c1 ZINC000147328726 CJ For-Sale Anodyne PDGFRB 20 50 O=Cc1ccc2c(c1)ncn2-c1cccc(-c2ccccc2)c1 ZINC000147328726 CJ For-Sale Anodyne HPGD 43 43 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive MME 37 42 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive ANPEP 47 33 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CASP3 16 43 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive BMP1 63 37 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive KLK3 93 42 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CTSB 91 51 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive PAPA1_CARPA 85 52 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CYSP_TRYCR 63 42 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CTSK 70 57 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CTSL 62 52 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive PGA 24 48 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CAPNS1 74 44 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive MMP11 45 33 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CTSS 39 57 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CAPN1 100 49 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CASP1 23 40 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CAPN2 150 50 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive PLAU 15 40 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CASP6 22 40 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CASP9 30 40 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive LAP3 41 34 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CTSC 44 45 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive CTRB_BOVIN 58 34 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive NPR 83 43 CCC[C@H](NC(=O)OCc1ccccc1)[C@@H](O)C#N ZINC000147328743 CD For-Sale Reactive PSMB5 49 38 CC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147328746 FC On-Demand Anodyne HRH2 16 42 CC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147328746 FC On-Demand Anodyne SFRP1 77 33 CC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147328746 FC On-Demand Anodyne WNT3 47 32 CN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)c1ccccc1 ZINC000147328767 DH For-Sale Anodyne AKR1C3 28 42 CN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)c1ccccc1 ZINC000147328767 DH For-Sale Anodyne PSBA 0 45 CS(=O)(=O)c1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147328783 FF For-Sale Reactive L3MBTL3 54 39 COc1cc(C)ccc1Oc1nc(N)nc2ccccc12 ZINC000147328803 CG For-Sale Anodyne DHFR 44 42 COc1cc(C)ccc1Oc1nc(N)nc2ccccc12 ZINC000147328803 CG For-Sale Anodyne FOLA 41 42 COc1cc(C)ccc1Oc1nc(N)nc2ccccc12 ZINC000147328803 CG For-Sale Anodyne DFR1 36 40 COc1cc(C)ccc1Oc1nc(N)nc2ccccc12 ZINC000147328803 CG For-Sale Anodyne DRTS_TOXGO 59 37 COc1cc(C)ccc1Oc1nc(N)nc2ccccc12 ZINC000147328803 CG For-Sale Anodyne DYR_PNECA 45 37 COc1cc(C)ccc1Oc1nc(N)nc2ccccc12 ZINC000147328803 CG For-Sale Anodyne DRTS_TRYCR 59 39 CC(C)Oc1ccccc1NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147328827 DI On-Demand Anodyne EPHX2 23 44 CCCCO[C@@H](C)C(=O)Nc1cccc(NS(C)(=O)=O)c1 ZINC000147328887 DE On-Demand Anodyne KCNK9 40 33 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne S1PR4 17 42 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne LPAR2 76 63 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne S1PR3 33 63 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne SLC2A1 28 47 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne PLA2G4B 81 39 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne FAAH 19 40 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne S1PR2 83 63 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne S1PR1 20 63 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne S1PR5 15 42 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne LEF 69 38 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne HT1 0 47 CCCCCOc1ccc(CNCCCCC(C)C)cc1 ZINC000147328915 CK For-Sale Anodyne LMGT2 0 47 CC[C@H]1CN(C(=O)Cc2cccc(F)c2)CC[C@@H]1N ZINC000147328941 CD On-Demand Anodyne DPP4 17 42 CC[C@H]1CN(C(=O)Cc2cccc(F)c2)CC[C@@H]1N ZINC000147328941 CD On-Demand Anodyne MLNR 31 42 CC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147328945 FC On-Demand Anodyne HRH2 16 42 CC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147328945 FC On-Demand Anodyne SFRP1 77 33 CC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147328945 FC On-Demand Anodyne WNT3 47 32 CNc1cccc(NCc2ccc(C)cc2)n1 ZINC000147328946 BG For-Sale Anodyne PETD 0 42 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive ANPEP 43 32 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CASP3 15 41 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive BMP1 18 42 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive KLK3 76 42 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CTSB 77 50 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive PAPA1_CARPA 70 49 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CYSP_TRYCR 63 42 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CTSK 52 51 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CTSL 48 49 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive PGA 24 48 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CAPNS1 67 44 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive MMP11 45 33 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CTSS 33 50 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CAPN1 92 47 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CASP1 23 40 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CAPN2 125 50 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CASP6 22 40 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CASP9 30 40 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CTSC 44 45 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive CTRB_BOVIN 58 34 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive NPR 65 42 CCC[C@@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147328950 CD For-Sale Reactive PSMB5 49 38 CCOC(=O)[C@@H]1CCCCN1C(=O)C1[C@H]2CCC[C@H]12 ZINC000147328966 CD On-Demand Anodyne FKBP1A 50 42 CS(=O)(=O)c1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147328975 FF For-Sale Reactive L3MBTL3 54 39 CCOC(=O)CCCNC(=O)c1cccc2c1OCCN2 ZINC000147328986 CD For-Sale Anodyne MLYCD 0 41 Nc1ccc([N+](=O)[O-])cc1COc1ccc(Cl)c(F)c1 ZINC000147328994 CH For-Sale Bother SNCA 48 40 CCCCCCCn1cnc(CCNCC)c1 ZINC000147329000 BG For-Sale Mild CPB2 32 49 CCCCCCCn1cnc(CCNCC)c1 ZINC000147329000 BG For-Sale Mild CPB1 22 41 CNC[C@H](C)C(=O)NN1CCCCC1 ZINC000147329032 AC For-Sale Anodyne Q8WS26_TRYCR 18 41 CC(C)Oc1ccccc1NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147329054 DI On-Demand Anodyne EPHX2 23 44 CNC(=O)CNC(=O)c1cn(-c2ccccc2)nc1-c1ccc2ccc(OC)cc2c1 ZINC000147329096 HG On-Demand Anodyne CDK2 19 54 CNC(=O)CNC(=O)c1cn(-c2ccccc2)nc1-c1ccc2ccc(OC)cc2c1 ZINC000147329096 HG On-Demand Anodyne CDK4 17 54 CCCCO[C@H](C)C(=O)Nc1cccc(NS(C)(=O)=O)c1 ZINC000147329104 DE On-Demand Anodyne KCNK9 40 33 CC(C)CCO[C@@H](C)C(=O)N1CCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000147329124 EH On-Demand Anodyne PRCP 62 44 CC[C@@H](N)C(=O)C1CCCCC1 ZINC000147329136 AD For-Sale Anodyne TPP2 30 41 CC[C@@H]1CN(C(=O)Cc2cccc(F)c2)CC[C@H]1N ZINC000147329151 CD On-Demand Anodyne DPP4 17 42 CC[C@@H]1CN(C(=O)Cc2cccc(F)c2)CC[C@H]1N ZINC000147329151 CD On-Demand Anodyne MLNR 31 42 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive MME 37 42 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive ANPEP 47 33 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CASP3 16 43 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive BMP1 18 42 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive KLK3 93 42 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CTSB 91 51 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive PAPA1_CARPA 85 52 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CYSP_TRYCR 63 42 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CTSK 70 57 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CTSL 62 52 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive PGA 24 48 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CAPNS1 74 44 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive MMP11 45 33 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CTSS 39 57 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CAPN1 100 49 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CASP1 23 40 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CAPN2 150 50 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive PLAU 15 40 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CASP6 22 40 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CASP9 30 40 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive LAP3 41 34 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CTSC 44 45 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive CTRB_BOVIN 58 34 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive NPR 83 43 CCC[C@H](NC(=O)OCc1ccccc1)[C@H](O)C#N ZINC000147329155 CD For-Sale Reactive PSMB5 49 38 CC(C)CCCCN[C@@H](C)C12CC3CC(CC(C3)C1)C2 ZINC000147329166 CK For-Sale Anodyne EPHX2 24 51 N#Cc1cccc(/C=C/C(=O)N2CCC[C@H]2CN2CCCC2)c1 ZINC000147329196 DF On-Demand Mild DPP4 16 45 N#Cc1cccc(/C=C/C(=O)N2CCC[C@H]2CN2CCCC2)c1 ZINC000147329196 DF On-Demand Mild UTS2R 44 29 N#Cc1cccc(/C=C/C(=O)N2CCC[C@H]2CN2CCCC2)c1 ZINC000147329196 DF On-Demand Mild CHRNA10 15 42 COc1ccccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147329235 CD On-Demand Anodyne OXTR 23 44 COc1ccccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147329235 CD On-Demand Anodyne AVPR1A 15 44 CNC[C@@H](C)C(=O)NN1CCCCC1 ZINC000147329238 AC For-Sale Anodyne Q8WS26_TRYCR 18 41 CC(C)Oc1ccccc1NC(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147329239 DI On-Demand Anodyne EPHX2 23 44 O=C(c1cccc2ccccc12)N1CCC[C@H](CCBr)C1 ZINC000147329298 EI For-Sale Reactive FAP 0 41 O=C(c1cccc2ccccc12)N1CCC[C@H](CCBr)C1 ZINC000147329298 EI For-Sale Reactive AKR1C3 0 49 O=C(c1cccc2ccccc12)N1CCC[C@H](CCBr)C1 ZINC000147329298 EI For-Sale Reactive L3MBTL1 0 40 O=C(c1cccc2ccccc12)N1CCC[C@H](CCBr)C1 ZINC000147329298 EI For-Sale Reactive L3MBTL3 19 40 O=C(c1cccc(CNS(=O)(=O)c2ccc(-c3ccccc3)cc2)c1)N1CCOCC1 ZINC000147329304 IG On-Demand Anodyne F2 20 42 O=C(c1cccc(CNS(=O)(=O)c2ccc(-c3ccccc3)cc2)c1)N1CCOCC1 ZINC000147329304 IG On-Demand Anodyne F10 22 43 O=C(c1cccc(CNS(=O)(=O)c2ccc(-c3ccccc3)cc2)c1)N1CCOCC1 ZINC000147329304 IG On-Demand Anodyne MMP13 21 45 O=C(c1cccc(CNS(=O)(=O)c2ccc(-c3ccccc3)cc2)c1)N1CCOCC1 ZINC000147329304 IG On-Demand Anodyne TRY2_BOVIN 93 46 O=C(c1cccc(CNS(=O)(=O)c2ccc(-c3ccccc3)cc2)c1)N1CCOCC1 ZINC000147329304 IG On-Demand Anodyne MMP2 18 45 O=C(c1cccc(CNS(=O)(=O)c2ccc(-c3ccccc3)cc2)c1)N1CCOCC1 ZINC000147329304 IG On-Demand Anodyne MMP9 15 40 O=C(c1cccc(CNS(=O)(=O)c2ccc(-c3ccccc3)cc2)c1)N1CCOCC1 ZINC000147329304 IG On-Demand Anodyne ST14 83 42 O=C(c1cccc(CNS(=O)(=O)c2ccc(-c3ccccc3)cc2)c1)N1CCOCC1 ZINC000147329304 IG On-Demand Anodyne AKR1C3 18 41 O=C(c1cccc(CNS(=O)(=O)c2ccc(-c3ccccc3)cc2)c1)N1CCOCC1 ZINC000147329304 IG On-Demand Anodyne TMPRSS6 40 33 Cc1nn(C(F)F)c(C)c1CC(=O)Nc1cccc(NS(C)(=O)=O)c1 ZINC000147329318 FE On-Demand Anodyne P2RX7 35 40 CC(C)CCO[C@H](C)C(=O)N1CCC[C@@H]1c1nc2ccccc2[nH]1 ZINC000147329331 EH On-Demand Anodyne PRCP 62 44 CC[C@H](N)C(=O)C1CCCCC1 ZINC000147329339 AD For-Sale Anodyne TPP2 30 41 CC(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147329350 FC On-Demand Anodyne ST14 44 33 CC(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147329350 FC On-Demand Anodyne AKR1C3 56 34 CC(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147329350 FC On-Demand Anodyne SFRP1 98 40 CC(=O)c1cccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147329350 FC On-Demand Anodyne WNT3 72 34 CC[C@H]1CN(C(=O)Cc2cccc(F)c2)CC[C@H]1N ZINC000147329352 CD On-Demand Anodyne DPP4 17 42 CC[C@H]1CN(C(=O)Cc2cccc(F)c2)CC[C@H]1N ZINC000147329352 CD On-Demand Anodyne MLNR 31 42 CC(C)CCCCN[C@H](C)C12CC3CC(CC(C3)C1)C2 ZINC000147329367 CK For-Sale Anodyne EPHX2 24 51 CCCCCCCCNS(=O)(=O)c1ccnc(NCC)c1 ZINC000147329412 DG For-Sale Mild ALOX15 41 38 CC(C)Oc1ccccc1NC(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147329431 DI On-Demand Anodyne EPHX2 23 44 CN(C)C(=O)Nc1ccns1 ZINC000147329477 AD For-Sale Anodyne PSBA 0 44 CN(C)C(=O)Nc1ccns1 ZINC000147329477 AD For-Sale Anodyne PPX1 0 42 O=C(c1cccc2ccccc12)N1CCC[C@@H](CCBr)C1 ZINC000147329493 EI For-Sale Reactive FAP 0 41 O=C(c1cccc2ccccc12)N1CCC[C@@H](CCBr)C1 ZINC000147329493 EI For-Sale Reactive AKR1C3 0 49 O=C(c1cccc2ccccc12)N1CCC[C@@H](CCBr)C1 ZINC000147329493 EI For-Sale Reactive L3MBTL1 0 40 O=C(c1cccc2ccccc12)N1CCC[C@@H](CCBr)C1 ZINC000147329493 EI For-Sale Reactive L3MBTL3 19 40 CC(C)CCO[C@@H](C)C(=O)N1CCC[C@H]1c1nc2ccccc2[nH]1 ZINC000147329531 EH On-Demand Anodyne PRCP 62 44 CC(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147329538 FC On-Demand Anodyne ST14 44 33 CC(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147329538 FC On-Demand Anodyne AKR1C3 56 34 CC(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147329538 FC On-Demand Anodyne SFRP1 98 40 CC(=O)c1cccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147329538 FC On-Demand Anodyne WNT3 72 34 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329564 EE On-Demand Anodyne TIMP3 40 32 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329564 EE On-Demand Anodyne HDAC8 16 42 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329564 EE On-Demand Anodyne HDAC10 52 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329564 EE On-Demand Anodyne HDAC1 16 45 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329564 EE On-Demand Anodyne HDAC2 30 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329564 EE On-Demand Anodyne HDAC3 30 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329564 EE On-Demand Anodyne HDAC6 28 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329564 EE On-Demand Anodyne HDAC11 57 43 C[C@H]1CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C[C@@H](C)O1 ZINC000147329593 DF On-Demand Anodyne CACNA1I 41 32 CC(C)CCO[C@H](C)C(=O)N1CCC[C@H]1c1nc2ccccc2[nH]1 ZINC000147329694 EH On-Demand Anodyne PRCP 62 44 CCNc1nc(Cl)nc(Oc2ccc(C)cc2OC)n1 ZINC000147329726 CG For-Sale Anodyne PPX1 0 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329750 EE On-Demand Anodyne CCKAR 22 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329750 EE On-Demand Anodyne TIMP3 40 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329750 EE On-Demand Anodyne HDAC8 16 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329750 EE On-Demand Anodyne HDAC10 52 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329750 EE On-Demand Anodyne HDAC1 16 45 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329750 EE On-Demand Anodyne HDAC2 30 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329750 EE On-Demand Anodyne HDAC3 30 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329750 EE On-Demand Anodyne HDAC6 28 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329750 EE On-Demand Anodyne CCKBR 15 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)C2CC2)c1 ZINC000147329750 EE On-Demand Anodyne HDAC11 57 43 CCCCCCCCNc1cc(Cl)ccc1C(=O)O ZINC000147329764 CJ For-Sale Mild RARB 18 43 CCCCCCCCNc1cc(Cl)ccc1C(=O)O ZINC000147329764 CJ For-Sale Mild HRP1_PLAFA 43 39 CCCCCCCCNc1cc(Cl)ccc1C(=O)O ZINC000147329764 CJ For-Sale Mild HNMT 42 36 CCCCCCCCNc1cc(Cl)ccc1C(=O)O ZINC000147329764 CJ For-Sale Mild AKR1C3 25 43 CCCCCCCCNc1cc(Cl)ccc1C(=O)O ZINC000147329764 CJ For-Sale Mild ASAH1 57 31 CCCCCCCCNc1cc(Cl)ccc1C(=O)O ZINC000147329764 CJ For-Sale Mild AKR1C2 60 43 CCCCCCCCNc1cc(Cl)ccc1C(=O)O ZINC000147329764 CJ For-Sale Mild OXER1 40 34 CCCCCCCCNc1cc(Cl)ccc1C(=O)O ZINC000147329764 CJ For-Sale Mild PSBA 0 43 C[C@H]1CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C[C@H](C)O1 ZINC000147329776 DF On-Demand Anodyne CACNA1I 41 32 CO[C@@H](C)CNNC(=O)OC(C)(C)C ZINC000147329811 BD For-Sale Reactive CTSK 22 41 O=C(c1ccc2ncccc2c1)N1CCC[C@H](CCBr)C1 ZINC000147329825 EH For-Sale Reactive CCR3 22 45 O=C(c1ccc2ncccc2c1)N1CCC[C@H](CCBr)C1 ZINC000147329825 EH For-Sale Reactive HPGD 45 38 O=C(c1ccc2ncccc2c1)N1CCC[C@H](CCBr)C1 ZINC000147329825 EH For-Sale Reactive MAP3K12 30 40 CNc1cc(Oc2ccc(C)cc2OC)cc([N+](=O)[O-])c1 ZINC000147329937 CH For-Sale Bother TBXA2R 0 47 CCCCCCCCNS(=O)(=O)c1cccnc1NCC ZINC000147329939 DG For-Sale Mild NPY5R 15 40 C[C@@H]1CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C[C@@H](C)O1 ZINC000147329951 DF On-Demand Anodyne CACNA1I 41 32 CO[C@H](C)CNNC(=O)OC(C)(C)C ZINC000147329971 BD For-Sale Reactive CTSK 22 41 Cc1nsc(NC(=O)N(C)C)c1C#N ZINC000147329995 BD For-Sale Mild PSBA 0 40 O=C(c1ccc2ncccc2c1)N1CCC[C@@H](CCBr)C1 ZINC000147330015 EH For-Sale Reactive CCR3 22 45 O=C(c1ccc2ncccc2c1)N1CCC[C@@H](CCBr)C1 ZINC000147330015 EH For-Sale Reactive HPGD 45 38 O=C(c1ccc2ncccc2c1)N1CCC[C@@H](CCBr)C1 ZINC000147330015 EH For-Sale Reactive MAP3K12 30 40 C[C@H]1CN(C(=O)c2ccc(NC(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)cc2)C[C@@H](C)O1 ZINC000147330078 HI On-Demand Anodyne MDM2 46 36 CCCOc1nc(N)nc(Oc2ccc(C)cc2OC)n1 ZINC000147330153 CE For-Sale Anodyne DHFR 34 42 CCCOc1nc(N)nc(Oc2ccc(C)cc2OC)n1 ZINC000147330153 CE For-Sale Anodyne DRTS_PLAFK 35 40 CCCOc1nc(N)nc(Oc2ccc(C)cc2OC)n1 ZINC000147330153 CE For-Sale Anodyne DRTS_TOXGO 53 39 CCCOc1nc(N)nc(Oc2ccc(C)cc2OC)n1 ZINC000147330153 CE For-Sale Anodyne DYR_PNECA 47 39 CCCOc1nc(N)nc(Oc2ccc(C)cc2OC)n1 ZINC000147330153 CE For-Sale Anodyne DRTS_TRYCR 45 32 CCCCCCCCNc1cc(OC)ccc1C(=O)O ZINC000147330160 CI For-Sale Mild RARB 21 40 CCCCCCCCNc1cc(OC)ccc1C(=O)O ZINC000147330160 CI For-Sale Mild MTNR1A 87 39 CCCCCCCCNc1cc(OC)ccc1C(=O)O ZINC000147330160 CI For-Sale Mild MTNR1B 77 39 CCCCCCCCNc1cc(OC)ccc1C(=O)O ZINC000147330160 CI For-Sale Mild PLA2G4B 87 40 CCCCCCCCNc1cc(OC)ccc1C(=O)O ZINC000147330160 CI For-Sale Mild SOAT1 40 41 CCCCCCCCNc1cc(OC)ccc1C(=O)O ZINC000147330160 CI For-Sale Mild FAAH 18 40 CCCCCCCCNc1cc(OC)ccc1C(=O)O ZINC000147330160 CI For-Sale Mild AKR1C3 34 56 CCCCCCCCNc1cc(OC)ccc1C(=O)O ZINC000147330160 CI For-Sale Mild ASAH1 44 31 CCCCCCCCNc1cc(OC)ccc1C(=O)O ZINC000147330160 CI For-Sale Mild AKR1C2 85 56 CCCCCCCCNc1cc(OC)ccc1C(=O)O ZINC000147330160 CI For-Sale Mild ACAT 0 47 NC(=O)CNC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147330170 DC For-Sale Anodyne F7 20 40 Cc1cc(Cl)nc2nc(N)nc(N)c12 ZINC000147330178 BD For-Sale Anodyne DHFR 36 43 Cc1cc(Cl)nc2nc(N)nc(N)c12 ZINC000147330178 BD For-Sale Anodyne DRTS_TOXGO 40 38 Cc1cc(Cl)nc2nc(N)nc(N)c12 ZINC000147330178 BD For-Sale Anodyne DYR_PNECA 46 38 CC(=O)Nc1ccc(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)cc1Cl ZINC000147330239 GG On-Demand Anodyne GRM4 47 46 CC(=O)Nc1ccc(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)cc1Cl ZINC000147330239 GG On-Demand Anodyne MAPK10 24 42 CC(=O)Nc1ccc(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)cc1Cl ZINC000147330239 GG On-Demand Anodyne MAPK8 15 42 CC(=O)Nc1ccc(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)cc1Cl ZINC000147330239 GG On-Demand Anodyne HEMY 47 34 CC(=O)Nc1ccc(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)cc1Cl ZINC000147330239 GG On-Demand Anodyne KCNK3 95 40 CC(=O)Nc1ccc(NC(=O)c2cccc(N3C(=O)CCC3=O)c2)cc1Cl ZINC000147330239 GG On-Demand Anodyne KCNK9 48 39 COC(=O)c1ccc(C)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147330246 GC On-Demand Anodyne CCR8 62 34 COC(=O)c1ccc(C)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147330246 GC On-Demand Anodyne SFRP1 69 32 COC(=O)c1ccc(C)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147330246 GC On-Demand Anodyne WNT3 41 30 CC(C)CCCCN[C@@H](C)c1ccc(CC(C)C)cc1 ZINC000147330257 CK For-Sale Anodyne LEF 21 42 CC(C)CCCCN[C@@H](C)c1ccc(CC(C)C)cc1 ZINC000147330257 CK For-Sale Anodyne SLC22A20 0 41 NC(=O)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147330345 CC For-Sale Anodyne HCAR1 0 41 CCCCCCCCNc1ccc(C(=O)O)c(Cl)c1 ZINC000147330389 CJ For-Sale Mild RARB 19 43 CCCCCCCCNc1ccc(C(=O)O)c(Cl)c1 ZINC000147330389 CJ For-Sale Mild THRB 47 35 CCCCCCCCNc1ccc(C(=O)O)c(Cl)c1 ZINC000147330389 CJ For-Sale Mild ASAH1 61 36 CCCCCCCCNc1ccc(C(=O)O)c(Cl)c1 ZINC000147330389 CJ For-Sale Mild AKR1C2 47 37 CCCCCCCCNc1ccc(C(=O)O)c(Cl)c1 ZINC000147330389 CJ For-Sale Mild AKR1C1 42 38 CCCCCCCCNc1ccc(C(=O)O)c(Cl)c1 ZINC000147330389 CJ For-Sale Mild ACAT 0 42 CCCCCCCCNc1ccc(C(=O)O)c(Cl)c1 ZINC000147330389 CJ For-Sale Mild PSBA 0 40 CCCCCCCCn1cnc(CCNCC)c1 ZINC000147330400 CG For-Sale Mild CPB2 32 49 CCCCCCCCn1cnc(CCNCC)c1 ZINC000147330400 CG For-Sale Mild CPB1 22 41 N#Cc1cccc(/C=C\C(=O)N2CCC[C@H]2CN2CCCC2)c1 ZINC000147330407 DF On-Demand Mild OPRK1 27 44 N#Cc1cccc(/C=C\C(=O)N2CCC[C@H]2CN2CCCC2)c1 ZINC000147330407 DF On-Demand Mild UTS2R 44 29 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000147330418 DD On-Demand Bother IRAK4 18 43 COC(=O)c1ccc(C)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147330448 GC On-Demand Anodyne CCR8 62 34 COC(=O)c1ccc(C)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147330448 GC On-Demand Anodyne SFRP1 69 32 COC(=O)c1ccc(C)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147330448 GC On-Demand Anodyne WNT3 41 30 CC(C)CCCCN[C@H](C)c1ccc(CC(C)C)cc1 ZINC000147330469 CK For-Sale Anodyne LEF 21 42 CC(C)CCCCN[C@H](C)c1ccc(CC(C)C)cc1 ZINC000147330469 CK For-Sale Anodyne SLC22A20 0 41 C[C@@H]1CN(C(=O)c2ccc(NC(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)cc2)C[C@@H](C)O1 ZINC000147330496 HI On-Demand Anodyne MDM2 46 36 Nc1ccc(COc2ccc(Cl)c(F)c2)cn1 ZINC000147330533 CG For-Sale Anodyne F9 20 41 COc1cc(C)ccc1Oc1nc(N)ncc1Br ZINC000147330546 DF For-Sale Anodyne DHFR 20 43 COc1cc(C)ccc1Oc1nc(N)ncc1Br ZINC000147330546 DF For-Sale Anodyne FOLA 47 43 COc1cc(C)ccc1Oc1nc(N)ncc1Br ZINC000147330546 DF For-Sale Anodyne DRTS_PLAFK 33 43 COc1cc(C)ccc1Oc1nc(N)ncc1Br ZINC000147330546 DF For-Sale Anodyne P2RX2 54 42 COc1cc(C)ccc1Oc1nc(N)ncc1Br ZINC000147330546 DF For-Sale Anodyne DFR1 21 42 COc1cc(C)ccc1Oc1nc(N)ncc1Br ZINC000147330546 DF For-Sale Anodyne P2RX3 32 42 COc1cc(C)ccc1Oc1nc(N)ncc1Br ZINC000147330546 DF For-Sale Anodyne DRTS_PLABA 39 43 COc1cc(C)ccc1Oc1nc(N)ncc1Br ZINC000147330546 DF For-Sale Anodyne DRTS_TOXGO 33 40 COc1cc(C)ccc1Oc1nc(N)ncc1Br ZINC000147330546 DF For-Sale Anodyne DFRA17 0 40 CCCCCCCCNS(=O)(=O)c1cnccc1NC ZINC000147330592 CF For-Sale Mild Q95J97_RABIT 0 42 CCCCCCCCCn1c(=O)oc2ccc(I)cc21 ZINC000147330604 GJ For-Sale Mild MIF 16 41 CCCCCCCCCn1c(=O)oc2ccc(I)cc21 ZINC000147330604 GJ For-Sale Mild TSPO 17 41 CCc1ccc(S(=O)(=O)NC[C@@H](CC)CC(=O)O)cc1 ZINC000147330611 CE On-Demand Anodyne LIMK2 29 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc([N+](=O)[O-])c1 ZINC000147330636 DD On-Demand Bother IRAK4 18 43 CN1CCN(C(=O)c2cccc3c2OCCN3)CC1=O ZINC000147330657 CC For-Sale Anodyne P2RX7 25 55 O=C(c1ccc(OC(F)F)cc1)N1CCC[C@H](CCBr)C1 ZINC000147330663 FH For-Sale Reactive GRM3 16 49 O=C(c1ccc(OC(F)F)cc1)N1CCC[C@H](CCBr)C1 ZINC000147330663 FH For-Sale Reactive L3MBTL3 41 37 CCOC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147330664 GC On-Demand Anodyne HRH2 16 45 CCOC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147330664 GC On-Demand Anodyne CCR8 47 38 CCOC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147330664 GC On-Demand Anodyne SFRP1 85 32 CCOC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147330664 GC On-Demand Anodyne WNT3 53 32 C[C@H]1CN(C(=O)c2ccc(NC(=O)c3ccc4c(c3)COC4)cc2)C[C@@H](C)O1 ZINC000147330745 GG On-Demand Anodyne L3MBTL3 19 41 CC[C@H](NC(=O)c1ccn(-c2cccc(F)c2)n1)c1ccccc1OCC(=O)NC ZINC000147330764 HG On-Demand Anodyne CTSA 49 36 Cc1cc(NCc2cccc(C(F)(F)F)c2)nc(-c2cccnc2)n1 ZINC000147330768 EI On-Demand Anodyne ROS1 58 40 COc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147330816 CD On-Demand Anodyne DRD4 43 33 COc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147330816 CD On-Demand Anodyne CCR3 20 44 COc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147330816 CD On-Demand Anodyne MTNR1A 41 43 COc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147330816 CD On-Demand Anodyne MTNR1B 34 40 COc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147330816 CD On-Demand Anodyne TAAR1 34 40 COc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147330816 CD On-Demand Anodyne LIMK2 22 40 CCc1ccc(S(=O)(=O)NC[C@H](CC)CC(=O)O)cc1 ZINC000147330820 CE On-Demand Anodyne LIMK2 29 42 O=c1oc2ccc(I)cc2n1CCCc1ccccc1 ZINC000147330842 GH For-Sale Anodyne MIF 20 51 O=c1oc2ccc(I)cc2n1CCCc1ccccc1 ZINC000147330842 GH For-Sale Anodyne SIGMAR1 21 53 CCOC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147330870 GC On-Demand Anodyne HRH2 16 45 CCOC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147330870 GC On-Demand Anodyne CCR8 47 38 CCOC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147330870 GC On-Demand Anodyne SFRP1 85 32 CCOC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147330870 GC On-Demand Anodyne WNT3 53 32 O=C(c1ccc(OC(F)F)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147330879 FH For-Sale Reactive GRM3 16 49 O=C(c1ccc(OC(F)F)cc1)N1CCC[C@@H](CCBr)C1 ZINC000147330879 FH For-Sale Reactive L3MBTL3 41 37 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(OCC(F)(F)F)nc1 ZINC000147330902 HI On-Demand Anodyne DGAT1 40 39 C[C@H]1CN(C(=O)c2ccc(NC(=O)c3ccc4c(c3)COC4)cc2)C[C@H](C)O1 ZINC000147330958 GG On-Demand Anodyne L3MBTL3 19 41 CC[C@@H](NC(=O)c1ccn(-c2cccc(F)c2)n1)c1ccccc1OCC(=O)NC ZINC000147330978 HG On-Demand Anodyne CTSA 49 36 CCCCCCCCNc1cnc(C(=O)O)cn1 ZINC000147330991 CF For-Sale Mild ASAH1 74 31 COc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147331000 CD On-Demand Anodyne DRD4 43 33 COc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147331000 CD On-Demand Anodyne CCR3 20 44 COc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147331000 CD On-Demand Anodyne MTNR1A 41 43 COc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147331000 CD On-Demand Anodyne MTNR1B 34 40 COc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147331000 CD On-Demand Anodyne TAAR1 34 40 COc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147331000 CD On-Demand Anodyne LIMK2 22 40 CC[C@H](CNS(=O)(=O)[C@@H](C)C(=O)OC)CC(=O)O ZINC000147331039 CB For-Sale Anodyne ENPEP 40 31 Cc1cc(S(=O)(=O)NCCNC(=O)N(C)C)ccc1Br ZINC000147331054 FD On-Demand Anodyne LEF 56 34 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(OCC(F)(F)F)nc1 ZINC000147331124 HI On-Demand Anodyne DGAT1 40 39 CCCCCCCCNc1ccc(F)cc1C(=O)O ZINC000147331201 CI For-Sale Mild RARB 18 43 CCCCCCCCNc1ccc(F)cc1C(=O)O ZINC000147331201 CI For-Sale Mild SOAT1 29 40 CCCCCCCCNc1ccc(F)cc1C(=O)O ZINC000147331201 CI For-Sale Mild ASAH1 83 33 CCCCCCCCNc1ccc(F)cc1C(=O)O ZINC000147331201 CI For-Sale Mild ACAT 0 54 CC[C@@H](CNS(=O)(=O)[C@@H](C)C(=O)OC)CC(=O)O ZINC000147331241 CB For-Sale Anodyne ENPEP 40 31 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CN2C(=O)CNC2=O)cc1 ZINC000147331243 FC On-Demand Anodyne HDAC11 40 34 CCCC[C@H](NCCCCC(C)C)c1ccc(F)cc1 ZINC000147331246 CK For-Sale Anodyne LEF 46 45 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(OCC(F)(F)F)nc1 ZINC000147331352 HI On-Demand Anodyne DGAT1 40 39 CCCCCCCCNc1nc(C)ccc1C(=O)O ZINC000147331378 CH For-Sale Mild RARB 15 40 CCCCCCCCNc1nc(C)ccc1C(=O)O ZINC000147331378 CH For-Sale Mild ASAH1 57 33 O=C(Nc1cccnc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147331385 EG For-Sale Anodyne AKR1C3 21 40 O=C(Nc1cccnc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147331385 EG For-Sale Anodyne NAMPT 32 48 CCCCCCCCn1c(=O)oc2ccc(I)cc21 ZINC000147331437 FJ For-Sale Mild MIF 16 41 CCCCCCCCn1c(=O)oc2ccc(I)cc21 ZINC000147331437 FJ For-Sale Mild TSPO 17 41 CCOc1cccc2cc([C@@H](C)NC(=O)N(C)Cc3cscn3)oc12 ZINC000147331439 FI On-Demand Anodyne BMP1 46 32 CCOc1cccc2cc([C@@H](C)NC(=O)N(C)Cc3cscn3)oc12 ZINC000147331439 FI On-Demand Anodyne CYP3A4 20 42 CCCC[C@@H](NCCCCC(C)C)c1ccc(F)cc1 ZINC000147331454 CK For-Sale Anodyne LEF 46 45 CC[C@H](CNS(=O)(=O)[C@H](C)C(=O)OC)CC(=O)O ZINC000147331456 CB For-Sale Anodyne ENPEP 40 31 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CN2C(=O)CNC2=O)cc1 ZINC000147331458 FC On-Demand Anodyne HDAC11 40 34 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2cccc(Br)c2)CC1 ZINC000147331467 IG On-Demand Anodyne ADRB1 18 48 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2cccc(Br)c2)CC1 ZINC000147331467 IG On-Demand Anodyne HTR1A 23 55 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2cccc(Br)c2)CC1 ZINC000147331467 IG On-Demand Anodyne SLC6A4 21 46 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2cccc(Br)c2)CC1 ZINC000147331467 IG On-Demand Anodyne ACOX1 17 40 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2cccc(Br)c2)CC1 ZINC000147331467 IG On-Demand Anodyne ABCB1 73 45 CC[C@@H]1CN(C(=O)c2ccccc2F)CC[C@@H]1N ZINC000147331510 CE On-Demand Anodyne SLC6A1 43 39 CC[C@@H]1CN(C(=O)c2ccccc2F)CC[C@@H]1N ZINC000147331510 CE On-Demand Anodyne L3MBTL1 0 40 CC[C@@H]1CN(C(=O)c2ccccc2F)CC[C@@H]1N ZINC000147331510 CE On-Demand Anodyne TP53BP1 0 40 NC(=O)c1ccc(OCC(=O)Nc2nc(-c3ccc4c(c3)OCCO4)cs2)cc1 ZINC000147331519 HF On-Demand Anodyne CHEK2 19 45 NC(=O)c1ccc(OCC(=O)Nc2nc(-c3ccc4c(c3)OCCO4)cs2)cc1 ZINC000147331519 HF On-Demand Anodyne CPT1A 17 45 NC(=O)c1ccc(OCC(=O)Nc2nc(-c3ccc4c(c3)OCCO4)cs2)cc1 ZINC000147331519 HF On-Demand Anodyne TGFBR1 22 43 CC(C)(C)OC(=O)NC[C@H](N)c1cccc(F)c1 ZINC000147331582 CE For-Sale Anodyne PAPA1_CARPA 43 47 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(OCC(F)(F)F)nc1 ZINC000147331588 HI On-Demand Anodyne DGAT1 40 39 CCCCCCCCNc1nccnc1C(=O)O ZINC000147331598 CF For-Sale Mild PLA2G4B 44 33 CCCCCCCCNc1nccnc1C(=O)O ZINC000147331598 CF For-Sale Mild ASAH1 78 33 O=C(Nc1cccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147331608 CG For-Sale Anodyne PPIA 41 51 O=C(Nc1cccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147331608 CG For-Sale Anodyne BCR 0 40 O=C(Nc1cccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147331608 CG For-Sale Anodyne AKR1C3 24 44 O=C(Nc1cccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147331608 CG For-Sale Anodyne BLM 0 40 O=C(Nc1cccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147331608 CG For-Sale Anodyne NAMPT 33 52 CCOc1cccc2cc([C@H](C)NC(=O)N(C)Cc3cscn3)oc12 ZINC000147331610 FI On-Demand Anodyne BMP1 46 32 CCOc1cccc2cc([C@H](C)NC(=O)N(C)Cc3cscn3)oc12 ZINC000147331610 FI On-Demand Anodyne CYP3A4 20 42 CC[C@@H](CNS(=O)(=O)[C@H](C)C(=O)OC)CC(=O)O ZINC000147331648 CB For-Sale Anodyne ENPEP 40 31 O=C(c1cc2ccccc2nc1O)N1CCC[C@@H]1Cc1ccccc1 ZINC000147331699 EH On-Demand Anodyne GRIN2B 43 42 O=C(c1cc2ccccc2nc1O)N1CCC[C@@H]1Cc1ccccc1 ZINC000147331699 EH On-Demand Anodyne TACR1 15 42 O=C(c1cc2ccccc2nc1O)N1CCC[C@@H]1Cc1ccccc1 ZINC000147331699 EH On-Demand Anodyne PREP 74 36 CC[C@H]1CN(C(=O)c2ccccc2F)CC[C@@H]1N ZINC000147331735 CE On-Demand Anodyne SLC6A1 43 39 CC[C@H]1CN(C(=O)c2ccccc2F)CC[C@@H]1N ZINC000147331735 CE On-Demand Anodyne L3MBTL1 0 40 CC[C@H]1CN(C(=O)c2ccccc2F)CC[C@@H]1N ZINC000147331735 CE On-Demand Anodyne TP53BP1 0 40 CCc1ncc(C(=O)Nc2cc([N+](=O)[O-])ccc2OC)s1 ZINC000147331772 DF On-Demand Bother KCNMA1 33 54 CCc1ncc(C(=O)Nc2cc([N+](=O)[O-])ccc2OC)s1 ZINC000147331772 DF On-Demand Bother WDR5 30 40 CN(C)C(=O)Oc1cc(Cl)ccc1N ZINC000147331795 BD For-Sale Anodyne NCEH1 72 47 CCCCCCCCNS(=O)(=O)c1ccc(NC)nc1 ZINC000147331801 CF For-Sale Mild ALOX15 56 45 O=C(NCC1CC1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147331821 DF For-Sale Anodyne CACNA1I 59 39 Nc1cccc(COc2ccc(Cl)c(F)c2)n1 ZINC000147331903 CG For-Sale Anodyne F9 15 40 O=C(c1cc2ccccc2nc1O)N1CCC[C@H]1Cc1ccccc1 ZINC000147331910 EH On-Demand Anodyne GRIN2B 43 42 O=C(c1cc2ccccc2nc1O)N1CCC[C@H]1Cc1ccccc1 ZINC000147331910 EH On-Demand Anodyne TACR1 15 42 O=C(c1cc2ccccc2nc1O)N1CCC[C@H]1Cc1ccccc1 ZINC000147331910 EH On-Demand Anodyne PREP 74 36 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CN2C(=O)CCC2=O)cc1 ZINC000147331919 FD On-Demand Anodyne HDAC10 43 38 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CN2C(=O)CCC2=O)cc1 ZINC000147331919 FD On-Demand Anodyne HDAC11 41 39 CC[C@@H]1CN(C(=O)c2ccccc2F)CC[C@H]1N ZINC000147331933 CE On-Demand Anodyne SLC6A1 43 39 CC[C@@H]1CN(C(=O)c2ccccc2F)CC[C@H]1N ZINC000147331933 CE On-Demand Anodyne L3MBTL1 0 40 CC[C@@H]1CN(C(=O)c2ccccc2F)CC[C@H]1N ZINC000147331933 CE On-Demand Anodyne TP53BP1 0 40 COc1ccc(CCn2c(=O)oc3ccc(I)cc32)cc1 ZINC000147331945 GG For-Sale Anodyne MIF 16 40 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147331949 HI On-Demand Anodyne ADRB1 18 43 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147331949 HI On-Demand Anodyne HTR1A 32 70 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147331949 HI On-Demand Anodyne HTR1D 17 44 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147331949 HI On-Demand Anodyne HTR1B 15 44 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147331949 HI On-Demand Anodyne SLC6A4 36 70 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147331949 HI On-Demand Anodyne ADRB3 19 53 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147331949 HI On-Demand Anodyne ABCB1 43 38 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147331949 HI On-Demand Anodyne CCR2 22 40 COc1ccccc1CN[C@H]1C2[C@H]3CC[C@H]2CN(C3)[C@H]1C(c1ccccc1)c1ccccc1 ZINC000147331950 IK Annotated Anodyne TACR1 20 75 COc1cc(C)ccc1Oc1nc(N)ncc1C ZINC000147332006 BE For-Sale Anodyne DHFR 24 44 COc1cc(C)ccc1Oc1nc(N)ncc1C ZINC000147332006 BE For-Sale Anodyne FOLA 46 44 COc1cc(C)ccc1Oc1nc(N)ncc1C ZINC000147332006 BE For-Sale Anodyne DRTS_PLAFK 38 44 COc1cc(C)ccc1Oc1nc(N)ncc1C ZINC000147332006 BE For-Sale Anodyne P2RX2 50 41 COc1cc(C)ccc1Oc1nc(N)ncc1C ZINC000147332006 BE For-Sale Anodyne DFR1 21 43 COc1cc(C)ccc1Oc1nc(N)ncc1C ZINC000147332006 BE For-Sale Anodyne P2RX3 30 41 COc1cc(C)ccc1Oc1nc(N)ncc1C ZINC000147332006 BE For-Sale Anodyne DRTS_PLABA 40 44 C[C@@H]1CCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147332027 BF For-Sale Anodyne PREP 94 38 O=C(NCC1CC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147332056 CF On-Demand Anodyne CACNA1H 24 43 O=C(NCC1CC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147332056 CF On-Demand Anodyne EPHX2 18 55 O=C(NCC1CC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147332056 CF On-Demand Anodyne CACNA1I 92 53 CC(=O)Nc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332066 GC On-Demand Anodyne EPHX2 21 42 CC(=O)Nc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332066 GC On-Demand Anodyne TGM2 31 41 CC(=O)Nc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332066 GC On-Demand Anodyne CA12 15 42 CC(=O)Nc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332066 GC On-Demand Anodyne F13A1 58 41 CC(=O)Nc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332066 GC On-Demand Anodyne IDO1 29 40 CC(=O)Nc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332066 GC On-Demand Anodyne SFRP1 60 32 CC(=O)Nc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332066 GC On-Demand Anodyne WNT3 44 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CN2C(=O)CCC2=O)cc1 ZINC000147332093 FD On-Demand Anodyne HDAC10 43 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CN2C(=O)CCC2=O)cc1 ZINC000147332093 FD On-Demand Anodyne HDAC11 41 39 CCCNc1ncc(COc2ccc(Cl)c(F)c2)s1 ZINC000147332119 DI For-Sale Anodyne LIMK1 20 41 CC[C@H]1CN(C(=O)c2ccccc2F)CC[C@H]1N ZINC000147332122 CE On-Demand Anodyne SLC6A1 43 39 CC[C@H]1CN(C(=O)c2ccccc2F)CC[C@H]1N ZINC000147332122 CE On-Demand Anodyne L3MBTL1 0 40 CC[C@H]1CN(C(=O)c2ccccc2F)CC[C@H]1N ZINC000147332122 CE On-Demand Anodyne TP53BP1 0 40 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147332136 HI On-Demand Anodyne ADRB2 44 53 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147332136 HI On-Demand Anodyne ADRB1 19 53 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147332136 HI On-Demand Anodyne HTR1A 42 70 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147332136 HI On-Demand Anodyne HTR1D 17 44 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147332136 HI On-Demand Anodyne HTR1B 15 44 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147332136 HI On-Demand Anodyne SLC6A4 36 70 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147332136 HI On-Demand Anodyne ADRB3 53 53 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147332136 HI On-Demand Anodyne ABCB1 53 38 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3cc(F)ccc23)CC1 ZINC000147332136 HI On-Demand Anodyne CCR2 75 40 CS(=O)(=O)Nc1ccc(F)cc1C(=O)Nc1ccc(CN2C(=O)CCC2=O)cc1 ZINC000147332189 HE On-Demand Anodyne PLA2G7 24 41 CS(=O)(=O)Nc1ccc(F)cc1C(=O)Nc1ccc(CN2C(=O)CCC2=O)cc1 ZINC000147332189 HE On-Demand Anodyne TRPV1 31 40 C[C@H]1CCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147332202 BF For-Sale Anodyne PREP 94 38 O=c1oc2ccc(I)cc2n1Cc1cc(F)ccc1F ZINC000147332235 GH For-Sale Anodyne MIF 19 57 Cc1ccc(Nc2ccccc2C(=O)Nc2cc(C)nn2C)cc1 ZINC000147332253 DI On-Demand Anodyne AKR1C3 26 53 Cc1ccc(Nc2ccccc2C(=O)Nc2cc(C)nn2C)cc1 ZINC000147332253 DI On-Demand Anodyne AKR1C2 53 41 Cc1ccc(Nc2ccccc2C(=O)Nc2cc(C)nn2C)cc1 ZINC000147332253 DI On-Demand Anodyne KCNK3 48 34 Cc1ccc(Nc2ccccc2C(=O)Nc2cc(C)nn2C)cc1 ZINC000147332253 DI On-Demand Anodyne KCNK9 49 34 CC(=O)Nc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332257 GC On-Demand Anodyne EPHX2 21 42 CC(=O)Nc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332257 GC On-Demand Anodyne TGM2 31 41 CC(=O)Nc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332257 GC On-Demand Anodyne CA12 15 42 CC(=O)Nc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332257 GC On-Demand Anodyne F13A1 58 41 CC(=O)Nc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332257 GC On-Demand Anodyne IDO1 29 40 CC(=O)Nc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332257 GC On-Demand Anodyne SFRP1 60 32 CC(=O)Nc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147332257 GC On-Demand Anodyne WNT3 44 32 CN(Cc1ccccc1)C(=O)CNC1(C(=O)O)CCC1 ZINC000147332262 CD For-Sale Anodyne TACR3 41 33 O=C(NN1CCCCC1)c1ccc2c(c1)CNCC2 ZINC000147332270 CD For-Sale Anodyne CNR1 58 36 O=C(NN1CCCCC1)c1ccc2c(c1)CNCC2 ZINC000147332270 CD For-Sale Anodyne PNMT 25 41 COc1cc(C)ccc1Oc1nc(N)ncc1F ZINC000147332332 BE For-Sale Anodyne DHFR 19 42 COc1cc(C)ccc1Oc1nc(N)ncc1F ZINC000147332332 BE For-Sale Anodyne FOLA 42 42 COc1cc(C)ccc1Oc1nc(N)ncc1F ZINC000147332332 BE For-Sale Anodyne DRTS_PLAFK 32 42 COc1cc(C)ccc1Oc1nc(N)ncc1F ZINC000147332332 BE For-Sale Anodyne P2RX2 48 39 COc1cc(C)ccc1Oc1nc(N)ncc1F ZINC000147332332 BE For-Sale Anodyne DRTS_PLABA 33 42 CC(C)c1nc(NN)cc(Oc2cccc([N+](=O)[O-])c2)n1 ZINC000147332382 CF For-Sale Bother ATSA 0 43 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne PPIA 27 42 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne LPL 41 32 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne KIT 21 62 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne MAPK14 0 65 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne RAF1 37 71 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne KDR 15 55 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne MTOR 15 41 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne EPHX2 17 50 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne PDGFRA 44 60 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne FLT3 74 77 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne CSF1R 25 63 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne Q8MMZ8_EIMTE 56 86 CC(C)(C)c1cc(NC(=O)Nc2ccc(C(=O)O)cc2)no1 ZINC000147332389 DG For-Sale Anodyne RET 28 62 C[C@@H]1CCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147332397 BF For-Sale Anodyne PREP 94 38 O=C(NC1CC1)C1CCN(C(=O)[C@H]2C[C@H]2c2cccc(Br)c2)CC1 ZINC000147332407 GG On-Demand Anodyne EPHX2 29 46 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000147332413 EF On-Demand Anodyne NPY2R 19 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000147332413 EF On-Demand Anodyne ENV 46 38 CCCCCCCCNS(=O)(=O)c1ccc(NCC)cc1 ZINC000147332431 DH For-Sale Mild ALOX15 61 47 CC(C)N(C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147332474 CF On-Demand Anodyne HCAR1 0 41 CC(C)N(C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147332474 CF On-Demand Anodyne PSBA 0 41 CC(C)CCCCN[C@@H](C)c1ccc2c(c1)NC(=O)CO2 ZINC000147332490 CG For-Sale Anodyne NR3C2 27 41 Cc1cc(C(=O)Nc2cc(S(C)(=O)=O)ccc2F)cc([N+](=O)[O-])c1 ZINC000147332527 FF On-Demand Bother WDR5 27 40 Nc1ccc(COc2ccc(Cl)c(F)c2)cc1[N+](=O)[O-] ZINC000147332554 CH For-Sale Bother F9 0 42 NNc1cc(Oc2cccc([N+](=O)[O-])c2)nc(C2CC2)n1 ZINC000147332586 CE For-Sale Bother ATSA 0 43 C[C@H]1CCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147332588 BF For-Sale Anodyne PREP 94 38 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000147332597 EF On-Demand Anodyne NPY2R 19 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(Cl)c(Cl)c1 ZINC000147332597 EF On-Demand Anodyne ENV 46 38 O=C(NC1CC1)C1CCN(C(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)CC1 ZINC000147332607 GG On-Demand Anodyne EPHX2 29 46 COc1cc(OCC(=O)Nc2cnc(-c3ccccc3)nc2)ccc1[N+](=O)[O-] ZINC000147332647 GG On-Demand Bother CETP 26 41 COc1cc(OCC(=O)Nc2cnc(-c3ccccc3)nc2)ccc1[N+](=O)[O-] ZINC000147332647 GG On-Demand Bother TAAR1 20 40 CCCCCCCCNc1nnccc1C(=O)O ZINC000147332648 CF For-Sale Mild ASAH1 63 32 O=C(CNC1(C(=O)O)CCC1)Nc1ccc2c(c1)OCO2 ZINC000147332677 CC For-Sale Anodyne LDLR 0 41 CC(C)CCCCN[C@H](C)c1ccc2c(c1)NC(=O)CO2 ZINC000147332686 CG For-Sale Anodyne NR3C2 27 41 CC(C)[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(C(C)(C)C)cc1 ZINC000147332761 FJ On-Demand Anodyne CYP3A4 18 44 CC[C@@H]1CCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147332788 CF For-Sale Anodyne PREP 82 37 CC[C@@H]1CCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147332788 CF For-Sale Anodyne ABHD11 0 40 CCOC(=O)c1[nH]c(C)c(C(=O)Nc2ccc(C(=O)OC(C)C)cc2)c1C ZINC000147332796 FH In-Stock Anodyne F3 50 33 CCOC(=O)c1[nH]c(C)c(C(=O)Nc2ccc(C(=O)OC(C)C)cc2)c1C ZINC000147332796 FH In-Stock Anodyne ACR 49 35 O=C(NC1CC1)C1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)CC1 ZINC000147332801 GG On-Demand Anodyne EPHX2 29 46 COCc1nc(C(=O)Nc2cc([N+](=O)[O-])ccc2C)cs1 ZINC000147332846 DF On-Demand Bother CACNA1D 53 33 COCc1nc(C(=O)Nc2cc([N+](=O)[O-])ccc2C)cs1 ZINC000147332846 DF On-Demand Bother KCNMA1 24 40 CCCCCCCCNS(=O)(=O)c1ccccc1NCC ZINC000147332851 DH For-Sale Mild ALOX15 35 41 COC(=O)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147332907 CD For-Sale Anodyne CACNA1I 44 35 COC(=O)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147332907 CD For-Sale Anodyne HCAR1 0 40 CC(C)[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(C(C)(C)C)cc1 ZINC000147332968 FJ On-Demand Anodyne CYP3A4 18 44 O=C(NC1CC1)C1CCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)CC1 ZINC000147332976 GG On-Demand Anodyne EPHX2 29 46 CC[C@H]1CCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147332980 CF For-Sale Anodyne PREP 82 37 CC[C@H]1CCCN1C(=O)C[C@@H]1CNc2ccccc21 ZINC000147332980 CF For-Sale Anodyne ABHD11 0 40 CCCCCCCCNc1cccc(F)c1C(=O)O ZINC000147333047 CI For-Sale Mild ASAH1 87 37 CCCCCCCCNc1cccc(F)c1C(=O)O ZINC000147333047 CI For-Sale Mild G3PG_TRYCR 0 44 CCCCCCCCNc1cccc(F)c1C(=O)O ZINC000147333047 CI For-Sale Mild ACAT 0 45 CCCCCCCCNc1cccc(F)c1C(=O)O ZINC000147333047 CI For-Sale Mild SAE1 0 44 COC(=O)c1cn(C(=O)OC(C)(C)C)c2ccc([N+](=O)[O-])cc12 ZINC000147333076 DG In-Stock Bother CTRB1 29 45 COC(=O)c1cn(C(=O)OC(C)(C)C)c2ccc([N+](=O)[O-])cc12 ZINC000147333076 DG In-Stock Bother F2RL3 47 34 CC(C)(C)OC(=O)N1CCC(OC(=O)Nc2ccccc2C(N)=O)CC1 ZINC000147333110 FF For-Sale Anodyne CHRM3 26 47 CC(C)(C)OC(=O)N1CCC(OC(=O)Nc2ccccc2C(N)=O)CC1 ZINC000147333110 FF For-Sale Anodyne CCR8 45 35 CC(C)(C)OC(=O)N1CCC(OC(=O)Nc2ccccc2C(N)=O)CC1 ZINC000147333110 FF For-Sale Anodyne GPR119 49 46 O=C(Nc1ccc(O)c(F)c1)c1cccc2c1OCCN2 ZINC000147333113 CF For-Sale Anodyne KCNK3 44 33 O=C(CNC1(C(=O)O)CCC1)Nc1nccs1 ZINC000147333126 CC For-Sale Anodyne MAP 0 45 O=C(CNC1(C(=O)O)CCC1)Nc1nccs1 ZINC000147333126 CC For-Sale Anodyne MAP1 128 43 CC[C@@H]1CCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147333127 CF For-Sale Anodyne PREP 82 37 CC[C@@H]1CCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147333127 CF For-Sale Anodyne ABHD11 0 40 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc3c(c2)OCCO3)C1 ZINC000147333164 GC On-Demand Anodyne PKM 36 47 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc3c(c2)OCCO3)C1 ZINC000147333164 GC On-Demand Anodyne SFRP1 46 31 CCCCCCCCNS(=O)(=O)c1ccccc1NC ZINC000147333190 CG For-Sale Mild ALOX15 35 41 Cn1ncc2c(N)nc(COc3ccc(Cl)c(F)c3)nc21 ZINC000147333202 DE For-Sale Anodyne Q9M629_MAIZE 61 37 C[C@H](N)CCC(=O)NN1CCCCC1 ZINC000147333219 AC For-Sale Anodyne DPP7 55 37 CCCCN(CCBr)c1nc2cc([N+](=O)[O-])ccc2[nH]1 ZINC000147333229 EG For-Sale Reactive GYRB 42 38 CC[C@H]1CCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147333264 CF For-Sale Anodyne PREP 82 37 CC[C@H]1CCCN1C(=O)C[C@H]1CNc2ccccc21 ZINC000147333264 CF For-Sale Anodyne ABHD11 0 40 O=C(NCC(F)(F)F)Nc1cccc(-c2cnc3cc(-c4ncccn4)ccn23)c1 ZINC000147333324 HI Annotated Anodyne BRAF 45 41 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne HTR1A 32 43 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne DRD2 48 43 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne DRD1 19 42 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne DRD4 40 30 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne HTR2A 26 41 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne HTR2C 29 41 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne ADRA1A 32 40 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne DRD3 59 43 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne HTR4 60 42 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne PDGFRB 65 39 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne HRP1_PLAFA 45 42 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne SRC 40 39 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne FLT1 19 42 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne KDR 18 41 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne SLC9A1 45 32 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne FLT4 41 38 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne AURKA 38 42 COc1cc2c(N)ncnc2cc1C(=O)NCCCN1CCN(C)CC1 ZINC000147333339 FC For-Sale Anodyne EHMT2 56 33 CCCCCCCCNc1c(C(=O)O)c(C)nn1C ZINC000147333367 CG For-Sale Mild ASAH1 50 32 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc3c(c2)OCCO3)C1 ZINC000147333369 GC On-Demand Anodyne PKM 36 47 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc3c(c2)OCCO3)C1 ZINC000147333369 GC On-Demand Anodyne SFRP1 46 31 C[C@@H](N)CCC(=O)NN1CCCCC1 ZINC000147333390 AC For-Sale Anodyne DPP7 55 37 Cc1c(Br)cccc1C(=O)Nc1ccc(Cl)cc1Br ZINC000147333407 HK For-Sale Anodyne F10 37 41 Cc1c(Br)cccc1C(=O)Nc1ccc(Cl)cc1Br ZINC000147333407 HK For-Sale Anodyne F12 0 40 Cc1c(Br)cccc1C(=O)Nc1ccc(Cl)cc1Br ZINC000147333407 HK For-Sale Anodyne KCNMA1 43 47 Cc1c(Br)cccc1C(=O)Nc1ccc(Cl)cc1Br ZINC000147333407 HK For-Sale Anodyne ACPS 0 43 Cc1c(Br)cccc1C(=O)Nc1ccc(Cl)cc1Br ZINC000147333407 HK For-Sale Anodyne DHOD 0 42 Cc1c(Br)cccc1C(=O)Nc1ccc(Cl)cc1Br ZINC000147333407 HK For-Sale Anodyne G2YM83_BOTF4 53 33 Cc1c(Br)cccc1C(=O)Nc1ccc(Cl)cc1Br ZINC000147333407 HK For-Sale Anodyne H9CNL0_SPOEX 0 57 COc1ccc([C@@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147333465 EH On-Demand Anodyne ACACA 52 35 COc1ccc([C@@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147333465 EH On-Demand Anodyne CYP3A4 17 43 CCCCCCCCNc1cccnc1C(=O)O ZINC000147333559 CH For-Sale Mild MAP1 30 43 CCCCCCCCNc1cccnc1C(=O)O ZINC000147333559 CH For-Sale Mild PLA2G4B 55 33 CCCCCCCCNc1cccnc1C(=O)O ZINC000147333559 CH For-Sale Mild ASAH1 61 33 O=C(CNC1(C(=O)O)CCC1)NCc1ccccc1 ZINC000147333560 CC For-Sale Anodyne NPFFR1 51 41 CC[C@H](CNS(=O)(=O)CCC(C)C)CC(=O)O ZINC000147333577 CD On-Demand Anodyne ENPEP 40 31 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne ADORA1 62 54 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne SLC29A1 56 35 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne ADORA2A 36 60 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne DNMT1 16 44 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne ADK 33 56 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne AHCY 114 57 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne P2RX4 46 47 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne P2RX1 58 44 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne P2RY1 32 47 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne ADCY5 43 39 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne AMD1 39 48 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne GAPDH 19 41 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne ITPR1 55 41 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne P2RY2 22 48 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne PRKACA 46 36 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne NS5B 36 53 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne ADORA3 72 56 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne OXGR1 146 54 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne RNASE1 44 35 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne DNMT3B 44 44 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne PANC 41 42 C/C=C1\O[C@H](n2cnc3c(N)ncnc32)[C@H](O)[C@@H]1O ZINC000147333651 CB For-Sale Anodyne DOT1L 76 44 CCNc1ncc(Br)c(Oc2ccc(C)cc2OC)n1 ZINC000147333673 EH For-Sale Anodyne P2RX2 44 32 COc1ccc([C@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147333685 EH On-Demand Anodyne ACACA 52 35 COc1ccc([C@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1 ZINC000147333685 EH On-Demand Anodyne CYP3A4 17 43 CC(C)c1nc(NN)cc(OCCN2CCCCC2)n1 ZINC000147333732 CD For-Sale Anodyne PSMB2 46 35 CC(C)c1nc(NN)cc(OCCN2CCCCC2)n1 ZINC000147333732 CD For-Sale Anodyne PSMB1 41 41 CC(C)c1nc(NN)cc(OCCN2CCCCC2)n1 ZINC000147333732 CD For-Sale Anodyne EHMT2 61 33 CC[C@@H](CNS(=O)(=O)CCC(C)C)CC(=O)O ZINC000147333752 CD On-Demand Anodyne ENPEP 40 31 CCCN(CCC)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147333815 CH On-Demand Anodyne HCAR1 0 40 NNc1cc(OCCN2CCCCC2)nc(C2CC2)n1 ZINC000147333951 CD For-Sale Anodyne PSMB2 45 36 NNc1cc(OCCN2CCCCC2)nc(C2CC2)n1 ZINC000147333951 CD For-Sale Anodyne PSMB1 40 36 NNc1cc(OCCN2CCCCC2)nc(C2CC2)n1 ZINC000147333951 CD For-Sale Anodyne EHMT2 57 38 O=C(NCc1ccccc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147334041 EG For-Sale Anodyne PPIA 26 43 O=C(NCc1ccccc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147334041 EG For-Sale Anodyne ANPEP 25 41 O=C(NCc1ccccc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147334041 EG For-Sale Anodyne ROCK2 18 49 O=C(NCc1ccccc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147334041 EG For-Sale Anodyne NCE103 19 49 O=C(NCc1ccccc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147334041 EG For-Sale Anodyne NAMPT 44 44 O=C(NCc1ccccc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147334041 EG For-Sale Anodyne PDS 55 41 CC[C@@H]1CN(C(=O)c2ccc3ncccc3c2)CC[C@@H]1N ZINC000147334047 CE On-Demand Anodyne CCR3 27 61 CC[C@@H]1CN(C(=O)c2ccc3ncccc3c2)CC[C@@H]1N ZINC000147334047 CE On-Demand Anodyne L3MBTL3 40 32 CC(C)[C@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147334064 DH On-Demand Anodyne CYP3A4 23 49 C=CS(=O)(=O)OC(c1ccc(C(O)(C(F)(F)F)C(F)(F)F)cc1)(C(F)(F)F)C(F)(F)F ZINC000147334106 KJ For-Sale Mild MLYCD 53 38 C=CS(=O)(=O)OC(c1ccc(C(O)(C(F)(F)F)C(F)(F)F)cc1)(C(F)(F)F)C(F)(F)F ZINC000147334106 KJ For-Sale Mild RORA 36 40 CCCCCCCCNc1ccc(C(=O)O)cc1F ZINC000147334162 CI For-Sale Mild RARB 26 52 CCCCCCCCNc1ccc(C(=O)O)cc1F ZINC000147334162 CI For-Sale Mild KCNQ1 0 40 CCCCCCCCNc1ccc(C(=O)O)cc1F ZINC000147334162 CI For-Sale Mild PLA2G4A 29 42 CCCCCCCCNc1ccc(C(=O)O)cc1F ZINC000147334162 CI For-Sale Mild S1PR4 15 41 CCCCCCCCNc1ccc(C(=O)O)cc1F ZINC000147334162 CI For-Sale Mild S1PR3 22 41 CCCCCCCCNc1ccc(C(=O)O)cc1F ZINC000147334162 CI For-Sale Mild PLA2G4B 69 42 CCCCCCCCNc1ccc(C(=O)O)cc1F ZINC000147334162 CI For-Sale Mild SOAT1 25 40 CCCCCCCCNc1ccc(C(=O)O)cc1F ZINC000147334162 CI For-Sale Mild ASAH1 90 37 CCCCCCCCNc1ccc(C(=O)O)cc1F ZINC000147334162 CI For-Sale Mild ACAT 0 51 CC(C)(C)c1nc(NN)cc(OCCN2CCCCC2)n1 ZINC000147334179 CD For-Sale Anodyne PSMB2 46 35 CC(C)(C)c1nc(NN)cc(OCCN2CCCCC2)n1 ZINC000147334179 CD For-Sale Anodyne PSMB5 16 41 CC(C)(C)c1nc(NN)cc(OCCN2CCCCC2)n1 ZINC000147334179 CD For-Sale Anodyne PSMB1 41 41 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne PPIA 42 46 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne GRIN2B 0 43 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne PTGER1 19 44 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne GUAB 0 51 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne ROCK2 20 49 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne EPHX2 21 45 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne CACNA1I 25 40 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne AKR1C3 27 42 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne NCE103 25 49 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne P96878_MYCTU 15 49 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne NAMPT 45 44 O=C(NCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147334219 DG On-Demand Anodyne PDS 60 40 CC[C@H]1CN(C(=O)c2ccc3ncccc3c2)CC[C@@H]1N ZINC000147334223 CE On-Demand Anodyne CCR3 27 61 CC[C@H]1CN(C(=O)c2ccc3ncccc3c2)CC[C@@H]1N ZINC000147334223 CE On-Demand Anodyne L3MBTL3 40 32 COc1ccc(C(=O)C2CCN(C(=O)c3ccc(C(N)=O)cn3)CC2)cc1 ZINC000147334231 FD On-Demand Anodyne SLC18A3 34 51 COc1ccc(C(=O)C2CCN(C(=O)c3ccc(C(N)=O)cn3)CC2)cc1 ZINC000147334231 FD On-Demand Anodyne PTR1 48 36 COc1ccc(C(=O)C2CCN(C(=O)c3ccc(C(N)=O)cn3)CC2)cc1 ZINC000147334231 FD On-Demand Anodyne L3MBTL3 45 36 COc1ccc(C(=O)C2CCN(C(=O)c3ccc(C(N)=O)cn3)CC2)cc1 ZINC000147334231 FD On-Demand Anodyne TRPC6 41 43 COc1ccc(C(=O)C2CCN(C(=O)c3ccc(C(N)=O)cn3)CC2)cc1 ZINC000147334231 FD On-Demand Anodyne TRPC3 22 43 CC(C)CCCCNCc1csc(Br)c1 ZINC000147334238 CI For-Sale Anodyne LEF 68 33 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(Cl)c2F)=NC12CCC(C(C)(C)C)CC2 ZINC000147334252 KK Annotated Anodyne GCGR 48 73 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(Cl)c2F)=NC12CCC(C(C)(C)C)CC2 ZINC000147334252 KK Annotated Anodyne GLP1R 21 51 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cccc(Cl)c2F)=NC12CCC(C(C)(C)C)CC2 ZINC000147334252 KK Annotated Anodyne GIPR 48 37 CC(C)[C@@H](NC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147334276 DH On-Demand Anodyne CYP3A4 23 49 CC(C)(O)c1cccc(CO)c1 ZINC000147334317 AD For-Sale Anodyne VIPR1 58 33 CCCCCCCCNc1ccc(C(=O)O)c(F)c1 ZINC000147334363 CI For-Sale Mild RARB 23 57 CCCCCCCCNc1ccc(C(=O)O)c(F)c1 ZINC000147334363 CI For-Sale Mild PLA2G4B 49 31 CCCCCCCCNc1ccc(C(=O)O)c(F)c1 ZINC000147334363 CI For-Sale Mild S1PR2 42 37 CCCCCCCCNc1ccc(C(=O)O)c(F)c1 ZINC000147334363 CI For-Sale Mild ASAH1 90 36 CCCCCCCCNc1ccc(C(=O)O)c(F)c1 ZINC000147334363 CI For-Sale Mild AKR1C2 43 35 CCCCCCCCNc1ccc(C(=O)O)c(F)c1 ZINC000147334363 CI For-Sale Mild ACAT 0 43 CC[C@@H]1CN(C(=O)c2ccc3ncccc3c2)CC[C@H]1N ZINC000147334388 CE On-Demand Anodyne CCR3 27 61 CC[C@@H]1CN(C(=O)c2ccc3ncccc3c2)CC[C@H]1N ZINC000147334388 CE On-Demand Anodyne L3MBTL3 40 32 CC(C)c1nc(NN)cc(OCC[C@@H]2CCCN2C)n1 ZINC000147334399 CD For-Sale Anodyne CHRNA10 59 36 Cc1cc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)ccc1Br ZINC000147334446 HD On-Demand Anodyne CTSC 16 40 CC(C)CCCCN[C@@H]1CCCc2c1[nH]c1ccccc21 ZINC000147334531 CJ For-Sale Anodyne EDNRB 45 34 CC[C@H]1CN(C(=O)c2ccc3ncccc3c2)CC[C@H]1N ZINC000147334600 CE On-Demand Anodyne CCR3 27 61 CC[C@H]1CN(C(=O)c2ccc3ncccc3c2)CC[C@H]1N ZINC000147334600 CE On-Demand Anodyne L3MBTL3 40 32 CC(C)c1nc(NN)cc(OCC[C@H]2CCCN2C)n1 ZINC000147334616 CD For-Sale Anodyne CHRNA10 59 36 CCN(C(=O)CCCOc1ccc2c(c1)CCC(=O)N2)c1cccnc1 ZINC000147334720 FG On-Demand Anodyne P2RY12 24 40 CC(C)CCCCN[C@H]1CCCc2c1[nH]c1ccccc21 ZINC000147334721 CJ For-Sale Anodyne EDNRB 45 34 COc1ccc(C2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147334788 GH On-Demand Anodyne ADRB2 20 55 COc1ccc(C2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147334788 GH On-Demand Anodyne ADRB1 23 48 COc1ccc(C2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147334788 GH On-Demand Anodyne HTR1A 27 74 COc1ccc(C2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147334788 GH On-Demand Anodyne SLC6A4 25 54 COc1ccc(C2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147334788 GH On-Demand Anodyne ADRB3 23 59 COc1ccc(C2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147334788 GH On-Demand Anodyne ACOX1 41 43 COc1ccc(C2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147334788 GH On-Demand Anodyne ABCB1 71 41 COc1ccc(C2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147334788 GH On-Demand Anodyne CARM1 46 33 CCCCCCCCNc1cc(C)nc(C)c1C(=O)O ZINC000147334802 CI For-Sale Mild ASAH1 60 32 CN1CCC[C@@H]1CCOc1cc(NN)nc(C2CC2)n1 ZINC000147334831 CD For-Sale Anodyne CHRNA10 64 37 CN1CCC[C@@H]1CCOc1cc(NN)nc(C2CC2)n1 ZINC000147334831 CD For-Sale Anodyne ACKR3 60 31 CCc1nc(CN(C)C(=O)N[C@@H](c2ccccc2)C(C)C)cs1 ZINC000147334855 EI On-Demand Anodyne CYP3A4 22 40 O=C(Nc1cc(Cl)cc(C(=O)O)c1)N[C@@H]1CCS(=O)(=O)C1 ZINC000147334867 ED On-Demand Anodyne EPHX2 27 45 CCCCNC(=O)C1CCN(C(=O)CN2CCc3ccccc32)CC1 ZINC000147334868 EE On-Demand Anodyne CCKAR 17 43 CCCCNC(=O)C1CCN(C(=O)CN2CCc3ccccc32)CC1 ZINC000147334868 EE On-Demand Anodyne TPP2 40 33 N[C@@H](Cc1ccc(O)c(O)c1)C(=O)NN1CCCCC1 ZINC000147334929 CC For-Sale Clean TH 0 43 N[C@@H](Cc1ccc(O)c(O)c1)C(=O)NN1CCCCC1 ZINC000147334929 CC For-Sale Clean OPRM1 27 41 N[C@@H](Cc1ccc(O)c(O)c1)C(=O)NN1CCCCC1 ZINC000147334929 CC For-Sale Clean OPRD1 25 41 N[C@@H](Cc1ccc(O)c(O)c1)C(=O)NN1CCCCC1 ZINC000147334929 CC For-Sale Clean YARS 74 35 N[C@@H](Cc1ccc(O)c(O)c1)C(=O)NN1CCCCC1 ZINC000147334929 CC For-Sale Clean ALOX15 23 56 N[C@@H](Cc1ccc(O)c(O)c1)C(=O)NN1CCCCC1 ZINC000147334929 CC For-Sale Clean DPP7 77 38 CC[C@@H]1CN(C(=O)c2ccc(C)c(F)c2)CC[C@@H]1N ZINC000147334970 CE On-Demand Anodyne L3MBTL3 65 36 COc1cc(NC(=O)CN2CCC(c3ccccn3)CC2)cc(OC)c1 ZINC000147334989 FF On-Demand Anodyne DRD4 32 67 COc1cc(NC(=O)CN2CCC(c3ccccn3)CC2)cc(OC)c1 ZINC000147334989 FF On-Demand Anodyne KCNA5 15 42 COc1cc(NC(=O)CN2CCC(c3ccccn3)CC2)cc(OC)c1 ZINC000147334989 FF On-Demand Anodyne NPY2R 28 41 COc1cc(NC(=O)CN2CCC(c3ccccn3)CC2)cc(OC)c1 ZINC000147334989 FF On-Demand Anodyne ACOX1 53 37 COc1cc(NC(=O)CN2CCC(c3ccccn3)CC2)cc(OC)c1 ZINC000147334989 FF On-Demand Anodyne NPY5R 19 40 COc1cc(NC(=O)CN2CCC(c3ccccn3)CC2)cc(OC)c1 ZINC000147334989 FF On-Demand Anodyne ZAP70 52 36 COc1cc(NC(=O)CN2CCC(c3ccccn3)CC2)cc(OC)c1 ZINC000147334989 FF On-Demand Anodyne MCHR1 42 38 COc1cc(NC(=O)CN2CCC(c3ccccn3)CC2)cc(OC)c1 ZINC000147334989 FF On-Demand Anodyne ALK 16 40 COc1ccc(C2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147335005 GH On-Demand Anodyne ADRB2 20 55 COc1ccc(C2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147335005 GH On-Demand Anodyne ADRB1 23 48 COc1ccc(C2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147335005 GH On-Demand Anodyne HTR1A 27 74 COc1ccc(C2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147335005 GH On-Demand Anodyne SLC6A4 25 54 COc1ccc(C2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147335005 GH On-Demand Anodyne ADRB3 23 59 COc1ccc(C2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147335005 GH On-Demand Anodyne ACOX1 41 43 COc1ccc(C2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147335005 GH On-Demand Anodyne ABCB1 71 41 COc1ccc(C2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)cc1 ZINC000147335005 GH On-Demand Anodyne CARM1 46 33 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@H]1O ZINC000147335025 EA For-Sale Mild POLA1 19 44 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@H]1O ZINC000147335025 EA For-Sale Mild P2RY6 158 63 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@H]1O ZINC000147335025 EA For-Sale Mild P2RY4 138 50 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@H]1O ZINC000147335025 EA For-Sale Mild P2RY1 29 48 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@H]1O ZINC000147335025 EA For-Sale Mild ATIC 27 41 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@H]1O ZINC000147335025 EA For-Sale Mild P2RY2 170 50 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@H]1O ZINC000147335025 EA For-Sale Mild P2RY14 89 52 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@H]1O ZINC000147335025 EA For-Sale Mild RNASE1 52 33 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@H]1O ZINC000147335025 EA For-Sale Mild GPR17 43 33 N#Cc1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)/C=C/c2cc(Cl)ccc2-n2cnnn2)cc1 ZINC000147335039 JH Annotated Mild CTSB 27 40 N#Cc1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)/C=C/c2cc(Cl)ccc2-n2cnnn2)cc1 ZINC000147335039 JH Annotated Mild F11 28 57 N#Cc1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)/C=C/c2cc(Cl)ccc2-n2cnnn2)cc1 ZINC000147335039 JH Annotated Mild CTRB_BOVIN 43 31 CN1CCC[C@H]1CCOc1cc(NN)nc(C2CC2)n1 ZINC000147335059 CD For-Sale Anodyne CHRNA10 64 37 CN1CCC[C@H]1CCOc1cc(NN)nc(C2CC2)n1 ZINC000147335059 CD For-Sale Anodyne ACKR3 60 31 CCc1nc(CN(C)C(=O)N[C@H](c2ccccc2)C(C)C)cs1 ZINC000147335069 EI On-Demand Anodyne CYP3A4 22 40 O=C(Nc1cc(Cl)cc(C(=O)O)c1)N[C@H]1CCS(=O)(=O)C1 ZINC000147335083 ED On-Demand Anodyne EPHX2 27 45 CC[C@H]1CN(C(=O)c2ccc(C)c(F)c2)CC[C@@H]1N ZINC000147335135 CE On-Demand Anodyne L3MBTL3 65 36 CCCCCCCCNc1cccc(Cl)c1C(=O)O ZINC000147335228 CJ For-Sale Mild SOAT1 15 40 CCCCCCCCNc1cccc(Cl)c1C(=O)O ZINC000147335228 CJ For-Sale Mild ASAH1 52 33 CCCCCCCCNc1cccc(Cl)c1C(=O)O ZINC000147335228 CJ For-Sale Mild G3PG_TRYCR 0 44 CCCCCCCCNc1cccc(Cl)c1C(=O)O ZINC000147335228 CJ For-Sale Mild ACAT 0 47 CCCCCCCCNc1cccc(Cl)c1C(=O)O ZINC000147335228 CJ For-Sale Mild SAE1 0 44 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@@H]1O ZINC000147335241 EA For-Sale Mild POLA1 19 44 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@@H]1O ZINC000147335241 EA For-Sale Mild P2RY6 158 63 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@@H]1O ZINC000147335241 EA For-Sale Mild P2RY4 138 50 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@@H]1O ZINC000147335241 EA For-Sale Mild P2RY1 29 48 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@@H]1O ZINC000147335241 EA For-Sale Mild ATIC 27 41 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@@H]1O ZINC000147335241 EA For-Sale Mild P2RY2 170 50 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@@H]1O ZINC000147335241 EA For-Sale Mild P2RY14 89 52 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@@H]1O ZINC000147335241 EA For-Sale Mild RNASE1 52 33 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](COP(=O)(O)O)[C@H](O)[C@@H]1O ZINC000147335241 EA For-Sale Mild GPR17 43 33 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2ccccc2)CC1 ZINC000147335263 FH On-Demand Anodyne ADRB2 16 48 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2ccccc2)CC1 ZINC000147335263 FH On-Demand Anodyne ADRB1 20 50 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2ccccc2)CC1 ZINC000147335263 FH On-Demand Anodyne HTR1A 29 70 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2ccccc2)CC1 ZINC000147335263 FH On-Demand Anodyne SLC6A4 25 54 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2ccccc2)CC1 ZINC000147335263 FH On-Demand Anodyne ADRB3 22 61 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2ccccc2)CC1 ZINC000147335263 FH On-Demand Anodyne ABCB1 64 44 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(OC(F)(F)F)cc2)C1 ZINC000147335270 HD On-Demand Anodyne CASR 26 43 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(OC(F)(F)F)cc2)C1 ZINC000147335270 HD On-Demand Anodyne EPHX2 28 45 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(OC(F)(F)F)cc2)C1 ZINC000147335270 HD On-Demand Anodyne SFRP1 121 36 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(OC(F)(F)F)cc2)C1 ZINC000147335270 HD On-Demand Anodyne WNT3 82 34 COc1ccc(OC)c(CNC2(C(=O)O)CCC2)c1 ZINC000147335283 CD On-Demand Anodyne MTNR1A 41 38 COc1ccc(OC)c(CNC2(C(=O)O)CCC2)c1 ZINC000147335283 CD On-Demand Anodyne MT-ND1 24 46 COc1ccc(OC)c(CNC2(C(=O)O)CCC2)c1 ZINC000147335283 CD On-Demand Anodyne AKR1C2 41 33 CN1CCC[C@H]1CCOc1cc(NN)nc(C(C)(C)C)n1 ZINC000147335287 CD For-Sale Anodyne CHRNA10 66 38 CCCCCNC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147335331 EG For-Sale Anodyne ASAH1 75 35 CCCCCNC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147335331 EG For-Sale Anodyne ACAT 0 51 CC[C@@H]1CN(C(=O)c2ccc(C)c(F)c2)CC[C@H]1N ZINC000147335336 CE On-Demand Anodyne L3MBTL3 65 36 Nc1cc(Br)ccc1C(=O)NN1CCCCC1 ZINC000147335399 CE For-Sale Anodyne CNR1 54 39 CCCCCCCCNc1ccc(C(=O)O)cc1Cl ZINC000147335424 CJ For-Sale Mild THRA 58 34 CCCCCCCCNc1ccc(C(=O)O)cc1Cl ZINC000147335424 CJ For-Sale Mild RARB 23 43 CCCCCCCCNc1ccc(C(=O)O)cc1Cl ZINC000147335424 CJ For-Sale Mild KCNQ1 0 40 CCCCCCCCNc1ccc(C(=O)O)cc1Cl ZINC000147335424 CJ For-Sale Mild PLA2G4B 69 42 CCCCCCCCNc1ccc(C(=O)O)cc1Cl ZINC000147335424 CJ For-Sale Mild ASAH1 56 36 CCCCCCCCNc1ccc(C(=O)O)cc1Cl ZINC000147335424 CJ For-Sale Mild ACAT 0 41 CCNc1ncnc(Oc2ccc(C)cc2OC)c1CC ZINC000147335429 CH For-Sale Anodyne PDE6A 43 36 CNC(=O)c1ccc(CN(C)C(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147335437 GF On-Demand Anodyne DRTS_PLAFK 20 45 CNC(=O)c1ccc(CN(C)C(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147335437 GF On-Demand Anodyne MTTP 42 38 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147335439 CA For-Sale Mild TOP1 54 38 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147335439 CA For-Sale Mild SLC29A1 52 35 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147335439 CA For-Sale Mild P2RY6 58 47 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147335439 CA For-Sale Mild TK1 33 40 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147335439 CA For-Sale Mild CDA 71 45 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147335439 CA For-Sale Mild P2RY4 45 39 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147335439 CA For-Sale Mild P2RY2 50 39 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147335439 CA For-Sale Mild P2RY14 64 40 CC(C)CCCCNC1CC(NC(=O)OC(C)(C)C)C1 ZINC000147335467 CG For-Sale Anodyne CTSK 24 41 CC(C)CCCCNC1CC(NC(=O)OC(C)(C)C)C1 ZINC000147335467 CG For-Sale Anodyne PGA5 44 38 CN1CCC[C@@H]1CCOc1cc(NN)nc(C(C)(C)C)n1 ZINC000147335519 CD For-Sale Anodyne CHRNA10 66 38 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc3c(c2)OCCCO3)C1 ZINC000147335541 GC On-Demand Anodyne PKM 34 43 CCCCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147335556 CG On-Demand Anodyne CACNA1H 24 40 CCCCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147335556 CG On-Demand Anodyne EPHX2 16 59 CCCCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147335556 CG On-Demand Anodyne ASAH1 64 35 CCCCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147335556 CG On-Demand Anodyne ACAT 0 52 CCCCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147335556 CG On-Demand Anodyne PSBA 0 41 CC[C@H]1CN(C(=O)c2ccc(C)c(F)c2)CC[C@H]1N ZINC000147335563 CE On-Demand Anodyne L3MBTL3 65 36 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@H]1O ZINC000147335638 CA For-Sale Mild TOP1 54 38 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@H]1O ZINC000147335638 CA For-Sale Mild SLC29A1 52 35 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@H]1O ZINC000147335638 CA For-Sale Mild P2RY6 58 47 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@H]1O ZINC000147335638 CA For-Sale Mild TK1 33 40 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@H]1O ZINC000147335638 CA For-Sale Mild CDA 71 45 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@H]1O ZINC000147335638 CA For-Sale Mild P2RY4 45 39 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@H]1O ZINC000147335638 CA For-Sale Mild P2RY2 50 39 N#Cc1cc(=O)[nH]c(=O)n1[C@@H]1O[C@H](CO)[C@H](O)[C@H]1O ZINC000147335638 CA For-Sale Mild P2RY14 64 40 CCCCCCCCNc1ccc(C(=O)O)nc1 ZINC000147335653 CH For-Sale Mild RARB 16 40 CCCCCCCCNc1ccc(C(=O)O)nc1 ZINC000147335653 CH For-Sale Mild PLA2G4B 58 35 CCCCCCCCNc1ccc(C(=O)O)nc1 ZINC000147335653 CH For-Sale Mild ASAH1 83 34 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne COMT 44 32 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne DHODH 26 40 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne CPN1 0 42 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne HDAC3 28 48 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne PTPN11 45 39 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne FEN1 0 42 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne E1 0 43 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne HK 0 49 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne RIPK1 34 40 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne P95276_MYCTO 0 43 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne PARP14 0 43 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne PARP15 0 40 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne KCNK3 85 40 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne KCNK9 74 40 NC(=O)Nc1cccc(-c2ccccc2)c1 ZINC000147335725 BF On-Demand Anodyne PARP10 0 43 CC(C)[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(F)cc1 ZINC000147335741 DH On-Demand Anodyne CYP3A4 15 42 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc3c(c2)OCCCO3)C1 ZINC000147335750 GC On-Demand Anodyne PKM 34 43 Cc1cccc(CN2C(=O)N/C(=C/c3c[nH]c4ccccc34)C2=O)c1 ZINC000147335834 EH In-Stock Anodyne HTR4 15 46 Cc1cc(C)n(-c2ccc(NC(=O)NC[C@@H](O)COc3c(C)cccc3C)cn2)n1 ZINC000147335850 HG On-Demand Anodyne ADRB1 46 36 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147335893 FF On-Demand Anodyne KCNQ2 92 47 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147335893 FF On-Demand Anodyne CSF1R 32 47 CC(C)[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(F)cc1 ZINC000147335921 DH On-Demand Anodyne CYP3A4 15 42 CC(=O)c1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147335983 CD For-Sale Anodyne AKR1C3 27 47 CC(=O)c1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147335983 CD For-Sale Anodyne KCNK3 92 38 CC(=O)c1cccc(NC(=O)CNC2(C(=O)O)CCC2)c1 ZINC000147335983 CD For-Sale Anodyne KCNK9 46 38 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147335988 EF On-Demand Anodyne TIMP3 47 30 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147335988 EF On-Demand Anodyne TNK2 49 35 O=C(CCC1CCNCC1)NN1CCCCC1 ZINC000147336055 BD For-Sale Anodyne F2R 30 46 O=C(CCC1CCNCC1)NN1CCCCC1 ZINC000147336055 BD For-Sale Anodyne GNAI1 0 40 O=C(CCC1CCNCC1)NN1CCCCC1 ZINC000147336055 BD For-Sale Anodyne GNAI3 0 40 O=C(CCC1CCNCC1)NN1CCCCC1 ZINC000147336055 BD For-Sale Anodyne GNAO1 0 40 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccccc1N1CCCCCC1 ZINC000147336071 FF On-Demand Anodyne CSF1R 32 47 COc1cc(C)ccc1Oc1nc(N)ncc1Cl ZINC000147336077 CF For-Sale Anodyne DHFR 22 42 COc1cc(C)ccc1Oc1nc(N)ncc1Cl ZINC000147336077 CF For-Sale Anodyne FOLA 45 42 COc1cc(C)ccc1Oc1nc(N)ncc1Cl ZINC000147336077 CF For-Sale Anodyne DRTS_PLAFK 35 42 COc1cc(C)ccc1Oc1nc(N)ncc1Cl ZINC000147336077 CF For-Sale Anodyne P2RX2 51 42 COc1cc(C)ccc1Oc1nc(N)ncc1Cl ZINC000147336077 CF For-Sale Anodyne DFR1 18 41 COc1cc(C)ccc1Oc1nc(N)ncc1Cl ZINC000147336077 CF For-Sale Anodyne P2RX3 31 45 COc1cc(C)ccc1Oc1nc(N)ncc1Cl ZINC000147336077 CF For-Sale Anodyne DRTS_PLABA 33 42 CN(Cc1cccc(C(F)(F)F)c1)C(=O)c1cc(F)ccc1NS(C)(=O)=O ZINC000147336092 HG On-Demand Anodyne TACR1 23 44 CN(Cc1cccc(C(F)(F)F)c1)C(=O)c1cc(F)ccc1NS(C)(=O)=O ZINC000147336092 HG On-Demand Anodyne TRPV1 77 43 CN(Cc1cccc(C(F)(F)F)c1)C(=O)c1cc(F)ccc1NS(C)(=O)=O ZINC000147336092 HG On-Demand Anodyne LIMK2 29 42 Cc1cc(C)n(-c2ccc(NC(=O)NC[C@H](O)COc3c(C)cccc3C)cn2)n1 ZINC000147336098 HG On-Demand Anodyne ADRB1 46 36 CCCCCCCCNc1nccc(C)c1C(=O)O ZINC000147336101 CH For-Sale Mild UTS2R 15 45 CCCCCCCCNc1nccc(C)c1C(=O)O ZINC000147336101 CH For-Sale Mild PLA2G4B 72 35 CCCCCCCCNc1nccc(C)c1C(=O)O ZINC000147336101 CH For-Sale Mild ASAH1 40 31 Cc1ccc(C(=O)N[C@@H]2CCCCC[C@@H]2C(=O)O)cc1Br ZINC000147336108 FH For-Sale Anodyne MAPK13 40 37 N#Cc1ccc(NC(=O)N2CCN(C=O)CC2)cc1 ZINC000147336126 CC For-Sale Mild PDGFRB 35 47 N#Cc1ccc(NC(=O)N2CCN(C=O)CC2)cc1 ZINC000147336126 CC For-Sale Mild TRPM8 17 48 O=C(Nc1cc(Cl)ccc1Br)c1ccncc1Cl ZINC000147336175 EI On-Demand Anodyne GRM4 33 42 O=C(Nc1cc(Cl)ccc1Br)c1ccncc1Cl ZINC000147336175 EI On-Demand Anodyne KCNMA1 25 44 O=C(Nc1cc(Cl)ccc1Br)c1ccncc1Cl ZINC000147336175 EI On-Demand Anodyne TYK2 23 49 O=C(Nc1cc(Cl)ccc1Br)c1ccncc1Cl ZINC000147336175 EI On-Demand Anodyne GPR35 25 40 O=C(c1cc2ncccn2n1)N1CCN(Cc2ccc(F)cc2Cl)CC1 ZINC000147336182 FE On-Demand Anodyne P2RX7 69 41 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147336186 EF On-Demand Anodyne OXTR 25 43 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147336186 EF On-Demand Anodyne AVPR1A 17 43 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147336186 EF On-Demand Anodyne TIMP3 47 30 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147336186 EF On-Demand Anodyne TNK2 49 35 CCCCc1ccc([C@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147336189 GK On-Demand Anodyne CYP3A4 18 42 FC(F)CNCC1CCCCCC1 ZINC000147336239 AF On-Demand Anodyne ADH4 0 45 CCC[C@@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147336244 CG On-Demand Anodyne CCKBR 52 36 CCC[C@@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147336244 CG On-Demand Anodyne CACNA1I 47 36 CCCCCCCCNS(=O)(=O)c1ccc(NCC)nc1 ZINC000147336315 DG For-Sale Mild ALOX15 48 41 Cc1ccc(C(=O)N[C@H]2CCCCC[C@@H]2C(=O)O)cc1Br ZINC000147336335 FH For-Sale Anodyne MAPK13 40 37 CC(C)CCCCNC(=O)CC1(C(=O)O)CCCCCC1 ZINC000147336381 CH For-Sale Anodyne CETP 0 41 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147336383 EF On-Demand Anodyne TIMP3 47 30 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147336383 EF On-Demand Anodyne TNK2 49 35 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2c(F)cccc2F)C1 ZINC000147336391 FC On-Demand Anodyne PKM 16 41 CCCCc1ccc([C@@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147336405 GK On-Demand Anodyne CYP3A4 18 42 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(O)(c2ccccc2)CC1 ZINC000147336433 FF On-Demand Anodyne HTR1A 23 57 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(O)(c2ccccc2)CC1 ZINC000147336433 FF On-Demand Anodyne ABCB1 62 61 CCC[C@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147336449 CG On-Demand Anodyne CCKBR 52 36 CCC[C@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147336449 CG On-Demand Anodyne CACNA1I 47 36 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(Cl)ccc2F)=NC12CCC(C(C)(C)C)CC2 ZINC000147336456 KK Annotated Anodyne GLP1R 22 54 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(Cl)ccc2F)=NC12CCC(C(C)(C)C)CC2 ZINC000147336456 KK Annotated Anodyne GIPR 66 42 CN1CCN(C(=O)Cc2ccc(NC(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)cc2)CC1 ZINC000147336491 HG On-Demand Anodyne MLNR 36 40 Cc1cc(C)n(-c2ccc(NC(=O)N[C@@H]3C[C@@H]3c3ccccc3)cn2)n1 ZINC000147336542 EH On-Demand Anodyne EPHX2 21 51 Cc1ccc(C(=O)N[C@@H]2CCCCC[C@H]2C(=O)O)cc1Br ZINC000147336544 FH For-Sale Anodyne MAPK13 40 37 Fc1cccc2c(NCCc3ccc(Cl)cc3)ncnc12 ZINC000147336577 DI For-Sale Anodyne HTT 0 59 Fc1cccc2c(NCCc3ccc(Cl)cc3)ncnc12 ZINC000147336577 DI For-Sale Anodyne MRGPRX1 16 41 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147336584 EF On-Demand Anodyne OXTR 25 43 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147336584 EF On-Demand Anodyne AVPR1A 17 43 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147336584 EF On-Demand Anodyne TIMP3 47 30 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147336584 EF On-Demand Anodyne TNK2 49 35 CN(Cc1cscn1)C(=O)N[C@@H](c1ccccc1)c1ccco1 ZINC000147336656 EH On-Demand Anodyne CYP3A4 20 46 CN1CCN(C(=O)Cc2ccc(NC(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)cc2)CC1 ZINC000147336682 HG On-Demand Anodyne MLNR 36 40 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCC2)cc1 ZINC000147336709 FD On-Demand Anodyne NPY2R 17 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCC2)cc1 ZINC000147336709 FD On-Demand Anodyne MTOR 16 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCC2)cc1 ZINC000147336709 FD On-Demand Anodyne L3MBTL3 76 40 COc1ccc(OC)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147336726 GC On-Demand Anodyne ADRA1D 19 49 COc1ccc(OC)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147336726 GC On-Demand Anodyne ADRA1A 15 49 COc1ccc(OC)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147336726 GC On-Demand Anodyne ADRA1B 26 49 CCCCCCCCNS(=O)(=O)c1ccnc(NC)c1 ZINC000147336735 CF For-Sale Mild ALOX15 42 38 Cc1ccc(C(=O)N[C@H]2CCCCC[C@H]2C(=O)O)cc1Br ZINC000147336744 FH For-Sale Anodyne MAPK13 40 37 CCC[C@H](NC(=O)c1csc(COC)n1)c1ccccc1 ZINC000147336755 DH On-Demand Anodyne TACR3 49 39 CCC[C@H](NC(=O)c1csc(COC)n1)c1ccccc1 ZINC000147336755 DH On-Demand Anodyne UTS2 53 33 CCOc1nc(N)nc(Oc2ccc(C)cc2OC)n1 ZINC000147336764 CD For-Sale Anodyne DHFR 45 43 CCOc1nc(N)nc(Oc2ccc(C)cc2OC)n1 ZINC000147336764 CD For-Sale Anodyne FOLA 41 42 CCOc1nc(N)nc(Oc2ccc(C)cc2OC)n1 ZINC000147336764 CD For-Sale Anodyne DRTS_PLAFK 40 41 CCOc1nc(N)nc(Oc2ccc(C)cc2OC)n1 ZINC000147336764 CD For-Sale Anodyne DRTS_TOXGO 64 40 CCOc1nc(N)nc(Oc2ccc(C)cc2OC)n1 ZINC000147336764 CD For-Sale Anodyne DYR_PNECA 56 40 CCOc1nc(N)nc(Oc2ccc(C)cc2OC)n1 ZINC000147336764 CD For-Sale Anodyne DRTS_TRYCR 49 35 CC[C@H]1CN(C(=O)CCS(=O)(=O)c2ccc3c(c2)OCCO3)CCO1 ZINC000147336774 FD On-Demand Anodyne PKM 32 41 Cc1cc(C)n(-c2ccc(NC(=O)N[C@H]3C[C@@H]3c3ccccc3)cn2)n1 ZINC000147336786 EH On-Demand Anodyne EPHX2 21 51 CN(Cc1cscn1)C(=O)N[C@H](c1ccccc1)c1ccco1 ZINC000147336883 EH On-Demand Anodyne CYP3A4 20 46 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCC2)cc1 ZINC000147336903 FD On-Demand Anodyne NPY2R 17 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCC2)cc1 ZINC000147336903 FD On-Demand Anodyne MTOR 16 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1ccc(C(=O)N2CCCC2)cc1 ZINC000147336903 FD On-Demand Anodyne L3MBTL3 76 40 CN1CCN(C(=O)Cc2ccc(NC(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)cc2)CC1 ZINC000147336904 HG On-Demand Anodyne MLNR 36 40 CN1CCN(C(=O)Cc2ccc(NC(=O)[C@H]3C[C@H]3c3cccc(Cl)c3)cc2)CC1 ZINC000147336904 HG On-Demand Anodyne MAPK1 22 41 COc1ccc(OC)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147336933 GC On-Demand Anodyne ADRA1D 19 49 COc1ccc(OC)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147336933 GC On-Demand Anodyne ADRA1A 15 49 COc1ccc(OC)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147336933 GC On-Demand Anodyne ADRA1B 26 49 CCCCCCCCNS(=O)(=O)c1ccnc(N)c1 ZINC000147336934 CE For-Sale Mild ALOX15 44 40 CCC[C@@H](NC(=O)c1csc(COC)n1)c1ccccc1 ZINC000147336947 DH On-Demand Anodyne TACR3 49 39 CCC[C@@H](NC(=O)c1csc(COC)n1)c1ccccc1 ZINC000147336947 DH On-Demand Anodyne UTS2 53 33 NCc1ccc(C(=O)NN2CCCCC2)o1 ZINC000147336960 BC For-Sale Anodyne CSF1R 0 41 Cc1cc(C)n(-c2ccc(NC(=O)N[C@@H]3C[C@H]3c3ccccc3)cn2)n1 ZINC000147336961 EH On-Demand Anodyne EPHX2 21 51 COc1cc(C)ccc1Oc1ncnc(N)c1C(C)C ZINC000147337011 CG For-Sale Anodyne P2RX2 41 36 Cc1cc(C)n(-c2ccc(NC(=O)N[C@H]3C[C@H]3c3ccccc3)cn2)n1 ZINC000147337075 EH On-Demand Anodyne EPHX2 21 51 COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1OC ZINC000147337187 GC On-Demand Anodyne ADRA1D 24 48 COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1OC ZINC000147337187 GC On-Demand Anodyne ADRA1A 17 48 COc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1OC ZINC000147337187 GC On-Demand Anodyne ADRA1B 34 48 C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)nc4)ccc23)c1 ZINC000147337229 JJ Annotated Mild EGFR 104 47 C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)nc4)ccc23)c1 ZINC000147337229 JJ Annotated Mild ERBB2 41 63 C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)nc4)ccc23)c1 ZINC000147337229 JJ Annotated Mild HDAC1 45 89 C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)nc4)ccc23)c1 ZINC000147337229 JJ Annotated Mild FBP1 0 44 C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)nc4)ccc23)c1 ZINC000147337229 JJ Annotated Mild ERBB4 63 40 C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)nc4)ccc23)c1 ZINC000147337229 JJ Annotated Mild EPHA8 15 47 C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)nc4)ccc23)c1 ZINC000147337229 JJ Annotated Mild EPHA5 22 47 C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)nc4)ccc23)c1 ZINC000147337229 JJ Annotated Mild MKNK1 20 47 C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)nc4)ccc23)c1 ZINC000147337229 JJ Annotated Mild DDR1 16 47 C#Cc1cccc(Nc2ncnc3cc(NC(=O)c4ccc(C(=O)Nc5ccccc5N)nc4)ccc23)c1 ZINC000147337229 JJ Annotated Mild MAPK4 0 47 CCCCCCCCNS(=O)(=O)c1cnccc1NCC ZINC000147337331 DG For-Sale Mild Q95J97_RABIT 0 40 Cc1cc(C)n(-c2ccc(NC(=O)N[C@@H]3CCCN(S(C)(=O)=O)C3)cn2)n1 ZINC000147337332 GD On-Demand Anodyne EPHX2 27 40 COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1OC ZINC000147337396 GC On-Demand Anodyne ADRA1D 24 48 COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1OC ZINC000147337396 GC On-Demand Anodyne ADRA1A 17 48 COc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1OC ZINC000147337396 GC On-Demand Anodyne ADRA1B 34 48 CCCNc1cccc(NC[C@@H]2CCCO2)n1 ZINC000147337449 BE For-Sale Anodyne TNK2 62 39 Cc1ccc(S(=O)(=O)OC[C@@H]2NC(=O)[C@H]2NC(=O)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)cc1 ZINC000147337505 KD For-Sale Mild REN 40 38 CC[C@H]1CN(C(=O)[C@@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337533 HD On-Demand Anodyne P2RY12 89 35 CC[C@H]1CN(C(=O)[C@@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337533 HD On-Demand Anodyne MC4R 58 41 CC[C@H]1CN(C(=O)[C@@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337533 HD On-Demand Anodyne CCR1 43 45 CC[C@H]1CN(C(=O)[C@@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337533 HD On-Demand Anodyne UTS2 45 36 Cc1cc(C)n(-c2ccc(NC(=O)N[C@H]3CCCN(S(C)(=O)=O)C3)cn2)n1 ZINC000147337545 GD On-Demand Anodyne EPHX2 27 40 CCCCCCCCNS(=O)(=O)c1cnccc1N ZINC000147337565 CE For-Sale Mild CA14 0 40 C[C@H](C(=O)NN1CCCCC1)[C@H](N)c1ccccc1 ZINC000147337570 CD For-Sale Anodyne KCNQ2 53 42 O=C(c1cc2ncccn2n1)N1CCN(Cc2cccc(Cl)c2)CC1 ZINC000147337649 FE On-Demand Anodyne DRD4 16 42 O=C(c1cc2ncccn2n1)N1CCN(Cc2cccc(Cl)c2)CC1 ZINC000147337649 FE On-Demand Anodyne FAAH 33 48 COc1cc(C)ccc1Oc1nc(N)cn2ccnc12 ZINC000147337666 CE For-Sale Anodyne SYK 27 40 COc1cc(C)ccc1Oc1nc(N)cn2ccnc12 ZINC000147337666 CE For-Sale Anodyne HIVRT 0 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(C)c(Cc3cccc(Cl)c3)s2)c1 ZINC000147337668 HJ On-Demand Bother CSNK1D 25 49 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(C)c(Cc3cccc(Cl)c3)s2)c1 ZINC000147337668 HJ On-Demand Bother TAAR1 24 42 CCCNc1cccc(NC[C@H]2CCCO2)n1 ZINC000147337674 BE For-Sale Anodyne TNK2 62 39 CC(C)CCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147337734 CG On-Demand Anodyne CACNA1H 24 40 CC(C)CCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147337734 CG On-Demand Anodyne CACNA1I 42 33 CC[C@@H]1CN(C(=O)[C@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337768 HD On-Demand Anodyne P2RY12 89 35 CC[C@@H]1CN(C(=O)[C@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337768 HD On-Demand Anodyne MC4R 58 41 CC[C@@H]1CN(C(=O)[C@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337768 HD On-Demand Anodyne CCR1 43 45 CC[C@@H]1CN(C(=O)[C@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337768 HD On-Demand Anodyne CCKBR 86 38 CC[C@@H]1CN(C(=O)[C@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337768 HD On-Demand Anodyne UTS2 45 36 CCCCCCCCNC(=O)c1cccnc1N ZINC000147337772 BF For-Sale Mild SCNN1A 33 40 CCCCCCCCNC(=O)c1cccnc1N ZINC000147337772 BF For-Sale Mild FAAH 24 42 CCCCCCCCNC(=O)c1cccnc1N ZINC000147337772 BF For-Sale Mild ASAH1 95 37 CCCCCCCCNC(=O)c1cccnc1N ZINC000147337772 BF For-Sale Mild ACAT 0 44 C[C@@H](C(=O)NN1CCCCC1)[C@H](N)c1ccccc1 ZINC000147337775 CD For-Sale Anodyne KCNQ2 53 42 Cc1c(O)cc2c(c1C)OCCC2 ZINC000147337781 AE For-Sale Anodyne ILK 0 40 Cc1cc(C)c(OCCN2CCCCC2)c(S(N)(=O)=O)c1 ZINC000147337807 DD For-Sale Anodyne HRH3 24 43 Cc1cc(C)c(OCCN2CCCCC2)c(S(N)(=O)=O)c1 ZINC000147337807 DD For-Sale Anodyne PSMB2 48 40 Cc1cc(C)c(OCCN2CCCCC2)c(S(N)(=O)=O)c1 ZINC000147337807 DD For-Sale Anodyne PSMB5 17 40 Cc1cc(C)c(OCCN2CCCCC2)c(S(N)(=O)=O)c1 ZINC000147337807 DD For-Sale Anodyne PSMB1 42 40 Cc1cc(C)n(-c2ccc(NC(=O)NCc3ccc(-n4ccnc4)c(F)c3)cn2)n1 ZINC000147337825 HH On-Demand Anodyne NOS2 75 34 Cc1cc(C)n(-c2ccc(NC(=O)NCc3ccc(-n4ccnc4)c(F)c3)cn2)n1 ZINC000147337825 HH On-Demand Anodyne NAMPT 27 47 CC(C)c1nc(NN)cc(OCCCc2ccccc2)n1 ZINC000147337876 CF For-Sale Anodyne SIGMAR1 15 40 Cc1ccc(S(=O)(=O)OC[C@@H]2NC(=O)[C@@H]2NC(=O)[C@H](NC(=O)OC(C)(C)C)c2ccccc2)cc1 ZINC000147337912 KD For-Sale Mild REN 40 38 CCCCCCCCNC(=O)c1ccnc(NCC)c1 ZINC000147337977 CH For-Sale Mild ASAH1 82 36 CCCCCCCCNC(=O)c1ccnc(NCC)c1 ZINC000147337977 CH For-Sale Mild KDM4E 24 42 CC[C@H]1CN(C(=O)[C@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337981 HD On-Demand Anodyne P2RY12 89 35 CC[C@H]1CN(C(=O)[C@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337981 HD On-Demand Anodyne MC4R 58 41 CC[C@H]1CN(C(=O)[C@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337981 HD On-Demand Anodyne CCR1 43 45 CC[C@H]1CN(C(=O)[C@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337981 HD On-Demand Anodyne CCKBR 86 38 CC[C@H]1CN(C(=O)[C@H](CCS(C)(=O)=O)NC(=O)c2ccc(Cl)cc2)CCO1 ZINC000147337981 HD On-Demand Anodyne UTS2 45 36 C[C@H](C(=O)NN1CCCCC1)[C@@H](N)c1ccccc1 ZINC000147337990 CD For-Sale Anodyne KCNQ2 53 42 COc1ccc([N+](=O)[O-])cc1CNC1(C(=O)O)CCC1 ZINC000147338088 CD For-Sale Bother CACNA1C 43 36 COc1ccc([N+](=O)[O-])cc1CNC1(C(=O)O)CCC1 ZINC000147338088 CD For-Sale Bother CACNA1D 73 33 COc1ccc([N+](=O)[O-])cc1CNC1(C(=O)O)CCC1 ZINC000147338088 CD For-Sale Bother KCNMA1 19 40 O=C(c1cc2ncccn2n1)N1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147338106 FE On-Demand Anodyne DRD4 35 41 O=C(c1cc2ncccn2n1)N1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147338106 FE On-Demand Anodyne LSS 18 53 O=C(c1cc2ncccn2n1)N1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147338106 FE On-Demand Anodyne FAAH 31 45 CCCCCCCCNC(=O)c1ccnc(NC)c1 ZINC000147338171 CG For-Sale Mild THRB 0 49 CCCCCCCCNC(=O)c1ccnc(NC)c1 ZINC000147338171 CG For-Sale Mild LPAR2 40 33 CCCCCCCCNC(=O)c1ccnc(NC)c1 ZINC000147338171 CG For-Sale Mild S1PR2 51 33 CCCCCCCCNC(=O)c1ccnc(NC)c1 ZINC000147338171 CG For-Sale Mild HDAC9 16 41 CCCCCCCCNC(=O)c1ccnc(NC)c1 ZINC000147338171 CG For-Sale Mild ASAH1 83 36 CCCCCCCCNC(=O)c1ccnc(NC)c1 ZINC000147338171 CG For-Sale Mild KDM4E 25 46 O=C(NCC1(O)CCCC1)c1cccc2c1OCCN2 ZINC000147338183 CD For-Sale Anodyne HCN1 52 34 O=C(NCC1(O)CCCC1)c1cccc2c1OCCN2 ZINC000147338183 CD For-Sale Anodyne HCN4 47 30 C[C@@H](C(=O)NN1CCCCC1)[C@@H](N)c1ccccc1 ZINC000147338185 CD For-Sale Anodyne KCNQ2 53 42 CC[C@H]1CN(C(=O)c2cc(S(=O)(=O)N(C)C)ccc2N2CCCC2)CCO1 ZINC000147338210 GD On-Demand Anodyne SLC6A9 29 44 CN(C)C(=O)NCCn1c(S)nc2ccccc2c1=O ZINC000147338253 CC For-Sale Anodyne POLR1A 60 34 CCCOCC(=O)NCCCCCCC(C)C ZINC000147338353 BG For-Sale Anodyne NOD1 62 40 CC(=O)Nc1cc(NC(=O)C(=O)NC[C@@H]2CCCCO2)ccc1F ZINC000147338371 ED On-Demand Anodyne ENV 42 35 O=C(NCC1(O)CCCCC1)c1cccc2c1OCCN2 ZINC000147338384 CD For-Sale Anodyne HCN1 54 36 O=C(NCC1(O)CCCCC1)c1cccc2c1OCCN2 ZINC000147338384 CD For-Sale Anodyne HCN4 50 32 CCCCCCCCNC(=O)c1cccnc1NCC ZINC000147338423 CH For-Sale Mild MERTK 32 41 CCCCCCCCNC(=O)c1cccnc1NCC ZINC000147338423 CH For-Sale Mild ASAH1 85 35 CC(=O)Nc1cc(NC(=O)C(=O)NC[C@H]2CCCCO2)ccc1F ZINC000147338589 ED On-Demand Anodyne ENV 42 35 CCCCCCCCNC(=O)c1ccnc(NCCC)c1 ZINC000147338611 CH For-Sale Mild LPAR2 58 34 CCCCCCCCNC(=O)c1ccnc(NCCC)c1 ZINC000147338611 CH For-Sale Mild S1PR2 76 35 CCCCCCCCNC(=O)c1ccnc(NCCC)c1 ZINC000147338611 CH For-Sale Mild ASAH1 82 36 CCCCCCCCNC(=O)c1ccnc(NCCC)c1 ZINC000147338611 CH For-Sale Mild KDM4E 24 42 CC(C)CCCCNC(=O)CC1(C(=O)O)CCCCC1 ZINC000147338791 CG For-Sale Anodyne CETP 17 41 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne OPRD1 19 46 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne FOLH1 45 33 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne ANPEP 17 47 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne EDNRB 22 45 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne EDNRA 22 46 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne CPB2 19 43 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne KLK3 62 35 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne PAPA1_CARPA 45 32 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne NTSR1 121 44 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne NTSR2 92 44 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne ADRBK1 16 49 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne HLA-A 97 50 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne MC5R 32 41 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne LNPEP 23 45 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne FURIN 63 45 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne SORT1 49 37 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne ENPEP 77 46 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne MC1R 24 41 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne CASP6 20 41 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne GART 42 31 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne SIRT1 34 51 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne F2RL1 57 36 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne DLG4 57 32 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne WDR5 30 49 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne NOD1 60 38 CC[C@H](C)[C@H](NC(=O)[C@H](N)Cc1cnc[nH]1)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCC(=O)O)C(=O)O ZINC000147338808 KA For-Sale Anodyne HPN 38 41 CCCCCCCCNC(=O)c1ccnc(N)c1 ZINC000147338823 BF For-Sale Mild KCNQ1 0 42 CCCCCCCCNC(=O)c1ccnc(N)c1 ZINC000147338823 BF For-Sale Mild S1PR2 44 31 CCCCCCCCNC(=O)c1ccnc(N)c1 ZINC000147338823 BF For-Sale Mild ASAH1 91 37 CCCCCCCCNC(=O)c1ccnc(N)c1 ZINC000147338823 BF For-Sale Mild ACAT 0 41 CCCCCCCCNC(=O)c1ccnc(N)c1 ZINC000147338823 BF For-Sale Mild KDM4E 34 47 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147338842 FA For-Sale Anodyne TOP1 58 39 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147338842 FA For-Sale Anodyne ADORA1 27 41 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147338842 FA For-Sale Anodyne SLC29A1 76 35 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147338842 FA For-Sale Anodyne P2RY6 63 63 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147338842 FA For-Sale Anodyne TK1 49 47 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147338842 FA For-Sale Anodyne CDA 76 46 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147338842 FA For-Sale Anodyne P2RY4 49 39 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147338842 FA For-Sale Anodyne P2RY2 51 39 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147338842 FA For-Sale Anodyne P2RY14 68 40 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147338842 FA For-Sale Anodyne RNASE1 15 45 O=C(Nc1ccc(I)cc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147338848 JI For-Sale Anodyne AKR1C3 18 41 O=C(Nc1ccc(I)cc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147338848 JI For-Sale Anodyne MTCA1 25 45 O=C(Nc1ccc(I)cc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147338848 JI For-Sale Anodyne P96878_MYCTU 25 45 O=C(Nc1cc(N2CCCS2(=O)=O)ccc1F)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147338913 HH On-Demand Anodyne CDK1 19 44 CC(=O)Nc1ccc(C)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147338957 GC On-Demand Anodyne CCR8 76 35 CC(=O)Nc1ccc(C)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147338957 GC On-Demand Anodyne SFRP1 57 31 CC(=O)Nc1ccc(C)c(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147338957 GC On-Demand Anodyne WNT3 41 31 CCOC(=O)c1ccc(NC(=O)CSCCC(=O)N2CCO[C@@H](CC)C2)cc1 ZINC000147338960 HF On-Demand Anodyne SLC27A1 18 42 N#Cc1cccc(OC2CCN(C(=O)C(N)=O)CC2)c1 ZINC000147338980 CC On-Demand Mild HRH1 22 48 N#Cc1cccc(OC2CCN(C(=O)C(N)=O)CC2)c1 ZINC000147338980 CC On-Demand Mild KCNH2 41 37 N#Cc1cccc(OC2CCN(C(=O)C(N)=O)CC2)c1 ZINC000147338980 CC On-Demand Mild PRSS2 71 33 N#Cc1cccc(OC2CCN(C(=O)C(N)=O)CC2)c1 ZINC000147338980 CC On-Demand Mild CCR3 32 48 N#Cc1cccc(OC2CCN(C(=O)C(N)=O)CC2)c1 ZINC000147338980 CC On-Demand Mild EPHX2 16 56 N#Cc1cccc(OC2CCN(C(=O)C(N)=O)CC2)c1 ZINC000147338980 CC On-Demand Mild TNKS 21 42 O=C(O)c1ccc(SCc2cccc(Cl)c2)cn1 ZINC000147338983 CH For-Sale Anodyne KMO 0 40 O=C(O)c1ccc(SCc2cccc(Cl)c2)cn1 ZINC000147338983 CH For-Sale Anodyne P4HTM 0 40 CCCCCCCCNC(=O)c1cc(Br)cnc1NCC ZINC000147338993 FI For-Sale Mild MERTK 25 42 CCCCCCCCNC(=O)c1cc(Br)cnc1NCC ZINC000147338993 FI For-Sale Mild ASAH1 68 34 Ic1ccc(-c2nccn2CCCc2ccccc2)cc1 ZINC000147339005 GJ For-Sale Anodyne PDE6D 17 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(C)c(Cc3ccccc3F)s2)c1 ZINC000147339008 HI On-Demand Bother TAAR1 24 41 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@H]2O)c(=O)[nH]1 ZINC000147339058 FA For-Sale Anodyne TOP1 58 39 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@H]2O)c(=O)[nH]1 ZINC000147339058 FA For-Sale Anodyne ADORA1 27 41 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@H]2O)c(=O)[nH]1 ZINC000147339058 FA For-Sale Anodyne SLC29A1 76 35 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@H]2O)c(=O)[nH]1 ZINC000147339058 FA For-Sale Anodyne P2RY6 63 63 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@H]2O)c(=O)[nH]1 ZINC000147339058 FA For-Sale Anodyne TK1 49 47 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@H]2O)c(=O)[nH]1 ZINC000147339058 FA For-Sale Anodyne CDA 76 46 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@H]2O)c(=O)[nH]1 ZINC000147339058 FA For-Sale Anodyne P2RY4 49 39 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@H]2O)c(=O)[nH]1 ZINC000147339058 FA For-Sale Anodyne P2RY2 51 39 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@H]2O)c(=O)[nH]1 ZINC000147339058 FA For-Sale Anodyne P2RY14 68 40 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@H](O)[C@H]2O)c(=O)[nH]1 ZINC000147339058 FA For-Sale Anodyne RNASE1 15 45 Cc1ccc(C(=O)O)cc1NC(=O)c1ocnc1C ZINC000147339088 CE On-Demand Anodyne MAPK14 43 39 Cc1ccc(C(=O)O)cc1NC(=O)c1ocnc1C ZINC000147339088 CE On-Demand Anodyne GPR35 51 36 C#CC(C)(C)NC(=O)OCc1ccccc1 ZINC000147339090 BE For-Sale Mild BMP1 43 33 C#CC(C)(C)NC(=O)OCc1ccccc1 ZINC000147339090 BE For-Sale Mild POL 0 42 C#CC(C)(C)NC(=O)OCc1ccccc1 ZINC000147339090 BE For-Sale Mild 17HSDCL 0 40 C#CC(C)(C)NC(=O)OCc1ccccc1 ZINC000147339090 BE For-Sale Mild HISB 0 40 O=C(Nc1cc(N2CCCS2(=O)=O)ccc1F)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147339094 HH On-Demand Anodyne CDK1 19 44 O=C(Nc1ccc(I)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339107 HI For-Sale Anodyne PPIA 23 49 O=C(Nc1ccc(I)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339107 HI For-Sale Anodyne EPHX2 17 44 O=C(Nc1ccc(I)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339107 HI For-Sale Anodyne CA12 16 45 O=C(Nc1ccc(I)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339107 HI For-Sale Anodyne AKR1C3 20 42 O=C(Nc1ccc(I)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339107 HI For-Sale Anodyne NCE103 20 42 O=C(Nc1ccc(I)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339107 HI For-Sale Anodyne MTCA1 25 45 O=C(Nc1ccc(I)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339107 HI For-Sale Anodyne P96878_MYCTU 25 45 O=C(Nc1ccc(I)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339107 HI For-Sale Anodyne HCAR1 0 42 O=C(Nc1ccc(I)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339107 HI For-Sale Anodyne Q25615_ONCVO 52 40 O=C(Nc1ccc(I)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339107 HI For-Sale Anodyne P95276_MYCTO 0 44 CC(=O)Nc1ccc(C)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147339118 GC On-Demand Anodyne CCR8 76 35 CC(=O)Nc1ccc(C)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147339118 GC On-Demand Anodyne SFRP1 57 31 CC(=O)Nc1ccc(C)c(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147339118 GC On-Demand Anodyne WNT3 41 31 CCCCCCCCNC(=O)c1ccc(C)cc1NC ZINC000147339158 CI For-Sale Mild S1PR2 46 35 CCCCCCCCNC(=O)c1ccc(C)cc1NC ZINC000147339158 CI For-Sale Mild PA2A1_NAJMO 0 42 CCCCCCCCNC(=O)c1ccc(C)cc1NC ZINC000147339158 CI For-Sale Mild ASAH1 92 38 CCCCCCCCNC(=O)c1ccc(C)cc1NC ZINC000147339158 CI For-Sale Mild ACAT 0 52 CCCCCCCCNC(=O)c1ccc(C)cc1NC ZINC000147339158 CI For-Sale Mild PSBA 0 40 CC[C@H](CNS(=O)(=O)Cc1cccc(C#N)c1)CC(=O)O ZINC000147339207 DD On-Demand Mild MMP12 0 43 Nc1nc(Oc2cccnc2)nc(N2CCCCC2)n1 ZINC000147339222 CD For-Sale Anodyne ERM 0 42 O=C(c1cc2ncccn2n1)N1CCN(Cc2cccc(C(F)(F)F)c2)CC1 ZINC000147339225 GF On-Demand Anodyne ABL1 21 40 O=C(c1cc2ncccn2n1)N1CCN(Cc2cccc(C(F)(F)F)c2)CC1 ZINC000147339225 GF On-Demand Anodyne FAAH 22 51 O=C(c1cc2ncccn2n1)N1CCN(Cc2cccc(C(F)(F)F)c2)CC1 ZINC000147339225 GF On-Demand Anodyne RBP4 16 42 O=C(c1cc2ncccn2n1)N1CCN(Cc2cccc(C(F)(F)F)c2)CC1 ZINC000147339225 GF On-Demand Anodyne SCD1 24 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(C)c(Cc3cccc(C)c3)s2)c1 ZINC000147339241 GJ On-Demand Bother CSNK1D 20 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(C)c(Cc3cccc(C)c3)s2)c1 ZINC000147339241 GJ On-Demand Bother SCD 15 40 CC(C)(C)OC(=O)NC[C@@H]1CCN(c2ccccc2F)C1 ZINC000147339304 CG On-Demand Anodyne ACACA 28 42 COc1cc(Cl)ccc1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147339318 FH For-Sale Reactive DRD2 36 40 COc1cc(Cl)ccc1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147339318 FH For-Sale Reactive HTR4 48 37 COc1cc(Cl)ccc1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147339318 FH For-Sale Reactive ACKR3 42 29 O=C(Nc1cccc(I)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147339319 JI For-Sale Anodyne PPIA 22 40 O=C(Nc1cccc(I)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147339319 JI For-Sale Anodyne AKR1C3 30 44 O=C(Nc1cccc(I)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147339319 JI For-Sale Anodyne KCNK3 50 33 O=C(Nc1cc(N2CCCS2(=O)=O)ccc1F)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147339333 HH On-Demand Anodyne CDK1 19 44 Cc1ccc2c(C3=CCN(C[C@@H](O)COc4cccc5[nH]ccc45)CC3)c[nH]c2c1 ZINC000147339357 HI On-Demand Anodyne ADRB2 33 46 Cc1ccc2c(C3=CCN(C[C@@H](O)COc4cccc5[nH]ccc45)CC3)c[nH]c2c1 ZINC000147339357 HI On-Demand Anodyne ADRB1 17 43 Cc1ccc2c(C3=CCN(C[C@@H](O)COc4cccc5[nH]ccc45)CC3)c[nH]c2c1 ZINC000147339357 HI On-Demand Anodyne HTR1A 36 60 Cc1ccc2c(C3=CCN(C[C@@H](O)COc4cccc5[nH]ccc45)CC3)c[nH]c2c1 ZINC000147339357 HI On-Demand Anodyne SLC6A4 35 47 Cc1ccc2c(C3=CCN(C[C@@H](O)COc4cccc5[nH]ccc45)CC3)c[nH]c2c1 ZINC000147339357 HI On-Demand Anodyne ADRB3 35 46 Cc1ccc2c(C3=CCN(C[C@@H](O)COc4cccc5[nH]ccc45)CC3)c[nH]c2c1 ZINC000147339357 HI On-Demand Anodyne ABCB1 40 38 CCCCCCCCNC(=O)c1nnc(N)s1 ZINC000147339380 CE For-Sale Mild ASAH1 81 34 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147339407 CF On-Demand Anodyne NPY2R 19 40 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147339407 CF On-Demand Anodyne CCKBR 27 40 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147339407 CF On-Demand Anodyne EPHX2 22 48 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147339407 CF On-Demand Anodyne AKR1C3 53 49 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147339407 CF On-Demand Anodyne RHOA 0 43 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147339407 CF On-Demand Anodyne PARP15 0 46 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147339407 CF On-Demand Anodyne KCNK3 89 53 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147339407 CF On-Demand Anodyne KCNK9 41 36 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147339407 CF On-Demand Anodyne PARP10 0 48 CC[C@@H](CNS(=O)(=O)Cc1cccc(C#N)c1)CC(=O)O ZINC000147339416 DD On-Demand Mild MMP12 0 43 Cc1ccc(Br)cc1S(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000147339419 HD On-Demand Anodyne CTSC 18 47 CC(C)(C)OC(=O)NC[C@H]1CCN(c2ccccc2F)C1 ZINC000147339461 CG On-Demand Anodyne ACACA 28 42 Cc1ccccc1-n1nc(C(=O)NCc2cccnc2-n2ccnc2)c2c1CCC2 ZINC000147339474 GG On-Demand Anodyne NOS2 92 33 COc1cc(Cl)ccc1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147339480 FH For-Sale Reactive DRD2 36 40 COc1cc(Cl)ccc1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147339480 FH For-Sale Reactive HTR4 48 37 COc1cc(Cl)ccc1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147339480 FH For-Sale Reactive ACKR3 42 29 Cc1cnn(CC(=O)N(CC(=O)Nc2ccccc2F)Cc2ccc(Cl)cc2)c1 ZINC000147339490 HH On-Demand Anodyne PLA2G7 78 40 Cc1cnn(CC(=O)N(CC(=O)Nc2ccccc2F)Cc2ccc(Cl)cc2)c1 ZINC000147339490 HH On-Demand Anodyne FFAR2 43 34 CCOc1cccc(Oc2cc(NN)nc(C(C)C)n2)c1 ZINC000147339493 CG For-Sale Anodyne ACACA 0 41 O=C(Nc1cccc(I)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339538 HI For-Sale Anodyne PPIA 33 60 O=C(Nc1cccc(I)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339538 HI For-Sale Anodyne P2RY1 0 47 O=C(Nc1cccc(I)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339538 HI For-Sale Anodyne EPHX2 18 43 O=C(Nc1cccc(I)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339538 HI For-Sale Anodyne AKR1C3 33 49 O=C(Nc1cccc(I)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339538 HI For-Sale Anodyne NCE103 16 40 O=C(Nc1cccc(I)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147339538 HI For-Sale Anodyne KCNK3 59 43 CCCCCCCCNC(=O)c1cc(NC)ccn1 ZINC000147339551 CG For-Sale Mild LPAR2 53 32 CCCCCCCCNC(=O)c1cc(NC)ccn1 ZINC000147339551 CG For-Sale Mild S1PR2 64 33 CCCCCCCCNC(=O)c1cc(NC)ccn1 ZINC000147339551 CG For-Sale Mild ASAH1 88 36 Cc1cc(C(=O)Nc2ccc3ccccc3n2)cc([N+](=O)[O-])c1 ZINC000147339577 DH On-Demand Bother KCNK3 40 34 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@@H]23)c1 ZINC000147339589 CF For-Sale Anodyne CCKBR 27 40 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@@H]23)c1 ZINC000147339589 CF For-Sale Anodyne RHOA 0 43 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@@H]23)c1 ZINC000147339589 CF For-Sale Anodyne PARP15 0 46 O=C(O)c1cccc(NC(=O)C2[C@H]3CCCC[C@@H]23)c1 ZINC000147339589 CF For-Sale Anodyne PARP10 0 48 CCCOCC(=O)NCc1cccnc1-n1ccnc1 ZINC000147339666 CD On-Demand Anodyne NOS2 84 35 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147339688 HG On-Demand Anodyne DRD4 42 35 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147339688 HG On-Demand Anodyne KCNK3 52 38 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147339688 HG On-Demand Anodyne KCNK9 42 38 CCCNc1cn2ccnc2c(Oc2cccnc2)n1 ZINC000147339757 CF For-Sale Anodyne HIVRT 0 40 CC[C@@H](C)c1ccc([C@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147339759 GK On-Demand Anodyne BMP1 47 33 CC[C@@H](C)c1ccc([C@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147339759 GK On-Demand Anodyne CYP3A4 17 43 O=C(O)c1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147339787 CF On-Demand Anodyne NPY2R 19 40 O=C(O)c1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147339787 CF On-Demand Anodyne CCKBR 27 40 O=C(O)c1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147339787 CF On-Demand Anodyne EPHX2 22 48 O=C(O)c1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147339787 CF On-Demand Anodyne AKR1C3 53 49 O=C(O)c1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147339787 CF On-Demand Anodyne RHOA 0 43 O=C(O)c1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147339787 CF On-Demand Anodyne PARP15 0 46 O=C(O)c1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147339787 CF On-Demand Anodyne KCNK3 89 53 O=C(O)c1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147339787 CF On-Demand Anodyne KCNK9 41 36 O=C(O)c1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147339787 CF On-Demand Anodyne PARP10 0 48 Cc1cccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147339826 HG On-Demand Anodyne DRD4 42 35 Cc1cccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147339826 HG On-Demand Anodyne KCNK3 52 38 Cc1cccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147339826 HG On-Demand Anodyne KCNK9 42 38 O=C(COc1cccc(Cl)c1)N1CCC[C@H](CCBr)C1 ZINC000147339848 FH For-Sale Reactive COLA 84 46 O=C(COc1cccc(Cl)c1)N1CCC[C@H](CCBr)C1 ZINC000147339848 FH For-Sale Reactive CPT1A 75 46 O=C(COc1cccc(Cl)c1)N1CCC[C@H](CCBr)C1 ZINC000147339848 FH For-Sale Reactive CPT2 45 46 CCCCCCCCNC(=O)c1cccnc1NC ZINC000147339854 CG For-Sale Mild S1PR2 42 33 CCCCCCCCNC(=O)c1cccnc1NC ZINC000147339854 CG For-Sale Mild ASAH1 87 36 CCN(CC)CC(=O)Nc1ccc(NC(=O)c2cccnc2)c(OC)c1 ZINC000147339882 FF On-Demand Anodyne GRM4 18 43 CCN(CC)CC(=O)Nc1ccc(NC(=O)c2cccnc2)c(OC)c1 ZINC000147339882 FF On-Demand Anodyne HDAC1 18 41 CCN(CC)CC(=O)Nc1ccc(NC(=O)c2cccnc2)c(OC)c1 ZINC000147339882 FF On-Demand Anodyne ABCB1 15 43 CCN(CC)CC(=O)Nc1ccc(NC(=O)c2cccnc2)c(OC)c1 ZINC000147339882 FF On-Demand Anodyne CSF1R 15 43 CCN(CC)CC(=O)Nc1ccc(NC(=O)c2cccnc2)c(OC)c1 ZINC000147339882 FF On-Demand Anodyne ENPP1 58 35 CCCCO[C@H](C)C(=O)NCc1cccnc1-n1ccnc1 ZINC000147339918 DE On-Demand Anodyne TBXAS1 42 39 CCCCO[C@H](C)C(=O)NCc1cccnc1-n1ccnc1 ZINC000147339918 DE On-Demand Anodyne CYP2C19 17 44 CC[C@H](C)c1ccc([C@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147339932 GK On-Demand Anodyne BMP1 47 33 CC[C@H](C)c1ccc([C@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147339932 GK On-Demand Anodyne CYP3A4 17 43 CC[C@H](CNS(=O)(=O)Cc1ccc(C#N)cc1)CC(=O)O ZINC000147339975 DD On-Demand Mild MMP12 0 46 CC[C@H](CNS(=O)(=O)Cc1ccc(C#N)cc1)CC(=O)O ZINC000147339975 DD On-Demand Mild CTRB_BOVIN 45 33 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1 ZINC000147339995 BD On-Demand Anodyne MAPK14 17 40 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1 ZINC000147339995 BD On-Demand Anodyne PRNP 31 42 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1 ZINC000147339995 BD On-Demand Anodyne NR1H4 15 48 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1 ZINC000147339995 BD On-Demand Anodyne CCKBR 0 41 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1 ZINC000147339995 BD On-Demand Anodyne AKR1C3 47 49 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1 ZINC000147339995 BD On-Demand Anodyne CYA 0 44 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1 ZINC000147339995 BD On-Demand Anodyne PARP15 0 43 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1 ZINC000147339995 BD On-Demand Anodyne KCNK3 106 49 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1 ZINC000147339995 BD On-Demand Anodyne KCNK9 90 49 Cc1ncoc1C(=O)Nc1cccc(C(=O)O)c1 ZINC000147339995 BD On-Demand Anodyne PARP10 0 43 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147339998 HG On-Demand Anodyne DRD4 42 35 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147339998 HG On-Demand Anodyne KCNK3 52 38 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147339998 HG On-Demand Anodyne KCNK9 42 38 CNc1cn2ccnc2c(Oc2cccnc2)n1 ZINC000147340000 BD For-Sale Anodyne HIVRT 0 43 O=C(Nc1cc(Cl)cc(C(=O)O)c1)Nc1ccccc1I ZINC000147340003 HI For-Sale Anodyne PPIA 26 48 O=C(Nc1cc(Cl)cc(C(=O)O)c1)Nc1ccccc1I ZINC000147340003 HI For-Sale Anodyne LPL 44 35 O=C(Nc1cc(Cl)cc(C(=O)O)c1)Nc1ccccc1I ZINC000147340003 HI For-Sale Anodyne AKR1C3 25 41 CCCCCCCCNC(=O)c1cc(N)ccc1[N+](=O)[O-] ZINC000147340018 CG For-Sale Mild ASAH1 75 34 O=C(COc1cccc(Cl)c1)N1CCC[C@@H](CCBr)C1 ZINC000147340021 FH For-Sale Reactive COLA 84 46 O=C(COc1cccc(Cl)c1)N1CCC[C@@H](CCBr)C1 ZINC000147340021 FH For-Sale Reactive CPT1A 75 46 O=C(COc1cccc(Cl)c1)N1CCC[C@@H](CCBr)C1 ZINC000147340021 FH For-Sale Reactive CPT2 45 46 CC[C@@H](C)c1ccc([C@@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147340062 GK On-Demand Anodyne BMP1 47 33 CC[C@@H](C)c1ccc([C@@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147340062 GK On-Demand Anodyne CYP3A4 17 43 CC[C@@H](CNS(=O)(=O)Cc1ccc(C#N)cc1)CC(=O)O ZINC000147340127 DD On-Demand Mild MMP12 0 46 CC[C@@H](CNS(=O)(=O)Cc1ccc(C#N)cc1)CC(=O)O ZINC000147340127 DD On-Demand Mild CTRB_BOVIN 45 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1-n1ccnc1 ZINC000147340147 ED On-Demand Anodyne PCSK5 52 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1-n1ccnc1 ZINC000147340147 ED On-Demand Anodyne FURIN 57 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1-n1ccnc1 ZINC000147340147 ED On-Demand Anodyne POLG_WNV 49 29 CCCCCCCCNC(=O)c1ccc(NCC)c(C)c1 ZINC000147340150 CJ For-Sale Mild FOLH1 19 43 CCCCCCCCNC(=O)c1ccc(NCC)c(C)c1 ZINC000147340150 CJ For-Sale Mild THRB 0 49 CCCCCCCCNC(=O)c1ccc(NCC)c(C)c1 ZINC000147340150 CJ For-Sale Mild KCNQ1 0 44 CCCCCCCCNC(=O)c1ccc(NCC)c(C)c1 ZINC000147340150 CJ For-Sale Mild ASAH1 74 36 CCCCCCCCNC(=O)c1ccc(NCC)c(C)c1 ZINC000147340150 CJ For-Sale Mild ACAT 0 46 CC[C@H](C)c1ccc([C@@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147340187 GK On-Demand Anodyne BMP1 47 33 CC[C@H](C)c1ccc([C@@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147340187 GK On-Demand Anodyne CYP3A4 17 43 O=C(O)CCCCCNC(=O)c1cccc(F)c1Cl ZINC000147340206 CF On-Demand Anodyne HDA106 0 44 O=C(O)C1(NCc2nc3ccccc3[nH]c2=O)CCC1 ZINC000147340211 CD For-Sale Anodyne PLAUR 38 40 O=C(O)C1(NCc2nc3ccccc3[nH]c2=O)CCC1 ZINC000147340211 CD For-Sale Anodyne STK33 52 39 COc1ccc2c(c1)OC[C@H](C(=O)NCCNC(=O)c1cccc(C)c1)C2 ZINC000147340225 FE On-Demand Anodyne DRD4 53 41 COc1ccc2c(c1)OC[C@H](C(=O)NCCNC(=O)c1cccc(C)c1)C2 ZINC000147340225 FE On-Demand Anodyne NQO2 26 40 COc1ccc2c(c1)OC[C@H](C(=O)NCCNC(=O)c1cccc(C)c1)C2 ZINC000147340225 FE On-Demand Anodyne CTSL 22 45 COc1ccc2c(c1)OC[C@H](C(=O)NCCNC(=O)c1cccc(C)c1)C2 ZINC000147340225 FE On-Demand Anodyne MTNR1A 54 43 COc1ccc2c(c1)OC[C@H](C(=O)NCCNC(=O)c1cccc(C)c1)C2 ZINC000147340225 FE On-Demand Anodyne MTNR1B 43 38 COc1ccc2c(c1)OC[C@H](C(=O)NCCNC(=O)c1cccc(C)c1)C2 ZINC000147340225 FE On-Demand Anodyne KCNK3 49 42 CSc1sc(/N=C/NC(=O)OC(C)(C)C)cc1S(=O)(=O)c1cccc(-c2c(C)cccc2N)c1 ZINC000147340238 KK For-Sale Mild C1S 57 58 O=C(NCC(F)(F)F)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147340244 CF For-Sale Anodyne HCAR1 0 41 CCCCCCCCNC(=O)c1cc(Cl)ccc1NC ZINC000147340310 CI For-Sale Mild CNR1 18 47 CCCCCCCCNC(=O)c1cc(Cl)ccc1NC ZINC000147340310 CI For-Sale Mild CNR2 15 47 CCCCCCCCNC(=O)c1cc(Cl)ccc1NC ZINC000147340310 CI For-Sale Mild S1PR2 48 33 CCCCCCCCNC(=O)c1cc(Cl)ccc1NC ZINC000147340310 CI For-Sale Mild ALPL 43 40 CCCCCCCCNC(=O)c1cc(Cl)ccc1NC ZINC000147340310 CI For-Sale Mild ASAH1 93 38 CCCCCCCCNC(=O)c1cc(Cl)ccc1NC ZINC000147340310 CI For-Sale Mild ACAT 0 46 CCCCCCCCNC(=O)c1cc(Cl)ccc1NC ZINC000147340310 CI For-Sale Mild PSBA 0 52 CC(C)c1ccc([C@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147340411 GK On-Demand Anodyne CYP3A4 20 44 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(C)(=O)=O)c1 ZINC000147340436 HE On-Demand Anodyne PLA2G7 43 39 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(C)(=O)=O)c1 ZINC000147340436 HE On-Demand Anodyne F2R 19 49 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(C)(=O)=O)c1 ZINC000147340436 HE On-Demand Anodyne NR1H4 19 41 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(C)(=O)=O)c1 ZINC000147340436 HE On-Demand Anodyne BRAF 17 40 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(C)(=O)=O)c1 ZINC000147340436 HE On-Demand Anodyne KCNK3 122 44 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(NS(C)(=O)=O)c1 ZINC000147340436 HE On-Demand Anodyne KCNK9 90 44 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne PPIA 16 44 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne KIT 16 44 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne TACR1 17 49 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne CNR2 17 41 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne JUN 20 41 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne LCK 39 41 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne MAPK14 29 46 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne TRPV1 19 42 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne KDR 20 44 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne CCR2 72 45 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne BLK 18 40 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne EPHX2 37 60 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne TEK 31 44 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne MCHR1 15 42 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne BMX 30 40 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne BTK 31 50 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne BRAF 41 43 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne TEC 15 40 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne TXK 25 40 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne TAAR1 45 44 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne AKR1C3 21 48 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne KCNK3 117 55 O=C(Nc1cccc(C(=O)NC2CCCCCC2)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1 ZINC000147340476 JK For-Sale Anodyne KCNK9 73 40 CCCCCCCCNC(=O)c1cc(F)c(NC)c(F)c1 ZINC000147340498 CI For-Sale Mild ASAH1 101 41 CCCCCCCCNC(=O)c1cc(F)c(NC)c(F)c1 ZINC000147340498 CI For-Sale Mild ACAT 0 60 CCCNc1cc(Oc2cccnc2)cc([N+](=O)[O-])c1 ZINC000147340515 CH For-Sale Bother ERO1A 0 40 CC(C)c1ccc([C@@H](NC(=O)N(C)Cc2cscn2)c2cccs2)cc1 ZINC000147340528 GK On-Demand Anodyne CYP3A4 20 44 O=C(Nc1ccc(CCN2CCOCC2)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147340601 GH On-Demand Anodyne EPHX2 29 43 O=C(Nc1ccc(CCN2CCOCC2)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147340601 GH On-Demand Anodyne NAMPT 20 45 C=CCCOCC(=O)Nc1ccc(OCc2cccnc2)c(Cl)c1 ZINC000147340607 EH On-Demand Mild EGFR 33 42 C=CCCOCC(=O)Nc1ccc(OCc2cccnc2)c(Cl)c1 ZINC000147340607 EH On-Demand Mild ERBB2 51 42 CCCCCCCCNC(=O)c1cccc(NCC)n1 ZINC000147340653 CH For-Sale Mild ASAH1 86 36 O=C(Nc1ccc(CCN2CCOCC2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147340785 GH On-Demand Anodyne EPHX2 29 43 O=C(Nc1ccc(CCN2CCOCC2)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147340785 GH On-Demand Anodyne NAMPT 20 45 CCCCCCCCNC(=O)c1cccc(NC)n1 ZINC000147340811 CG For-Sale Mild ASAH1 92 37 C[C@H](OCCCNC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147340861 EG On-Demand Anodyne BMP1 42 33 Cc1ccc(C(=O)NCCCCCC(=O)O)cc1Br ZINC000147340893 EG On-Demand Anodyne HDAC9 33 41 Cc1ccc(C(=O)NCCCCCC(=O)O)cc1Br ZINC000147340893 EG On-Demand Anodyne HDA106 0 49 CCOc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147340953 EH For-Sale Reactive AVPR1A 21 46 CCOc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147340953 EH For-Sale Reactive GRM3 18 55 CCOc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147340953 EH For-Sale Reactive L3MBTL3 57 38 CCCCCCCCNC(=O)c1cc(NCC)ccn1 ZINC000147340965 CH For-Sale Mild ASAH1 87 35 CNc1nc(Oc2cccnc2)nc(N2CCOCC2)n1 ZINC000147340966 CC For-Sale Anodyne PIK3CA 37 50 CNc1nc(Oc2cccnc2)nc(N2CCOCC2)n1 ZINC000147340966 CC For-Sale Anodyne MTOR 29 44 CNc1nc(Oc2cccnc2)nc(N2CCOCC2)n1 ZINC000147340966 CC For-Sale Anodyne PIK3CG 25 44 CNc1nc(Oc2cccnc2)nc(N2CCOCC2)n1 ZINC000147340966 CC For-Sale Anodyne EPHB4 41 37 O=C(Nc1ccc(CCN2CCOCC2)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147340995 GH On-Demand Anodyne EPHX2 29 43 O=C(Nc1ccc(CCN2CCOCC2)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147340995 GH On-Demand Anodyne NAMPT 20 45 C[C@@H](OCCCNC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147341004 EG On-Demand Anodyne BMP1 42 33 CCOc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147341074 EH For-Sale Reactive AVPR1A 21 46 CCOc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147341074 EH For-Sale Reactive GRM3 18 55 CCOc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147341074 EH For-Sale Reactive L3MBTL3 57 38 O=C(Nc1ccc(CCN2CCOCC2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147341164 GH On-Demand Anodyne EPHX2 29 43 O=C(Nc1ccc(CCN2CCOCC2)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147341164 GH On-Demand Anodyne NAMPT 20 45 CCCCCCCCNC(=O)c1ccc(NC)nc1 ZINC000147341172 CG On-Demand Mild FOLH1 23 44 CCCCCCCCNC(=O)c1ccc(NC)nc1 ZINC000147341172 CG On-Demand Mild THRB 0 50 CCCCCCCCNC(=O)c1ccc(NC)nc1 ZINC000147341172 CG On-Demand Mild LPAR2 40 36 CCCCCCCCNC(=O)c1ccc(NC)nc1 ZINC000147341172 CG On-Demand Mild S1PR2 55 36 CCCCCCCCNC(=O)c1ccc(NC)nc1 ZINC000147341172 CG On-Demand Mild EPHX2 38 40 CCCCCCCCNC(=O)c1ccc(NC)nc1 ZINC000147341172 CG On-Demand Mild ASAH1 87 37 CCCCCCCCNC(=O)c1cnc(NC)c(Cl)c1 ZINC000147341293 CH For-Sale Mild LPAR2 57 40 CCCCCCCCNC(=O)c1cnc(NC)c(Cl)c1 ZINC000147341293 CH For-Sale Mild S1PR3 27 40 CCCCCCCCNC(=O)c1cnc(NC)c(Cl)c1 ZINC000147341293 CH For-Sale Mild S1PR2 64 40 CCCCCCCCNC(=O)c1cnc(NC)c(Cl)c1 ZINC000147341293 CH For-Sale Mild ASAH1 82 38 CCOc1ccccc1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147341306 EH For-Sale Reactive HCN1 69 41 CCOc1ccccc1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147341306 EH For-Sale Reactive HCN4 53 41 O=C(O)CCCCCNC(=O)C1[C@@H]2CCCC[C@@H]12 ZINC000147341333 CE On-Demand Anodyne EPHX2 23 44 Cc1cc(C)c(OCc2ccncc2Cl)c(S(N)(=O)=O)c1 ZINC000147341337 EF For-Sale Anodyne CA14 25 40 CCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1OCC ZINC000147341339 HD On-Demand Anodyne ADRA1D 17 40 CCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1OCC ZINC000147341339 HD On-Demand Anodyne ADRA1B 22 40 CCOc1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1OCC ZINC000147341339 HD On-Demand Anodyne SSTR5 41 36 CC(C)CCCCNCc1ccc2c(c1)CC(C)(C)O2 ZINC000147341437 CI For-Sale Anodyne LEF 58 36 CCCCCCCCNC(=O)c1cc(Cl)nc(NCC)c1 ZINC000147341445 DI For-Sale Mild ASAH1 81 36 CCOc1ccccc1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147341454 EH For-Sale Reactive HCN1 69 41 CCOc1ccccc1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147341454 EH For-Sale Reactive HCN4 53 41 O=C(O)CCCCCNC(=O)C1[C@H]2CCCC[C@@H]12 ZINC000147341484 CE For-Sale Anodyne EPHX2 23 44 CCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1OCC ZINC000147341507 HD On-Demand Anodyne ADRA1D 17 40 CCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1OCC ZINC000147341507 HD On-Demand Anodyne ADRA1B 22 40 CCOc1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1OCC ZINC000147341507 HD On-Demand Anodyne SSTR5 41 36 CC[C@@H]1CN(C(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147341591 CE On-Demand Anodyne MLNR 31 40 CC[C@@H]1CN(C(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147341591 CE On-Demand Anodyne EPHX2 48 38 CCCCCCCCNC(=O)c1cccc(N)n1 ZINC000147341630 BF For-Sale Mild GRIA1 45 34 CCCCCCCCNC(=O)c1cccc(N)n1 ZINC000147341630 BF For-Sale Mild FAAH 17 40 CCCCCCCCNC(=O)c1cccc(N)n1 ZINC000147341630 BF For-Sale Mild PA2A1_NAJMO 0 40 CCCCCCCCNC(=O)c1cccc(N)n1 ZINC000147341630 BF For-Sale Mild ASAH1 97 38 CCCCCCCCNC(=O)c1cccc(N)n1 ZINC000147341630 BF For-Sale Mild ACAT 0 48 COc1ccc(-n2nc(C)c3c(Br)ccnc32)cc1 ZINC000147341678 DH For-Sale Anodyne NPBWR1 23 42 O=C(O)CCCCCNC(=O)C1[C@H]2CCCC[C@H]12 ZINC000147341684 CE On-Demand Anodyne EPHX2 23 44 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147341776 CE On-Demand Anodyne MLNR 31 40 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147341776 CE On-Demand Anodyne EPHX2 48 38 CCCCCCCCNC(=O)c1cnccc1NCCC ZINC000147341822 CH For-Sale Mild S1PR2 44 37 CCCCCCCCNC(=O)c1cnccc1NCCC ZINC000147341822 CH For-Sale Mild ASAH1 82 35 CC[C@@H]1CN(C(=O)Nc2ccc(F)cc2)CC[C@H]1N ZINC000147341928 CE On-Demand Anodyne MLNR 31 40 CC[C@@H]1CN(C(=O)Nc2ccc(F)cc2)CC[C@H]1N ZINC000147341928 CE On-Demand Anodyne EPHX2 48 38 CCc1sc(C(C)(C)C)nc1-c1ccccc1 ZINC000147341986 BJ For-Sale Anodyne PTGDR2 37 43 Cc1ccnc(Cl)c1NC(=O)c1cccc2c1OCCN2 ZINC000147342041 DG For-Sale Anodyne G2YM83_BOTF4 74 38 CCCCCCCCNC(=O)c1ccc(C)cc1N ZINC000147342068 CH For-Sale Mild ASAH1 93 37 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2)CC[C@H]1N ZINC000147342069 CE On-Demand Anodyne MLNR 31 40 CC[C@H]1CN(C(=O)Nc2ccc(F)cc2)CC[C@H]1N ZINC000147342069 CE On-Demand Anodyne EPHX2 48 38 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(C)c(Cc3cccc(F)c3)s2)c1 ZINC000147342113 HI On-Demand Bother CSNK1D 19 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(C)c(Cc3cccc(F)c3)s2)c1 ZINC000147342113 HI On-Demand Bother TAAR1 26 40 CC(C)(C)OC(=O)NCCCNCC(F)F ZINC000147342183 BD On-Demand Anodyne CTSK 24 48 Cc1cc(N2CCOCC2)ccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147342209 FD On-Demand Anodyne HRH3 18 44 Cc1cc(N2CCOCC2)ccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147342209 FD On-Demand Anodyne TTK 25 41 C[C@@H](CC(=O)O)NC(=O)c1cccc(F)c1Cl ZINC000147342223 CE On-Demand Anodyne DAC 50 39 C[C@@H](CC(=O)O)NC(=O)c1cccc(F)c1Cl ZINC000147342223 CE On-Demand Anodyne CTSA 51 33 CC(C)[C@@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147342225 CG On-Demand Anodyne HCAR1 0 41 COc1ccc([N+](=O)[O-])cc1S(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000147342233 GC On-Demand Bother ADRA1D 15 52 COc1ccc([N+](=O)[O-])cc1S(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000147342233 GC On-Demand Bother ADRA1B 22 52 COc1ccc([N+](=O)[O-])cc1S(=O)(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1 ZINC000147342233 GC On-Demand Bother TBXA2R 16 43 CC[C@@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147342283 CF On-Demand Anodyne CCKAR 26 42 CC[C@@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147342283 CF On-Demand Anodyne EPHX2 24 40 CC[C@@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147342283 CF On-Demand Anodyne P2RY14 42 37 CC[C@@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147342283 CF On-Demand Anodyne KCNK3 52 39 CC[C@@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147342283 CF On-Demand Anodyne KCNK9 44 39 CCCCCCCCNC(=O)c1cccc(N)c1[N+](=O)[O-] ZINC000147342289 CG For-Sale Mild ASAH1 77 36 CSc1nn(-c2ccccc2)c2cc(NC(=O)NC3CCNCC3)ccc12 ZINC000147342314 GH Annotated Anodyne KHK 0 78 CN(C(=O)Oc1ccc(I)cc1)c1ccccc1 ZINC000147342340 FH For-Sale Anodyne LIPE 28 56 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(C)c(Cc3ccc(F)cc3)s2)c1 ZINC000147342364 HI On-Demand Bother CSNK1D 20 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(C)c(Cc3ccc(F)cc3)s2)c1 ZINC000147342364 HI On-Demand Bother ACAT 40 36 C[C@H](CC(=O)O)NC(=O)c1cccc(F)c1Cl ZINC000147342371 CE On-Demand Anodyne DAC 50 39 C[C@H](CC(=O)O)NC(=O)c1cccc(F)c1Cl ZINC000147342371 CE On-Demand Anodyne CTSA 51 33 CC(C)[C@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147342376 CG On-Demand Anodyne HCAR1 0 41 Cc1cc(N2CCOCC2)ccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147342429 FD On-Demand Anodyne HRH3 18 44 Cc1cc(N2CCOCC2)ccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147342429 FD On-Demand Anodyne TTK 25 41 COc1ccc([N+](=O)[O-])cc1S(=O)(=O)N[C@H]1CCCN(S(C)(=O)=O)C1 ZINC000147342454 GC On-Demand Bother ADRA1D 15 52 COc1ccc([N+](=O)[O-])cc1S(=O)(=O)N[C@H]1CCCN(S(C)(=O)=O)C1 ZINC000147342454 GC On-Demand Bother ADRA1B 22 52 COc1ccc([N+](=O)[O-])cc1S(=O)(=O)N[C@H]1CCCN(S(C)(=O)=O)C1 ZINC000147342454 GC On-Demand Bother TBXA2R 16 43 COCc1nc(C(=O)N[C@H](c2ccccc2)c2ccc(Cl)cc2)cs1 ZINC000147342460 FI On-Demand Anodyne UTS2 43 33 CC[C@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147342501 CF On-Demand Anodyne CCKAR 26 42 CC[C@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147342501 CF On-Demand Anodyne EPHX2 24 40 CC[C@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147342501 CF On-Demand Anodyne P2RY14 42 37 CC[C@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147342501 CF On-Demand Anodyne KCNK3 52 39 CC[C@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147342501 CF On-Demand Anodyne KCNK9 44 39 CCCCCCCCNC(=O)c1nnc(NCCC)s1 ZINC000147342569 CG For-Sale Mild ASAH1 72 33 CSc1nn(-c2ccccc2)c2cc(N3CCCNCC3)ccc12 ZINC000147342589 EH Annotated Anodyne CHRNA4 35 42 CSc1nn(-c2ccccc2)c2cc(N3CCCNCC3)ccc12 ZINC000147342589 EH Annotated Anodyne KHK 0 91 Cc1ccc(O)c(C(=O)Nc2ccc(Cl)cc2Br)c1 ZINC000147342677 EI For-Sale Anodyne F10 29 56 Cc1ccc(O)c(C(=O)Nc2ccc(Cl)cc2Br)c1 ZINC000147342677 EI For-Sale Anodyne KCNMA1 57 59 Cc1ccc(O)c(C(=O)Nc2ccc(Cl)cc2Br)c1 ZINC000147342677 EI For-Sale Anodyne PYK 42 37 Cc1ccc(O)c(C(=O)Nc2ccc(Cl)cc2Br)c1 ZINC000147342677 EI For-Sale Anodyne TMPRSS4 0 50 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(N3CCCC3=O)cc2)C1 ZINC000147342699 HC On-Demand Anodyne AKR1C3 30 58 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(-c3csnn3)cc1)C2 ZINC000147342726 FG On-Demand Anodyne ROCK2 52 59 Cc1ccc2c(c1)O[C@H](CO)CN2C ZINC000147342747 AD For-Sale Anodyne NISCH 25 51 CCCCCCCCNC(=O)c1cc(F)c(N)c(F)c1 ZINC000147342756 CH For-Sale Mild ASAH1 104 42 CC[C@@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@H]1N ZINC000147342772 CF On-Demand Anodyne CCKAR 26 42 CC[C@@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@H]1N ZINC000147342772 CF On-Demand Anodyne EPHX2 24 40 CC[C@@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@H]1N ZINC000147342772 CF On-Demand Anodyne P2RY14 42 37 CC[C@@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@H]1N ZINC000147342772 CF On-Demand Anodyne KCNK3 52 39 CC[C@@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@H]1N ZINC000147342772 CF On-Demand Anodyne KCNK9 44 39 Cc1ccccc1-c1noc(CNC2(C(=O)O)CCC2)n1 ZINC000147342785 CE For-Sale Anodyne S1PR5 16 40 O=C(Nc1nc(C(F)(F)F)cs1)c1csc(-c2ccccc2F)n1 ZINC000147342800 FJ On-Demand Anodyne MPL 70 38 CC[C@H](CNS(=O)(=O)C[C@@H](C)c1ccccc1)CC(=O)O ZINC000147342843 DE For-Sale Anodyne GRIA4 22 43 CCN(CC)CCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147342853 DF On-Demand Anodyne CACNA1H 24 41 CSc1nn(-c2ccccc2)c2cc(N3CC(N4CCNCC4)C3)ccc12 ZINC000147342877 GF Annotated Anodyne KHK 0 80 CNC(=O)c1cccc(NC(=O)C2CCN(c3ncnc4sc(C)c(C)c34)CC2)c1 ZINC000147342879 HH On-Demand Anodyne LIMK2 66 53 CC[C@H](NC(=O)C[C@@H]1CNc2ccccc21)C(=O)O ZINC000147342886 CD On-Demand Anodyne ACE2 57 33 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc(N3CCCC3=O)cc2)C1 ZINC000147342918 HC On-Demand Anodyne AKR1C3 30 58 CC[C@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@H]1N ZINC000147342961 CF On-Demand Anodyne CCKAR 26 42 CC[C@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@H]1N ZINC000147342961 CF On-Demand Anodyne EPHX2 24 40 CC[C@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@H]1N ZINC000147342961 CF On-Demand Anodyne P2RY14 42 37 CC[C@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@H]1N ZINC000147342961 CF On-Demand Anodyne KCNK3 52 39 CC[C@H]1CN(C(=O)Nc2cccc(C)c2)CC[C@H]1N ZINC000147342961 CF On-Demand Anodyne KCNK9 44 39 CCCCCCCCNC(=O)c1ccc(NCC)nn1 ZINC000147342964 CF For-Sale Mild KCNQ1 0 40 CCCCCCCCNC(=O)c1ccc(NCC)nn1 ZINC000147342964 CF For-Sale Mild SCD1 17 46 CCCCCCCCNC(=O)c1ccc(NCC)nn1 ZINC000147342964 CF For-Sale Mild ASAH1 88 37 C[C@@H](CC(=O)O)NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147343005 BD For-Sale Anodyne FFAR1 0 41 C[C@@H](CC(=O)O)NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147343005 BD For-Sale Anodyne GPR88 0 52 CC[C@H](NC(=O)c1cc2ccc(F)cc2s1)C(=O)O ZINC000147343012 CF On-Demand Anodyne PIN1 51 52 COc1ccc(Br)cc1CNC1(C(=O)O)CCC1 ZINC000147343044 DF On-Demand Anodyne QRFPR 42 35 CC[C@@H](CNS(=O)(=O)C[C@@H](C)c1ccccc1)CC(=O)O ZINC000147343046 DE For-Sale Anodyne GRIA4 22 43 COc1cc2c(cc1OC)CCN(C[C@@H](O)COc1cccc3[nH]ccc13)CC2 ZINC000147343057 GG On-Demand Anodyne ADRB2 19 53 COc1cc2c(cc1OC)CCN(C[C@@H](O)COc1cccc3[nH]ccc13)CC2 ZINC000147343057 GG On-Demand Anodyne ADRB1 23 52 COc1cc2c(cc1OC)CCN(C[C@@H](O)COc1cccc3[nH]ccc13)CC2 ZINC000147343057 GG On-Demand Anodyne HTR1A 26 65 COc1cc2c(cc1OC)CCN(C[C@@H](O)COc1cccc3[nH]ccc13)CC2 ZINC000147343057 GG On-Demand Anodyne SLC6A4 25 53 COc1cc2c(cc1OC)CCN(C[C@@H](O)COc1cccc3[nH]ccc13)CC2 ZINC000147343057 GG On-Demand Anodyne ADRB3 16 53 COc1cc2c(cc1OC)CCN(C[C@@H](O)COc1cccc3[nH]ccc13)CC2 ZINC000147343057 GG On-Demand Anodyne ACOX1 29 43 COc1cc2c(cc1OC)CCN(C[C@@H](O)COc1cccc3[nH]ccc13)CC2 ZINC000147343057 GG On-Demand Anodyne ABCB1B 46 32 COc1cc2c(cc1OC)CCN(C[C@@H](O)COc1cccc3[nH]ccc13)CC2 ZINC000147343057 GG On-Demand Anodyne ABCB1 93 40 CC[C@@H](NC(=O)C[C@@H]1CNc2ccccc21)C(=O)O ZINC000147343067 CD On-Demand Anodyne ACE2 57 33 CC(C)CCCCNCc1ccncn1 ZINC000147343091 BE For-Sale Anodyne FDFT1 0 41 CSc1nn(-c2ccccc2)c2cc(N3CCN(C(=O)[C@@H]4CCCNC4)CC3)ccc12 ZINC000147343107 IG Annotated Anodyne KHK 0 82 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(S(N)(=O)=O)cc2)C1 ZINC000147343137 GB On-Demand Anodyne CA1 17 42 C[N+](C)(C)CCCCCCCCCCC(=O)O ZINC000147343163 BG For-Sale Anodyne FABP3 36 43 C[N+](C)(C)CCCCCCCCCCC(=O)O ZINC000147343163 BG For-Sale Anodyne FABP5 18 54 C[N+](C)(C)CCCCCCCCCCC(=O)O ZINC000147343163 BG For-Sale Anodyne BBOX1 72 48 CCCCCCCCNC(=O)c1cc(Br)cnc1NC ZINC000147343186 EH For-Sale Mild LPAR2 50 35 CCCCCCCCNC(=O)c1cc(Br)cnc1NC ZINC000147343186 EH For-Sale Mild S1PR2 58 35 CCCCCCCCNC(=O)c1cc(Br)cnc1NC ZINC000147343186 EH For-Sale Mild MERTK 17 40 CCCCCCCCNC(=O)c1cc(Br)cnc1NC ZINC000147343186 EH For-Sale Mild ASAH1 75 35 CN(C)C(=O)c1ccc(Oc2ccccc2)c(N)c1 ZINC000147343214 CF For-Sale Anodyne SRD5A2 0 41 CN(C)C(=O)c1ccc(Oc2ccccc2)c(N)c1 ZINC000147343214 CF For-Sale Anodyne TSPO 50 33 CN(C)C(=O)c1ccc(Oc2ccccc2)c(N)c1 ZINC000147343214 CF For-Sale Anodyne TRY1_BOVIN 22 43 CN(C)C(=O)c1ccc(Oc2ccccc2)c(N)c1 ZINC000147343214 CF For-Sale Anodyne MT-ND1 18 44 C[C@H](CC(=O)O)NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147343227 BD For-Sale Anodyne FFAR1 0 41 C[C@H](CC(=O)O)NC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147343227 BD For-Sale Anodyne GPR88 0 52 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343250 FG On-Demand Anodyne DRD4 44 34 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343250 FG On-Demand Anodyne CTSL 18 40 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343250 FG On-Demand Anodyne CTSV 17 41 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343250 FG On-Demand Anodyne MDM2 41 31 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343250 FG On-Demand Anodyne KCNK3 48 38 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343250 FG On-Demand Anodyne KCNK9 44 46 CC[C@H](CNS(=O)(=O)C[C@H](C)c1ccccc1)CC(=O)O ZINC000147343254 DE For-Sale Anodyne GRIA4 22 43 CN(Cc1cscn1)C(=O)NC1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147343256 GH On-Demand Anodyne DRD4 31 45 CN(Cc1cscn1)C(=O)NC1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147343256 GH On-Demand Anodyne SIGMAR1 25 49 CN(Cc1cscn1)C(=O)NC1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147343256 GH On-Demand Anodyne SSTR5 48 38 CN(Cc1cscn1)C(=O)NC1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147343256 GH On-Demand Anodyne CCR1 19 43 CN(Cc1cscn1)C(=O)NC1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147343256 GH On-Demand Anodyne CXCR3 30 41 CN(Cc1cscn1)C(=O)NC1CCN(Cc2ccc(Cl)cc2)CC1 ZINC000147343256 GH On-Demand Anodyne MCHR1 48 50 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCc2cccc(-c3cncnc3)c2)cc(N2CCCC2=O)c1 ZINC000147343272 KI Annotated Anodyne CTSD 58 67 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCc2cccc(-c3cncnc3)c2)cc(N2CCCC2=O)c1 ZINC000147343272 KI Annotated Anodyne BACE2 71 64 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCc2cccc(-c3cncnc3)c2)cc(N2CCCC2=O)c1 ZINC000147343272 KI Annotated Anodyne BACE1 96 80 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCc2cccc(-c3cncnc3)c2)cc(N2CCCC2=O)c1 ZINC000147343272 KI Annotated Anodyne PLM1_PLAFA 57 41 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCc2cccc(-c3cncnc3)c2)cc(N2CCCC2=O)c1 ZINC000147343272 KI Annotated Anodyne PLM2_PLAFA 36 45 CSc1nn(-c2ccccc2)c2cc(N3CCN(C(=O)[C@H]4CCCNC4)CC3)ccc12 ZINC000147343293 IG Annotated Anodyne KHK 0 82 CC[C@H](NC(=O)C[C@H]1CNc2ccccc21)C(=O)O ZINC000147343301 CD On-Demand Anodyne ACE2 57 33 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)N2CCOCC2)CC1 ZINC000147343319 GA On-Demand Anodyne P2RY12 55 37 CCNc1cccc(NCc2ccncc2)n1 ZINC000147343335 BF For-Sale Anodyne GPR39 0 45 C[C@H]1NC(=S)N(c2ccc(OCc3ccccc3F)cc2)C1=O ZINC000147343342 EG On-Demand Anodyne GYS1 48 33 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc(S(N)(=O)=O)cc2)C1 ZINC000147343352 GB On-Demand Anodyne CA1 17 42 CCCCCCCCNC(=O)c1cc(Br)cnc1N ZINC000147343390 EH For-Sale Mild ASAH1 81 36 CC[C@@H](C)[C@H](N)C(=O)NN1CCCCC1 ZINC000147343422 BC For-Sale Anodyne TPP2 41 44 C[C@@H](CC(=O)O)NC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147343442 BD For-Sale Anodyne FFAR1 0 41 C[C@@H](CC(=O)O)NC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147343442 BD For-Sale Anodyne GPR88 0 52 Cc1cccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343476 FG On-Demand Anodyne DRD4 44 34 Cc1cccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343476 FG On-Demand Anodyne CTSL 18 40 Cc1cccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343476 FG On-Demand Anodyne CTSV 17 41 Cc1cccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343476 FG On-Demand Anodyne MDM2 41 31 Cc1cccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343476 FG On-Demand Anodyne KCNK3 48 38 Cc1cccc(C(=O)NCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147343476 FG On-Demand Anodyne KCNK9 44 46 CC[C@@H](CNS(=O)(=O)C[C@H](C)c1ccccc1)CC(=O)O ZINC000147343483 DE For-Sale Anodyne GRIA4 22 43 CCc1nc(CN(C)C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cs1 ZINC000147343492 HI On-Demand Anodyne DRD4 29 45 CCc1nc(CN(C)C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cs1 ZINC000147343492 HI On-Demand Anodyne SIGMAR1 23 47 CCc1nc(CN(C)C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cs1 ZINC000147343492 HI On-Demand Anodyne SSTR5 56 36 CCc1nc(CN(C)C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cs1 ZINC000147343492 HI On-Demand Anodyne CCR1 17 43 CCc1nc(CN(C)C(=O)NC2CCN(Cc3ccc(Cl)cc3)CC2)cs1 ZINC000147343492 HI On-Demand Anodyne MCHR1 45 44 CSc1nn(-c2ccccc2)c2cc(N3CCN(Cc4ccncc4)CC3)ccc12 ZINC000147343504 HI Annotated Anodyne HTR1A 17 44 CSc1nn(-c2ccccc2)c2cc(N3CCN(Cc4ccncc4)CC3)ccc12 ZINC000147343504 HI Annotated Anodyne DRD1 22 43 CSc1nn(-c2ccccc2)c2cc(N3CCN(Cc4ccncc4)CC3)ccc12 ZINC000147343504 HI Annotated Anodyne DRD4 42 40 CSc1nn(-c2ccccc2)c2cc(N3CCN(Cc4ccncc4)CC3)ccc12 ZINC000147343504 HI Annotated Anodyne KHK 0 65 C[C@H]1CN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2F)C[C@@H](C)O1 ZINC000147343510 GE On-Demand Anodyne NPY2R 58 35 C[C@H]1CN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2F)C[C@@H](C)O1 ZINC000147343510 GE On-Demand Anodyne ENV 42 34 CC[C@@H](NC(=O)C[C@H]1CNc2ccccc21)C(=O)O ZINC000147343516 CD On-Demand Anodyne ACE2 57 33 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)c(OC)c1 ZINC000147343517 FG For-Sale Reactive OXTR 30 46 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)c(OC)c1 ZINC000147343517 FG For-Sale Reactive GRM3 16 48 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)c(OC)c1 ZINC000147343517 FG For-Sale Reactive RORC 43 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)N2CCOCC2)CC1 ZINC000147343528 GA On-Demand Anodyne P2RY12 55 37 CCCCNC(=O)C1CCN(C(=O)c2ccccc2NS(C)(=O)=O)CC1 ZINC000147343531 GD On-Demand Anodyne EPHX2 21 43 CCCCNC(=O)C1CCN(C(=O)c2ccccc2NS(C)(=O)=O)CC1 ZINC000147343531 GD On-Demand Anodyne CCR8 67 35 CCCCCCCCNC(=O)c1cnc(C)cc1NC ZINC000147343595 CH For-Sale Mild MERTK 20 41 CCCCCCCCNC(=O)c1cnc(C)cc1NC ZINC000147343595 CH For-Sale Mild ASAH1 77 33 CC[C@@H]1c2ccsc2CCN1C(=O)c1ccc(-c2nnc(-c3ccc(C)cc3)o2)cc1 ZINC000147343609 IK Annotated Anodyne TRPM8 16 43 CC[C@H](C)[C@H](N)C(=O)NN1CCCCC1 ZINC000147343649 BC For-Sale Anodyne TPP2 41 44 C[C@H](CC(=O)O)NC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147343654 BD For-Sale Anodyne FFAR1 0 41 C[C@H](CC(=O)O)NC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147343654 BD For-Sale Anodyne GPR88 0 52 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147343668 FG On-Demand Anodyne DRD4 44 34 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147343668 FG On-Demand Anodyne CTSL 18 40 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147343668 FG On-Demand Anodyne CTSV 17 41 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147343668 FG On-Demand Anodyne MDM2 41 31 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147343668 FG On-Demand Anodyne KCNK3 48 38 Cc1cccc(C(=O)NCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147343668 FG On-Demand Anodyne KCNK9 44 46 COC(=O)CN(Cc1ccccc1)C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147343691 HD On-Demand Bother COLA 42 34 COC(=O)CN(Cc1ccccc1)C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147343691 HD On-Demand Bother MMP2 22 41 COC(=O)CN(Cc1ccccc1)C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147343691 HD On-Demand Bother MMP8 40 41 COC(=O)CN(Cc1ccccc1)C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147343691 HD On-Demand Bother MMP9 25 41 COC(=O)CN(Cc1ccccc1)C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147343691 HD On-Demand Bother MMP1 36 41 COC(=O)CN(Cc1ccccc1)C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147343691 HD On-Demand Bother LIMK2 45 41 CSc1nn(-c2ccccc2)c2cc(N3CC[C@H](N4CCNCC4)C3)ccc12 ZINC000147343701 GG Annotated Anodyne KHK 0 77 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)c(OC)c1 ZINC000147343732 FG For-Sale Reactive OXTR 22 46 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)c(OC)c1 ZINC000147343732 FG For-Sale Reactive GRM3 16 48 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)c(OC)c1 ZINC000147343732 FG For-Sale Reactive RORC 43 40 O=C(O)c1cc(Cl)cc(NC(=O)N2CCC(O)CC2)c1 ZINC000147343762 CE On-Demand Anodyne CACNA1H 42 37 O=C(O)c1cc(Cl)cc(NC(=O)N2CCC(O)CC2)c1 ZINC000147343762 CE On-Demand Anodyne EPHX2 18 42 O=C(O)c1cc(Cl)cc(NC(=O)N2CCC(O)CC2)c1 ZINC000147343762 CE On-Demand Anodyne CACNA1I 49 36 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(C(N)=O)cc2)C1 ZINC000147343768 FB On-Demand Anodyne HRH2 15 41 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(C(N)=O)cc2)C1 ZINC000147343768 FB On-Demand Anodyne SFRP1 76 33 CS(=O)(=O)N1CCC[C@H](NS(=O)(=O)c2ccc(C(N)=O)cc2)C1 ZINC000147343768 FB On-Demand Anodyne WNT3 47 31 COc1cccc(C(=O)Nc2cc(Cl)ccc2Br)c1O ZINC000147343776 FI For-Sale Anodyne CPT1A 43 30 COc1cccc(C(=O)Nc2cc(Cl)ccc2Br)c1O ZINC000147343776 FI For-Sale Anodyne PYGL 15 40 COc1cccc(C(=O)Nc2cc(Cl)ccc2Br)c1O ZINC000147343776 FI For-Sale Anodyne GRM4 23 42 COc1cccc(C(=O)Nc2cc(Cl)ccc2Br)c1O ZINC000147343776 FI For-Sale Anodyne KCNMA1 45 49 COc1cccc(C(=O)Nc2cc(Cl)ccc2Br)c1O ZINC000147343776 FI For-Sale Anodyne ACPS 0 40 COc1cccc(C(=O)Nc2cc(Cl)ccc2Br)c1O ZINC000147343776 FI For-Sale Anodyne GPR35 46 33 COc1cccc(C(=O)Nc2cc(Cl)ccc2Br)c1O ZINC000147343776 FI For-Sale Anodyne KCNK3 61 45 COc1cccc(C(=O)Nc2cc(Cl)ccc2Br)c1O ZINC000147343776 FI For-Sale Anodyne KCNK9 55 45 COc1cccc(C(=O)Nc2cc(Cl)ccc2Br)c1O ZINC000147343776 FI For-Sale Anodyne BRPF1 0 41 CC[C@H]1c2ccsc2CCN1C(=O)c1ccc(-c2nnc(-c3ccc(C)cc3)o2)cc1 ZINC000147343799 IK Annotated Anodyne TRPM8 16 43 O=c1oc2cc(I)ccc2n1Cc1cccc(F)c1 ZINC000147343817 FG For-Sale Anodyne MIF 22 55 CCCNc1nc(Oc2cccnc2)c2ccccc2n1 ZINC000147343825 CH For-Sale Anodyne SLC2A1 0 41 CCCNc1nc(Oc2cccnc2)c2ccccc2n1 ZINC000147343825 CH For-Sale Anodyne HT1 0 41 CCCNc1nc(Oc2cccnc2)c2ccccc2n1 ZINC000147343825 CH For-Sale Anodyne LMGT2 0 41 Cc1ccc(CNC(=O)[C@H](C)Cc2cccc(F)c2)cc1F ZINC000147343839 DH On-Demand Anodyne ANPEP 28 52 Cc1ccc(CNC(=O)[C@H](C)Cc2cccc(F)c2)cc1F ZINC000147343839 DH On-Demand Anodyne TRPV1 43 41 Cc1ccc(CNC(=O)[C@H](C)Cc2cccc(F)c2)cc1F ZINC000147343839 DH On-Demand Anodyne PAPA1_CARPA 15 41 Cc1ccc(CNC(=O)[C@H](C)Cc2cccc(F)c2)cc1F ZINC000147343839 DH On-Demand Anodyne CTSL 19 41 Cc1ccc(CNC(=O)[C@H](C)Cc2cccc(F)c2)cc1F ZINC000147343839 DH On-Demand Anodyne CPA1 15 40 Cc1ccc(CNC(=O)[C@H](C)Cc2cccc(F)c2)cc1F ZINC000147343839 DH On-Demand Anodyne CTSS 15 41 Cc1ccc(CNC(=O)[C@H](C)Cc2cccc(F)c2)cc1F ZINC000147343839 DH On-Demand Anodyne ACE2 44 33 Cc1ccc(CNC(=O)[C@H](C)Cc2cccc(F)c2)cc1F ZINC000147343839 DH On-Demand Anodyne AMP1_PLAFQ 47 36 Cc1ccc(CNC(=O)[C@H](C)Cc2cccc(F)c2)cc1F ZINC000147343839 DH On-Demand Anodyne LEF 111 46 Cc1ccc(CNC(=O)[C@H](C)Cc2cccc(F)c2)cc1F ZINC000147343839 DH On-Demand Anodyne CARM1 55 35 CCCCCCCCNC(=O)c1nnc(NCC)s1 ZINC000147343854 CG For-Sale Mild ASAH1 72 33 CSc1nn(-c2ccccc2)c2cc(N3CC[C@@H](N4CCNCC4)C3)ccc12 ZINC000147343907 GG Annotated Anodyne KHK 0 77 O=C(Nc1ccc(-c2csnn2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147343920 GI On-Demand Anodyne PRNP 54 33 O=C(Nc1ccc(-c2csnn2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147343920 GI On-Demand Anodyne GRM4 48 35 O=C(Nc1ccc(-c2csnn2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147343920 GI On-Demand Anodyne NR2E3 44 34 O=C(Nc1ccc(-c2csnn2)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147343920 GI On-Demand Anodyne SMO 19 41 C[C@@H]1CN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2F)C[C@@H](C)O1 ZINC000147343980 GE On-Demand Anodyne NPY2R 58 35 C[C@@H]1CN(c2ccc(NC(=O)C(=O)NC[C@@H]3CCCCO3)cc2F)C[C@@H](C)O1 ZINC000147343980 GE On-Demand Anodyne ENV 42 34 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc(C(N)=O)cc2)C1 ZINC000147344004 FB On-Demand Anodyne HRH2 15 41 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc(C(N)=O)cc2)C1 ZINC000147344004 FB On-Demand Anodyne SFRP1 76 33 CS(=O)(=O)N1CCC[C@@H](NS(=O)(=O)c2ccc(C(N)=O)cc2)C1 ZINC000147344004 FB On-Demand Anodyne WNT3 47 31 CCCCCCCCNC(=O)c1ccc(NCC)cc1 ZINC000147344032 CI For-Sale Mild FOLH1 30 50 CCCCCCCCNC(=O)c1ccc(NCC)cc1 ZINC000147344032 CI For-Sale Mild KCNQ1 0 56 CCCCCCCCNC(=O)c1ccc(NCC)cc1 ZINC000147344032 CI For-Sale Mild HDAC6 17 46 CCCCCCCCNC(=O)c1ccc(NCC)cc1 ZINC000147344032 CI For-Sale Mild S1PR2 45 36 CCCCCCCCNC(=O)c1ccc(NCC)cc1 ZINC000147344032 CI For-Sale Mild EPHX2 19 40 CCCCCCCCNC(=O)c1ccc(NCC)cc1 ZINC000147344032 CI For-Sale Mild HDA106 0 45 CCCCCCCCNC(=O)c1ccc(NCC)cc1 ZINC000147344032 CI For-Sale Mild CNGA1 0 42 CCCCCCCCNC(=O)c1ccc(NCC)cc1 ZINC000147344032 CI For-Sale Mild ENPP2 27 40 CCCCCCCCNC(=O)c1ccc(NCC)cc1 ZINC000147344032 CI For-Sale Mild ASAH1 100 40 CCCCCCCCNC(=O)c1ccc(NCC)cc1 ZINC000147344032 CI For-Sale Mild ACAT 0 45 CCCCCCCCNC(=O)c1ccc(NCC)cc1 ZINC000147344032 CI For-Sale Mild PSBA 0 40 CC[C@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147344068 DE On-Demand Anodyne TBXA2R 52 41 CC[C@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147344068 DE On-Demand Anodyne TBXAS1 34 47 O=C(Nc1cc(Cl)ccc1Br)c1ccccc1O ZINC000147344097 EI For-Sale Anodyne F10 27 41 O=C(Nc1cc(Cl)ccc1Br)c1ccccc1O ZINC000147344097 EI For-Sale Anodyne GRM4 24 40 O=C(Nc1cc(Cl)ccc1Br)c1ccccc1O ZINC000147344097 EI For-Sale Anodyne KCNMA1 61 75 O=C(Nc1cc(Cl)ccc1Br)c1ccccc1O ZINC000147344097 EI For-Sale Anodyne ACPS 0 43 O=C(Nc1cc(Cl)ccc1Br)c1ccccc1O ZINC000147344097 EI For-Sale Anodyne Q25615_ONCVO 55 35 O=C(Nc1cc(Cl)ccc1Br)c1ccccc1O ZINC000147344097 EI For-Sale Anodyne TMPRSS4 0 45 CN(CC(=O)O)S(=O)(=O)Cc1ccccc1C(F)(F)F ZINC000147344129 DD On-Demand Anodyne RORC 17 40 COc1cc(C(=O)CCC2CCCCC2)c(OC)cc1Cl ZINC000147344146 DJ For-Sale Anodyne HTR4 90 69 CCc1nc(CN(C)C(=O)N[C@@H](CN2CCOCC2)c2ccccc2)cs1 ZINC000147344156 GF On-Demand Anodyne CASR 55 42 CCc1nc(CN(C)C(=O)N[C@@H](CN2CCOCC2)c2ccccc2)cs1 ZINC000147344156 GF On-Demand Anodyne CYP3A4 21 42 CCCCCCCCNC(=O)c1cc(Cl)ccc1NCC ZINC000147344245 DJ For-Sale Mild CNR1 19 46 CCCCCCCCNC(=O)c1cc(Cl)ccc1NCC ZINC000147344245 DJ For-Sale Mild CNR2 16 46 CCCCCCCCNC(=O)c1cc(Cl)ccc1NCC ZINC000147344245 DJ For-Sale Mild ALPL 42 39 CCCCCCCCNC(=O)c1cc(Cl)ccc1NCC ZINC000147344245 DJ For-Sale Mild ASAH1 91 38 CCCCCCCCNC(=O)c1cc(Cl)ccc1NCC ZINC000147344245 DJ For-Sale Mild ACAT 0 45 CCCCCCCCNC(=O)c1cc(Cl)ccc1NCC ZINC000147344245 DJ For-Sale Mild PSBA 0 51 CC[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147344284 DE On-Demand Anodyne TBXA2R 52 41 CC[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1)CC(=O)O ZINC000147344284 DE On-Demand Anodyne TBXAS1 34 47 CCc1nc(CN(C)C(=O)N[C@H](CN2CCOCC2)c2ccccc2)cs1 ZINC000147344319 GF On-Demand Anodyne CASR 55 42 CCc1nc(CN(C)C(=O)N[C@H](CN2CCOCC2)c2ccccc2)cs1 ZINC000147344319 GF On-Demand Anodyne CYP3A4 21 42 CSc1nn(-c2ccccc2)c2cc(N3CCN(C4CNC4)CC3)ccc12 ZINC000147344336 GF Annotated Anodyne KHK 0 81 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(CCN3CCOCC3)cc1)C2 ZINC000147344377 GF On-Demand Anodyne ROCK2 34 49 O=C(Nc1ncccc1Br)c1cccc2c1OCCN2 ZINC000147344398 EF For-Sale Anodyne G2YM83_BOTF4 59 33 CCCCCCCCNC(=O)c1cnccc1NCC ZINC000147344405 CH For-Sale Mild ASAH1 82 35 O=C(Nc1cc(Br)cc(C(=O)O)c1)Nc1ccccc1Br ZINC000147344443 HJ For-Sale Anodyne PPIA 22 41 O=C(Nc1cc(Br)cc(C(=O)O)c1)Nc1ccccc1Br ZINC000147344443 HJ For-Sale Anodyne LPL 43 33 O=C(Nc1cc(Br)cc(C(=O)O)c1)Nc1ccccc1Br ZINC000147344443 HJ For-Sale Anodyne P95276_MYCTO 0 41 N[C@H](CCC(=O)O)C(=O)NN1CCCCC1 ZINC000147344472 BB For-Sale Anodyne GRM8 25 45 N[C@H](CCC(=O)O)C(=O)NN1CCCCC1 ZINC000147344472 BB For-Sale Anodyne GRIK3 15 45 N[C@H](CCC(=O)O)C(=O)NN1CCCCC1 ZINC000147344472 BB For-Sale Anodyne DPP7 40 36 Cc1cc(C)c(OCCCN2CCCC2)c(S(N)(=O)=O)c1 ZINC000147344475 DD For-Sale Anodyne HRH3 59 40 Cc1cc(C)c(OCCCN2CCCC2)c(S(N)(=O)=O)c1 ZINC000147344475 DD For-Sale Anodyne HNMT 44 36 CC[C@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147344501 CD On-Demand Anodyne CAPN1 21 42 COCc1nc(C(=O)N2CCN(CC(=O)Nc3cccc(C)c3C)CC2)cs1 ZINC000147344532 HE On-Demand Anodyne TRPC6 46 34 CCN(CC)Cc1ccccc1CNC(=O)N(C)Cc1cscn1 ZINC000147344554 EG On-Demand Anodyne BMP1 50 34 CSc1nn(-c2ccccc2)c2cc(N3CCN([C@@H]4CCNC4)CC3)ccc12 ZINC000147344555 GG Annotated Anodyne KHK 0 89 CCCCCCCCNC(=O)c1cnccc1NC ZINC000147344608 CG For-Sale Mild FAAH 16 42 CCCCCCCCNC(=O)c1cnccc1NC ZINC000147344608 CG For-Sale Mild ASAH1 88 37 CCCNc1cccc(NCc2ccncc2)n1 ZINC000147344642 BF For-Sale Anodyne GPR39 0 46 N[C@@H](CCC(=O)O)C(=O)NN1CCCCC1 ZINC000147344654 BB For-Sale Anodyne GRM8 25 45 N[C@@H](CCC(=O)O)C(=O)NN1CCCCC1 ZINC000147344654 BB For-Sale Anodyne GRIK3 15 45 N[C@@H](CCC(=O)O)C(=O)NN1CCCCC1 ZINC000147344654 BB For-Sale Anodyne DPP7 40 36 CNC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147344663 GB On-Demand Anodyne HRH2 15 41 CNC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147344663 GB On-Demand Anodyne SFRP1 64 33 CNC(=O)c1ccc(S(=O)(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147344663 GB On-Demand Anodyne WNT3 41 32 CC[C@@H](CNS(=O)(=O)c1ccc(F)cc1)CC(=O)O ZINC000147344671 CD On-Demand Anodyne CAPN1 21 42 O=C(Nc1cc(Cl)cc(C(=O)O)c1)Nc1ccccc1Br ZINC000147344683 FI For-Sale Anodyne PPIA 33 50 O=C(Nc1cc(Cl)cc(C(=O)O)c1)Nc1ccccc1Br ZINC000147344683 FI For-Sale Anodyne LPL 43 33 O=C(Nc1cc(Cl)cc(C(=O)O)c1)Nc1ccccc1Br ZINC000147344683 FI For-Sale Anodyne P2RY1 21 41 O=C(Nc1cc(Cl)cc(C(=O)O)c1)Nc1ccccc1Br ZINC000147344683 FI For-Sale Anodyne ITGA4 46 41 O=C(Nc1cc(Cl)cc(C(=O)O)c1)Nc1ccccc1Br ZINC000147344683 FI For-Sale Anodyne AKR1C3 29 41 CSc1nn(-c2ccccc2)c2cc(N3CCN([C@H]4CCNC4)CC3)ccc12 ZINC000147344741 GG Annotated Anodyne KHK 0 89 COc1ccc([N+](=O)[O-])c(C(=O)Nc2nc(C)c(Cc3ccccc3Cl)s2)c1 ZINC000147344796 HJ On-Demand Bother TAAR1 22 40 CCCCCCCCNC(=O)c1ccc(NC)nn1 ZINC000147344813 CF For-Sale Mild S1PR2 41 36 CCCCCCCCNC(=O)c1ccc(NC)nn1 ZINC000147344813 CF For-Sale Mild SCD1 18 47 CCCCCCCCNC(=O)c1ccc(NC)nn1 ZINC000147344813 CF For-Sale Mild ASAH1 92 37 Oc1ccc(CNCC(F)F)cc1 ZINC000147344824 AD On-Demand Anodyne H9TVJ1_CHISP 44 35 c1cc(OCC2CC2)c2cc[nH]c2c1 ZINC000147344849 AF For-Sale Anodyne HTR1A 24 52 c1cc(OCC2CC2)c2cc[nH]c2c1 ZINC000147344849 AF For-Sale Anodyne IL5 54 35 CNC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147344863 GB On-Demand Anodyne HRH2 15 41 CNC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147344863 GB On-Demand Anodyne SFRP1 64 33 CNC(=O)c1ccc(S(=O)(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cc1 ZINC000147344863 GB On-Demand Anodyne WNT3 41 32 O=C(Nc1ccc(Br)cc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147344925 HJ For-Sale Anodyne EPHX2 20 43 O=C(Nc1ccc(Br)cc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147344925 HJ For-Sale Anodyne CA12 19 49 O=C(Nc1ccc(Br)cc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147344925 HJ For-Sale Anodyne CA9 19 45 O=C(Nc1ccc(Br)cc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147344925 HJ For-Sale Anodyne AKR1C3 26 51 O=C(Nc1ccc(Br)cc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147344925 HJ For-Sale Anodyne IDO1 18 44 O=C(Nc1ccc(Br)cc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147344925 HJ For-Sale Anodyne MTCA1 37 49 O=C(Nc1ccc(Br)cc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147344925 HJ For-Sale Anodyne P96878_MYCTU 42 49 O=C(Nc1ccc(Br)cc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147344925 HJ For-Sale Anodyne P95276_MYCTO 0 42 CSc1nn(-c2ccccc2)c2cc(N3CCN([C@@H]4CCNC4)C3=O)ccc12 ZINC000147344952 GG Annotated Anodyne KHK 0 63 O=C1CCC[C@H](C(=O)OCc2ccccc2)N1 ZINC000147344979 BD On-Demand Anodyne FKBP1A 34 43 O=C1CCC[C@H](C(=O)OCc2ccccc2)N1 ZINC000147344979 BD On-Demand Anodyne HDAC3 15 41 O=C1CCC[C@H](C(=O)OCc2ccccc2)N1 ZINC000147344979 BD On-Demand Anodyne SLC12A5 64 44 O=c1oc2cc(I)ccc2n1Cc1cc(F)ccc1F ZINC000147344984 GH For-Sale Anodyne MIF 16 46 COc1cc(C(=O)Cl)c(Cl)cc1Cl ZINC000147345007 BG For-Sale Reactive HTR4 51 39 CCN(CC)c1ccc(CNCCCCC(C)C)cc1 ZINC000147345034 CI For-Sale Clean S1PR2 30 40 CCN(CC)c1ccc(CNCCCCC(C)C)cc1 ZINC000147345034 CI For-Sale Clean LEF 67 34 CC(C)(C)c1ccc(CNCC(F)F)cc1 ZINC000147345077 BG On-Demand Anodyne PETD 0 40 CCCCCCCCNC(=O)c1ccc(C)cc1NCC ZINC000147345080 CJ For-Sale Mild PA2A1_NAJMO 0 42 CCCCCCCCNC(=O)c1ccc(C)cc1NCC ZINC000147345080 CJ For-Sale Mild ASAH1 75 36 OC[C@@H]1C[C@@H]1c1ccc(I)cc1 ZINC000147345084 CE For-Sale Anodyne SLC6A1 19 41 O=[N+]([O-])c1cccc(CCl)c1O ZINC000147345091 AE For-Sale Reactive COLA 89 33 O=[N+]([O-])c1cccc(CCl)c1O ZINC000147345091 AE For-Sale Reactive PQSD 0 52 Nc1nc(F)nc2ccccc12 ZINC000147345104 AD For-Sale Anodyne DHFR 15 46 Nc1nc(F)nc2ccccc12 ZINC000147345104 AD For-Sale Anodyne FOLA 16 46 Nc1nc(F)nc2ccccc12 ZINC000147345104 AD For-Sale Anodyne HTR3A 15 46 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne TYMS 17 40 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne F9 21 45 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne TACR1 19 41 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne CMA1 64 35 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne CTRA_BOVIN 52 44 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne FCER2 60 32 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne PAPA1_CARPA 63 40 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne CTSL 38 40 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne CACNA1B 28 41 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne CTRB1 42 36 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne CAPNS1 41 31 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne REN 40 38 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne CTSS 25 40 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne CAPN1 44 37 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne PIN1 48 35 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne FPR1 55 41 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne CTRB_BOVIN 67 39 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne CYP3A4 36 45 CC(C)(C)OC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345124 GH On-Demand Anodyne BLA1_STEMA 47 36 CCNC(=O)n1ccc(O)cc1=O ZINC000147345146 AC For-Sale Anodyne ASAH1 77 43 O=C(Nc1ccc(Br)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345150 FI For-Sale Anodyne PPIA 23 49 O=C(Nc1ccc(Br)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345150 FI For-Sale Anodyne EPHX2 18 44 O=C(Nc1ccc(Br)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345150 FI For-Sale Anodyne AKR1C3 25 48 O=C(Nc1ccc(Br)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345150 FI For-Sale Anodyne IDO1 20 41 O=C(Nc1ccc(Br)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345150 FI For-Sale Anodyne MTCA1 25 45 O=C(Nc1ccc(Br)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345150 FI For-Sale Anodyne P96878_MYCTU 25 45 O=C(Nc1ccc(Br)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345150 FI For-Sale Anodyne HCAR1 0 42 O=C(Nc1ccc(Br)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345150 FI For-Sale Anodyne P95276_MYCTO 0 44 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne HRH2 29 41 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne LTA4H 47 50 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne RARB 15 45 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne HRH3 77 47 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne MMP13 29 40 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne PLA2G4A 22 43 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne PLA2G4B 100 43 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne LIPE 23 47 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne FAAH 32 45 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne LIPA 48 35 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne MMP1 15 43 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne PSMB2 54 42 CCCCOc1ccc(OC(=O)N2CCCCC2)cc1 ZINC000147345161 CH For-Sale Anodyne PSMB1 46 42 CSc1nn(-c2ccccc2)c2cc(N3CCN([C@H]4CCNC4)C3=O)ccc12 ZINC000147345175 GG Annotated Anodyne KHK 0 63 O=C(O)/C=C/c1ccc(NC(=O)C2[C@H]3CCCC[C@H]23)cc1 ZINC000147345188 CG On-Demand Anodyne MMP1 0 45 O=C(c1ccc2c(c1)CCO2)N1CCC[C@H](CCBr)C1 ZINC000147345196 EG For-Sale Reactive GPR183 0 47 OC[C@H]1C[C@@H]1c1ccc(I)cc1 ZINC000147345240 CE For-Sale Anodyne SLC6A1 19 41 CCCCCCCCNC(=O)c1cnc(C)cc1N ZINC000147345272 CG For-Sale Mild MERTK 21 41 CCCCCCCCNC(=O)c1cnc(C)cc1N ZINC000147345272 CG For-Sale Mild ASAH1 81 34 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne ALOX5 26 53 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne MAOB 40 42 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne PPARG 28 44 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne PTGER2 34 40 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne ADRB3 20 42 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne LTA4H 15 44 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne EDNRA 21 50 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne PTGER4 31 40 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne PTGER3 41 35 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne CTSB 22 41 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne CAPN1 24 41 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne CAPN2 49 41 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne ACE2 24 43 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne ACR 27 40 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne FFAR1 64 46 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne PTGES 15 45 CCOC(=O)C[C@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345328 DG For-Sale Anodyne PDS 73 37 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne TYMS 17 40 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne F9 21 45 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne TACR1 19 41 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne CMA1 64 35 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne CTRA_BOVIN 52 44 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne FCER2 60 32 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne PAPA1_CARPA 63 40 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne CTSL 38 40 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne CACNA1B 28 41 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne CTRB1 42 36 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne CAPNS1 41 31 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne REN 40 38 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne CTSS 25 40 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne CAPN1 44 37 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne PIN1 48 35 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne FPR1 55 41 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne CTRB_BOVIN 67 39 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne CYP3A4 36 45 CC(C)(C)OC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc2ncsc2c1 ZINC000147345330 GH On-Demand Anodyne BLA1_STEMA 47 36 O=C(Nc1cccc(Br)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147345389 HJ For-Sale Anodyne EGFR 39 42 O=C(Nc1cccc(Br)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147345389 HJ For-Sale Anodyne PPIA 38 44 O=C(Nc1cccc(Br)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147345389 HJ For-Sale Anodyne KIT 16 43 O=C(Nc1cccc(Br)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147345389 HJ For-Sale Anodyne KDR 15 43 O=C(Nc1cccc(Br)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147345389 HJ For-Sale Anodyne EPHX2 25 47 O=C(Nc1cccc(Br)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147345389 HJ For-Sale Anodyne TAAR1 19 43 O=C(Nc1cccc(Br)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147345389 HJ For-Sale Anodyne AKR1C3 39 50 O=C(Nc1cccc(Br)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147345389 HJ For-Sale Anodyne P95276_MYCTO 0 45 O=C(Nc1cccc(Br)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147345389 HJ For-Sale Anodyne KCNK3 88 37 O=C(Nc1cccc(Br)c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147345389 HJ For-Sale Anodyne KCNK9 48 36 O=C(O)/C=C/c1ccc(NC(=O)C2[C@H]3CCCC[C@@H]23)cc1 ZINC000147345392 CG For-Sale Anodyne MMP1 0 45 O=C(c1ccc2c(c1)CCO2)N1CCC[C@@H](CCBr)C1 ZINC000147345428 EG For-Sale Reactive GPR183 0 47 CCCCCCCCNC(=O)c1cc(NCCC)ccn1 ZINC000147345473 CH For-Sale Mild LPAR2 55 34 CCCCCCCCNC(=O)c1cc(NCCC)ccn1 ZINC000147345473 CH For-Sale Mild S1PR2 71 37 CCCCCCCCNC(=O)c1cc(NCCC)ccn1 ZINC000147345473 CH For-Sale Mild ASAH1 93 36 OC[C@@H]1C[C@H]1c1ccc(I)cc1 ZINC000147345475 CE For-Sale Anodyne SLC6A1 19 41 O=C(NC1CCCCC1)N1CCC1 ZINC000147345504 AD In-Stock Anodyne AMPC 16 42 CCOC(=O)C[C@@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345536 DG For-Sale Anodyne PTGER2 34 40 CCOC(=O)C[C@@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345536 DG For-Sale Anodyne EDNRA 21 50 CCOC(=O)C[C@@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345536 DG For-Sale Anodyne PTGER4 31 40 CCOC(=O)C[C@@H](O)c1cccc(OCc2ccccc2)c1 ZINC000147345536 DG For-Sale Anodyne PTGES 15 45 O=C(O)/C=C/c1ccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)cc1 ZINC000147345591 CG On-Demand Anodyne MMP1 0 45 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne PPIA 40 61 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne KIT 16 40 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne PTGER3 15 45 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne P2RY1 0 48 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne KDR 15 42 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne EPHX2 21 43 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne TAAR1 18 40 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne AKR1C3 40 50 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne NCE103 15 41 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne HCAR1 0 40 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne P95276_MYCTO 0 41 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne PSBA 0 40 O=C(Nc1cccc(Br)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147345609 FI For-Sale Anodyne KCNK3 62 44 Cc1cccc(OCCNC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147345611 DG On-Demand Bother DRD4 40 33 Cc1cccc(OCCNC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147345611 DG On-Demand Bother CACNA1D 46 36 Cc1cccc(OCCNC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147345611 DG On-Demand Bother MTNR1B 20 43 Cc1cccc(OCCNC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147345611 DG On-Demand Bother ACR 21 40 CCCc1c(-c2ccc(O)cc2)c(=O)oc2cc(O)ccc12 ZINC000147345615 CH For-Sale Anodyne ESR1 38 63 CCCc1c(-c2ccc(O)cc2)c(=O)oc2cc(O)ccc12 ZINC000147345615 CH For-Sale Anodyne ALDH2 57 36 CCCc1c(-c2ccc(O)cc2)c(=O)oc2cc(O)ccc12 ZINC000147345615 CH For-Sale Anodyne ESR2 28 63 CCCc1c(-c2ccc(O)cc2)c(=O)oc2cc(O)ccc12 ZINC000147345615 CH For-Sale Anodyne HSD17B3 51 67 CCCc1c(-c2ccc(O)cc2)c(=O)oc2cc(O)ccc12 ZINC000147345615 CH For-Sale Anodyne NQO1 70 45 C[C@H]1CC[C@@H](C)CN1C(=O)c1cccc2c1OCCN2 ZINC000147345649 CF For-Sale Anodyne HCRTR1 58 36 CC(C)(C(=O)N1CCC[C@H](CCBr)C1)c1ccccc1 ZINC000147345658 EH For-Sale Reactive CHRM2 21 40 CC(C)(C(=O)N1CCC[C@H](CCBr)C1)c1ccccc1 ZINC000147345658 EH For-Sale Reactive CHRM1 22 40 CC(C)(C(=O)N1CCC[C@H](CCBr)C1)c1ccccc1 ZINC000147345658 EH For-Sale Reactive CHRM3 37 40 CC(C)(C(=O)N1CCC[C@H](CCBr)C1)c1ccccc1 ZINC000147345658 EH For-Sale Reactive AMY2 45 32 OC[C@H]1C[C@H]1c1ccc(I)cc1 ZINC000147345683 CE For-Sale Anodyne SLC6A1 19 41 CCN(Cc1cccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)c1)C(C)=O ZINC000147345687 HH On-Demand Anodyne DRTS_PLAFK 20 44 CCN(Cc1cccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)c1)C(C)=O ZINC000147345687 HH On-Demand Anodyne PTGER3 32 46 CCN(Cc1cccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)c1)C(C)=O ZINC000147345687 HH On-Demand Anodyne KCNK3 75 37 CCN(Cc1cccc(NC(=O)c2cccn(Cc3ccccc3)c2=O)c1)C(C)=O ZINC000147345687 HH On-Demand Anodyne KCNK9 59 35 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild FDPS 37 41 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild FOLH1 30 50 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild THRB 0 58 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild KCNQ1 0 52 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild S1PR4 36 40 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild S1PR3 42 40 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild FAAH 0 42 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild S1PR2 72 40 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild S1PR1 20 40 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild EPHX2 19 43 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild S1PR5 24 40 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild HDA106 0 45 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild CNGA1 0 45 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild ENPP2 30 46 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild ASAH1 89 40 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild ACAT 0 45 CCCCCCCCNC(=O)c1ccc(NCCC)cc1 ZINC000147345709 CJ For-Sale Mild PSBA 0 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccccc2CN2CCc3ccccc32)c1 ZINC000147345733 HI On-Demand Bother AKR1C2 25 43 CCNc1cccc(NCc2cccnc2)n1 ZINC000147345764 BF For-Sale Anodyne TBXAS1 0 44 CCNc1cccc(NCc2cccnc2)n1 ZINC000147345764 BF For-Sale Anodyne LTB4R 0 40 CCNc1cccc(NCc2cccnc2)n1 ZINC000147345764 BF For-Sale Anodyne CLK4 16 44 CN(CC(=O)O)S(=O)(=O)Cc1ccccc1Cl ZINC000147345819 CD On-Demand Anodyne CXCL8 38 40 CC(=O)N1CCCc2cc(S(=O)(=O)N[C@@H]3CCCN(S(C)(=O)=O)C3)ccc21 ZINC000147345823 HC On-Demand Anodyne SFRP1 89 33 CC(=O)N1CCCc2cc(S(=O)(=O)N[C@@H]3CCCN(S(C)(=O)=O)C3)ccc21 ZINC000147345823 HC On-Demand Anodyne WNT3 56 33 C[C@H]1CC[C@H](C)N(C(=O)c2cccc3c2OCCN3)C1 ZINC000147345847 CF For-Sale Anodyne HCRTR1 58 36 CC(C)(C(=O)N1CCC[C@@H](CCBr)C1)c1ccccc1 ZINC000147345903 EH For-Sale Reactive CHRM2 21 40 CC(C)(C(=O)N1CCC[C@@H](CCBr)C1)c1ccccc1 ZINC000147345903 EH For-Sale Reactive CHRM1 22 40 CC(C)(C(=O)N1CCC[C@@H](CCBr)C1)c1ccccc1 ZINC000147345903 EH For-Sale Reactive CHRM3 37 40 CC(C)(C(=O)N1CCC[C@@H](CCBr)C1)c1ccccc1 ZINC000147345903 EH For-Sale Reactive AMY2 45 32 O=C1NC(=O)c2ccccc2/C1=C/Nc1ccccc1 ZINC000147345914 CE On-Demand Anodyne CASP8 15 45 O=C1NC(=O)c2ccccc2/C1=C/Nc1ccccc1 ZINC000147345914 CE On-Demand Anodyne CASP7 26 45 O=C1NC(=O)c2ccccc2/C1=C/Nc1ccccc1 ZINC000147345914 CE On-Demand Anodyne CDK4 51 50 Cc1nnc(CNC(=O)c2ccccc2S(=O)(=O)N2CCCCC2)o1 ZINC000147345915 FD On-Demand Anodyne LPL 47 38 Cc1nnc(CNC(=O)c2ccccc2S(=O)(=O)N2CCCCC2)o1 ZINC000147345915 FD On-Demand Anodyne EPHX2 23 41 CCCCCCCCNC(=O)c1ccc(NC)cc1 ZINC000147345936 CH For-Sale Mild FOLH1 31 51 CCCCCCCCNC(=O)c1ccc(NC)cc1 ZINC000147345936 CH For-Sale Mild THRB 0 60 CCCCCCCCNC(=O)c1ccc(NC)cc1 ZINC000147345936 CH For-Sale Mild LPAR2 44 39 CCCCCCCCNC(=O)c1ccc(NC)cc1 ZINC000147345936 CH For-Sale Mild HDAC6 16 50 CCCCCCCCNC(=O)c1ccc(NC)cc1 ZINC000147345936 CH For-Sale Mild FAAH 15 43 CCCCCCCCNC(=O)c1ccc(NC)cc1 ZINC000147345936 CH For-Sale Mild S1PR2 67 39 CCCCCCCCNC(=O)c1ccc(NC)cc1 ZINC000147345936 CH For-Sale Mild EPHX2 18 46 CCCCCCCCNC(=O)c1ccc(NC)cc1 ZINC000147345936 CH For-Sale Mild HDAC9 18 40 CCCCCCCCNC(=O)c1ccc(NC)cc1 ZINC000147345936 CH For-Sale Mild ASAH1 102 40 CCNc1nc(Cl)nc(Oc2cccnc2)n1 ZINC000147345939 CE For-Sale Anodyne Q31945_CHEAL 0 40 CCNc1nc(Cl)nc(Oc2cccnc2)n1 ZINC000147345939 CE For-Sale Anodyne PPX1 0 47 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne AVPR1A 15 44 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne CPT1A 40 39 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne PYGL 19 40 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne PRNP 16 43 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne GRM4 38 43 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne NR1H4 17 44 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne TYK2 22 41 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne CSF1R 15 40 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne ACPS 0 43 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne TAAR1 18 42 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne AKR1C3 45 42 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne NR2E3 64 42 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne AKR1C2 72 42 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne SMO 27 42 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne GALE 0 45 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne Q25615_ONCVO 59 36 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne KCNK3 102 46 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1F ZINC000147346022 DH On-Demand Anodyne KCNK9 75 38 CC(=O)N1CCCc2cc(S(=O)(=O)N[C@H]3CCCN(S(C)(=O)=O)C3)ccc21 ZINC000147346054 HC On-Demand Anodyne SFRP1 89 33 CC(=O)N1CCCc2cc(S(=O)(=O)N[C@H]3CCCN(S(C)(=O)=O)C3)ccc21 ZINC000147346054 HC On-Demand Anodyne WNT3 56 33 C[C@@H]1CC[C@@H](C)N(C(=O)c2cccc3c2OCCN3)C1 ZINC000147346058 CF For-Sale Anodyne HCRTR1 58 36 CCCCCCCCNC(=O)c1cc(N)nc(Cl)c1 ZINC000147346093 CG On-Demand Mild SCNN1A 40 43 CCCCCCCCNC(=O)c1cc(N)nc(Cl)c1 ZINC000147346093 CG On-Demand Mild ASAH1 90 38 CNc1cc(Oc2cccnc2)cc([N+](=O)[O-])c1 ZINC000147346148 BF For-Sale Bother ERO1A 0 41 CCOC(=O)NCC(=O)Nc1cccc(CN(CC)C(C)=O)c1 ZINC000147346164 DD On-Demand Anodyne NAMPT 15 40 Cc1nc(-c2cccc(NC(=O)C(=O)NCC(C)(C)N3CCC[C@H](C)C3)c2)oc1C ZINC000147346168 HH On-Demand Anodyne PDE8B 43 31 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne RARA 33 47 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne COLA 40 37 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne CPT1A 55 40 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne CPT2 45 36 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne F3 44 31 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne NR1H4 22 49 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne P4HTM 0 41 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne FABH 0 41 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne AKR1C3 36 40 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne AKR1C2 39 40 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne KCNK3 82 40 Cc1ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1Br ZINC000147346244 FH On-Demand Anodyne KCNK9 49 38 CC[C@H](NC(=O)c1c(OC)cccc1[N+](=O)[O-])C(=O)O ZINC000147346248 CD For-Sale Bother COLA 71 34 CC[C@H](NC(=O)c1c(OC)cccc1[N+](=O)[O-])C(=O)O ZINC000147346248 CD For-Sale Bother ACE2 42 33 CC[C@H](NC(=O)c1c(OC)cccc1[N+](=O)[O-])C(=O)O ZINC000147346248 CD For-Sale Bother ALS 30 45 C[C@H]1CC[C@@H](C)N(C(=O)c2cccc3c2OCCN3)C1 ZINC000147346262 CF For-Sale Anodyne HCRTR1 58 36 CCCCCCCCNC(=O)c1nc(NC)ccc1Cl ZINC000147346280 CH For-Sale Mild S1PR2 42 35 CCCCCCCCNC(=O)c1nc(NC)ccc1Cl ZINC000147346280 CH For-Sale Mild ASAH1 84 40 Cc1nc(-c2cccc(NC(=O)C(=O)NCC(C)(C)N3CCC[C@@H](C)C3)c2)oc1C ZINC000147346376 HH On-Demand Anodyne PDE8B 43 31 COCc1nc(C(=O)Nc2nc3c(s2)C[C@H](C)CC3)cs1 ZINC000147346414 DG On-Demand Anodyne SLC27A1 26 40 C=CCCOCC(=O)N1CCC(NS(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147346434 FD On-Demand Mild TGM2 17 44 C=CCCOCC(=O)N1CCC(NS(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147346434 FD On-Demand Mild F13A1 21 44 C=CCCOCC(=O)N1CCC(NS(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147346434 FD On-Demand Mild CCR8 68 40 C=CCCOCC(=O)N1CCC(NS(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147346434 FD On-Demand Mild SFRP1 117 38 C=CCCOCC(=O)N1CCC(NS(=O)(=O)c2ccc(F)cc2)CC1 ZINC000147346434 FD On-Demand Mild WNT3 80 38 CC(C)(C)CC[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147346465 KK Annotated Anodyne GCGR 56 73 CC(C)(C)CC[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147346465 KK Annotated Anodyne GLP1R 25 73 CC(C)(C)CC[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147346465 KK Annotated Anodyne GIPR 60 42 Oc1ccc2c(F)c(F)c(F)c(F)c2c1 ZINC000147346467 BG For-Sale Anodyne ESR2 32 44 Cc1nc(C)c(C(=O)Nc2ccc(F)c(C(=O)O)c2)o1 ZINC000147346479 CE On-Demand Anodyne DGAT1 22 40 Cc1nc(C)c(C(=O)Nc2ccc(F)c(C(=O)O)c2)o1 ZINC000147346479 CE On-Demand Anodyne Q25615_ONCVO 41 30 Cc1nc(C)c(C(=O)Nc2ccc(F)c(C(=O)O)c2)o1 ZINC000147346479 CE On-Demand Anodyne KCNK3 42 32 FC(F)(F)c1cnc(N(CCBr)C2CCCC2)c(Cl)c1 ZINC000147346482 FJ For-Sale Reactive TRPM8 41 35 CC(C)CCCCNCc1cccc(Br)c1 ZINC000147346524 CI For-Sale Anodyne FDFT1 0 47 CC(C)CCCCNCc1cccc(Br)c1 ZINC000147346524 CI For-Sale Anodyne LEF 76 41 CCCCCCCCNC(=O)c1cnccc1N ZINC000147346533 BF For-Sale Mild FAAH 17 45 CCCCCCCCNC(=O)c1cnccc1N ZINC000147346533 BF For-Sale Mild PA2A1_NAJMO 0 40 CCCCCCCCNC(=O)c1cnccc1N ZINC000147346533 BF For-Sale Mild ASAH1 91 37 COCc1nc(C(=O)Nc2nc3c(s2)C[C@@H](C)CC3)cs1 ZINC000147346590 DG On-Demand Anodyne SLC27A1 26 40 O=C(CCNC1(C(=O)O)CCC1)Nc1ccccc1 ZINC000147346663 CD For-Sale Anodyne LTA4H 18 40 O=C(CCNC1(C(=O)O)CCC1)Nc1ccccc1 ZINC000147346663 CD For-Sale Anodyne HDAC10 20 45 O=C(CCNC1(C(=O)O)CCC1)Nc1ccccc1 ZINC000147346663 CD For-Sale Anodyne HDAC2 17 45 O=C(CCNC1(C(=O)O)CCC1)Nc1ccccc1 ZINC000147346663 CD For-Sale Anodyne HDAC3 22 45 O=C(CCNC1(C(=O)O)CCC1)Nc1ccccc1 ZINC000147346663 CD For-Sale Anodyne HDAC6 16 45 O=C(CCNC1(C(=O)O)CCC1)Nc1ccccc1 ZINC000147346663 CD For-Sale Anodyne PFHDAC1 0 45 CCN(CCCNC(=O)[C@H]1c2ccccc2C(=O)N(Cc2ccc(F)cc2)[C@H]1c1ccc(OC)cc1)Cc1ccccc1 ZINC000147346685 KK In-Stock Anodyne TSHR 50 35 CCN(CCCNC(=O)[C@H]1c2ccccc2C(=O)N(Cc2ccc(F)cc2)[C@H]1c1ccc(OC)cc1)Cc1ccccc1 ZINC000147346685 KK In-Stock Anodyne ACHE 0 42 CCCCCCCCNC(=O)c1ccc(N)nc1 ZINC000147346734 BF For-Sale Mild FOLH1 24 44 CCCCCCCCNC(=O)c1ccc(N)nc1 ZINC000147346734 BF For-Sale Mild THRB 0 51 CCCCCCCCNC(=O)c1ccc(N)nc1 ZINC000147346734 BF For-Sale Mild KCNQ1 0 46 CCCCCCCCNC(=O)c1ccc(N)nc1 ZINC000147346734 BF For-Sale Mild FAAH 17 44 CCCCCCCCNC(=O)c1ccc(N)nc1 ZINC000147346734 BF For-Sale Mild S1PR2 40 36 CCCCCCCCNC(=O)c1ccc(N)nc1 ZINC000147346734 BF For-Sale Mild EPHX2 36 57 CCCCCCCCNC(=O)c1ccc(N)nc1 ZINC000147346734 BF For-Sale Mild ASAH1 93 37 CCCCCCCCNC(=O)c1ccc(N)nc1 ZINC000147346734 BF For-Sale Mild ACAT 0 43 COC(=O)/C=C/C(=O)OCCN1CCCCC1 ZINC000147346746 BC For-Sale Anodyne HTR4 18 50 COC(=O)/C=C/C(=O)OCCN1CCCCC1 ZINC000147346746 BC For-Sale Anodyne HCAR2 30 42 COC(=O)/C=C/C(=O)OCCN1CCCCC1 ZINC000147346746 BC For-Sale Anodyne PSMB2 44 33 CC(C)CCCCN[C@@H](C)CCC(=O)O ZINC000147346748 BF For-Sale Anodyne FOLH1 39 40 CC(C)CCCCN[C@@H](C)CCC(=O)O ZINC000147346748 BF For-Sale Anodyne Q6UB75_PIG 0 40 CC(C)CCN1C(=O)c2ccc(I)cc2S1(=O)=O ZINC000147346758 GE For-Sale Anodyne ELANE 16 41 COCc1nc(C(=O)N[C@@H](CC(C)C)c2ccccc2)cs1 ZINC000147346794 DH On-Demand Anodyne PTGER3 78 41 COCc1nc(C(=O)N[C@@H](CC(C)C)c2ccccc2)cs1 ZINC000147346794 DH On-Demand Anodyne CTSK 19 46 COCc1nc(C(=O)N[C@@H](CC(C)C)c2ccccc2)cs1 ZINC000147346794 DH On-Demand Anodyne TACR3 44 37 COCc1nc(C(=O)N[C@@H](CC(C)C)c2ccccc2)cs1 ZINC000147346794 DH On-Demand Anodyne CAPNS1 48 32 COCc1nc(C(=O)N[C@@H](CC(C)C)c2ccccc2)cs1 ZINC000147346794 DH On-Demand Anodyne CAPN2 49 32 COCc1nc(C(=O)N[C@@H](CC(C)C)c2ccccc2)cs1 ZINC000147346794 DH On-Demand Anodyne NPR 48 33 Cc1cc(C)c(OCCn2ccnc2)c(S(N)(=O)=O)c1 ZINC000147346815 CD For-Sale Anodyne TBXAS1 31 44 CCN(CCCNC(=O)[C@@H]1c2ccccc2C(=O)N(Cc2ccc(F)cc2)[C@H]1c1ccc(OC)cc1)Cc1ccccc1 ZINC000147346885 KK In-Stock Anodyne TSHR 50 35 CCN(CCCNC(=O)[C@@H]1c2ccccc2C(=O)N(Cc2ccc(F)cc2)[C@H]1c1ccc(OC)cc1)Cc1ccccc1 ZINC000147346885 KK In-Stock Anodyne ACHE 0 42 CCCCCCCCNC(=O)c1cccc(F)c1NCC ZINC000147346937 CI For-Sale Mild ASAH1 101 39 CCCCCCCCNC(=O)c1cccc(F)c1NCC ZINC000147346937 CI For-Sale Mild ACAT 0 47 CCCCCCCCNC(=O)c1cccc(F)c1NCC ZINC000147346937 CI For-Sale Mild PSBA 0 40 CC(C)CCCCN[C@H](C)CCC(=O)O ZINC000147346946 BF For-Sale Anodyne FOLH1 39 40 CC(C)CCCCN[C@H](C)CCC(=O)O ZINC000147346946 BF For-Sale Anodyne Q6UB75_PIG 0 40 CSc1nn(-c2ccccc2)c2cc(N3CCN(C(=O)c4ccccn4)CC3)ccc12 ZINC000147346993 II Annotated Anodyne KHK 0 64 COCc1nc(C(=O)N[C@H](CC(C)C)c2ccccc2)cs1 ZINC000147346997 DH On-Demand Anodyne PTGER4 21 41 COCc1nc(C(=O)N[C@H](CC(C)C)c2ccccc2)cs1 ZINC000147346997 DH On-Demand Anodyne PTGER3 78 41 COCc1nc(C(=O)N[C@H](CC(C)C)c2ccccc2)cs1 ZINC000147346997 DH On-Demand Anodyne CTSK 19 46 COCc1nc(C(=O)N[C@H](CC(C)C)c2ccccc2)cs1 ZINC000147346997 DH On-Demand Anodyne TACR3 44 37 COCc1nc(C(=O)N[C@H](CC(C)C)c2ccccc2)cs1 ZINC000147346997 DH On-Demand Anodyne CAPNS1 48 32 COCc1nc(C(=O)N[C@H](CC(C)C)c2ccccc2)cs1 ZINC000147346997 DH On-Demand Anodyne CAPN2 49 32 COCc1nc(C(=O)N[C@H](CC(C)C)c2ccccc2)cs1 ZINC000147346997 DH On-Demand Anodyne NPR 48 33 CN(Cc1cscn1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147346998 FE On-Demand Anodyne CASR 47 38 O=C[C@@H](O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]1O)[C@@H](O)[C@H](O)[C@H](O)CO ZINC000147347006 EA For-Sale Mild FIMH 76 40 CCCCOc1ccc2cc3cc(I)c(=O)c(I)c-3oc2c1 ZINC000147347014 KK For-Sale Anodyne ALDH2 59 32 CCCCOc1ccc2cc3cc(I)c(=O)c(I)c-3oc2c1 ZINC000147347014 KK For-Sale Anodyne CA7 15 55 O=C(O)C1(NCc2ccc(OC(F)(F)F)cc2)CCC1 ZINC000147347041 CF On-Demand Anodyne GRIN2B 26 43 O=C(O)C1(NCc2ccc(OC(F)(F)F)cc2)CCC1 ZINC000147347041 CF On-Demand Anodyne SCN9A 0 42 CCOc1cccc([N+](=O)[O-])c1C(=O)N[C@@H](CC)C(=O)O ZINC000147347087 CD On-Demand Bother COLA 43 32 CCOc1cccc([N+](=O)[O-])c1C(=O)N[C@@H](CC)C(=O)O ZINC000147347087 CD On-Demand Bother ACE2 44 33 CC(C)/C=C/NC(=O)OC(C)(C)C ZINC000147347101 AF For-Sale Anodyne CTSK 20 46 N#Cc1cc(F)cc(OCc2ccccc2)c1 ZINC000147347141 BG On-Demand Mild MAOB 26 53 N#Cc1cc(F)cc(OCc2ccccc2)c1 ZINC000147347141 BG On-Demand Mild GRM5 31 45 N#Cc1cc(F)cc(OCc2ccccc2)c1 ZINC000147347141 BG On-Demand Mild FFAR1 19 43 CCCCCCCCNC(=O)c1cccc(F)c1NC ZINC000147347148 CH For-Sale Mild ASAH1 103 40 CN(Cc1cscn1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147347193 FE On-Demand Anodyne CASR 47 38 CCCNc1cccc(NCc2cccnc2)n1 ZINC000147347208 BF For-Sale Anodyne TBXAS1 0 42 CCCNc1cccc(NCc2cccnc2)n1 ZINC000147347208 BF For-Sale Anodyne FDFT1 0 40 CCCNc1cccc(NCc2cccnc2)n1 ZINC000147347208 BF For-Sale Anodyne CLK4 15 43 FC(F)CNCc1ccccc1OC(F)F ZINC000147347210 BF On-Demand Anodyne PHES 0 55 CSc1nn(-c2ccccc2)c2cc(N3CCN(Cc4cccnc4)CC3)ccc12 ZINC000147347223 HI Annotated Anodyne DRD4 37 44 CSc1nn(-c2ccccc2)c2cc(N3CCN(Cc4cccnc4)CC3)ccc12 ZINC000147347223 HI Annotated Anodyne KHK 0 61 Cc1cc(C)c(OCCCn2ccnc2)c(S(N)(=O)=O)c1 ZINC000147347228 DD For-Sale Anodyne TBXAS1 40 42 Cc1cc(C)c(OCCCn2ccnc2)c(S(N)(=O)=O)c1 ZINC000147347228 DD For-Sale Anodyne QPCT 41 35 CCCCCCCCNC(=O)c1ccc(NCCC)nn1 ZINC000147347329 CG For-Sale Mild LPAR2 44 34 CCCCCCCCNC(=O)c1ccc(NCCC)nn1 ZINC000147347329 CG For-Sale Mild S1PR2 65 36 CCCCCCCCNC(=O)c1ccc(NCCC)nn1 ZINC000147347329 CG For-Sale Mild SCD1 15 46 CCCCCCCCNC(=O)c1ccc(NCCC)nn1 ZINC000147347329 CG For-Sale Mild ASAH1 88 37 CC[C@H](NC(=O)c1cc(C)cc(Cl)c1)C(=O)O ZINC000147347344 CE On-Demand Anodyne CCKAR 0 44 CC[C@H](NC(=O)c1cc(C)cc(Cl)c1)C(=O)O ZINC000147347344 CE On-Demand Anodyne CCKBR 26 41 CC[C@H](NC(=O)c1cc(C)cc(Cl)c1)C(=O)O ZINC000147347344 CE On-Demand Anodyne CTSV 25 45 Cc1ncoc1C(=O)Nc1ccc(F)c(C(=O)O)c1 ZINC000147347369 CE On-Demand Anodyne KCNK3 89 36 Cc1ncoc1C(=O)Nc1ccc(F)c(C(=O)O)c1 ZINC000147347369 CE On-Demand Anodyne KCNK9 47 35 N[C@H](CC(=O)NN1CCCCC1)c1ccccc1 ZINC000147347410 BD For-Sale Anodyne KCNQ2 49 35 N[C@H](CC(=O)NN1CCCCC1)c1ccccc1 ZINC000147347410 BD For-Sale Anodyne DPP7 37 40 CSc1nn(-c2ccccc2)c2cc(N3CCN(C(=O)[C@@H]4CCCN4)CC3)ccc12 ZINC000147347419 HG Annotated Anodyne KHK 0 76 O=C(NCCc1cccs1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147347433 FH For-Sale Anodyne ADAM17 0 40 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(NC(=O)c3ccc(F)cc3)cc2)C1 ZINC000147347449 HG On-Demand Anodyne TGM2 73 41 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(NC(=O)c3ccc(F)cc3)cc2)C1 ZINC000147347449 HG On-Demand Anodyne F13A1 82 41 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(NC(=O)c3ccc(F)cc3)cc2)C1 ZINC000147347449 HG On-Demand Anodyne NAMPT 31 41 CCCCCCCCNC(=O)c1cccc(NCCC)n1 ZINC000147347463 CH For-Sale Mild S1PR2 53 37 CCCCCCCCNC(=O)c1cccc(NCCC)n1 ZINC000147347463 CH For-Sale Mild ASAH1 86 36 O=C(Nc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1Cl)c1ccco1 ZINC000147347465 HK On-Demand Anodyne GRM4 23 47 O=C(Nc1ccc2oc(=O)[nH]c2c1)c1cccnc1Oc1ccc(Cl)cc1Cl ZINC000147347486 HJ On-Demand Anodyne UGCG 34 41 O=C(Nc1ccc2oc(=O)[nH]c2c1)c1cccnc1Oc1ccc(Cl)cc1Cl ZINC000147347486 HJ On-Demand Anodyne GRM4 50 42 O=C(Nc1ccc2oc(=O)[nH]c2c1)c1cccnc1Oc1ccc(Cl)cc1Cl ZINC000147347486 HJ On-Demand Anodyne NR2E3 63 35 O=C(Nc1ccc2oc(=O)[nH]c2c1)c1cccnc1Oc1ccc(Cl)cc1Cl ZINC000147347486 HJ On-Demand Anodyne SHH 42 37 c1ccc(CCNc2ncc3ccccc3n2)cc1 ZINC000147347517 BG For-Sale Anodyne STAT6 41 48 c1ccc(CCNc2ncc3ccccc3n2)cc1 ZINC000147347517 BG For-Sale Anodyne MRGPRX1 17 41 c1ccc(CCNc2ncc3ccccc3n2)cc1 ZINC000147347517 BG For-Sale Anodyne PETD 0 43 Cc1cc(NC(=O)c2ccccc2NS(=O)(=O)c2cccc([N+](=O)[O-])c2)n(C)n1 ZINC000147347571 HF On-Demand Bother PRTN3 47 35 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne AVPR1A 18 46 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne DHODH 27 42 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne PYGL 27 41 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne JAK1 0 44 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne GRM4 51 45 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne NR1H4 17 52 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne TYK2 28 44 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne CSF1R 19 42 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne ENV 42 32 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne ACPS 0 41 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne TAAR1 15 40 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne NR2E3 67 42 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne SHH 59 43 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne AKR1C2 59 39 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne SMO 29 45 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne GALE 0 43 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne Q25615_ONCVO 55 33 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne KCNK3 97 49 O=C(O)c1cc(NC(=O)c2cccc(F)c2Cl)ccc1Cl ZINC000147347587 EI On-Demand Anodyne KCNK9 75 38 CN(C)C1(CNc2cc(C(=O)O)ccc2N)CCCC1 ZINC000147347588 CE For-Sale Anodyne RARA 41 32 CN(C)C1(CNc2cc(C(=O)O)ccc2N)CCCC1 ZINC000147347588 CE For-Sale Anodyne RARG 40 36 CN(C)C1(CNc2cc(C(=O)O)ccc2N)CCCC1 ZINC000147347588 CE For-Sale Anodyne RXRG 51 33 CN(C)C1(CNc2cc(C(=O)O)ccc2N)CCCC1 ZINC000147347588 CE For-Sale Anodyne RARB 41 36 CN(C)C1(CNc2cc(C(=O)O)ccc2N)CCCC1 ZINC000147347588 CE For-Sale Anodyne RXRB 50 33 N[C@@H](CC(=O)NN1CCCCC1)c1ccccc1 ZINC000147347599 BD For-Sale Anodyne KCNQ2 49 35 N[C@@H](CC(=O)NN1CCCCC1)c1ccccc1 ZINC000147347599 BD For-Sale Anodyne DPP7 37 40 CSc1nn(-c2ccccc2)c2cc(N3CCN(C(=O)[C@H]4CCCN4)CC3)ccc12 ZINC000147347633 HG Annotated Anodyne KHK 0 76 CCCCCCCCNC(=O)c1cnc(C)cc1NCC ZINC000147347635 CH For-Sale Mild MERTK 23 42 CCCCCCCCNC(=O)c1cnc(C)cc1NCC ZINC000147347635 CH For-Sale Mild ASAH1 75 33 O=C(NCCc1cccs1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147347656 DG On-Demand Anodyne ADAM17 0 40 O=C(Nc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1Cl)c1ccco1 ZINC000147347661 HK On-Demand Anodyne GRM4 23 47 COCc1nc(C(=O)N[C@@H](c2ccc(Cl)cc2)C2CC2)cs1 ZINC000147347679 EH On-Demand Anodyne AKT1 23 41 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(CCN3CCCC3)cc2)C1 ZINC000147347702 HF On-Demand Anodyne HRH3 19 42 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(CCN3CCCC3)cc2)C1 ZINC000147347702 HF On-Demand Anodyne BIRC2 56 39 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(COc2cccc(F)c2)c1 ZINC000147347720 GG On-Demand Anodyne F10 16 44 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne RARA 21 40 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne MAOB 19 42 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne AVPR2 33 42 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne AVPR1A 22 42 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne CPT1A 54 40 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne CPT2 45 36 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne PRNP 31 41 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne F3 45 31 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne NR1H4 22 47 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne P4HTM 0 42 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne CSF1R 26 52 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne FABH 0 40 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne BTK 21 40 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne TAAR1 27 47 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne AKR1C3 34 41 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne SHH 58 39 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne AKR1C2 32 41 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne SMO 28 40 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne KCNK3 102 42 Cc1ccc(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)cc1Br ZINC000147347768 FI On-Demand Anodyne KCNK9 53 39 O=C(NN1CCCCC1)c1ccc2c(c1)CCCN2 ZINC000147347829 CE For-Sale Anodyne CNR1 61 38 CCCCCCCCNC(=O)c1nnc(NC)s1 ZINC000147347840 CF For-Sale Mild ASAH1 80 36 O=C(Nc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1Cl)c1ccco1 ZINC000147347867 HK On-Demand Anodyne GRM4 23 47 CCc1nn(-c2ccccc2)c2cc(N3CCC(N4CCNCC4)CC3)ccc12 ZINC000147347872 GG Annotated Anodyne KHK 0 85 CCCCCCCCCCCC[C@@H](Oc1cccc([N+](=O)[O-])c1)C(=O)OCC ZINC000147347887 GK For-Sale Mild INHA 35 53 CCCCCCCCCCCC[C@@H](Oc1cccc([N+](=O)[O-])c1)C(=O)OCC ZINC000147347887 GK For-Sale Mild CACNA1C 70 50 CCCCCCCCCCCC[C@@H](Oc1cccc([N+](=O)[O-])c1)C(=O)OCC ZINC000147347887 GK For-Sale Mild TBXA2R 18 41 CCCCCCCCCCCC[C@@H](Oc1cccc([N+](=O)[O-])c1)C(=O)OCC ZINC000147347887 GK For-Sale Mild CACNA1D 105 50 CCCCCCCCCCCC[C@@H](Oc1cccc([N+](=O)[O-])c1)C(=O)OCC ZINC000147347887 GK For-Sale Mild ACR 17 42 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(CCN3CCCC3)cc2)C1 ZINC000147347918 HF On-Demand Anodyne HRH3 19 42 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(CCN3CCCC3)cc2)C1 ZINC000147347918 HF On-Demand Anodyne BIRC2 56 39 CNc1nc(Oc2cccnc2)nc(-n2cncn2)n1 ZINC000147347953 CC For-Sale Anodyne PDE4A 15 43 C=C[C@H]1[C@H](O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)[C@H]2O)OC=C2C(=O)OCC[C@H]21 ZINC000147347966 KA Annotated Mild VEGFA 40 42 C=C[C@H]1[C@H](O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O[C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)[C@H]2O)OC=C2C(=O)OCC[C@H]21 ZINC000147347966 KA Annotated Mild FIMH 59 33 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(COc2cccc(F)c2)c1 ZINC000147347972 GG On-Demand Anodyne F10 16 44 Cc1cc(NC(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(F)c2)n(C)n1 ZINC000147347984 HG On-Demand Anodyne PRTN3 59 39 Cc1nc(C)c(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)o1 ZINC000147347988 CF On-Demand Anodyne SORT1 23 40 Cc1nc(C)c(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)o1 ZINC000147347988 CF On-Demand Anodyne AGPAT2 52 39 Cc1nc(C)c(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)o1 ZINC000147347988 CF On-Demand Anodyne CSF1R 22 42 Cc1nc(C)c(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)o1 ZINC000147347988 CF On-Demand Anodyne NR2E3 61 35 Cc1nc(C)c(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)o1 ZINC000147347988 CF On-Demand Anodyne SHH 65 47 Cc1nc(C)c(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)o1 ZINC000147347988 CF On-Demand Anodyne SMO 25 43 Cc1nc(C)c(C(=O)Nc2ccc(Cl)c(C(=O)O)c2)o1 ZINC000147347988 CF On-Demand Anodyne KCNK3 40 35 O[C@H](CNCCCN1CCOCC1)COc1cccc2[nH]ccc12 ZINC000147348022 ED On-Demand Anodyne ADRB2 17 54 O[C@H](CNCCCN1CCOCC1)COc1cccc2[nH]ccc12 ZINC000147348022 ED On-Demand Anodyne ADRB1 37 54 O[C@H](CNCCCN1CCOCC1)COc1cccc2[nH]ccc12 ZINC000147348022 ED On-Demand Anodyne HTR1A 20 54 O[C@H](CNCCCN1CCOCC1)COc1cccc2[nH]ccc12 ZINC000147348022 ED On-Demand Anodyne SLC6A4 19 41 O[C@H](CNCCCN1CCOCC1)COc1cccc2[nH]ccc12 ZINC000147348022 ED On-Demand Anodyne ADRB3 21 45 CCc1nn(-c2ccccc2)c2cc(-c3ccc(OC4CCNCC4)cc3)ccc12 ZINC000147348069 GK Annotated Anodyne KHK 0 66 CCCCCCCCNC(=O)c1cnc(NCC)c(Cl)c1 ZINC000147348070 DI For-Sale Mild ASAH1 74 38 C/C=C/[C@@H]1C[C@@H](O)CC(=O)O1 ZINC000147348083 AC For-Sale Anodyne HMGCR 75 49 CC[C@@H]1OCC(=O)[C@H]1NC(=O)OC(C)(C)C ZINC000147348111 BD For-Sale Anodyne CTSK 28 43 CCCCCCCCCCCC[C@H](Oc1cccc([N+](=O)[O-])c1)C(=O)OCC ZINC000147348142 GK For-Sale Mild INHA 35 53 CCCCCCCCCCCC[C@H](Oc1cccc([N+](=O)[O-])c1)C(=O)OCC ZINC000147348142 GK For-Sale Mild CACNA1C 70 50 CCCCCCCCCCCC[C@H](Oc1cccc([N+](=O)[O-])c1)C(=O)OCC ZINC000147348142 GK For-Sale Mild TBXA2R 18 41 CCCCCCCCCCCC[C@H](Oc1cccc([N+](=O)[O-])c1)C(=O)OCC ZINC000147348142 GK For-Sale Mild CACNA1D 105 50 CCCCCCCCCCCC[C@H](Oc1cccc([N+](=O)[O-])c1)C(=O)OCC ZINC000147348142 GK For-Sale Mild ACR 17 42 CC[C@H](NCC(F)F)c1ccc(O)cc1 ZINC000147348150 BF For-Sale Anodyne ESR1 16 41 CC[C@H](NCC(F)F)c1ccc(O)cc1 ZINC000147348150 BF For-Sale Anodyne NMUR2 0 42 CC(C)(C)OC(=O)N1CCN(Cc2ccccc2)C[C@H]1CC(=O)O ZINC000147348175 EF In-Stock Anodyne DRD4 43 37 CC(C)(C)OC(=O)N1CCN(Cc2ccccc2)C[C@H]1CC(=O)O ZINC000147348175 EF In-Stock Anodyne SIGMAR1 57 45 CC(C)(C)OC(=O)N1CCN(Cc2ccccc2)C[C@H]1CC(=O)O ZINC000147348175 EF In-Stock Anodyne CACNA1G 32 40 Cc1cc(NC(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(C)c2)n(C)n1 ZINC000147348204 HG On-Demand Anodyne PRTN3 50 37 Cc1cc(NC(=O)c2ccccc2NS(=O)(=O)c2ccc(F)c(C)c2)n(C)n1 ZINC000147348204 HG On-Demand Anodyne LEF 32 40 O=C(O)c1cc(NC(=O)C2[C@H]3CCCC[C@H]23)ccc1Cl ZINC000147348211 CG On-Demand Anodyne NPY2R 24 41 O=C(O)c1cc(NC(=O)C2[C@H]3CCCC[C@H]23)ccc1Cl ZINC000147348211 CG On-Demand Anodyne ENV 41 32 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348243 HI On-Demand Anodyne ADRB2 15 48 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348243 HI On-Demand Anodyne ADRB1 18 44 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348243 HI On-Demand Anodyne HTR1A 36 71 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348243 HI On-Demand Anodyne HTR1D 21 44 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348243 HI On-Demand Anodyne HTR1B 19 44 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348243 HI On-Demand Anodyne SLC6A4 45 71 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348243 HI On-Demand Anodyne ADRB3 20 54 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348243 HI On-Demand Anodyne ABCB1 46 38 O[C@@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348243 HI On-Demand Anodyne CCR2 22 40 CC[C@H](CNS(=O)(=O)c1ccccc1C)CC(=O)O ZINC000147348264 CD On-Demand Anodyne ITGAV 44 46 CC[C@H](CNS(=O)(=O)c1ccccc1C)CC(=O)O ZINC000147348264 CD On-Demand Anodyne ITGA2 0 43 CCCCCCCCNC(=O)c1cnc(N)c(Cl)c1 ZINC000147348276 CG For-Sale Mild SCNN1A 24 41 CCCCCCCCNC(=O)c1cnc(N)c(Cl)c1 ZINC000147348276 CG For-Sale Mild ASAH1 87 39 CCc1nn(-c2ccccc2)c2cc(OC3CN(C4CCNCC4)C3)ccc12 ZINC000147348290 GG Annotated Anodyne KHK 0 66 C[C@H]1CCC[C@H](C)N1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147348299 DH For-Sale Anodyne CACNA1I 48 36 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCC(C)CC3)cc1)C2 ZINC000147348318 HH On-Demand Anodyne MTNR1A 15 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCC(C)CC3)cc1)C2 ZINC000147348318 HH On-Demand Anodyne MTNR1B 16 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCC(C)CC3)cc1)C2 ZINC000147348318 HH On-Demand Anodyne ROCK2 28 50 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCC(C)CC3)cc1)C2 ZINC000147348318 HH On-Demand Anodyne EPHX2 17 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCC(C)CC3)cc1)C2 ZINC000147348318 HH On-Demand Anodyne L3MBTL3 54 36 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCC(C)CC3)cc1)C2 ZINC000147348318 HH On-Demand Anodyne TRPC6 31 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)N3CCC(C)CC3)cc1)C2 ZINC000147348318 HH On-Demand Anodyne TRPC3 24 43 COC(=O)/C=C/C(=O)OCCCN1CCOCC1 ZINC000147348347 CB For-Sale Anodyne PAOX 17 43 CC[C@@H](NCC(F)F)c1ccc(O)cc1 ZINC000147348355 BF For-Sale Anodyne ESR1 16 41 CC[C@@H](NCC(F)F)c1ccc(O)cc1 ZINC000147348355 BF For-Sale Anodyne NMUR2 0 42 O=C(O)c1cc(NC(=O)C2[C@H]3CCCC[C@@H]23)ccc1Cl ZINC000147348414 CG For-Sale Anodyne NPY2R 24 41 O=C(O)c1cc(NC(=O)C2[C@H]3CCCC[C@@H]23)ccc1Cl ZINC000147348414 CG For-Sale Anodyne ENV 41 32 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348466 HI On-Demand Anodyne ADRB2 15 48 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348466 HI On-Demand Anodyne ADRB1 18 44 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348466 HI On-Demand Anodyne HTR1A 36 71 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348466 HI On-Demand Anodyne HTR1D 21 44 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348466 HI On-Demand Anodyne HTR1B 19 44 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348466 HI On-Demand Anodyne SLC6A4 45 71 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348466 HI On-Demand Anodyne ADRB3 20 54 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348466 HI On-Demand Anodyne ABCB1 46 38 O[C@H](COc1cccc2[nH]ccc12)CN1CCC(c2c[nH]c3ccc(F)cc23)CC1 ZINC000147348466 HI On-Demand Anodyne CCR2 22 40 CC[C@@H](CNS(=O)(=O)c1ccccc1C)CC(=O)O ZINC000147348468 CD On-Demand Anodyne ITGAV 44 46 CC[C@@H](CNS(=O)(=O)c1ccccc1C)CC(=O)O ZINC000147348468 CD On-Demand Anodyne ITGA2 0 43 CCCCCCCCNC(=O)c1nc(N)ccc1Cl ZINC000147348479 CG For-Sale Mild CNR1 15 46 CCCCCCCCNC(=O)c1nc(N)ccc1Cl ZINC000147348479 CG For-Sale Mild SCNN1A 75 45 CCCCCCCCNC(=O)c1nc(N)ccc1Cl ZINC000147348479 CG For-Sale Mild ASAH1 92 40 C[C@@H]1CCC[C@@H](C)N1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147348489 DH For-Sale Anodyne CACNA1I 48 36 CCc1nn(-c2ccccc2)c2cc(N3CC[C@H](N4CCNCC4)C3)ccc12 ZINC000147348510 GG Annotated Anodyne KHK 0 75 COc1ccc(Br)cc1CNCC(F)F ZINC000147348589 CF On-Demand Anodyne PHES 0 49 CC(C)N1CC[C@@H](Oc2ccccc2)C1 ZINC000147348600 BF On-Demand Anodyne HRH3 32 56 COc1ccc(S(=O)(=O)Nc2ccccc2C(=O)Nc2cc(C)nn2C)cc1 ZINC000147348603 HF On-Demand Anodyne PRTN3 70 45 COc1ccc(S(=O)(=O)Nc2ccccc2C(=O)Nc2cc(C)nn2C)cc1 ZINC000147348603 HF On-Demand Anodyne FFAR4 19 42 COc1ccc(S(=O)(=O)Nc2ccccc2C(=O)Nc2cc(C)nn2C)cc1 ZINC000147348603 HF On-Demand Anodyne CREBBP 24 42 COc1ccc(S(=O)(=O)Nc2ccccc2C(=O)Nc2cc(C)nn2C)cc1 ZINC000147348603 HF On-Demand Anodyne BRD9 24 42 CC(C)CCCCN[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348607 CF For-Sale Anodyne CA2 80 43 CC(C)CCCCN[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348607 CF For-Sale Anodyne CA1 65 40 CC(C)CCCCN[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348607 CF For-Sale Anodyne CA7 52 38 CC(C)CCCCN[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348607 CF For-Sale Anodyne CA4 49 37 CC(C)CCCCN[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348607 CF For-Sale Anodyne CA12 48 41 CC(C)CCCCN[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348607 CF For-Sale Anodyne CA9 55 41 CC(C)CCCCN[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348607 CF For-Sale Anodyne CYNT 45 34 CC(C)CCCCN[C@@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348607 CF For-Sale Anodyne P96878_MYCTU 33 41 O=C(O)c1cc(NC(=O)C2[C@@H]3CCCC[C@@H]23)ccc1Cl ZINC000147348612 CG On-Demand Anodyne NPY2R 24 41 O=C(O)c1cc(NC(=O)C2[C@@H]3CCCC[C@@H]23)ccc1Cl ZINC000147348612 CG On-Demand Anodyne ENV 41 32 CN(C)C1(CNc2cccc(C(=O)O)c2N)CCCC1 ZINC000147348658 CE For-Sale Anodyne AKR1C2 44 38 CCCCCCCCC(=O)[C@@H]1COc2ccccc21 ZINC000147348661 CI For-Sale Mild LASR 57 39 CCCCCCCCC(=O)[C@@H]1COc2ccccc21 ZINC000147348661 CI For-Sale Mild CQSS 50 31 COc1cc(CBr)cc(I)c1OC ZINC000147348665 FG For-Sale Anodyne DRTS_TOXGO 40 33 CCO[C@H]1CCCN(S(=O)(=O)c2cc(CNC(C)=O)ccc2OC)C1 ZINC000147348679 FD On-Demand Anodyne TSHR 40 30 COCCOc1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)cc1F ZINC000147348680 HE On-Demand Anodyne MET 57 37 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CA2 66 48 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne PTGS2 63 50 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CA6 25 41 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CA1 57 42 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CA7 42 44 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CA13 33 41 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CA5B 31 40 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CA5A 33 40 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CA14 25 40 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CA12 57 44 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CA9 68 48 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CAH_METTE 52 41 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne CYNT 41 44 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne NCE103 26 44 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne MTCA1 33 40 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne P96878_MYCTU 35 40 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne MTCA2 34 40 Cc1cc(N)n(-c2ccc(S(N)(=O)=O)cc2)n1 ZINC000147348686 CC For-Sale Anodyne A6YCJ1_9METZ 40 44 CCCCCCCCNC(=O)c1ccc([N+](=O)[O-])c(N)c1 ZINC000147348696 CG For-Sale Mild FOLH1 17 43 CCCCCCCCNC(=O)c1ccc([N+](=O)[O-])c(N)c1 ZINC000147348696 CG For-Sale Mild ASAH1 73 34 CC[C@H](CNS(=O)(=O)c1cc(Cl)ccc1C)CC(=O)O ZINC000147348697 DE On-Demand Anodyne PTGDR2 28 41 CCc1nn(-c2ccccc2)c2cc(N3CC[C@@H](N4CCNCC4)C3)ccc12 ZINC000147348734 GG Annotated Anodyne KHK 0 75 Cc1cc(NC(=O)Nc2ccc(N3CCN(C)CC3)cc2C)n(-c2ccccn2)n1 ZINC000147348737 HG On-Demand Anodyne TNF 41 35 Cc1cc(NC(=O)Nc2ccc(N3CCN(C)CC3)cc2C)n(-c2ccccn2)n1 ZINC000147348737 HG On-Demand Anodyne MAPK7 22 40 NCCCCNC(=O)C[C@@H]1CNc2ccccc21 ZINC000147348784 BD For-Sale Anodyne POLG_WNV 50 31 Cc1cc(C)c(OCCN2CCCC2)c(S(N)(=O)=O)c1 ZINC000147348800 CD For-Sale Anodyne HRH3 16 43 Cc1cc(C)c(OCCN2CCCC2)c(S(N)(=O)=O)c1 ZINC000147348800 CD For-Sale Anodyne PSMB2 46 38 CC(C)CCCCN[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348837 CF For-Sale Anodyne CA2 80 43 CC(C)CCCCN[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348837 CF For-Sale Anodyne CA1 65 40 CC(C)CCCCN[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348837 CF For-Sale Anodyne CA7 52 38 CC(C)CCCCN[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348837 CF For-Sale Anodyne CA4 49 37 CC(C)CCCCN[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348837 CF For-Sale Anodyne CA12 48 41 CC(C)CCCCN[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348837 CF For-Sale Anodyne CA9 55 41 CC(C)CCCCN[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348837 CF For-Sale Anodyne CYNT 45 34 CC(C)CCCCN[C@H](C)c1ccc(S(N)(=O)=O)cc1 ZINC000147348837 CF For-Sale Anodyne P96878_MYCTU 33 41 Cc1ncoc1C(=O)Nc1ccc(Cl)c(C(=O)O)c1 ZINC000147348859 CF On-Demand Anodyne GRM4 46 38 Cc1ncoc1C(=O)Nc1ccc(Cl)c(C(=O)O)c1 ZINC000147348859 CF On-Demand Anodyne AGPAT2 43 37 Cc1ncoc1C(=O)Nc1ccc(Cl)c(C(=O)O)c1 ZINC000147348859 CF On-Demand Anodyne TYK2 43 34 Cc1ncoc1C(=O)Nc1ccc(Cl)c(C(=O)O)c1 ZINC000147348859 CF On-Demand Anodyne CSF1R 22 41 Cc1ncoc1C(=O)Nc1ccc(Cl)c(C(=O)O)c1 ZINC000147348859 CF On-Demand Anodyne SHH 64 43 Cc1ncoc1C(=O)Nc1ccc(Cl)c(C(=O)O)c1 ZINC000147348859 CF On-Demand Anodyne KCNK3 70 40 Cc1ncoc1C(=O)Nc1ccc(Cl)c(C(=O)O)c1 ZINC000147348859 CF On-Demand Anodyne KCNK9 44 35 CCCCCCCCC(=O)[C@H]1COc2ccccc21 ZINC000147348872 CI For-Sale Mild LASR 57 39 CCCCCCCCC(=O)[C@H]1COc2ccccc21 ZINC000147348872 CI For-Sale Mild CQSS 50 31 CC[C@@H](CNS(=O)(=O)c1cc(Cl)ccc1C)CC(=O)O ZINC000147348911 DE On-Demand Anodyne PTGDR2 28 41 COCCOc1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)cc1F ZINC000147348913 HE On-Demand Anodyne MET 57 37 C=CCNC(=O)c1cccc(S(=O)(=O)N2CCC[C@@H](OCC)C2)c1 ZINC000147348925 FD On-Demand Mild TGM2 53 36 C=CCNC(=O)c1cccc(S(=O)(=O)N2CCC[C@@H](OCC)C2)c1 ZINC000147348925 FD On-Demand Mild F13A1 46 34 C=CCNC(=O)c1cccc(S(=O)(=O)N2CCC[C@@H](OCC)C2)c1 ZINC000147348925 FD On-Demand Mild AKR1C3 57 39 CCCCCCCCNC(=O)c1nc(C(C)C)ncc1N ZINC000147348930 CG For-Sale Mild ASAH1 85 35 CCc1nn(-c2ccccc2)c2cc(N3CCN(C4CNC4)CC3)ccc12 ZINC000147348969 FF Annotated Anodyne KHK 0 85 NCCCCNC(=O)C[C@H]1CNc2ccccc21 ZINC000147348988 BD For-Sale Anodyne POLG_WNV 50 31 CCOC(=O)/C=C/C(=O)OCCN1CCOCC1 ZINC000147348990 CB For-Sale Anodyne HCAR2 24 49 COc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1Br ZINC000147349019 GH On-Demand Anodyne BMP1 55 35 CC(C)CCCCN[C@@H](C)c1ccc(C(C)(C)C)cc1 ZINC000147349069 CK For-Sale Anodyne LEF 21 42 Cc1ccc(C(=O)NCc2cccc(C(=O)O)c2)cc1Br ZINC000147349108 EG On-Demand Anodyne DRD4 40 32 Cc1ccc(C(=O)NCc2cccc(C(=O)O)c2)cc1Br ZINC000147349108 EG On-Demand Anodyne CHRM3 17 43 Cc1ccc(C(=O)NCc2cccc(C(=O)O)c2)cc1Br ZINC000147349108 EG On-Demand Anodyne MMP13 20 55 Cc1ccc(C(=O)NCc2cccc(C(=O)O)c2)cc1Br ZINC000147349108 EG On-Demand Anodyne PPARD 17 41 Cc1ccc(C(=O)NCc2cccc(C(=O)O)c2)cc1Br ZINC000147349108 EG On-Demand Anodyne ROCK2 17 45 Cc1ccc(C(=O)NCc2cccc(C(=O)O)c2)cc1Br ZINC000147349108 EG On-Demand Anodyne E1 0 43 Cc1ccc(C(=O)NCc2cccc(C(=O)O)c2)cc1Br ZINC000147349108 EG On-Demand Anodyne KDM4E 24 44 C=CCNC(=O)c1cccc(S(=O)(=O)N2CCC[C@H](OCC)C2)c1 ZINC000147349146 FD On-Demand Mild TGM2 53 36 C=CCNC(=O)c1cccc(S(=O)(=O)N2CCC[C@H](OCC)C2)c1 ZINC000147349146 FD On-Demand Mild F13A1 46 34 C=CCNC(=O)c1cccc(S(=O)(=O)N2CCC[C@H](OCC)C2)c1 ZINC000147349146 FD On-Demand Mild AKR1C3 57 39 CCCCCCCCNC(=O)c1cc(Cl)nc(NC)c1 ZINC000147349163 CH For-Sale Mild ASAH1 82 37 COc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1Br ZINC000147349219 GH On-Demand Anodyne BMP1 55 35 CC(C)CCCCN[C@H](C)c1ccc(C(C)(C)C)cc1 ZINC000147349241 CK For-Sale Anodyne LEF 21 42 Nc1ccc(C(=O)NN2CCCCC2)cc1Br ZINC000147349318 CE For-Sale Anodyne CNR1 59 37 Cc1nc(C)c(C(=O)NCc2cccc(C(=O)O)c2)o1 ZINC000147349339 CD On-Demand Anodyne MMP13 23 45 Cc1nc(C)c(C(=O)NCc2cccc(C(=O)O)c2)o1 ZINC000147349339 CD On-Demand Anodyne CARM1 50 32 COC(=O)C1(c2cccc(OCc3ccccc3)c2)CCCC1 ZINC000147349345 DI For-Sale Anodyne ALOX5 29 43 COC(=O)C1(c2cccc(OCc3ccccc3)c2)CCCC1 ZINC000147349345 DI For-Sale Anodyne MAOB 49 41 COC(=O)C1(c2cccc(OCc3ccccc3)c2)CCCC1 ZINC000147349345 DI For-Sale Anodyne CHRM3 26 41 COC(=O)C1(c2cccc(OCc3ccccc3)c2)CCCC1 ZINC000147349345 DI For-Sale Anodyne LTA4H 21 43 COC(=O)C1(c2cccc(OCc3ccccc3)c2)CCCC1 ZINC000147349345 DI For-Sale Anodyne PTGER4 18 40 COC(=O)C1(c2cccc(OCc3ccccc3)c2)CCCC1 ZINC000147349345 DI For-Sale Anodyne ALOX5AP 22 40 COC(=O)C1(c2cccc(OCc3ccccc3)c2)CCCC1 ZINC000147349345 DI For-Sale Anodyne ADAM17 36 60 COC(=O)C1(c2cccc(OCc3ccccc3)c2)CCCC1 ZINC000147349345 DI For-Sale Anodyne GYS1 46 34 COC(=O)C1(c2cccc(OCc3ccccc3)c2)CCCC1 ZINC000147349345 DI For-Sale Anodyne FFAR1 70 46 COC(=O)C1(c2cccc(OCc3ccccc3)c2)CCCC1 ZINC000147349345 DI For-Sale Anodyne SLC12A5 75 39 COC(=O)C1(c2cccc(OCc3ccccc3)c2)CCCC1 ZINC000147349345 DI For-Sale Anodyne PDS 66 35 C[C@H]1C[C@@H](C)CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147349369 DH On-Demand Anodyne CACNA1H 40 35 C[C@H]1C[C@@H](C)CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147349369 DH On-Demand Anodyne CACNA1I 42 33 CCCCCCCCNC(=O)c1ccc(NC)c(C)c1 ZINC000147349405 CI For-Sale Mild FOLH1 19 44 CCCCCCCCNC(=O)c1ccc(NC)c(C)c1 ZINC000147349405 CI For-Sale Mild KCNQ1 0 42 CCCCCCCCNC(=O)c1ccc(NC)c(C)c1 ZINC000147349405 CI For-Sale Mild S1PR2 51 36 CCCCCCCCNC(=O)c1ccc(NC)c(C)c1 ZINC000147349405 CI For-Sale Mild PA2A1_NAJMO 0 40 CCCCCCCCNC(=O)c1ccc(NC)c(C)c1 ZINC000147349405 CI For-Sale Mild ASAH1 89 37 CCCCCCCCNC(=O)c1ccc(NC)c(C)c1 ZINC000147349405 CI For-Sale Mild ACAT 0 47 COc1cccc2sc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)nc12 ZINC000147349526 EH On-Demand Bother KCNK9 40 38 CCc1nn(-c2ccccc2)c2cc(N3CCN([C@@H]4CCNC4)C3=O)ccc12 ZINC000147349528 GG Annotated Anodyne KHK 0 68 CCCCCCCN1C(=O)[C@@H](C)Oc2cc(I)ccc21 ZINC000147349544 GI For-Sale Mild FSHR 41 32 CCCCCCCN1C(=O)[C@@H](C)Oc2cc(I)ccc21 ZINC000147349544 GI For-Sale Mild PPARG 0 40 CC[C@H](CNS(=O)(=O)c1cccnc1)CC(=O)O ZINC000147349578 CC On-Demand Anodyne TBXAS1 60 42 CC[C@H](CNS(=O)(=O)c1cccnc1)CC(=O)O ZINC000147349578 CC On-Demand Anodyne NAMPT 37 41 Cc1cc(NC(=O)c2ccccc2Nc2ccc(OC(F)F)cc2)n(C)n1 ZINC000147349585 FI On-Demand Anodyne AKR1C3 20 40 Cc1cc(NC(=O)c2ccccc2Nc2ccc(OC(F)F)cc2)n(C)n1 ZINC000147349585 FI On-Demand Anodyne AKR1C2 63 40 O=C(O)c1cccc(CNC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147349595 CE On-Demand Anodyne F2 20 42 O=C(O)c1cccc(CNC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147349595 CE On-Demand Anodyne P2RX7 16 40 O=C(O)c1cccc(CNC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147349595 CE On-Demand Anodyne PREP 22 44 O=C(O)c1cccc(CNC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147349595 CE On-Demand Anodyne TMPRSS11D 52 33 CCCCCCCCNC(=O)c1nc(NCC)ccc1Cl ZINC000147349596 DI For-Sale Mild ASAH1 82 39 Cc1nn(C(F)F)c(C)c1CC(=O)NCCC(=O)N1CCOCC1 ZINC000147349604 EC On-Demand Anodyne P2RX7 26 40 C[C@H]1C[C@H](C)CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147349614 DH On-Demand Anodyne CACNA1H 40 35 C[C@H]1C[C@H](C)CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147349614 DH On-Demand Anodyne CACNA1I 42 33 CCCCCCCC(=O)SCC/C=C/COC(=O)[C@@H](NC(=O)c1csc(-c2csc(C)n2)n1)C(C)C ZINC000147349620 KK Annotated Mild HDAC4 0 43 CCc1nn(-c2ccccc2)c2cc(N3CCN([C@H]4CCNC4)C3=O)ccc12 ZINC000147349676 GG Annotated Anodyne KHK 0 68 CCc1ncc(C(=O)Nc2nc3cc(OC)c(OC)cc3s2)s1 ZINC000147349708 EH On-Demand Anodyne CSNK1D 44 42 CCc1ncc(C(=O)Nc2nc3cc(OC)c(OC)cc3s2)s1 ZINC000147349708 EH On-Demand Anodyne PIK3CG 17 43 CC(C)[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC=C[C@H](OS(C)(=O)=O)C1 ZINC000147349711 GD For-Sale Mild PGA5 40 35 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cccc2cccnc12 ZINC000147349715 GH On-Demand Anodyne LCK 25 42 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cccc2cccnc12 ZINC000147349715 GH On-Demand Anodyne MAPK14 15 42 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cccc2cccnc12 ZINC000147349715 GH On-Demand Anodyne P2RY1 29 48 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cccc2cccnc12 ZINC000147349715 GH On-Demand Anodyne FLT3 15 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cccc2cccnc12 ZINC000147349715 GH On-Demand Anodyne AURKA 15 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cccc2cccnc12 ZINC000147349715 GH On-Demand Anodyne MAPK7 26 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cccc2cccnc12 ZINC000147349715 GH On-Demand Anodyne WNT3 18 41 CC[C@@H](CNS(=O)(=O)c1cccnc1)CC(=O)O ZINC000147349767 CC On-Demand Anodyne TBXAS1 60 42 CC[C@@H](CNS(=O)(=O)c1cccnc1)CC(=O)O ZINC000147349767 CC On-Demand Anodyne NAMPT 37 41 CCCCCCCCNC(=O)c1cc(C)ccc1NCC ZINC000147349772 CJ For-Sale Mild PA2A1_NAJMO 0 42 CCCCCCCCNC(=O)c1cc(C)ccc1NCC ZINC000147349772 CJ For-Sale Mild ASAH1 73 36 CCCCCCCCNC(=O)c1cc(C)ccc1NCC ZINC000147349772 CJ For-Sale Mild ACAT 0 48 C[C@@H]1C[C@@H](C)CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147349788 DH On-Demand Anodyne CACNA1H 40 35 C[C@@H]1C[C@@H](C)CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147349788 DH On-Demand Anodyne CACNA1I 42 33 CCCCCCCN1C(=O)[C@H](C)Oc2cc(I)ccc21 ZINC000147349802 GI For-Sale Mild FSHR 41 32 CCCCCCCN1C(=O)[C@H](C)Oc2cc(I)ccc21 ZINC000147349802 GI For-Sale Mild PPARG 0 40 CNc1cccc(NCc2cccc(F)c2)n1 ZINC000147349811 BF For-Sale Anodyne HAO2 17 40 O=C(O)c1cccc(CNC(=O)C2[C@H]3CCCC[C@@H]23)c1 ZINC000147349825 CE For-Sale Anodyne F2 20 42 O=C(O)c1cccc(CNC(=O)C2[C@H]3CCCC[C@@H]23)c1 ZINC000147349825 CE For-Sale Anodyne P2RX7 16 40 O=C(O)c1cccc(CNC(=O)C2[C@H]3CCCC[C@@H]23)c1 ZINC000147349825 CE For-Sale Anodyne PREP 22 44 O=C(O)c1cccc(CNC(=O)C2[C@H]3CCCC[C@@H]23)c1 ZINC000147349825 CE For-Sale Anodyne TMPRSS11D 52 33 COc1cc2nc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)sc2cc1OC ZINC000147349864 FH On-Demand Bother LCK 22 40 COc1cc2nc(NC(=O)c3cc(C)cc([N+](=O)[O-])c3)sc2cc1OC ZINC000147349864 FH On-Demand Bother CSNK1D 24 41 CCOc1c(Br)cc(CNCCCCC(C)C)cc1OC ZINC000147349880 FJ For-Sale Anodyne LPAR2 51 55 CCOc1c(Br)cc(CNCCCCC(C)C)cc1OC ZINC000147349880 FJ For-Sale Anodyne S1PR2 50 55 CCOc1c(Br)cc(CNCCCCC(C)C)cc1OC ZINC000147349880 FJ For-Sale Anodyne LEF 41 33 CC(C)[C@@H](NC(=O)OC(C)(C)C)C(=O)N1CC=C[C@@H](OS(C)(=O)=O)C1 ZINC000147349884 GD For-Sale Mild PGA5 40 35 CCc1nn(-c2ccccc2)c2cc(N3CCN(C4CCNCC4)C3=O)ccc12 ZINC000147349905 GH Annotated Anodyne KHK 0 67 CCCCCCCCNC(=O)c1cc(C)ccc1NC ZINC000147350011 CI For-Sale Mild S1PR2 46 35 CCCCCCCCNC(=O)c1cc(C)ccc1NC ZINC000147350011 CI For-Sale Mild PA2A1_NAJMO 0 42 CCCCCCCCNC(=O)c1cc(C)ccc1NC ZINC000147350011 CI For-Sale Mild ASAH1 88 37 CCCCCCCCNC(=O)c1cc(C)ccc1NC ZINC000147350011 CI For-Sale Mild PSBA 0 40 O=C(O)c1cccc(CNC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147350022 CE On-Demand Anodyne F2 20 42 O=C(O)c1cccc(CNC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147350022 CE On-Demand Anodyne P2RX7 16 40 O=C(O)c1cccc(CNC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147350022 CE On-Demand Anodyne PREP 22 44 O=C(O)c1cccc(CNC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147350022 CE On-Demand Anodyne TMPRSS11D 52 33 O=C(NCc1ccccn1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147350065 FF For-Sale Anodyne NAMPT 22 41 COCc1nc(C(=O)Nc2nc3cc(OC)c(OC)cc3s2)cs1 ZINC000147350071 FG On-Demand Anodyne CSNK1D 36 42 CCCCCCNCCCCC(C)C ZINC000147350089 AH For-Sale Anodyne ADH1A 0 47 CCCCCCNCCCCC(C)C ZINC000147350089 AH For-Sale Anodyne ADH7 0 44 CCCCCCNCCCCC(C)C ZINC000147350089 AH For-Sale Anodyne S1PR3 21 50 CCCCCCNCCCCC(C)C ZINC000147350089 AH For-Sale Anodyne S1PR2 47 50 CCCCCCNCCCCC(C)C ZINC000147350089 AH For-Sale Anodyne ADH1B 0 47 CCCCCCNCCCCC(C)C ZINC000147350089 AH For-Sale Anodyne ADH1C 0 47 CCCCCCNCCCCC(C)C ZINC000147350089 AH For-Sale Anodyne Q6UB75_PIG 47 39 CCCCCCNCCCCC(C)C ZINC000147350089 AH For-Sale Anodyne Q8WS26_TRYCR 41 42 CCCCCCNCCCCC(C)C ZINC000147350089 AH For-Sale Anodyne FPPS 0 42 CCCCCCNCCCCC(C)C ZINC000147350089 AH For-Sale Anodyne SPPS 0 42 CCc1nn(-c2ccccc2)c2cc(N3CC[C@@]4(CCNC4)C3)ccc12 ZINC000147350163 EH Annotated Anodyne KHK 0 67 Cc1ncoc1C(=O)NCc1cccc(C(=O)O)c1 ZINC000147350271 CD On-Demand Anodyne MMP13 24 45 Cc1ncoc1C(=O)NCc1cccc(C(=O)O)c1 ZINC000147350271 CD On-Demand Anodyne KDM4E 31 41 CCc1ccc(NC(=O)C2(C(=O)Nc3ccc(F)cc3)CC2)cc1F ZINC000147350298 EH On-Demand Anodyne MET 28 49 CCc1ccc(NC(=O)C2(C(=O)Nc3ccc(F)cc3)CC2)cc1F ZINC000147350298 EH On-Demand Anodyne ENV 43 34 CCc1ccc(NC(=O)C2(C(=O)Nc3ccc(F)cc3)CC2)cc1F ZINC000147350298 EH On-Demand Anodyne AXL 39 40 O=C(NCc1ccccn1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147350304 DF On-Demand Anodyne PPIA 40 40 O=C(NCc1ccccn1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147350304 DF On-Demand Anodyne GRM4 44 40 O=C(NCc1ccccn1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147350304 DF On-Demand Anodyne EPHX2 15 42 O=C(NCc1ccccn1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147350304 DF On-Demand Anodyne NAMPT 20 41 FC(F)(F)COc1ccc(CCBr)cc1 ZINC000147350372 CH For-Sale Reactive TAAR1 17 44 CCc1nn(-c2ccccc2)c2cc(N3CC[C@]4(CCNC4)C3)ccc12 ZINC000147350373 EH Annotated Anodyne KHK 0 67 CCOc1ccc([C@@H](C)NCC(F)F)cc1 ZINC000147350417 BG On-Demand Anodyne ACACA 35 47 CCOc1ccc([C@@H](C)NCC(F)F)cc1 ZINC000147350417 BG On-Demand Anodyne ACACB 19 47 CCCNc1cccc(NCc2cccc(F)c2)n1 ZINC000147350458 CH For-Sale Anodyne NAMPT 0 40 CCCCCCCCNC(=O)c1ccccc1NN ZINC000147350484 CG For-Sale Mild CNR1 15 42 CCCCCCCCNC(=O)c1ccccc1NN ZINC000147350484 CG For-Sale Mild DRD3 17 40 CCCCCCCCNC(=O)c1ccccc1NN ZINC000147350484 CG For-Sale Mild CDC25B 15 41 CCCCCCCCNC(=O)c1ccccc1NN ZINC000147350484 CG For-Sale Mild GRIA1 40 33 CCCCCCCCNC(=O)c1ccccc1NN ZINC000147350484 CG For-Sale Mild FAAH 15 42 CCCCCCCCNC(=O)c1ccccc1NN ZINC000147350484 CG For-Sale Mild S1PR2 43 38 CCCCCCCCNC(=O)c1ccccc1NN ZINC000147350484 CG For-Sale Mild EPHX2 28 40 CCCCCCCCNC(=O)c1ccccc1NN ZINC000147350484 CG For-Sale Mild ASAH1 105 42 CCCCCCCCNC(=O)c1ccccc1NN ZINC000147350484 CG For-Sale Mild POLR1A 53 35 CC[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147350501 CE On-Demand Anodyne CCKAR 44 40 CC[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147350501 CE On-Demand Anodyne CCKBR 0 41 CC[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147350501 CE On-Demand Anodyne ACE2 58 33 CC[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147350501 CE On-Demand Anodyne DAC 40 38 CC(C)(C)OC(=O)N[C@@H]1CCCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)C1 ZINC000147350557 GH On-Demand Anodyne MDM2 71 33 CC(C)(C)OC(=O)N[C@@H]1CCCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)C1 ZINC000147350557 GH On-Demand Anodyne NPBWR1 43 32 O=C(O)C1(NCc2cc(Cl)ccc2OC(F)F)CCC1 ZINC000147350560 DG For-Sale Anodyne PDEC 0 40 CCNC(=O)Nc1cc2cccc(CNC(=O)c3ccncc3)c2cn1 ZINC000147350601 EF For-Sale Anodyne TRPV1 28 42 CCNC(=O)Nc1cc2cccc(CNC(=O)c3ccncc3)c2cn1 ZINC000147350601 EF For-Sale Anodyne ROCK2 19 40 CCc1nn(-c2ccccc2)c2cc(-c3ccc([C@@H]4CCNC4)cc3)ccc12 ZINC000147350618 FK Annotated Anodyne KHK 0 64 O=C(NN1CCCCC1)c1cccc2c1CCCN2 ZINC000147350623 CE For-Sale Anodyne CNR1 54 33 CCOc1ccc([C@H](C)NCC(F)F)cc1 ZINC000147350630 BG On-Demand Anodyne ACACA 35 47 CCOc1ccc([C@H](C)NCC(F)F)cc1 ZINC000147350630 BG On-Demand Anodyne ACACB 19 47 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(c2oc(-c3ccco3)nc2C#N)CC1 ZINC000147350650 HD On-Demand Mild P2RY12 174 36 CS(=O)(=O)c1ccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cn1 ZINC000147350666 HD On-Demand Anodyne ROCK2 20 40 CS(=O)(=O)c1ccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cn1 ZINC000147350666 HD On-Demand Anodyne NAMPT 49 38 CC[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147350685 CE On-Demand Anodyne CCKAR 44 40 CC[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147350685 CE On-Demand Anodyne CCKBR 0 41 CC[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147350685 CE On-Demand Anodyne ACE2 58 33 CC[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147350685 CE On-Demand Anodyne DAC 40 38 CCCCCCCCNC(=O)c1ccnc(NN)c1 ZINC000147350692 CE For-Sale Mild ASAH1 85 36 CCCCCCCCNC(=O)c1ccnc(NN)c1 ZINC000147350692 CE For-Sale Mild KDM4E 25 45 O=C1NC(=O)/C(=C\c2ccc3ccccc3c2)N1 ZINC000147350704 BE For-Sale Anodyne GSK3B 15 65 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne LPL 33 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne LCK 28 49 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne P2RY1 15 45 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne PIK3CA 19 43 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne PRNP 56 47 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne KDR 18 49 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne MTOR 40 44 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne HCK 23 45 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne PIK3CG 16 40 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne FLT3 23 47 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne CSF1R 20 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne AURKA 18 46 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cnc(-c2ccccc2)nc1 ZINC000147350791 HH On-Demand Anodyne MAPK7 29 42 CCc1nn(-c2ccccc2)c2cc(-c3ccc([C@H]4CCNC4)cc3)ccc12 ZINC000147350826 FK Annotated Anodyne KHK 0 64 CC(C)(C)c1cc(O)ccc1OC(=O)c1ccccc1 ZINC000147350842 CH For-Sale Anodyne ELANE 15 40 CS(=O)(=O)c1ccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cn1 ZINC000147350859 HD On-Demand Anodyne ROCK2 20 40 CS(=O)(=O)c1ccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cn1 ZINC000147350859 HD On-Demand Anodyne NAMPT 49 38 CC[C@@H](NC(=O)c1ccc(Br)cc1OC)C(=O)O ZINC000147350913 DE On-Demand Anodyne FOLH1 29 42 CC[C@@H](NC(=O)c1ccc(Br)cc1OC)C(=O)O ZINC000147350913 DE On-Demand Anodyne ACE2 41 32 CC(C)(C)OC(=O)N[C@@H]1CCCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)C1 ZINC000147350961 GH On-Demand Anodyne MDM2 71 33 CC(C)(C)OC(=O)N[C@@H]1CCCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)C1 ZINC000147350961 GH On-Demand Anodyne NPBWR1 43 32 COc1ccc(Cl)cc1C(=O)N[C@@H](C)Cc1ccc(O)cc1 ZINC000147350976 DG On-Demand Anodyne AVPR1A 22 40 COc1ccc(Cl)cc1C(=O)N[C@@H](C)Cc1ccc(O)cc1 ZINC000147350976 DG On-Demand Anodyne GRIA1 42 33 COc1ccc(Cl)cc1C(=O)N[C@@H](C)Cc1ccc(O)cc1 ZINC000147350976 DG On-Demand Anodyne KCNMA1 29 48 COc1ccc(Cl)cc1C(=O)N[C@@H](C)Cc1ccc(O)cc1 ZINC000147350976 DG On-Demand Anodyne CPT1B 44 38 COc1ccc(Cl)cc1C(=O)N[C@@H](C)Cc1ccc(O)cc1 ZINC000147350976 DG On-Demand Anodyne U38 0 45 COc1ccc(Cl)cc1C(=O)N[C@@H](C)Cc1ccc(O)cc1 ZINC000147350976 DG On-Demand Anodyne ACPS 0 41 COc1ccc(Cl)cc1C(=O)N[C@@H](C)Cc1ccc(O)cc1 ZINC000147350976 DG On-Demand Anodyne PSBA 0 40 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1nc(C)c(C)s1 ZINC000147351009 FG On-Demand Anodyne SLC27A1 22 50 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(S(C)(=O)=O)nc3)c2)CCO1 ZINC000147351056 HE On-Demand Anodyne CCR3 22 40 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(S(C)(=O)=O)nc3)c2)CCO1 ZINC000147351056 HE On-Demand Anodyne NAMPT 45 42 Cc1nn(-c2ccccc2)c2cc(N3CC[C@H](N4CCNCC4)C3)ccc12 ZINC000147351072 FF Annotated Anodyne KHK 0 88 CCCCCCCCNC(=O)c1cccc(NN)n1 ZINC000147351080 CE For-Sale Mild EPHX2 22 40 CCCCCCCCNC(=O)c1cccc(NN)n1 ZINC000147351080 CE For-Sale Mild ASAH1 90 36 CC[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351154 BD For-Sale Anodyne ACE 33 42 CC[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351154 BD For-Sale Anodyne MME 36 42 CC[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351154 BD For-Sale Anodyne ACE2 68 37 CC[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351154 BD For-Sale Anodyne GPR88 0 51 Cc1cc(C(=O)N2CCC[C@H](CCBr)C2)ccc1[N+](=O)[O-] ZINC000147351167 FH For-Sale Reactive L3MBTL1 0 41 CCOCCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147351185 DF On-Demand Anodyne CACNA1I 40 33 COc1ccc(Cl)cc1C(=O)N[C@H](C)Cc1ccc(O)cc1 ZINC000147351199 DG On-Demand Anodyne AVPR1A 22 40 COc1ccc(Cl)cc1C(=O)N[C@H](C)Cc1ccc(O)cc1 ZINC000147351199 DG On-Demand Anodyne GRIA1 42 33 COc1ccc(Cl)cc1C(=O)N[C@H](C)Cc1ccc(O)cc1 ZINC000147351199 DG On-Demand Anodyne KCNMA1 29 48 COc1ccc(Cl)cc1C(=O)N[C@H](C)Cc1ccc(O)cc1 ZINC000147351199 DG On-Demand Anodyne CPT1B 44 38 COc1ccc(Cl)cc1C(=O)N[C@H](C)Cc1ccc(O)cc1 ZINC000147351199 DG On-Demand Anodyne U38 0 45 COc1ccc(Cl)cc1C(=O)N[C@H](C)Cc1ccc(O)cc1 ZINC000147351199 DG On-Demand Anodyne ACPS 0 41 COc1ccc(Cl)cc1C(=O)N[C@H](C)Cc1ccc(O)cc1 ZINC000147351199 DG On-Demand Anodyne PSBA 0 40 C[C@H](NC(=O)OCCCl)C(=O)O ZINC000147351247 AC For-Sale Reactive SLC15A1 44 36 C[C@H](NC(=O)OCCCl)C(=O)O ZINC000147351247 AC For-Sale Reactive SLC15A2 0 47 Cc1nn(-c2ccccc2)c2cc(N3CC[C@@H](N4CCNCC4)C3)ccc12 ZINC000147351270 FF Annotated Anodyne KHK 0 88 Cc1cc(C(=O)NCc2ccc(OC(F)F)cc2)cc([N+](=O)[O-])c1 ZINC000147351292 EG On-Demand Bother U38 0 44 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(S(C)(=O)=O)nc3)c2)CCO1 ZINC000147351293 HE On-Demand Anodyne CCR3 22 40 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc(S(C)(=O)=O)nc3)c2)CCO1 ZINC000147351293 HE On-Demand Anodyne NAMPT 45 42 CCCCCCCCNC(=O)c1cc(Br)cnc1NN ZINC000147351315 EG For-Sale Mild ASAH1 68 34 CCCCCCCCCC[C@@H](C)C(C)C ZINC000147351329 BK For-Sale Mild CQSS 55 41 COC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147351330 DH On-Demand Anodyne PPIA 15 42 COC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147351330 DH On-Demand Anodyne F10 26 44 COC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147351330 DH On-Demand Anodyne ECR 42 33 COC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147351330 DH On-Demand Anodyne NR1H4 22 40 COC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147351330 DH On-Demand Anodyne FABH 0 42 COC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147351330 DH On-Demand Anodyne PAGA 0 42 COC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147351330 DH On-Demand Anodyne KCNK3 83 42 COC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147351330 DH On-Demand Anodyne KCNK9 64 42 COC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147351330 DH On-Demand Anodyne FAS 15 43 Cc1nn(Cc2ccccc2)c(C)c1CNC(=O)N(C)Cc1cscn1 ZINC000147351331 FG On-Demand Anodyne P2RX7 15 43 CC[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351341 BD For-Sale Anodyne ACE 33 42 CC[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351341 BD For-Sale Anodyne MME 36 42 CC[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351341 BD For-Sale Anodyne ACE2 68 37 CC[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351341 BD For-Sale Anodyne GPR88 0 51 Cc1cc(C(=O)N2CCC[C@@H](CCBr)C2)ccc1[N+](=O)[O-] ZINC000147351365 FH For-Sale Reactive L3MBTL1 0 41 CN(C(=O)Oc1ccnc2ccccc12)c1ccccc1 ZINC000147351395 CH For-Sale Anodyne LIPE 16 43 CCNC(=O)N[C@@H]1C[C@H]1c1cccc(OC)c1 ZINC000147351405 BD On-Demand Anodyne DRD4 42 32 CCNC(=O)N[C@@H]1C[C@H]1c1cccc(OC)c1 ZINC000147351405 BD On-Demand Anodyne MTNR1A 49 43 CCNC(=O)N[C@@H]1C[C@H]1c1cccc(OC)c1 ZINC000147351405 BD On-Demand Anodyne MTNR1B 47 42 CCNC(=O)N[C@@H]1C[C@H]1c1cccc(OC)c1 ZINC000147351405 BD On-Demand Anodyne EPHX2 15 49 CCNC(=O)N[C@@H]1C[C@H]1c1cccc(OC)c1 ZINC000147351405 BD On-Demand Anodyne KDM1A 17 42 CC[C@H](NC(=O)[C@H]1Oc2ccccc2O[C@@H]1C)C(=O)O ZINC000147351470 CD On-Demand Anodyne MME 29 40 CC[C@H](NC(=O)[C@H]1Oc2ccccc2O[C@@H]1C)C(=O)O ZINC000147351470 CD On-Demand Anodyne ACE2 65 35 CCCCCCCCNC(=O)c1cccc(F)c1NN ZINC000147351481 CG For-Sale Mild EPHX2 0 40 CCCCCCCCNC(=O)c1cccc(F)c1NN ZINC000147351481 CG For-Sale Mild ASAH1 102 39 COCCC[C@H](N)C(=O)NN1CCCCC1 ZINC000147351508 BC For-Sale Anodyne DPP7 40 35 Cc1nn(-c2ccccc2)c2cc(-c3ccc(N4CCNCC4)cc3)ccc12 ZINC000147351519 FI Annotated Anodyne BMPR1A 0 43 Cc1nn(-c2ccccc2)c2cc(-c3ccc(N4CCNCC4)cc3)ccc12 ZINC000147351519 FI Annotated Anodyne ACVRL1 0 43 Cc1nn(-c2ccccc2)c2cc(-c3ccc(N4CCNCC4)cc3)ccc12 ZINC000147351519 FI Annotated Anodyne ACVR1 60 43 Cc1nn(-c2ccccc2)c2cc(-c3ccc(N4CCNCC4)cc3)ccc12 ZINC000147351519 FI Annotated Anodyne KHK 0 82 CCCCCCCCCC[C@H](C)C(C)C ZINC000147351540 BK For-Sale Mild CQSS 55 41 CC[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351544 BD For-Sale Anodyne ACE 33 42 CC[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351544 BD For-Sale Anodyne MME 36 42 CC[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351544 BD For-Sale Anodyne ACE2 68 37 CC[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351544 BD For-Sale Anodyne GPR88 0 51 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne LCK 30 43 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne MAPK14 23 45 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne PIK3CA 38 51 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne JAK2 18 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne MAPKAPK5 49 35 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne MTOR 74 51 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne HCK 17 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne PIK3CG 36 44 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne FLT3 19 43 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne CSF1R 19 44 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne AURKA 19 43 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne STAT6 63 33 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147351667 HF On-Demand Anodyne DGAT1 50 46 CC(C)[C@H](NC(=O)c1csc(-c2cscn2)n1)C(=O)NCCC(=O)NO ZINC000147351683 GD Annotated Mild HDAC3 0 63 CCCCCCCCNC(=O)c1cc(F)c(NN)c(F)c1 ZINC000147351690 CG For-Sale Mild ASAH1 100 40 CNCc1cnc(Oc2ccc(Cl)c(F)c2)c(Cl)c1 ZINC000147351695 DI For-Sale Anodyne SLC6A4 15 57 COCCC[C@@H](N)C(=O)NN1CCCCC1 ZINC000147351707 BC For-Sale Anodyne DPP7 40 35 CC[C@H](NC(=O)[C@@H]1Oc2ccccc2O[C@@H]1C)C(=O)O ZINC000147351709 CD On-Demand Anodyne MME 29 40 CC[C@H](NC(=O)[C@@H]1Oc2ccccc2O[C@@H]1C)C(=O)O ZINC000147351709 CD On-Demand Anodyne ACE2 65 35 Cc1nn(-c2ccccc2)c2cc(N3CCN(C4CNC4)CC3)ccc12 ZINC000147351731 EE Annotated Anodyne KHK 0 76 CC[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351732 BD For-Sale Anodyne ACE 33 42 CC[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351732 BD For-Sale Anodyne MME 36 42 CC[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351732 BD For-Sale Anodyne ACE2 68 37 CC[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147351732 BD For-Sale Anodyne GPR88 0 51 CC(C)Oc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147351735 FI For-Sale Reactive GRM3 16 52 CC(C)Oc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147351735 FI For-Sale Reactive L3MBTL3 48 37 Nc1nc(Oc2cccnc2)nc(N2CCOCC2)n1 ZINC000147351754 CC For-Sale Anodyne PIK3CA 39 55 Nc1nc(Oc2cccnc2)nc(N2CCOCC2)n1 ZINC000147351754 CC For-Sale Anodyne MTOR 21 43 Nc1nc(Oc2cccnc2)nc(N2CCOCC2)n1 ZINC000147351754 CC For-Sale Anodyne PIK3CG 21 43 CCOc1c(Br)cc(CNCCCCC(C)C)cc1Br ZINC000147351812 HK For-Sale Anodyne LPAR2 55 50 CCOc1c(Br)cc(CNCCCCC(C)C)cc1Br ZINC000147351812 HK For-Sale Anodyne S1PR2 55 50 CCOc1c(Br)cc(CNCCCCC(C)C)cc1Br ZINC000147351812 HK For-Sale Anodyne LEF 65 33 O=C(NC[C@@H]1CCCO1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147351823 CE On-Demand Anodyne CACNA1I 63 37 CCCCCCCCNC(=O)c1cnccc1NN ZINC000147351895 CE For-Sale Mild ASAH1 87 36 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCCC2)nc1 ZINC000147351905 GG On-Demand Anodyne LCK 27 42 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCCC2)nc1 ZINC000147351905 GG On-Demand Anodyne HCK 16 42 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCCC2)nc1 ZINC000147351905 GG On-Demand Anodyne FLT3 17 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCCC2)nc1 ZINC000147351905 GG On-Demand Anodyne CSF1R 22 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(N2CCCC2)nc1 ZINC000147351905 GG On-Demand Anodyne DGAT1 37 43 CC[C@H](NC(=O)c1ccc(C)c(Br)c1)C(=O)O ZINC000147351925 DE On-Demand Anodyne CA2 28 43 CC(C)Oc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147351939 FI For-Sale Reactive GRM3 16 52 CC(C)Oc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147351939 FI For-Sale Reactive L3MBTL3 48 37 CC[C@@H]1CN(C(=O)Nc2ccccc2OC)CC[C@@H]1N ZINC000147351977 CE On-Demand Anodyne SMO 22 46 Cc1nn(-c2ccccc2)c2cc(N3CC(N4CCNCC4)C3)ccc12 ZINC000147351979 EE Annotated Anodyne KHK 0 82 COc1ccc2[nH]cc(C3=CCN(C[C@@H](O)COc4cccc5[nH]ccc45)CC3)c2c1 ZINC000147352012 HI On-Demand Anodyne ADRB1 17 42 COc1ccc2[nH]cc(C3=CCN(C[C@@H](O)COc4cccc5[nH]ccc45)CC3)c2c1 ZINC000147352012 HI On-Demand Anodyne HTR1A 28 56 COc1ccc2[nH]cc(C3=CCN(C[C@@H](O)COc4cccc5[nH]ccc45)CC3)c2c1 ZINC000147352012 HI On-Demand Anodyne SLC6A4 33 44 O=C(NC[C@H]1CCCO1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147352041 CE On-Demand Anodyne CACNA1I 63 37 O=C(NC1CCCC1)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1 ZINC000147352078 GH On-Demand Anodyne MAPK14 35 41 O=C(NC1CCCC1)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1 ZINC000147352078 GH On-Demand Anodyne MAPK13 68 32 COc1ccc(CCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352117 EI On-Demand Anodyne SLC6A1 21 41 COc1ccc(CCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352117 EI On-Demand Anodyne SCNN1A 78 43 COc1ccc(CCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352117 EI On-Demand Anodyne MTNR1A 62 43 COc1ccc(CCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352117 EI On-Demand Anodyne MTNR1B 54 43 COc1ccc(CCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352117 EI On-Demand Anodyne SLC6A5 18 41 COc1ccc(CCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352117 EI On-Demand Anodyne MCHR1 15 46 COc1ccc(CCCNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352117 EI On-Demand Anodyne CRTM 40 36 CC[C@@H](NC(=O)c1ccc(C)c(Br)c1)C(=O)O ZINC000147352118 DE On-Demand Anodyne CA2 28 43 CCCCCCCCNC(=O)c1cnc(NN)c(Cl)c1 ZINC000147352138 CG For-Sale Mild ASAH1 86 38 Cc1nc(-c2nc(C(=O)N[C@H](C(=O)NCCCC(=O)NO)C(C)C)cs2)cs1 ZINC000147352160 ID Annotated Mild HDAC3 31 71 CC[C@H]1CN(C(=O)Nc2ccccc2OC)CC[C@@H]1N ZINC000147352175 CE On-Demand Anodyne SMO 22 46 Cc1nn(-c2ccccc2)c2cc(N3CCN([C@@H]4CCNC4)CC3)ccc12 ZINC000147352210 FF Annotated Anodyne KHK 0 78 Cc1cccc(C)c1OC[C@H](O)CNC(=O)Nc1ccc(S(C)(=O)=O)nc1 ZINC000147352220 GD On-Demand Anodyne ADRB1 59 39 COc1ccc(CCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352313 EI On-Demand Anodyne SLC6A1 21 41 COc1ccc(CCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352313 EI On-Demand Anodyne SCNN1A 78 43 COc1ccc(CCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352313 EI On-Demand Anodyne MTNR1A 62 43 COc1ccc(CCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352313 EI On-Demand Anodyne MTNR1B 54 43 COc1ccc(CCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352313 EI On-Demand Anodyne SLC6A5 18 41 COc1ccc(CCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352313 EI On-Demand Anodyne MCHR1 15 46 COc1ccc(CCCNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1 ZINC000147352313 EI On-Demand Anodyne CRTM 40 36 Cc1nn(C(F)F)c(C)c1CC(=O)N1CCN(C(=O)Nc2ccc(F)cc2)CC1 ZINC000147352317 HF On-Demand Anodyne P2RX7 28 40 CCCCCCCCNC(=O)c1cnc(C)cc1NN ZINC000147352351 CF For-Sale Mild MERTK 17 40 CCCCCCCCNC(=O)c1cnc(C)cc1NN ZINC000147352351 CF For-Sale Mild ASAH1 79 33 CC[C@@H]1CN(C(=O)Nc2ccccc2OC)CC[C@H]1N ZINC000147352352 CE On-Demand Anodyne SMO 22 46 Nc1cccc(/C=C/C(=O)NN2CCCCC2)c1 ZINC000147352383 BD For-Sale Anodyne HDAC8 55 41 Nc1cccc(/C=C/C(=O)NN2CCCCC2)c1 ZINC000147352383 BD For-Sale Anodyne HDAC1 25 41 Nc1cccc(/C=C/C(=O)NN2CCCCC2)c1 ZINC000147352383 BD For-Sale Anodyne HDAC6 35 41 Cc1cccc(C)c1OC[C@@H](O)CNC(=O)Nc1ccc(S(C)(=O)=O)nc1 ZINC000147352424 GD On-Demand Anodyne ADRB1 59 39 Cc1nn(-c2ccccc2)c2cc(N3CCN([C@H]4CCNC4)CC3)ccc12 ZINC000147352443 FF Annotated Anodyne KHK 0 78 CC(C)CCO[C@@H](C)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147352461 EF On-Demand Anodyne CASR 49 36 CCN1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147352472 DE For-Sale Anodyne CACNA1H 49 39 CCN1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147352472 DE For-Sale Anodyne CACNA1I 50 35 CC(C)c1nc(NN)cc(OC[C@@H]2CCCCN2C)n1 ZINC000147352479 CD For-Sale Anodyne CHRNA10 71 40 CC(C)CCCCNCc1ccc(SC(F)(F)F)cc1 ZINC000147352486 DK For-Sale Anodyne LEF 74 37 COc1ccc(CCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147352521 EI On-Demand Anodyne SCNN1A 78 43 COc1ccc(CCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147352521 EI On-Demand Anodyne MTNR1A 62 43 COc1ccc(CCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147352521 EI On-Demand Anodyne MTNR1B 54 43 COc1ccc(CCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147352521 EI On-Demand Anodyne SLC6A5 18 41 COc1ccc(CCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147352521 EI On-Demand Anodyne MCHR1 15 46 COc1ccc(CCCNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)cc1 ZINC000147352521 EI On-Demand Anodyne CRTM 40 36 CC[C@H]1CN(C(=O)Nc2ccccc2OC)CC[C@H]1N ZINC000147352550 CE On-Demand Anodyne SMO 22 46 CCCCCCCCNC(=O)c1ccc(NN)nn1 ZINC000147352556 CD For-Sale Mild ASAH1 91 37 COCc1nc(C(=O)N(C)Cc2ccc(OCc3ccccc3)c(OC)c2)cs1 ZINC000147352564 HI On-Demand Anodyne DRTS_PLAFK 27 45 COCc1nc(C(=O)N(C)Cc2ccc(OCc3ccccc3)c(OC)c2)cs1 ZINC000147352564 HI On-Demand Anodyne PTGER1 42 46 COCc1nc(C(=O)N(C)Cc2ccc(OCc3ccccc3)c(OC)c2)cs1 ZINC000147352564 HI On-Demand Anodyne PTGER4 24 44 CCCOc1ccc(Cl)cc1NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147352565 HH On-Demand Bother PTGDR2 25 40 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne TBXA2R 22 41 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne BMP1 67 37 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne KCNA5 0 47 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne MMP13 62 42 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne ADAM17 31 40 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne MMP16 0 42 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne MMP2 45 46 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne MMP3 55 43 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne MMP8 35 45 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne MMP14 26 52 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne MMP9 54 52 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne MMP12 32 45 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne MMP7 51 55 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne ADAMTS4 41 38 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne MMP1 59 45 CC[C@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352594 DD On-Demand Anodyne Q9JN24_ECOLX 0 42 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cccc(C(=O)N(C)C)c1 ZINC000147352611 GG On-Demand Anodyne LCK 21 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1cccc(C(=O)N(C)C)c1 ZINC000147352611 GG On-Demand Anodyne FLT3 17 43 N[C@H](C(=O)NN1CCCCC1)c1cccs1 ZINC000147352617 BD For-Sale Anodyne DPP7 23 42 CC(C)CCO[C@H](C)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147352655 EF On-Demand Anodyne CASR 49 36 Cc1[nH]c2cc([C@@H]3CCCCN3C(=O)c3ccccc3N)nn2c(=O)c1C ZINC000147352663 FF Annotated Anodyne COLA 44 33 Cc1[nH]c2cc([C@@H]3CCCCN3C(=O)c3ccccc3N)nn2c(=O)c1C ZINC000147352663 FF Annotated Anodyne CPT1A 43 33 CCN(C)c1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNC(C)(C)c2cccc(OC)c2)cc(N2CCCC2=O)c1 ZINC000147352677 KJ Annotated Anodyne CTSD 66 65 CCN(C)c1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNC(C)(C)c2cccc(OC)c2)cc(N2CCCC2=O)c1 ZINC000147352677 KJ Annotated Anodyne BACE2 69 65 CCN(C)c1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNC(C)(C)c2cccc(OC)c2)cc(N2CCCC2=O)c1 ZINC000147352677 KJ Annotated Anodyne BACE1 85 65 CCN(C)c1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNC(C)(C)c2cccc(OC)c2)cc(N2CCCC2=O)c1 ZINC000147352677 KJ Annotated Anodyne PLM1_PLAFA 70 64 CCN(C)c1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNC(C)(C)c2cccc(OC)c2)cc(N2CCCC2=O)c1 ZINC000147352677 KJ Annotated Anodyne PLM2_PLAFA 39 64 Cc1nn(-c2ccccc2)c2cc(N3CCN(C4CCNCC4)CC3)ccc12 ZINC000147352681 GG Annotated Anodyne KHK 0 84 CC(C)c1nc(NN)cc(OC[C@H]2CCCCN2C)n1 ZINC000147352719 CD For-Sale Anodyne CHRNA10 71 40 CCCCCCCCNC(=O)c1cc(Cl)ccc1NN ZINC000147352735 CH For-Sale Mild CNR1 18 54 CCCCCCCCNC(=O)c1cc(Cl)ccc1NN ZINC000147352735 CH For-Sale Mild EPHX2 0 47 CCCCCCCCNC(=O)c1cc(Cl)ccc1NN ZINC000147352735 CH For-Sale Mild ALPL 44 40 CCCCCCCCNC(=O)c1cc(Cl)ccc1NN ZINC000147352735 CH For-Sale Mild ASAH1 93 38 COc1ccc(CCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147352776 FG On-Demand Anodyne SCNN1A 49 41 COc1ccc(CCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147352776 FG On-Demand Anodyne NQO2 36 42 COc1ccc(CCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147352776 FG On-Demand Anodyne MTNR1A 103 45 COc1ccc(CCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147352776 FG On-Demand Anodyne MTNR1B 92 42 COc1ccc(CCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147352776 FG On-Demand Anodyne ROCK2 27 43 CC[C@@H]1CN(C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147352785 BE On-Demand Anodyne NPY2R 36 41 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne TBXA2R 22 41 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne BMP1 67 37 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne KCNA5 0 47 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne MMP13 62 42 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne ADAM17 31 40 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne MMP16 0 42 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne MMP2 45 46 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne MMP3 55 43 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne MMP8 35 45 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne MMP14 26 52 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne MMP9 54 52 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne MMP12 32 45 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne MMP7 51 55 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne ADAMTS4 41 38 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne MMP1 59 45 CC[C@@H](CNS(=O)(=O)c1ccc(OC)cc1)CC(=O)O ZINC000147352789 DD On-Demand Anodyne Q9JN24_ECOLX 0 42 N[C@@H](C(=O)NN1CCCCC1)c1cccs1 ZINC000147352837 BD For-Sale Anodyne DPP7 23 42 CS(=O)(=O)c1ccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)cn1 ZINC000147352839 EE On-Demand Anodyne EPHX2 25 41 CC(C)CCO[C@@H](C)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147352844 EF On-Demand Anodyne CASR 49 36 Cc1[nH]c2cc([C@@H]3CCCCN3C(=O)c3ccccc3)nn2c(=O)c1C ZINC000147352879 FG Annotated Anodyne COLA 95 37 Cc1[nH]c2cc([C@@H]3CCCCN3C(=O)c3ccccc3)nn2c(=O)c1C ZINC000147352879 FG Annotated Anodyne CPT1A 92 37 O=C(O)c1cc(Cl)cc(NC(=O)N2CCCCCCC2)c1 ZINC000147352915 DH On-Demand Anodyne EPHX2 15 46 O=C(O)c1cc(Cl)cc(NC(=O)N2CCCCCCC2)c1 ZINC000147352915 DH On-Demand Anodyne HCAR1 0 42 CCCCCCCCNC(=O)c1cc(C)ccc1NN ZINC000147352942 CG For-Sale Mild ASAH1 91 37 CC(=O)Nc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1Cl ZINC000147352956 FD On-Demand Anodyne ENV 42 35 CN1CCCC[C@@H]1COc1cc(NN)nc(C2CC2)n1 ZINC000147352999 CD For-Sale Anodyne CHRNA10 73 42 CC[C@H]1CN(C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147353002 BE On-Demand Anodyne NPY2R 36 41 Nc1c(F)cccc1C(=O)NN1CCCCC1 ZINC000147353022 BD For-Sale Anodyne CNR1 50 31 CC[C@H](CNS(=O)(=O)c1cccc(Cl)c1)CC(=O)O ZINC000147353034 DE On-Demand Anodyne TBXA2R 42 34 CC[C@H](CNS(=O)(=O)c1cccc(Cl)c1)CC(=O)O ZINC000147353034 DE On-Demand Anodyne FBP1 32 42 CC(C)CCO[C@H](C)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147353050 EF On-Demand Anodyne CASR 49 36 CS(=O)(=O)c1ccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)cn1 ZINC000147353055 EE On-Demand Anodyne EPHX2 25 41 O=C(O)C1(NCCS(=O)(=O)c2ccc(Br)cc2)CCC1 ZINC000147353082 FD For-Sale Anodyne LIG1 0 40 CC(C)CCCCN[C@@H]1CCCC[C@@H]1c1ccccc1 ZINC000147353090 CK For-Sale Anodyne GRIA4 19 48 Ic1cccc(-c2cnn(CCCc3ccccc3)c2)c1 ZINC000147353109 GJ For-Sale Anodyne SIGMAR1 16 50 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne DRD2 23 53 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne DRD4 22 46 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne ACHE 23 40 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne HTR4 66 47 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne GRIN2B 52 39 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne LTA4H 58 46 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne HRH3 28 41 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne SIGMAR1 60 64 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne NPY1R 41 38 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne CCR3 44 37 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne COLA 50 39 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne CPT1A 47 39 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne CHRNA10 62 45 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne GRIN3A 0 47 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne CYP2J2 48 34 O=C(O)CCN1CCC(COc2ccccc2)CC1 ZINC000147353123 CE In-Stock Anodyne MEN1 48 37 CCCCCCCCNC(=O)c1ccc(C)cc1NN ZINC000147353154 CG For-Sale Mild EPHX2 0 40 CCCCCCCCNC(=O)c1ccc(C)cc1NN ZINC000147353154 CG For-Sale Mild ASAH1 94 38 CC(=O)Nc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1Cl ZINC000147353189 FD On-Demand Anodyne ENV 42 35 CC[C@@H]1CN(C(=O)Nc2ccccc2)CC[C@H]1N ZINC000147353196 BE On-Demand Anodyne NPY2R 36 41 CNCc1cnccc1Oc1ccc(Cl)c(F)c1 ZINC000147353202 CG For-Sale Anodyne SLC6A4 26 62 CN1CCCC[C@H]1COc1cc(NN)nc(C2CC2)n1 ZINC000147353225 CD For-Sale Anodyne CHRNA10 73 42 CC[C@@H](CNS(=O)(=O)c1cccc(Cl)c1)CC(=O)O ZINC000147353249 DE On-Demand Anodyne TBXA2R 42 34 CC[C@@H](CNS(=O)(=O)c1cccc(Cl)c1)CC(=O)O ZINC000147353249 DE On-Demand Anodyne FBP1 32 42 CS(=O)(=O)c1ccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)cn1 ZINC000147353263 EE On-Demand Anodyne EPHX2 25 41 Cc1nc(C)c(C(=O)Nc2cccc(OCC(=O)O)c2)o1 ZINC000147353277 CE On-Demand Anodyne FABP4 59 41 Cc1nc(C)c(C(=O)Nc2cccc(OCC(=O)O)c2)o1 ZINC000147353277 CE On-Demand Anodyne FABP5 28 40 Cc1nc(C)c(C(=O)Nc2cccc(OCC(=O)O)c2)o1 ZINC000147353277 CE On-Demand Anodyne KCNK3 74 38 Cc1nc(C)c(C(=O)Nc2cccc(OCC(=O)O)c2)o1 ZINC000147353277 CE On-Demand Anodyne KCNK9 78 36 CC(C)CCCCN[C@H]1CCCC[C@@H]1c1ccccc1 ZINC000147353294 CK For-Sale Anodyne GRIA4 19 48 O=C(O)c1cc(Cl)cc(NC(=O)N2CCSCC2)c1 ZINC000147353353 DF On-Demand Anodyne HCAR1 0 40 CCCCCCCCNC(=O)c1cc(NN)ccn1 ZINC000147353367 CE For-Sale Mild ASAH1 90 35 CC[C@H]1CN(C(=O)Nc2ccccc2)CC[C@H]1N ZINC000147353410 BE On-Demand Anodyne NPY2R 36 41 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H](c1ccc3c(c1)OCCO3)C1CC1)C2 ZINC000147353433 GG On-Demand Anodyne ROCK2 19 41 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(Cl)c1N1CCOCC1 ZINC000147353443 GD On-Demand Anodyne MAPK8 18 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(Cl)c1N1CCOCC1 ZINC000147353443 GD On-Demand Anodyne TNK2 22 42 CS(=O)(=O)c1ccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)cn1 ZINC000147353461 EE On-Demand Anodyne EPHX2 25 41 CNCc1cnc(C)cc1Oc1ccc(Cl)c(F)c1 ZINC000147353463 CH For-Sale Anodyne SLC6A2 15 63 CNCc1cnc(C)cc1Oc1ccc(Cl)c(F)c1 ZINC000147353463 CH For-Sale Anodyne SLC6A4 23 64 CN1CCCC[C@H]1COc1cc(NN)nc(C(C)(C)C)n1 ZINC000147353474 CD For-Sale Anodyne CHRNA10 72 41 CC(C)CCCCN[C@@H]1CCCC[C@H]1c1ccccc1 ZINC000147353478 CK For-Sale Anodyne GRIA4 19 48 O=C(O)COc1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147353481 CF On-Demand Anodyne FABP4 45 35 O=C(O)COc1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147353481 CF On-Demand Anodyne COLA 59 41 O=C(O)COc1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147353481 CF On-Demand Anodyne CPT1A 55 41 O=C(O)COc1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147353481 CF On-Demand Anodyne EPHX2 23 46 O=C(O)COc1cccc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147353481 CF On-Demand Anodyne KCNK3 24 42 CCC(=O)c1ccc(NC(=O)CCl)cc1 ZINC000147353531 BE For-Sale Reactive ACR 41 32 CCC(=O)c1ccc(NC(=O)CCl)cc1 ZINC000147353531 BE For-Sale Reactive PPO2 15 45 CCC(=O)c1ccc(NC(=O)CCl)cc1 ZINC000147353531 BE For-Sale Reactive SLC27A1 17 42 COc1ccc(Br)c(C(=O)N2CCC[C@H](CCBr)C2)c1 ZINC000147353537 HI For-Sale Reactive GRM3 16 48 CCCCCCCCNC(=O)c1ccc(NN)cc1 ZINC000147353556 CG For-Sale Mild FOLH1 30 50 CCCCCCCCNC(=O)c1ccc(NN)cc1 ZINC000147353556 CG For-Sale Mild THRB 0 58 CCCCCCCCNC(=O)c1ccc(NN)cc1 ZINC000147353556 CG For-Sale Mild HDAC6 15 46 CCCCCCCCNC(=O)c1ccc(NN)cc1 ZINC000147353556 CG For-Sale Mild S1PR2 51 38 CCCCCCCCNC(=O)c1ccc(NN)cc1 ZINC000147353556 CG For-Sale Mild EPHX2 19 45 CCCCCCCCNC(=O)c1ccc(NN)cc1 ZINC000147353556 CG For-Sale Mild ASAH1 101 40 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H](c1ccc3c(c1)OCCO3)C1CC1)C2 ZINC000147353581 GG On-Demand Anodyne ROCK2 19 41 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(Cl)c1N1CCOCC1 ZINC000147353601 GD On-Demand Anodyne MAPK8 18 42 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(Cl)c1N1CCOCC1 ZINC000147353601 GD On-Demand Anodyne TNK2 22 42 COc1cccc(CS(=O)(=O)N(C)CC(=O)O)c1 ZINC000147353609 CC On-Demand Anodyne MMP13 23 40 COc1cccc(CS(=O)(=O)N(C)CC(=O)O)c1 ZINC000147353609 CC On-Demand Anodyne MTNR1A 47 45 COc1cccc(CS(=O)(=O)N(C)CC(=O)O)c1 ZINC000147353609 CC On-Demand Anodyne MTNR1B 38 45 COc1cccc(CS(=O)(=O)N(C)CC(=O)O)c1 ZINC000147353609 CC On-Demand Anodyne MMP3 16 47 COc1cccc(CS(=O)(=O)N(C)CC(=O)O)c1 ZINC000147353609 CC On-Demand Anodyne HSD17B2 27 43 COc1cccc(CS(=O)(=O)N(C)CC(=O)O)c1 ZINC000147353609 CC On-Demand Anodyne FFAR1 17 40 COc1cccc(CS(=O)(=O)N(C)CC(=O)O)c1 ZINC000147353609 CC On-Demand Anodyne AKR1C3 15 43 COc1cccc(CS(=O)(=O)N(C)CC(=O)O)c1 ZINC000147353609 CC On-Demand Anodyne DAGLA 27 40 NC(=O)[C@H]1CCCN1C(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147353616 FD For-Sale Anodyne TRHR 54 33 C=CCCOCC(=O)Nc1cccc(CN2CCCCC2)c1 ZINC000147353634 DG On-Demand Mild HRH2 53 46 COc1ccc(Br)c(C(=O)N2CCC[C@@H](CCBr)C2)c1 ZINC000147353687 HI For-Sale Reactive GRM3 16 48 CCCCCCCCNC(=O)c1cc(Cl)nc(NN)c1 ZINC000147353712 CG For-Sale Mild ASAH1 84 36 CC(C)N(CCCCOCC(=O)OC(C)(C)C)c1cnc(-c2ccccc2)c(-c2ccccc2)n1 ZINC000147353720 JK In-Stock Anodyne AMY2 44 32 NC(=O)c1ccc(OCC(=O)Nc2ncc(Cc3ccc(F)cc3)s2)cc1 ZINC000147353725 GF On-Demand Anodyne SCD1 40 44 NC(=O)c1ccc(OCC(=O)Nc2ncc(Cc3ccc(F)cc3)s2)cc1 ZINC000147353725 GF On-Demand Anodyne SCD 34 44 CC(C)CCCCN[C@H]1CCCC[C@H]1c1ccccc1 ZINC000147353734 CK For-Sale Anodyne GRIA4 19 48 O=C(O)COc1cccc(NC(=O)C2[C@H]3CCCC[C@@H]23)c1 ZINC000147353737 CF For-Sale Anodyne COLA 59 41 CN1CCCC[C@@H]1COc1cc(NN)nc(C(C)(C)C)n1 ZINC000147353758 CD For-Sale Anodyne CHRNA10 72 41 CS(=O)(=O)c1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cn1 ZINC000147353759 GC On-Demand Anodyne JAK3 15 47 CS(=O)(=O)c1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)cn1 ZINC000147353759 GC On-Demand Anodyne EPHX2 43 40 NC(=O)[C@@H]1CCCN1C(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147353772 FD For-Sale Anodyne TRHR 54 33 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H](c1ccc3c(c1)OCCO3)C1CC1)C2 ZINC000147353778 GG On-Demand Anodyne ROCK2 19 41 Cc1nn(-c2ccccc2)c2cc(N3CCN(c4ccncc4)CC3)ccc12 ZINC000147353796 FI Annotated Anodyne KHK 0 74 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1nc(C(F)(F)F)cs1 ZINC000147353800 GH On-Demand Anodyne LCK 16 40 O=C(CNC(=O)Nc1cccc(CN2C(=O)CNC2=O)c1)Nc1ccc(F)cc1 ZINC000147353826 GD On-Demand Anodyne NPY1R 28 45 O=C(CNC(=O)Nc1cccc(CN2C(=O)CNC2=O)c1)Nc1ccc(F)cc1 ZINC000147353826 GD On-Demand Anodyne CCR3 55 39 Cc1ccc2nc(-c3ccc(NC(=O)[C@H]4CCCN4C(=O)c4cccs4)cc3)sc2c1 ZINC000147353900 IK On-Demand Anodyne F2 15 42 Cc1ccc2nc(-c3ccc(NC(=O)[C@H]4CCCN4C(=O)c4cccs4)cc3)sc2c1 ZINC000147353900 IK On-Demand Anodyne APP 20 45 CCCCCCCCNC(=O)c1ccc(NN)c(C)c1 ZINC000147353918 CG For-Sale Mild FOLH1 16 43 CCCCCCCCNC(=O)c1ccc(NN)c(C)c1 ZINC000147353918 CG For-Sale Mild ASAH1 87 36 CS(=O)(=O)c1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cn1 ZINC000147353943 GC On-Demand Anodyne JAK3 15 47 CS(=O)(=O)c1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)cn1 ZINC000147353943 GC On-Demand Anodyne EPHX2 43 40 O=C(O)COc1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147353965 CF On-Demand Anodyne FABP4 45 35 O=C(O)COc1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147353965 CF On-Demand Anodyne COLA 59 41 O=C(O)COc1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147353965 CF On-Demand Anodyne CPT1A 55 41 O=C(O)COc1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147353965 CF On-Demand Anodyne EPHX2 23 46 O=C(O)COc1cccc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147353965 CF On-Demand Anodyne KCNK3 24 42 Cc1nn(-c2ccccc2)c2cc(N3CCN(C4CCNCC4)C3=O)ccc12 ZINC000147354003 GG Annotated Anodyne KHK 0 61 O=C(N[C@H](c1ccc2c(c1)OCCO2)C1CC1)c1ccc2c(c1)COC2 ZINC000147354007 FG On-Demand Anodyne AKT1 23 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354047 EE On-Demand Anodyne KLK3 46 36 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354047 EE On-Demand Anodyne CTSK 38 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354047 EE On-Demand Anodyne PCSK5 51 33 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354047 EE On-Demand Anodyne FURIN 46 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354047 EE On-Demand Anodyne POLG_WNV 68 31 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354047 EE On-Demand Anodyne HPN 46 32 Cc1cc2nc(-c3ccc(N(C)C)cc3)cn2cc1Br ZINC000147354069 EI For-Sale Anodyne APP 19 63 COc1cc(C(=O)Nc2nc3ccccc3[nH]2)ccc1F ZINC000147354082 CF On-Demand Anodyne CSNK1D 29 48 COc1cc(C(=O)Nc2nc3ccccc3[nH]2)ccc1F ZINC000147354082 CF On-Demand Anodyne CPT1A 45 31 COc1cc(C(=O)Nc2nc3ccccc3[nH]2)ccc1F ZINC000147354082 CF On-Demand Anodyne CSNK1E 36 47 COc1cc(C(=O)Nc2nc3ccccc3[nH]2)ccc1F ZINC000147354082 CF On-Demand Anodyne PDGFRA 40 34 COc1cc(C(=O)Nc2nc3ccccc3[nH]2)ccc1F ZINC000147354082 CF On-Demand Anodyne FABH 0 40 COc1cc(C(=O)Nc2nc3ccccc3[nH]2)ccc1F ZINC000147354082 CF On-Demand Anodyne SHH 24 44 COc1cc(C(=O)Nc2nc3ccccc3[nH]2)ccc1F ZINC000147354082 CF On-Demand Anodyne STK33 56 45 COc1cc(C(=O)Nc2nc3ccccc3[nH]2)ccc1F ZINC000147354082 CF On-Demand Anodyne GLMU 0 40 CCCCCCCCNC(=O)c1nc(NN)ccc1Cl ZINC000147354119 CG For-Sale Mild SCNN1A 44 41 CCCCCCCCNC(=O)c1nc(NN)ccc1Cl ZINC000147354119 CG For-Sale Mild ASAH1 86 39 Cc1ncoc1C(=O)Nc1cccc(OCC(=O)O)c1 ZINC000147354198 CD On-Demand Anodyne FABP4 50 39 Cc1ncoc1C(=O)Nc1cccc(OCC(=O)O)c1 ZINC000147354198 CD On-Demand Anodyne KCNK3 87 38 Cc1ncoc1C(=O)Nc1cccc(OCC(=O)O)c1 ZINC000147354198 CD On-Demand Anodyne KCNK9 81 38 CC(C)(C)c1ccc(CCC(=O)N2CCc3[nH]c4ccccc4c3C2)cc1 ZINC000147354216 FJ On-Demand Anodyne DRD5 22 41 CC(C)(C)c1ccc(CCC(=O)N2CCc3[nH]c4ccccc4c3C2)cc1 ZINC000147354216 FJ On-Demand Anodyne SSTR4 50 35 CC(C)(C)c1ccc(CCC(=O)N2CCc3[nH]c4ccccc4c3C2)cc1 ZINC000147354216 FJ On-Demand Anodyne GPBAR1 18 44 CCN1CCN(c2ccc3c(C)nn(-c4ccccc4)c3c2)CC1 ZINC000147354244 DG Annotated Anodyne HTR1A 29 47 CCN1CCN(c2ccc3c(C)nn(-c4ccccc4)c3c2)CC1 ZINC000147354244 DG Annotated Anodyne DRD2 17 42 CCN1CCN(c2ccc3c(C)nn(-c4ccccc4)c3c2)CC1 ZINC000147354244 DG Annotated Anodyne DRD1 0 42 CCN1CCN(c2ccc3c(C)nn(-c4ccccc4)c3c2)CC1 ZINC000147354244 DG Annotated Anodyne DRD4 28 42 CCN1CCN(c2ccc3c(C)nn(-c4ccccc4)c3c2)CC1 ZINC000147354244 DG Annotated Anodyne HTR2A 20 40 CCN1CCN(c2ccc3c(C)nn(-c4ccccc4)c3c2)CC1 ZINC000147354244 DG Annotated Anodyne DRD3 15 42 CCN1CCN(c2ccc3c(C)nn(-c4ccccc4)c3c2)CC1 ZINC000147354244 DG Annotated Anodyne PLK1 0 40 CCN1CCN(c2ccc3c(C)nn(-c4ccccc4)c3c2)CC1 ZINC000147354244 DG Annotated Anodyne KHK 0 70 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354265 EE On-Demand Anodyne NPY1R 18 44 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354265 EE On-Demand Anodyne KLK3 46 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354265 EE On-Demand Anodyne CTSK 38 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354265 EE On-Demand Anodyne PCSK5 51 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354265 EE On-Demand Anodyne FURIN 46 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354265 EE On-Demand Anodyne POLG_WNV 68 31 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1cccc(NC(C)=O)c1 ZINC000147354265 EE On-Demand Anodyne HPN 46 32 Nc1nc(-c2sccc2Br)nc(N2CCCC2)n1 ZINC000147354295 EF For-Sale Anodyne ERM 0 40 O[C@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354331 FE On-Demand Anodyne ADRB2 50 54 O[C@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354331 FE On-Demand Anodyne ADRB1 0 54 O[C@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354331 FE On-Demand Anodyne HTR1A 28 58 O[C@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354331 FE On-Demand Anodyne DRD4 39 45 O[C@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354331 FE On-Demand Anodyne ADRB3 52 54 O[C@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354331 FE On-Demand Anodyne ACOX1 25 41 O[C@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354331 FE On-Demand Anodyne ABCB1 64 46 O=C(NCc1cccnc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147354419 FF For-Sale Anodyne GYRB 0 42 O=C(NCc1cccnc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147354419 FF For-Sale Anodyne CHRNA7 37 45 O=C(NCc1cccnc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147354419 FF For-Sale Anodyne ROCK2 20 45 O=C(NCc1cccnc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147354419 FF For-Sale Anodyne ACHP_LYMST 20 41 O=C(NCc1cccnc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147354419 FF For-Sale Anodyne NAMPT 100 61 C[C@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147354433 BD On-Demand Anodyne DAC 53 41 Cc1nn(-c2ccccc2)c2cc(N3CCN(C(C)C)CC3)ccc12 ZINC000147354441 EH Annotated Anodyne PLK1 15 42 Cc1nn(-c2ccccc2)c2cc(N3CCN(C(C)C)CC3)ccc12 ZINC000147354441 EH Annotated Anodyne KHK 0 70 Cc1nc(NC(=O)c2ccc(Cl)cc2)sc1-c1nc2ccccc2n1C(F)F ZINC000147354444 HK On-Demand Anodyne PIK3CG 15 41 Cc1nc(NC(=O)c2ccc(Cl)cc2)sc1-c1nc2ccccc2n1C(F)F ZINC000147354444 HK On-Demand Anodyne IMDH_CRYPV 33 42 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354469 EE On-Demand Anodyne NPY1R 18 44 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354469 EE On-Demand Anodyne KLK3 46 36 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354469 EE On-Demand Anodyne CTSK 38 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354469 EE On-Demand Anodyne PCSK5 51 33 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354469 EE On-Demand Anodyne FURIN 46 35 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354469 EE On-Demand Anodyne POLG_WNV 68 31 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354469 EE On-Demand Anodyne HPN 46 32 Fc1ccc(Cn2cc(-c3cccc(I)c3)cn2)cc1 ZINC000147354554 GI For-Sale Anodyne ADORA2B 20 40 Fc1ccc(Cn2cc(-c3cccc(I)c3)cn2)cc1 ZINC000147354554 GI For-Sale Anodyne ALK 0 48 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354560 FE On-Demand Anodyne ADRB2 50 54 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354560 FE On-Demand Anodyne ADRB1 0 54 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354560 FE On-Demand Anodyne HTR1A 28 58 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354560 FE On-Demand Anodyne DRD4 39 45 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354560 FE On-Demand Anodyne ADRB3 52 54 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354560 FE On-Demand Anodyne ACOX1 25 41 O[C@@H](COc1cccc2[nH]ccc12)CN1CCN(c2ccccn2)CC1 ZINC000147354560 FE On-Demand Anodyne ABCB1 64 46 COc1ccc(CNC2(C(=O)O)CCC2)cc1C#N ZINC000147354596 CD On-Demand Mild S1PR1 0 42 Cc1nccn1-c1ccc(CNC(=O)Nc2ccc(S(C)(=O)=O)nc2)cc1F ZINC000147354609 HE On-Demand Anodyne NAMPT 42 38 O=C(CN1CCOCC1)Nc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147354632 HC On-Demand Anodyne MTOR 80 36 O=C(CN1CCOCC1)Nc1ccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)cc1 ZINC000147354632 HC On-Demand Anodyne EPHX2 20 42 O=C(NCc1cccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147354645 DF On-Demand Anodyne GYRB 0 40 O=C(NCc1cccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147354645 DF On-Demand Anodyne PPIA 40 40 O=C(NCc1cccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147354645 DF On-Demand Anodyne TBXAS1 45 39 O=C(NCc1cccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147354645 DF On-Demand Anodyne CHRNA7 39 40 O=C(NCc1cccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147354645 DF On-Demand Anodyne ROCK2 21 45 O=C(NCc1cccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147354645 DF On-Demand Anodyne NAMPT 102 61 C[C@@H](NC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147354651 BD On-Demand Anodyne DAC 53 41 Cc1nn(-c2ccccc2)c2cc(N3CCN[C@H](C)C3)ccc12 ZINC000147354652 DG Annotated Anodyne KHK 0 76 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354667 EE On-Demand Anodyne NPY1R 18 44 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354667 EE On-Demand Anodyne KLK3 46 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354667 EE On-Demand Anodyne CTSK 38 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354667 EE On-Demand Anodyne PCSK5 51 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354667 EE On-Demand Anodyne FURIN 46 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354667 EE On-Demand Anodyne POLG_WNV 68 31 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1cccc(NC(C)=O)c1 ZINC000147354667 EE On-Demand Anodyne HPN 46 32 O=C(CC1CCNCC1)NN1CCCCC1 ZINC000147354680 BC For-Sale Anodyne F2R 24 40 CC[C@@H]1CN(C(=O)Nc2ccccc2F)CC[C@@H]1N ZINC000147354734 CE On-Demand Anodyne RBP4 55 38 O=C(CN1CCOCC1)Nc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147354841 HC On-Demand Anodyne MTOR 80 36 O=C(CN1CCOCC1)Nc1ccc(NC(=O)C(=O)NC[C@H]2CCCCO2)cc1 ZINC000147354841 HC On-Demand Anodyne EPHX2 20 42 O=C(NCc1ccncc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147354844 FF For-Sale Anodyne FLT1 29 42 O=C(NCc1ccncc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147354844 FF For-Sale Anodyne ROCK2 23 52 O=C(NCc1ccncc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147354844 FF For-Sale Anodyne EPHB4 25 40 O=C(NCc1ccncc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147354844 FF For-Sale Anodyne NAMPT 50 42 Cc1cccc(Cl)c1NC(=O)c1cccc2c1OCCN2 ZINC000147354847 DH For-Sale Anodyne LCK 35 40 CS(=O)(=O)c1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cn1 ZINC000147354854 HG On-Demand Anodyne ROCK2 24 45 CS(=O)(=O)c1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cn1 ZINC000147354854 HG On-Demand Anodyne MET 49 45 CS(=O)(=O)c1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cn1 ZINC000147354854 HG On-Demand Anodyne CYP2C9 15 42 CS(=O)(=O)c1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cn1 ZINC000147354854 HG On-Demand Anodyne NAMPT 76 45 CN(C)Cc1cccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)c1 ZINC000147354855 EF On-Demand Anodyne CCR3 43 37 CN(C)Cc1cccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)c1 ZINC000147354855 EF On-Demand Anodyne NAMPT 0 50 CN(C)Cc1cccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)c1 ZINC000147354855 EF On-Demand Anodyne PSBA 0 40 Cc1nn(-c2ccccc2)c2cc(N3CCN[C@@H](C)C3)ccc12 ZINC000147354861 DG Annotated Anodyne KHK 0 76 FC(F)(F)c1ccc2c(c1)[C@@H]1C=CC[C@H]1[C@@H](c1ccccc1)N2 ZINC000147354880 DK In-Stock Clean KIF11 23 60 CC[C@H]1CN(C(=O)Nc2ccccc2F)CC[C@@H]1N ZINC000147354884 CE On-Demand Anodyne RBP4 55 38 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(=O)n(C)c1 ZINC000147354955 FE On-Demand Anodyne LPL 46 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(=O)n(C)c1 ZINC000147354955 FE On-Demand Anodyne HRH3 0 41 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147354957 CH On-Demand Anodyne ACE 47 39 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147354957 CH On-Demand Anodyne MME 47 39 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147354957 CH On-Demand Anodyne NPY1R 29 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147354957 CH On-Demand Anodyne GZMB 48 29 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147354957 CH On-Demand Anodyne XIAP 31 41 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147354957 CH On-Demand Anodyne BIRC2 41 38 CCCCCCCCCCCCN(C[C@@H](O)CCl)C[C@@H](O)CCl ZINC000147354965 FI For-Sale Reactive CQSS 41 31 Cc1cn2nc([C@@H]3CCCCN3C(=O)c3ccccc3NS(C)(=O)=O)cc2nc1C ZINC000147354996 IG Annotated Anodyne COLA 56 39 Cc1cn2nc([C@@H]3CCCCN3C(=O)c3ccccc3NS(C)(=O)=O)cc2nc1C ZINC000147354996 IG Annotated Anodyne CPT1A 55 39 COc1ccc([C@H](NCC(F)F)c2ccccc2)cc1 ZINC000147355000 CH On-Demand Anodyne AOC3 20 41 O=C(NCc1ccncc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147355072 DF On-Demand Anodyne PPIA 29 43 O=C(NCc1ccncc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147355072 DF On-Demand Anodyne FLT1 40 39 O=C(NCc1ccncc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147355072 DF On-Demand Anodyne KDR 15 41 O=C(NCc1ccncc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147355072 DF On-Demand Anodyne ROCK2 22 52 O=C(NCc1ccncc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147355072 DF On-Demand Anodyne NAMPT 53 42 CC[C@@H]1CN(C(=O)Nc2ccccc2F)CC[C@H]1N ZINC000147355082 CE On-Demand Anodyne RBP4 55 38 COc1nn(-c2ccccc2)c2cc(N3CCN([C@@H]4CCNC4)CC3)ccc12 ZINC000147355096 GF Annotated Anodyne KHK 0 90 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147355103 CH On-Demand Anodyne ACE 47 39 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147355103 CH On-Demand Anodyne MME 47 39 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147355103 CH On-Demand Anodyne NPY1R 29 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147355103 CH On-Demand Anodyne GZMB 48 29 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147355103 CH On-Demand Anodyne XIAP 31 41 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H]1CCc2ccccc21 ZINC000147355103 CH On-Demand Anodyne BIRC2 41 38 CCCCCCCCCCCCN(C[C@H](O)CCl)C[C@@H](O)CCl ZINC000147355135 FI For-Sale Reactive CQSS 41 31 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCOCC1(C)C)C2 ZINC000147355136 DD On-Demand Anodyne MT-ND4 40 30 COc1ccc([C@@H](NCC(F)F)c2ccccc2)cc1 ZINC000147355216 CH On-Demand Anodyne AOC3 20 41 CC(C)CCCCN[C@@H]1CCN(CCc2ccccc2)C1 ZINC000147355243 CH For-Sale Anodyne DRD2 15 42 CC(C)CCCCN[C@@H]1CCN(CCc2ccccc2)C1 ZINC000147355243 CH For-Sale Anodyne DRD4 23 44 CC(C)CCCCN[C@@H]1CCN(CCc2ccccc2)C1 ZINC000147355243 CH For-Sale Anodyne OPRM1 15 45 CC(C)CCCCN[C@@H]1CCN(CCc2ccccc2)C1 ZINC000147355243 CH For-Sale Anodyne SLC18A2 36 40 CC(C)CCCCN[C@@H]1CCN(CCc2ccccc2)C1 ZINC000147355243 CH For-Sale Anodyne GRIN2B 15 45 CC(C)CCCCN[C@@H]1CCN(CCc2ccccc2)C1 ZINC000147355243 CH For-Sale Anodyne SIGMAR1 61 52 CC(C)CCCCN[C@@H]1CCN(CCc2ccccc2)C1 ZINC000147355243 CH For-Sale Anodyne BIRC2 82 44 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(OCC(=O)OC)cc2)C1 ZINC000147355288 FD On-Demand Anodyne MMP13 75 41 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(OCC(=O)OC)cc2)C1 ZINC000147355288 FD On-Demand Anodyne ADAM17 59 47 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(OCC(=O)OC)cc2)C1 ZINC000147355288 FD On-Demand Anodyne MMP3 67 41 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(OCC(=O)OC)cc2)C1 ZINC000147355288 FD On-Demand Anodyne MMP9 38 41 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(OCC(=O)OC)cc2)C1 ZINC000147355288 FD On-Demand Anodyne MMP7 64 39 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(OCC(=O)OC)cc2)C1 ZINC000147355288 FD On-Demand Anodyne MMP1 73 41 CC[C@H]1CN(C(=O)Nc2ccccc2F)CC[C@H]1N ZINC000147355293 CE On-Demand Anodyne RBP4 55 38 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147355314 BD For-Sale Anodyne SLC15A1 0 40 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147355314 BD For-Sale Anodyne GPR88 0 54 COc1nn(-c2ccccc2)c2cc(N3CCN([C@H]4CCNC4)CC3)ccc12 ZINC000147355315 GF Annotated Anodyne KHK 0 90 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355322 CH On-Demand Anodyne ACE 47 39 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355322 CH On-Demand Anodyne MME 47 39 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355322 CH On-Demand Anodyne NPY1R 29 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355322 CH On-Demand Anodyne GZMB 48 29 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355322 CH On-Demand Anodyne XIAP 31 41 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355322 CH On-Demand Anodyne BIRC2 41 38 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(S(C)(=O)=O)nc1 ZINC000147355338 HE On-Demand Anodyne LCK 23 42 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(S(C)(=O)=O)nc1 ZINC000147355338 HE On-Demand Anodyne HCK 17 40 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(S(C)(=O)=O)nc1 ZINC000147355338 HE On-Demand Anodyne FLT3 15 40 CCCCCCCCn1c([C@@H](C)O)nc2cc(N)ccc21 ZINC000147355387 CI For-Sale Mild TLR8 0 40 CCCCCCCCn1c([C@@H](C)O)nc2cc(N)ccc21 ZINC000147355387 CI For-Sale Mild OXER1 46 32 CCCCCCCCCCCCN(C[C@H](O)CCl)C[C@H](O)CCl ZINC000147355394 FI For-Sale Reactive CQSS 41 31 Cc1ccccc1-n1nc(C(=O)NCc2ccc(N3CCCC3)nc2)c2c1CCC2 ZINC000147355425 HH On-Demand Anodyne CNR1 50 32 COc1ccc(CNCC(F)F)c(O)c1 ZINC000147355431 BD For-Sale Clean PHES 0 41 CC(C)CCCCN[C@H]1CCN(CCc2ccccc2)C1 ZINC000147355434 CH For-Sale Anodyne DRD2 15 42 CC(C)CCCCN[C@H]1CCN(CCc2ccccc2)C1 ZINC000147355434 CH For-Sale Anodyne DRD4 23 44 CC(C)CCCCN[C@H]1CCN(CCc2ccccc2)C1 ZINC000147355434 CH For-Sale Anodyne OPRM1 15 45 CC(C)CCCCN[C@H]1CCN(CCc2ccccc2)C1 ZINC000147355434 CH For-Sale Anodyne SLC18A2 36 40 CC(C)CCCCN[C@H]1CCN(CCc2ccccc2)C1 ZINC000147355434 CH For-Sale Anodyne GRIN2B 15 45 CC(C)CCCCN[C@H]1CCN(CCc2ccccc2)C1 ZINC000147355434 CH For-Sale Anodyne SIGMAR1 61 52 CC(C)CCCCN[C@H]1CCN(CCc2ccccc2)C1 ZINC000147355434 CH For-Sale Anodyne BIRC2 82 44 CC(C)N1CCN(C[C@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355440 DD On-Demand Anodyne ADRB2 19 51 CC(C)N1CCN(C[C@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355440 DD On-Demand Anodyne ADRB1 22 60 CC(C)N1CCN(C[C@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355440 DD On-Demand Anodyne HTR1A 25 60 CC(C)N1CCN(C[C@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355440 DD On-Demand Anodyne SLC6A4 23 52 CC(C)N1CCN(C[C@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355440 DD On-Demand Anodyne ADRB3 21 57 CC(C)N1CCN(C[C@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355440 DD On-Demand Anodyne ACOX1 44 46 CC(C)N1CCN(C[C@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355440 DD On-Demand Anodyne ABCB1 65 44 Cc1cc(Cl)cc(C(=O)Nc2nc3ccccc3[nH]2)c1 ZINC000147355484 CH On-Demand Anodyne KCNN3 36 42 Cc1cc(Cl)cc(C(=O)Nc2nc3ccccc3[nH]2)c1 ZINC000147355484 CH On-Demand Anodyne NR2E3 65 38 Cc1cc(Cl)cc(C(=O)Nc2nc3ccccc3[nH]2)c1 ZINC000147355484 CH On-Demand Anodyne SHH 25 46 Cc1cc(Cl)cc(C(=O)Nc2nc3ccccc3[nH]2)c1 ZINC000147355484 CH On-Demand Anodyne STK33 56 44 Cc1cc(Cl)cc(C(=O)Nc2nc3ccccc3[nH]2)c1 ZINC000147355484 CH On-Demand Anodyne KCNK3 49 38 Cc1cc(Cl)cc(C(=O)Nc2nc3ccccc3[nH]2)c1 ZINC000147355484 CH On-Demand Anodyne KCNK9 28 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355495 CH On-Demand Anodyne ACE 47 39 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355495 CH On-Demand Anodyne MME 47 39 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355495 CH On-Demand Anodyne TRPV1 23 42 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355495 CH On-Demand Anodyne NPY1R 29 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355495 CH On-Demand Anodyne SCN9A 33 52 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355495 CH On-Demand Anodyne GZMB 48 29 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355495 CH On-Demand Anodyne XIAP 31 41 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H]1CCc2ccccc21 ZINC000147355495 CH On-Demand Anodyne BIRC2 41 38 CC[C@@H]1CN(C(=O)Oc2ccccc2)CC[C@@H]1N ZINC000147355503 BE For-Sale Anodyne NPY2R 15 48 CC[C@@H]1CN(C(=O)Oc2ccccc2)CC[C@@H]1N ZINC000147355503 BE For-Sale Anodyne CHRNA4 0 44 CC[C@@H]1CN(C(=O)Oc2ccccc2)CC[C@@H]1N ZINC000147355503 BE For-Sale Anodyne MGLL 0 42 CC[C@@H]1CN(C(=O)Oc2ccccc2)CC[C@@H]1N ZINC000147355503 BE For-Sale Anodyne ABHD6 0 42 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2cccs2)c1 ZINC000147355509 GF On-Demand Anodyne KCNK3 60 52 O=C(NC[C@@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2cccs2)c1 ZINC000147355509 GF On-Demand Anodyne KCNK9 39 52 C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147355537 BD For-Sale Anodyne SLC15A1 0 40 C[C@@H](NC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147355537 BD For-Sale Anodyne GPR88 0 54 CCC(=O)c1cccc(NC(=O)N2CCC(Oc3ccccc3Cl)CC2)c1 ZINC000147355541 GK On-Demand Anodyne P2RY12 20 40 CCC(=O)c1cccc(NC(=O)N2CCC(Oc3ccccc3Cl)CC2)c1 ZINC000147355541 GK On-Demand Anodyne CCR3 44 38 CCC(=O)c1cccc(NC(=O)N2CCC(Oc3ccccc3Cl)CC2)c1 ZINC000147355541 GK On-Demand Anodyne EPHX2 50 50 CCC(=O)c1cccc(NC(=O)N2CCC(Oc3ccccc3Cl)CC2)c1 ZINC000147355541 GK On-Demand Anodyne P2RY14 42 34 CCC(=O)c1cccc(NC(=O)N2CCC(Oc3ccccc3Cl)CC2)c1 ZINC000147355541 GK On-Demand Anodyne SCD1 44 79 CCC(=O)c1cccc(NC(=O)N2CCC(Oc3ccccc3Cl)CC2)c1 ZINC000147355541 GK On-Demand Anodyne SCD 26 47 CCC(=O)c1cccc(NC(=O)N2CCC(Oc3ccccc3Cl)CC2)c1 ZINC000147355541 GK On-Demand Anodyne KCNK3 42 34 CC1(C)COCCN1C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147355557 CG On-Demand Anodyne MDM2 79 34 CCCCCCCCn1c([C@H](C)O)nc2cc(N)ccc21 ZINC000147355572 CI For-Sale Mild TLR8 0 40 CCCCCCCCn1c([C@H](C)O)nc2cc(N)ccc21 ZINC000147355572 CI For-Sale Mild OXER1 46 32 C=Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147355597 FE Annotated Mild HDAC1 0 78 C=Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147355597 FE Annotated Mild HDAC6 22 78 CC(C)N1CCN(C[C@@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355668 DD On-Demand Anodyne ADRB2 19 51 CC(C)N1CCN(C[C@@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355668 DD On-Demand Anodyne ADRB1 22 60 CC(C)N1CCN(C[C@@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355668 DD On-Demand Anodyne HTR1A 25 60 CC(C)N1CCN(C[C@@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355668 DD On-Demand Anodyne SLC6A4 23 52 CC(C)N1CCN(C[C@@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355668 DD On-Demand Anodyne ADRB3 21 57 CC(C)N1CCN(C[C@@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355668 DD On-Demand Anodyne ACOX1 44 46 CC(C)N1CCN(C[C@@H](O)COc2cccc3[nH]ccc23)CC1 ZINC000147355668 DD On-Demand Anodyne ABCB1 65 44 CC[C@H]1CN(C(=O)Oc2ccccc2)CC[C@@H]1N ZINC000147355703 BE For-Sale Anodyne NPY2R 15 48 CC[C@H]1CN(C(=O)Oc2ccccc2)CC[C@@H]1N ZINC000147355703 BE For-Sale Anodyne CHRNA4 0 44 CC[C@H]1CN(C(=O)Oc2ccccc2)CC[C@@H]1N ZINC000147355703 BE For-Sale Anodyne MGLL 0 42 CC[C@H]1CN(C(=O)Oc2ccccc2)CC[C@@H]1N ZINC000147355703 BE For-Sale Anodyne ABHD6 0 42 Cc1nn(C(F)F)c(C)c1CC(=O)NCc1ccc(N2CCCC2)nc1 ZINC000147355710 FF On-Demand Anodyne P2RX7 52 44 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2cccs2)c1 ZINC000147355719 GF On-Demand Anodyne KCNK3 60 52 O=C(NC[C@H]1CCCCO1)C(=O)Nc1cccc(NC(=O)c2cccs2)c1 ZINC000147355719 GF On-Demand Anodyne KCNK9 39 52 C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147355720 BD For-Sale Anodyne SLC15A1 0 40 C[C@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147355720 BD For-Sale Anodyne GPR88 0 54 CC1(C)COCCN1C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147355751 CG On-Demand Anodyne MDM2 79 34 CC(C)(C)CC[C@H](c1ccc(C(=O)NCc2nn[nH]n2)cc1)N1C(=O)C(c2cc(F)cc(F)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147355773 KK Annotated Anodyne GLP1R 15 69 CC(C)c1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147355793 FF Annotated Mild HDAC1 26 75 CC(C)c1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147355793 FF Annotated Mild HDAC6 26 74 CC(C)c1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147355793 FF Annotated Mild HDA106 0 40 CCCCCCCCn1c(C)nc2cc(N)ccc21 ZINC000147355810 CI For-Sale Mild TLR8 0 45 Cc1ncccc1NC(=O)c1cccc2c1OCCN2 ZINC000147355824 CE For-Sale Anodyne G2YM83_BOTF4 81 42 C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147355878 BD For-Sale Anodyne SLC15A1 0 40 C[C@@H](NC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147355878 BD For-Sale Anodyne GPR88 0 54 CS(=O)(=O)c1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cn1 ZINC000147355895 GF On-Demand Anodyne NAMPT 41 36 CC[C@@H]1CN(C(=O)Oc2ccccc2)CC[C@H]1N ZINC000147355902 BE For-Sale Anodyne NPY2R 15 48 CC[C@@H]1CN(C(=O)Oc2ccccc2)CC[C@H]1N ZINC000147355902 BE For-Sale Anodyne CHRNA4 0 44 CC[C@@H]1CN(C(=O)Oc2ccccc2)CC[C@H]1N ZINC000147355902 BE For-Sale Anodyne MGLL 0 42 CC[C@@H]1CN(C(=O)Oc2ccccc2)CC[C@H]1N ZINC000147355902 BE For-Sale Anodyne ABHD6 0 42 CCCCCN1C[C@@H](O)C[C@H]1C(=O)OC ZINC000147355935 BC On-Demand Anodyne GBA2 57 41 CCCCCN1C[C@@H](O)C[C@H]1C(=O)OC ZINC000147355935 BC On-Demand Anodyne P0504H10.9 0 41 CCCCCN1C[C@@H](O)C[C@H]1C(=O)OC ZINC000147355935 BC On-Demand Anodyne SIS 0 42 C[C@H]1OCC[C@H]1Nc1ccc2c(c1)Cc1ccccc1-2 ZINC000147355945 CH For-Sale Anodyne GALE 0 40 CCCNc1nc(OC)nc(Oc2cccc(Cl)c2Cl)n1 ZINC000147355962 EH For-Sale Anodyne ALS 37 41 CC1(C)COCCN1C(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147355972 CG On-Demand Anodyne MDM2 79 34 CCO[C@@H]1CCCN(S(=O)(=O)c2cc3c(cc2F)NC(=O)CC3)C1 ZINC000147355974 FD On-Demand Anodyne PKM 34 42 CCCCCCCCn1c(CCC)nc2cc(N)ccc21 ZINC000147355982 CJ For-Sale Mild HDAC10 21 48 CCCCCCCCn1c(CCC)nc2cc(N)ccc21 ZINC000147355982 CJ For-Sale Mild HDAC1 0 49 CCCCCCCCn1c(CCC)nc2cc(N)ccc21 ZINC000147355982 CJ For-Sale Mild HDAC4 22 48 CCCCCCCCn1c(CCC)nc2cc(N)ccc21 ZINC000147355982 CJ For-Sale Mild HDAC5 29 48 CCCCCCCCn1c(CCC)nc2cc(N)ccc21 ZINC000147355982 CJ For-Sale Mild HDAC9 23 48 CCCCCCCCn1c(CCC)nc2cc(N)ccc21 ZINC000147355982 CJ For-Sale Mild HDAC11 22 48 CCCCCCCCn1c(CCC)nc2cc(N)ccc21 ZINC000147355982 CJ For-Sale Mild HDAC7 33 48 CCCCCCCCn1c(CCC)nc2cc(N)ccc21 ZINC000147355982 CJ For-Sale Mild TLR8 0 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(-n2cccn2)c(F)c1 ZINC000147355989 HH On-Demand Anodyne NPY2R 67 36 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(-n2cccn2)c(F)c1 ZINC000147355989 HH On-Demand Anodyne KDR 15 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc(-n2cccn2)c(F)c1 ZINC000147355989 HH On-Demand Anodyne FLT3 17 41 CC(C)C1CCC2(CC1)N=C(c1cc(Cl)cc(Cl)c1)C(=O)N2[C@H](CCC(C)(C)C)c1ccc(C(=O)NCc2nn[nH]n2)cc1 ZINC000147355998 KK Annotated Anodyne GCGR 22 81 CC(C)C1CCC2(CC1)N=C(c1cc(Cl)cc(Cl)c1)C(=O)N2[C@H](CCC(C)(C)C)c1ccc(C(=O)NCc2nn[nH]n2)cc1 ZINC000147355998 KK Annotated Anodyne GLP1R 16 73 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1Cc1ccccc1)NO ZINC000147356019 HG Annotated Mild MAP 0 42 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1Cc1ccccc1)NO ZINC000147356019 HG Annotated Mild HDAC8 29 42 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1Cc1ccccc1)NO ZINC000147356019 HG Annotated Mild HDAC10 39 43 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1Cc1ccccc1)NO ZINC000147356019 HG Annotated Mild HDAC2 31 42 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1Cc1ccccc1)NO ZINC000147356019 HG Annotated Mild HDAC5 15 40 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1Cc1ccccc1)NO ZINC000147356019 HG Annotated Mild HDAC6 36 42 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1Cc1ccccc1)NO ZINC000147356019 HG Annotated Mild HDAC11 15 40 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1Cc1ccccc1)NO ZINC000147356019 HG Annotated Mild HDA106 0 46 O=C(O)c1cc(Cl)cc(NC(=O)N2CCC(CO)CC2)c1 ZINC000147356047 DE On-Demand Anodyne CACNA1H 43 35 O=C(O)c1cc(Cl)cc(NC(=O)N2CCC(CO)CC2)c1 ZINC000147356047 DE On-Demand Anodyne CACNA1I 46 37 Cc1ccc(C(=O)N[C@@H](C)C(=O)O)cc1Br ZINC000147356072 CD On-Demand Anodyne CA2 18 54 Cc1ccc(C(=O)N[C@@H](C)C(=O)O)cc1Br ZINC000147356072 CD On-Demand Anodyne CA4 15 53 Cc1ccc(C(=O)N[C@@H](C)C(=O)O)cc1Br ZINC000147356072 CD On-Demand Anodyne SLC15A2 0 43 CC[C@H]1CN(C(=O)Oc2ccccc2)CC[C@H]1N ZINC000147356100 BE For-Sale Anodyne NPY2R 15 48 CC[C@H]1CN(C(=O)Oc2ccccc2)CC[C@H]1N ZINC000147356100 BE For-Sale Anodyne CHRNA4 0 44 CC[C@H]1CN(C(=O)Oc2ccccc2)CC[C@H]1N ZINC000147356100 BE For-Sale Anodyne MGLL 0 42 CC[C@H]1CN(C(=O)Oc2ccccc2)CC[C@H]1N ZINC000147356100 BE For-Sale Anodyne ABHD6 0 42 CS(=O)(=O)c1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cn1 ZINC000147356108 GF On-Demand Anodyne NAMPT 41 36 CC[C@H](NC(=O)c1cc(C(F)(F)F)ccc1Br)C(=O)O ZINC000147356114 FG On-Demand Anodyne MTTP 48 33 CCO[C@H]1CCCN(S(=O)(=O)c2cc3c(cc2F)NC(=O)CC3)C1 ZINC000147356168 FD On-Demand Anodyne PKM 34 42 C[C@@H]1OCC[C@H]1Nc1ccc2c(c1)Cc1ccccc1-2 ZINC000147356174 CH For-Sale Anodyne GALE 0 40 COc1nc(N)nc(Oc2cccc(Cl)c2Cl)n1 ZINC000147356191 CF For-Sale Anodyne ALS 49 44 CCCCCCCCn1cnc2cc(N)ccc21 ZINC000147356211 BH For-Sale Mild NR1I2 32 54 CCCCCCCCn1cnc2cc(N)ccc21 ZINC000147356211 BH For-Sale Mild ICMT 37 41 CC(C)(C)CC[C@H](c1ccc(C(=O)NCc2nn[nH]n2)cc1)N1C(=O)C(c2cc(F)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147356228 KK Annotated Anodyne GLP1R 17 75 COCCOc1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c(C)c1 ZINC000147356231 FG On-Demand Bother TAAR1 18 41 COCCOc1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c(C)c1 ZINC000147356231 FG On-Demand Bother AKR1C3 15 41 COCCOc1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])c(C)c1 ZINC000147356231 FG On-Demand Bother AKR1C2 42 43 Cc1ccccc1NC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147356240 EI For-Sale Anodyne EPHX1 0 42 Cc1ccccc1NC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147356240 EI For-Sale Anodyne LPL 54 37 Cc1ccccc1NC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147356240 EI For-Sale Anodyne DDX3X 0 52 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1N1CCOCC1 ZINC000147356249 EC On-Demand Anodyne PCSK5 53 32 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1N1CCOCC1 ZINC000147356249 EC On-Demand Anodyne FURIN 50 33 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1N1CCOCC1 ZINC000147356249 EC On-Demand Anodyne SCN10A 23 45 Cc1cc(F)cc(NC(=O)c2cccc3c2OCCN3)c1 ZINC000147356253 CG For-Sale Anodyne KCNK3 70 35 Cc1cc(F)cc(NC(=O)c2cccc3c2OCCN3)c1 ZINC000147356253 CG For-Sale Anodyne KCNK9 66 35 CCc1ncc(C(=O)N(C)Cc2ccc(OCc3ccccc3)c(OC)c2)s1 ZINC000147356254 GJ On-Demand Anodyne DRTS_PLAFK 31 45 CCc1ncc(C(=O)N(C)Cc2ccc(OCc3ccccc3)c(OC)c2)s1 ZINC000147356254 GJ On-Demand Anodyne PTGER1 51 46 CCc1ncc(C(=O)N(C)Cc2ccc(OCc3ccccc3)c(OC)c2)s1 ZINC000147356254 GJ On-Demand Anodyne PTGER4 25 46 CCc1ncc(C(=O)N(C)Cc2ccc(OCc3ccccc3)c(OC)c2)s1 ZINC000147356254 GJ On-Demand Anodyne MT-ND1 23 41 CCc1ncc(C(=O)N(C)Cc2ccc(OCc3ccccc3)c(OC)c2)s1 ZINC000147356254 GJ On-Demand Anodyne HSD17B2 29 42 N#Cc1ccc(N2CCN(C(=O)c3cnn(-c4ccccc4Cl)c3)CC2)nc1 ZINC000147356268 GF On-Demand Mild SMO 18 41 Nc1cccc(CC(=O)NCc2sccc2Br)c1 ZINC000147356301 EF For-Sale Anodyne MAPK8 0 43 Cc1ccc(C(=O)N[C@H](C)C(=O)O)cc1Br ZINC000147356307 CD On-Demand Anodyne CA2 18 54 Cc1ccc(C(=O)N[C@H](C)C(=O)O)cc1Br ZINC000147356307 CD On-Demand Anodyne CA4 15 53 Cc1ccc(C(=O)N[C@H](C)C(=O)O)cc1Br ZINC000147356307 CD On-Demand Anodyne SLC15A2 0 43 CS(=O)(=O)c1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cn1 ZINC000147356335 GF On-Demand Anodyne NAMPT 41 36 O=C(Nc1ccccc1)Nc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147356355 GF On-Demand Anodyne EPHX2 22 42 O=C(Nc1ccccc1)Nc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147356355 GF On-Demand Anodyne DGAT1 15 40 O=C(Nc1ccccc1)Nc1cccc(NC(=O)C(=O)NC[C@@H]2CCCCO2)c1 ZINC000147356355 GF On-Demand Anodyne KCNK3 47 41 C[C@H]1OCC[C@@H]1Nc1ccc2c(c1)Cc1ccccc1-2 ZINC000147356381 CH For-Sale Anodyne GALE 0 40 CCCCNC(=O)N1CC[C@H](N)[C@H](CC)C1 ZINC000147356385 BD On-Demand Anodyne ASAH1 59 32 CCCCCCCCn1c(CO)nc2cc(N)ccc21 ZINC000147356423 CG For-Sale Mild HDAC1 0 48 CCCCCCCCn1c(CO)nc2cc(N)ccc21 ZINC000147356423 CG For-Sale Mild HDAC4 15 42 CCCCCCCCn1c(CO)nc2cc(N)ccc21 ZINC000147356423 CG For-Sale Mild HDAC5 27 42 CCCCCCCCn1c(CO)nc2cc(N)ccc21 ZINC000147356423 CG For-Sale Mild HDAC9 19 42 CCCCCCCCn1c(CO)nc2cc(N)ccc21 ZINC000147356423 CG For-Sale Mild HDAC11 17 42 CCCCCCCCn1c(CO)nc2cc(N)ccc21 ZINC000147356423 CG For-Sale Mild HDAC7 30 42 CCOC(=O)c1cc(C)cc(N)n1 ZINC000147356450 AD For-Sale Anodyne NOS1 30 44 CCOC(=O)c1cc(C)cc(N)n1 ZINC000147356450 AD For-Sale Anodyne NOS2 20 47 CCOC(=O)c1cc(C)cc(N)n1 ZINC000147356450 AD For-Sale Anodyne NOS3 29 47 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1N1CCOCC1 ZINC000147356466 EC On-Demand Anodyne PCSK5 53 32 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1N1CCOCC1 ZINC000147356466 EC On-Demand Anodyne FURIN 50 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1N1CCOCC1 ZINC000147356466 EC On-Demand Anodyne SCN10A 23 45 Cc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147356471 DH On-Demand Anodyne EPHX1 0 42 Cc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147356471 DH On-Demand Anodyne PPIA 31 48 Cc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147356471 DH On-Demand Anodyne LPL 56 37 Cc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147356471 DH On-Demand Anodyne CXCL8 43 33 Cc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147356471 DH On-Demand Anodyne PTGER3 24 44 Cc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147356471 DH On-Demand Anodyne ITGA4 47 40 Cc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147356471 DH On-Demand Anodyne AKR1C3 38 41 Cc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147356471 DH On-Demand Anodyne DDX3X 0 52 N#Cc1ccc(N2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147356480 FG On-Demand Mild SSTR1 15 44 N#Cc1ccc(N2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147356480 FG On-Demand Mild SMO 15 47 N#Cc1ccc(N2CCN(C(=O)[C@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147356480 FG On-Demand Mild NPBWR1 66 40 CS(=O)(=O)c1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cn1 ZINC000147356546 GF On-Demand Anodyne NAMPT 41 36 O=C(NN1CCCCC1)c1ccc2c(c1)CCN2 ZINC000147356553 BD For-Sale Anodyne CNR1 58 36 O=C(Nc1ccccc1)Nc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147356570 GF On-Demand Anodyne EPHX2 22 42 O=C(Nc1ccccc1)Nc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147356570 GF On-Demand Anodyne DGAT1 15 40 O=C(Nc1ccccc1)Nc1cccc(NC(=O)C(=O)NC[C@H]2CCCCO2)c1 ZINC000147356570 GF On-Demand Anodyne KCNK3 47 41 C[C@@H]1OCC[C@@H]1Nc1ccc2c(c1)Cc1ccccc1-2 ZINC000147356579 CH For-Sale Anodyne GALE 0 40 CCCCNC(=O)N1CC[C@@H](N)[C@H](CC)C1 ZINC000147356610 BD On-Demand Anodyne ASAH1 59 32 C[C@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147356612 BD On-Demand Anodyne SLC15A2 0 40 N#Cc1ccc(N2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147356709 FG On-Demand Mild SMO 17 47 N#Cc1ccc(N2CCN(C(=O)[C@@H]3C[C@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147356709 FG On-Demand Mild NPBWR1 66 40 Cc1nc2cc([C@@H]3CCCCN3C(=O)c3ccccc3NS(C)(=O)=O)nn2c(C)c1C ZINC000147356749 IG Annotated Anodyne COLA 78 39 Cc1nc2cc([C@@H]3CCCCN3C(=O)c3ccccc3NS(C)(=O)=O)nn2c(C)c1C ZINC000147356749 IG Annotated Anodyne CPT1A 76 39 COc1nn(-c2ccccc2)c2cc(N3CCN(c4ccncc4)CC3)ccc12 ZINC000147356792 GH Annotated Anodyne KHK 0 71 CCCCNC(=O)N1CC[C@H](N)[C@@H](CC)C1 ZINC000147356793 BD On-Demand Anodyne ASAH1 59 32 O=C(NC1CC1)c1ccc(-c2cnc3c(NCC4CC4)nccn23)cc1 ZINC000147356809 EG Annotated Anodyne MAPK11 26 43 O=C(NC1CC1)c1ccc(-c2cnc3c(NCC4CC4)nccn23)cc1 ZINC000147356809 EG Annotated Anodyne MAPK14 26 43 O=C(NC1CC1)c1ccc(-c2cnc3c(NCC4CC4)nccn23)cc1 ZINC000147356809 EG Annotated Anodyne IKBKB 22 43 O=C(NC1CC1)c1ccc(-c2cnc3c(NCC4CC4)nccn23)cc1 ZINC000147356809 EG Annotated Anodyne MAPK13 88 34 O=C(NC1CC1)c1ccc(-c2cnc3c(NCC4CC4)nccn23)cc1 ZINC000147356809 EG Annotated Anodyne MAPKAPK5 38 40 O=C(NC1CC1)c1ccc(-c2cnc3c(NCC4CC4)nccn23)cc1 ZINC000147356809 EG Annotated Anodyne TTK 56 49 C[C@@H](NC(=O)C1[C@H]2CCCC[C@H]12)C(=O)O ZINC000147356817 BD On-Demand Anodyne SLC15A2 0 40 CCCCCCCCn1c(C(C)C)nc2cc(N)ccc21 ZINC000147356855 CK For-Sale Mild TLR8 0 40 CN(CC(=O)O)S(=O)(=O)Cc1cccc(C(F)(F)F)c1 ZINC000147356893 DD On-Demand Anodyne TACR1 22 42 C=CCOc1ccccc1CNCC(F)F ZINC000147356909 BF On-Demand Mild PHES 0 57 N#Cc1ccc(N2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147356915 FG On-Demand Mild SSTR1 15 44 N#Cc1ccc(N2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147356915 FG On-Demand Mild SMO 15 47 N#Cc1ccc(N2CCN(C(=O)[C@@H]3C[C@@H]3c3cccc(Cl)c3)CC2)nc1 ZINC000147356915 FG On-Demand Mild NPBWR1 66 40 COCc1nc(C(=O)N2CCN(CC(=O)NC(C)C)CC2)cs1 ZINC000147356933 EC On-Demand Anodyne TRPC6 58 37 COCCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147356958 CE On-Demand Anodyne HRH2 17 40 COCCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147356958 CE On-Demand Anodyne CACNA1I 44 34 O=C(O)C1(NCc2nc(-c3ccccn3)no2)CCC1 ZINC000147356965 CD For-Sale Anodyne LUCI_PHOPE 26 45 CCCCNC(=O)N1CC[C@@H](N)[C@@H](CC)C1 ZINC000147356987 BD On-Demand Anodyne ASAH1 59 32 Cc1cccc(N2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357023 GG On-Demand Anodyne ADRB2 17 56 Cc1cccc(N2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357023 GG On-Demand Anodyne ADRB1 21 50 Cc1cccc(N2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357023 GG On-Demand Anodyne HTR1A 37 60 Cc1cccc(N2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357023 GG On-Demand Anodyne HTR2A 17 43 Cc1cccc(N2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357023 GG On-Demand Anodyne HTR2C 21 43 Cc1cccc(N2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357023 GG On-Demand Anodyne SLC6A4 30 60 Cc1cccc(N2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357023 GG On-Demand Anodyne ACOX1 34 44 Cc1cccc(N2CCN(C[C@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357023 GG On-Demand Anodyne ABCB1 89 65 C[C@H](NC(=O)C1[C@H]2CCCC[C@@H]12)C(=O)O ZINC000147357030 BD For-Sale Anodyne SLC15A2 0 40 CCCCCCCCn1c(CC)nc2cc(N)ccc21 ZINC000147357059 CJ For-Sale Mild HDAC10 17 41 CCCCCCCCn1c(CC)nc2cc(N)ccc21 ZINC000147357059 CJ For-Sale Mild HDAC1 0 45 CCCCCCCCn1c(CC)nc2cc(N)ccc21 ZINC000147357059 CJ For-Sale Mild HDAC4 18 41 CCCCCCCCn1c(CC)nc2cc(N)ccc21 ZINC000147357059 CJ For-Sale Mild HDAC5 26 41 CCCCCCCCn1c(CC)nc2cc(N)ccc21 ZINC000147357059 CJ For-Sale Mild HDAC9 18 41 CCCCCCCCn1c(CC)nc2cc(N)ccc21 ZINC000147357059 CJ For-Sale Mild HDAC11 18 41 CCCCCCCCn1c(CC)nc2cc(N)ccc21 ZINC000147357059 CJ For-Sale Mild HDAC7 33 41 CCCCCCCCn1c(CC)nc2cc(N)ccc21 ZINC000147357059 CJ For-Sale Mild TLR8 0 43 Fc1cccc(Cn2cc(-c3ccccc3I)cn2)c1 ZINC000147357075 GI For-Sale Anodyne ADORA2B 19 47 Fc1cccc(Cn2cc(-c3ccccc3I)cn2)c1 ZINC000147357075 GI For-Sale Anodyne ALK 15 45 CC(C)CCCCNCc1ccccc1N ZINC000147357157 BG For-Sale Anodyne GPM3 0 48 O=C(Nc1cc(Br)cc(C(=O)O)c1)NC1CCCCCC1 ZINC000147357183 FH For-Sale Anodyne EPHX2 36 51 Cc1cccc(N2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357237 GG On-Demand Anodyne ADRB2 17 56 Cc1cccc(N2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357237 GG On-Demand Anodyne ADRB1 21 50 Cc1cccc(N2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357237 GG On-Demand Anodyne HTR1A 37 60 Cc1cccc(N2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357237 GG On-Demand Anodyne HTR2A 17 43 Cc1cccc(N2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357237 GG On-Demand Anodyne HTR2C 21 43 Cc1cccc(N2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357237 GG On-Demand Anodyne SLC6A4 30 60 Cc1cccc(N2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357237 GG On-Demand Anodyne ACOX1 34 44 Cc1cccc(N2CCN(C[C@@H](O)COc3cccc4[nH]ccc34)CC2)c1C ZINC000147357237 GG On-Demand Anodyne ABCB1 89 65 C[C@@H](NC(=O)C1[C@H]2CCCC[C@@H]12)C(=O)O ZINC000147357239 BD For-Sale Anodyne SLC15A2 0 40 O=C(CCCC1CCN(C(=O)c2cc3ccccc3s2)CC1)NO ZINC000147357267 EG For-Sale Mild AKR1C3 16 40 Cc1nc(-c2nc(C(=O)NCCCCC(=O)NO)cs2)cs1 ZINC000147357307 ED Annotated Mild HDAC8 20 43 Cc1nc(-c2nc(C(=O)NCCCCC(=O)NO)cs2)cs1 ZINC000147357307 ED Annotated Mild HDAC10 36 47 Cc1nc(-c2nc(C(=O)NCCCCC(=O)NO)cs2)cs1 ZINC000147357307 ED Annotated Mild HDAC1 28 48 Cc1nc(-c2nc(C(=O)NCCCCC(=O)NO)cs2)cs1 ZINC000147357307 ED Annotated Mild HDAC2 24 45 Cc1nc(-c2nc(C(=O)NCCCCC(=O)NO)cs2)cs1 ZINC000147357307 ED Annotated Mild HDAC4 19 41 Cc1nc(-c2nc(C(=O)NCCCCC(=O)NO)cs2)cs1 ZINC000147357307 ED Annotated Mild HDAC6 28 47 Cc1nc(-c2nc(C(=O)NCCCCC(=O)NO)cs2)cs1 ZINC000147357307 ED Annotated Mild HDAC9 43 41 Cc1nc(-c2nc(C(=O)NCCCCC(=O)NO)cs2)cs1 ZINC000147357307 ED Annotated Mild HDA106 0 44 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2nc(-c3ccccc3F)cs2)C1 ZINC000147357321 HH On-Demand Anodyne MPL 44 37 COCC[C@H](N)C(=O)NN1CCCCC1 ZINC000147357400 BB For-Sale Anodyne DPP7 45 37 CCOC(=O)c1cnn(-c2cccc(NC(=O)N3CCC[C@@H](OCC)C3)c2)c1C ZINC000147357432 HG On-Demand Anodyne P2RY12 50 40 CCOC(=O)c1cnn(-c2cccc(NC(=O)N3CCC[C@@H](OCC)C3)c2)c1C ZINC000147357432 HG On-Demand Anodyne P2RY14 43 33 O=C(Nc1cc(Cl)cc(C(=O)O)c1)NC1CCCCCC1 ZINC000147357449 DH For-Sale Anodyne EPHX2 57 63 O=C(Nc1cc(Cl)cc(C(=O)O)c1)NC1CCCCCC1 ZINC000147357449 DH For-Sale Anodyne CXCR3 15 51 Cc1ncoc1C(=O)N[C@H](C)C(=O)O ZINC000147357480 AC On-Demand Anodyne SLC15A1 40 32 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA2 90 44 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA6 17 41 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA1 78 44 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA7 61 43 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA13 27 41 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA5B 38 41 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA4 53 42 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA5A 33 41 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA14 47 43 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA12 61 46 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA9 71 46 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CAH_METTE 29 41 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CYNT 40 39 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne NCE103 26 40 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA15 17 41 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne MTCA1 15 41 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne CA 0 41 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne A6YCJ1_9METZ 23 41 C[C@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357506 CC On-Demand Anodyne Q5TU56_ANOGA 0 41 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2nc(-c3ccccc3F)cs2)C1 ZINC000147357507 HH On-Demand Anodyne MPL 44 37 CC(C)c1csc(NC(=O)NCC(=O)Nc2ccc(F)cc2)n1 ZINC000147357570 EG On-Demand Anodyne ROCK1 17 43 CC(C)c1csc(NC(=O)NCC(=O)Nc2ccc(F)cc2)n1 ZINC000147357570 EG On-Demand Anodyne F7 30 40 COCC[C@@H](N)C(=O)NN1CCCCC1 ZINC000147357601 BB For-Sale Anodyne DPP7 45 37 CC[C@H](NC(=O)[C@@H]1CCCO[C@H]1c1ccccc1)C(=O)O ZINC000147357625 CE On-Demand Anodyne ACE2 51 33 CC[C@H](NC(=O)[C@@H]1CCCO[C@H]1c1ccccc1)C(=O)O ZINC000147357625 CE On-Demand Anodyne XIAP 49 32 CC[C@H](NC(=O)[C@@H]1CCCO[C@H]1c1ccccc1)C(=O)O ZINC000147357625 CE On-Demand Anodyne BIRC2 45 32 CCOC(=O)c1cnn(-c2cccc(NC(=O)N3CCC[C@H](OCC)C3)c2)c1C ZINC000147357678 HG On-Demand Anodyne P2RY12 50 40 CCOC(=O)c1cnn(-c2cccc(NC(=O)N3CCC[C@H](OCC)C3)c2)c1C ZINC000147357678 HG On-Demand Anodyne P2RY14 43 33 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA2 90 44 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA6 17 41 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA1 78 44 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA7 61 43 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA13 27 41 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA5B 38 41 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA4 53 42 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA5A 33 41 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA14 47 43 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA12 61 46 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA9 71 46 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CAH_METTE 29 41 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CYNT 40 39 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne NCE103 26 40 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA15 17 41 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne MTCA1 15 41 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne CA 0 41 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne A6YCJ1_9METZ 23 41 C[C@@H]1OCC[C@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357679 CC On-Demand Anodyne Q5TU56_ANOGA 0 41 CN(Cc1ccc(C(=O)O)cc1)C(=O)C1[C@H]2CCCC[C@H]12 ZINC000147357703 CF On-Demand Anodyne STAT5A 0 41 CCOC1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147357750 DG On-Demand Anodyne EPHX2 16 43 CCOC1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1 ZINC000147357750 DG On-Demand Anodyne MDM2 95 33 CC(C)(C)CC[C@H](c1ccc(C(=O)NCc2nn[nH]n2)cc1)N1C(=O)C(c2cccc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147357757 KK Annotated Anodyne GLP1R 16 73 O=S1(=O)N=C(N(CCBr)C2CCCC2)c2ccccc21 ZINC000147357776 FF For-Sale Reactive KCNA3 48 58 COc1nn(-c2ccccc2)c2cc(N3CC(N4CCNCC4)C3)ccc12 ZINC000147357828 FE Annotated Anodyne KHK 0 76 O=C(C[C@@H]1CCCNC1)NN1CCCCC1 ZINC000147357835 BC For-Sale Anodyne CPN1 0 40 CC[C@H](NC(=O)[C@H]1CCCO[C@H]1c1ccccc1)C(=O)O ZINC000147357856 CE On-Demand Anodyne ACE2 51 33 CC[C@H](NC(=O)[C@H]1CCCO[C@H]1c1ccccc1)C(=O)O ZINC000147357856 CE On-Demand Anodyne XIAP 49 32 CC[C@H](NC(=O)[C@H]1CCCO[C@H]1c1ccccc1)C(=O)O ZINC000147357856 CE On-Demand Anodyne BIRC2 45 32 O=C(NCc1cccs1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147357895 DG On-Demand Anodyne PPIA 16 41 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA2 90 44 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA6 17 41 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA1 78 44 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA7 61 43 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA13 27 41 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA5B 38 41 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA4 53 42 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA5A 33 41 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA14 47 43 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA12 61 46 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA9 71 46 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CAH_METTE 29 41 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CYNT 40 39 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne NCE103 26 40 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA15 17 41 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne MTCA1 15 41 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne CA 0 41 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne A6YCJ1_9METZ 23 41 C[C@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147357902 CC On-Demand Anodyne Q5TU56_ANOGA 0 41 CN(Cc1ccc(C(=O)O)cc1)C(=O)C1[C@H]2CCCC[C@@H]12 ZINC000147357932 CF For-Sale Anodyne STAT5A 0 41 COc1ccc(CCNc2cc(Cl)ccc2Br)cc1 ZINC000147357956 EJ For-Sale Anodyne PTGDR 28 41 COCc1nc(C(=O)NCC2(N(C)C)CCCCCC2)cs1 ZINC000147357979 EF On-Demand Anodyne SLC6A5 15 44 Cc1[nH]c2cc([C@@H]3CCCCN3C(=O)c3ccccc3O)nn2c(=O)c1C ZINC000147357985 FF Annotated Anodyne COLA 44 36 Cc1[nH]c2cc([C@@H]3CCCCN3C(=O)c3ccccc3O)nn2c(=O)c1C ZINC000147357985 FF Annotated Anodyne CPT1A 43 36 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(S(=O)(=O)N3CCCCC3)cc2)C1 ZINC000147358018 HE On-Demand Anodyne PKM 15 41 O=C(CNC(=O)Nc1cnc(-c2ccccc2)nc1)Nc1ccc(F)cc1 ZINC000147358045 FG On-Demand Anodyne ROCK2 16 41 O=C(CNC(=O)Nc1cnc(-c2ccccc2)nc1)Nc1ccc(F)cc1 ZINC000147358045 FG On-Demand Anodyne MTOR 16 40 O=C(CNC(=O)Nc1cnc(-c2ccccc2)nc1)Nc1ccc(F)cc1 ZINC000147358045 FG On-Demand Anodyne PRMT3 19 40 O=C(CNC(=O)Nc1cnc(-c2ccccc2)nc1)Nc1ccc(F)cc1 ZINC000147358045 FG On-Demand Anodyne NAMPT 26 40 O=C(C[C@H]1CCCNC1)NN1CCCCC1 ZINC000147358051 BC For-Sale Anodyne CPN1 0 40 CCOc1ccccc1CNC1(C(=O)O)CCC1 ZINC000147358110 BE For-Sale Anodyne HCN1 55 38 CCOc1ccccc1CNC1(C(=O)O)CCC1 ZINC000147358110 BE For-Sale Anodyne HCN4 47 37 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA2 90 44 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA6 17 41 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA1 78 44 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA7 61 43 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA13 27 41 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA5B 38 41 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA4 53 42 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA5A 33 41 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA14 47 43 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA12 61 46 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA9 71 46 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CAH_METTE 29 41 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CYNT 40 39 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne NCE103 26 40 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA15 17 41 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne MTCA1 15 41 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne CA 0 41 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne A6YCJ1_9METZ 23 41 C[C@@H]1OCC[C@@H]1NCc1ccc(S(N)(=O)=O)cc1 ZINC000147358116 CC On-Demand Anodyne Q5TU56_ANOGA 0 41 CN(Cc1ccc(C(=O)O)cc1)C(=O)C1[C@@H]2CCCC[C@@H]12 ZINC000147358148 CF On-Demand Anodyne STAT5A 0 41 O=C(c1ccc2ccccc2n1)N1CCC[C@H](CCBr)C1 ZINC000147358192 EH For-Sale Reactive SMO 40 39 CCO[C@H]1CCCN(S(=O)(=O)c2ccc(S(=O)(=O)N3CCCCC3)cc2)C1 ZINC000147358209 HE On-Demand Anodyne PKM 15 41 Cc1nn(-c2ccccc2)c(C)c1NC(=O)NCC(=O)Nc1ccc(F)cc1 ZINC000147358268 GG On-Demand Anodyne P2RX7 29 64 Cc1nn(-c2ccccc2)c(C)c1NC(=O)NCC(=O)Nc1ccc(F)cc1 ZINC000147358268 GG On-Demand Anodyne FPR2 53 38 COc1ccc(C)cc1NC(=O)CN(Cc1cccc(Cl)c1)S(=O)(=O)c1ccc(C)cc1 ZINC000147358282 JJ In-Stock Anodyne BMP1 41 41 COc1ccc(C)cc1NC(=O)CN(Cc1cccc(Cl)c1)S(=O)(=O)c1ccc(C)cc1 ZINC000147358282 JJ In-Stock Anodyne MMP2 19 47 COc1ccc(C)cc1NC(=O)CN(Cc1cccc(Cl)c1)S(=O)(=O)c1ccc(C)cc1 ZINC000147358282 JJ In-Stock Anodyne MMP8 36 47 COc1ccc(C)cc1NC(=O)CN(Cc1cccc(Cl)c1)S(=O)(=O)c1ccc(C)cc1 ZINC000147358282 JJ In-Stock Anodyne MMP9 23 48 COc1ccc(C)cc1NC(=O)CN(Cc1cccc(Cl)c1)S(=O)(=O)c1ccc(C)cc1 ZINC000147358282 JJ In-Stock Anodyne KCNMA1 17 42 COc1ccc(C)cc1NC(=O)CN(Cc1cccc(Cl)c1)S(=O)(=O)c1ccc(C)cc1 ZINC000147358282 JJ In-Stock Anodyne MMP1 27 47 COc1ccc(C)cc1NC(=O)CN(Cc1cccc(Cl)c1)S(=O)(=O)c1ccc(C)cc1 ZINC000147358282 JJ In-Stock Anodyne DAGLA 29 45 CCCCCCCCN1[C@H]2CC[C@H]1CC(=O)C2 ZINC000147358286 BH On-Demand Mild GBA2 45 32 CCCCCCCCN1[C@H]2CC[C@H]1CC(=O)C2 ZINC000147358286 BH On-Demand Mild LASR 53 36 CCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147358297 CG On-Demand Anodyne PPARA 24 40 CCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147358297 CG On-Demand Anodyne CACNA1I 55 35 Fc1ccc(F)c(Cn2cc(-c3ccccc3I)cn2)c1 ZINC000147358395 GI For-Sale Anodyne ALK 15 56 CCc1cccc(Cc2cnc(NC(=O)COc3ccc(C(N)=O)cc3)s2)c1 ZINC000147358404 GG On-Demand Anodyne SCD1 43 46 CCc1cccc(Cc2cnc(NC(=O)COc3ccc(C(N)=O)cc3)s2)c1 ZINC000147358404 GG On-Demand Anodyne SCD 41 50 Cc1cc(OCC(=O)NC2CCCC2)ccc1S(N)(=O)=O ZINC000147358423 DD For-Sale Anodyne FAAH 24 40 Cc1cc(OCC(=O)NC2CCCC2)ccc1S(N)(=O)=O ZINC000147358423 DD For-Sale Anodyne EPHX2 23 42 Cc1cc(OCC(=O)NC2CCCC2)ccc1S(N)(=O)=O ZINC000147358423 DD For-Sale Anodyne LUXN 0 53 Cc1cc(OCC(=O)NC2CCCC2)ccc1S(N)(=O)=O ZINC000147358423 DD For-Sale Anodyne ADIPOR1 0 40 Cc1cc(OCC(=O)NC2CCCC2)ccc1S(N)(=O)=O ZINC000147358423 DD For-Sale Anodyne ADIPOR2 0 40 O=C(c1ccc2ccccc2n1)N1CCC[C@@H](CCBr)C1 ZINC000147358424 EH For-Sale Reactive SMO 40 39 CCc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147358437 FE Annotated Mild HDA106 0 41 Cc1cc(NC(=O)c2cccc3c2OCCN3)ccn1 ZINC000147358465 CE For-Sale Anodyne TYK2 52 34 Cc1cc(NC(=O)c2cccc3c2OCCN3)ccn1 ZINC000147358465 CE For-Sale Anodyne KCNK3 76 36 Cc1cc(NC(=O)c2cccc3c2OCCN3)ccn1 ZINC000147358465 CE For-Sale Anodyne KCNK9 66 35 C[C@@H]1CCCN(Cc2csc(NC(=O)NCC(=O)Nc3ccc(F)cc3)n2)C1 ZINC000147358524 HG On-Demand Anodyne CCR3 114 43 Cc1cc(C(=O)N[C@@H]2CCOc3ccccc32)cc([N+](=O)[O-])c1 ZINC000147358543 DG On-Demand Bother LUXR 25 41 CNc1cn2ccnc2c(Oc2cccc(Cl)c2Cl)n1 ZINC000147358589 DH For-Sale Anodyne HIVRT 0 46 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccnc2N2CCOCC2)C1 ZINC000147358695 HD On-Demand Anodyne MTOR 47 34 Cc1cc(C(=O)N[C@H]2CCOc3ccccc32)cc([N+](=O)[O-])c1 ZINC000147358722 DG On-Demand Bother LUXR 25 41 O=C(c1ccc([N+](=O)[O-])cc1)N1CCC[C@H](CCBr)C1 ZINC000147358731 EG For-Sale Reactive L3MBTL3 51 38 C[C@H]1CCCN(Cc2csc(NC(=O)NCC(=O)Nc3ccc(F)cc3)n2)C1 ZINC000147358747 HG On-Demand Anodyne CCR3 114 43 CN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147358783 CF On-Demand Anodyne CACNA1I 49 34 O=C(Cc1ccc(F)cc1Cl)[C@@H]1COc2ccccc21 ZINC000147358792 CH For-Sale Anodyne P2RX7 50 42 CCCCCCC[C@@H](Cc1ccc(F)c(F)c1)NCC ZINC000147358802 CJ For-Sale Mild Q6UB75_PIG 0 50 COc1ccc(CCCN(C)C(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147358830 GI On-Demand Anodyne NPBWR1 60 41 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147358835 CE On-Demand Anodyne DRD4 42 32 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147358835 CE On-Demand Anodyne CCKAR 23 42 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147358835 CE On-Demand Anodyne CCR3 33 52 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147358835 CE On-Demand Anodyne MTNR1A 34 45 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147358835 CE On-Demand Anodyne MTNR1B 39 44 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147358835 CE On-Demand Anodyne CCKBR 0 42 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147358835 CE On-Demand Anodyne TAAR1 35 41 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147358835 CE On-Demand Anodyne LIMK2 34 46 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147358835 CE On-Demand Anodyne KCNK3 41 35 CCN(CC)CCOc1ccccc1NC(=O)C(=O)NC[C@@H]1CCCCO1 ZINC000147358899 GE On-Demand Anodyne AMY2 60 40 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccnc2N2CCOCC2)C1 ZINC000147358900 HD On-Demand Anodyne MTOR 47 34 CC(C)Oc1cccc(CC(=O)N[C@@H](CN2CCOCC2)c2ccccc2)c1 ZINC000147358910 GG On-Demand Anodyne CASR 51 41 CC(C)Oc1cccc(CC(=O)N[C@@H](CN2CCOCC2)c2ccccc2)c1 ZINC000147358910 GG On-Demand Anodyne TACR2 27 40 COc1ccc(CNCC(F)F)cc1Cl ZINC000147358922 BF On-Demand Anodyne PDE5A 26 44 COc1ccc(CNCC(F)F)cc1Cl ZINC000147358922 BF On-Demand Anodyne PDE6A 47 36 COc1ccc(CNCC(F)F)cc1Cl ZINC000147358922 BF On-Demand Anodyne TTR 0 41 Cc1nn(-c2ccccc2)c2cc(N3CC[C@@H](N)C3)ccc12 ZINC000147358931 CF Annotated Anodyne KHK 0 63 O=C(c1ccc([N+](=O)[O-])cc1)N1CCC[C@@H](CCBr)C1 ZINC000147358953 EG For-Sale Reactive L3MBTL3 51 38 COCc1nc(C(=O)N[C@@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147358959 FI On-Demand Anodyne MME 59 35 COCc1nc(C(=O)N[C@@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147358959 FI On-Demand Anodyne ANPEP 57 34 COCc1nc(C(=O)N[C@@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147358959 FI On-Demand Anodyne PAPA1_CARPA 43 35 COCc1nc(C(=O)N[C@@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147358959 FI On-Demand Anodyne CTSL 19 40 COCc1nc(C(=O)N[C@@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147358959 FI On-Demand Anodyne TACR3 44 37 COCc1nc(C(=O)N[C@@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147358959 FI On-Demand Anodyne CAPNS1 47 32 COCc1nc(C(=O)N[C@@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147358959 FI On-Demand Anodyne CAPN1 42 36 O=C(Cc1ccc(F)cc1Cl)[C@H]1COc2ccccc21 ZINC000147358991 CH For-Sale Anodyne P2RX7 50 42 CCCCCCC[C@H](Cc1ccc(F)c(F)c1)NCC ZINC000147358995 CJ For-Sale Mild Q6UB75_PIG 0 50 NC(=O)c1ccc(OCC(=O)Nc2ncc(Cc3cccc(F)c3)s2)cc1 ZINC000147359036 GF On-Demand Anodyne SCD1 42 46 NC(=O)c1ccc(OCC(=O)Nc2ncc(Cc3cccc(F)c3)s2)cc1 ZINC000147359036 GF On-Demand Anodyne SCD 40 48 Cc1cc(OCc2cccc(C#N)c2)ccc1S(N)(=O)=O ZINC000147359048 DE For-Sale Mild MAOB 53 55 Cc1cc(OCc2cccc(C#N)c2)ccc1S(N)(=O)=O ZINC000147359048 DE For-Sale Mild ADAMTS4 22 50 Cc1cc(OCc2cccc(C#N)c2)ccc1S(N)(=O)=O ZINC000147359048 DE For-Sale Mild FFAR1 48 39 CCN(CC)CCOc1ccccc1NC(=O)C(=O)NC[C@H]1CCCCO1 ZINC000147359050 GE On-Demand Anodyne AMY2 60 40 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147359073 CE On-Demand Anodyne DRD4 42 32 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147359073 CE On-Demand Anodyne CCKAR 23 42 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147359073 CE On-Demand Anodyne CCR3 33 52 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147359073 CE On-Demand Anodyne MTNR1A 34 45 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147359073 CE On-Demand Anodyne MTNR1B 39 44 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147359073 CE On-Demand Anodyne CCKBR 0 42 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147359073 CE On-Demand Anodyne TAAR1 35 41 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147359073 CE On-Demand Anodyne LIMK2 34 46 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147359073 CE On-Demand Anodyne KCNK3 41 35 Cc1nn(-c2ccccc2)c2cc(N3CC[C@H](N)C3)ccc12 ZINC000147359105 CF Annotated Anodyne KHK 0 63 CC(C)Oc1cccc(CC(=O)N[C@H](CN2CCOCC2)c2ccccc2)c1 ZINC000147359144 GG On-Demand Anodyne CASR 51 41 CC(C)Oc1cccc(CC(=O)N[C@H](CN2CCOCC2)c2ccccc2)c1 ZINC000147359144 GG On-Demand Anodyne TACR2 27 40 COCc1nc(C(=O)N[C@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147359163 FI On-Demand Anodyne MME 59 35 COCc1nc(C(=O)N[C@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147359163 FI On-Demand Anodyne ANPEP 57 34 COCc1nc(C(=O)N[C@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147359163 FI On-Demand Anodyne PAPA1_CARPA 43 35 COCc1nc(C(=O)N[C@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147359163 FI On-Demand Anodyne CTSL 19 40 COCc1nc(C(=O)N[C@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147359163 FI On-Demand Anodyne TACR3 44 37 COCc1nc(C(=O)N[C@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147359163 FI On-Demand Anodyne CAPNS1 47 32 COCc1nc(C(=O)N[C@H](Cc2ccccc2)c2ccccc2)cs1 ZINC000147359163 FI On-Demand Anodyne CAPN1 42 36 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359258 CE On-Demand Anodyne DRD4 42 32 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359258 CE On-Demand Anodyne CCKAR 23 42 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359258 CE On-Demand Anodyne CCR3 33 52 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359258 CE On-Demand Anodyne MTNR1A 34 45 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359258 CE On-Demand Anodyne MTNR1B 39 44 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359258 CE On-Demand Anodyne CCKBR 0 42 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359258 CE On-Demand Anodyne TAAR1 35 41 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359258 CE On-Demand Anodyne LIMK2 34 46 CC[C@@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359258 CE On-Demand Anodyne KCNK3 41 35 COc1nn(-c2ccccc2)c2cc(N3CCN(C4CNC4)CC3)ccc12 ZINC000147359317 FE Annotated Anodyne KHK 0 82 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc3c1OCO3)C2 ZINC000147359325 EE On-Demand Anodyne EDNRB 45 35 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc3c1OCO3)C2 ZINC000147359325 EE On-Demand Anodyne MTNR1A 45 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1cccc3c1OCO3)C2 ZINC000147359325 EE On-Demand Anodyne ROCK2 26 41 NCC1[C@H]2CC[C@H]1CN(Cc1ccccc1)C2 ZINC000147359340 BE For-Sale Anodyne DRD2 15 43 NCC1[C@H]2CC[C@H]1CN(Cc1ccccc1)C2 ZINC000147359340 BE For-Sale Anodyne ACHE 22 46 NCC1[C@H]2CC[C@H]1CN(Cc1ccccc1)C2 ZINC000147359340 BE For-Sale Anodyne DRD3 21 40 NCC1[C@H]2CC[C@H]1CN(Cc1ccccc1)C2 ZINC000147359340 BE For-Sale Anodyne SIGMAR1 61 47 CC(C)[C@H](NC(=O)c1csc(-c2cscn2)n1)C(=O)NCCCC(=O)NO ZINC000147359351 HD Annotated Mild HDAC3 32 70 CCn1cc(I)c(=O)n(Cc2ccc(F)cc2Cl)c1=O ZINC000147359379 HE For-Sale Anodyne P2RX7 57 41 CC[C@@H]1CCCCN1C(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147359437 FH For-Sale Anodyne ABHD11 0 40 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359484 CE On-Demand Anodyne DRD4 42 32 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359484 CE On-Demand Anodyne CCKAR 23 42 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359484 CE On-Demand Anodyne CCR3 33 52 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359484 CE On-Demand Anodyne MTNR1A 34 45 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359484 CE On-Demand Anodyne MTNR1B 39 44 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359484 CE On-Demand Anodyne CCKBR 0 42 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359484 CE On-Demand Anodyne TAAR1 35 41 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359484 CE On-Demand Anodyne LIMK2 34 46 CC[C@H]1CN(C(=O)Nc2cccc(OC)c2)CC[C@H]1N ZINC000147359484 CE On-Demand Anodyne KCNK3 41 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359498 FE On-Demand Anodyne ACACA 17 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359498 FE On-Demand Anodyne CTSK 41 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359498 FE On-Demand Anodyne F7 20 52 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359498 FE On-Demand Anodyne HDAC11 46 34 COCCOc1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1Cl ZINC000147359546 GH On-Demand Anodyne ROCK2 32 49 CN(C[C@H]1CCCN1C)C(=O)c1cccc2c1OCCN2 ZINC000147359605 CD For-Sale Anodyne CHRNA10 44 33 CN(C[C@H]1CCCN1C)C(=O)c1cccc2c1OCCN2 ZINC000147359605 CD For-Sale Anodyne ACKR3 54 36 COc1ccc(C)cc1CNC1(C(=O)O)CCC1 ZINC000147359639 BE On-Demand Anodyne QRFPR 40 34 CC[C@H]1CCCCN1C(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147359646 FH For-Sale Anodyne ABHD11 0 40 Cc1ncoc1C(=O)NCc1cc(C(=O)O)c(C)o1 ZINC000147359690 CD For-Sale Anodyne LIG1 0 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359705 FE On-Demand Anodyne ACACA 17 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359705 FE On-Demand Anodyne CTSK 41 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359705 FE On-Demand Anodyne F7 23 52 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359705 FE On-Demand Anodyne HDAC11 46 34 CN(C[C@@H]1CCCN1C)C(=O)c1cccc2c1OCCN2 ZINC000147359809 CD For-Sale Anodyne CHRNA10 44 33 CN(C[C@@H]1CCCN1C)C(=O)c1cccc2c1OCCN2 ZINC000147359809 CD For-Sale Anodyne ACKR3 54 36 COc1nn(-c2ccccc2)c2cc(-c3ccc(N4CCNCC4)cc3)ccc12 ZINC000147359824 GI Annotated Anodyne TGFBR1 0 47 COc1nn(-c2ccccc2)c2cc(-c3ccc(N4CCNCC4)cc3)ccc12 ZINC000147359824 GI Annotated Anodyne ACVR1 64 47 CC(C)CCCCN[C@@H]1CC[C@H](NC(=O)OC(C)(C)C)C1 ZINC000147359843 CH For-Sale Anodyne CTSK 22 40 CC(C)CCCCN[C@@H]1CC[C@H](NC(=O)OC(C)(C)C)C1 ZINC000147359843 CH For-Sale Anodyne PGA5 42 37 CC[C@@H]1CCCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147359855 DH On-Demand Anodyne CACNA1I 51 35 O=C(O)CCCCCCNC(=O)c1cccc(F)c1Cl ZINC000147359905 DG On-Demand Anodyne HDA106 0 44 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359906 FE On-Demand Anodyne ACACA 17 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359906 FE On-Demand Anodyne CTSK 41 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359906 FE On-Demand Anodyne F7 23 52 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147359906 FE On-Demand Anodyne HDAC11 46 34 CC(C)c1nc(NN)cc(OCc2cccc(Cl)c2)n1 ZINC000147359950 CG For-Sale Anodyne MAOB 27 44 COc1nn(-c2ccccc2)c2cc(N3CCN(C4CCNCC4)C3=O)ccc12 ZINC000147360009 GG Annotated Anodyne KHK 0 67 CC(C)CCCCN[C@H]1CC[C@H](NC(=O)OC(C)(C)C)C1 ZINC000147360045 CH For-Sale Anodyne CTSK 22 40 CC(C)CCCCN[C@H]1CC[C@H](NC(=O)OC(C)(C)C)C1 ZINC000147360045 CH For-Sale Anodyne PGA5 42 37 Nc1ccccc1CNCC(F)F ZINC000147360046 AD For-Sale Anodyne PHES 42 32 CC[C@H]1CCCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147360065 DH On-Demand Anodyne CACNA1I 51 35 CNC(=O)c1cc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)ccc1Cl ZINC000147360104 HE On-Demand Anodyne ENV 40 31 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147360113 FE On-Demand Anodyne ACACA 17 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147360113 FE On-Demand Anodyne CTSK 41 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147360113 FE On-Demand Anodyne F7 20 52 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(NC(=O)C2CC2)cc1 ZINC000147360113 FE On-Demand Anodyne HDAC11 46 34 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc2c(c1)C(=O)NC2=O ZINC000147360137 FG On-Demand Anodyne CASP3 0 44 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc2c(c1)C(=O)NC2=O ZINC000147360137 FG On-Demand Anodyne CASP2 23 44 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc2c(c1)C(=O)NC2=O ZINC000147360137 FG On-Demand Anodyne HRH3 0 43 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc2c(c1)C(=O)NC2=O ZINC000147360137 FG On-Demand Anodyne CDK4 36 45 O=C(O)CCCCCCNC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147360165 CF For-Sale Anodyne PLD1 15 46 O=C(O)CCCCCCNC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147360165 CF For-Sale Anodyne EPHX2 26 42 O=C(O)CCCCCCNC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147360165 CF For-Sale Anodyne HDA106 0 40 O=C(O)CCCCCCNC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147360165 CF For-Sale Anodyne NAMPT 17 48 O=C(O)CCCCCCNC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147360165 CF For-Sale Anodyne GPR88 0 42 CC(C)(C)[C@@H](CN1CCc2ccccc2C1)NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147360190 HF On-Demand Anodyne NOD1 29 40 CC(C)(C)[C@@H](CN1CCc2ccccc2C1)NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147360190 HF On-Demand Anodyne NOD2 47 43 CC[C@H](CNS(=O)(=O)c1ccc(F)c(Cl)c1)CC(=O)O ZINC000147360193 DE On-Demand Anodyne TBXA2R 47 38 CC[C@H](CNS(=O)(=O)c1ccc(F)c(Cl)c1)CC(=O)O ZINC000147360193 DE On-Demand Anodyne LEF 57 40 NNc1cc(OCc2cccc(Cl)c2)nc(C2CC2)n1 ZINC000147360200 CF For-Sale Anodyne MAOB 26 40 CCc1nn(-c2ccccc2)c2nc(N3CCN(c4cccnc4)CC3)ncc12 ZINC000147360220 GG Annotated Anodyne KHK 0 47 CC(C)CCCCN[C@@H]1CC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000147360262 CH For-Sale Anodyne CTSK 22 40 CC(C)CCCCN[C@@H]1CC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000147360262 CH For-Sale Anodyne PGA5 42 37 CCCCCCCC[C@@H](Cc1ccc(F)c(F)c1)NCC ZINC000147360293 CK For-Sale Mild Q6UB75_PIG 0 50 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(S(=O)(=O)N3CCCC3)cc2)C1 ZINC000147360305 HD On-Demand Anodyne PKM 18 42 CNC(=O)c1cc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)ccc1Cl ZINC000147360323 HE On-Demand Anodyne ENV 40 31 CCCC[C@H](NC(N)=O)C(=O)N(C)CC(=O)Nc1c(C)cc(C)cc1C ZINC000147360368 FE On-Demand Anodyne NOD1 66 32 CC[C@H](NC(=O)[C@@H](C)N1[C@@H](C)CC[C@@H]1C)C(=O)O ZINC000147360371 CD For-Sale Anodyne RIR1_HHV11 41 31 CC[C@H](NC(=O)[C@@H](C)N1[C@@H](C)CC[C@@H]1C)C(=O)O ZINC000147360371 CD For-Sale Anodyne ACE2 50 33 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCN(C)CC2)cc1C ZINC000147360376 HI On-Demand Anodyne LPL 45 38 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCN(C)CC2)cc1C ZINC000147360376 HI On-Demand Anodyne KCNQ2 63 36 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCN(C)CC2)cc1C ZINC000147360376 HI On-Demand Anodyne PRNP 20 40 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCN(C)CC2)cc1C ZINC000147360376 HI On-Demand Anodyne FLT3 17 46 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCN(C)CC2)cc1C ZINC000147360376 HI On-Demand Anodyne CSF1R 23 50 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCN(C)CC2)cc1C ZINC000147360376 HI On-Demand Anodyne MAPK7 18 40 O=C(O)CCCCCCNC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147360398 CF For-Sale Anodyne PLD1 15 46 O=C(O)CCCCCCNC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147360398 CF For-Sale Anodyne EPHX2 26 42 O=C(O)CCCCCCNC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147360398 CF For-Sale Anodyne HDA106 0 40 O=C(O)CCCCCCNC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147360398 CF For-Sale Anodyne NAMPT 17 48 O=C(O)CCCCCCNC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147360398 CF For-Sale Anodyne GPR88 0 42 CC[C@@H](CNS(=O)(=O)c1ccc(F)c(Cl)c1)CC(=O)O ZINC000147360400 DE On-Demand Anodyne TBXA2R 47 38 CC[C@@H](CNS(=O)(=O)c1ccc(F)c(Cl)c1)CC(=O)O ZINC000147360400 DE On-Demand Anodyne LEF 57 40 CC(C)(C)[C@H](CN1CCc2ccccc2C1)NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147360408 HF On-Demand Anodyne NOD1 29 40 CC(C)(C)[C@H](CN1CCc2ccccc2C1)NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147360408 HF On-Demand Anodyne NOD2 47 43 CC[C@H]1CN(C(=O)c2ccccc2SCC(=O)Nc2cccc(OC)c2)CCO1 ZINC000147360424 HH On-Demand Anodyne CASR 15 42 CC[C@H]1CN(C(=O)c2ccccc2SCC(=O)Nc2cccc(OC)c2)CCO1 ZINC000147360424 HH On-Demand Anodyne CCR3 16 48 CC[C@H]1CN(C(=O)c2ccccc2SCC(=O)Nc2cccc(OC)c2)CCO1 ZINC000147360424 HH On-Demand Anodyne MTNR1B 20 40 CC[C@H]1CN(C(=O)c2ccccc2SCC(=O)Nc2cccc(OC)c2)CCO1 ZINC000147360424 HH On-Demand Anodyne KCNK3 40 34 Cc1nn(-c2ccccc2)c2nc(C3CCN(C(=O)C4CCNCC4)CC3)nc(O)c12 ZINC000147360439 HF Annotated Anodyne KHK 0 51 CC(C)CCCCN[C@H]1CC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000147360476 CH For-Sale Anodyne CTSK 22 40 CC(C)CCCCN[C@H]1CC[C@@H](NC(=O)OC(C)(C)C)C1 ZINC000147360476 CH For-Sale Anodyne PGA5 42 37 CCCCCCCC[C@H](Cc1ccc(F)c(F)c1)NCC ZINC000147360493 CK For-Sale Mild Q6UB75_PIG 0 50 CN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CCCC1 ZINC000147360495 CG On-Demand Anodyne CACNA1I 41 33 CCO[C@H]1CCCN(S(=O)(=O)c2ccc(S(=O)(=O)N3CCCC3)cc2)C1 ZINC000147360506 HD On-Demand Anodyne PKM 18 42 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne DHODH 15 42 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne P2RY12 30 44 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne F10 23 42 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne KIT 20 47 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne JUN 24 40 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne LCK 31 41 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne ATF1 60 41 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne KDR 28 43 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne MTTP 41 32 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne NFKB1 55 41 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne CSF1R 21 46 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne TEK 36 41 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne BTK 25 41 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne KCNK3 37 40 Cc1c(C(=O)Nc2ccc(Cl)cc2)cnn1-c1cccc(C(F)(F)F)c1 ZINC000147360543 GK On-Demand Anodyne PDS 20 48 CCCC[C@@H](NC(N)=O)C(=O)N(C)CC(=O)Nc1c(C)cc(C)cc1C ZINC000147360574 FE On-Demand Anodyne NOD1 66 32 CC[C@H](NC(=O)[C@H](C)N1[C@@H](C)CC[C@@H]1C)C(=O)O ZINC000147360583 CD For-Sale Anodyne RIR1_HHV11 41 31 CC[C@H](NC(=O)[C@H](C)N1[C@@H](C)CC[C@@H]1C)C(=O)O ZINC000147360583 CD For-Sale Anodyne ACE2 50 33 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147360589 CF For-Sale Anodyne PLD1 15 46 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147360589 CF For-Sale Anodyne EPHX2 26 42 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147360589 CF For-Sale Anodyne HDA106 0 40 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147360589 CF For-Sale Anodyne NAMPT 17 48 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147360589 CF For-Sale Anodyne GPR88 0 42 Cc1nc(N)sc1C(=O)NN1CCCCC1 ZINC000147360608 BD For-Sale Anodyne CNR1 15 40 Cc1nn(-c2ccccc2)c2nc(C3CCN([C@@H]4CCNC4)CC3)nc(O)c12 ZINC000147360627 GE Annotated Anodyne KHK 0 48 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360649 FG On-Demand Anodyne MME 40 35 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360649 FG On-Demand Anodyne ANPEP 41 33 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360649 FG On-Demand Anodyne CASR 49 38 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360649 FG On-Demand Anodyne TACR2 33 47 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360649 FG On-Demand Anodyne CAPN1 28 45 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360649 FG On-Demand Anodyne CAPN2 26 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360649 FG On-Demand Anodyne ACE2 69 35 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360649 FG On-Demand Anodyne PGA5 47 33 CC(=O)N[C@@H]1[C@@H](O)CN(C)C[C@H]1O ZINC000147360772 AA For-Sale Anodyne NA 45 36 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147360779 CF For-Sale Anodyne PLD1 15 46 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147360779 CF For-Sale Anodyne EPHX2 26 42 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147360779 CF For-Sale Anodyne HDA106 0 40 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147360779 CF For-Sale Anodyne NAMPT 17 48 O=C(O)CCCCCCNC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147360779 CF For-Sale Anodyne GPR88 0 42 O=C(O)C1(NCc2cc(=O)oc3cc(O)ccc23)CCC1 ZINC000147360798 CD For-Sale Anodyne HSD17B3 41 45 Brc1ccc(Br)c(-c2nc3ccccc3s2)c1 ZINC000147360805 FK For-Sale Anodyne LUCI_PHOPY 16 44 Brc1ccc(Br)c(-c2nc3ccccc3s2)c1 ZINC000147360805 FK For-Sale Anodyne LUCI_PHOPE 23 44 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360826 FG On-Demand Anodyne MME 40 35 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360826 FG On-Demand Anodyne ANPEP 41 33 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360826 FG On-Demand Anodyne CASR 49 38 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360826 FG On-Demand Anodyne TACR2 33 47 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360826 FG On-Demand Anodyne CAPN1 28 45 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360826 FG On-Demand Anodyne CAPN2 26 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360826 FG On-Demand Anodyne ACE2 69 35 C[C@H](Cc1cccc(F)c1)C(=O)N[C@@H](CN1CCOCC1)c1ccccc1 ZINC000147360826 FG On-Demand Anodyne PGA5 47 33 Cc1nn(-c2ccccc2)c2nc(C3CCN([C@H]4CCNC4)CC3)nc(O)c12 ZINC000147360838 GE Annotated Anodyne KHK 0 48 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccc(F)cc1Cl)NO ZINC000147360921 JI Annotated Mild HDAC6 21 75 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne ESR1 82 40 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne ACHE 20 46 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne KCNH2 16 43 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne ESR2 59 41 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne LTA4H 58 47 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne HRH3 84 55 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne SIGMAR1 21 43 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne YES1 18 40 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne TNK2 19 40 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne PSMB2 62 49 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne PSMB5 22 52 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne PSMB1 55 52 Cc1cc(OCCN2CCCCC2)ccc1S(N)(=O)=O ZINC000147360953 CD For-Sale Anodyne TBK1 16 40 Cc1ccc(C(=O)NCCCCCCC(=O)O)cc1Br ZINC000147360954 EH On-Demand Anodyne HDAC10 17 41 Cc1ccc(C(=O)NCCCCCCC(=O)O)cc1Br ZINC000147360954 EH On-Demand Anodyne HDAC1 21 45 Cc1ccc(C(=O)NCCCCCCC(=O)O)cc1Br ZINC000147360954 EH On-Demand Anodyne HDAC2 18 45 Cc1ccc(C(=O)NCCCCCCC(=O)O)cc1Br ZINC000147360954 EH On-Demand Anodyne HDAC3 21 45 Cc1ccc(C(=O)NCCCCCCC(=O)O)cc1Br ZINC000147360954 EH On-Demand Anodyne HDAC4 18 45 Cc1ccc(C(=O)NCCCCCCC(=O)O)cc1Br ZINC000147360954 EH On-Demand Anodyne HDAC5 20 42 Cc1ccc(C(=O)NCCCCCCC(=O)O)cc1Br ZINC000147360954 EH On-Demand Anodyne HDAC6 20 45 Cc1ccc(C(=O)NCCCCCCC(=O)O)cc1Br ZINC000147360954 EH On-Demand Anodyne HDAC9 33 41 Cc1ccc(C(=O)NCCCCCCC(=O)O)cc1Br ZINC000147360954 EH On-Demand Anodyne HDA106 0 49 CN(Cc1cscn1)C(=O)N[C@@H](CCCc1ccccc1)c1ccccc1 ZINC000147360960 GK On-Demand Anodyne BMP1 51 36 CN(Cc1cscn1)C(=O)N[C@@H](CCCc1ccccc1)c1ccccc1 ZINC000147360960 GK On-Demand Anodyne CYP3A4 21 47 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361020 FG On-Demand Anodyne MME 40 35 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361020 FG On-Demand Anodyne ANPEP 41 33 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361020 FG On-Demand Anodyne CASR 49 38 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361020 FG On-Demand Anodyne TACR2 33 47 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361020 FG On-Demand Anodyne CAPN1 28 45 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361020 FG On-Demand Anodyne CAPN2 26 40 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361020 FG On-Demand Anodyne ACE2 69 35 C[C@@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361020 FG On-Demand Anodyne PGA5 47 33 Cc1nn(-c2ccccc2)c2nc(C3CCN(C4CCNCC4)CC3)nc(O)c12 ZINC000147361036 GF Annotated Anodyne KHK 0 52 CC[C@H]1CN(C(=O)c2cccc(NS(=O)(=O)c3ccc(F)c(F)c3)c2)CCO1 ZINC000147361091 HG On-Demand Anodyne TRY2_BOVIN 54 33 CC[C@H]1CN(C(=O)c2cccc(NS(=O)(=O)c3ccc(F)c(F)c3)c2)CCO1 ZINC000147361091 HG On-Demand Anodyne ST14 40 32 CC[C@H]1CN(C(=O)c2cccc(NS(=O)(=O)c3ccc(F)c(F)c3)c2)CCO1 ZINC000147361091 HG On-Demand Anodyne SFRP1 52 34 CC[C@H]1CN(C(=O)c2cccc(NS(=O)(=O)c3ccc(F)c(F)c3)c2)CCO1 ZINC000147361091 HG On-Demand Anodyne WNT3 53 34 O=S(=O)(Nc1nnc(Cc2ccc(Cl)cc2)s1)c1ccc(F)c(Cl)c1 ZINC000147361125 HI On-Demand Anodyne CA2 36 46 O=S(=O)(Nc1nnc(Cc2ccc(Cl)cc2)s1)c1ccc(F)c(Cl)c1 ZINC000147361125 HI On-Demand Anodyne CA1 37 46 O=S(=O)(Nc1nnc(Cc2ccc(Cl)cc2)s1)c1ccc(F)c(Cl)c1 ZINC000147361125 HI On-Demand Anodyne CA4 60 46 O=S(=O)(Nc1nnc(Cc2ccc(Cl)cc2)s1)c1ccc(F)c(Cl)c1 ZINC000147361125 HI On-Demand Anodyne CA9 17 46 O=S(=O)(Nc1nnc(Cc2ccc(Cl)cc2)s1)c1ccc(F)c(Cl)c1 ZINC000147361125 HI On-Demand Anodyne A6YCJ1_9METZ 24 45 CN(Cc1cscn1)C(=O)N[C@H](CCCc1ccccc1)c1ccccc1 ZINC000147361153 GK On-Demand Anodyne BMP1 51 36 CN(Cc1cscn1)C(=O)N[C@H](CCCc1ccccc1)c1ccccc1 ZINC000147361153 GK On-Demand Anodyne CYP3A4 21 47 CC(=O)N[C@H]1[C@@H](O)CN(C)C[C@H]1O ZINC000147361177 AA For-Sale Anodyne NA 45 36 CN(C)C(=O)NCCn1c(CCCl)nc2ccccc21 ZINC000147361192 CE For-Sale Reactive HDAC1 15 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361219 FG On-Demand Anodyne MME 40 35 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361219 FG On-Demand Anodyne ANPEP 41 33 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361219 FG On-Demand Anodyne CASR 49 38 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361219 FG On-Demand Anodyne TACR2 33 47 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361219 FG On-Demand Anodyne CAPN1 28 45 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361219 FG On-Demand Anodyne CAPN2 26 40 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361219 FG On-Demand Anodyne ACE2 69 35 C[C@H](Cc1cccc(F)c1)C(=O)N[C@H](CN1CCOCC1)c1ccccc1 ZINC000147361219 FG On-Demand Anodyne PGA5 47 33 CCc1nn(-c2ccccc2)c2nc(C3CCNCC3)nc(O)c12 ZINC000147361249 DF Annotated Anodyne KHK 0 48 NCC(=O)NCC(=O)NN1CCCCC1 ZINC000147361253 BA For-Sale Anodyne UREB 0 48 CC[C@H](NC(=O)c1ccc(Br)c(Cl)c1)C(=O)O ZINC000147361258 DF On-Demand Anodyne CA2 30 52 CC[C@H](NC(=O)c1ccc(Br)c(Cl)c1)C(=O)O ZINC000147361258 DF On-Demand Anodyne CA4 22 52 CC[C@H](NC(=O)c1ccc(Br)c(Cl)c1)C(=O)O ZINC000147361258 DF On-Demand Anodyne KMO 0 41 CCCCCCCCOc1cc(N(C)C)ccc1N ZINC000147361304 CI For-Sale Mild THRA 56 38 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne PRCP 17 46 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne NPY1R 23 47 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne KLK3 71 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne CTSK 32 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne NPFFR2 41 38 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne C3AR1 56 36 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne HLA-DRB1 46 41 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne SOAT1 25 44 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne PCSK5 41 34 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne FURIN 59 33 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne CAPN2 45 34 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne POLG_WNV 83 35 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne UTS2 40 42 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361308 FH On-Demand Anodyne NPFFR1 56 38 CC[C@H]1CN(C(=O)c2cc(S(=O)(=O)N3CCOCC3)ccc2F)CCO1 ZINC000147361322 GD On-Demand Anodyne CNR1 18 41 CC[C@H]1CN(C(=O)c2cc(S(=O)(=O)N3CCOCC3)ccc2F)CCO1 ZINC000147361322 GD On-Demand Anodyne CNR2 19 41 CC[C@H]1CN(C(=O)c2cc(S(=O)(=O)N3CCOCC3)ccc2F)CCO1 ZINC000147361322 GD On-Demand Anodyne PKM 41 38 O=C(O)CCCCCCNC(=O)C1[C@@H]2CCCC[C@@H]12 ZINC000147361347 CF On-Demand Anodyne EPHX2 23 44 Cc1cc(OCC2(CC#N)CC2)ccc1S(N)(=O)=O ZINC000147361381 CD For-Sale Mild TRPV4 44 34 NC(=O)c1ccsc1NC(=O)CNC1(C(=O)O)CCC1 ZINC000147361409 CC For-Sale Anodyne MAPK8 26 52 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccc([N+](=O)[O-])cc1)NO ZINC000147361415 IG Annotated Mild HDAC6 19 77 O=C(O)c1sc(O)c2ncccc12 ZINC000147361416 AD For-Sale Anodyne KDM4A 0 51 O=C(O)c1sc(O)c2ncccc12 ZINC000147361416 AD For-Sale Anodyne KDM4C 0 51 O=C(O)c1sc(O)c2ncccc12 ZINC000147361416 AD For-Sale Anodyne KDM4E 15 51 O=C(O)c1sc(O)c2ncccc12 ZINC000147361416 AD For-Sale Anodyne KDM3A 0 51 O=C(O)c1sc(O)c2ncccc12 ZINC000147361416 AD For-Sale Anodyne KDM6B 0 51 O=C(O)c1sc(O)c2ncccc12 ZINC000147361416 AD For-Sale Anodyne FTO 0 51 CC(=O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147361421 CD On-Demand Anodyne CCR3 29 46 CC(=O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147361421 CD On-Demand Anodyne GUAB 0 48 CC(=O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147361421 CD On-Demand Anodyne EPHX2 15 41 CC(=O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147361421 CD On-Demand Anodyne AKR1C3 23 47 CC(=O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147361421 CD On-Demand Anodyne PRMT3 53 35 CC(=O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147361421 CD On-Demand Anodyne IMDH_CRYPV 42 37 CC(=O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147361421 CD On-Demand Anodyne PSBA 0 47 CC(=O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147361421 CD On-Demand Anodyne KCNK3 75 39 CC(=O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147361421 CD On-Demand Anodyne KCNK9 50 37 CC(=O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147361421 CD On-Demand Anodyne PARP10 0 42 O=C(Nc1[nH]ncc1Br)c1ccccc1Cl ZINC000147361435 DG On-Demand Anodyne BDKRB1 18 55 O=C(Nc1[nH]ncc1Br)c1ccccc1Cl ZINC000147361435 DG On-Demand Anodyne EPHB3 43 37 O=C(Nc1[nH]ncc1Br)c1ccccc1Cl ZINC000147361435 DG On-Demand Anodyne NR2E3 66 36 O=C(Nc1[nH]ncc1Br)c1ccccc1Cl ZINC000147361435 DG On-Demand Anodyne SMO 26 45 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne PRCP 17 46 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne NPY1R 23 47 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne KLK3 71 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne CTSK 32 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne NPFFR2 41 38 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne C3AR1 56 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne HLA-DRB1 46 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne SOAT1 25 44 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne PCSK5 41 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne FURIN 59 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne CAPN2 45 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne POLG_WNV 83 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne UTS2 40 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361473 FH On-Demand Anodyne NPFFR1 56 38 Nc1cc2ccccc2cc1C(=O)NN1CCCCC1 ZINC000147361477 CF For-Sale Anodyne CNR1 50 31 CCc1nn(-c2ccccc2)c2nc(C3CCN([C@@H]4CCNC4)CC3)nc(O)c12 ZINC000147361478 GF Annotated Anodyne KHK 0 55 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne ACE 57 43 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne MME 93 43 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne LTA4H 40 36 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne ANPEP 68 40 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne KCNA5 0 41 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne CCKAR 50 43 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne CPA1 41 43 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne CCR3 29 40 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne PYGL 26 40 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne ECE1 43 36 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne CAPN1 43 43 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne CAPN2 64 35 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne ACE2 85 43 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne FPR1 45 35 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne NPR 57 34 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne SLC15A2 0 40 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne BLA1_STEMA 51 35 CCc1ccccc1C(=O)N[C@@H](CC)C(=O)O ZINC000147361506 BD On-Demand Anodyne DAC 40 39 CCCCCC(=O)OC=C(Cl)Cl ZINC000147361515 BG For-Sale Anodyne FABP5 15 41 CCCCCC(=O)OC=C(Cl)Cl ZINC000147361515 BG For-Sale Anodyne CQSS 59 36 COC(=O)c1ccc(O)c(NN)c1 ZINC000147361518 AC For-Sale Anodyne CA7 23 52 COC(=O)c1ccc(O)c(NN)c1 ZINC000147361518 AC For-Sale Anodyne CA14 28 52 C=Cc1ccc(S(=O)(=O)N[C@H](C)C(=O)OC)cc1 ZINC000147361523 CD On-Demand Anodyne MMP13 29 44 C=Cc1ccc(S(=O)(=O)N[C@H](C)C(=O)OC)cc1 ZINC000147361523 CD On-Demand Anodyne MMP2 26 49 C=Cc1ccc(S(=O)(=O)N[C@H](C)C(=O)OC)cc1 ZINC000147361523 CD On-Demand Anodyne MMP9 18 49 C=Cc1ccc(S(=O)(=O)N[C@H](C)C(=O)OC)cc1 ZINC000147361523 CD On-Demand Anodyne MMP12 18 43 C=Cc1ccc(S(=O)(=O)N[C@H](C)C(=O)OC)cc1 ZINC000147361523 CD On-Demand Anodyne MMP7 21 43 C=Cc1ccc(S(=O)(=O)N[C@H](C)C(=O)OC)cc1 ZINC000147361523 CD On-Demand Anodyne LEF 27 41 CC(=O)Nc1ccc(C)c(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)c1 ZINC000147361528 HG On-Demand Anodyne ROCK2 19 40 O=C(O)CCCCCCNC(=O)C1[C@H]2CCCC[C@@H]12 ZINC000147361549 CF For-Sale Anodyne EPHX2 23 44 CC(C)Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147361625 GF Annotated Mild MAP 0 40 CC(C)Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147361625 GF Annotated Mild MAP1 47 40 CC(C)Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147361625 GF Annotated Mild HDAC6 29 80 CCc1nn(-c2ccccc2)c2nc(C3CCN([C@H]4CCNC4)CC3)nc(O)c12 ZINC000147361657 GF Annotated Anodyne KHK 0 55 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne PRCP 17 46 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne NPY1R 23 47 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne KLK3 71 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne CTSK 32 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne NPFFR2 41 38 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne C3AR1 56 36 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne HLA-DRB1 46 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne SOAT1 25 44 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne PCSK5 41 34 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne FURIN 59 33 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne CAPN2 45 34 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne POLG_WNV 83 35 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne UTS2 40 42 CCCC[C@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361665 FH On-Demand Anodyne NPFFR1 56 38 O=C(c1csc(-c2ccccn2)n1)N1CCC(OCc2ccccc2)CC1 ZINC000147361677 GI On-Demand Anodyne GRIN2B 48 47 O=C(c1csc(-c2ccccn2)n1)N1CCC(OCc2ccccc2)CC1 ZINC000147361677 GI On-Demand Anodyne COLA 18 46 O=C(c1csc(-c2ccccn2)n1)N1CCC(OCc2ccccc2)CC1 ZINC000147361677 GI On-Demand Anodyne CPT1A 17 46 O=C(c1csc(-c2ccccn2)n1)N1CCC(OCc2ccccc2)CC1 ZINC000147361677 GI On-Demand Anodyne TRPC6 48 35 O=c1[nH]c([C@H](F)C(F)(F)F)nc2ccccc12 ZINC000147361678 BE For-Sale Anodyne TNKS 30 53 O=c1[nH]c([C@H](F)C(F)(F)F)nc2ccccc12 ZINC000147361678 BE For-Sale Anodyne TNKS2 21 53 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne ACE 40 42 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne OPRM1 26 43 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne OPRD1 28 46 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne MME 85 48 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne LTA4H 16 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne ANPEP 74 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne EDNRA 21 49 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne TACR1 29 52 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CTSD 46 48 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne HRAS 51 38 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne FCER2 71 39 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CASP3 44 67 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne BMP1 24 52 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne RNPEP 28 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CASP8 24 52 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne KLK3 127 71 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CTSB 104 68 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne PAPA1_CARPA 91 63 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CYSP_TRYCR 83 63 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CCKAR 15 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CTSK 78 72 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CTSL 67 62 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CPA1 27 40 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CACNA1B 45 37 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne PGA 35 46 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne F2R 17 45 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne NPFFR2 40 32 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne TIMP3 45 33 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne C3AR1 35 43 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne HLA-A 55 40 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CAPNS1 101 65 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne MMP2 25 44 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne MMP3 61 51 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne MMP8 26 45 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne MMP14 17 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne HLA-DRB1 85 48 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne REN 70 54 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne REN1 49 48 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne HDAC6 15 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne LNPEP 18 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne MMP11 65 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne TGM1 23 40 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CTSS 54 72 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne GHSR 19 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CAPN1 163 73 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne MMP9 35 45 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CASP1 49 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CAPN2 202 70 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne ACE2 62 38 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne PLAU 34 45 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CASP6 65 49 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CASP9 64 49 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne BACE1 15 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne POLG_HCV1 22 46 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne LAP3 30 45 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne TPSAB1 48 42 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne MMP1 40 46 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne FPR1 73 50 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne NPR 119 59 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne AMP1_PLAFQ 44 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne R1A_CVHSA 21 42 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne CASP10 38 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne NAAA 56 37 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne SIRT1 15 40 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne PSMB5 74 63 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne NPFFR1 40 32 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne Q9NAW4_PLAFA 57 40 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](C)CO ZINC000147361728 DD On-Demand Anodyne HPN 44 33 CCCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147361734 CG On-Demand Anodyne PPARA 32 41 CCCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147361734 CG On-Demand Anodyne CACNA1I 50 34 CC(=O)Nc1ccc(C)c(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)c1 ZINC000147361745 HG On-Demand Anodyne ROCK2 19 40 O=C(O)CCCCCCNC(=O)C1[C@H]2CCCC[C@H]12 ZINC000147361752 CF On-Demand Anodyne EPHX2 23 44 c1ccc(CSC2CCC2)cc1 ZINC000147361821 AG On-Demand Anodyne SLC18A2 38 42 c1ccc(CSC2CCC2)cc1 ZINC000147361821 AG On-Demand Anodyne QRFPR 40 40 CC(=O)c1ccc(NC(=O)NCCNC(=O)N(C)C)cc1 ZINC000147361838 CD On-Demand Anodyne PSBA 0 44 CCOc1ccc(OCCNC2(C(=O)O)CCC2)cc1 ZINC000147361842 CE For-Sale Anodyne LTA4H 17 40 CCOc1ccc(OCCNC2(C(=O)O)CCC2)cc1 ZINC000147361842 CE For-Sale Anodyne PLA2G4B 70 34 Cc1cc(OCCN2CCN(C)CC2)ccc1S(N)(=O)=O ZINC000147361845 DC For-Sale Anodyne LTA4H 46 47 Cc1cc(OCCN2CCN(C)CC2)ccc1S(N)(=O)=O ZINC000147361845 DC For-Sale Anodyne HRH3 38 44 Cc1cc(OCCN2CCN(C)CC2)ccc1S(N)(=O)=O ZINC000147361845 DC For-Sale Anodyne PSMB2 47 37 Cc1cc(OCCN2CCN(C)CC2)ccc1S(N)(=O)=O ZINC000147361845 DC For-Sale Anodyne PSMB1 42 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne PRCP 17 46 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne NPY1R 23 47 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne KLK3 71 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne CTSK 32 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne NPFFR2 41 38 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne C3AR1 56 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne HLA-DRB1 46 41 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne SOAT1 25 44 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne PCSK5 41 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne FURIN 59 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne CAPN2 45 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne POLG_WNV 83 35 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne UTS2 40 42 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](c1ccccc1)c1ccc(Cl)cc1 ZINC000147361873 FH On-Demand Anodyne NPFFR1 56 38 CCc1nn(-c2ccccc2)c2nc(C3CCN(C4CCNCC4)CC3)nc(O)c12 ZINC000147361882 HG Annotated Anodyne KHK 0 54 O=c1[nH]c([C@@H](F)C(F)(F)F)nc2ccccc12 ZINC000147361885 BE For-Sale Anodyne TNKS 30 53 O=c1[nH]c([C@@H](F)C(F)(F)F)nc2ccccc12 ZINC000147361885 BE For-Sale Anodyne TNKS2 21 53 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne ACE 40 42 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne OPRM1 26 43 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne OPRD1 28 46 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne MME 85 48 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne LTA4H 16 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne ANPEP 74 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne EDNRA 21 49 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne TACR1 29 52 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CTSD 46 48 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne HRAS 51 38 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne FCER2 71 39 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CASP3 44 67 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne BMP1 24 52 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne RNPEP 28 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CASP8 24 52 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne KLK3 127 71 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CTSB 104 68 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne PAPA1_CARPA 91 63 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CYSP_TRYCR 83 63 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CCKAR 15 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CTSK 78 72 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CTSL 67 62 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CPA1 27 40 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CACNA1B 45 37 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne PGA 35 46 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne F2R 17 45 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne NPFFR2 40 32 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne TIMP3 45 33 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne C3AR1 35 43 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne HLA-A 55 40 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CAPNS1 101 65 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne MMP2 25 44 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne MMP3 61 51 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne MMP8 26 45 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne MMP14 17 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne HLA-DRB1 85 48 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne REN 70 54 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne REN1 49 48 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne HDAC6 15 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne LNPEP 18 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne MMP11 65 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne TGM1 23 40 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CTSS 54 72 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne GHSR 19 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CAPN1 163 73 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne MMP9 35 45 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CASP1 49 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CAPN2 202 70 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne ACE2 62 38 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne PLAU 34 45 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CASP6 65 49 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CASP9 64 49 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne BACE1 15 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne POLG_HCV1 22 46 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne LAP3 30 45 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne TPSAB1 48 42 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne MMP1 40 46 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne FPR1 73 50 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne NPR 119 59 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne AMP1_PLAFQ 44 47 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne R1A_CVHSA 21 42 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne CASP10 38 41 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne NAAA 56 37 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne SIRT1 15 40 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne PSMB5 74 63 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne NPFFR1 40 32 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne Q9NAW4_PLAFA 57 40 CC(C)C[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@H](C)CO ZINC000147361936 DD On-Demand Anodyne HPN 44 33 CC(=O)Nc1ccc(C)c(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)c1 ZINC000147361937 HG On-Demand Anodyne CHRM3 15 41 CC(=O)Nc1ccc(C)c(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)c1 ZINC000147361937 HG On-Demand Anodyne CCR3 31 43 CNc1nc(Nc2cc(F)c(C(=O)N3CC[C@H](OC)C3)cc2OC)ncc1C(F)(F)F ZINC000147361977 IG Annotated Anodyne TTK 19 57 CNc1nc(Nc2cc(F)c(C(=O)N3CC[C@H](OC)C3)cc2OC)ncc1C(F)(F)F ZINC000147361977 IG Annotated Anodyne LRRK2 97 75 CCCCCCCCN1[C@H]2CC[C@H]1CC(NC)C2 ZINC000147361978 CH For-Sale Mild GBA2 42 33 CCO[C@@H]1CCCN(S(=O)(=O)c2cc(NC(C)=O)ccc2OC)C1 ZINC000147362023 FD On-Demand Anodyne TSHR 62 34 CCO[C@@H]1CCCN(S(=O)(=O)c2cc(NC(C)=O)ccc2OC)C1 ZINC000147362023 FD On-Demand Anodyne CPT1A 56 38 CCO[C@@H]1CCCN(S(=O)(=O)c2cc(NC(C)=O)ccc2OC)C1 ZINC000147362023 FD On-Demand Anodyne CPT2 49 38 CCO[C@@H]1CCCN(S(=O)(=O)c2cc(NC(C)=O)ccc2OC)C1 ZINC000147362023 FD On-Demand Anodyne CPT1B 52 36 Cc1cc(O[C@@H](C)C(=O)NC2CC2)ccc1S(N)(=O)=O ZINC000147362042 CC For-Sale Anodyne EPHX2 17 40 Cc1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147362059 BD For-Sale Anodyne ADRA1B 0 45 CC(C)(C)OC(=O)N1CCC(NCCc2c(Cl)ncnc2Cl)CC1 ZINC000147362075 GG For-Sale Anodyne GPR119 56 44 CCc1nn(-c2ccccc2)c2nc(C3CCN(C(=O)C4CCNCC4)CC3)nc(O)c12 ZINC000147362108 IF Annotated Anodyne KHK 0 47 CC(=O)Nc1ccc(C)c(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)c1 ZINC000147362119 HG On-Demand Anodyne CHRM3 15 41 CC(=O)Nc1ccc(C)c(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)c1 ZINC000147362119 HG On-Demand Anodyne CCR3 31 43 CNc1nc(Nc2cc(F)c(C(=O)N3CC[C@@H](OC)C3)cc2OC)ncc1C(F)(F)F ZINC000147362130 IG Annotated Anodyne TTK 19 57 CNc1nc(Nc2cc(F)c(C(=O)N3CC[C@@H](OC)C3)cc2OC)ncc1C(F)(F)F ZINC000147362130 IG Annotated Anodyne LRRK2 97 75 C[C@](N)(C(=O)NN1CCCCC1)c1ccccc1 ZINC000147362186 BD For-Sale Anodyne AMY2 56 34 C[C@](N)(C(=O)NN1CCCCC1)c1ccccc1 ZINC000147362186 BD For-Sale Anodyne LYPLA1 0 40 C[C@](N)(C(=O)NN1CCCCC1)c1ccccc1 ZINC000147362186 BD For-Sale Anodyne LYPLA2 24 40 C[C@](N)(C(=O)NN1CCCCC1)c1ccccc1 ZINC000147362186 BD For-Sale Anodyne ABHD11 0 40 CCO[C@H]1CCCN(S(=O)(=O)c2cc(NC(C)=O)ccc2OC)C1 ZINC000147362253 FD On-Demand Anodyne TSHR 62 34 CCO[C@H]1CCCN(S(=O)(=O)c2cc(NC(C)=O)ccc2OC)C1 ZINC000147362253 FD On-Demand Anodyne CPT1A 56 38 CCO[C@H]1CCCN(S(=O)(=O)c2cc(NC(C)=O)ccc2OC)C1 ZINC000147362253 FD On-Demand Anodyne CPT2 49 38 CCO[C@H]1CCCN(S(=O)(=O)c2cc(NC(C)=O)ccc2OC)C1 ZINC000147362253 FD On-Demand Anodyne CPT1B 52 36 Cc1cc(O[C@H](C)C(=O)NC2CC2)ccc1S(N)(=O)=O ZINC000147362277 CC For-Sale Anodyne EPHX2 17 40 O=C(O)CC[C@H](NS(=O)(=O)c1ccccc1[N+](=O)[O-])C(=O)O ZINC000147362289 EC On-Demand Anodyne COLA 79 35 O=C(O)CC[C@H](NS(=O)(=O)c1ccccc1[N+](=O)[O-])C(=O)O ZINC000147362289 EC On-Demand Anodyne NAALAD2 47 40 O=C(O)CC[C@H](NS(=O)(=O)c1ccccc1[N+](=O)[O-])C(=O)O ZINC000147362289 EC On-Demand Anodyne ITGAV 68 41 Cc1nn(-c2ccccc2)c2nc(-c3ccc(N4CCNCC4)cc3)cc(CO)c12 ZINC000147362330 GG Annotated Anodyne ACVR1 49 34 Cc1nn(-c2ccccc2)c2nc(-c3ccc(N4CCNCC4)cc3)cc(CO)c12 ZINC000147362330 GG Annotated Anodyne KHK 0 50 CCc1sc(NC(=O)COc2ccc(C(N)=O)cc2)nc1-c1ccccc1 ZINC000147362349 GG On-Demand Anodyne ADORA1 17 49 CCc1sc(NC(=O)COc2ccc(C(N)=O)cc2)nc1-c1ccccc1 ZINC000147362349 GG On-Demand Anodyne DHODH 15 44 CCc1sc(NC(=O)COc2ccc(C(N)=O)cc2)nc1-c1ccccc1 ZINC000147362349 GG On-Demand Anodyne ADORA2A 18 44 CCc1sc(NC(=O)COc2ccc(C(N)=O)cc2)nc1-c1ccccc1 ZINC000147362349 GG On-Demand Anodyne ADORA2B 33 41 CCc1sc(NC(=O)COc2ccc(C(N)=O)cc2)nc1-c1ccccc1 ZINC000147362349 GG On-Demand Anodyne RORC 19 41 C[C@@](N)(C(=O)NN1CCCCC1)c1ccccc1 ZINC000147362398 BD For-Sale Anodyne AMY2 56 34 C[C@@](N)(C(=O)NN1CCCCC1)c1ccccc1 ZINC000147362398 BD For-Sale Anodyne LYPLA1 0 40 C[C@@](N)(C(=O)NN1CCCCC1)c1ccccc1 ZINC000147362398 BD For-Sale Anodyne LYPLA2 24 40 C[C@@](N)(C(=O)NN1CCCCC1)c1ccccc1 ZINC000147362398 BD For-Sale Anodyne ABHD11 0 40 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362413 CE On-Demand Anodyne PDGFRB 49 37 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362413 CE On-Demand Anodyne MMP13 41 47 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362413 CE On-Demand Anodyne MMP3 47 42 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362413 CE On-Demand Anodyne MMP9 41 47 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362413 CE On-Demand Anodyne EPHX2 54 40 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362413 CE On-Demand Anodyne ACR 30 40 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362413 CE On-Demand Anodyne MMP1 46 47 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362413 CE On-Demand Anodyne MCHR1 15 42 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362413 CE On-Demand Anodyne ELOVL6 0 42 COc1ccc(-c2ccc3c(N4CCOC[C@@H]4C)nc(N4CCC[C@@H](CO)C4)nc3n2)cc1CO ZINC000147362425 JF Annotated Anodyne MTOR 35 63 O=C(CCCCNC(=O)c1csc(-c2nccs2)n1)NO ZINC000147362464 ED Annotated Mild HDAC8 17 43 O=C(CCCCNC(=O)c1csc(-c2nccs2)n1)NO ZINC000147362464 ED Annotated Mild HDAC10 32 47 O=C(CCCCNC(=O)c1csc(-c2nccs2)n1)NO ZINC000147362464 ED Annotated Mild HDAC1 27 64 O=C(CCCCNC(=O)c1csc(-c2nccs2)n1)NO ZINC000147362464 ED Annotated Mild HDAC2 21 43 O=C(CCCCNC(=O)c1csc(-c2nccs2)n1)NO ZINC000147362464 ED Annotated Mild HDAC6 28 64 O=C(CCCCNC(=O)c1csc(-c2nccs2)n1)NO ZINC000147362464 ED Annotated Mild HDAC9 40 36 O=C(CCCCNC(=O)c1csc(-c2nccs2)n1)NO ZINC000147362464 ED Annotated Mild HDA106 0 42 CCN(CC(=O)Nc1c(Cl)cccc1Cl)C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147362500 HJ On-Demand Anodyne EPHX2 19 40 Cc1cc(OCC(=O)NC2CC2)ccc1S(N)(=O)=O ZINC000147362508 CC For-Sale Anodyne LUXN 0 48 Cc1cc(OCC(=O)NC2CC2)ccc1S(N)(=O)=O ZINC000147362508 CC For-Sale Anodyne ADIPOR1 0 43 Cc1cc(OCC(=O)NC2CC2)ccc1S(N)(=O)=O ZINC000147362508 CC For-Sale Anodyne ADIPOR2 0 43 CCc1ncc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCCC2)s1 ZINC000147362513 FJ On-Demand Anodyne KCNQ2 68 45 CCc1ncc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCCC2)s1 ZINC000147362513 FJ On-Demand Anodyne TEK 25 50 CCc1ncc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCCC2)s1 ZINC000147362513 FJ On-Demand Anodyne TAAR1 22 41 CCc1ncc(C(=O)Nc2cc(C(F)(F)F)ccc2N2CCCC2)s1 ZINC000147362513 FJ On-Demand Anodyne LIPG 49 34 O=C(O)CC[C@@H](NS(=O)(=O)c1ccccc1[N+](=O)[O-])C(=O)O ZINC000147362524 EC On-Demand Anodyne FOLH1 47 38 O=C(O)CC[C@@H](NS(=O)(=O)c1ccccc1[N+](=O)[O-])C(=O)O ZINC000147362524 EC On-Demand Anodyne COLA 99 40 O=C(O)CC[C@@H](NS(=O)(=O)c1ccccc1[N+](=O)[O-])C(=O)O ZINC000147362524 EC On-Demand Anodyne NAALAD2 53 41 O=C(O)CC[C@@H](NS(=O)(=O)c1ccccc1[N+](=O)[O-])C(=O)O ZINC000147362524 EC On-Demand Anodyne MMP2 19 40 O=C(O)CC[C@@H](NS(=O)(=O)c1ccccc1[N+](=O)[O-])C(=O)O ZINC000147362524 EC On-Demand Anodyne ITGAV 65 44 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362590 CE On-Demand Anodyne PDGFRB 46 37 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362590 CE On-Demand Anodyne MMP13 37 42 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362590 CE On-Demand Anodyne MMP3 40 42 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362590 CE On-Demand Anodyne MMP9 40 42 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362590 CE On-Demand Anodyne EPHX2 54 40 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362590 CE On-Demand Anodyne ACR 30 40 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362590 CE On-Demand Anodyne MMP1 37 47 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147362590 CE On-Demand Anodyne ELOVL6 0 42 Cc1ccc(F)c(-c2cccc(C(=O)O)c2)c1F ZINC000147362632 BH For-Sale Anodyne DHODH 41 33 Cc1ccc(F)c(-c2cccc(C(=O)O)c2)c1F ZINC000147362632 BH For-Sale Anodyne PTGER1 26 45 Cc1ccc(F)c(-c2cccc(C(=O)O)c2)c1F ZINC000147362632 BH For-Sale Anodyne TTR 0 41 Cc1ccc(F)c(-c2cccc(C(=O)O)c2)c1F ZINC000147362632 BH For-Sale Anodyne AKR1C3 40 40 CC(=O)NC1[C@@H](O)CN(C)C[C@@H]1O ZINC000147362665 AA For-Sale Anodyne NA 45 36 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1nc(C)c(C)o1 ZINC000147362682 DH On-Demand Anodyne LPL 58 36 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1nc(C)c(C)o1 ZINC000147362682 DH On-Demand Anodyne CSF1R 17 41 Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147362696 ED Annotated Mild HDAC8 16 40 Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147362696 ED Annotated Mild HDAC4 16 40 Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147362696 ED Annotated Mild HDAC6 29 77 Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147362696 ED Annotated Mild HDA106 0 42 CCN(CC(=O)Nc1c(Cl)cccc1Cl)C(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147362736 HJ On-Demand Anodyne EPHX2 19 40 NCCN[C@H](CCC(=O)O)C(=O)O ZINC000147362765 AA For-Sale Anodyne FOLH1 73 56 NCCN[C@H](CCC(=O)O)C(=O)O ZINC000147362765 AA For-Sale Anodyne CPB2 54 45 NCCN[C@H](CCC(=O)O)C(=O)O ZINC000147362765 AA For-Sale Anodyne NAALAD2 74 55 NCCN[C@H](CCC(=O)O)C(=O)O ZINC000147362765 AA For-Sale Anodyne GRM8 24 45 NCCN[C@H](CCC(=O)O)C(=O)O ZINC000147362765 AA For-Sale Anodyne GRIK3 20 45 NCCN[C@H](CCC(=O)O)C(=O)O ZINC000147362765 AA For-Sale Anodyne DLG4 62 35 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147362807 CE On-Demand Anodyne PDGFRB 46 37 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147362807 CE On-Demand Anodyne MMP13 37 42 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147362807 CE On-Demand Anodyne MMP3 40 42 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147362807 CE On-Demand Anodyne MMP9 40 42 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147362807 CE On-Demand Anodyne EPHX2 54 40 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147362807 CE On-Demand Anodyne ACR 30 40 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147362807 CE On-Demand Anodyne MMP1 37 47 CC[C@@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147362807 CE On-Demand Anodyne ELOVL6 0 42 CC(C)CCCCNCCc1ccccc1 ZINC000147362813 BH For-Sale Anodyne SIGMAR1 19 70 CC(C)CCCCNCCc1ccccc1 ZINC000147362813 BH For-Sale Anodyne SLC2A1 0 44 CC(C)CCCCNCCc1ccccc1 ZINC000147362813 BH For-Sale Anodyne S1PR2 17 48 CC(C)CCCCNCCc1ccccc1 ZINC000147362813 BH For-Sale Anodyne AMP1_PLAFQ 27 41 CC(C)CCCCNCCc1ccccc1 ZINC000147362813 BH For-Sale Anodyne TAAR1 15 52 CC(C)CCCCNCCc1ccccc1 ZINC000147362813 BH For-Sale Anodyne HT1 0 44 CC(C)CCCCNCCc1ccccc1 ZINC000147362813 BH For-Sale Anodyne GPM3 0 48 CC(C)CCCCNCCc1ccccc1 ZINC000147362813 BH For-Sale Anodyne LMGT2 0 44 COC(=O)Nc1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)/C=C/c2cc(Cl)ccc2-n2cnnn2)cc1 ZINC000147362833 KH Annotated Anodyne FCER2 46 35 COC(=O)Nc1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)/C=C/c2cc(Cl)ccc2-n2cnnn2)cc1 ZINC000147362833 KH Annotated Anodyne TIMP3 56 33 COC(=O)Nc1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)/C=C/c2cc(Cl)ccc2-n2cnnn2)cc1 ZINC000147362833 KH Annotated Anodyne F11 32 70 COC(=O)Nc1ccc(NC(=O)[C@H](Cc2ccccc2)NC(=O)/C=C/c2cc(Cl)ccc2-n2cnnn2)cc1 ZINC000147362833 KH Annotated Anodyne FPR1 55 38 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne LTA4H 35 43 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne CA1 23 41 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne P2RY1 29 53 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne RAF1 67 50 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne KDR 34 48 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne MTNR1B 17 50 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne NPY5R 27 42 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne SLC1A1 19 40 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne CFTR 26 40 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne SLC1A3 17 40 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne EPHX2 25 40 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne ACR 21 49 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne SLC1A2 38 40 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne TEK 57 48 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne BRAF 18 41 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne KCNK3 18 40 CN(C)C(=O)Nc1ccc(Oc2cccc(C(F)(F)F)c2)cc1 ZINC000147362864 DJ For-Sale Anodyne PDS 45 45 CC(=O)NC1[C@H](O)CN(C)C[C@H]1O ZINC000147362883 AA For-Sale Anodyne NA 45 36 CCCS(=O)(=O)NC1CCN(C(=O)c2cccn(Cc3ccccc3)c2=O)CC1 ZINC000147362884 HD On-Demand Anodyne MLNR 25 41 CCCS(=O)(=O)NC1CCN(C(=O)c2cccn(Cc3ccccc3)c2=O)CC1 ZINC000147362884 HD On-Demand Anodyne CCR8 93 38 CCCS(=O)(=O)NC1CCN(C(=O)c2cccn(Cc3ccccc3)c2=O)CC1 ZINC000147362884 HD On-Demand Anodyne SFRP1 81 39 CCCS(=O)(=O)NC1CCN(C(=O)c2cccn(Cc3ccccc3)c2=O)CC1 ZINC000147362884 HD On-Demand Anodyne WNT3 52 34 CCCCc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147362903 GG Annotated Mild MAP1 16 41 C[C@@H](CN(C)C(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147362935 CD For-Sale Anodyne GPR88 0 57 CCN(CC(=O)Nc1c(Cl)cccc1Cl)C(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147362960 HJ On-Demand Anodyne EPHX2 19 40 CCC[C@H](NC(N)=O)C(=O)Nc1nc(-c2ccccc2)c(CC)s1 ZINC000147362992 EG On-Demand Anodyne PTGDR2 16 45 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147363005 CE On-Demand Anodyne PDGFRB 46 37 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147363005 CE On-Demand Anodyne MMP13 37 42 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147363005 CE On-Demand Anodyne MMP3 40 42 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147363005 CE On-Demand Anodyne MMP9 40 42 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147363005 CE On-Demand Anodyne EPHX2 54 40 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147363005 CE On-Demand Anodyne ACR 30 40 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147363005 CE On-Demand Anodyne MMP1 37 47 CC[C@H]1CN(C(=O)Nc2ccc(OC)cc2)CC[C@H]1N ZINC000147363005 CE On-Demand Anodyne ELOVL6 0 42 CCCCCNCCCCC(C)C ZINC000147363057 AH For-Sale Anodyne ADH1A 0 43 CCCCCNCCCCC(C)C ZINC000147363057 AH For-Sale Anodyne ADH7 0 41 CCCCCNCCCCC(C)C ZINC000147363057 AH For-Sale Anodyne S1PR3 17 47 CCCCCNCCCCC(C)C ZINC000147363057 AH For-Sale Anodyne S1PR2 40 47 CCCCCNCCCCC(C)C ZINC000147363057 AH For-Sale Anodyne ADH1B 0 43 CCCCCNCCCCC(C)C ZINC000147363057 AH For-Sale Anodyne ADH1C 0 43 CCCCCNCCCCC(C)C ZINC000147363057 AH For-Sale Anodyne Q6UB75_PIG 40 35 CCCCCNCCCCC(C)C ZINC000147363057 AH For-Sale Anodyne FPPS 0 41 CCCCCNCCCCC(C)C ZINC000147363057 AH For-Sale Anodyne SPPS 46 39 Cc1cccc(NC(=O)c2cccc3c2OCCN3)c1O ZINC000147363081 CF For-Sale Anodyne G2YM83_BOTF4 59 34 CCCS(=O)(=O)NC1CCN(C(=O)CNC(=O)OCC)CC1 ZINC000147363109 EC On-Demand Anodyne CCR8 54 36 C[C@H](CN(C)C(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147363153 CD For-Sale Anodyne GPR88 0 57 O=C(O)C1(NCCCc2nc(-c3cccs3)no2)CCC1 ZINC000147363159 DE For-Sale Anodyne ETHR 29 40 CCOC(=O)c1ccc(/N=C/c2cc(C)cc(Br)c2)cc1 ZINC000147363168 EJ For-Sale Anodyne ACR 19 42 CC[C@@H]1CN(C(=O)NC2CC2)CC[C@@H]1N ZINC000147363193 BC For-Sale Anodyne EPHX2 20 40 CC(=O)Nc1ccc(C)c(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)c1 ZINC000147363201 GF On-Demand Anodyne MAPK14 34 43 O=C(CNc1ccc(Cl)cc1Cl)Nc1ccc(N2CCCCC2)cc1 ZINC000147363203 GK For-Sale Anodyne CNR1 54 33 O=C(CNc1ccc(Cl)cc1Cl)Nc1ccc(N2CCCCC2)cc1 ZINC000147363203 GK For-Sale Anodyne F10 22 40 O=C(CNc1ccc(Cl)cc1Cl)Nc1ccc(N2CCCCC2)cc1 ZINC000147363203 GK For-Sale Anodyne LPL 26 40 O=C(CNc1ccc(Cl)cc1Cl)Nc1ccc(N2CCCCC2)cc1 ZINC000147363203 GK For-Sale Anodyne CNR2 19 41 O=C(CNc1ccc(Cl)cc1Cl)Nc1ccc(N2CCCCC2)cc1 ZINC000147363203 GK For-Sale Anodyne HNMT 42 32 O=C(CNc1ccc(Cl)cc1Cl)Nc1ccc(N2CCCCC2)cc1 ZINC000147363203 GK For-Sale Anodyne EPHX2 15 42 CCC[C@@H](NC(N)=O)C(=O)Nc1nc(-c2ccccc2)c(CC)s1 ZINC000147363214 EG On-Demand Anodyne PTGDR2 16 45 O=C(Nc1nc2ccccc2[nH]1)c1ccc(Br)c(Cl)c1 ZINC000147363225 FI On-Demand Anodyne KCNN3 36 43 O=C(Nc1nc2ccccc2[nH]1)c1ccc(Br)c(Cl)c1 ZINC000147363225 FI On-Demand Anodyne HPSE 16 46 O=C(Nc1nc2ccccc2[nH]1)c1ccc(Br)c(Cl)c1 ZINC000147363225 FI On-Demand Anodyne NR2E3 67 40 O=C(Nc1nc2ccccc2[nH]1)c1ccc(Br)c(Cl)c1 ZINC000147363225 FI On-Demand Anodyne SHH 31 48 O=C(Nc1nc2ccccc2[nH]1)c1ccc(Br)c(Cl)c1 ZINC000147363225 FI On-Demand Anodyne STK33 56 44 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne F2 60 51 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne OPRM1 16 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne CELA1 46 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne ELANE 45 36 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne TRHR 58 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne HLA-DRB3 63 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne CTRA_BOVIN 41 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne TRY1_BOVIN 96 48 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne NTSR1 80 36 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne NTSR2 66 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne MAP1 103 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne CELA2A 41 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne LGMN 54 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne TPP2 44 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne XIAP 47 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363256 FD On-Demand Anodyne TMPRSS11D 45 36 Nc1nc(Oc2cccc(Cl)c2Cl)c2ccccc2n1 ZINC000147363262 DI For-Sale Anodyne DHFR 18 43 FC(F)CNCc1cncn1C1CC1 ZINC000147363306 BD For-Sale Anodyne CAMC 0 44 C[C@@H](CN(C)C(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147363339 CD For-Sale Anodyne GPR88 0 57 COc1ccc2nc(CCl)n(CCNC(=O)N(C)C)c2n1 ZINC000147363363 DD For-Sale Reactive PDE10A 33 42 CC(C)CCCCNCc1ccc(-c2ccc(F)cc2)o1 ZINC000147363377 CK For-Sale Anodyne LEF 46 33 CC[C@H]1CN(C(=O)NC2CC2)CC[C@@H]1N ZINC000147363409 BC For-Sale Anodyne EPHX2 20 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne F2 60 51 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne OPRM1 16 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne CELA1 46 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne ELANE 45 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne TRHR 58 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne HLA-DRB3 63 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne CTRA_BOVIN 41 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne TRY1_BOVIN 96 48 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne NTSR1 80 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne NTSR2 66 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne MAP1 103 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne CELA2A 41 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne LGMN 54 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne TPP2 44 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne XIAP 47 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1nccs1 ZINC000147363422 FD On-Demand Anodyne TMPRSS11D 45 36 CCc1ncc(C(=O)N(C)Cc2ccc3c(c2)OCO3)s1 ZINC000147363434 DF On-Demand Anodyne NOS2 71 36 CCc1ncc(C(=O)N(C)Cc2ccc3c(c2)OCO3)s1 ZINC000147363434 DF On-Demand Anodyne HSD17B2 25 41 CCc1cn(C)c2c(N3CCCC3=O)cc(C(=O)N[C@@H](Cc3ccccc3)[C@@H](O)CNCc3cccc(OC)c3)cc12 ZINC000147363468 KI Annotated Anodyne CTSD 59 69 CCc1cn(C)c2c(N3CCCC3=O)cc(C(=O)N[C@@H](Cc3ccccc3)[C@@H](O)CNCc3cccc(OC)c3)cc12 ZINC000147363468 KI Annotated Anodyne BACE2 71 69 CCc1cn(C)c2c(N3CCCC3=O)cc(C(=O)N[C@@H](Cc3ccccc3)[C@@H](O)CNCc3cccc(OC)c3)cc12 ZINC000147363468 KI Annotated Anodyne BACE1 89 81 CCc1cn(C)c2c(N3CCCC3=O)cc(C(=O)N[C@@H](Cc3ccccc3)[C@@H](O)CNCc3cccc(OC)c3)cc12 ZINC000147363468 KI Annotated Anodyne PLM1_PLAFA 55 44 CCc1cn(C)c2c(N3CCCC3=O)cc(C(=O)N[C@@H](Cc3ccccc3)[C@@H](O)CNCc3cccc(OC)c3)cc12 ZINC000147363468 KI Annotated Anodyne PLM2_PLAFA 30 54 C#CCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147363476 CB For-Sale Mild CA2 27 42 C[C@H](CN(C)C(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147363550 CD For-Sale Anodyne GPR88 0 57 Cc1nc(-c2nc(C(=O)N[C@H](C(=O)NCCC(=O)NO)C(C)C)cs2)cs1 ZINC000147363580 HD Annotated Mild HDAC3 17 64 CC[C@@H]1CN(C(=O)NC2CC2)CC[C@H]1N ZINC000147363606 BC For-Sale Anodyne EPHX2 20 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne F2 60 51 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne OPRM1 16 43 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne CELA1 46 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne ELANE 45 36 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne TRHR 58 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne HLA-DRB3 63 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne CTRA_BOVIN 41 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne TRY1_BOVIN 96 48 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne NTSR1 80 36 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne NTSR2 66 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne MAP1 103 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne CELA2A 41 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne LGMN 54 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne TPP2 44 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne XIAP 47 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363623 FD On-Demand Anodyne TMPRSS11D 45 36 CCCCCCCCNC(=O)[C@@H]1CC[C@H](N)[C@H](C)C1 ZINC000147363632 CG For-Sale Mild EPHX2 40 40 CCCCCCCCNC(=O)[C@@H]1CC[C@H](N)[C@H](C)C1 ZINC000147363632 CG For-Sale Mild TPP2 26 40 CCCCCCCCNC(=O)[C@@H]1CC[C@H](N)[C@H](C)C1 ZINC000147363632 CG For-Sale Mild ASAH1 49 32 CC(=O)Nc1ccc(C)c(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)c1 ZINC000147363642 HJ On-Demand Anodyne ROCK2 28 46 CC(=O)Nc1ccc(C)c(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)c1 ZINC000147363642 HJ On-Demand Anodyne MET 39 43 CC(=O)Nc1ccc(C)c(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)c1 ZINC000147363642 HJ On-Demand Anodyne DDR2 16 40 CC(=O)Nc1ccc(C)c(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)c1 ZINC000147363642 HJ On-Demand Anodyne NAMPT 46 44 COc1ccc2c(c1)cc(C(=O)Cl)n2C ZINC000147363645 BF For-Sale Reactive PTGS2 37 42 COc1ccc2c(c1)cc(C(=O)Cl)n2C ZINC000147363645 BF For-Sale Reactive AKR1C3 30 42 COc1ccc2c(c1)cc(C(=O)Cl)n2C ZINC000147363645 BF For-Sale Reactive PYK 24 48 CC(C)CCCCNCc1ccc(OCCC(C)C)cc1 ZINC000147363670 CK For-Sale Anodyne LTA4H 18 42 CC(C)CCCCNCc1ccc(OCCC(C)C)cc1 ZINC000147363670 CK For-Sale Anodyne LPAR2 42 50 CC(C)CCCCNCc1ccc(OCCC(C)C)cc1 ZINC000147363670 CK For-Sale Anodyne S1PR3 17 50 CC(C)CCCCNCc1ccc(OCCC(C)C)cc1 ZINC000147363670 CK For-Sale Anodyne SLC2A1 26 43 CC(C)CCCCNCc1ccc(OCCC(C)C)cc1 ZINC000147363670 CK For-Sale Anodyne S1PR2 43 50 CC(C)CCCCNCc1ccc(OCCC(C)C)cc1 ZINC000147363670 CK For-Sale Anodyne LEF 77 40 CC(C)CCCCNCc1ccc(OCCC(C)C)cc1 ZINC000147363670 CK For-Sale Anodyne HT1 0 43 CC(C)CCCCNCc1ccc(OCCC(C)C)cc1 ZINC000147363670 CK For-Sale Anodyne GPM3 0 51 CC(C)CCCCNCc1ccc(OCCC(C)C)cc1 ZINC000147363670 CK For-Sale Anodyne O69638_MYCTO 0 47 CC(C)CCCCNCc1ccc(OCCC(C)C)cc1 ZINC000147363670 CK For-Sale Anodyne LMGT2 0 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(-n3cccn3)c(F)c2)c1 ZINC000147363787 FG On-Demand Bother TAAR1 27 47 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne F2 60 51 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne OPRM1 16 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne CELA1 46 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne ELANE 45 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne TRHR 58 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne HLA-DRB3 63 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne CTRA_BOVIN 41 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne TRY1_BOVIN 96 48 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne NTSR1 80 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne NTSR2 66 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne MAP1 103 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne CELA2A 41 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne LGMN 54 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne TPP2 44 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne XIAP 47 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1nccs1 ZINC000147363799 FD On-Demand Anodyne TMPRSS11D 45 36 CC[C@H]1CN(C(=O)NC2CC2)CC[C@H]1N ZINC000147363804 BC For-Sale Anodyne EPHX2 20 40 CC(=O)c1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147363860 CD For-Sale Anodyne ABCB1 0 41 CC(=O)c1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147363860 CD For-Sale Anodyne HCN1 73 34 CC(=O)c1ccccc1OCCNC1(C(=O)O)CCC1 ZINC000147363860 CD For-Sale Anodyne HCN4 52 34 CCCCC1CCC(NC(=O)Nc2cc(NC(C)=O)ccc2C)CC1 ZINC000147363861 EJ On-Demand Anodyne EPHX2 47 45 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147363875 DD On-Demand Anodyne ANPEP 37 40 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147363875 DD On-Demand Anodyne FCER2 42 36 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147363875 DD On-Demand Anodyne KLK3 52 34 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147363875 DD On-Demand Anodyne CTSK 25 40 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147363875 DD On-Demand Anodyne CAPNS1 51 36 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147363875 DD On-Demand Anodyne HLA-DRB1 46 34 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147363875 DD On-Demand Anodyne CTSS 20 40 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147363875 DD On-Demand Anodyne CAPN1 80 38 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147363875 DD On-Demand Anodyne CAPN2 103 39 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147363875 DD On-Demand Anodyne FPR1 59 37 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147363875 DD On-Demand Anodyne NPR 66 33 Cc1cccc(CNCCCCC(C)C)c1 ZINC000147363880 BH For-Sale Anodyne FDFT1 0 48 Cc1cccc(CNCCCCC(C)C)c1 ZINC000147363880 BH For-Sale Anodyne SLC6A13 0 47 Cc1cccc(CNCCCCC(C)C)c1 ZINC000147363880 BH For-Sale Anodyne LEF 74 41 Cc1cccc(CNCCCCC(C)C)c1 ZINC000147363880 BH For-Sale Anodyne GPM3 0 49 C#CCNC(=O)[C@H](C)Oc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147363897 CC For-Sale Mild CA2 34 41 C#CCNC(=O)[C@H](C)Oc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147363897 CC For-Sale Mild CA14 16 41 C[C@H](Cc1ccsc1)NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147363909 DI On-Demand Anodyne MDM2 63 33 COC(=O)N[C@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147364066 DD On-Demand Anodyne ANPEP 37 40 COC(=O)N[C@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147364066 DD On-Demand Anodyne FCER2 42 36 COC(=O)N[C@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147364066 DD On-Demand Anodyne KLK3 52 34 COC(=O)N[C@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147364066 DD On-Demand Anodyne CTSK 25 40 COC(=O)N[C@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147364066 DD On-Demand Anodyne CAPNS1 51 36 COC(=O)N[C@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147364066 DD On-Demand Anodyne HLA-DRB1 46 34 COC(=O)N[C@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147364066 DD On-Demand Anodyne CTSS 20 40 COC(=O)N[C@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147364066 DD On-Demand Anodyne CAPN1 80 38 COC(=O)N[C@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147364066 DD On-Demand Anodyne CAPN2 103 39 COC(=O)N[C@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147364066 DD On-Demand Anodyne FPR1 59 37 COC(=O)N[C@H](CC(C)C)C(=O)Nc1nnc2ccccn12 ZINC000147364066 DD On-Demand Anodyne NPR 66 33 Cc1cc(C(=O)NCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147364079 CD On-Demand Bother DRD4 49 40 Cc1cc(C(=O)NCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147364079 CD On-Demand Bother ADRA1A 22 40 Cc1cc(C(=O)NCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147364079 CD On-Demand Bother PLD2 56 35 CCCCCCCCNC(=O)[C@@H]1CC[C@@H](N)[C@H](C)C1 ZINC000147364083 CG For-Sale Mild EPHX2 40 40 CCCCCCCCNC(=O)[C@@H]1CC[C@@H](N)[C@H](C)C1 ZINC000147364083 CG For-Sale Mild TPP2 26 40 CCCCCCCCNC(=O)[C@@H]1CC[C@@H](N)[C@H](C)C1 ZINC000147364083 CG For-Sale Mild ASAH1 49 32 CC(C)CCCCNS(=O)(=O)c1ccc(C(=O)O)cc1 ZINC000147364094 CE For-Sale Anodyne CA2 25 40 CC(C)CCCCNS(=O)(=O)c1ccc(C(=O)O)cc1 ZINC000147364094 CE For-Sale Anodyne TBXA2R 45 35 CC(C)CCCCNS(=O)(=O)c1ccc(C(=O)O)cc1 ZINC000147364094 CE For-Sale Anodyne TBXAS1 47 43 CC(C)CCCCNS(=O)(=O)c1ccc(C(=O)O)cc1 ZINC000147364094 CE For-Sale Anodyne CASP3 0 42 C#CCNC(=O)[C@@H](C)Oc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147364107 CC For-Sale Mild CA2 34 41 C#CCNC(=O)[C@@H](C)Oc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147364107 CC For-Sale Mild CA14 16 41 C[C@H](O)c1ccc(NC(=O)NCCNC(=O)N(C)C)cc1 ZINC000147364218 CD For-Sale Anodyne PSBA 0 53 Cc1c(CN2CCSCC2)cccc1NC(=O)[C@@H](C)N1CCc2ccccc21 ZINC000147364227 GH On-Demand Anodyne KCNQ2 50 33 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccccc1Cl)NO ZINC000147364241 IH Annotated Mild HDAC10 20 40 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccccc1Cl)NO ZINC000147364241 IH Annotated Mild HDAC6 26 76 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccccc1Cl)NO ZINC000147364241 IH Annotated Mild HDA106 0 42 O=C(O)C1(NCCCOc2ccccc2)CCC1 ZINC000147364279 BE For-Sale Anodyne DRD4 19 44 O=C(O)C1(NCCCOc2ccccc2)CCC1 ZINC000147364279 BE For-Sale Anodyne HRH2 23 40 O=C(O)C1(NCCCOc2ccccc2)CCC1 ZINC000147364279 BE For-Sale Anodyne LTA4H 30 44 O=C(O)C1(NCCCOc2ccccc2)CCC1 ZINC000147364279 BE For-Sale Anodyne PLA2G4B 57 32 C=CC[C@]1(C)C[C@@H](c2cccc(Cl)c2)[C@@H](c2ccc(Cl)cc2)OC1=O ZINC000147364304 GK For-Sale Mild TP53 27 44 C=CC[C@]1(C)C[C@@H](c2cccc(Cl)c2)[C@@H](c2ccc(Cl)cc2)OC1=O ZINC000147364304 GK For-Sale Mild MDM2 161 44 CNCc1ccc(Oc2ccc(Cl)c(F)c2)nc1C ZINC000147364309 CH For-Sale Anodyne SLC6A4 15 55 C[C@H](Cc1ccsc1)NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147364319 DI On-Demand Anodyne MDM2 63 33 CC(C)OCC(=O)Nc1ccc2nc3n(c(=O)c2c1)CCC3 ZINC000147364359 DD On-Demand Anodyne ACHE 16 46 CC(C)OCC(=O)Nc1ccc2nc3n(c(=O)c2c1)CCC3 ZINC000147364359 DD On-Demand Anodyne MCHR1 30 41 CC[C@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147364396 BD For-Sale Anodyne ACE 33 42 CC[C@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147364396 BD For-Sale Anodyne MME 36 42 CC[C@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147364396 BD For-Sale Anodyne ACE2 68 37 CC[C@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147364396 BD For-Sale Anodyne GPR88 0 51 Cc1c(CN2CCSCC2)cccc1NC(=O)[C@H](C)N1CCc2ccccc21 ZINC000147364448 GH On-Demand Anodyne KCNQ2 50 33 C[C@@H](O)c1ccc(NC(=O)NCCNC(=O)N(C)C)cc1 ZINC000147364451 CD For-Sale Anodyne PSBA 0 53 O=C(O)C1(NCc2nc(-c3ccccc3)no2)CCC1 ZINC000147364501 CD For-Sale Anodyne NPPA 41 48 COCc1nc(C(=O)Nc2ccc(-n3cnc4ccccc43)cc2)cs1 ZINC000147364519 FH On-Demand Anodyne F9 37 45 COCc1nc(C(=O)Nc2ccc(-n3cnc4ccccc43)cc2)cs1 ZINC000147364519 FH On-Demand Anodyne PDGFRB 15 42 CCCCCCCCNC(=O)[C@@H]1CCC[C@H](C)[C@@H]1N ZINC000147364531 CG For-Sale Mild TPP2 27 43 CCCCCCCCNC(=O)[C@@H]1CCC[C@H](C)[C@@H]1N ZINC000147364531 CG For-Sale Mild ASAH1 48 32 O=C(CNC(=O)Nc1nc(CN2CCCCC2)cs1)Nc1ccc(F)cc1 ZINC000147364545 GG On-Demand Anodyne CCR3 53 38 CC[C@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147364637 BD For-Sale Anodyne ACE 33 42 CC[C@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147364637 BD For-Sale Anodyne MME 36 42 CC[C@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147364637 BD For-Sale Anodyne ACE2 68 37 CC[C@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147364637 BD For-Sale Anodyne GPR88 0 51 C[C@H](O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147364639 CD For-Sale Anodyne ACAT 0 40 C[C@H](O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147364639 CD For-Sale Anodyne PSBA 0 43 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1cccc(CN2CCSCC2)c1C ZINC000147364692 GG On-Demand Anodyne ANPEP 33 40 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1cccc(CN2CCSCC2)c1C ZINC000147364692 GG On-Demand Anodyne CAPNS1 50 31 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1cccc(CN2CCSCC2)c1C ZINC000147364692 GG On-Demand Anodyne CAPN1 42 37 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1cccc(CN2CCSCC2)c1C ZINC000147364692 GG On-Demand Anodyne CAPN2 60 34 COC(=O)N[C@@H](CC(C)C)C(=O)Nc1cccc(CN2CCSCC2)c1C ZINC000147364692 GG On-Demand Anodyne FPR1 45 31 CCN[C@@H]1c2ccccc2C[C@@H]1O ZINC000147364768 AD For-Sale Anodyne POL 0 43 CCN[C@@H]1c2ccccc2C[C@@H]1O ZINC000147364768 AD For-Sale Anodyne PLM1_PLAFA 41 41 CCN[C@@H]1c2ccccc2C[C@@H]1O ZINC000147364768 AD For-Sale Anodyne PLM2_PLAFA 23 41 CCN[C@@H]1c2ccccc2C[C@@H]1O ZINC000147364768 AD For-Sale Anodyne Q8IM16_PLAF7 0 41 O=C(CNC(=O)Nc1nc(CN2CCOCC2)cs1)Nc1ccc(F)cc1 ZINC000147364779 GD On-Demand Anodyne PIK3CA 21 41 O=C(CNC(=O)Nc1nc(CN2CCOCC2)cs1)Nc1ccc(F)cc1 ZINC000147364779 GD On-Demand Anodyne MTOR 50 41 O=C(CNC(=O)Nc1nc(CN2CCOCC2)cs1)Nc1ccc(F)cc1 ZINC000147364779 GD On-Demand Anodyne EPHX2 19 45 O=C(CNC(=O)Nc1nc(CN2CCOCC2)cs1)Nc1ccc(F)cc1 ZINC000147364779 GD On-Demand Anodyne PIK3CG 16 41 CCCCCCCCCn1cc(C)c(I)n1 ZINC000147364781 EJ For-Sale Mild ADA 32 46 O=C(Nc1ccc2nc3n(c(=O)c2c1)CCC3)c1cccn(Cc2ccccc2)c1=O ZINC000147364844 HF On-Demand Anodyne ACHE 18 42 O=C(Nc1ccc2nc3n(c(=O)c2c1)CCC3)c1cccn(Cc2ccccc2)c1=O ZINC000147364844 HF On-Demand Anodyne NR2E3 61 34 O=C(Nc1ccc2nc3n(c(=O)c2c1)CCC3)c1cccn(Cc2ccccc2)c1=O ZINC000147364844 HF On-Demand Anodyne POLR1A 72 37 C[C@@H](O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147364861 CD For-Sale Anodyne ACAT 0 40 C[C@@H](O)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147364861 CD For-Sale Anodyne PSBA 0 43 O=C(O)C1CCC(NC(=O)[C@H]2C[C@H]2c2ccccc2)CC1 ZINC000147364882 CF For-Sale Anodyne EPHX2 22 44 O=C(O)C1CCC(NC(=O)[C@H]2C[C@H]2c2ccccc2)CC1 ZINC000147364882 CF For-Sale Anodyne GPR88 0 41 CCCCCCCCNC(=O)[C@@H]1CCC[C@@H](C)[C@@H]1N ZINC000147364930 CG For-Sale Mild TPP2 27 43 CCCCCCCCNC(=O)[C@@H]1CCC[C@@H](C)[C@@H]1N ZINC000147364930 CG For-Sale Mild ASAH1 48 32 CC[C@@H]1CN(C(=O)Nc2cccc(F)c2)CC[C@@H]1N ZINC000147364949 CE On-Demand Anodyne CCR3 52 42 CC[C@@H]1CN(C(=O)Nc2cccc(F)c2)CC[C@@H]1N ZINC000147364949 CE On-Demand Anodyne MLNR 26 40 COc1ccc(C)cc1-n1ccc(C(=O)Nc2ccc(C)cn2)n1 ZINC000147364964 DG On-Demand Anodyne F10 50 36 COc1ccc(C)cc1-n1ccc(C(=O)Nc2ccc(C)cn2)n1 ZINC000147364964 DG On-Demand Anodyne GCK 25 40 COc1ccc(C)cc1-n1ccc(C(=O)Nc2ccc(C)cn2)n1 ZINC000147364964 DG On-Demand Anodyne LUCI_LUCLA 39 53 O=C(O)C1CCC(NC(=O)[C@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147365074 CF For-Sale Anodyne EPHX2 22 44 O=C(O)C1CCC(NC(=O)[C@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147365074 CF For-Sale Anodyne GPR88 0 41 CCOC(=O)NCC(=O)Nc1ccc2nc3n(c(=O)c2c1)CCC3 ZINC000147365076 ED On-Demand Anodyne ACHE 17 47 CN[C@@H]1CCN(c2ccc(N)cn2)C1 ZINC000147365123 AC In-Stock Anodyne HRH4 80 54 Cc1c(CN2CCSCC2)cccc1NC(=O)[C@@H]1CCCN1Cc1ccccc1 ZINC000147365129 HI On-Demand Anodyne SIGMAR1 25 44 Cc1c(CN2CCSCC2)cccc1NC(=O)[C@@H]1CCCN1Cc1ccccc1 ZINC000147365129 HI On-Demand Anodyne CCR3 30 42 CC[C@H](NC(=O)c1cc(C)ccc1Br)C(=O)O ZINC000147365145 DE On-Demand Anodyne ACE2 44 32 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCCN(C)C)nc12 ZINC000147365154 GD For-Sale Clean ADORA2B 18 47 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCCN(C)C)nc12 ZINC000147365154 GD For-Sale Clean CASR 26 46 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCCN(C)C)nc12 ZINC000147365154 GD For-Sale Clean PIK3CA 30 47 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCCN(C)C)nc12 ZINC000147365154 GD For-Sale Clean MTOR 38 47 COc1ccc(N2CCOCC2)c2sc(NC(=O)NCCN(C)C)nc12 ZINC000147365154 GD For-Sale Clean PIK3CG 29 47 CC[C@H]1CN(C(=O)Nc2cccc(F)c2)CC[C@@H]1N ZINC000147365162 CE On-Demand Anodyne CCR3 52 42 CC[C@H]1CN(C(=O)Nc2cccc(F)c2)CC[C@@H]1N ZINC000147365162 CE On-Demand Anodyne MLNR 26 40 Cc1ccc(NC(=O)Cc2c(C)nn(C(F)F)c2C)nc1 ZINC000147365193 CF On-Demand Anodyne P2RX7 34 42 O=C(O)C1CCC(NC(=O)[C@@H]2C[C@H]2c2ccccc2)CC1 ZINC000147365302 CF For-Sale Anodyne EPHX2 22 44 O=C(O)C1CCC(NC(=O)[C@@H]2C[C@H]2c2ccccc2)CC1 ZINC000147365302 CF For-Sale Anodyne GPR88 0 41 CN[C@H]1CCN(c2ccc(N)cn2)C1 ZINC000147365303 AC In-Stock Anodyne HRH4 80 54 CS(=O)(=O)NCCC(=O)Nc1ccc2nc3n(c(=O)c2c1)CCC3 ZINC000147365307 FC On-Demand Anodyne ACHE 17 44 CS(=O)(=O)NCCC(=O)Nc1ccc2nc3n(c(=O)c2c1)CCC3 ZINC000147365307 FC On-Demand Anodyne TERT 17 41 Cc1c(CN2CCSCC2)cccc1NC(=O)[C@H]1CCCN1Cc1ccccc1 ZINC000147365341 HI On-Demand Anodyne SIGMAR1 25 44 Cc1c(CN2CCSCC2)cccc1NC(=O)[C@H]1CCCN1Cc1ccccc1 ZINC000147365341 HI On-Demand Anodyne CCR3 30 42 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccccc1)NO ZINC000147365342 HG Annotated Mild HDAC10 45 49 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccccc1)NO ZINC000147365342 HG Annotated Mild HDAC2 31 44 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccccc1)NO ZINC000147365342 HG Annotated Mild HDAC4 15 42 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccccc1)NO ZINC000147365342 HG Annotated Mild HDAC5 16 42 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccccc1)NO ZINC000147365342 HG Annotated Mild HDAC6 40 44 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccccc1)NO ZINC000147365342 HG Annotated Mild HDA106 0 49 CCCCCCCCNC(=O)[C@@H]1CC[C@H](C)[C@H](N)C1 ZINC000147365355 CG For-Sale Mild EPHX2 39 40 CCCCCCCCNC(=O)[C@@H]1CC[C@H](C)[C@H](N)C1 ZINC000147365355 CG For-Sale Mild TPP2 26 40 CCCCCCCCNC(=O)[C@@H]1CC[C@H](C)[C@H](N)C1 ZINC000147365355 CG For-Sale Mild ASAH1 49 32 CC[C@@H]1CN(C(=O)Nc2cccc(F)c2)CC[C@H]1N ZINC000147365370 CE On-Demand Anodyne CCR3 52 42 CC[C@@H]1CN(C(=O)Nc2cccc(F)c2)CC[C@H]1N ZINC000147365370 CE On-Demand Anodyne MLNR 26 40 O=C(O)C1CCC(NC(=O)[C@@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147365472 CF For-Sale Anodyne EPHX2 22 44 O=C(O)C1CCC(NC(=O)[C@@H]2C[C@@H]2c2ccccc2)CC1 ZINC000147365472 CF For-Sale Anodyne GPR88 0 41 O=C(c1ccc2c(c1)COC2)N1CCC[C@H](CCBr)C1 ZINC000147365520 EG For-Sale Reactive L3MBTL3 51 35 CC[C@H]1CN(C(=O)Nc2cccc(F)c2)CC[C@H]1N ZINC000147365585 CE On-Demand Anodyne CCR3 52 42 CC[C@H]1CN(C(=O)Nc2cccc(F)c2)CC[C@H]1N ZINC000147365585 CE On-Demand Anodyne MLNR 26 40 NC(=O)c1ccc(CC(=O)N2CCCCC2)cc1 ZINC000147365655 BD On-Demand Anodyne DPP7 51 35 NC(=O)c1ccc(CC(=O)N2CCCCC2)cc1 ZINC000147365655 BD On-Demand Anodyne KCNJ1 40 36 Cc1ccc(C(=O)NC2CCC(C(=O)O)CC2)cc1Br ZINC000147365691 EG In-Stock Anodyne MAPK11 43 42 Cc1ccc(C(=O)NC2CCC(C(=O)O)CC2)cc1Br ZINC000147365691 EG In-Stock Anodyne MAPK14 59 46 Cc1ccc(C(=O)NC2CCC(C(=O)O)CC2)cc1Br ZINC000147365691 EG In-Stock Anodyne MAPK13 80 40 Cc1ccc(C(=O)NC2CCC(C(=O)O)CC2)cc1Br ZINC000147365691 EG In-Stock Anodyne HSPB1 0 46 O=C(c1ccc2c(c1)COC2)N1CCC[C@@H](CCBr)C1 ZINC000147365706 EG For-Sale Reactive L3MBTL3 51 35 CCCCCCCCNC(=O)[C@@H]1CC[C@@H](C)[C@H](N)C1 ZINC000147365761 CG For-Sale Mild EPHX2 39 40 CCCCCCCCNC(=O)[C@@H]1CC[C@@H](C)[C@H](N)C1 ZINC000147365761 CG For-Sale Mild TPP2 26 40 CCCCCCCCNC(=O)[C@@H]1CC[C@@H](C)[C@H](N)C1 ZINC000147365761 CG For-Sale Mild ASAH1 49 32 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365778 ED On-Demand Anodyne OPRM1 23 42 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365778 ED On-Demand Anodyne CTSK 23 40 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365778 ED On-Demand Anodyne CHRNA6 0 47 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365778 ED On-Demand Anodyne NPFFR2 40 32 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365778 ED On-Demand Anodyne PCSK5 54 35 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365778 ED On-Demand Anodyne FURIN 55 35 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365778 ED On-Demand Anodyne POLG_WNV 72 32 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365778 ED On-Demand Anodyne NPFFR1 61 32 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365778 ED On-Demand Anodyne NOD2 42 37 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147365809 GG On-Demand Anodyne PIK3CA 37 42 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147365809 GG On-Demand Anodyne JAK2 15 42 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147365809 GG On-Demand Anodyne MAPKAPK5 45 34 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147365809 GG On-Demand Anodyne MTOR 74 43 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147365809 GG On-Demand Anodyne TTK 18 41 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147365809 GG On-Demand Anodyne EPHB4 51 33 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147365809 GG On-Demand Anodyne STAT6 60 38 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147365809 GG On-Demand Anodyne DGAT1 53 47 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365999 ED On-Demand Anodyne OPRM1 23 42 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365999 ED On-Demand Anodyne CTSK 23 40 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365999 ED On-Demand Anodyne CHRNA6 0 47 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365999 ED On-Demand Anodyne NPFFR2 40 32 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365999 ED On-Demand Anodyne PCSK5 54 35 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365999 ED On-Demand Anodyne FURIN 55 35 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365999 ED On-Demand Anodyne POLG_WNV 72 32 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365999 ED On-Demand Anodyne NPFFR1 61 32 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCc2ccccc2C1 ZINC000147365999 ED On-Demand Anodyne NOD2 42 37 CCC(CC)CN1C(=O)C(=O)c2cccc(F)c21 ZINC000147366030 BF For-Sale Anodyne ALDH1A1 50 36 CCCCCC(=O)[C@@H]1Cc2ccccc2O1 ZINC000147366056 BG For-Sale Anodyne TPP2 51 33 CCCCCC(=O)[C@@H]1Cc2ccccc2O1 ZINC000147366056 BG For-Sale Anodyne CQSS 50 31 CCCCCCCCNC(=O)[C@@H]1C[C@H](N)CC[C@@H]1C ZINC000147366134 CG For-Sale Mild EPHX2 42 40 CCCCCCCCNC(=O)[C@@H]1C[C@H](N)CC[C@@H]1C ZINC000147366134 CG For-Sale Mild TPP2 26 40 CCCCCCCCNC(=O)[C@@H]1C[C@H](N)CC[C@@H]1C ZINC000147366134 CG For-Sale Mild ASAH1 50 34 C[C@H](N)c1nc(C(=O)NN2CCCCC2)cs1 ZINC000147366208 CD For-Sale Anodyne CNR1 16 43 O=C(Nc1cc(Br)ccc1O)c1cccc2c1OCCN2 ZINC000147366231 EG For-Sale Anodyne KCNMA1 18 40 CCCCCC(=O)[C@H]1Cc2ccccc2O1 ZINC000147366255 BG For-Sale Anodyne TPP2 51 33 CCCCCC(=O)[C@H]1Cc2ccccc2O1 ZINC000147366255 BG For-Sale Anodyne CQSS 50 31 CC(=O)SC[C@H](CCC(=O)C(C)C)C(=O)N1CCC[C@@H]1C(=O)O ZINC000147366275 ED For-Sale Anodyne ACE 67 48 CC(=O)SC[C@H](CCC(=O)C(C)C)C(=O)N1CCC[C@@H]1C(=O)O ZINC000147366275 ED For-Sale Anodyne REN 19 53 COCCOc1ccccc1CNC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147366285 FH On-Demand Anodyne P2RX7 50 34 CCNC/C=C/C(=O)O ZINC000147366305 AC For-Sale Anodyne GABRR2 0 42 CCNC/C=C/C(=O)O ZINC000147366305 AC For-Sale Anodyne TSPAN17 0 44 COC(=O)COc1cccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c1 ZINC000147366306 EF On-Demand Anodyne CCKAR 37 41 COC(=O)COc1cccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c1 ZINC000147366306 EF On-Demand Anodyne CCR3 17 44 COC(=O)COc1cccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c1 ZINC000147366306 EF On-Demand Anodyne CCKBR 42 38 COC(=O)COc1cccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c1 ZINC000147366306 EF On-Demand Anodyne EPHX2 47 45 COC(=O)COc1cccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c1 ZINC000147366306 EF On-Demand Anodyne KCNK3 40 34 CC(C)CCCCN[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000147366350 CI For-Sale Anodyne DRD2 0 44 CC(C)CCCCN[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000147366350 CI For-Sale Anodyne DRD4 37 45 CC(C)CCCCN[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000147366350 CI For-Sale Anodyne ACHE 24 43 CC(C)CCCCN[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000147366350 CI For-Sale Anodyne DRD3 23 45 CC(C)CCCCN[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000147366350 CI For-Sale Anodyne SIGMAR1 57 51 CC(C)CCCCN[C@@H]1CCCN(Cc2ccccc2)C1 ZINC000147366350 CI For-Sale Anodyne BIRC2 42 48 C[C@@H](N)c1nc(C(=O)NN2CCCCC2)cs1 ZINC000147366420 CD For-Sale Anodyne CNR1 16 43 CC(C)(C)c1[nH]c(SCc2cccc(F)c2F)nc(=O)c1C#N ZINC000147366428 EH Annotated Mild CXCR2 27 72 Cc1ccc(O)c(NC(=O)c2cccc3c2OCCN3)c1 ZINC000147366441 CF For-Sale Anodyne KCNMA1 35 45 CC(C)CCO[C@@H](C)C(=O)NCc1ccccc1OC(F)(F)F ZINC000147366442 EH On-Demand Anodyne ANPEP 17 40 CCCCCCC[C@@H](Cc1ccc(F)c(F)c1)NCCC ZINC000147366460 CK For-Sale Mild S1PR2 44 37 CC(=O)SC[C@@H](CCC(=O)C(C)C)C(=O)N1CCC[C@@H]1C(=O)O ZINC000147366498 ED For-Sale Anodyne ACE 67 48 CC(=O)SC[C@@H](CCC(=O)C(C)C)C(=O)N1CCC[C@@H]1C(=O)O ZINC000147366498 ED For-Sale Anodyne REN 19 53 O=C(CCCCNC(=O)c1csc(-c2cscn2)n1)NO ZINC000147366522 ED Annotated Mild HDAC8 18 43 O=C(CCCCNC(=O)c1csc(-c2cscn2)n1)NO ZINC000147366522 ED Annotated Mild HDAC10 32 47 O=C(CCCCNC(=O)c1csc(-c2cscn2)n1)NO ZINC000147366522 ED Annotated Mild HDAC1 25 45 O=C(CCCCNC(=O)c1csc(-c2cscn2)n1)NO ZINC000147366522 ED Annotated Mild HDAC2 22 43 O=C(CCCCNC(=O)c1csc(-c2cscn2)n1)NO ZINC000147366522 ED Annotated Mild HDAC6 27 47 O=C(CCCCNC(=O)c1csc(-c2cscn2)n1)NO ZINC000147366522 ED Annotated Mild HDAC9 40 37 O=C(CCCCNC(=O)c1csc(-c2cscn2)n1)NO ZINC000147366522 ED Annotated Mild HDA106 0 42 COCCOc1ccccc1CNC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147366529 FH On-Demand Anodyne P2RX7 50 34 CCCCCCCCNC(=O)[C@@H]1C[C@@H](N)CC[C@@H]1C ZINC000147366536 CG For-Sale Mild EPHX2 42 40 CCCCCCCCNC(=O)[C@@H]1C[C@@H](N)CC[C@@H]1C ZINC000147366536 CG For-Sale Mild TPP2 26 40 CCCCCCCCNC(=O)[C@@H]1C[C@@H](N)CC[C@@H]1C ZINC000147366536 CG For-Sale Mild ASAH1 50 34 COC(=O)COc1cccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147366551 EF On-Demand Anodyne CCKAR 37 41 COC(=O)COc1cccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147366551 EF On-Demand Anodyne CCR3 17 44 COC(=O)COc1cccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147366551 EF On-Demand Anodyne CCKBR 42 38 COC(=O)COc1cccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147366551 EF On-Demand Anodyne EPHX2 47 45 COC(=O)COc1cccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c1 ZINC000147366551 EF On-Demand Anodyne KCNK3 40 34 CC(C)CCCCN[C@H]1CCCN(Cc2ccccc2)C1 ZINC000147366556 CI For-Sale Anodyne DRD2 0 44 CC(C)CCCCN[C@H]1CCCN(Cc2ccccc2)C1 ZINC000147366556 CI For-Sale Anodyne DRD4 37 45 CC(C)CCCCN[C@H]1CCCN(Cc2ccccc2)C1 ZINC000147366556 CI For-Sale Anodyne ACHE 24 43 CC(C)CCCCN[C@H]1CCCN(Cc2ccccc2)C1 ZINC000147366556 CI For-Sale Anodyne DRD3 23 45 CC(C)CCCCN[C@H]1CCCN(Cc2ccccc2)C1 ZINC000147366556 CI For-Sale Anodyne SIGMAR1 57 51 CC(C)CCCCN[C@H]1CCCN(Cc2ccccc2)C1 ZINC000147366556 CI For-Sale Anodyne BIRC2 42 48 CCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147366615 CC For-Sale Anodyne MAOA 20 40 Cc1ccc(NC(=O)c2cccc3c2OCCN3)c(C)n1 ZINC000147366646 CF For-Sale Anodyne G2YM83_BOTF4 51 33 COC(=O)COc1cccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000147366661 EF On-Demand Anodyne CCKAR 37 41 COC(=O)COc1cccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000147366661 EF On-Demand Anodyne CCR3 17 44 COC(=O)COc1cccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000147366661 EF On-Demand Anodyne CCKBR 42 38 COC(=O)COc1cccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000147366661 EF On-Demand Anodyne EPHX2 47 45 COC(=O)COc1cccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c1 ZINC000147366661 EF On-Demand Anodyne KCNK3 40 34 CC(C)CCO[C@H](C)C(=O)NCc1ccccc1OC(F)(F)F ZINC000147366666 EH On-Demand Anodyne ANPEP 17 40 CCCCCCC[C@H](Cc1ccc(F)c(F)c1)NCCC ZINC000147366678 CK For-Sale Mild S1PR2 44 37 CC(=O)SC[C@H](CCC(=O)C(C)C)C(=O)N1CCC[C@H]1C(=O)O ZINC000147366683 ED For-Sale Anodyne ACE 67 48 CC(=O)SC[C@H](CCC(=O)C(C)C)C(=O)N1CCC[C@H]1C(=O)O ZINC000147366683 ED For-Sale Anodyne REN 19 53 COCCOc1ccccc1CNC(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147366688 FH On-Demand Anodyne P2RX7 50 34 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne F2 37 44 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne KLK3 44 35 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne TRY2_BOVIN 76 35 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne CTSK 20 42 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne F11 15 40 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne PCSK5 60 38 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne FURIN 83 40 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne F7 21 41 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne ST14 78 34 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne LEF 31 42 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne POLG_WNV 58 32 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne NPFFR1 52 35 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne TMPRSS11D 41 35 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366778 GD On-Demand Anodyne TMPRSS6 64 30 C[C@@H](N)C(=O)Oc1ccc(O)cc1 ZINC000147366815 AC For-Sale Anodyne CA14 0 42 C[C@@H](N)C(=O)Oc1ccc(O)cc1 ZINC000147366815 AC For-Sale Anodyne SLC1A6 47 30 C[C@@H](N)C(=O)Oc1ccc(O)cc1 ZINC000147366815 AC For-Sale Anodyne SLC1A7 47 30 C[C@@H](N)C(=O)Oc1ccc(O)cc1 ZINC000147366815 AC For-Sale Anodyne IMPA2 0 40 Cc1cccc(NC(=O)C(=O)NCc2ccc(C(=O)N3C[C@H](C)O[C@H](C)C3)cc2)c1 ZINC000147366849 HE On-Demand Anodyne KCNK3 46 35 O=C(Nc1ccc(Cl)c(Br)c1)c1cccc2c1OCCN2 ZINC000147366870 FI For-Sale Anodyne NR2E3 62 32 COC(=O)COc1cccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c1 ZINC000147366873 EF On-Demand Anodyne CCKAR 37 41 COC(=O)COc1cccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c1 ZINC000147366873 EF On-Demand Anodyne CCR3 17 44 COC(=O)COc1cccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c1 ZINC000147366873 EF On-Demand Anodyne CCKBR 46 41 COC(=O)COc1cccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c1 ZINC000147366873 EF On-Demand Anodyne EPHX2 47 45 COC(=O)COc1cccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c1 ZINC000147366873 EF On-Demand Anodyne KCNK3 40 34 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne HTR1A 108 53 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne ADRA2A 16 44 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne DRD2 90 53 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne DRD1 31 46 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne DRD4 51 48 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne ADRA1D 92 48 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne HTR1B 19 40 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne HTR2A 48 46 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne HTR2C 21 41 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne ADRA1A 82 48 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne ADRA1B 74 48 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne DRD3 86 46 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne HTR7 65 47 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne HSD11B1 15 40 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne HTR6 27 40 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne TACR3 21 42 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne ABCB1 29 41 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne PKM 36 40 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne TGM2 36 41 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne PTGDR2 29 42 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne F13A1 46 41 COc1ccccc1N1CCN(S(=O)(=O)c2cccc(CC(=O)O)c2)CC1 ZINC000147366879 GD On-Demand Anodyne AKR1C3 58 49 CC(=O)SC[C@@H](CCC(=O)C(C)C)C(=O)N1CCC[C@H]1C(=O)O ZINC000147366935 ED For-Sale Anodyne ACE 67 48 CC(=O)SC[C@@H](CCC(=O)C(C)C)C(=O)N1CCC[C@H]1C(=O)O ZINC000147366935 ED For-Sale Anodyne REN 19 53 CCNc1cc(Oc2cccc(Cl)c2Cl)cc([N+](=O)[O-])c1 ZINC000147366963 EK For-Sale Bother TBXA2R 21 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne F2 37 44 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne KLK3 44 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne TRY2_BOVIN 76 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne CTSK 20 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne F11 15 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne PCSK5 60 38 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne FURIN 83 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne F7 21 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne ST14 78 34 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne LEF 31 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne POLG_WNV 58 32 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne NPFFR1 52 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne TMPRSS11D 41 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(S(=O)(=O)NC(C)C)c1 ZINC000147366988 GD On-Demand Anodyne TMPRSS6 64 30 c1ncc(-c2noc([C@H]3C[C@@H]4CC[C@@H]3N4)n2)s1 ZINC000147366996 BD For-Sale Anodyne CHRNA7 0 40 CCCCCCCCNC(=O)CCC1CCC(N)CC1 ZINC000147367002 CH For-Sale Mild FAAH 0 49 CCCCCCCCNC(=O)CCC1CCC(N)CC1 ZINC000147367002 CH For-Sale Mild EPHX2 40 50 CCCCCCCCNC(=O)CCC1CCC(N)CC1 ZINC000147367002 CH For-Sale Mild ASAH1 72 38 CCCCCCCCNC(=O)CCC1CCC(N)CC1 ZINC000147367002 CH For-Sale Mild LASR 48 34 CCCCCCCCNC(=O)CCC1CCC(N)CC1 ZINC000147367002 CH For-Sale Mild NOD1 37 40 Cc1cccc(NC(=O)C(=O)NCc2ccc(C(=O)N3C[C@H](C)O[C@@H](C)C3)cc2)c1 ZINC000147367004 HE On-Demand Anodyne KCNK3 46 35 COC(=O)COc1cccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147367064 GC On-Demand Anodyne CCR3 52 44 COC(=O)COc1cccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147367064 GC On-Demand Anodyne EPHX2 57 48 CC[C@H](CNS(=O)(=O)c1c(C)cc(C)cc1C)CC(=O)O ZINC000147367068 DE On-Demand Anodyne NR3C1 0 44 CC[C@H](CNS(=O)(=O)c1c(C)cc(C)cc1C)CC(=O)O ZINC000147367068 DE On-Demand Anodyne NR3C2 29 44 CC[C@H](CNS(=O)(=O)c1c(C)cc(C)cc1C)CC(=O)O ZINC000147367068 DE On-Demand Anodyne ITGAV 40 41 CC[C@H](CNS(=O)(=O)c1c(C)cc(C)cc1C)CC(=O)O ZINC000147367068 DE On-Demand Anodyne KCS20 0 40 CC[C@H](CNS(=O)(=O)c1c(C)cc(C)cc1C)CC(=O)O ZINC000147367068 DE On-Demand Anodyne FAE1 0 40 O=C(NCC1CCC1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147367098 EG For-Sale Anodyne CACNA1I 57 35 C[C@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367178 CC For-Sale Anodyne CA2 67 51 C[C@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367178 CC For-Sale Anodyne CA1 60 51 C[C@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367178 CC For-Sale Anodyne CA7 44 43 C[C@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367178 CC For-Sale Anodyne CA4 41 39 C[C@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367178 CC For-Sale Anodyne CA12 53 46 C[C@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367178 CC For-Sale Anodyne CA9 56 44 C[C@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367178 CC For-Sale Anodyne CAH_METTE 27 43 C[C@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367178 CC For-Sale Anodyne MTCA1 47 40 C[C@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367178 CC For-Sale Anodyne P96878_MYCTU 57 40 CCCCCCCCNC(=O)C[C@@H]1CCCC[C@@H]1N ZINC000147367209 CG For-Sale Mild EPHX2 36 44 CCCCCCCCNC(=O)C[C@@H]1CCCC[C@@H]1N ZINC000147367209 CG For-Sale Mild ASAH1 64 36 CCCCCCCCNC(=O)C[C@@H]1CCCC[C@@H]1N ZINC000147367209 CG For-Sale Mild LASR 44 31 CN(CCC(=O)O)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147367265 BD For-Sale Anodyne FFAR1 0 41 CN(CCC(=O)O)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147367265 BD For-Sale Anodyne GPR88 0 49 Cc1[nH]c(SCc2cccc(F)c2F)nc(=O)c1C#N ZINC000147367277 CF Annotated Mild CTSB 15 42 Cc1[nH]c(SCc2cccc(F)c2F)nc(=O)c1C#N ZINC000147367277 CF Annotated Mild CXCR2 29 76 Cc1[nH]c(SCc2cccc(F)c2F)nc(=O)c1C#N ZINC000147367277 CF Annotated Mild NS5B 22 40 CC[C@@H](CNS(=O)(=O)c1c(C)cc(C)cc1C)CC(=O)O ZINC000147367279 DE On-Demand Anodyne NR3C1 0 44 CC[C@@H](CNS(=O)(=O)c1c(C)cc(C)cc1C)CC(=O)O ZINC000147367279 DE On-Demand Anodyne NR3C2 29 44 CC[C@@H](CNS(=O)(=O)c1c(C)cc(C)cc1C)CC(=O)O ZINC000147367279 DE On-Demand Anodyne ITGAV 40 41 CC[C@@H](CNS(=O)(=O)c1c(C)cc(C)cc1C)CC(=O)O ZINC000147367279 DE On-Demand Anodyne KCS20 0 40 CC[C@@H](CNS(=O)(=O)c1c(C)cc(C)cc1C)CC(=O)O ZINC000147367279 DE On-Demand Anodyne FAE1 0 40 COC(=O)COc1cccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147367282 GC On-Demand Anodyne CCR3 52 44 COC(=O)COc1cccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147367282 GC On-Demand Anodyne EPHX2 57 48 O=C(CNC(=O)Nc1cccnc1N1CCCC1)Nc1ccc(F)cc1 ZINC000147367305 FF On-Demand Anodyne KCNQ2 62 43 O=C(CNC(=O)Nc1cccnc1N1CCCC1)Nc1ccc(F)cc1 ZINC000147367305 FF On-Demand Anodyne TRPV1 21 40 O=C(CNC(=O)Nc1cccnc1N1CCCC1)Nc1ccc(F)cc1 ZINC000147367305 FF On-Demand Anodyne P2RY1 49 41 O=C(NCC1CCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147367315 CF On-Demand Anodyne CACNA1H 24 42 O=C(NCC1CCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147367315 CF On-Demand Anodyne CCR3 28 40 O=C(NCC1CCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147367315 CF On-Demand Anodyne EPHX2 18 60 O=C(NCC1CCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147367315 CF On-Demand Anodyne CACNA1I 92 48 CC(C)N1C(=O)COc2ccc(Cl)cc21 ZINC000147367360 BE In-Stock Anodyne SLC5A2 36 47 C[C@@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367369 CC For-Sale Anodyne CA2 67 51 C[C@@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367369 CC For-Sale Anodyne CA1 60 51 C[C@@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367369 CC For-Sale Anodyne CA7 44 43 C[C@@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367369 CC For-Sale Anodyne CA4 41 39 C[C@@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367369 CC For-Sale Anodyne CA12 53 46 C[C@@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367369 CC For-Sale Anodyne CA9 56 44 C[C@@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367369 CC For-Sale Anodyne CAH_METTE 27 43 C[C@@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367369 CC For-Sale Anodyne MTCA1 47 40 C[C@@H]1OCC[C@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367369 CC For-Sale Anodyne P96878_MYCTU 57 40 CC(C)(O)Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147367399 GD Annotated Mild HDAC1 24 78 CC(C)(O)Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147367399 GD Annotated Mild HDAC3 51 78 CC(C)(O)Cc1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147367399 GD Annotated Mild HDAC6 23 78 c1ncc(-c2noc([C@H]3C[C@H]4CC[C@@H]3N4)n2)s1 ZINC000147367411 BD For-Sale Anodyne CHRNA7 0 40 C[C@]1(CNC(=O)c2cccc3c2OCCN3)CCCO1 ZINC000147367428 CD For-Sale Anodyne HCN1 52 34 C[C@]1(CNC(=O)c2cccc3c2OCCN3)CCCO1 ZINC000147367428 CD For-Sale Anodyne HCN4 48 32 CN(CCC(=O)O)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147367438 BD For-Sale Anodyne FFAR1 0 41 CN(CCC(=O)O)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147367438 BD For-Sale Anodyne GPR88 0 49 CCCCCCCCNC(=O)C[C@H]1CCCC[C@@H]1N ZINC000147367455 CG For-Sale Mild EPHX2 36 44 CCCCCCCCNC(=O)C[C@H]1CCCC[C@@H]1N ZINC000147367455 CG For-Sale Mild ASAH1 64 36 CCCCCCCCNC(=O)C[C@H]1CCCC[C@@H]1N ZINC000147367455 CG For-Sale Mild LASR 44 31 COC(=O)COc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147367534 GF On-Demand Anodyne NOS2 63 33 COC(=O)COc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147367534 GF On-Demand Anodyne ROCK2 29 46 COC(=O)COc1cccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147367534 GF On-Demand Anodyne NAMPT 34 41 CNC(=O)CNC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147367558 ED For-Sale Anodyne F7 21 41 C[C@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367566 CC For-Sale Anodyne CA2 67 51 C[C@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367566 CC For-Sale Anodyne CA1 60 51 C[C@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367566 CC For-Sale Anodyne CA7 44 43 C[C@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367566 CC For-Sale Anodyne CA4 41 39 C[C@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367566 CC For-Sale Anodyne CA12 53 46 C[C@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367566 CC For-Sale Anodyne CA9 56 44 C[C@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367566 CC For-Sale Anodyne CAH_METTE 27 43 C[C@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367566 CC For-Sale Anodyne MTCA1 47 40 C[C@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367566 CC For-Sale Anodyne P96878_MYCTU 57 40 CCc1ncc(C(=O)Nc2cccc(S(=O)(=O)N3CCN(CC)CC3)c2)s1 ZINC000147367598 HE On-Demand Anodyne TGM2 43 33 CCc1ncc(C(=O)Nc2cccc(S(=O)(=O)N3CCN(CC)CC3)c2)s1 ZINC000147367598 HE On-Demand Anodyne F13A1 48 39 COCCOc1ccccc1CNC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147367619 FF On-Demand Anodyne MTNR1A 44 40 COCCOc1ccccc1CNC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147367619 FF On-Demand Anodyne ROCK2 31 42 CNc1nc(Oc2cccc(Cl)c2Cl)nc(N(C)C)n1 ZINC000147367621 DG For-Sale Anodyne ALS 15 40 CCCCCCCCNC(=O)C[C@@H]1CCCC[C@H]1N ZINC000147367638 CG For-Sale Mild EPHX2 36 44 CCCCCCCCNC(=O)C[C@@H]1CCCC[C@H]1N ZINC000147367638 CG For-Sale Mild ASAH1 64 36 CCCCCCCCNC(=O)C[C@@H]1CCCC[C@H]1N ZINC000147367638 CG For-Sale Mild LASR 44 31 C[C@@]1(CNC(=O)c2cccc3c2OCCN3)CCCO1 ZINC000147367640 CD For-Sale Anodyne HCN1 52 34 C[C@@]1(CNC(=O)c2cccc3c2OCCN3)CCCO1 ZINC000147367640 CD For-Sale Anodyne HCN4 48 32 CN(CCC(=O)O)C(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147367659 BD For-Sale Anodyne FFAR1 0 41 CN(CCC(=O)O)C(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147367659 BD For-Sale Anodyne GPR88 0 49 CSCC[C@@H](C)NC=O ZINC000147367720 AC For-Sale Anodyne ADH1A 0 50 CSCC[C@@H](C)NC=O ZINC000147367720 AC For-Sale Anodyne ADH1B 0 50 CSCC[C@@H](C)NC=O ZINC000147367720 AC For-Sale Anodyne ADH1C 0 50 CN(CCC(=O)O)C(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147367778 BD For-Sale Anodyne FFAR1 0 41 CN(CCC(=O)O)C(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147367778 BD For-Sale Anodyne GPR88 0 49 CCCCCCCCNC(=O)C[C@H]1CCCC[C@H]1N ZINC000147367794 CG For-Sale Mild EPHX2 36 44 CCCCCCCCNC(=O)C[C@H]1CCCC[C@H]1N ZINC000147367794 CG For-Sale Mild ASAH1 64 36 CCCCCCCCNC(=O)C[C@H]1CCCC[C@H]1N ZINC000147367794 CG For-Sale Mild LASR 44 31 CCCCNS(=O)(=O)c1cccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147367796 GG On-Demand Bother TBXA2R 20 41 CCCCNS(=O)(=O)c1cccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147367796 GG On-Demand Bother KCNK3 72 39 CCCCNS(=O)(=O)c1cccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)c1 ZINC000147367796 GG On-Demand Bother KCNK9 44 39 C[C@@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367841 CC For-Sale Anodyne CA2 67 51 C[C@@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367841 CC For-Sale Anodyne CA1 60 51 C[C@@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367841 CC For-Sale Anodyne CA7 44 43 C[C@@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367841 CC For-Sale Anodyne CA4 41 39 C[C@@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367841 CC For-Sale Anodyne CA12 53 46 C[C@@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367841 CC For-Sale Anodyne CA9 56 44 C[C@@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367841 CC For-Sale Anodyne CAH_METTE 27 43 C[C@@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367841 CC For-Sale Anodyne MTCA1 47 40 C[C@@H]1OCC[C@@H]1Nc1ccc(S(N)(=O)=O)cc1 ZINC000147367841 CC For-Sale Anodyne P96878_MYCTU 57 40 CNC(=O)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147367862 CC On-Demand Anodyne CACNA1I 42 36 CSCC[C@H](C)NC=O ZINC000147367941 AC For-Sale Anodyne ADH1A 0 50 CSCC[C@H](C)NC=O ZINC000147367941 AC For-Sale Anodyne ADH1B 0 50 CSCC[C@H](C)NC=O ZINC000147367941 AC For-Sale Anodyne ADH1C 0 50 CCCCCCCCNC(=O)[C@@H]1C[C@H](C)CC[C@@H]1N ZINC000147367985 CG For-Sale Mild EPHX2 42 40 CCCCCCCCNC(=O)[C@@H]1C[C@H](C)CC[C@@H]1N ZINC000147367985 CG For-Sale Mild TPP2 31 43 CCCCCCCCNC(=O)[C@@H]1C[C@H](C)CC[C@@H]1N ZINC000147367985 CG For-Sale Mild ASAH1 83 35 C[C@H]1OCC[C@H]1Nc1cccc(S(N)(=O)=O)c1 ZINC000147368049 CC For-Sale Anodyne CA2 18 44 C[C@H]1OCC[C@H]1Nc1cccc(S(N)(=O)=O)c1 ZINC000147368049 CC For-Sale Anodyne CA4 20 44 CCOC(=O)c1ccc(C#N)c(I)c1 ZINC000147368062 DE In-Stock Mild CA14 0 54 CN(CCC(=O)O)C(=O)C1[C@H]2CCCC[C@H]12 ZINC000147368092 BD On-Demand Anodyne PHF8 0 40 O=C(NCc1cccc2c1OCO2)c1cnn(-c2ccccc2Cl)c1 ZINC000147368106 FG On-Demand Anodyne P2RX7 15 45 O=C(NCc1cccc2c1OCO2)c1cnn(-c2ccccc2Cl)c1 ZINC000147368106 FG On-Demand Anodyne SCN2A 18 41 O=C(NCc1cccc2c1OCO2)c1cnn(-c2ccccc2Cl)c1 ZINC000147368106 FG On-Demand Anodyne SCN10A 37 41 CCNc1nc(OC)nc(Oc2cccc(Cl)c2Cl)n1 ZINC000147368185 DG For-Sale Anodyne ALS 46 42 C[C@@H]1OCC[C@H]1Nc1cccc(S(N)(=O)=O)c1 ZINC000147368246 CC For-Sale Anodyne CA2 18 44 C[C@@H]1OCC[C@H]1Nc1cccc(S(N)(=O)=O)c1 ZINC000147368246 CC For-Sale Anodyne CA4 20 44 COc1ccc(-c2ccc(C)c(N)c2)nc1 ZINC000147368268 BF For-Sale Anodyne CYP11B1 15 52 CN(CCC(=O)O)C(=O)C1[C@H]2CCCC[C@@H]12 ZINC000147368294 BD For-Sale Anodyne PHF8 0 40 COC(=O)c1cc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc(C(=O)OC)c1 ZINC000147368327 HE On-Demand Anodyne CCR3 41 38 COC(=O)c1cc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc(C(=O)OC)c1 ZINC000147368327 HE On-Demand Anodyne FUCA1 18 40 COC(=O)c1cc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc(C(=O)OC)c1 ZINC000147368327 HE On-Demand Anodyne EPHX2 15 44 COC(=O)c1cc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc(C(=O)OC)c1 ZINC000147368327 HE On-Demand Anodyne F7 26 40 COC(=O)c1cc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc(C(=O)OC)c1 ZINC000147368327 HE On-Demand Anodyne PRMT3 19 44 CCc1cncnc1-c1ccco1 ZINC000147368363 AE For-Sale Anodyne ADORA1 17 42 CCc1cncnc1-c1ccco1 ZINC000147368363 AE For-Sale Anodyne ADORA2A 18 42 CCc1cncnc1-c1ccco1 ZINC000147368363 AE For-Sale Anodyne ADORA2B 16 42 CCCCCCCCNC(=O)[C@@H]1C[C@@H](C)CC[C@@H]1N ZINC000147368425 CG For-Sale Mild EPHX2 42 40 CCCCCCCCNC(=O)[C@@H]1C[C@@H](C)CC[C@@H]1N ZINC000147368425 CG For-Sale Mild TPP2 31 43 CCCCCCCCNC(=O)[C@@H]1C[C@@H](C)CC[C@@H]1N ZINC000147368425 CG For-Sale Mild ASAH1 83 35 C[C@H]1OCC[C@@H]1Nc1cccc(S(N)(=O)=O)c1 ZINC000147368441 CC For-Sale Anodyne CA2 18 44 C[C@H]1OCC[C@@H]1Nc1cccc(S(N)(=O)=O)c1 ZINC000147368441 CC For-Sale Anodyne CA4 20 44 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(-c3ccc(NC(C)=O)cc3)cc2)C1 ZINC000147368472 HH On-Demand Anodyne TIMP3 47 31 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(-c3ccc(NC(C)=O)cc3)cc2)C1 ZINC000147368472 HH On-Demand Anodyne TGM2 63 43 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(-c3ccc(NC(C)=O)cc3)cc2)C1 ZINC000147368472 HH On-Demand Anodyne F13A1 89 43 CCO[C@@H]1CCCN(S(=O)(=O)c2ccc(-c3ccc(NC(C)=O)cc3)cc2)C1 ZINC000147368472 HH On-Demand Anodyne NAMPT 29 44 O=C1c2cc(I)ccc2CCN1Cc1cc(F)ccc1F ZINC000147368477 GH For-Sale Anodyne P2RX7 22 42 CN(CCC(=O)O)C(=O)C1[C@@H]2CCCC[C@@H]12 ZINC000147368491 BD On-Demand Anodyne PHF8 0 40 C[C@@H]1CCC[C@H](NC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147368502 FH For-Sale Anodyne EPHX2 42 39 COc1ccc2nc(CCl)n(CCNC(=O)N(C)C)c2c1 ZINC000147368609 DE For-Sale Reactive DRD4 43 32 COc1ccc2nc(CCl)n(CCNC(=O)N(C)C)c2c1 ZINC000147368609 DE For-Sale Reactive MTNR1A 43 37 COc1ccc2nc(CCl)n(CCNC(=O)N(C)C)c2c1 ZINC000147368609 DE For-Sale Reactive SCD 18 41 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(NC2CC2)nc1 ZINC000147368616 GH On-Demand Anodyne MRGPRX1 46 41 C[C@@H]1OCC[C@@H]1Nc1cccc(S(N)(=O)=O)c1 ZINC000147368618 CC For-Sale Anodyne CA2 18 44 C[C@@H]1OCC[C@@H]1Nc1cccc(S(N)(=O)=O)c1 ZINC000147368618 CC For-Sale Anodyne CA4 20 44 COc1ccccc1CC(=O)N1CCC[C@H](CCBr)C1 ZINC000147368637 EG For-Sale Reactive TACR1 16 41 COc1ccccc1CC(=O)N1CCC[C@H](CCBr)C1 ZINC000147368637 EG For-Sale Reactive CCR3 17 50 COc1ccccc1CC(=O)N1CCC[C@H](CCBr)C1 ZINC000147368637 EG For-Sale Reactive MBTPS1 49 33 COc1ccccc1CC(=O)N1CCC[C@H](CCBr)C1 ZINC000147368637 EG For-Sale Reactive ACKR3 64 33 COC(=O)COc1cccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147368668 GH On-Demand Anodyne CCR3 28 41 CCO[C@H]1CCCN(S(=O)(=O)c2ccc(-c3ccc(NC(C)=O)cc3)cc2)C1 ZINC000147368688 HH On-Demand Anodyne TIMP3 47 31 CCO[C@H]1CCCN(S(=O)(=O)c2ccc(-c3ccc(NC(C)=O)cc3)cc2)C1 ZINC000147368688 HH On-Demand Anodyne TGM2 63 43 CCO[C@H]1CCCN(S(=O)(=O)c2ccc(-c3ccc(NC(C)=O)cc3)cc2)C1 ZINC000147368688 HH On-Demand Anodyne F13A1 89 43 CCO[C@H]1CCCN(S(=O)(=O)c2ccc(-c3ccc(NC(C)=O)cc3)cc2)C1 ZINC000147368688 HH On-Demand Anodyne NAMPT 29 44 C[C@H]1CCC[C@H](NC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147368711 FH For-Sale Anodyne EPHX2 42 39 CCCCCCCCNC(=O)[C@@H]1CCC[C@H](N)[C@@H]1C ZINC000147368822 CG For-Sale Mild TPP2 27 43 CCCCCCCCNC(=O)[C@@H]1CCC[C@H](N)[C@@H]1C ZINC000147368822 CG For-Sale Mild ASAH1 50 34 Cc1ccc2c(c1)nc(CCCl)n2CCNC(=O)N(C)C ZINC000147368832 DE For-Sale Reactive HDAC1 0 41 COc1ccccc1CC(=O)N1CCC[C@@H](CCBr)C1 ZINC000147368835 EG For-Sale Reactive TACR1 16 41 COc1ccccc1CC(=O)N1CCC[C@@H](CCBr)C1 ZINC000147368835 EG For-Sale Reactive CCR3 17 50 COc1ccccc1CC(=O)N1CCC[C@@H](CCBr)C1 ZINC000147368835 EG For-Sale Reactive MBTPS1 49 33 COc1ccccc1CC(=O)N1CCC[C@@H](CCBr)C1 ZINC000147368835 EG For-Sale Reactive ACKR3 64 33 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(OC)c1OC ZINC000147368837 DD On-Demand Anodyne GRIA1 47 31 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(OC)c1OC ZINC000147368837 DD On-Demand Anodyne PCSK5 55 35 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(OC)c1OC ZINC000147368837 DD On-Demand Anodyne FURIN 61 36 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(OC)c1OC ZINC000147368837 DD On-Demand Anodyne POLG_WNV 66 36 COC(=O)COc1cccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)c1 ZINC000147368865 GH On-Demand Anodyne CCR3 28 41 C[C@@H]1CCC[C@@H](NC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147368874 FH For-Sale Anodyne EPHX2 42 39 NS(=O)(=O)c1ccc(NC2CCN(Cc3cscn3)CC2)c([N+](=O)[O-])c1 ZINC000147368926 GD On-Demand Bother SCN5A 45 37 FC(F)CNCc1ccc(OCc2ccccc2)cc1 ZINC000147368964 CH On-Demand Anodyne MAOB 27 50 FC(F)CNCc1ccc(OCc2ccccc2)cc1 ZINC000147368964 CH On-Demand Anodyne LTA4H 30 47 FC(F)CNCc1ccc(OCc2ccccc2)cc1 ZINC000147368964 CH On-Demand Anodyne SLC15A1 0 40 FC(F)CNCc1ccc(OCc2ccccc2)cc1 ZINC000147368964 CH On-Demand Anodyne TAAR1 21 50 FC(F)CNCc1ccc(OCc2ccccc2)cc1 ZINC000147368964 CH On-Demand Anodyne FFAR1 33 45 COc1cc(Br)ccc1C(=O)NCCCCC(=O)O ZINC000147368972 EE On-Demand Anodyne DRD2 15 41 COc1cc(Br)ccc1C(=O)NCCCCC(=O)O ZINC000147368972 EE On-Demand Anodyne FOLH1 47 53 COc1cc(Br)ccc1C(=O)NCCCCC(=O)O ZINC000147368972 EE On-Demand Anodyne HDA106 0 42 CC[C@H](NC(=O)c1cc(Cl)cc([N+](=O)[O-])c1)C(=O)O ZINC000147368985 CD On-Demand Bother CCKBR 77 41 Cc1cc(OCC(=O)NCC#N)ccc1S(N)(=O)=O ZINC000147368988 CB For-Sale Mild TRPV4 40 30 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(OC)c1OC ZINC000147369041 DD On-Demand Anodyne GRIA1 47 31 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(OC)c1OC ZINC000147369041 DD On-Demand Anodyne PCSK5 55 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(OC)c1OC ZINC000147369041 DD On-Demand Anodyne FURIN 61 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(OC)c1OC ZINC000147369041 DD On-Demand Anodyne POLG_WNV 66 36 COC(=O)COc1cccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147369067 GH On-Demand Anodyne CCR3 28 41 C[C@H]1CCC[C@@H](NC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147369083 FH For-Sale Anodyne EPHX2 42 39 CO[C@@H](CCl)c1cccc([N+](=O)[O-])c1 ZINC000147369088 BF For-Sale Reactive CACNA1C 54 37 CO[C@@H](CCl)c1cccc([N+](=O)[O-])c1 ZINC000147369088 BF For-Sale Reactive CACNA1D 85 37 CC(C)=CCC/C(C)=C\CC/C(C)=C\CCO ZINC000147369143 BJ For-Sale Anodyne GGPS1 55 50 CC(C)=CCC/C(C)=C\CC/C(C)=C\CCO ZINC000147369143 BJ For-Sale Anodyne FDFT1 28 61 CC(C)=CCC/C(C)=C\CC/C(C)=C\CCO ZINC000147369143 BJ For-Sale Anodyne LSS 26 41 O=C(c1ccc2c(c1)OCO2)N1CCC[C@H](CCBr)C1 ZINC000147369146 EG For-Sale Reactive SSTR3 96 33 O=C(c1ccc2c(c1)OCO2)N1CCC[C@H](CCBr)C1 ZINC000147369146 EG For-Sale Reactive L3MBTL3 47 35 O=C(O)CCCCNC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147369171 CE For-Sale Anodyne PLD1 15 44 O=C(O)CCCCNC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147369171 CE For-Sale Anodyne EPHX2 21 40 O=C(O)CCCCNC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147369171 CE For-Sale Anodyne NAMPT 19 48 O=C(O)CCCCNC(=O)[C@H]1C[C@H]1c1ccccc1 ZINC000147369171 CE For-Sale Anodyne GPR88 0 43 COc1cccc2c1c(-c1ccc(C(C)C)cc1)nc(=O)n2C(C)C ZINC000147369201 EJ For-Sale Anodyne CASR 37 47 CC(=O)N1CCC(NCC(F)F)CC1 ZINC000147369212 BC For-Sale Anodyne EPHX2 16 47 CCCCCCCCNC(=O)[C@@H]1CCC[C@@H](N)[C@@H]1C ZINC000147369252 CG For-Sale Mild TPP2 27 43 CCCCCCCCNC(=O)[C@@H]1CCC[C@@H](N)[C@@H]1C ZINC000147369252 CG For-Sale Mild ASAH1 50 34 C[C@H](N)c1ccc(NC(=O)NCCNC(=O)N(C)C)cc1 ZINC000147369253 CD For-Sale Anodyne P96878_MYCTU 16 40 C[C@H](N)c1ccc(NC(=O)NCCNC(=O)N(C)C)cc1 ZINC000147369253 CD For-Sale Anodyne PSBA 0 51 CC(C)CCCCNS(=O)(=O)c1cccc(C(=O)O)c1 ZINC000147369256 CE For-Sale Anodyne HTR7 21 41 CC(C)CCCCNS(=O)(=O)c1cccc(C(=O)O)c1 ZINC000147369256 CE For-Sale Anodyne CASP3 0 40 CC(C)CCCCNS(=O)(=O)c1cccc(C(=O)O)c1 ZINC000147369256 CE For-Sale Anodyne FBP1 29 40 CC(C)CCCCNS(=O)(=O)c1cccc(C(=O)O)c1 ZINC000147369256 CE For-Sale Anodyne AKR1C3 65 61 COC(=O)COc1cccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)c1 ZINC000147369257 GH On-Demand Anodyne CCR3 28 41 C[C@@H]1CCC[C@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147369284 DH On-Demand Anodyne EPHX2 42 47 CO[C@H](CCl)c1cccc([N+](=O)[O-])c1 ZINC000147369303 BF For-Sale Reactive CACNA1C 54 37 CO[C@H](CCl)c1cccc([N+](=O)[O-])c1 ZINC000147369303 BF For-Sale Reactive CACNA1D 85 37 O=C(c1ccc2c(c1)OCO2)N1CCC[C@@H](CCBr)C1 ZINC000147369373 EG For-Sale Reactive SSTR3 96 33 O=C(c1ccc2c(c1)OCO2)N1CCC[C@@H](CCBr)C1 ZINC000147369373 EG For-Sale Reactive L3MBTL3 47 35 O=C(O)CCCCNC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147369389 CE For-Sale Anodyne PLD1 15 44 O=C(O)CCCCNC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147369389 CE For-Sale Anodyne EPHX2 21 40 O=C(O)CCCCNC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147369389 CE For-Sale Anodyne NAMPT 19 48 O=C(O)CCCCNC(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147369389 CE For-Sale Anodyne GPR88 0 43 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccc(F)cc1)NO ZINC000147369425 HG Annotated Mild HDAC10 27 40 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccc(F)cc1)NO ZINC000147369425 HG Annotated Mild HDAC1 23 65 O=C(CCCCNC(=O)c1nc(-c2nccs2)sc1-c1ccc(F)cc1)NO ZINC000147369425 HG Annotated Mild HDA106 0 40 COCc1nc(C(=O)N[C@@H](Cc2ccc(OC)cc2)c2ccc(OC)cc2)cs1 ZINC000147369459 HI On-Demand Anodyne SOAT1 19 48 C[C@@H](N)c1ccc(NC(=O)NCCNC(=O)N(C)C)cc1 ZINC000147369461 CD For-Sale Anodyne P96878_MYCTU 16 40 C[C@@H](N)c1ccc(NC(=O)NCCNC(=O)N(C)C)cc1 ZINC000147369461 CD For-Sale Anodyne PSBA 0 51 Cc1ccc(F)c(C[C@@H]2CCCCN2)c1F ZINC000147369507 BF For-Sale Anodyne LTA4H 0 41 Cc1ccc(F)c(C[C@@H]2CCCCN2)c1F ZINC000147369507 BF For-Sale Anodyne CHRNA10 31 41 C[C@H]1CCC[C@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147369512 DH On-Demand Anodyne EPHX2 42 47 CCCC(=O)N1CCC[C@@H](C(=O)Nc2cccc(CN3CCSCC3)c2C)C1 ZINC000147369558 HH On-Demand Anodyne CCR8 37 43 O=C(O)CCCCNC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147369567 CE For-Sale Anodyne PLD1 15 44 O=C(O)CCCCNC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147369567 CE For-Sale Anodyne EPHX2 21 40 O=C(O)CCCCNC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147369567 CE For-Sale Anodyne NAMPT 19 48 O=C(O)CCCCNC(=O)[C@@H]1C[C@H]1c1ccccc1 ZINC000147369567 CE For-Sale Anodyne GPR88 0 43 Cc1cc(OCCN2CCOCC2)ccc1S(N)(=O)=O ZINC000147369621 DC For-Sale Anodyne ESR1 58 36 Cc1cc(OCCN2CCOCC2)ccc1S(N)(=O)=O ZINC000147369621 DC For-Sale Anodyne ESR2 41 36 Cc1cc(OCCN2CCOCC2)ccc1S(N)(=O)=O ZINC000147369621 DC For-Sale Anodyne LTA4H 39 47 Cc1cc(OCCN2CCOCC2)ccc1S(N)(=O)=O ZINC000147369621 DC For-Sale Anodyne THRB 0 47 Cc1cc(OCCN2CCOCC2)ccc1S(N)(=O)=O ZINC000147369621 DC For-Sale Anodyne HRH3 34 57 Cc1cc(OCCN2CCOCC2)ccc1S(N)(=O)=O ZINC000147369621 DC For-Sale Anodyne SRC 15 44 Cc1cc(OCCN2CCOCC2)ccc1S(N)(=O)=O ZINC000147369621 DC For-Sale Anodyne EPHX2 16 40 Cc1cc(OCCN2CCOCC2)ccc1S(N)(=O)=O ZINC000147369621 DC For-Sale Anodyne PSMB2 46 35 Cc1cc(OCCN2CCOCC2)ccc1S(N)(=O)=O ZINC000147369621 DC For-Sale Anodyne PSMB1 41 38 Cc1cc(OCCN2CCOCC2)ccc1S(N)(=O)=O ZINC000147369621 DC For-Sale Anodyne TBK1 23 41 COCc1nc(C(=O)N[C@H](Cc2ccc(OC)cc2)c2ccc(OC)cc2)cs1 ZINC000147369654 HI On-Demand Anodyne SOAT1 19 48 CCCCCCCCNC(=O)[C@H]1[C@@H](N)CCC[C@H]1C ZINC000147369675 CG For-Sale Mild TPP2 27 43 CCCCCCCCNC(=O)[C@H]1[C@@H](N)CCC[C@H]1C ZINC000147369675 CG For-Sale Mild ASAH1 49 34 C[C@H](N)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147369687 CD For-Sale Anodyne PSBA 0 43 O=C(Cc1ccc(Cl)c(Cl)c1)N1CCC[C@H](CCBr)C1 ZINC000147369713 GJ For-Sale Reactive OPRM1 0 47 O=C(Cc1ccc(Cl)c(Cl)c1)N1CCC[C@H](CCBr)C1 ZINC000147369713 GJ For-Sale Reactive OPRK1 53 49 O=C(Cc1ccc(Cl)c(Cl)c1)N1CCC[C@H](CCBr)C1 ZINC000147369713 GJ For-Sale Reactive CCR3 35 42 CC[C@H](NC(=O)[C@@H]1[C@H]2CCc3ccccc3[C@@H]21)C(=O)O ZINC000147369724 CD For-Sale Anodyne ACE2 44 32 CC[C@H](NC(=O)[C@@H]1[C@H]2CCc3ccccc3[C@@H]21)C(=O)O ZINC000147369724 CD For-Sale Anodyne GZMB 40 32 Cc1ccc(F)c(C[C@H]2CCCCN2)c1F ZINC000147369725 BF For-Sale Anodyne LTA4H 0 41 Cc1ccc(F)c(C[C@H]2CCCCN2)c1F ZINC000147369725 BF For-Sale Anodyne CHRNA10 31 41 C[C@@H]1CCC[C@@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147369728 DH On-Demand Anodyne EPHX2 42 47 O=C(O)CCCCNC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147369781 CE For-Sale Anodyne PLD1 15 44 O=C(O)CCCCNC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147369781 CE For-Sale Anodyne EPHX2 21 40 O=C(O)CCCCNC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147369781 CE For-Sale Anodyne NAMPT 19 48 O=C(O)CCCCNC(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147369781 CE For-Sale Anodyne GPR88 0 43 CC[C@H](CNS(=O)(=O)c1ccc(F)c(F)c1)CC(=O)O ZINC000147369790 DD On-Demand Anodyne TBXA2R 48 35 CC[C@H](CNS(=O)(=O)c1ccc(F)c(F)c1)CC(=O)O ZINC000147369790 DD On-Demand Anodyne LEF 60 42 C[C@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147369825 CI For-Sale Anodyne MAOB 23 49 C[C@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147369825 CI For-Sale Anodyne LTA4H 15 45 C[C@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147369825 CI For-Sale Anodyne ACACA 30 45 C[C@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147369825 CI For-Sale Anodyne ACE2 21 41 C[C@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147369825 CI For-Sale Anodyne TAAR1 22 47 C[C@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147369825 CI For-Sale Anodyne FFAR1 28 43 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne ESR1 47 35 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne ACHE 27 42 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne HTR2A 15 40 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne SLC6A4 16 43 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne HTR3A 25 48 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne KCNH2 15 48 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne LTA4H 41 44 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne HRH3 117 64 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne SIGMAR1 30 48 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne BCHE 21 41 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne HNMT 49 36 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne PSMB2 51 40 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne PSMB1 45 43 Cc1cc(OCCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147369869 CD For-Sale Anodyne MEN1 43 39 C[C@@H](N)c1cccc(NC(=O)NCCNC(=O)N(C)C)c1 ZINC000147369912 CD For-Sale Anodyne PSBA 0 43 O=C(Cc1ccc(Cl)c(Cl)c1)N1CCC[C@@H](CCBr)C1 ZINC000147369922 GJ For-Sale Reactive OPRM1 0 47 O=C(Cc1ccc(Cl)c(Cl)c1)N1CCC[C@@H](CCBr)C1 ZINC000147369922 GJ For-Sale Reactive OPRK1 53 49 O=C(Cc1ccc(Cl)c(Cl)c1)N1CCC[C@@H](CCBr)C1 ZINC000147369922 GJ For-Sale Reactive CCR3 35 42 COc1ccc2cc(CNCCCCC(C)C)ccc2c1 ZINC000147369942 CJ For-Sale Anodyne SLC6A13 0 45 COc1ccc2cc(CNCCCCC(C)C)ccc2c1 ZINC000147369942 CJ For-Sale Anodyne LEF 79 45 COc1ccc2cc(CNCCCCC(C)C)ccc2c1 ZINC000147369942 CJ For-Sale Anodyne GPM3 0 59 C[C@H]1CCC[C@@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147369945 DH On-Demand Anodyne EPHX2 42 47 CCC(CC)CN1C(=O)C(=O)c2ccccc21 ZINC000147369989 BF For-Sale Anodyne ALDH1A1 76 58 CCC(CC)CN1C(=O)C(=O)c2ccccc21 ZINC000147369989 BF For-Sale Anodyne ALDH3A1 48 58 CCC(CC)CN1C(=O)C(=O)c2ccccc21 ZINC000147369989 BF For-Sale Anodyne CES1 26 56 CC[C@@H](CNS(=O)(=O)c1ccc(F)c(F)c1)CC(=O)O ZINC000147369994 DD On-Demand Anodyne TBXA2R 48 35 CC[C@@H](CNS(=O)(=O)c1ccc(F)c(F)c1)CC(=O)O ZINC000147369994 DD On-Demand Anodyne LEF 60 42 Cc1ccc(C(=O)NCCCCC(=O)O)cc1Br ZINC000147370000 DF On-Demand Anodyne FOLH1 40 40 Cc1ccc(C(=O)NCCCCC(=O)O)cc1Br ZINC000147370000 DF On-Demand Anodyne HDAC1 19 43 Cc1ccc(C(=O)NCCCCC(=O)O)cc1Br ZINC000147370000 DF On-Demand Anodyne HDAC2 15 43 Cc1ccc(C(=O)NCCCCC(=O)O)cc1Br ZINC000147370000 DF On-Demand Anodyne HDAC3 21 43 Cc1ccc(C(=O)NCCCCC(=O)O)cc1Br ZINC000147370000 DF On-Demand Anodyne HDAC5 15 40 Cc1ccc(C(=O)NCCCCC(=O)O)cc1Br ZINC000147370000 DF On-Demand Anodyne HDA106 0 47 NCc1cc(C(=O)NN2CCCCC2)ccn1 ZINC000147370003 BC For-Sale Anodyne CNR1 59 37 NCc1cc(C(=O)NN2CCCCC2)ccn1 ZINC000147370003 BC For-Sale Anodyne KDM4E 32 41 C[C@@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147370048 CI For-Sale Anodyne MAOB 23 49 C[C@@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147370048 CI For-Sale Anodyne LTA4H 15 45 C[C@@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147370048 CI For-Sale Anodyne ACACA 30 45 C[C@@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147370048 CI For-Sale Anodyne ACE2 21 41 C[C@@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147370048 CI For-Sale Anodyne TAAR1 22 47 C[C@@H](NCC(F)F)c1ccc(OCc2ccccc2)cc1 ZINC000147370048 CI For-Sale Anodyne FFAR1 28 43 CCCCCCCCNC(=O)[C@@H]1[C@@H](C)CCC[C@@H]1N ZINC000147370054 CG For-Sale Mild TPP2 27 43 CCCCCCCCNC(=O)[C@@H]1[C@@H](C)CCC[C@@H]1N ZINC000147370054 CG For-Sale Mild ASAH1 49 34 Nc1ncc(Cl)c(Oc2cccc(Cl)c2Cl)n1 ZINC000147370056 CH For-Sale Anodyne DFR1 18 41 CSCC[C@@H](C)NC(=O)CN ZINC000147370064 AC On-Demand Anodyne SLC15A2 0 48 Cc1cc(NC(=O)NCC(=O)Nc2ccc(F)cc2)n(-c2ccccn2)n1 ZINC000147370102 FE On-Demand Anodyne SLC11A2 41 37 CC[C@H](NC(=O)[C@H]1[C@H]2c3ccccc3CC[C@H]21)C(=O)O ZINC000147370110 CD For-Sale Anodyne ACE2 44 32 CC[C@H](NC(=O)[C@H]1[C@H]2c3ccccc3CC[C@H]21)C(=O)O ZINC000147370110 CD For-Sale Anodyne GZMB 40 32 O=C(NCC1CCCC1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147370136 EG For-Sale Anodyne CACNA1I 57 35 CN(C)c1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1 ZINC000147370145 EG For-Sale Reactive L3MBTL3 60 39 CC(C)CCCCNS(=O)(=O)c1ccc(CC(=O)O)cc1 ZINC000147370166 DE For-Sale Anodyne TBXA2R 54 41 CC(C)CCCCNS(=O)(=O)c1ccc(CC(=O)O)cc1 ZINC000147370166 DE For-Sale Anodyne TBXAS1 45 45 CC(C)CCCCNS(=O)(=O)c1ccc(CC(=O)O)cc1 ZINC000147370166 DE For-Sale Anodyne ALOX15 33 41 CSCC[C@H](C)NC(=O)CN ZINC000147370277 AC On-Demand Anodyne SLC15A2 0 48 O=C(NCC1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147370337 CG On-Demand Anodyne CACNA1H 24 42 O=C(NCC1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147370337 CG On-Demand Anodyne CCR3 30 42 O=C(NCC1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147370337 CG On-Demand Anodyne EPHX2 18 63 O=C(NCC1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147370337 CG On-Demand Anodyne CACNA1I 92 48 CN(C)c1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1 ZINC000147370347 EG For-Sale Reactive L3MBTL3 60 39 CC(C)CCCCNS(=O)(=O)c1cc(C(=O)O)ccc1F ZINC000147370375 DF For-Sale Anodyne LEF 61 40 COC(=O)c1cc2cc(NC(=O)N[C@@H]3C[C@@H]3c3ccccc3)ccc2o1 ZINC000147370395 FH On-Demand Anodyne EPHX2 26 41 NC1CCC(C(=O)NN2CCCCC2)CC1 ZINC000147370456 BD For-Sale Anodyne EPHX2 16 44 CCCCCCCCNC(=O)[C@@H]1CC[C@H](N)C[C@@H]1C ZINC000147370472 CG For-Sale Mild EPHX2 43 40 CCCCCCCCNC(=O)[C@@H]1CC[C@H](N)C[C@@H]1C ZINC000147370472 CG For-Sale Mild TPP2 31 41 CCCCCCCCNC(=O)[C@@H]1CC[C@H](N)C[C@@H]1C ZINC000147370472 CG For-Sale Mild ASAH1 55 35 O=C(NCC1CCCCC1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147370580 FH For-Sale Anodyne CACNA1I 47 33 CCOC(=O)c1c[nH]cc1-c1ccc(Br)cc1 ZINC000147370588 CH For-Sale Anodyne PRKCZ 21 40 COC(=O)c1cc2cc(NC(=O)N[C@H]3C[C@@H]3c3ccccc3)ccc2o1 ZINC000147370592 FH On-Demand Anodyne EPHX2 26 41 Cc1cc(OCC(=O)NCCC#N)ccc1S(N)(=O)=O ZINC000147370614 CC For-Sale Mild TRPV4 40 31 CC[C@H](NC(=O)c1cccc(F)c1Br)C(=O)O ZINC000147370624 DE For-Sale Anodyne MME 43 41 CC[C@H](NC(=O)c1cccc(F)c1Br)C(=O)O ZINC000147370624 DE For-Sale Anodyne ACE2 68 36 CC[C@H](NC(=O)c1cccc(F)c1Br)C(=O)O ZINC000147370624 DE For-Sale Anodyne NPR 44 35 CC[C@H](NC(=O)c1cccc(F)c1Br)C(=O)O ZINC000147370624 DE For-Sale Anodyne DAC 40 38 CC(C)COC[C@H](O)CN1CCN(c2cccc(C(F)(F)F)c2)CC1 ZINC000147370626 FF On-Demand Anodyne HTR1A 15 47 CC(C)COC[C@H](O)CN1CCN(c2cccc(C(F)(F)F)c2)CC1 ZINC000147370626 FF On-Demand Anodyne ABCB1 48 40 CC[C@H](CNS(=O)(=O)c1ccc(C(N)=O)cc1)CC(=O)O ZINC000147370670 DC On-Demand Anodyne CA2 27 40 O=C(NCC1CCCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147370788 DH For-Sale Anodyne CACNA1H 22 41 O=C(NCC1CCCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147370788 DH For-Sale Anodyne CCR3 29 44 O=C(NCC1CCCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147370788 DH For-Sale Anodyne EPHX2 17 65 O=C(NCC1CCCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147370788 DH For-Sale Anodyne CACNA1I 87 47 COC(=O)c1cc2cc(NC(=O)N[C@@H]3C[C@H]3c3ccccc3)ccc2o1 ZINC000147370792 FH On-Demand Anodyne EPHX2 26 41 CC(C)COC[C@@H](O)CN1CCN(c2cccc(C(F)(F)F)c2)CC1 ZINC000147370826 FF On-Demand Anodyne HTR1A 15 47 CC(C)COC[C@@H](O)CN1CCN(c2cccc(C(F)(F)F)c2)CC1 ZINC000147370826 FF On-Demand Anodyne ABCB1 48 40 O=C(O)C1(n2nnnc2COc2cccc(Cl)c2)CCC1 ZINC000147370833 DD For-Sale Anodyne VCP 24 42 CCOC(=O)c1n[nH]c2ccc(-c3ccccc3)cc2c1=O ZINC000147370842 CF For-Sale Anodyne GSK3B 18 55 CCOC(=O)c1n[nH]c2ccc(-c3ccccc3)cc2c1=O ZINC000147370842 CF For-Sale Anodyne GSK3A 28 55 CCOC(=O)c1n[nH]c2ccc(-c3ccccc3)cc2c1=O ZINC000147370842 CF For-Sale Anodyne ADORA3 33 42 CCOC(=O)c1n[nH]c2ccc(-c3ccccc3)cc2c1=O ZINC000147370842 CF For-Sale Anodyne AKT1 35 40 CCOC(=O)c1n[nH]c2ccc(-c3ccccc3)cc2c1=O ZINC000147370842 CF For-Sale Anodyne SLC5A2 16 40 CCOC(=O)c1n[nH]c2ccc(-c3ccccc3)cc2c1=O ZINC000147370842 CF For-Sale Anodyne TTK 34 43 CCOC(=O)c1n[nH]c2ccc(-c3ccccc3)cc2c1=O ZINC000147370842 CF For-Sale Anodyne HAO2 53 34 C#Cc1cccc(Nc2ncnc3ccc(OCc4ccc(C(=O)Nc5ccccc5N)cc4)cc23)c1 ZINC000147370860 JK Annotated Mild EGFR 99 47 C#Cc1cccc(Nc2ncnc3ccc(OCc4ccc(C(=O)Nc5ccccc5N)cc4)cc23)c1 ZINC000147370860 JK Annotated Mild MAP2K5 15 51 C#Cc1cccc(Nc2ncnc3ccc(OCc4ccc(C(=O)Nc5ccccc5N)cc4)cc23)c1 ZINC000147370860 JK Annotated Mild HDAC2 29 45 C#Cc1cccc(Nc2ncnc3ccc(OCc4ccc(C(=O)Nc5ccccc5N)cc4)cc23)c1 ZINC000147370860 JK Annotated Mild FBP1 0 47 C#Cc1cccc(Nc2ncnc3ccc(OCc4ccc(C(=O)Nc5ccccc5N)cc4)cc23)c1 ZINC000147370860 JK Annotated Mild ERBB4 50 51 C#Cc1cccc(Nc2ncnc3ccc(OCc4ccc(C(=O)Nc5ccccc5N)cc4)cc23)c1 ZINC000147370860 JK Annotated Mild EPHA8 15 51 C#Cc1cccc(Nc2ncnc3ccc(OCc4ccc(C(=O)Nc5ccccc5N)cc4)cc23)c1 ZINC000147370860 JK Annotated Mild EPHA5 24 51 C#Cc1cccc(Nc2ncnc3ccc(OCc4ccc(C(=O)Nc5ccccc5N)cc4)cc23)c1 ZINC000147370860 JK Annotated Mild MKNK1 25 51 C#Cc1cccc(Nc2ncnc3ccc(OCc4ccc(C(=O)Nc5ccccc5N)cc4)cc23)c1 ZINC000147370860 JK Annotated Mild DDR1 16 51 C#Cc1cccc(Nc2ncnc3ccc(OCc4ccc(C(=O)Nc5ccccc5N)cc4)cc23)c1 ZINC000147370860 JK Annotated Mild MAPK4 0 51 CC[C@@H](CNS(=O)(=O)c1ccc(C(N)=O)cc1)CC(=O)O ZINC000147370870 DC On-Demand Anodyne CA2 27 40 COCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147370877 DB For-Sale Anodyne CA2 30 43 COCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147370877 DB For-Sale Anodyne CA1 21 43 COCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147370877 DB For-Sale Anodyne CA9 21 43 COCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147370877 DB For-Sale Anodyne NCE103 16 41 CCCCCCCCNC(=O)[C@@H]1CC[C@@H](N)C[C@@H]1C ZINC000147370883 CG For-Sale Mild EPHX2 43 40 CCCCCCCCNC(=O)[C@@H]1CC[C@@H](N)C[C@@H]1C ZINC000147370883 CG For-Sale Mild TPP2 31 41 CCCCCCCCNC(=O)[C@@H]1CC[C@@H](N)C[C@@H]1C ZINC000147370883 CG For-Sale Mild ASAH1 55 35 Clc1cccc(NCc2nc(-c3cncs3)no2)c1 ZINC000147370914 CG For-Sale Anodyne CD38 19 41 CCNCc1cnccc1Oc1ccc(Cl)c(F)c1 ZINC000147370977 CH For-Sale Anodyne SLC6A4 16 50 CC(C)C[C@@H](C)NC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147371001 EH For-Sale Anodyne ANPEP 27 51 COC(=O)c1cc2cc(NC(=O)N[C@H]3C[C@H]3c3ccccc3)ccc2o1 ZINC000147371016 FH On-Demand Anodyne EPHX2 26 41 CCOC(=O)c1cc(-c2cccnc2)n[nH]c1=O ZINC000147371018 BD In-Stock Anodyne CYP2A6 37 43 NC(=O)c1ccc(OCC(=O)Nc2cccc(N3CCCC3)c2)cc1 ZINC000147371021 EE On-Demand Anodyne COLA 32 42 NC(=O)c1ccc(OCC(=O)Nc2cccc(N3CCCC3)c2)cc1 ZINC000147371021 EE On-Demand Anodyne CPT1A 25 42 NC(=O)c1ccc(OCC(=O)Nc2cccc(N3CCCC3)c2)cc1 ZINC000147371021 EE On-Demand Anodyne MCHR1 20 44 NC(=O)c1ccc(OCC(=O)Nc2cccc(N3CCCC3)c2)cc1 ZINC000147371021 EE On-Demand Anodyne HIF1A 24 47 Cc1cccc2c1c(-c1ccc(C(C)C)cc1)nc(=O)n2C(C)C ZINC000147371032 DK For-Sale Anodyne CASR 30 47 CN(Cc1ccoc1)C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147371043 CH On-Demand Anodyne MDM2 74 34 C[C@]1(CNC(=O)c2cc(F)ccc2O)CCCO1 ZINC000147371143 CD On-Demand Anodyne HCN4 48 32 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(-n3cccn3)c(F)c2)C1 ZINC000147371149 HF On-Demand Anodyne NPY2R 65 35 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(F)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147371151 KK Annotated Anodyne GLP1R 24 62 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2cc(F)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147371151 KK Annotated Anodyne GIPR 64 43 CCOc1ccc2cc(C(=O)Nc3cccc(CN4CCSCC4)c3C)[nH]c2c1 ZINC000147371177 HJ On-Demand Anodyne MRGPRX1 40 36 CC(C)C[C@H](C)NC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147371209 EH For-Sale Anodyne ANPEP 27 51 COC(=O)[C@H]1CCCN(C(=O)c2ccc(C)cc2F)C1 ZINC000147371212 CE On-Demand Anodyne SLC6A1 50 36 COC(=O)[C@H]1CCCN(C(=O)c2ccc(C)cc2F)C1 ZINC000147371212 CE On-Demand Anodyne HCRTR2 24 46 CN[C@@H](C)c1cccc(NC(=O)NCCNC(N)=O)c1 ZINC000147371231 CC For-Sale Anodyne F7 30 43 CN[C@@H](C)c1cccc(NC(=O)NCCNC(N)=O)c1 ZINC000147371231 CC For-Sale Anodyne ACAT 0 40 COC(=O)c1cc2cc(NC(=O)N[C@@H]3CCCN(S(C)(=O)=O)C3)ccc2o1 ZINC000147371246 GD On-Demand Anodyne EPHX2 41 38 CCCS(=O)(=O)N[C@@H](C)C(=O)Nc1cccc(N2CCCC2)c1 ZINC000147371252 ED On-Demand Anodyne LPL 41 33 CCCS(=O)(=O)N[C@@H](C)C(=O)Nc1cccc(N2CCCC2)c1 ZINC000147371252 ED On-Demand Anodyne KCNQ2 63 42 CCOC(=O)c1cc2cc([N+](=O)[O-])ccc2nn1 ZINC000147371262 BD For-Sale Bother CACNA1C 54 41 CCOC(=O)c1cc2cc([N+](=O)[O-])ccc2nn1 ZINC000147371262 BD For-Sale Bother CACNA1D 82 40 CCOC(=O)c1cc2cc([N+](=O)[O-])ccc2nn1 ZINC000147371262 BD For-Sale Bother CTRB1 29 44 CCOC(=O)c1cc2cc([N+](=O)[O-])ccc2nn1 ZINC000147371262 BD For-Sale Bother KCNMA1 16 40 CN(Cc1ccoc1)C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147371281 CH On-Demand Anodyne MDM2 74 34 NCCCC(=O)NN1CCCCC1 ZINC000147371315 AC For-Sale Anodyne ABAT 43 36 CCCCCCCCNC(=O)CC[C@@H]1CCC[C@H](N)C1 ZINC000147371318 CH For-Sale Mild EPHX2 43 44 CCCCCCCCNC(=O)CC[C@@H]1CCC[C@H](N)C1 ZINC000147371318 CH For-Sale Mild LASR 48 34 C[C@@]1(CNC(=O)c2cc(F)ccc2O)CCCO1 ZINC000147371347 CD On-Demand Anodyne HCN4 48 32 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(-n3cccn3)c(F)c2)C1 ZINC000147371358 HF On-Demand Anodyne NPY2R 65 35 Clc1ccc2c(N(CCBr)C3CCCC3)ccnc2c1 ZINC000147371395 FK For-Sale Reactive HRP1_PLAFA 95 41 Clc1ccc2c(N(CCBr)C3CCCC3)ccnc2c1 ZINC000147371395 FK For-Sale Reactive HNMT 56 36 COC(=O)[C@@H]1CCCN(C(=O)c2ccc(C)cc2F)C1 ZINC000147371398 CE On-Demand Anodyne SLC6A1 50 36 COC(=O)[C@@H]1CCCN(C(=O)c2ccc(C)cc2F)C1 ZINC000147371398 CE On-Demand Anodyne HCRTR2 24 46 CC(C)C[C@@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147371434 CH For-Sale Anodyne ANPEP 17 40 COC(=O)c1cc2cc(NC(=O)N[C@H]3CCCN(S(C)(=O)=O)C3)ccc2o1 ZINC000147371439 GD On-Demand Anodyne EPHX2 41 38 CN[C@H](C)c1cccc(NC(=O)NCCNC(N)=O)c1 ZINC000147371474 CC For-Sale Anodyne F7 30 43 CN[C@H](C)c1cccc(NC(=O)NCCNC(N)=O)c1 ZINC000147371474 CC For-Sale Anodyne ACAT 0 40 CN(Cc1ccoc1)C(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147371510 CH On-Demand Anodyne MDM2 74 34 COCCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147371532 DC For-Sale Anodyne CA2 25 44 COCCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147371532 DC For-Sale Anodyne CA1 20 44 COCCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147371532 DC For-Sale Anodyne CA12 15 44 COCCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147371532 DC For-Sale Anodyne CA9 21 41 CCCCCCCCNC(=O)CC[C@H]1CCC[C@H](N)C1 ZINC000147371537 CH For-Sale Mild EPHX2 43 44 CCCCCCCCNC(=O)CC[C@H]1CCC[C@H](N)C1 ZINC000147371537 CH For-Sale Mild LASR 48 34 CC(C)C[C@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147371632 CH For-Sale Anodyne ANPEP 17 40 CC(C)CCCCNS(=O)(=O)c1ccc(F)c(C(=O)O)c1 ZINC000147371671 DF For-Sale Anodyne TBXA2R 52 38 CC(C)CCCCNS(=O)(=O)c1ccc(F)c(C(=O)O)c1 ZINC000147371671 DF For-Sale Anodyne TBXAS1 35 41 CC(C)CCCCNS(=O)(=O)c1ccc(F)c(C(=O)O)c1 ZINC000147371671 DF For-Sale Anodyne CASP3 15 51 CC(C)CCCCNS(=O)(=O)c1ccc(F)c(C(=O)O)c1 ZINC000147371671 DF For-Sale Anodyne LEF 56 48 CCNc1cn2ccnc2c(Oc2cccc(Cl)c2Cl)n1 ZINC000147371675 DI For-Sale Anodyne HIVRT 0 44 CCN[C@@H](C)c1ccc(NC(=O)NCCNC(N)=O)cc1 ZINC000147371696 CD For-Sale Anodyne F7 33 43 CN(Cc1ccoc1)C(=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147371724 CH On-Demand Anodyne MDM2 74 34 C[C@]1(CNC(=O)c2cccc3c2OCCN3)CCCS1 ZINC000147371732 CF For-Sale Anodyne HCN1 51 33 C[C@]1(CNC(=O)c2cccc3c2OCCN3)CCCS1 ZINC000147371732 CF For-Sale Anodyne HCN4 46 30 CCCCCCCCNC(=O)CC[C@@H]1CCC[C@@H](N)C1 ZINC000147371737 CH For-Sale Mild EPHX2 43 44 CCCCCCCCNC(=O)CC[C@@H]1CCC[C@@H](N)C1 ZINC000147371737 CH For-Sale Mild LASR 48 34 CCN[C@H](C)c1ccc(NC(=O)NCCNC(N)=O)cc1 ZINC000147371886 CD For-Sale Anodyne F7 33 43 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1cccc(CN(C)C)c1 ZINC000147371889 FI On-Demand Anodyne LPL 56 36 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1cccc(CN(C)C)c1 ZINC000147371889 FI On-Demand Anodyne KCNQ2 65 36 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1cccc(CN(C)C)c1 ZINC000147371889 FI On-Demand Anodyne PTGER3 24 41 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1cccc(CN(C)C)c1 ZINC000147371889 FI On-Demand Anodyne BCR 0 40 Cc1cc(N2CCCC2)ccc1NC(=O)Nc1cccc(CN(C)C)c1 ZINC000147371889 FI On-Demand Anodyne DDX3X 0 42 CCCCC(=O)[C@@H]1Cc2ccccc2O1 ZINC000147371898 BF For-Sale Anodyne TPP2 51 33 C[C@@]1(CNC(=O)c2cccc3c2OCCN3)CCCS1 ZINC000147371910 CF For-Sale Anodyne HCN1 51 33 C[C@@]1(CNC(=O)c2cccc3c2OCCN3)CCCS1 ZINC000147371910 CF For-Sale Anodyne HCN4 46 30 CCCCCCCCNC(=O)CC[C@H]1CCC[C@@H](N)C1 ZINC000147371923 CH For-Sale Mild EPHX2 43 44 CCCCCCCCNC(=O)CC[C@H]1CCC[C@@H](N)C1 ZINC000147371923 CH For-Sale Mild LASR 48 34 CSc1ccc([C@H](C)NC(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147371947 GI On-Demand Anodyne DRTS_PLAFK 19 42 CSc1ccc([C@H](C)NC(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147371947 GI On-Demand Anodyne PTGER4 30 46 CSc1ccc([C@H](C)NC(=O)c2cccn(Cc3ccccc3)c2=O)cc1 ZINC000147371947 GI On-Demand Anodyne PTGDR 33 45 Cc1c(CN2CCSCC2)cccc1NC(=O)c1[nH]c2ccc(F)cc2c1Cl ZINC000147372008 HK On-Demand Anodyne MRGPRX1 42 36 NCCC1[C@@H]2CN(Cc3ccccc3)C[C@@H]12 ZINC000147372018 BD For-Sale Anodyne DRD3 15 40 CCCCCCCCNC(=O)CC1CCC(N)CC1 ZINC000147372069 CG For-Sale Mild EPHX2 42 47 CCCCCCCCNC(=O)CC1CCC(N)CC1 ZINC000147372069 CG For-Sale Mild ASAH1 80 40 CCCCCCCCNC(=O)CC1CCC(N)CC1 ZINC000147372069 CG For-Sale Mild LASR 46 33 COC1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147372071 DF For-Sale Anodyne CACNA1H 43 36 COC1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147372071 DF For-Sale Anodyne EPHX2 27 42 COC1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147372071 DF For-Sale Anodyne CACNA1I 53 37 CCCCC(=O)[C@H]1Cc2ccccc2O1 ZINC000147372073 BF For-Sale Anodyne TPP2 51 33 CCCNc1cc(Oc2cccc(C(F)(F)F)c2)ncn1 ZINC000147372109 CI For-Sale Anodyne PDS 41 35 CN[C@@H](C)c1ccc(NC(=O)NCCNC(N)=O)cc1 ZINC000147372123 CC For-Sale Anodyne F7 34 45 CN[C@@H](C)c1ccc(NC(=O)NCCNC(N)=O)cc1 ZINC000147372123 CC For-Sale Anodyne P96878_MYCTU 29 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H]1CCCC[C@@H]1C(C)(C)C ZINC000147372129 DF On-Demand Anodyne HDAC4 15 42 COc1cccc2c1C[C@@H](CO)CO2 ZINC000147372186 AD For-Sale Anodyne HTR1B 27 58 NC(=O)c1cc(NC(=O)NCC(=O)Nc2ccc(F)cc2)ccc1Cl ZINC000147372224 FE On-Demand Anodyne F7 26 48 NC(=O)c1cc(NC(=O)NCC(=O)Nc2ccc(F)cc2)ccc1Cl ZINC000147372224 FE On-Demand Anodyne PRMT3 33 42 NC(=O)c1cc(NC(=O)NCC(=O)Nc2ccc(F)cc2)ccc1Cl ZINC000147372224 FE On-Demand Anodyne IMDH_CRYPV 25 42 CCCCCCCCNC(=O)C[C@@H]1CCC[C@H](N)C1 ZINC000147372299 CG For-Sale Mild EPHX2 41 46 CCCCCCCCNC(=O)C[C@@H]1CCC[C@H](N)C1 ZINC000147372299 CG For-Sale Mild ASAH1 59 34 CN[C@H](C)c1ccc(NC(=O)NCCNC(N)=O)cc1 ZINC000147372309 CC For-Sale Anodyne F7 34 45 CN[C@H](C)c1ccc(NC(=O)NCCNC(N)=O)cc1 ZINC000147372309 CC For-Sale Anodyne P96878_MYCTU 29 40 CN1CCC(NC(=O)Nc2cc(Br)cc(C(=O)O)c2)CC1 ZINC000147372326 FE For-Sale Anodyne EPHX2 54 47 CN1CCC(NC(=O)Nc2cc(Br)cc(C(=O)O)c2)CC1 ZINC000147372326 FE For-Sale Anodyne CXCR3 19 43 C[C@@H](CNC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147372353 CD On-Demand Anodyne ITGAV 48 40 C[C@@H](CNC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147372353 CD On-Demand Anodyne DAC 50 42 CCNc1cc(Oc2cccc(C(F)(F)F)c2)nc(N)n1 ZINC000147372389 CG For-Sale Anodyne PDS 40 35 Cc1cc(OCCn2ccnc2)ccc1S(N)(=O)=O ZINC000147372417 CC For-Sale Anodyne CYP19A1 31 45 Cc1cc(OCCn2ccnc2)ccc1S(N)(=O)=O ZINC000147372417 CC For-Sale Anodyne TBXAS1 50 55 Cc1cc(OCCn2ccnc2)ccc1S(N)(=O)=O ZINC000147372417 CC For-Sale Anodyne CYP17A1 15 41 Cc1cc(OCCn2ccnc2)ccc1S(N)(=O)=O ZINC000147372417 CC For-Sale Anodyne HMOX2 21 43 COc1cccc2c1C[C@H](CO)CO2 ZINC000147372443 AD For-Sale Anodyne HTR1A 20 66 COc1cccc2c1C[C@H](CO)CO2 ZINC000147372443 AD For-Sale Anodyne HTR1B 27 58 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(Cn2cncn2)c1 ZINC000147372460 GF On-Demand Anodyne KCNK3 47 34 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(Cn2cncn2)c1 ZINC000147372460 GF On-Demand Anodyne KCNK9 49 34 CNCc1cccnc1Oc1ccc(Cl)c(F)c1 ZINC000147372470 CG For-Sale Anodyne SLC6A4 16 58 NCCC1[C@H]2CN(Cc3ccccc3)C[C@H]12 ZINC000147372482 BD For-Sale Anodyne DRD3 15 40 NCCC1[C@H]2CN(Cc3ccccc3)C[C@H]12 ZINC000147372482 BD For-Sale Anodyne SIGMAR1 44 47 CCCCCCCCNC(=O)C[C@H]1CCC[C@H](N)C1 ZINC000147372505 CG For-Sale Mild EPHX2 41 46 CCCCCCCCNC(=O)C[C@H]1CCC[C@H](N)C1 ZINC000147372505 CG For-Sale Mild ASAH1 59 34 C[C@H](CNC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147372523 CD On-Demand Anodyne ITGAV 48 40 C[C@H](CNC(=O)c1cccc(F)c1Cl)C(=O)O ZINC000147372523 CD On-Demand Anodyne DAC 50 42 CN1CCC(NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147372524 DE On-Demand Anodyne CACNA1H 24 41 CN1CCC(NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147372524 DE On-Demand Anodyne EPHX2 55 59 CN1CCC(NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147372524 DE On-Demand Anodyne TYRO3 41 41 CCCC[C@H](NC(N)=O)C(=O)N[C@H]1CCCC[C@@H]1C(C)(C)C ZINC000147372534 DF On-Demand Anodyne HDAC4 15 42 Cc1ccc(F)c(CCC(=O)O)c1F ZINC000147372586 BE In-Stock Anodyne FFAR1 49 45 C[C@H](NC(=O)N(C)Cc1cscn1)c1nnc2ccccn12 ZINC000147372594 DE On-Demand Anodyne CYP3A4 17 43 CCNc1nccc(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147372628 CH For-Sale Anodyne PDS 41 36 CSC1=NC(=O)/C(=C/c2ccc(C)cc2)S1 ZINC000147372632 BG For-Sale Clean HPGD 16 42 NC(=O)c1ccc(OCC(=O)Nc2cccc(Cn3cncn3)c2)cc1 ZINC000147372653 FD On-Demand Anodyne HIS3 41 41 NC(=O)c1ccc(OCC(=O)Nc2cccc(Cn3cncn3)c2)cc1 ZINC000147372653 FD On-Demand Anodyne HIF1A 25 41 CCCCCCCCNC(=O)C[C@@H]1CCC[C@@H](N)C1 ZINC000147372703 CG For-Sale Mild EPHX2 41 46 CCCCCCCCNC(=O)C[C@@H]1CCC[C@@H](N)C1 ZINC000147372703 CG For-Sale Mild ASAH1 59 34 CC[C@H](NC(=O)CCNC(=O)[C@@H]1C[C@H]1C)C(=O)O ZINC000147372710 CC For-Sale Anodyne NOD1 61 35 O=C(c1ccc2c(c1)COC2)N1CCC[C@@H]1C1CCCC1 ZINC000147372715 CH On-Demand Anodyne PREP 25 41 CCN[C@@H](C)c1cccc(NC(=O)NCCNC(N)=O)c1 ZINC000147372717 CD For-Sale Anodyne F7 29 42 COc1cc(Br)ccc1C(=O)NC[C@H](C)C(=O)O ZINC000147372724 DD On-Demand Anodyne FOLH1 25 42 COc1cc(Br)ccc1C(=O)NC[C@H](C)C(=O)O ZINC000147372724 DD On-Demand Anodyne KCNA3 25 47 COc1cc(Br)ccc1C(=O)NC[C@H](C)C(=O)O ZINC000147372724 DD On-Demand Anodyne ITGAV 42 40 COc1cc(Br)ccc1C(=O)NC[C@H](C)C(=O)O ZINC000147372724 DD On-Demand Anodyne GPR35 40 33 CC[C@H](C(=O)OC)c1c(F)ccc(C)c1F ZINC000147372784 BF For-Sale Anodyne LEF 60 35 C[C@@H](NC(=O)N(C)Cc1cscn1)c1nnc2ccccn12 ZINC000147372786 DE On-Demand Anodyne CYP3A4 17 43 CC(C)OC(=O)[C@@H](COS(C)(=O)=O)NC(=O)OC(C)(C)C ZINC000147372803 EC For-Sale Mild PAPA1_CARPA 47 37 CC(C)OC(=O)[C@@H](COS(C)(=O)=O)NC(=O)OC(C)(C)C ZINC000147372803 EC For-Sale Mild CTSK 17 42 CC(C)OC(=O)[C@@H](COS(C)(=O)=O)NC(=O)OC(C)(C)C ZINC000147372803 EC For-Sale Mild FPR1 42 36 CNc1cc(Oc2cccc(C(F)(F)F)c2)nc(C)n1 ZINC000147372830 CH For-Sale Anodyne PDS 40 34 Cc1cc(OCCCn2ccnc2)ccc1S(N)(=O)=O ZINC000147372855 CD For-Sale Anodyne CYP19A1 27 50 Cc1cc(OCCCn2ccnc2)ccc1S(N)(=O)=O ZINC000147372855 CD For-Sale Anodyne TBXAS1 56 49 Cc1cc(OCCCn2ccnc2)ccc1S(N)(=O)=O ZINC000147372855 CD For-Sale Anodyne HMOX1 19 49 Cc1cc(OCCCn2ccnc2)ccc1S(N)(=O)=O ZINC000147372855 CD For-Sale Anodyne HMOX2 52 48 Cc1cc(OCCCn2ccnc2)ccc1S(N)(=O)=O ZINC000147372855 CD For-Sale Anodyne QPCT 40 39 C[C@H](c1ccc(C(=O)NCc2nn[nH]n2)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147372910 KK Annotated Anodyne GCGR 30 80 C[C@H](c1ccc(C(=O)NCc2nn[nH]n2)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147372910 KK Annotated Anodyne GLP1R 18 71 CCCCCCCCNC(=O)C[C@H]1CCC[C@@H](N)C1 ZINC000147372914 CG For-Sale Mild EPHX2 41 46 CCCCCCCCNC(=O)C[C@H]1CCC[C@@H](N)C1 ZINC000147372914 CG For-Sale Mild ASAH1 59 34 CC[C@H](NC(=O)CCNC(=O)[C@H]1C[C@H]1C)C(=O)O ZINC000147372928 CC For-Sale Anodyne NOD1 61 35 COc1cc(Br)ccc1C(=O)NC[C@@H](C)C(=O)O ZINC000147372938 DD On-Demand Anodyne FOLH1 25 42 COc1cc(Br)ccc1C(=O)NC[C@@H](C)C(=O)O ZINC000147372938 DD On-Demand Anodyne KCNA3 25 47 COc1cc(Br)ccc1C(=O)NC[C@@H](C)C(=O)O ZINC000147372938 DD On-Demand Anodyne ITGAV 42 40 COc1cc(Br)ccc1C(=O)NC[C@@H](C)C(=O)O ZINC000147372938 DD On-Demand Anodyne GPR35 40 33 CCC[C@H](NC(N)=O)C(=O)Nc1cccc(Cn2cncn2)c1 ZINC000147372954 DD On-Demand Anodyne HIS3 65 36 CCN[C@H](C)c1cccc(NC(=O)NCCNC(N)=O)c1 ZINC000147372966 CD For-Sale Anodyne F7 29 42 CC[C@@H](C(=O)OC)c1c(F)ccc(C)c1F ZINC000147372973 BF For-Sale Anodyne LEF 60 35 CC(C)OC(=O)[C@H](COS(C)(=O)=O)NC(=O)OC(C)(C)C ZINC000147372988 EC For-Sale Mild PAPA1_CARPA 47 37 CC(C)OC(=O)[C@H](COS(C)(=O)=O)NC(=O)OC(C)(C)C ZINC000147372988 EC For-Sale Mild CTSK 22 42 CC(C)OC(=O)[C@H](COS(C)(=O)=O)NC(=O)OC(C)(C)C ZINC000147372988 EC For-Sale Mild FPR1 42 36 CCc1ncc(C(=O)NCc2ccc(S(=O)(=O)N3CCCCC3)cc2)s1 ZINC000147373054 GF On-Demand Anodyne EPHX2 19 41 CCc1ncc(C(=O)NCc2ccc(S(=O)(=O)N3CCCCC3)cc2)s1 ZINC000147373054 GF On-Demand Anodyne TGM2 51 41 CCc1ncc(C(=O)NCc2ccc(S(=O)(=O)N3CCCCC3)cc2)s1 ZINC000147373054 GF On-Demand Anodyne NAMPT 129 63 CN(Cc1cscn1)C(=O)N[C@H](c1ccccc1)c1nccn1C ZINC000147373062 EF On-Demand Anodyne CYP3A4 18 41 CCCCC[C@H](NCCCCC(C)C)c1ccccc1 ZINC000147373063 CK For-Sale Anodyne SOAT1 21 48 CNc1ncc(C)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147373101 CH For-Sale Anodyne LCK 28 42 CNc1ncc(C)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147373101 CH For-Sale Anodyne P2RY1 15 44 CNc1ncc(C)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147373101 CH For-Sale Anodyne TEK 30 41 CNc1ncc(C)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147373101 CH For-Sale Anodyne PDS 41 33 CCC[C@@H](NC(N)=O)C(=O)Nc1cccc(Cn2cncn2)c1 ZINC000147373124 DD On-Demand Anodyne HIS3 65 36 CCCCCCCCNC(=O)[C@@H]1CCC[C@H](CCN)C1 ZINC000147373150 CH For-Sale Mild EPHX2 28 40 CCCCCCCCNC(=O)[C@@H]1CCC[C@H](CCN)C1 ZINC000147373150 CH For-Sale Mild TPP2 22 40 CN(C)C(=O)NCCn1c(CCCl)nc2cc(F)ccc21 ZINC000147373162 DE For-Sale Reactive HDAC1 0 40 Cc1ccc([N+](=O)[O-])cc1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147373190 FH For-Sale Reactive SLC27A4 42 31 NC(=O)[C@H]1CCCN1Cc1cccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)c1 ZINC000147373194 HE On-Demand Anodyne NPY1R 27 41 NC(=O)[C@H]1CCCN1Cc1cccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)c1 ZINC000147373194 HE On-Demand Anodyne CCR3 110 40 COC(=O)COc1cccc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000147373195 HE On-Demand Anodyne ADRB2 25 44 COC(=O)COc1cccc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000147373195 HE On-Demand Anodyne ADRB1 59 43 COC(=O)COc1cccc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000147373195 HE On-Demand Anodyne ADRB3 17 44 COC(=O)COc1cccc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c1 ZINC000147373195 HE On-Demand Anodyne ACOX1 47 38 CCCCC[C@@H](NCCCCC(C)C)c1ccccc1 ZINC000147373198 CK For-Sale Anodyne SOAT1 21 48 CC(C)(C)CC[C@H](c1ccc(C(=O)NCc2nn[nH]n2)cc1)N1C(=O)C(c2ccc(F)cc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147373200 KK Annotated Anodyne GLP1R 15 67 C[C@@H](CNC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147373202 BD For-Sale Anodyne GPR88 0 46 CN(Cc1cscn1)C(=O)N[C@@H](c1ccccc1)c1nccn1C ZINC000147373293 EF On-Demand Anodyne CYP3A4 18 41 CCNc1ncc(Cl)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147373296 DI For-Sale Anodyne PDS 45 38 CCCCCCCCNC(=O)[C@H]1CCC[C@H](CCN)C1 ZINC000147373331 CH For-Sale Mild EPHX2 28 40 CCCCCCCCNC(=O)[C@H]1CCC[C@H](CCN)C1 ZINC000147373331 CH For-Sale Mild TPP2 22 40 Cc1ccc([N+](=O)[O-])cc1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147373383 FH For-Sale Reactive SLC27A4 42 31 C[C@H](CNC(=O)[C@@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147373403 BD For-Sale Anodyne GPR88 0 46 COC(=O)COc1cccc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000147373409 HE On-Demand Anodyne ADRB2 25 44 COC(=O)COc1cccc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000147373409 HE On-Demand Anodyne ADRB1 59 43 COC(=O)COc1cccc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000147373409 HE On-Demand Anodyne ADRB3 17 44 COC(=O)COc1cccc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c1 ZINC000147373409 HE On-Demand Anodyne ACOX1 47 38 Nc1nonc1C(=O)NN1CCCCC1 ZINC000147373428 BB For-Sale Anodyne CNR1 53 33 Cc1c(CN2CCSCC2)cccc1NC(=O)C1CCN(CC(F)(F)F)CC1 ZINC000147373465 HH On-Demand Anodyne CACNA1G 33 40 CCCCCCCCNC(=O)[C@@H]1CCC[C@@H](CCN)C1 ZINC000147373504 CH For-Sale Mild EPHX2 28 40 CCCCCCCCNC(=O)[C@@H]1CCC[C@@H](CCN)C1 ZINC000147373504 CH For-Sale Mild TPP2 22 40 CNc1ncc(Cl)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147373517 DH For-Sale Anodyne PDS 43 37 Cc1cc(CNCC(F)F)ccc1F ZINC000147373529 BE On-Demand Anodyne LEF 57 43 C[C@@H](CNC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147373573 BD For-Sale Anodyne GPR88 0 46 O=C(CCCc1ccc2c(c1)-c1ccccc1C2)N1C[C@H]2CC[C@H]1C2 ZINC000147373585 EJ On-Demand Anodyne PREP 47 38 CC[C@H](CNS(=O)(=O)c1cc(C#N)ccc1C)CC(=O)O ZINC000147373611 DD On-Demand Mild TBXA2R 0 44 CCCCCCCCNC(=O)[C@H]1CCC[C@@H](CCN)C1 ZINC000147373628 CH For-Sale Mild EPHX2 28 40 CCCCCCCCNC(=O)[C@H]1CCC[C@@H](CCN)C1 ZINC000147373628 CH For-Sale Mild TPP2 22 40 Cc1cc(OCc2nc(C)c(C)s2)ccc1S(N)(=O)=O ZINC000147373713 DE For-Sale Anodyne Q50565_METTH 0 41 C[C@H](CNC(=O)[C@H]1C[C@@H]1c1ccccc1)C(=O)O ZINC000147373747 BD For-Sale Anodyne GPR88 0 46 CCCCCCCCNC(=O)[C@@H]1CCC[C@H](CN)C1 ZINC000147373764 CG For-Sale Mild TPP2 32 42 CC[C@@H](CNS(=O)(=O)c1cc(C#N)ccc1C)CC(=O)O ZINC000147373767 DD On-Demand Mild TBXA2R 0 44 CCc1ncc(C(=O)Nc2nc(-c3ccc(CCCNC(C)=O)cc3)cs2)s1 ZINC000147373783 HI On-Demand Anodyne ROCK1 21 43 O=C(CCOc1ccccc1)N1CCC[C@H](CCBr)C1 ZINC000147373807 EG For-Sale Reactive HRH3 17 48 O=C(CCOc1ccccc1)N1CCC[C@H](CCBr)C1 ZINC000147373807 EG For-Sale Reactive COLA 75 37 O=C(CCOc1ccccc1)N1CCC[C@H](CCBr)C1 ZINC000147373807 EG For-Sale Reactive CPT1A 70 37 O=C(CCOc1ccccc1)N1CCC[C@H](CCBr)C1 ZINC000147373807 EG For-Sale Reactive CPT2 44 37 O=C(CCOc1ccccc1)N1CCC[C@H](CCBr)C1 ZINC000147373807 EG For-Sale Reactive PREP 51 36 Cc1c(CN2CCSCC2)cccc1NC(=O)c1c[nH]cc1-c1ccccc1 ZINC000147373841 GJ On-Demand Anodyne MRGPRX1 42 43 Cc1c([C@@H](C)NCCCCC(C)C)sc2ccccc12 ZINC000147373858 CK For-Sale Anodyne TRPM8 33 41 CC(C)(C)NCc1cnccc1Oc1ccc(Cl)c(F)c1 ZINC000147373868 DJ For-Sale Anodyne SLC6A4 15 47 CCCCCCCCNC(=O)[C@H]1CCC[C@H](CN)C1 ZINC000147373898 CG For-Sale Mild TPP2 32 42 O=C(CCOc1ccccc1)N1CCC[C@@H](CCBr)C1 ZINC000147373935 EG For-Sale Reactive HRH3 17 48 O=C(CCOc1ccccc1)N1CCC[C@@H](CCBr)C1 ZINC000147373935 EG For-Sale Reactive COLA 75 37 O=C(CCOc1ccccc1)N1CCC[C@@H](CCBr)C1 ZINC000147373935 EG For-Sale Reactive CPT1A 70 37 O=C(CCOc1ccccc1)N1CCC[C@@H](CCBr)C1 ZINC000147373935 EG For-Sale Reactive CPT2 44 37 O=C(CCOc1ccccc1)N1CCC[C@@H](CCBr)C1 ZINC000147373935 EG For-Sale Reactive PREP 51 36 Cc1c([C@H](C)NCCCCC(C)C)sc2ccccc12 ZINC000147373968 CK For-Sale Anodyne TRPM8 33 41 Cc1ccc(C(=O)NC[C@@H](C)C(=O)O)cc1Br ZINC000147373987 DE On-Demand Anodyne F3 62 34 Cc1ccc(C(=O)NC[C@@H](C)C(=O)O)cc1Br ZINC000147373987 DE On-Demand Anodyne ITGAV 65 43 CN(C)C(=O)CN(C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147374003 DD For-Sale Anodyne PSBA 0 41 CCNc1ncc(C)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147374015 CI For-Sale Anodyne PDS 40 35 Fc1cc(Oc2ccncc2CNC2CC2)ccc1Cl ZINC000147374068 CH For-Sale Anodyne SLC6A4 15 49 CCCCCCCCNC(=O)[C@@H]1CCC[C@@H](CN)C1 ZINC000147374077 CG For-Sale Mild TPP2 32 42 Cc1ccc(C(=O)NC[C@H](C)C(=O)O)cc1Br ZINC000147374095 DE On-Demand Anodyne F3 62 34 Cc1ccc(C(=O)NC[C@H](C)C(=O)O)cc1Br ZINC000147374095 DE On-Demand Anodyne ITGAV 65 43 CC(C)(C)OC(=O)N1CC[C@H](Nc2cccc(Br)c2)C1 ZINC000147374209 EH On-Demand Anodyne ITGAL 42 34 CC(C)(C)OC(=O)N1CC[C@H](Nc2cccc(Br)c2)C1 ZINC000147374209 EH On-Demand Anodyne PTPN2 45 31 CC(C)(C)OC(=O)N1CC[C@H](Nc2cccc(Br)c2)C1 ZINC000147374209 EH On-Demand Anodyne EPHX2 15 43 CC(C)(C)OC(=O)N1CC[C@H](Nc2cccc(Br)c2)C1 ZINC000147374209 EH On-Demand Anodyne CCR8 15 41 CC(C)(C)OC(=O)N1CC[C@H](Nc2cccc(Br)c2)C1 ZINC000147374209 EH On-Demand Anodyne GPR119 45 47 CC(C)(C)OC(=O)N1CC[C@H](Nc2cccc(Br)c2)C1 ZINC000147374209 EH On-Demand Anodyne SFRP1 72 42 CC(C)(C)OC(=O)N1CC[C@H](Nc2cccc(Br)c2)C1 ZINC000147374209 EH On-Demand Anodyne WNT3 58 38 Cc1cccnc1NC(=O)NCC(=O)Nc1ccc(F)cc1 ZINC000147374216 DE On-Demand Anodyne PPIA 40 40 CCCCCCCCNC(=O)[C@H]1CCC[C@@H](CN)C1 ZINC000147374256 CG For-Sale Mild TPP2 32 42 CC(C)NCc1cnccc1Oc1ccc(Cl)c(F)c1 ZINC000147374289 CI For-Sale Anodyne SLC6A4 16 49 CC(C)(C)OC(=O)N1CC[C@@H](Nc2cccc(Br)c2)C1 ZINC000147374342 EH On-Demand Anodyne ITGAL 42 34 CC(C)(C)OC(=O)N1CC[C@@H](Nc2cccc(Br)c2)C1 ZINC000147374342 EH On-Demand Anodyne PTPN2 45 31 CC(C)(C)OC(=O)N1CC[C@@H](Nc2cccc(Br)c2)C1 ZINC000147374342 EH On-Demand Anodyne EPHX2 15 43 CC(C)(C)OC(=O)N1CC[C@@H](Nc2cccc(Br)c2)C1 ZINC000147374342 EH On-Demand Anodyne CCR8 15 41 CC(C)(C)OC(=O)N1CC[C@@H](Nc2cccc(Br)c2)C1 ZINC000147374342 EH On-Demand Anodyne GPR119 45 47 CC(C)(C)OC(=O)N1CC[C@@H](Nc2cccc(Br)c2)C1 ZINC000147374342 EH On-Demand Anodyne SFRP1 72 42 CC(C)(C)OC(=O)N1CC[C@@H](Nc2cccc(Br)c2)C1 ZINC000147374342 EH On-Demand Anodyne WNT3 58 38 COC(=O)COc1cccc(NC(=O)NCc2ccc(-n3ccnc3C)c(F)c2)c1 ZINC000147374376 HG On-Demand Anodyne ROCK2 25 42 O=C(C(=O)N1CCC(C(=O)Nc2nccs2)CC1)c1ccc2c(c1)CCC2 ZINC000147374377 GF On-Demand Anodyne MAP1 47 44 CCNC(=O)CN1CCN(C(=O)c2cccc(CN3CCCC3)c2)CC1 ZINC000147374411 FD On-Demand Anodyne HRH2 31 41 CCNC(=O)CN1CCN(C(=O)c2cccc(CN3CCCC3)c2)CC1 ZINC000147374411 FD On-Demand Anodyne AVPR1B 15 40 CCNC(=O)CN1CCN(C(=O)c2cccc(CN3CCCC3)c2)CC1 ZINC000147374411 FD On-Demand Anodyne CHRM3 15 42 CCNC(=O)CN1CCN(C(=O)c2cccc(CN3CCCC3)c2)CC1 ZINC000147374411 FD On-Demand Anodyne TRY2_BOVIN 51 35 CCNC(=O)CN1CCN(C(=O)c2cccc(CN3CCCC3)c2)CC1 ZINC000147374411 FD On-Demand Anodyne FAAH 17 50 CCNC(=O)CN1CCN(C(=O)c2cccc(CN3CCCC3)c2)CC1 ZINC000147374411 FD On-Demand Anodyne PARP1 20 46 CCNC(=O)CN1CCN(C(=O)c2cccc(CN3CCCC3)c2)CC1 ZINC000147374411 FD On-Demand Anodyne NPFFR1 43 33 CCCCCCCCNC(=O)CC1CCC(CN)CC1 ZINC000147374435 CH For-Sale Mild EPHX2 42 45 CCCCCCCCNC(=O)CC1CCC(CN)CC1 ZINC000147374435 CH For-Sale Mild ASAH1 72 39 CCCCCCCCNC(=O)CC1CCC(CN)CC1 ZINC000147374435 CH For-Sale Mild LASR 45 32 CCCCCCCCNC(=O)CC1CCC(CN)CC1 ZINC000147374435 CH For-Sale Mild NOD1 45 38 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne PLG 21 41 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne PRSS1 17 40 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne ACE 46 45 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne OPRM1 53 38 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne OPRD1 52 38 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne F10 20 50 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne MME 118 44 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne ANPEP 65 36 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne TACR1 17 44 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CTSD 21 41 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne MC4R 50 42 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CTRA_BOVIN 19 47 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne FCER2 94 43 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CTSB 89 50 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne PAPA1_CARPA 80 53 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CYSP_TRYCR 67 41 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CTSK 34 48 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CTSL 86 53 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CPA1 15 40 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CACNA1B 64 38 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne NPFFR2 54 45 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne TIMP3 88 46 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CTRB1 40 38 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne TACR3 22 41 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne MC3R 57 42 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CAPNS1 66 38 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne MMP2 23 54 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne MMP3 36 40 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne MMP8 26 43 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne GRIA1 56 49 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne ECE1 19 41 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne HLA-DRB1 86 41 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne REN 56 40 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne PCSK5 55 38 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne FURIN 81 46 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne PTPRA 48 34 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne PTPN1 16 41 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CTSS 48 53 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CAPN1 102 52 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne MMP9 31 46 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CAPN2 132 48 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne ACE2 84 44 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne MC1R 92 42 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne PLAU 34 40 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne BACE1 21 40 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CTSV 54 47 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne TPSAB1 23 40 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne PROC 54 47 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne MMP1 48 51 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne FPR1 79 40 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne CTRB_BOVIN 62 39 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne NPR 68 36 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne AMP1_PLAFQ 49 40 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne PSMB5 64 51 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne BLA1_STEMA 78 40 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne KISS1R 81 43 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne POLG_WNV 64 35 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne STAT3 38 43 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne QRFPR 46 38 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne PSMB8 71 38 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne NPFFR1 73 45 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne TMPRSS11D 52 43 CCOc1ccc(C[C@@H](NC(=O)c2ccccc2)C(=O)N[C@@H](Cc2ccccc2)C(=O)NCc2ccc(CN)cc2)cc1 ZINC000147374437 KH For-Sale Anodyne PDS 78 41 CCNc1cncc(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147374510 CH For-Sale Anodyne PDS 42 34 COc1cc(S(C)(=O)=O)ccc1CN ZINC000147374517 BC For-Sale Anodyne PTGS2 25 43 COCc1nc(C(=O)NCc2cn(-c3ccccc3)nc2-c2ccccc2)cs1 ZINC000147374518 HI On-Demand Anodyne CDK2 15 41 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne ESR1 81 38 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne ACHE 19 44 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne KCNH2 16 42 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne ESR2 57 40 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne LTA4H 60 48 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne HRH3 80 54 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne SIGMAR1 16 41 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne YES1 18 41 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne TNK2 18 41 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne PSMB2 59 47 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne PSMB1 53 50 Cc1cc(OCCN2CCCC2)ccc1S(N)(=O)=O ZINC000147374576 CD For-Sale Anodyne TBK1 15 41 CCCCCCCCn1c(SCC(=O)O)n[nH]c1=O ZINC000147374610 CE For-Sale Mild CSNK2A2 15 40 CCCCCCCCn1c(SCC(=O)O)n[nH]c1=O ZINC000147374610 CE For-Sale Mild ASAH1 42 29 CC(C)/C=C/c1sc(-c2nccs2)nc1C(=O)NCCCCC(=O)NO ZINC000147374848 GG Annotated Mild HDA106 0 40 CC[C@H](c1ccc(C(=O)NCc2nn[nH]n2)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147374908 KK Annotated Anodyne GCGR 29 85 CC[C@H](c1ccc(C(=O)NCc2nn[nH]n2)cc1)N1C(=O)C(c2cc(Cl)cc(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147374908 KK Annotated Anodyne GLP1R 17 72 CCN(CC)S(=O)(=O)c1ccc(CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147374913 HF On-Demand Bother MMP2 16 46 CCN(CC)S(=O)(=O)c1ccc(CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147374913 HF On-Demand Bother MMP8 35 46 CCN(CC)S(=O)(=O)c1ccc(CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147374913 HF On-Demand Bother MMP9 18 46 CCN(CC)S(=O)(=O)c1ccc(CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147374913 HF On-Demand Bother MMP1 27 46 CCN(CC)S(=O)(=O)c1ccc(CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147374913 HF On-Demand Bother NAMPT 41 40 CCOC(=O)c1ccc(-c2n[nH]c3ncccc23)[nH]1 ZINC000147374915 CE For-Sale Anodyne PRKCQ 45 34 CNc1nc(OC)nc(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147374928 DF For-Sale Anodyne PDS 41 34 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne ALOX5 19 42 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne ACE 39 50 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne PPARG 44 51 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne PPARA 46 51 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne FOLH1 15 40 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne MME 88 42 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne ANPEP 86 38 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne FCER2 40 31 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne PAPA1_CARPA 47 33 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne CPA1 86 43 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne SLC15A1 0 43 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne CAPNS1 50 36 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne CAPN1 52 41 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne CAPN2 48 37 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne ACE2 67 41 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne LAP3 45 39 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne CPA3 0 43 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne FPR1 58 40 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne POL 0 43 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne NPR 67 36 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne AMP1_PLAFQ 52 40 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne SLC15A2 0 41 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne SLC22A20 0 42 CC(C)CO[C@H](Cc1ccccc1)C(=O)O ZINC000147374939 BE In-Stock Anodyne BLAIMP-1 0 48 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CA2 144 73 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne PTGS2 20 40 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CA6 30 40 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CA1 123 63 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CA7 65 52 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CA13 24 40 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CA5B 72 52 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CA4 126 66 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CA5A 78 52 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CA14 49 42 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CA12 109 73 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CA9 119 68 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CAH_METTE 27 40 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne CYNT 48 42 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne NCE103 68 53 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne MTCA1 62 73 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne P96878_MYCTU 80 73 NS(=O)(=O)c1ccc(NC(=O)NCC(=O)Nc2ccc(F)cc2)cc1 ZINC000147374956 FD On-Demand Anodyne NAMPT 34 40 CCCCCCCCNC(=N)C1CCCCC1 ZINC000147374978 BI For-Sale Mild GNAI1 0 50 CCCCCCCCNC(=N)C1CCCCC1 ZINC000147374978 BI For-Sale Mild GNAI3 0 50 CCCCCCCCNC(=N)C1CCCCC1 ZINC000147374978 BI For-Sale Mild GNAO1 0 50 CCCCCCCCNC(=N)C1CCCCC1 ZINC000147374978 BI For-Sale Mild ASAH1 60 33 CN(C)C(=O)NCCn1c(CCCl)nc2cc(Cl)ccc21 ZINC000147375069 EF For-Sale Reactive HDAC1 0 41 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2nccs2)CC1 ZINC000147375125 FD On-Demand Anodyne P2RY12 62 33 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2nccs2)CC1 ZINC000147375125 FD On-Demand Anodyne MAP1 91 41 CCNC(=O)CN1CCN(C(=O)c2[nH]c3ccc(F)cc3c2Cl)CC1 ZINC000147375130 FD On-Demand Anodyne MPO 21 42 CCCCCCCCNC(=N)c1ccccc1 ZINC000147375137 BH For-Sale Mild ASAH1 94 43 CCNc1cc(Oc2cccc(C(F)(F)F)c2)ncn1 ZINC000147375160 CH For-Sale Anodyne PDS 42 37 Cc1c(CN2CCSCC2)cccc1NC(=O)c1c(Cl)c2ccccc2n1C ZINC000147375184 HJ On-Demand Anodyne MRGPRX1 42 37 CN(Cc1cccs1)C(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147375234 FH For-Sale Anodyne HCAR3 16 42 COC(=O)c1cc2c(CN3CC[C@@H](O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147375280 GF For-Sale Anodyne CCR3 43 37 COC(=O)c1cc2c(CN3CC[C@@H](O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147375280 GF For-Sale Anodyne MLNR 66 37 COC(=O)c1cc2c(CN3CC[C@@H](O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147375280 GF For-Sale Anodyne MCHR1 25 40 CCCCc1ccc(Br)c([N+](=O)[O-])c1 ZINC000147375288 CH For-Sale Anodyne INHA 37 45 CN(Cc1cccs1)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147375432 DH On-Demand Anodyne HCAR3 15 40 COC(=O)c1cc2c(CN3CC[C@H](O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147375445 GF For-Sale Anodyne CCR3 43 37 COC(=O)c1cc2c(CN3CC[C@H](O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147375445 GF For-Sale Anodyne MLNR 66 37 COC(=O)c1cc2c(CN3CC[C@H](O)C3)cn(Cc3ccc(F)cc3)c2cn1 ZINC000147375445 GF For-Sale Anodyne MCHR1 25 40 CNS(=O)(=O)c1ccc(C(=O)Nc2cccc(CN3CCSCC3)c2C)o1 ZINC000147375474 HE On-Demand Anodyne LPL 42 34 CNS(=O)(=O)c1ccc(C(=O)Nc2cccc(CN3CCSCC3)c2C)o1 ZINC000147375474 HE On-Demand Anodyne MAPK8 21 40 CC[C@H](CNS(=O)(=O)c1ccc(C)cc1)CC(=O)O ZINC000147375482 CD On-Demand Anodyne TBXAS1 30 40 O=C(CNC(=O)N1CCOCC1)Nc1ccc(F)cc1 ZINC000147375558 CC On-Demand Anodyne MTOR 27 44 O=C(CNC(=O)N1CCOCC1)Nc1ccc(F)cc1 ZINC000147375558 CC On-Demand Anodyne EPHX2 34 57 O=C(CNC(=O)N1CCOCC1)Nc1ccc(F)cc1 ZINC000147375558 CC On-Demand Anodyne AKR1C3 25 46 CCCn1c(=O)n(-c2ccc3c(c2)OCO3)c2ncc(NC(=O)OCC)cc21 ZINC000147375590 GF For-Sale Anodyne ADORA2B 21 41 CC[C@@H](CNS(=O)(=O)c1ccc(C)cc1)CC(=O)O ZINC000147375618 CD On-Demand Anodyne TBXAS1 30 40 CNc1ncc(Br)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147375652 EI For-Sale Anodyne P2RY1 15 43 CNc1ncc(Br)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147375652 EI For-Sale Anodyne PDS 41 33 CN(Cc1ccsc1)C(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147375661 FH For-Sale Anodyne HCAR3 24 42 CN(C)C(=O)NCCn1c(CCCl)nc2cc(Br)ccc21 ZINC000147375746 FF For-Sale Reactive HDAC10 25 41 CN(C)C(=O)NCCn1c(CCCl)nc2cc(Br)ccc21 ZINC000147375746 FF For-Sale Reactive HDAC1 15 42 CN(C)C(=O)NCCn1c(CCCl)nc2cc(Br)ccc21 ZINC000147375746 FF For-Sale Reactive HDAC2 16 41 CN(C)C(=O)NCCn1c(CCCl)nc2cc(Br)ccc21 ZINC000147375746 FF For-Sale Reactive HDAC3 15 41 CN(C)C(=O)NCCn1c(CCCl)nc2cc(Br)ccc21 ZINC000147375746 FF For-Sale Reactive HDAC4 28 41 CN(C)C(=O)NCCn1c(CCCl)nc2cc(Br)ccc21 ZINC000147375746 FF For-Sale Reactive HDAC5 38 41 CN(C)C(=O)NCCn1c(CCCl)nc2cc(Br)ccc21 ZINC000147375746 FF For-Sale Reactive HDAC9 32 41 CN(C)C(=O)NCCn1c(CCCl)nc2cc(Br)ccc21 ZINC000147375746 FF For-Sale Reactive HDAC11 29 41 CN(C)C(=O)NCCn1c(CCCl)nc2cc(Br)ccc21 ZINC000147375746 FF For-Sale Reactive HDAC7 36 41 CCNC(=O)CN1CCN(C(=O)C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)CC1 ZINC000147375764 HC On-Demand Anodyne MMP13 29 46 CCNC(=O)CN1CCN(C(=O)C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)CC1 ZINC000147375764 HC On-Demand Anodyne APP 37 40 CCNC(=O)CN1CCN(C(=O)C2(S(=O)(=O)c3ccc(Cl)cc3)CC2)CC1 ZINC000147375764 HC On-Demand Anodyne MMP14 30 40 O=C(Nc1ccc(Cl)cc1Br)c1cccc2c1OCCN2 ZINC000147375783 FI For-Sale Anodyne KCNMA1 23 42 O=C(Nc1ccc(Cl)cc1Br)c1cccc2c1OCCN2 ZINC000147375783 FI For-Sale Anodyne G2YM83_BOTF4 51 32 O=[N+]([O-])c1cnc(Nc2ccc3c(c2)OCO3)c([N+](=O)[O-])c1 ZINC000147375787 DE For-Sale Bother DYRK2 40 36 CCOc1ccc(S(=O)(=O)NC[C@@H](CC)CC(=O)O)cc1 ZINC000147375837 DD On-Demand Anodyne MMP13 30 40 CCOc1ccc(S(=O)(=O)NC[C@@H](CC)CC(=O)O)cc1 ZINC000147375837 DD On-Demand Anodyne MMP14 22 40 CCOc1ccc(S(=O)(=O)NC[C@@H](CC)CC(=O)O)cc1 ZINC000147375837 DD On-Demand Anodyne ADAMTS4 49 38 CN(Cc1ccsc1)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147375872 DH On-Demand Anodyne HCAR3 23 40 O=C(Nc1cc(Cl)ccc1Br)c1cccc2c1OCCN2 ZINC000147375951 FI For-Sale Anodyne KCNMA1 19 44 O=C(Nc1cc(Cl)ccc1Br)c1cccc2c1OCCN2 ZINC000147375951 FI For-Sale Anodyne G2YM83_BOTF4 51 32 O=C(NCCc1ccc(Br)s1)c1cccc(OC(F)F)c1 ZINC000147375976 GI On-Demand Anodyne DRD4 44 34 CCOC[C@H](C)NC(=O)Nc1ccc2c(c1)oc1ccccc12 ZINC000147375977 DI On-Demand Anodyne ECE1 19 41 CCOC[C@H](C)NC(=O)Nc1ccc2c(c1)oc1ccccc12 ZINC000147375977 DI On-Demand Anodyne MMP12 34 40 CCOc1ccc(S(=O)(=O)NC[C@H](CC)CC(=O)O)cc1 ZINC000147376011 DD On-Demand Anodyne MMP13 30 40 CCOc1ccc(S(=O)(=O)NC[C@H](CC)CC(=O)O)cc1 ZINC000147376011 DD On-Demand Anodyne MMP14 22 40 CCOc1ccc(S(=O)(=O)NC[C@H](CC)CC(=O)O)cc1 ZINC000147376011 DD On-Demand Anodyne ADAMTS4 49 38 CCCNc1nccc(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147376107 CI For-Sale Anodyne PDS 40 35 CC[C@H](CNS(=O)(=O)c1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147376214 DD On-Demand Bother CACNA1D 51 33 CC[C@H](CNS(=O)(=O)c1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147376214 DD On-Demand Bother COLA 22 41 CCN(C[C@@H](C)C(=O)O)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147376225 CE For-Sale Anodyne GPR88 0 55 CCc1c(N)ncnc1Oc1cccc(C(F)(F)F)c1 ZINC000147376281 CG For-Sale Anodyne PDS 40 35 CC(C)CCCCNS(=O)(=O)Cc1cccc(C(=O)O)c1 ZINC000147376306 DF For-Sale Anodyne FOLH1 17 43 CC(C)CCCCNS(=O)(=O)Cc1cccc(C(=O)O)c1 ZINC000147376306 DF For-Sale Anodyne TRY2_BOVIN 69 31 CC(C)CCCCNS(=O)(=O)Cc1cccc(C(=O)O)c1 ZINC000147376306 DF For-Sale Anodyne MMP3 15 40 CC(C)CCCCNS(=O)(=O)Cc1cccc(C(=O)O)c1 ZINC000147376306 DF For-Sale Anodyne AKR1C3 48 44 CC(C)CCCCNS(=O)(=O)Cc1cccc(C(=O)O)c1 ZINC000147376306 DF For-Sale Anodyne TMPRSS11D 60 39 CC[C@@H](CNS(=O)(=O)c1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147376357 DD On-Demand Bother CACNA1D 51 33 CC[C@@H](CNS(=O)(=O)c1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147376357 DD On-Demand Bother COLA 22 41 CCN(C[C@H](C)C(=O)O)C(=O)[C@@H]1C[C@@H]1c1ccccc1 ZINC000147376358 CE For-Sale Anodyne GPR88 0 55 CN(C)C(=O)NCCn1c(CCCl)nc2cc(I)ccc21 ZINC000147376390 HF For-Sale Reactive HDAC1 0 40 CNC(=O)CCCOc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147376419 CC For-Sale Anodyne CA2 24 40 CNC(=O)CCCOc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147376419 CC For-Sale Anodyne P2RY12 0 46 CNC(=O)CCCOc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147376419 CC For-Sale Anodyne CA1 21 40 COc1ccc2cc(CNC(=O)NCC(=O)Nc3ccc(F)cc3)ccc2c1 ZINC000147376438 GG On-Demand Anodyne MTNR1A 49 40 COc1ccc2cc(CNC(=O)NCC(=O)Nc3ccc(F)cc3)ccc2c1 ZINC000147376438 GG On-Demand Anodyne MTNR1B 42 40 COc1ccc2cc(CNC(=O)NCC(=O)Nc3ccc(F)cc3)ccc2c1 ZINC000147376438 GG On-Demand Anodyne ROCK2 34 44 COc1ccc2cc(CNC(=O)NCC(=O)Nc3ccc(F)cc3)ccc2c1 ZINC000147376438 GG On-Demand Anodyne CA9 16 42 COc1ccc2cc(CNC(=O)NCC(=O)Nc3ccc(F)cc3)ccc2c1 ZINC000147376438 GG On-Demand Anodyne ENPP1 55 31 CC(C)CCCCNCc1cc([N+](=O)[O-])c(F)cc1F ZINC000147376465 CH For-Sale Bother LEF 50 35 CNc1ncnc(Oc2cccc(C(F)(F)F)c2)c1C ZINC000147376478 CH For-Sale Anodyne P2RY1 15 44 CNc1ncnc(Oc2cccc(C(F)(F)F)c2)c1C ZINC000147376478 CH For-Sale Anodyne PDS 42 33 C[C@H](NC(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147376491 CF On-Demand Anodyne CACNA1I 46 34 CCN(C[C@@H](C)C(=O)O)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147376550 CE For-Sale Anodyne GPR88 0 55 Cc1cc(C(=O)NCc2ccc(S(=O)(=O)N3CCCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147376568 HG On-Demand Bother EPHX2 30 43 Cc1cc(C(=O)NCc2ccc(S(=O)(=O)N3CCCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147376568 HG On-Demand Bother TGM2 39 41 Cc1cc(C(=O)NCc2ccc(S(=O)(=O)N3CCCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147376568 HG On-Demand Bother NAMPT 95 56 CC[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147376580 CD On-Demand Anodyne ITGAV 43 31 CC[C@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147376580 CD On-Demand Anodyne Q9JN24_ECOLX 0 44 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000147376602 HI On-Demand Anodyne TACR3 16 44 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000147376602 HI On-Demand Anodyne MCHR1 16 45 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cc(-c2ccc(F)cc2)n[nH]1 ZINC000147376602 HI On-Demand Anodyne MRGPRX1 46 44 Cc1cc(OCCC(=O)N(C)C)ccc1S(N)(=O)=O ZINC000147376640 CC For-Sale Anodyne THRA 0 40 C[C@@H](NC(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147376725 CF On-Demand Anodyne CACNA1I 46 34 CCN(C[C@H](C)C(=O)O)C(=O)[C@H]1C[C@@H]1c1ccccc1 ZINC000147376734 CE For-Sale Anodyne GPR88 0 55 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(F)c(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147376751 KK Annotated Anodyne GLP1R 23 57 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccc(F)c(Cl)c2)=NC12CCC(C(C)(C)C)CC2 ZINC000147376751 KK Annotated Anodyne GIPR 76 43 O=C(O)C1(n2nnnc2-c2ccc(Cl)cc2Cl)CCC1 ZINC000147376764 DF For-Sale Anodyne HSD11B1 22 43 O=C(O)C1(n2nnnc2-c2ccc(Cl)cc2Cl)CCC1 ZINC000147376764 DF For-Sale Anodyne ALPL 41 32 O=C(O)C1(n2nnnc2-c2ccc(Cl)cc2Cl)CCC1 ZINC000147376764 DF For-Sale Anodyne DPP8 63 34 O=C(O)C1(n2nnnc2-c2ccc(Cl)cc2Cl)CCC1 ZINC000147376764 DF For-Sale Anodyne DPP9 61 34 CNc1nc(C)cc(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147376769 CH For-Sale Anodyne PDS 41 32 CC[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147376791 CD On-Demand Anodyne ITGAV 43 31 CC[C@@H](CNS(=O)(=O)c1ccccc1)CC(=O)O ZINC000147376791 CD On-Demand Anodyne Q9JN24_ECOLX 0 44 Cc1c(CN2CCSCC2)cccc1NC(=O)C1CCN(S(N)(=O)=O)CC1 ZINC000147376826 HD On-Demand Anodyne EPHX2 34 42 O=C(CNC(=O)NCc1ccc(OC(F)(F)F)cc1)Nc1ccc(F)cc1 ZINC000147376867 GG On-Demand Anodyne P2RY1 61 39 O=C(CNC(=O)NCc1ccc(OC(F)(F)F)cc1)Nc1ccc(F)cc1 ZINC000147376867 GG On-Demand Anodyne EPHX2 57 47 CC[C@@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147376897 CD On-Demand Anodyne CHRM2 28 41 CC[C@@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147376897 CD On-Demand Anodyne MMP13 63 49 CC[C@@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147376897 CD On-Demand Anodyne ADAM17 35 45 CC[C@@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147376897 CD On-Demand Anodyne MMP8 39 49 CC[C@@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147376897 CD On-Demand Anodyne MMP9 43 50 CC[C@@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147376897 CD On-Demand Anodyne MMP7 74 49 CC[C@@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147376897 CD On-Demand Anodyne MMP1 72 47 CC[C@@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147376897 CD On-Demand Anodyne AKR1C3 0 40 CC[C@H](CNS(=O)(=O)c1ccc(Cl)c(Cl)c1)CC(=O)O ZINC000147377003 EF On-Demand Anodyne TBXA2R 41 33 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(Nc2ncccn2)c1 ZINC000147377017 HI On-Demand Anodyne BTK 48 35 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(Nc2ncccn2)c1 ZINC000147377017 HI On-Demand Anodyne MRGPRX1 45 40 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(Nc2ncccn2)c1 ZINC000147377017 HI On-Demand Anodyne KCNK3 46 34 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H](C(=O)Nc3ccccn3)C2)cc1 ZINC000147377021 GD On-Demand Anodyne CPT1A 118 46 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H](C(=O)Nc3ccccn3)C2)cc1 ZINC000147377021 GD On-Demand Anodyne CPT2 40 33 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H](C(=O)Nc3ccccn3)C2)cc1 ZINC000147377021 GD On-Demand Anodyne MAP3K12 28 40 CC[C@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147377097 CD On-Demand Anodyne CHRM2 28 41 CC[C@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147377097 CD On-Demand Anodyne MMP13 63 49 CC[C@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147377097 CD On-Demand Anodyne ADAM17 35 45 CC[C@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147377097 CD On-Demand Anodyne MMP8 39 49 CC[C@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147377097 CD On-Demand Anodyne MMP9 43 50 CC[C@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147377097 CD On-Demand Anodyne MMP7 74 49 CC[C@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147377097 CD On-Demand Anodyne MMP1 72 47 CC[C@H]1CN(S(=O)(=O)c2ccc(OC)cc2)CC[C@@H]1N ZINC000147377097 CD On-Demand Anodyne AKR1C3 0 40 CC(C)S(=O)(=O)NC(=O)Cc1csc(-c2ccc(Cl)cc2Cl)n1 ZINC000147377121 GH On-Demand Anodyne ALPL 43 39 CC(C)S(=O)(=O)NC(=O)Cc1csc(-c2ccc(Cl)cc2Cl)n1 ZINC000147377121 GH On-Demand Anodyne DPP8 62 33 CC(C)S(=O)(=O)NC(=O)Cc1csc(-c2ccc(Cl)cc2Cl)n1 ZINC000147377121 GH On-Demand Anodyne DPP9 62 33 CCCCCCCCN1CCC[C@H](NC2CC2)C1=O ZINC000147377143 CG For-Sale Mild LASR 46 33 CCN(CC)CCCOC(=O)c1ccc2[nH]c3ccc(C(=O)OCCCN(CC)CC)cc3c2c1 ZINC000147377149 JK Annotated Anodyne AMY2 42 39 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(-n2ccnc2)nc1 ZINC000147377196 GG On-Demand Anodyne MRGPRX1 44 39 CNc1ncc(F)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147377214 CG For-Sale Anodyne PDS 42 33 CC[C@@H](CNS(=O)(=O)c1ccc(Cl)c(Cl)c1)CC(=O)O ZINC000147377235 EF On-Demand Anodyne TBXA2R 41 33 NC(=O)c1ccc(OCC(=O)N2CCC[C@H](C(=O)Nc3ccccn3)C2)cc1 ZINC000147377242 GD On-Demand Anodyne CPT1A 118 46 NC(=O)c1ccc(OCC(=O)N2CCC[C@H](C(=O)Nc3ccccn3)C2)cc1 ZINC000147377242 GD On-Demand Anodyne CPT2 40 33 NC(=O)c1ccc(OCC(=O)N2CCC[C@H](C(=O)Nc3ccccn3)C2)cc1 ZINC000147377242 GD On-Demand Anodyne MAP3K12 28 40 CCCCCCCCN1CCC[C@@H](NC2CC2)C1=O ZINC000147377349 CG For-Sale Mild LASR 46 33 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(C(N)=O)c1 ZINC000147377425 FF On-Demand Anodyne SLC9A1 22 40 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(C(N)=O)c1 ZINC000147377425 FF On-Demand Anodyne KCNK3 44 35 Cc1cc(C)n([C@@H](C)C(=O)N2CCC[C@H](C(=O)Nc3ccccn3)C2)n1 ZINC000147377441 FE On-Demand Anodyne MAP3K12 29 41 O=[N+]([O-])c1cc(SSc2ccc(F)c([N+](=O)[O-])c2)ccc1F ZINC000147377442 EJ For-Sale Reactive PDE7A 19 41 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccccc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147377470 KK Annotated Anodyne GCGR 47 77 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccccc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147377470 KK Annotated Anodyne GLP1R 22 55 C[C@H](c1ccc(C(=O)NCCC(=O)O)cc1)N1C(=O)C(c2ccccc2)=NC12CCC(C(C)(C)C)CC2 ZINC000147377470 KK Annotated Anodyne GIPR 67 39 CC(C)CCCCNS(=O)(=O)c1ccc(O)c(C(=O)O)c1 ZINC000147377478 DE For-Sale Anodyne CASP3 31 64 CC(C)CCCCNS(=O)(=O)c1ccc(O)c(C(=O)O)c1 ZINC000147377478 DE For-Sale Anodyne MGRA 0 40 CCCCCCCCN1CCC[C@H](NCC)C1=O ZINC000147377581 CF For-Sale Mild LASR 47 33 Cc1cc(C)n([C@H](C)C(=O)N2CCC[C@H](C(=O)Nc3ccccn3)C2)n1 ZINC000147377664 FE On-Demand Anodyne MAP3K12 29 41 CC(C)CCCCNS(=O)(=O)c1ccc(Br)c(C(=O)O)c1 ZINC000147377713 GG For-Sale Anodyne CASP3 24 48 CC(C)CCCCNS(=O)(=O)c1ccc(Br)c(C(=O)O)c1 ZINC000147377713 GG For-Sale Anodyne LEF 16 42 Cc1cc(OCCc2cccnc2)ccc1S(N)(=O)=O ZINC000147377770 CD For-Sale Anodyne CA7 18 44 Cc1cc(OCCc2cccnc2)ccc1S(N)(=O)=O ZINC000147377770 CD For-Sale Anodyne CA12 15 44 Cc1cc(OCCc2cccnc2)ccc1S(N)(=O)=O ZINC000147377770 CD For-Sale Anodyne CA9 15 44 CCCCCCCCN1CCC[C@@H](NCC)C1=O ZINC000147377827 CF For-Sale Mild LASR 47 33 CCNc1nc(Cl)nc(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147377846 DH For-Sale Anodyne PETD 0 42 CCNc1nc(Cl)nc(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147377846 DH For-Sale Anodyne PDS 43 36 CCNc1nc(Cl)nc(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147377846 DH For-Sale Anodyne PPX1 0 42 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(OCC(N)=O)c1 ZINC000147377872 GF On-Demand Anodyne DRD4 42 33 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(OCC(N)=O)c1 ZINC000147377872 GF On-Demand Anodyne SLC9A1 60 36 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(OCC(N)=O)c1 ZINC000147377872 GF On-Demand Anodyne MRGPRX1 42 38 CC[C@H](CNS(=O)(=O)c1ccc(F)c(C#N)c1)CC(=O)O ZINC000147377878 DD On-Demand Mild LEF 54 38 Cc1cc(C)n([C@@H](C)C(=O)N2CCC[C@@H](C(=O)Nc3ccccn3)C2)n1 ZINC000147377903 FE On-Demand Anodyne MAP3K12 29 41 CCc1ncc(C(=O)NCc2ccc(S(=O)(=O)N(CC)CC)cc2)s1 ZINC000147377963 GF On-Demand Anodyne NAMPT 79 45 CCCCCCCCN1CC[C@H](NC2CC2)C1=O ZINC000147377992 CF For-Sale Mild LASR 48 34 COc1ccc(C(F)(F)c2cc(NCCC(F)(F)F)c3ncc(-c4ccc(C(=O)NC5CC5)c(C)c4)n3n2)cc1 ZINC000147378026 KK Annotated Anodyne TTK 15 67 COc1ccc2c(c1)nc(CCl)n2CCNC(=O)N(C)C ZINC000147378054 DE For-Sale Reactive DRD4 42 32 COc1ccc2c(c1)nc(CCl)n2CCNC(=O)N(C)C ZINC000147378054 DE For-Sale Reactive MTNR1A 42 36 CC[C@@H](CNS(=O)(=O)c1ccc(F)c(C#N)c1)CC(=O)O ZINC000147378076 DD On-Demand Mild LEF 54 38 O=C(NS(=O)(=O)c1cccnc1)[C@@H](OCC(F)(F)F)c1ccccc1 ZINC000147378091 FE In-Stock Anodyne KCNA5 42 35 CCCCCCCCOc1ccc(CN)nc1 ZINC000147378132 BG For-Sale Mild THRA 41 38 CCCCCCCCOc1ccc(CN)nc1 ZINC000147378132 BG For-Sale Mild PLA2G4B 93 41 CCCCCCCCOc1ccc(CN)nc1 ZINC000147378132 BG For-Sale Mild CYP1A2 17 42 CCCCCCCCOc1ccc(CN)nc1 ZINC000147378132 BG For-Sale Mild CYP2C19 24 42 Cc1cc(C)n([C@H](C)C(=O)N2CCC[C@@H](C(=O)Nc3ccccn3)C2)n1 ZINC000147378137 FE On-Demand Anodyne MAP3K12 29 41 CCCCCCCCN1CC[C@@H](NC2CC2)C1=O ZINC000147378213 CF For-Sale Mild LASR 48 34 CCNc1ncc(F)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147378293 DH For-Sale Anodyne PDS 40 35 O=C(NS(=O)(=O)c1cccnc1)[C@H](OCC(F)(F)F)c1ccccc1 ZINC000147378295 FE In-Stock Anodyne KCNA5 42 35 O=C(C(=O)N1CCC[C@@H](C(=O)Nc2ccccn2)C1)c1ccc2c(c1)CCC2 ZINC000147378369 GF On-Demand Anodyne MAPK10 15 48 CCOC(=O)c1nnc2ccc([N+](=O)[O-])cc2c1Cl ZINC000147378384 CE In-Stock Bother CACNA1C 49 42 CCOC(=O)c1nnc2ccc([N+](=O)[O-])cc2c1Cl ZINC000147378384 CE In-Stock Bother ELANE 0 56 CCOC(=O)c1nnc2ccc([N+](=O)[O-])cc2c1Cl ZINC000147378384 CE In-Stock Bother CACNA1D 76 39 CCOC(=O)c1nnc2ccc([N+](=O)[O-])cc2c1Cl ZINC000147378384 CE In-Stock Bother CTRB1 34 51 CCOC(=O)c1nnc2ccc([N+](=O)[O-])cc2c1Cl ZINC000147378384 CE In-Stock Bother KCNMA1 23 47 CCOC(=O)c1nnc2ccc([N+](=O)[O-])cc2c1Cl ZINC000147378384 CE In-Stock Bother SLC5A2 0 43 CCOC(=O)c1nnc2ccc([N+](=O)[O-])cc2c1Cl ZINC000147378384 CE In-Stock Bother F2RL3 52 32 CCCCCCCCN1CCC[C@H](NCCC)C1=O ZINC000147378422 CG For-Sale Mild LASR 46 33 CC[C@H](NS(=O)(=O)c1cccc(C(F)(F)F)c1C)C(=O)O ZINC000147378489 EE For-Sale Anodyne ITGAV 65 44 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne F2 21 42 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne CELA1 69 53 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne ELANE 98 47 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne HLA-DRB3 60 36 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne CMA1 39 41 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne CTRA_BOVIN 25 44 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne CACNA1B 18 46 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne HLA-A 48 36 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne LGMN 93 38 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne CTRC 15 52 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne TPP2 43 46 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne XIAP 53 47 COC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C)C(C)C ZINC000147378501 ED For-Sale Anodyne BRCA1 64 35 CCc1c(NC)ncnc1Oc1cccc(C(F)(F)F)c1 ZINC000147378516 CH For-Sale Anodyne PDS 44 35 Cc1cc(OCc2ccc(C#N)cc2)ccc1S(N)(=O)=O ZINC000147378543 DE For-Sale Mild MAOB 48 52 O=C(N[C@@H](Cc1ccc(O)cc1)c1nc2ccccc2[nH]1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147378598 HI On-Demand Anodyne OPRM1 17 47 O=C(N[C@@H](Cc1ccc(O)cc1)c1nc2ccccc2[nH]1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147378598 HI On-Demand Anodyne F11 48 35 O=C(N[C@@H](Cc1ccc(O)cc1)c1nc2ccccc2[nH]1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147378598 HI On-Demand Anodyne PTPN1 45 54 O=C(C(=O)N1CCC[C@H](C(=O)Nc2ccccn2)C1)c1ccc2c(c1)CCC2 ZINC000147378627 GF On-Demand Anodyne MAPK10 15 48 Fc1cc(Oc2cncc(CNC3CC3)n2)ccc1Cl ZINC000147378637 CG For-Sale Anodyne GRIN2B 0 46 CCCCCCCCN1CCC[C@@H](NCCC)C1=O ZINC000147378640 CG For-Sale Mild LASR 46 33 COc1ccc(CCCC(=O)NS(=O)(=O)C(C)C)cc1 ZINC000147378673 CD On-Demand Anodyne BMP1 74 44 COc1ccc(CCCC(=O)NS(=O)(=O)C(C)C)cc1 ZINC000147378673 CD On-Demand Anodyne MMP13 36 47 COc1ccc(CCCC(=O)NS(=O)(=O)C(C)C)cc1 ZINC000147378673 CD On-Demand Anodyne MMP3 43 41 COc1ccc(CCCC(=O)NS(=O)(=O)C(C)C)cc1 ZINC000147378673 CD On-Demand Anodyne MMP8 27 47 COc1ccc(CCCC(=O)NS(=O)(=O)C(C)C)cc1 ZINC000147378673 CD On-Demand Anodyne MMP9 35 43 COc1ccc(CCCC(=O)NS(=O)(=O)C(C)C)cc1 ZINC000147378673 CD On-Demand Anodyne MMP12 31 47 COc1ccc(CCCC(=O)NS(=O)(=O)C(C)C)cc1 ZINC000147378673 CD On-Demand Anodyne IAP 0 40 COc1ccc(CCCC(=O)NS(=O)(=O)C(C)C)cc1 ZINC000147378673 CD On-Demand Anodyne MMP1 49 39 c1cn2cc(-c3ccc4cn[nH]c4c3)nc(Nc3ccc(N4CCCOCC4)cc3)c2n1 ZINC000147378682 II Annotated Anodyne SYK 51 93 c1cn2cc(-c3ccc4cn[nH]c4c3)nc(Nc3ccc(N4CCCOCC4)cc3)c2n1 ZINC000147378682 II Annotated Anodyne MAPKAPK5 62 46 c1cn2cc(-c3ccc4cn[nH]c4c3)nc(Nc3ccc(N4CCCOCC4)cc3)c2n1 ZINC000147378682 II Annotated Anodyne STAT6 61 37 CNc1nc(Cl)nc(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147378728 DG For-Sale Anodyne PDS 42 36 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccn(CC(N)=O)n1)C2 ZINC000147378752 EC On-Demand Anodyne ROCK2 34 46 COc1ccccc1Cc1nnnn1C1(C(=O)O)CCC1 ZINC000147378802 CD For-Sale Anodyne CCR8 28 40 CC[C@@H]1CN(S(=O)(=O)c2ccc(C)cc2C)CC[C@@H]1N ZINC000147378837 CE On-Demand Anodyne EPHX2 33 50 CCCCCCCCN1CC[C@H](NC(C)C)C1=O ZINC000147378855 CF For-Sale Mild LASR 49 36 C[C@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147378856 BD For-Sale Anodyne SLC15A1 0 40 C[C@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147378856 BD For-Sale Anodyne GPR88 0 54 OC[C@@H]1NC[C@H]2C[C@@H]21 ZINC000147378859 AB For-Sale Anodyne GLA 0 43 OC[C@@H]1NC[C@H]2C[C@@H]21 ZINC000147378859 AB For-Sale Anodyne GANAB 0 43 OC[C@@H]1NC[C@H]2C[C@@H]21 ZINC000147378859 AB For-Sale Anodyne GANC 0 43 OC[C@@H]1NC[C@H]2C[C@@H]21 ZINC000147378859 AB For-Sale Anodyne GAA 19 43 OC[C@@H]1NC[C@H]2C[C@@H]21 ZINC000147378859 AB For-Sale Anodyne AGLC 0 43 OC[C@@H]1NC[C@H]2C[C@@H]21 ZINC000147378859 AB For-Sale Anodyne MAL62 0 44 OC[C@@H]1NC[C@H]2C[C@@H]21 ZINC000147378859 AB For-Sale Anodyne Q43014_PRUAV 0 43 OC[C@@H]1NC[C@H]2C[C@@H]21 ZINC000147378859 AB For-Sale Anodyne AGL 0 44 OC[C@@H]1NC[C@H]2C[C@@H]21 ZINC000147378859 AB For-Sale Anodyne Q9GPQ4_TRYVI 0 44 OC[C@@H]1NC[C@H]2C[C@@H]21 ZINC000147378859 AB For-Sale Anodyne SGA1 0 44 COc1ccc(Nc2nc(-c3ccc4cc[nH]c4c3)cn3ccnc23)cc1OC ZINC000147378936 GJ For-Sale Anodyne EPHB4 27 41 COc1ccc(Nc2nc(-c3ccc4cc[nH]c4c3)cn3ccnc23)cc1OC ZINC000147378936 GJ For-Sale Anodyne ENPP1 51 32 CNc1cccc(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147378953 CH For-Sale Anodyne PDS 42 33 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccnc1N1CCCCC1)C2 ZINC000147379023 FG On-Demand Anodyne ROCK2 39 47 C[C@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147379047 BD For-Sale Anodyne SLC15A1 0 40 C[C@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147379047 BD For-Sale Anodyne GPR88 0 54 CC[C@H]1CN(S(=O)(=O)c2ccc(C)cc2C)CC[C@@H]1N ZINC000147379052 CE On-Demand Anodyne EPHX2 33 50 CCCCCCCCN1CC[C@@H](NC(C)C)C1=O ZINC000147379073 CF For-Sale Mild LASR 49 36 COc1ccccc1-n1c(=O)[nH]c2cccnc21 ZINC000147379218 BD For-Sale Anodyne HTR1A 25 46 COc1ccccc1-n1c(=O)[nH]c2cccnc21 ZINC000147379218 BD For-Sale Anodyne ADRA1A 16 46 COc1ccccc1-n1c(=O)[nH]c2cccnc21 ZINC000147379218 BD For-Sale Anodyne ADRA1B 17 46 COc1ccccc1-n1c(=O)[nH]c2cccnc21 ZINC000147379218 BD For-Sale Anodyne HTR7 22 43 O=C(NCCN1C(=O)c2ccccc2C1=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147379232 EE On-Demand Anodyne EPHX2 22 46 CCCCCCCCN1CCC[C@H](NC(C)C)C1=O ZINC000147379266 CG For-Sale Mild LASR 48 35 C[C@H](NC(=O)C1[C@@H]2CCCC[C@@H]12)C(=O)O ZINC000147379285 BD On-Demand Anodyne SLC15A2 0 40 CC(C)CC[C@H](O)[C@@H](C)[C@H]1CC[C@@H]([C@@H]2CC=C3C[C@@H](O)CC[C@]3(C)C2=O)[C@]1(C)CCO ZINC000147379294 IJ Annotated Anodyne RORC 0 53 C=C(NC(=O)OC(C)(C)C)C(=O)OC(C)C ZINC000147379351 BD In-Stock Anodyne CTSK 0 43 Nc1ccc([N+](=O)[O-])c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147379384 CG For-Sale Bother PPXII 0 42 CN(Cc1cscn1)C(=O)NCc1ccc(Oc2ccc(F)cc2)cc1 ZINC000147379395 FI On-Demand Anodyne BMP1 29 42 COc1cc(OCC(=O)N2CCC[C@H](C(=O)Nc3ccccc3)C2)ccc1[N+](=O)[O-] ZINC000147379399 HF On-Demand Bother CPT1A 51 40 COc1cc(OCC(=O)N2CCC[C@H](C(=O)Nc3ccccc3)C2)ccc1[N+](=O)[O-] ZINC000147379399 HF On-Demand Bother CPT2 43 37 COc1cc(OCC(=O)N2CCC[C@H](C(=O)Nc3ccccc3)C2)ccc1[N+](=O)[O-] ZINC000147379399 HF On-Demand Bother MMP7 21 44 COc1cc(OCC(=O)N2CCC[C@H](C(=O)Nc3ccccc3)C2)ccc1[N+](=O)[O-] ZINC000147379399 HF On-Demand Bother ALK 16 44 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)c(Cl)c3)cs2)s1 ZINC000147379414 GJ On-Demand Anodyne MPL 46 42 CCc1ncc(C(=O)Nc2nc(-c3ccc(OC)c(Cl)c3)cs2)s1 ZINC000147379414 GJ On-Demand Anodyne TRPA1 17 41 O=[N+]([O-])c1ccc(F)nc1Nc1ccc2c(c1)OCO2 ZINC000147379422 CF For-Sale Bother DYRK2 41 37 O=C(NCCN1C(=O)c2ccccc2C1=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147379439 EE On-Demand Anodyne EPHX2 22 46 O=C(Nc1cccc(Br)c1O)c1cccc2c1OCCN2 ZINC000147379456 EG For-Sale Anodyne G2YM83_BOTF4 52 32 CCCCCCCCN1CCC[C@@H](NC(C)C)C1=O ZINC000147379477 CG For-Sale Mild LASR 48 35 CCCC[C@H](NC(N)=O)C(=O)N(C)Cc1ccc(C#N)cc1 ZINC000147379565 DD On-Demand Mild CTRB_BOVIN 52 37 COc1cc(OCC(=O)N2CCC[C@@H](C(=O)Nc3ccccc3)C2)ccc1[N+](=O)[O-] ZINC000147379613 HF On-Demand Bother CPT1A 51 40 COc1cc(OCC(=O)N2CCC[C@@H](C(=O)Nc3ccccc3)C2)ccc1[N+](=O)[O-] ZINC000147379613 HF On-Demand Bother CPT2 43 37 COc1cc(OCC(=O)N2CCC[C@@H](C(=O)Nc3ccccc3)C2)ccc1[N+](=O)[O-] ZINC000147379613 HF On-Demand Bother MMP7 21 44 COc1cc(OCC(=O)N2CCC[C@@H](C(=O)Nc3ccccc3)C2)ccc1[N+](=O)[O-] ZINC000147379613 HF On-Demand Bother ALK 16 44 CNc1cc(Oc2cccc(C(F)(F)F)c2)nc(N)n1 ZINC000147379638 CF For-Sale Anodyne PDS 42 33 O=C(NCCN1C(=O)c2ccccc2C1=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147379662 EE On-Demand Anodyne EPHX2 22 46 Cn1cc(NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147379694 CE On-Demand Anodyne MAPK10 15 48 CC(C)(C)c1nc(NN)cc(SCc2ccccc2)n1 ZINC000147379703 CG For-Sale Anodyne PTR1 15 47 CCCCCCCCN1CCC[C@H](NC)C1=O ZINC000147379712 BF For-Sale Mild LASR 48 34 CCCC[C@@H](NC(N)=O)C(=O)N(C)Cc1ccc(C#N)cc1 ZINC000147379794 DD On-Demand Mild CTRB_BOVIN 52 37 CC(=O)N1CCC[C@H]1C(=O)Nc1cccc(CN2CCSCC2)c1C ZINC000147379797 FE On-Demand Anodyne LGMN 63 33 CC(=O)N1CCC[C@H]1C(=O)Nc1cccc(CN2CCSCC2)c1C ZINC000147379797 FE On-Demand Anodyne XIAP 39 42 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1F ZINC000147379800 EG For-Sale Reactive GRM3 16 47 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1F ZINC000147379800 EG For-Sale Reactive HRH3 26 41 COc1ccc(C(=O)N2CCC[C@H](CCBr)C2)cc1F ZINC000147379800 EG For-Sale Reactive ACKR3 69 37 CCNc1ncc(Br)c(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147379855 FI For-Sale Anodyne PDS 40 35 O=C(NCCN1C(=O)c2ccccc2C1=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147379877 EE On-Demand Anodyne EPHX2 22 46 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NC(C)C)cc1C)C2 ZINC000147379914 GG On-Demand Anodyne ROCK2 31 47 CCCCCCCCN1CCC[C@@H](NC)C1=O ZINC000147379916 BF For-Sale Mild LASR 48 34 CCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H](C(=O)Nc2ccccn2)C1 ZINC000147379948 ED On-Demand Anodyne P2RY12 134 34 CCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H](C(=O)Nc2ccccn2)C1 ZINC000147379948 ED On-Demand Anodyne TRY1_BOVIN 46 33 CCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H](C(=O)Nc2ccccn2)C1 ZINC000147379948 ED On-Demand Anodyne CTSK 20 40 CCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H](C(=O)Nc2ccccn2)C1 ZINC000147379948 ED On-Demand Anodyne DPP7 43 34 CC(C)CC[C@H](O)[C@@H](CO)[C@H]1CC[C@@H]([C@@H]2CC=C3C[C@@H](O)CC[C@]3(C)C2=O)[C@]1(C)CCO ZINC000147379956 JH Annotated Anodyne RORC 0 45 CC(=O)N1CCC[C@@H]1C(=O)Nc1cccc(CN2CCSCC2)c1C ZINC000147379975 FE On-Demand Anodyne LGMN 63 33 CC(=O)N1CCC[C@@H]1C(=O)Nc1cccc(CN2CCSCC2)c1C ZINC000147379975 FE On-Demand Anodyne XIAP 39 42 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1F ZINC000147380019 EG For-Sale Reactive GRM3 16 47 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1F ZINC000147380019 EG For-Sale Reactive HRH3 26 41 COc1ccc(C(=O)N2CCC[C@@H](CCBr)C2)cc1F ZINC000147380019 EG For-Sale Reactive ACKR3 69 37 Cc1ccc(NC(=O)c2cccc3c2OCCN3)cn1 ZINC000147380025 CE For-Sale Anodyne G2YM83_BOTF4 52 34 Cc1ccc(S(=O)(=O)NCCCCC(C)C)cc1C(=O)O ZINC000147380168 DF For-Sale Anodyne TBXAS1 34 40 Cc1ccc(S(=O)(=O)NCCCCC(C)C)cc1C(=O)O ZINC000147380168 DF For-Sale Anodyne CASP3 18 52 Cc1ccc(S(=O)(=O)NCCCCC(C)C)cc1C(=O)O ZINC000147380168 DF For-Sale Anodyne LEF 48 34 CC(C)=CC[C@H](O)[C@@H](C)[C@H]1CC[C@@H]([C@@H]2CC=C3C[C@@H](O)CC[C@]3(C)C2=O)[C@]1(C)CCO ZINC000147380194 IJ Annotated Anodyne RORC 0 40 Cc1cc(NC(=O)c2cccc3c2OCCN3)ccc1O ZINC000147380213 CF For-Sale Anodyne AVPR2 15 40 Cc1cc(NC(=O)c2cccc3c2OCCN3)ccc1O ZINC000147380213 CF For-Sale Anodyne KCNK3 66 38 Cc1cc(NC(=O)c2cccc3c2OCCN3)ccc1O ZINC000147380213 CF For-Sale Anodyne KCNK9 66 36 O=C(c1ccc2c(c1)CCC2)N1CCC[C@H](CCBr)C1 ZINC000147380217 EH For-Sale Reactive L3MBTL3 58 36 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(NC(=O)c3ccco3)c(C)c1)C2 ZINC000147380306 HI On-Demand Anodyne ROCK2 27 45 CCNc1cc(Oc2cccc(C(F)(F)F)c2)nc(C)n1 ZINC000147380326 CI For-Sale Anodyne PDS 42 34 Cc1ccc2[nH]c(C(=O)Nc3cccc(CN4CCSCC4)c3C)cc2c1 ZINC000147380336 GJ On-Demand Anodyne PYGL 70 43 Cc1ccc2[nH]c(C(=O)Nc3cccc(CN4CCSCC4)c3C)cc2c1 ZINC000147380336 GJ On-Demand Anodyne PYGM 20 43 CCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H](C(=O)Nc2ccccn2)C1 ZINC000147380339 ED On-Demand Anodyne P2RY12 134 34 CCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H](C(=O)Nc2ccccn2)C1 ZINC000147380339 ED On-Demand Anodyne TRY1_BOVIN 46 33 CCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H](C(=O)Nc2ccccn2)C1 ZINC000147380339 ED On-Demand Anodyne CTSK 20 40 CCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H](C(=O)Nc2ccccn2)C1 ZINC000147380339 ED On-Demand Anodyne DPP7 43 34 CC[C@H](CNS(=O)(=O)c1ccc(Cl)cc1OC)CC(=O)O ZINC000147380431 EE On-Demand Anodyne COLA 66 37 CC[C@H](CNS(=O)(=O)c1ccc(Cl)cc1OC)CC(=O)O ZINC000147380431 EE On-Demand Anodyne CPT1A 59 37 CC[C@H](CNS(=O)(=O)c1ccc(Cl)cc1OC)CC(=O)O ZINC000147380431 EE On-Demand Anodyne CPT1B 71 34 CC[C@H](CNS(=O)(=O)c1ccc(Cl)cc1OC)CC(=O)O ZINC000147380431 EE On-Demand Anodyne PTGDR2 41 39 CCCC[C@H](NC(N)=O)C(=O)N(CCC)Cc1ccc(C#N)cc1 ZINC000147380441 EF On-Demand Mild CTRB_BOVIN 50 36 O=C(c1ccc2c(c1)CCC2)N1CCC[C@@H](CCBr)C1 ZINC000147380443 EH For-Sale Reactive L3MBTL3 58 36 CCOc1cc(C=O)cc(OCC)c1OC ZINC000147380482 BE For-Sale Anodyne TUBB1 50 45 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(NC(=O)c3ccco3)c(C)c1)C2 ZINC000147380511 HI On-Demand Anodyne ROCK2 27 45 COc1ccc(CNC(=O)Cc2csc(-c3ccc(C(F)(F)F)cc3)n2)cc1 ZINC000147380526 HJ On-Demand Anodyne PPARG 18 52 COc1ccc(CNC(=O)Cc2csc(-c3ccc(C(F)(F)F)cc3)n2)cc1 ZINC000147380526 HJ On-Demand Anodyne AVPR1B 21 43 COc1ccc(CNC(=O)Cc2csc(-c3ccc(C(F)(F)F)cc3)n2)cc1 ZINC000147380526 HJ On-Demand Anodyne PPARA 42 52 COc1ccc(CNC(=O)Cc2csc(-c3ccc(C(F)(F)F)cc3)n2)cc1 ZINC000147380526 HJ On-Demand Anodyne TRPV1 20 41 COc1ccc(CNC(=O)Cc2csc(-c3ccc(C(F)(F)F)cc3)n2)cc1 ZINC000147380526 HJ On-Demand Anodyne CSNK1D 29 45 COc1ccc(CNC(=O)Cc2csc(-c3ccc(C(F)(F)F)cc3)n2)cc1 ZINC000147380526 HJ On-Demand Anodyne PPARD 67 51 COc1ccc(CNC(=O)Cc2csc(-c3ccc(C(F)(F)F)cc3)n2)cc1 ZINC000147380526 HJ On-Demand Anodyne CA9 18 45 Cc1c(CN2CCSCC2)cccc1NC(=O)C(=O)Nc1ccc(Cl)cc1 ZINC000147380581 HH On-Demand Anodyne F10 16 52 CCn1nc(C)c2c1CCN([C@@H](C(=O)NC)c1ccccc1)[C@H]2CCc1cccc(C)c1 ZINC000147380627 IJ Annotated Anodyne HCRTR1 44 81 CCCC[C@@H](NC(N)=O)C(=O)N(CCC)Cc1ccc(C#N)cc1 ZINC000147380631 EF On-Demand Mild CTRB_BOVIN 50 36 CC[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1OC)CC(=O)O ZINC000147380643 EE On-Demand Anodyne COLA 66 37 CC[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1OC)CC(=O)O ZINC000147380643 EE On-Demand Anodyne CPT1A 59 37 CC[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1OC)CC(=O)O ZINC000147380643 EE On-Demand Anodyne CPT1B 71 34 CC[C@@H](CNS(=O)(=O)c1ccc(Cl)cc1OC)CC(=O)O ZINC000147380643 EE On-Demand Anodyne PTGDR2 41 39 O=C(c1ccc2nccnc2c1)N1CCC[C@H](CCBr)C1 ZINC000147380682 EG For-Sale Reactive CCR3 0 41 O=C(c1ccc2nccnc2c1)N1CCC[C@H](CCBr)C1 ZINC000147380682 EG For-Sale Reactive ECE2 0 43 O=C(c1ccc2nccnc2c1)N1CCC[C@H](CCBr)C1 ZINC000147380682 EG For-Sale Reactive L3MBTL3 47 35 O=C(c1ccc2nccnc2c1)N1CCC[C@H](CCBr)C1 ZINC000147380682 EG For-Sale Reactive HPGD 47 40 O=C(NC1CCN(c2ccccc2)CC1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147380693 EH On-Demand Anodyne SIGMAR1 19 40 Cc1cc(NC(=O)c2ccc3c(c2)COC3)ccc1NC(=O)c1ccco1 ZINC000147380716 FI On-Demand Anodyne MAPK14 17 46 Cc1cc(NC(=O)c2ccc3c(c2)COC3)ccc1NC(=O)c1ccco1 ZINC000147380716 FI On-Demand Anodyne KCNK3 52 52 CCNc1ncnc(Oc2cccc(C(F)(F)F)c2)c1C ZINC000147380760 CI For-Sale Anodyne PDS 40 35 C[C@H](Cl)c1nc2cnccc2n1CCNC(=O)N(C)C ZINC000147380847 CE For-Sale Reactive PTAFR 38 40 O=C(NC1CCN(c2ccccc2)CC1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147380874 EH On-Demand Anodyne SIGMAR1 19 40 O=C(NC1CCN(c2ccccc2)CC1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147380874 EH On-Demand Anodyne SCN5A 19 41 O=C(c1ccc2nccnc2c1)N1CCC[C@@H](CCBr)C1 ZINC000147380897 EG For-Sale Reactive CCR3 0 41 O=C(c1ccc2nccnc2c1)N1CCC[C@@H](CCBr)C1 ZINC000147380897 EG For-Sale Reactive ECE2 0 43 O=C(c1ccc2nccnc2c1)N1CCC[C@@H](CCBr)C1 ZINC000147380897 EG For-Sale Reactive L3MBTL3 47 35 O=C(c1ccc2nccnc2c1)N1CCC[C@@H](CCBr)C1 ZINC000147380897 EG For-Sale Reactive HPGD 47 40 O=C(Nc1cn[nH]c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147380958 CE On-Demand Anodyne PPIA 16 43 C[C@@H]1CCCN1CCc1ccc(-c2ccc(CCn3cnnn3)cc2)cc1 ZINC000147381027 FH Annotated Anodyne KCNH2 21 57 CCOc1nc(N)nc(Oc2cccc(C(F)(F)F)c2)n1 ZINC000147381029 DF For-Sale Anodyne PDS 42 39 C[C@@H](Cl)c1nc2cnccc2n1CCNC(=O)N(C)C ZINC000147381045 CE For-Sale Reactive PTAFR 38 40 O=C(NC1CCN(c2ccccc2)CC1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147381139 EH On-Demand Anodyne SIGMAR1 17 40 O=C(NC1CCN(c2ccccc2)CC1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147381139 EH On-Demand Anodyne SCN5A 19 41 CCc1nc(COc2ccc(S(N)(=O)=O)c(C)c2)no1 ZINC000147381144 CD For-Sale Anodyne ACACB 0 42 CCN(C(=O)Nc1cc(Br)cc(C(=O)O)c1)C1CCCC1 ZINC000147381213 FH For-Sale Anodyne ACE 40 32 CC[C@H](NS(=O)(=O)c1cc(Cl)c(Br)s1)C(=O)O ZINC000147381236 FE For-Sale Anodyne ITGAV 55 36 C[C@@H]1CCCN1CCc1ccc(-c2ccc(CCn3ncnn3)cc2)cc1 ZINC000147381240 FH Annotated Anodyne HTR3A 17 42 C[C@@H]1CCCN1CCc1ccc(-c2ccc(CCn3ncnn3)cc2)cc1 ZINC000147381240 FH Annotated Anodyne HRH3 94 67 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cnn(C)c1-n1cccc1 ZINC000147381258 GG On-Demand Anodyne MRGPRX1 41 38 N[C@H](CCC(=O)NN1CCCCC1)c1ccccc1 ZINC000147381411 CD For-Sale Anodyne KCNQ2 44 37 N[C@H](CCC(=O)NN1CCCCC1)c1ccccc1 ZINC000147381411 CD For-Sale Anodyne DPP7 62 42 CCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CCCC1 ZINC000147381435 DH For-Sale Anodyne ACE 49 38 CCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CCCC1 ZINC000147381435 DH For-Sale Anodyne PYGL 21 40 CCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CCCC1 ZINC000147381435 DH For-Sale Anodyne CACNA1I 50 34 CCCCCCCCN1CCC[C@H](NC(C)C)C1 ZINC000147381446 CH For-Sale Mild BIRC2 42 33 c1cc(-c2cn3ccnc3c(Nc3ccc(N4CCOCC4)cc3)n2)c2cn[nH]c2c1 ZINC000147381503 HH For-Sale Anodyne SYK 43 69 c1cc(-c2cn3ccnc3c(Nc3ccc(N4CCOCC4)cc3)n2)c2cn[nH]c2c1 ZINC000147381503 HH For-Sale Anodyne MAPKAPK5 59 44 c1cc(-c2cn3ccnc3c(Nc3ccc(N4CCOCC4)cc3)n2)c2cn[nH]c2c1 ZINC000147381503 HH For-Sale Anodyne EPHB4 25 49 c1cc(-c2cn3ccnc3c(Nc3ccc(N4CCOCC4)cc3)n2)c2cn[nH]c2c1 ZINC000147381503 HH For-Sale Anodyne STAT6 74 39 O=C(N[C@H]1C[C@H]1c1ccccc1)N[C@@H]1CCCOc2ccc(F)cc21 ZINC000147381522 EH On-Demand Anodyne EPHX2 20 43 COc1ccc(C)cc1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147381558 EH For-Sale Reactive GRM3 16 41 COc1ccc(C)cc1C(=O)N1CCC[C@H](CCBr)C1 ZINC000147381558 EH For-Sale Reactive ACKR3 44 31 N[C@@H](CCC(=O)NN1CCCCC1)c1ccccc1 ZINC000147381576 CD For-Sale Anodyne KCNQ2 44 37 N[C@@H](CCC(=O)NN1CCCCC1)c1ccccc1 ZINC000147381576 CD For-Sale Anodyne DPP7 62 42 CCCCCCCCN1CCC[C@@H](NC(C)C)C1 ZINC000147381664 CH For-Sale Mild BIRC2 42 33 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(CN3CCC[C@@H]3C(N)=O)c1)C2 ZINC000147381683 HE On-Demand Anodyne ROCK2 25 41 CCCNc1cc(Oc2ccc3c(c2)OCO3)ncn1 ZINC000147381720 CF For-Sale Anodyne CLK1 51 40 CCCNc1cc(Oc2ccc3c(c2)OCO3)ncn1 ZINC000147381720 CF For-Sale Anodyne CLK2 40 35 CCCNc1cc(Oc2ccc3c(c2)OCO3)ncn1 ZINC000147381720 CF For-Sale Anodyne CLK4 65 35 CCCNc1cc(Oc2ccc3c(c2)OCO3)ncn1 ZINC000147381720 CF For-Sale Anodyne DYRK2 53 40 CC(C)CCCCNS(=O)(=O)c1cnn(CC(=O)O)c1 ZINC000147381743 DD For-Sale Anodyne TBXAS1 34 40 O=C(N[C@H]1C[C@@H]1c1ccccc1)N[C@@H]1CCCOc2ccc(F)cc21 ZINC000147381759 EH On-Demand Anodyne EPHX2 20 43 COc1ccc(C)cc1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147381774 EH For-Sale Reactive GRM3 16 41 COc1ccc(C)cc1C(=O)N1CCC[C@@H](CCBr)C1 ZINC000147381774 EH For-Sale Reactive ACKR3 44 31 Cc1cc(OCc2ncccn2)ccc1S(N)(=O)=O ZINC000147381807 CD For-Sale Anodyne CA2 17 42 Cc1cc(OCc2ncccn2)ccc1S(N)(=O)=O ZINC000147381807 CD For-Sale Anodyne CA7 23 42 Cc1cc(OCc2ncccn2)ccc1S(N)(=O)=O ZINC000147381807 CD For-Sale Anodyne CA12 16 42 Cc1cc(OCc2ncccn2)ccc1S(N)(=O)=O ZINC000147381807 CD For-Sale Anodyne CA9 18 42 CCCCCCCCNc1scnc1C(=O)O ZINC000147381889 CH For-Sale Mild MAP1 22 41 CCCCCCCCNc1scnc1C(=O)O ZINC000147381889 CH For-Sale Mild ASAH1 56 30 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCC[C@@H]3C(N)=O)c1)C2 ZINC000147381905 HE On-Demand Anodyne ROCK2 25 41 CCNc1cc(Oc2ccc3c(c2)OCO3)nc(N)n1 ZINC000147381958 CE For-Sale Anodyne DYRK2 48 37 NC(=O)C(=O)N1CC[C@H](Oc2ccccc2Cl)C1 ZINC000147381959 CC On-Demand Anodyne SCD1 44 55 NC(=O)C(=O)N1CC[C@H](Oc2ccccc2Cl)C1 ZINC000147381959 CC On-Demand Anodyne SCD 27 50 NCCc1ccc(C(=O)NN2CCCCC2)cc1 ZINC000147381966 BD For-Sale Anodyne CNR1 55 34 O=C(N[C@@H]1CCCOc2ccc(F)cc21)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147381976 EH On-Demand Anodyne EPHX2 20 43 CC[C@@H](CNS(=O)(=O)c1ccc2c(c1)CCC2)CC(=O)O ZINC000147381979 DD On-Demand Anodyne CA7 15 40 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc2[nH]c(=O)c(=O)[nH]c2c1 ZINC000147381996 HE On-Demand Anodyne MRGPRX1 47 45 O=C(c1coc2ccccc12)N1CCC[C@H](CCBr)C1 ZINC000147382068 EI For-Sale Reactive INHA 78 36 NC(=O)C(=O)N1CC[C@@H](Oc2ccccc2Cl)C1 ZINC000147382135 CC On-Demand Anodyne SCD1 44 55 NC(=O)C(=O)N1CC[C@@H](Oc2ccccc2Cl)C1 ZINC000147382135 CC On-Demand Anodyne SCD 27 50 Cc1cccc(NC(=O)c2cccc3c2OCCN3)c1Br ZINC000147382178 EH For-Sale Anodyne G2YM83_BOTF4 68 35 O=C(N[C@@H]1CCCOc2ccc(F)cc21)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147382179 EH On-Demand Anodyne EPHX2 20 43 Cc1ccc(NS(C)(=O)=O)c(C(=O)N(C)Cc2cccc(C(F)(F)F)c2)c1 ZINC000147382251 HH On-Demand Anodyne TACR1 20 45 Cc1ccc(NS(C)(=O)=O)c(C(=O)N(C)Cc2cccc(C(F)(F)F)c2)c1 ZINC000147382251 HH On-Demand Anodyne TRPV1 56 40 Cc1ccc(NS(C)(=O)=O)c(C(=O)N(C)Cc2cccc(C(F)(F)F)c2)c1 ZINC000147382251 HH On-Demand Anodyne HSP90AB1 16 43 Cc1ccc(NS(C)(=O)=O)c(C(=O)N(C)Cc2cccc(C(F)(F)F)c2)c1 ZINC000147382251 HH On-Demand Anodyne HSD17B2 25 42 Cc1ccc(NS(C)(=O)=O)c(C(=O)N(C)Cc2cccc(C(F)(F)F)c2)c1 ZINC000147382251 HH On-Demand Anodyne LIMK2 17 40 O=C(c1coc2ccccc12)N1CCC[C@@H](CCBr)C1 ZINC000147382270 EI For-Sale Reactive INHA 78 36 CCCc1cc(C(=O)Nc2cccc(CN3CCSCC3)c2C)n[nH]1 ZINC000147382276 FG On-Demand Anodyne MRGPRX1 43 40 CC[C@@H]1CCCCN1CCS(=O)(=O)c1cccc(C#N)c1 ZINC000147382310 DF On-Demand Mild CHRNA10 34 46 O=C(O)c1c(F)ccc2ccccc12 ZINC000147382356 AF For-Sale Anodyne KCNJ11 87 36 O=C(O)c1c(F)ccc2ccccc12 ZINC000147382356 AF For-Sale Anodyne CYP73A1 0 63 NCC(=O)N1CC[C@H](Oc2ccccc2Cl)C1 ZINC000147382360 CD On-Demand Anodyne SCD1 38 51 NCC(=O)N1CC[C@H](Oc2ccccc2Cl)C1 ZINC000147382360 CD On-Demand Anodyne SCD 27 50 Cc1nc(-c2ccc(NC(=O)c3cccc(N4C(=O)CCC4=O)c3)cc2)cs1 ZINC000147382382 GI On-Demand Anodyne PRNP 69 38 Cc1nc(-c2ccc(NC(=O)c3cccc(N4C(=O)CCC4=O)c3)cc2)cs1 ZINC000147382382 GI On-Demand Anodyne KCNK3 67 35 Cc1nc(-c2ccc(NC(=O)c3cccc(N4C(=O)CCC4=O)c3)cc2)cs1 ZINC000147382382 GI On-Demand Anodyne KCNK9 41 35 O=S(=O)(NCc1ccc(-n2ccnc2)c(F)c1)c1cccc2cnccc12 ZINC000147382424 GG On-Demand Anodyne P2RX7 29 47 O=S(=O)(NCc1ccc(-n2ccnc2)c(F)c1)c1cccc2cnccc12 ZINC000147382424 GG On-Demand Anodyne Q95J97_RABIT 0 48 CCOc1nc(NC)nc(Oc2ccc3c(c2)OCO3)n1 ZINC000147382477 CD For-Sale Anodyne CLK4 52 32 Cc1cc(OCC(=O)N2CCCC2)ccc1S(N)(=O)=O ZINC000147382486 CC For-Sale Anodyne HTR1D 16 41 Cc1cc(OCC(=O)N2CCCC2)ccc1S(N)(=O)=O ZINC000147382486 CC For-Sale Anodyne HTR1B 18 41 Cc1cc(OCC(=O)N2CCCC2)ccc1S(N)(=O)=O ZINC000147382486 CC For-Sale Anodyne COLA 32 41 Cc1cc(OCC(=O)N2CCCC2)ccc1S(N)(=O)=O ZINC000147382486 CC For-Sale Anodyne CPT1A 29 41 Cc1cc(OCC(=O)N2CCCC2)ccc1S(N)(=O)=O ZINC000147382486 CC For-Sale Anodyne GPR183 0 51 CC[C@H]1CCCCN1CCS(=O)(=O)c1cccc(C#N)c1 ZINC000147382510 DF On-Demand Mild CHRNA10 34 46 NNc1cc(Sc2ccccc2[N+](=O)[O-])nc(C2CC2)n1 ZINC000147382539 DF For-Sale Bother PDE7A 19 46 NCC(=O)N1CC[C@@H](Oc2ccccc2Cl)C1 ZINC000147382605 CD On-Demand Anodyne SCD1 38 51 NCC(=O)N1CC[C@@H](Oc2ccccc2Cl)C1 ZINC000147382605 CD On-Demand Anodyne SCD 27 50 CCOc1ccc([C@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1OCC ZINC000147382614 GI On-Demand Anodyne BMP1 55 35 CCOc1ccc([C@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1OCC ZINC000147382614 GI On-Demand Anodyne CYP3A4 15 43 O=C(NCC1(CO)CCCC1)c1cccc2c1OCCN2 ZINC000147382642 CD For-Sale Anodyne HCN1 51 34 O=C(NCC1(CO)CCCC1)c1cccc2c1OCCN2 ZINC000147382642 CD For-Sale Anodyne HCN4 47 30 CC[C@H](NS(=O)(=O)c1cc(Br)c(C)cc1Br)C(=O)O ZINC000147382643 HF On-Demand Anodyne ITGAV 65 42 CC[C@H](NS(=O)(=O)c1cc(Br)c(C)cc1Br)C(=O)O ZINC000147382643 HF On-Demand Anodyne LEF 38 42 CCC(=O)Nc1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147382645 HH On-Demand Anodyne CCR3 24 41 CCC(=O)Nc1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147382645 HH On-Demand Anodyne EPHX2 22 40 CCC(=O)Nc1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147382645 HH On-Demand Anodyne NAMPT 35 40 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)N(C)C)CC1 ZINC000147382694 EB On-Demand Anodyne P2RY12 151 36 C=CCOc1ccc(C(=O)Nc2cccc(CN3CCSCC3)c2C)cc1OC ZINC000147382697 HI On-Demand Mild SLC9A1 67 40 C=CCOc1ccc(C(=O)Nc2cccc(CN3CCSCC3)c2C)cc1OC ZINC000147382697 HI On-Demand Mild MRGPRX1 45 43 CNc1cn2ccnc2c(Oc2ccc3c(c2)OCO3)n1 ZINC000147382725 CE For-Sale Anodyne HIVRT 0 41 COc1ccc(-c2cc3[nH]c(C(=O)O)cc3o2)cc1 ZINC000147382731 CG For-Sale Anodyne CYP1B1 19 45 COc1ccc(-c2cc3[nH]c(C(=O)O)cc3o2)cc1 ZINC000147382731 CG For-Sale Anodyne CYP1A1 18 45 COc1ccc(-c2cc3[nH]c(C(=O)O)cc3o2)cc1 ZINC000147382731 CG For-Sale Anodyne TUBB2B 41 41 CCn1cc(NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147382754 DF On-Demand Anodyne CACNA1I 41 31 Cc1cc(OCC(=O)N2CCCCC2)ccc1S(N)(=O)=O ZINC000147382763 DD For-Sale Anodyne HTR1D 15 41 Cc1cc(OCC(=O)N2CCCCC2)ccc1S(N)(=O)=O ZINC000147382763 DD For-Sale Anodyne HTR1B 18 41 Cc1cc(OCC(=O)N2CCCCC2)ccc1S(N)(=O)=O ZINC000147382763 DD For-Sale Anodyne COLA 27 40 Cc1cc(OCC(=O)N2CCCCC2)ccc1S(N)(=O)=O ZINC000147382763 DD For-Sale Anodyne CPT1A 25 40 Cc1cc(OCC(=O)N2CCCCC2)ccc1S(N)(=O)=O ZINC000147382763 DD For-Sale Anodyne GPR183 0 50 CN(CCS(=O)(=O)c1cccc(C#N)c1)c1ccccc1 ZINC000147382767 DE For-Sale Mild KCNA5 0 45 CC(C)c1nc(NN)cc(Sc2ccccc2[N+](=O)[O-])n1 ZINC000147382776 DF For-Sale Bother PDE7A 19 47 Cc1cccnc1C(=O)N1CCC[C@H]1C ZINC000147382779 BE On-Demand Anodyne HCRTR1 44 35 Cc1cccnc1C(=O)N1CCC[C@H]1C ZINC000147382779 BE On-Demand Anodyne TRPC3 34 41 CCOc1ccc([C@@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1OCC ZINC000147382846 GI On-Demand Anodyne BMP1 55 35 CCOc1ccc([C@@H](NC(=O)N(C)Cc2cscn2)C(C)C)cc1OCC ZINC000147382846 GI On-Demand Anodyne CYP3A4 15 43 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne RARA 33 42 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne AVPR2 66 42 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne AVPR1A 36 52 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne F2R 0 43 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne CPT1A 43 39 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne PRNP 25 40 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne GRM4 35 40 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne NR1H4 25 47 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne MTTP 54 36 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne AKR1C3 46 40 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne NR2E3 62 38 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne SHH 43 41 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne AKR1C2 73 37 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne SMO 34 40 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne GALE 0 40 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne Q25615_ONCVO 53 32 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne KCNK3 114 45 Cc1cc(NC(=O)c2cccc(F)c2Cl)ccc1C(=O)O ZINC000147382861 DH On-Demand Anodyne KCNK9 84 40 CCC(=O)Nc1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147382884 HH On-Demand Anodyne CCR3 24 41 CCC(=O)Nc1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147382884 HH On-Demand Anodyne EPHX2 22 40 CCC(=O)Nc1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147382884 HH On-Demand Anodyne NAMPT 35 40 CC(C)CCCCNS(=O)(=O)c1cnn(CCC(=O)O)c1 ZINC000147382888 DD For-Sale Anodyne TBXAS1 35 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)N(C)C)CC1 ZINC000147382913 EB On-Demand Anodyne P2RY12 151 36 CCNc1ncc(Cl)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147382944 CG For-Sale Anodyne DYRK1A 31 43 CCNc1ncc(Cl)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147382944 CG For-Sale Anodyne CLK1 41 43 CCNc1ncc(Cl)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147382944 CG For-Sale Anodyne CLK2 37 43 CCNc1ncc(Cl)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147382944 CG For-Sale Anodyne CLK4 58 43 CCNc1ncc(Cl)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147382944 CG For-Sale Anodyne DYRK1B 28 43 CCCCCCCCNC(=O)c1cc(S(=O)(=O)Cl)cn1C ZINC000147382979 EG For-Sale Unstable ASAH1 96 38 Cc1cccnc1C(=O)N1CCC[C@@H]1C ZINC000147382998 BE On-Demand Anodyne HCRTR1 44 35 Cc1cccnc1C(=O)N1CCC[C@@H]1C ZINC000147382998 BE On-Demand Anodyne TRPC3 34 41 CC(C)CNC(=O)c1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)cc1 ZINC000147383044 HF On-Demand Anodyne F3 80 34 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne RARA 29 45 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne AVPR2 31 40 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne AVPR1A 20 40 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne F3 66 33 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne NR1H4 18 49 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne P4HTM 0 45 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne PLAU 15 40 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne CSF1R 16 41 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne TAAR1 38 43 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne AKR1C3 38 44 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne AKR1C2 41 44 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne KCNK3 105 43 Cc1ccc(C(=O)Nc2ccc(C(=O)O)c(C)c2)cc1Br ZINC000147383095 EI On-Demand Anodyne KCNK9 56 41 CCCNc1cc(Oc2ccc3c(c2)OCO3)nc(N)n1 ZINC000147383142 CE For-Sale Anodyne EDNRA 15 42 CCCNc1cc(Oc2ccc3c(c2)OCO3)nc(N)n1 ZINC000147383142 CE For-Sale Anodyne DYRK2 41 38 CC(C)CCCCNS(=O)(=O)Cc1ccc(C(=O)O)cc1 ZINC000147383146 DF For-Sale Anodyne RARB 16 50 CC(C)CCCCNS(=O)(=O)Cc1ccc(C(=O)O)cc1 ZINC000147383146 DF For-Sale Anodyne PLA2G4A 40 37 CC(C)CCCCNS(=O)(=O)Cc1ccc(C(=O)O)cc1 ZINC000147383146 DF For-Sale Anodyne TMPRSS11D 73 39 CCC(=O)Nc1ccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147383148 GG On-Demand Anodyne EPHX2 40 44 COC(=O)c1ccc(C(=O)Nc2cccc(CN3CCSCC3)c2C)s1 ZINC000147383156 GH On-Demand Anodyne MRGPRX1 40 36 CN(C(C)(C)C)S(=O)(=O)CCNC(=O)OCc1ccccc1 ZINC000147383158 ED On-Demand Anodyne CTSB 43 39 CN(C(C)(C)C)S(=O)(=O)CCNC(=O)OCc1ccccc1 ZINC000147383158 ED On-Demand Anodyne PAPA1_CARPA 56 39 CN(C(C)(C)C)S(=O)(=O)CCNC(=O)OCc1ccccc1 ZINC000147383158 ED On-Demand Anodyne CYSP_TRYCR 47 37 CN(C(C)(C)C)S(=O)(=O)CCNC(=O)OCc1ccccc1 ZINC000147383158 ED On-Demand Anodyne CTSK 22 40 CN(C(C)(C)C)S(=O)(=O)CCNC(=O)OCc1ccccc1 ZINC000147383158 ED On-Demand Anodyne CAPNS1 56 35 CN(C(C)(C)C)S(=O)(=O)CCNC(=O)OCc1ccccc1 ZINC000147383158 ED On-Demand Anodyne CTSS 15 47 CN(C(C)(C)C)S(=O)(=O)CCNC(=O)OCc1ccccc1 ZINC000147383158 ED On-Demand Anodyne CAPN1 66 41 CN(C(C)(C)C)S(=O)(=O)CCNC(=O)OCc1ccccc1 ZINC000147383158 ED On-Demand Anodyne CAPN2 96 35 CN(C(C)(C)C)S(=O)(=O)CCNC(=O)OCc1ccccc1 ZINC000147383158 ED On-Demand Anodyne NPR 74 45 CCCCCCCCNC(=O)c1csc(S(=O)(=O)Cl)c1 ZINC000147383183 EH For-Sale Unstable KCNQ1 0 41 CCCCCCCCNC(=O)c1csc(S(=O)(=O)Cl)c1 ZINC000147383183 EH For-Sale Unstable ASAH1 80 34 CC(C)CNC(=O)c1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)cc1 ZINC000147383249 HF On-Demand Anodyne F3 80 34 CCCCCCCCNC(=O)c1cc(S(=O)(=O)Cl)c[nH]1 ZINC000147383379 DG For-Sale Unstable ALPL 40 34 CCCCCCCCNC(=O)c1cc(S(=O)(=O)Cl)c[nH]1 ZINC000147383379 DG For-Sale Unstable ASAH1 84 37 CCC(=O)Nc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147383393 HJ On-Demand Anodyne ROCK2 31 51 CCC(=O)Nc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147383393 HJ On-Demand Anodyne MET 56 46 CCC(=O)Nc1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147383393 HJ On-Demand Anodyne NAMPT 68 52 C[C@@H](CCN)C(=O)NN1CCCCC1 ZINC000147383540 AC For-Sale Anodyne DPP7 21 41 Cc1cc(NC(=O)C2[C@H]3CCCC[C@H]23)ccc1C(=O)O ZINC000147383551 CG On-Demand Anodyne HRH3 0 41 Cc1cc(NC(=O)C2[C@H]3CCCC[C@H]23)ccc1C(=O)O ZINC000147383551 CG On-Demand Anodyne EPHX2 16 41 CCNc1ncc(C)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147383555 CF For-Sale Anodyne CLK4 40 36 S=c1[nH]ccn1Cc1cnc[nH]1 ZINC000147383582 AD For-Sale Anodyne DBH 61 46 CCCCCCCCNC(=O)c1csc(S(=O)(=O)Cl)c1C ZINC000147383587 FI For-Sale Unstable ASAH1 91 36 C[C@H](CCN)C(=O)NN1CCCCC1 ZINC000147383757 AC For-Sale Anodyne DPP7 21 41 CCCNc1ncc(Cl)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147383768 DG For-Sale Anodyne DYRK1A 25 44 CCCNc1ncc(Cl)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147383768 DG For-Sale Anodyne CLK1 36 44 CCCNc1ncc(Cl)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147383768 DG For-Sale Anodyne CLK2 31 44 CCCNc1ncc(Cl)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147383768 DG For-Sale Anodyne CLK4 46 44 CCCNc1ncc(Cl)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147383768 DG For-Sale Anodyne DYRK1B 23 44 Cc1cc(NC(=O)C2[C@H]3CCCC[C@@H]23)ccc1C(=O)O ZINC000147383777 CG For-Sale Anodyne HRH3 0 41 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(NC(N)=O)cc1 ZINC000147383824 GG On-Demand Anodyne PRNP 46 35 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(NC(N)=O)cc1 ZINC000147383824 GG On-Demand Anodyne MRGPRX1 46 43 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(NC(N)=O)cc1 ZINC000147383824 GG On-Demand Anodyne NOD2 44 39 CCCCCCCCNC(=O)c1n[nH]c(C)c1S(=O)(=O)Cl ZINC000147383825 EF For-Sale Unstable ASAH1 63 34 CCCNc1cncc(Oc2ccc3c(c2)OCO3)n1 ZINC000147383938 CF For-Sale Anodyne DYRK2 42 39 Cc1cc(C(=O)N2CCN([C@@H]3CCS(=O)(=O)C3)CC2)cc([N+](=O)[O-])c1 ZINC000147383944 FC On-Demand Bother L3MBTL3 46 38 Cc1cc(NC(=O)C2[C@@H]3CCCC[C@@H]23)ccc1C(=O)O ZINC000147383988 CG On-Demand Anodyne HRH3 0 41 Cc1cc(NC(=O)C2[C@@H]3CCCC[C@@H]23)ccc1C(=O)O ZINC000147383988 CG On-Demand Anodyne EPHX2 16 41 CCCCCCCCNC(=O)c1cc(S(=O)(=O)Cl)c(C)o1 ZINC000147384077 EH For-Sale Unstable ASAH1 87 33 COC(=O)c1cc2cc(NC(=O)NC[C@@H](O)COc3c(C)cccc3C)ccc2o1 ZINC000147384093 HG On-Demand Anodyne ADRB1 41 32 CCNC(=O)CCOc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147384119 CC For-Sale Anodyne CA2 28 40 CCNC(=O)CCOc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147384119 CC For-Sale Anodyne CA1 21 40 Cc1cc(C(=O)N2CCN([C@H]3CCS(=O)(=O)C3)CC2)cc([N+](=O)[O-])c1 ZINC000147384173 FC On-Demand Bother L3MBTL3 46 38 Cc1cc(NC(=O)c2ocnc2C)ccc1C(=O)O ZINC000147384190 CE On-Demand Anodyne NR1H4 16 41 Cc1cc(NC(=O)c2ocnc2C)ccc1C(=O)O ZINC000147384190 CE On-Demand Anodyne IMPDH2 0 40 Cc1cc(NC(=O)c2ocnc2C)ccc1C(=O)O ZINC000147384190 CE On-Demand Anodyne AKR1C2 40 33 Cc1cc(NC(=O)c2ocnc2C)ccc1C(=O)O ZINC000147384190 CE On-Demand Anodyne DGAT1 22 40 Cc1cc(NC(=O)c2ocnc2C)ccc1C(=O)O ZINC000147384190 CE On-Demand Anodyne KCNK3 71 35 Cc1cc(NC(=O)c2ocnc2C)ccc1C(=O)O ZINC000147384190 CE On-Demand Anodyne KCNK9 48 36 CCCCO[C@@H](C)C(=O)NC1CCN(C(=O)C(C)C)CC1 ZINC000147384198 CD On-Demand Anodyne EPHX2 23 45 CC(C)CCCCNS(=O)(=O)c1ccc(C(=O)O)cn1 ZINC000147384252 DD For-Sale Anodyne P4HTM 0 40 CCCCCCCCNC(=O)Cc1ccc(S(=O)(=O)Cl)s1 ZINC000147384269 FH For-Sale Unstable ASAH1 81 36 COC(=O)c1cc2cc(NC(=O)NC[C@H](O)COc3c(C)cccc3C)ccc2o1 ZINC000147384330 HG On-Demand Anodyne ADRB1 41 32 CS(=O)(=O)NC[C@@H]1CCCCN1C(=O)c1ccc(Oc2cccnc2)cc1 ZINC000147384336 GE On-Demand Anodyne CPT1A 53 35 CCCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147384354 DC For-Sale Anodyne CA2 32 40 CCCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147384354 DC For-Sale Anodyne CA1 27 40 CCCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147384354 DC For-Sale Anodyne MTNR1A 37 42 CCCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147384354 DC For-Sale Anodyne PLA2G4B 68 34 CCCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147384354 DC For-Sale Anodyne CA12 19 40 CCCCNC(=O)COc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147384354 DC For-Sale Anodyne CA9 23 40 NC(=O)CCCC(=O)NNc1ccc([N+](=O)[O-])cc1 ZINC000147384360 CC On-Demand Reactive CA4 15 41 NC(=O)CCCC(=O)NNc1ccc([N+](=O)[O-])cc1 ZINC000147384360 CC On-Demand Reactive ACR 20 40 CCCCO[C@H](C)C(=O)NC1CCN(C(=O)C(C)C)CC1 ZINC000147384370 CD On-Demand Anodyne EPHX2 23 45 CCCNc1nc(C)cc(Oc2ccc3c(c2)OCO3)n1 ZINC000147384395 CG For-Sale Anodyne DYRK1A 23 41 CCCNc1nc(C)cc(Oc2ccc3c(c2)OCO3)n1 ZINC000147384395 CG For-Sale Anodyne CLK1 33 41 CCCNc1nc(C)cc(Oc2ccc3c(c2)OCO3)n1 ZINC000147384395 CG For-Sale Anodyne DYRK2 49 41 C[C@@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147384446 BD For-Sale Anodyne SLC15A1 0 40 C[C@@H](NC(=O)[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147384446 BD For-Sale Anodyne GPR88 0 54 N#Cc1cccc(S(=O)(=O)CCN2CCC[C@@H]2C(N)=O)c1 ZINC000147384483 DC On-Demand Mild ITGA4 59 34 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne ACE 66 46 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne MME 93 59 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne LTA4H 26 45 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne ANPEP 78 43 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne RNPEP 25 45 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne CTSB 45 47 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne CPA1 38 46 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne SLC15A1 0 41 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne C3AR1 55 34 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne CAPNS1 47 36 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne MMP3 36 44 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne HLA-DRB1 42 35 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne CAPN1 70 41 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne CAPN2 105 41 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne ENPEP 68 33 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne ACE2 91 46 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne CTSC 27 40 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne FPR1 50 38 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne NPR 70 43 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne XIAP 63 34 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne AMPX_VIBPR 0 45 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne KIF11 0 41 CC[C@H](NC(=O)[C@@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384490 CD On-Demand Anodyne SLC15A2 0 49 FC(F)(F)c1cnc(N(CCBr)C2CCCCC2)c(Cl)c1 ZINC000147384516 GK For-Sale Reactive TRPM8 40 35 CS(=O)(=O)NC[C@H]1CCCCN1C(=O)c1ccc(Oc2cccnc2)cc1 ZINC000147384552 GE On-Demand Anodyne CPT1A 53 35 NC(=O)[C@H]1CCCN1Cc1cccc(NC(=O)c2ccc3c(c2)COC3)c1 ZINC000147384598 FE On-Demand Anodyne PLAU 17 44 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(C(=O)C(C)C)CC1 ZINC000147384611 EC On-Demand Anodyne EPHX2 17 47 CCCC[C@H](NC(N)=O)C(=O)NC1CCN(C(=O)C(C)C)CC1 ZINC000147384611 EC On-Demand Anodyne NOD1 41 33 CC(=O)N1C(=O)/C(=C\c2ccccc2)NC(=O)[C@@H]1Cc1ccccc1 ZINC000147384667 EE For-Sale Anodyne GALR1 43 31 C[C@@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147384682 BD For-Sale Anodyne SLC15A1 0 40 C[C@@H](NC(=O)[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147384682 BD For-Sale Anodyne GPR88 0 54 N#Cc1cccc(S(=O)(=O)CCN2CCC[C@H]2C(N)=O)c1 ZINC000147384698 DC On-Demand Mild ITGA4 59 34 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne ACE 66 46 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne MME 93 59 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne LTA4H 26 45 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne ANPEP 78 43 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne RNPEP 25 45 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne CTSB 45 47 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne CPA1 38 46 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne SLC15A1 0 41 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne C3AR1 55 34 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne CAPNS1 47 36 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne MMP3 36 44 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne HLA-DRB1 42 35 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne CAPN1 70 41 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne CAPN2 105 41 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne ENPEP 68 33 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne ACE2 91 46 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne CTSC 27 40 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne FPR1 50 38 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne NPR 70 43 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne XIAP 63 34 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne AMPX_VIBPR 0 45 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne KIF11 0 41 CC[C@H](NC(=O)[C@H](C)[C@@H](N)c1ccccc1)C(=O)O ZINC000147384704 CD On-Demand Anodyne SLC15A2 0 49 CCCCCCCCNC(=O)c1cccc2c1OCCN2 ZINC000147384732 CH For-Sale Mild ASAH1 75 34 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCCC[C@@H]1CBr ZINC000147384774 GE For-Sale Reactive CASP3 92 40 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCCC[C@@H]1CBr ZINC000147384774 GE For-Sale Reactive PKM 45 53 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCCC[C@@H]1CBr ZINC000147384774 GE For-Sale Reactive CASP7 102 39 COc1ccc([C@H](NC(=O)Cc2cccc(OC(C)C)c2)C2CC2)cc1 ZINC000147384790 FI On-Demand Anodyne MTNR1A 58 44 COc1ccc([C@H](NC(=O)Cc2cccc(OC(C)C)c2)C2CC2)cc1 ZINC000147384790 FI On-Demand Anodyne MTNR1B 51 44 COc1ccc([C@H](NC(=O)Cc2cccc(OC(C)C)c2)C2CC2)cc1 ZINC000147384790 FI On-Demand Anodyne FFAR1 18 40 Cc1cccc(C(=O)O)c1N1CCCC1 ZINC000147384805 BE For-Sale Anodyne SLC6A1 55 38 Cc1cccc(C(=O)O)c1N1CCCC1 ZINC000147384805 BE For-Sale Anodyne FABP4 39 40 Cc1cccc(C(=O)O)c1N1CCCC1 ZINC000147384805 BE For-Sale Anodyne AKR1C2 23 43 Cc1cccc(C(=O)O)c1N1CCCC1 ZINC000147384805 BE For-Sale Anodyne BRPF1 0 40 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(C(=O)C(C)C)CC1 ZINC000147384823 EC On-Demand Anodyne EPHX2 17 47 CCCC[C@@H](NC(N)=O)C(=O)NC1CCN(C(=O)C(C)C)CC1 ZINC000147384823 EC On-Demand Anodyne NOD1 41 33 Nc1cc(Oc2ccc3c(c2)OCO3)ncn1 ZINC000147384866 BD For-Sale Anodyne CLK4 45 32 COc1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1Cl ZINC000147384868 GG On-Demand Anodyne PDE5A 24 42 CCCCCCCCNC(=O)c1cc(S(=O)(=O)Cl)c(Br)o1 ZINC000147384882 HI For-Sale Unstable ASAH1 82 34 CCCCC[C@H](Br)[C@H](Br)C[C@@H](Br)[C@@H](Br)CCCCCCCC(=O)OC ZINC000147384964 KK For-Sale Reactive ENPP2 28 43 CCCCC[C@H](Br)[C@H](Br)C[C@@H](Br)[C@@H](Br)CCCCCCCC(=O)OC ZINC000147384964 KK For-Sale Reactive NOD1 58 36 CCCCC[C@H](Br)[C@H](Br)C[C@@H](Br)[C@@H](Br)CCCCCCCC(=O)OC ZINC000147384964 KK For-Sale Reactive CQSS 63 39 COc1ccc([C@H](NC(=O)[C@@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147384980 EI On-Demand Anodyne CTSL 33 42 COc1ccc([C@H](NC(=O)[C@@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147384980 EI On-Demand Anodyne CTSS 25 42 COc1ccc([C@H](NC(=O)[C@@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147384980 EI On-Demand Anodyne ACE2 52 36 COc1ccc([C@H](NC(=O)[C@@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147384980 EI On-Demand Anodyne PSMB8 46 33 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCCC[C@H]1CBr ZINC000147385010 GE For-Sale Reactive CASP3 92 40 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCCC[C@H]1CBr ZINC000147385010 GE For-Sale Reactive PKM 45 53 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCCC[C@H]1CBr ZINC000147385010 GE For-Sale Reactive CASP7 102 39 COc1cccc(CCC(=O)Nc2cccc(CN3CCSCC3)c2C)c1 ZINC000147385030 GI On-Demand Anodyne DRD4 40 32 COc1cccc(CCC(=O)Nc2cccc(CN3CCSCC3)c2C)c1 ZINC000147385030 GI On-Demand Anodyne HRH2 29 42 COc1cccc(CCC(=O)Nc2cccc(CN3CCSCC3)c2C)c1 ZINC000147385030 GI On-Demand Anodyne PTGER3 20 41 COc1cccc(CCC(=O)Nc2cccc(CN3CCSCC3)c2C)c1 ZINC000147385030 GI On-Demand Anodyne CCR3 22 42 COc1cccc(CCC(=O)Nc2cccc(CN3CCSCC3)c2C)c1 ZINC000147385030 GI On-Demand Anodyne ABCB1 20 40 COc1cccc(CCC(=O)Nc2cccc(CN3CCSCC3)c2C)c1 ZINC000147385030 GI On-Demand Anodyne HCAR2 19 45 C[C@@H](NC(=O)C1[C@@H]2CCCC[C@@H]12)C(=O)O ZINC000147385034 BD On-Demand Anodyne SLC15A2 0 40 CCCNc1ncc(Br)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147385068 FH For-Sale Anodyne CLK2 29 41 CCCNc1ncc(Br)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147385068 FH For-Sale Anodyne CLK4 29 41 CCCC[C@H](NC(N)=O)C(=O)NCc1ccnc(N2CCOCC2)c1 ZINC000147385079 EC On-Demand Anodyne PCSK5 53 35 CCCC[C@H](NC(N)=O)C(=O)NCc1ccnc(N2CCOCC2)c1 ZINC000147385079 EC On-Demand Anodyne FURIN 47 35 CCCC[C@H](NC(N)=O)C(=O)NCc1ccnc(N2CCOCC2)c1 ZINC000147385079 EC On-Demand Anodyne SMG1 40 34 CCCCCCCCNC(=O)c1cc(S(N)(=O)=O)c(Br)o1 ZINC000147385091 GF For-Sale Mild ASAH1 86 37 COC(=O)c1cc2cc(NC(=O)NCc3ccc(-n4ccnc4)c(F)c3)ccc2o1 ZINC000147385212 HH On-Demand Anodyne NOS2 79 33 COC(=O)c1cc2cc(NC(=O)NCc3ccc(-n4ccnc4)c(F)c3)ccc2o1 ZINC000147385212 HH On-Demand Anodyne ROCK2 15 40 COc1ccnc(N[C@@H]2CCNC2)c1 ZINC000147385218 AC For-Sale Anodyne CHEK2 20 46 COc1ccnc(N[C@@H]2CCNC2)c1 ZINC000147385218 AC For-Sale Anodyne PRKD1 44 37 COc1ccnc(N[C@@H]2CCNC2)c1 ZINC000147385218 AC For-Sale Anodyne IRAK4 32 42 COc1ccc([C@@H](NC(=O)[C@@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147385237 EI On-Demand Anodyne CTSL 33 42 COc1ccc([C@@H](NC(=O)[C@@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147385237 EI On-Demand Anodyne CTSS 25 42 COc1ccc([C@@H](NC(=O)[C@@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147385237 EI On-Demand Anodyne ACE2 52 36 COc1ccc([C@@H](NC(=O)[C@@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147385237 EI On-Demand Anodyne PSMB8 46 33 CC[C@@H]1CN(S(=O)(=O)c2cccc(C)c2)CC[C@@H]1N ZINC000147385242 CD On-Demand Anodyne AKR1C3 42 37 COC(=O)c1c(C)[nH]c(C(=O)Nc2cccc(CN3CCSCC3)c2C)c1C ZINC000147385252 HH On-Demand Anodyne MRGPRX1 40 35 CCCCCCCCNC(=O)c1cc(S(N)(=O)=O)c[nH]1 ZINC000147385277 DD For-Sale Mild CA2 32 60 CCCCCCCCNC(=O)c1cc(S(N)(=O)=O)c[nH]1 ZINC000147385277 DD For-Sale Mild ASAH1 88 37 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccnc(N2CCOCC2)c1 ZINC000147385279 EC On-Demand Anodyne PCSK5 53 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccnc(N2CCOCC2)c1 ZINC000147385279 EC On-Demand Anodyne FURIN 47 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccnc(N2CCOCC2)c1 ZINC000147385279 EC On-Demand Anodyne SMG1 40 34 O=C1CCCc2cc(S(=O)(=O)NCc3ccc(-n4ccnc4)c(F)c3)ccc2N1 ZINC000147385323 HF On-Demand Anodyne PKM 28 43 CN(C)Cc1cccc(-c2cnc(N)c(-c3nc4ccccc4[nH]3)n2)c1 ZINC000147385328 EG For-Sale Anodyne ATM 34 57 CN(C)Cc1cccc(-c2cnc(N)c(-c3nc4ccccc4[nH]3)n2)c1 ZINC000147385328 EG For-Sale Anodyne ATR 15 57 CN(C)Cc1cccc(-c2cnc(N)c(-c3nc4ccccc4[nH]3)n2)c1 ZINC000147385328 EG For-Sale Anodyne RET 23 40 O=C(c1cc(Cl)ccc1F)N(Cc1ccccc1)c1ccccc1 ZINC000147385331 EK For-Sale Anodyne ALDH1A1 23 40 O=C(c1cc(Cl)ccc1F)N(Cc1ccccc1)c1ccccc1 ZINC000147385331 EK For-Sale Anodyne NS5B 19 42 CCCNc1nccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147385332 CF For-Sale Anodyne DYRK1A 30 44 CCCNc1nccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147385332 CF For-Sale Anodyne CLK1 42 44 CCCNc1nccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147385332 CF For-Sale Anodyne CLK2 38 44 CCCNc1nccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147385332 CF For-Sale Anodyne CLK4 53 44 CCCNc1nccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147385332 CF For-Sale Anodyne DYRK2 41 39 CCCNc1nccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147385332 CF For-Sale Anodyne DYRK1B 28 44 COc1ccccc1Sc1cc(NN)nc(C(C)C)n1 ZINC000147385376 CG For-Sale Anodyne ALS 40 38 COC(=O)c1cc2cc(NC(=O)N3C[C@H](c4ccccc4)O[C@H](C)C3)ccc2o1 ZINC000147385427 GI On-Demand Anodyne GYRB 18 40 COc1ccnc(N[C@H]2CCNC2)c1 ZINC000147385436 AC For-Sale Anodyne CHEK2 20 46 COc1ccnc(N[C@H]2CCNC2)c1 ZINC000147385436 AC For-Sale Anodyne PRKD1 44 37 COc1ccnc(N[C@H]2CCNC2)c1 ZINC000147385436 AC For-Sale Anodyne IRAK4 32 42 COc1ccc([C@@H](NC(=O)[C@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147385454 EI On-Demand Anodyne CTSL 33 42 COc1ccc([C@@H](NC(=O)[C@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147385454 EI On-Demand Anodyne CTSS 25 42 COc1ccc([C@@H](NC(=O)[C@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147385454 EI On-Demand Anodyne ACE2 52 36 COc1ccc([C@@H](NC(=O)[C@H](C)Cc2cccc(F)c2)C2CC2)cc1 ZINC000147385454 EI On-Demand Anodyne PSMB8 46 33 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccnc2Oc2ccccc2)C1 ZINC000147385458 HG On-Demand Anodyne P2RY1 47 39 CCN(Cc1ccc(OC)c(OC)c1)C(=O)c1cc(C)cc([N+](=O)[O-])c1 ZINC000147385465 FH On-Demand Bother MT-ND1 25 41 Cc1cc(OCCc2ccncc2)ccc1S(N)(=O)=O ZINC000147385466 CD For-Sale Anodyne CA2 19 45 Cc1cc(OCCc2ccncc2)ccc1S(N)(=O)=O ZINC000147385466 CD For-Sale Anodyne CA1 15 45 Cc1cc(OCCc2ccncc2)ccc1S(N)(=O)=O ZINC000147385466 CD For-Sale Anodyne CA7 22 45 Cc1cc(OCCc2ccncc2)ccc1S(N)(=O)=O ZINC000147385466 CD For-Sale Anodyne CA12 15 45 Cc1cc(OCCc2ccncc2)ccc1S(N)(=O)=O ZINC000147385466 CD For-Sale Anodyne CA9 18 45 CC[C@H]1CN(S(=O)(=O)c2cccc(C)c2)CC[C@@H]1N ZINC000147385471 CD On-Demand Anodyne AKR1C3 42 37 CCCCCCCCNC(=O)c1cc(S(N)(=O)=O)c(C)o1 ZINC000147385485 DE On-Demand Mild ASAH1 77 35 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cc(Cl)cn1C ZINC000147385499 FH On-Demand Anodyne MRGPRX1 31 40 COC(=O)Cc1csc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)n1 ZINC000147385527 FE On-Demand Anodyne ROCK2 35 46 COc1cc([N+](=O)[O-])ccc1S(=O)(=O)NCc1ccc(-n2ccnc2)c(F)c1 ZINC000147385531 HE On-Demand Bother CYP19A1 16 41 CCNc1cccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147385608 CG For-Sale Anodyne CLK4 40 34 CCNc1cccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147385608 CG For-Sale Anodyne DYRK2 47 38 COC(=O)c1cc2cc(NC(=O)N3C[C@H](C)O[C@@H](c4ccccc4)C3)ccc2o1 ZINC000147385633 GI On-Demand Anodyne GYRB 18 40 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccnc2Oc2ccccc2)C1 ZINC000147385688 HG On-Demand Anodyne P2RY1 47 39 CCCCCCCCNC(=O)Cc1ccc(S(N)(=O)=O)s1 ZINC000147385700 EE On-Demand Mild CA2 27 52 CCCCCCCCNC(=O)Cc1ccc(S(N)(=O)=O)s1 ZINC000147385700 EE On-Demand Mild CA5B 44 39 CCCCCCCCNC(=O)Cc1ccc(S(N)(=O)=O)s1 ZINC000147385700 EE On-Demand Mild CA5A 45 35 CCCCCCCCNC(=O)Cc1ccc(S(N)(=O)=O)s1 ZINC000147385700 EE On-Demand Mild NCE103 16 40 CCCCCCCCNC(=O)Cc1ccc(S(N)(=O)=O)s1 ZINC000147385700 EE On-Demand Mild ASAH1 92 37 Cc1cc(OCCc2ccccn2)ccc1S(N)(=O)=O ZINC000147385703 CD For-Sale Anodyne CA7 18 40 COCc1nc(C(=O)N(C)Cc2ccc3cc(OC)ccc3c2)cs1 ZINC000147385705 FH On-Demand Anodyne HSD17B2 26 44 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(C[S@](C)=O)c1 ZINC000147385740 HH On-Demand Anodyne MRGPRX1 41 39 FCOc1ccc(Cl)cc1Cl ZINC000147385768 AG For-Sale Anodyne FABI 15 47 FCOc1ccc(Cl)cc1Cl ZINC000147385768 AG For-Sale Anodyne CBR1 15 47 Cc1cc([N+](=O)[O-])c(OCCN2CCN(C(=O)OC(C)(C)C)CC2)cc1Cl ZINC000147385780 GG For-Sale Anodyne HTR4 18 40 CC(C)CCCCNS(=O)(=O)c1ccc(Cl)c(C(=O)O)c1 ZINC000147385784 EG For-Sale Anodyne TBXA2R 45 37 CC(C)CCCCNS(=O)(=O)c1ccc(Cl)c(C(=O)O)c1 ZINC000147385784 EG For-Sale Anodyne TBXAS1 34 42 CC(C)CCCCNS(=O)(=O)c1ccc(Cl)c(C(=O)O)c1 ZINC000147385784 EG For-Sale Anodyne HTR7 21 40 CC(C)CCCCNS(=O)(=O)c1ccc(Cl)c(C(=O)O)c1 ZINC000147385784 EG For-Sale Anodyne CASP3 25 49 NCCCCNC(=O)COc1ccc2ccc(=O)oc2c1 ZINC000147385799 CD On-Demand Anodyne MAOA 46 47 NCCCCNC(=O)COc1ccc2ccc(=O)oc2c1 ZINC000147385799 CD On-Demand Anodyne MAOB 30 49 NCCCCNC(=O)COc1ccc2ccc(=O)oc2c1 ZINC000147385799 CD On-Demand Anodyne CA7 28 53 NCCCCNC(=O)COc1ccc2ccc(=O)oc2c1 ZINC000147385799 CD On-Demand Anodyne CA12 0 53 NCCCCNC(=O)COc1ccc2ccc(=O)oc2c1 ZINC000147385799 CD On-Demand Anodyne CA9 0 53 CCCNc1nc(Cl)nc(Oc2ccc3c(c2)OCO3)n1 ZINC000147385828 DF For-Sale Anodyne DYRK2 43 38 COC(=O)c1cc2cc(NC(=O)N3C[C@@H](C)O[C@H](c4ccccc4)C3)ccc2o1 ZINC000147385843 GI On-Demand Anodyne GYRB 18 40 COc1ccc(CCCC(=O)NS(=O)(=O)CC2CCCCC2)cc1 ZINC000147385848 FG On-Demand Anodyne BMP1 36 45 COc1ccc(CCCC(=O)NS(=O)(=O)CC2CCCCC2)cc1 ZINC000147385848 FG On-Demand Anodyne MMP2 73 36 COc1ccc(CCCC(=O)NS(=O)(=O)CC2CCCCC2)cc1 ZINC000147385848 FG On-Demand Anodyne MMP3 41 44 COc1ccc(CCCC(=O)NS(=O)(=O)CC2CCCCC2)cc1 ZINC000147385848 FG On-Demand Anodyne MMP8 26 43 COc1ccc(CCCC(=O)NS(=O)(=O)CC2CCCCC2)cc1 ZINC000147385848 FG On-Demand Anodyne MMP9 28 43 COc1ccc(CCCC(=O)NS(=O)(=O)CC2CCCCC2)cc1 ZINC000147385848 FG On-Demand Anodyne MMP1 46 43 NCCCCC(=O)NN1CCCCC1 ZINC000147385905 AC For-Sale Anodyne APHA 40 37 Cc1cc(OCC(=O)NC(C)(C)C)ccc1S(N)(=O)=O ZINC000147385927 DC For-Sale Anodyne HDAC8 0 41 Cc1cccc(OC[C@@H](C)NC(=O)c2ccc3c(c2)COC3)c1 ZINC000147385957 DG On-Demand Anodyne PIN1 20 40 CC[C@H](CNS(=O)(=O)c1ccc(Br)c(C)c1)CC(=O)O ZINC000147385976 FF On-Demand Anodyne LEF 58 40 Cc1cc([N+](=O)[O-])c(OC2CCN(C(=O)OC(C)(C)C)CC2)cc1Cl ZINC000147385984 FI For-Sale Anodyne GPR119 43 42 COC(=O)c1cc2cc(NC(=O)N3C[C@H](C)O[C@H](c4ccccc4)C3)ccc2o1 ZINC000147386048 GI On-Demand Anodyne GYRB 18 40 COc1cccc2ccc(CNCCCCC(C)C)nc12 ZINC000147386079 CI For-Sale Anodyne MCHR1 0 43 CCCCCCCCNC(=O)c1csc(S(N)(=O)=O)c1C ZINC000147386133 EF For-Sale Mild ASAH1 93 36 O=C(O)c1ccc(CNC(=O)[C@H]2C[C@H]2c2ccccc2)o1 ZINC000147386134 CE For-Sale Anodyne GPR88 0 41 CCN(CC)CCOc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147386154 CD For-Sale Anodyne ERG2 17 44 CCN(CC)CCOc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147386154 CD For-Sale Anodyne CA7 16 41 CCN(CC)CCOc1ccc(S(N)(=O)=O)c(C)c1 ZINC000147386154 CD For-Sale Anodyne SQLE 41 31 CC[C@@H](CNS(=O)(=O)c1ccc(Br)c(C)c1)CC(=O)O ZINC000147386187 FF On-Demand Anodyne LEF 58 40 Cc1ccc(C(=O)NNC(=O)NC2CCN(C(=O)c3ccccc3)CC2)s1 ZINC000147386199 GE On-Demand Reactive MAPK11 28 41 Cc1ccc(C(=O)NNC(=O)NC2CCN(C(=O)c3ccccc3)CC2)s1 ZINC000147386199 GE On-Demand Reactive EPHX2 38 54 Cc1ccc(C(=O)NNC(=O)NC2CCN(C(=O)c3ccccc3)CC2)s1 ZINC000147386199 GE On-Demand Reactive CCR8 51 34 Cc1ccc(C(=O)NNC(=O)NC2CCN(C(=O)c3ccccc3)CC2)s1 ZINC000147386199 GE On-Demand Reactive SFRP1 68 42 Cc1ccc(C(=O)NNC(=O)NC2CCN(C(=O)c3ccccc3)CC2)s1 ZINC000147386199 GE On-Demand Reactive L3MBTL3 63 34 COCCn1nc(C(=O)Nc2cccc(CN3CCSCC3)c2C)ccc1=O ZINC000147386278 HD On-Demand Anodyne MRGPRX1 44 39 COc1ccc2nc([C@H](C)Cl)n(CCNC(N)=O)c2c1 ZINC000147386284 CE For-Sale Reactive DRD4 42 32 COc1ccc2nc([C@H](C)Cl)n(CCNC(N)=O)c2c1 ZINC000147386284 CE For-Sale Reactive MTNR1A 37 42 COc1ccc2nc([C@H](C)Cl)n(CCNC(N)=O)c2c1 ZINC000147386284 CE For-Sale Reactive SCD 17 41 COc1ccc2nc([C@H](C)Cl)n(CCNC(N)=O)c2c1 ZINC000147386284 CE For-Sale Reactive PROKR1 65 35 CCCCCCCCNC(=O)c1n[nH]c(C)c1S(N)(=O)=O ZINC000147386303 DD For-Sale Mild ASAH1 63 33 O=C(O)c1ccc(CNC(=O)[C@H]2C[C@@H]2c2ccccc2)o1 ZINC000147386326 CE For-Sale Anodyne GPR88 0 41 C[C@@H](C=O)NCc1ccccc1 ZINC000147386334 AD For-Sale Mild CPA1 28 44 C[C@@H](C=O)NCc1ccccc1 ZINC000147386334 AD For-Sale Mild ACPP 0 43 C[C@@H](C=O)NCc1ccccc1 ZINC000147386334 AD For-Sale Mild SLC1A6 45 29 C[C@@H](C=O)NCc1ccccc1 ZINC000147386334 AD For-Sale Mild CAPN1 43 36 C[C@@H](C=O)NCc1ccccc1 ZINC000147386334 AD For-Sale Mild SLC1A7 45 29 CC[C@H](CNS(=O)(=O)c1ccccc1[N+](=O)[O-])CC(=O)O ZINC000147386377 DD On-Demand Bother COLA 86 41 CC[C@@H]1CN(S(=O)(=O)c2cc(C)ccc2C)CC[C@@H]1N ZINC000147386411 CE On-Demand Anodyne EPHX2 26 42 CN(Cc1cscn1)C(=O)NC1CCN(C(=O)c2ccccc2)CC1 ZINC000147386439 FF On-Demand Anodyne EPHX2 19 44 COC(=O)Cc1csc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)n1 ZINC000147386445 FG On-Demand Anodyne CPT1A 28 41 CCCCCCCCNC(=O)c1csc(S(N)(=O)=O)c1 ZINC000147386479 DE On-Demand Mild CA2 26 67 CCCCCCCCNC(=O)c1csc(S(N)(=O)=O)c1 ZINC000147386479 DE On-Demand Mild KCNQ1 0 41 CCCCCCCCNC(=O)c1csc(S(N)(=O)=O)c1 ZINC000147386479 DE On-Demand Mild ASAH1 76 33 CCCCCCCCNC(=O)c1csc(S(N)(=O)=O)c1 ZINC000147386479 DE On-Demand Mild ACAT 0 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne KLK3 61 37 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne CTSL 22 44 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne TIMP3 40 32 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne HDAC10 43 38 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne MMP2 17 41 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne MMP3 39 44 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne HDAC1 17 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne PCSK5 41 33 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne FURIN 52 36 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne HDAC11 46 38 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne S1PR5 16 44 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne POLG_WNV 62 36 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386488 CD On-Demand Anodyne NPFFR1 40 32 O=C(O)c1ccc(CNC(=O)[C@@H]2C[C@H]2c2ccccc2)o1 ZINC000147386535 CE For-Sale Anodyne GPR88 0 41 COc1ccc2nc([C@@H](C)Cl)n(CCNC(N)=O)c2c1 ZINC000147386543 CE For-Sale Reactive DRD4 42 32 COc1ccc2nc([C@@H](C)Cl)n(CCNC(N)=O)c2c1 ZINC000147386543 CE For-Sale Reactive MTNR1A 37 42 COc1ccc2nc([C@@H](C)Cl)n(CCNC(N)=O)c2c1 ZINC000147386543 CE For-Sale Reactive SCD 17 41 COc1ccc2nc([C@@H](C)Cl)n(CCNC(N)=O)c2c1 ZINC000147386543 CE For-Sale Reactive PROKR1 65 35 CC[C@@H](CNS(=O)(=O)c1ccccc1[N+](=O)[O-])CC(=O)O ZINC000147386584 DD On-Demand Bother COLA 86 41 CC[C@H]1CN(S(=O)(=O)c2cc(C)ccc2C)CC[C@@H]1N ZINC000147386598 CE On-Demand Anodyne EPHX2 26 42 COC(=O)Cc1csc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)n1 ZINC000147386656 FG On-Demand Anodyne CPT1A 28 41 CCCCCCCCNC(=O)c1cc(S(N)(=O)=O)cn1C ZINC000147386673 DD On-Demand Mild ASAH1 86 38 CCc1nc(CN(C)C(=O)NC2CCN(C(=O)c3ccccc3)CC2)cs1 ZINC000147386682 GG On-Demand Anodyne EPHX2 19 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne KLK3 61 37 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne CTSL 22 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne TIMP3 40 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne HDAC10 43 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne MMP2 17 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne MMP3 39 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne HDAC1 17 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne PCSK5 41 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne FURIN 52 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne HDAC11 46 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne S1PR5 16 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne POLG_WNV 62 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(COC)c1 ZINC000147386689 CD On-Demand Anodyne NPFFR1 40 32 CC(=O)Nc1cc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)ccc1C ZINC000147386694 HG On-Demand Anodyne CCR3 34 41 O=c1nc2n(cc1COCc1ccccc1)[C@@H]1O[C@H](CO)[C@@H](O)[C@@H]1O2 ZINC000147386703 EB Annotated Anodyne ADORA1 43 44 O=c1nc2n(cc1COCc1ccccc1)[C@@H]1O[C@H](CO)[C@@H](O)[C@@H]1O2 ZINC000147386703 EB Annotated Anodyne SLC29A1 80 38 O=c1nc2n(cc1COCc1ccccc1)[C@@H]1O[C@H](CO)[C@@H](O)[C@@H]1O2 ZINC000147386703 EB Annotated Anodyne ADORA2A 34 40 O=c1nc2n(cc1COCc1ccccc1)[C@@H]1O[C@H](CO)[C@@H](O)[C@@H]1O2 ZINC000147386703 EB Annotated Anodyne CDA 52 33 O=c1nc2n(cc1COCc1ccccc1)[C@@H]1O[C@H](CO)[C@@H](O)[C@@H]1O2 ZINC000147386703 EB Annotated Anodyne FIMH 73 40 CCC(=O)[C@@H]1Cc2ccccc2O1 ZINC000147386720 AD For-Sale Anodyne TPP2 57 34 Nc1nc(Oc2ccc3c(c2)OCO3)c2ccccc2n1 ZINC000147386729 CF For-Sale Anodyne EDNRA 15 43 Nc1nc(Oc2ccc3c(c2)OCO3)c2ccccc2n1 ZINC000147386729 CF For-Sale Anodyne HSP90AB1 0 45 CC(=O)NCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147386730 CD On-Demand Anodyne CACNA1H 24 41 CC(=O)NCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147386730 CD On-Demand Anodyne HCAR1 0 40 O=C(O)c1ccc(CNC(=O)[C@@H]2C[C@@H]2c2ccccc2)o1 ZINC000147386761 CE For-Sale Anodyne GPR88 0 41 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cnc2sccn2c1=O ZINC000147386764 HF On-Demand Anodyne MRGPRX1 43 38 COC(=O)COc1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147386793 HE On-Demand Anodyne CYP26A1 18 42 COC(=O)Cc1csc(NC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)n1 ZINC000147386861 FG On-Demand Anodyne CPT1A 28 41 CC(=O)Nc1cc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)ccc1C ZINC000147386901 HG On-Demand Anodyne CCR3 34 41 CCC(=O)[C@H]1Cc2ccccc2O1 ZINC000147386939 AD For-Sale Anodyne TPP2 57 34 O=C1CC[C@@H]2C[C@@H](C(=O)O)N[C@H]2C1 ZINC000147386975 AC For-Sale Anodyne CAD 45 36 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cnc2n(c1=O)CCS2 ZINC000147386988 HE On-Demand Anodyne MRGPRX1 44 40 CC[C@@H](C)[C@@H](N)C(=O)NN1CCCCC1 ZINC000147387026 BC For-Sale Anodyne TPP2 41 44 Cc1cc(OCCCC(=O)N(C)C)ccc1S(N)(=O)=O ZINC000147387030 DC For-Sale Anodyne THRA 25 41 Cc1cc(OCCCC(=O)N(C)C)ccc1S(N)(=O)=O ZINC000147387030 DC For-Sale Anodyne P2RY12 0 45 COC(=O)Cc1csc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)n1 ZINC000147387081 FG On-Demand Anodyne CPT1A 28 41 O=C1CC[C@@H]2C[C@H](C(=O)O)N[C@H]2C1 ZINC000147387166 AC For-Sale Anodyne CAD 45 36 O=C(c1cccc2ncccc12)N1CCC[C@@H]1CCCBr ZINC000147387169 EI For-Sale Reactive HCRTR1 30 48 O=C(c1cccc2ncccc12)N1CCC[C@@H]1CCCBr ZINC000147387169 EI For-Sale Reactive PREP 35 43 O=C(c1cccc2ncccc12)N1CCC[C@@H]1CCCBr ZINC000147387169 EI For-Sale Reactive HCRTR2 38 48 O=C(c1cccc2ncccc12)N1CCC[C@@H]1CCCBr ZINC000147387169 EI For-Sale Reactive FAP 0 52 CCNc1nc(C)cc(Oc2ccc3c(c2)OCO3)n1 ZINC000147387184 CF For-Sale Anodyne DYRK2 54 39 CC[C@H](C)[C@@H](N)C(=O)NN1CCCCC1 ZINC000147387213 BC For-Sale Anodyne TPP2 41 44 COC(=O)c1ccccc1CNCC(F)F ZINC000147387249 BD For-Sale Anodyne PHES 0 41 O=C1CCc2cc(S(=O)(=O)NCc3ccc(-n4ccnc4)c(F)c3)c(F)cc2N1 ZINC000147387254 HF On-Demand Anodyne PKM 43 47 CC(C)CCCCNCc1cnccn1 ZINC000147387255 BE For-Sale Anodyne FDFT1 0 45 C/C(C(=O)O)=C(/C)c1ccc2ccccc2c1 ZINC000147387281 BH For-Sale Anodyne CYP2A5 0 43 c1cnc2oc(NC3CCNCC3)nc2c1 ZINC000147387315 BD For-Sale Anodyne SSTR5 33 49 O=C(c1cccc2ncccc12)N1CCC[C@H]1CCCBr ZINC000147387376 EI For-Sale Reactive HCRTR1 30 48 O=C(c1cccc2ncccc12)N1CCC[C@H]1CCCBr ZINC000147387376 EI For-Sale Reactive PREP 35 43 O=C(c1cccc2ncccc12)N1CCC[C@H]1CCCBr ZINC000147387376 EI For-Sale Reactive HCRTR2 38 48 O=C(c1cccc2ncccc12)N1CCC[C@H]1CCCBr ZINC000147387376 EI For-Sale Reactive FAP 0 52 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(-n2cncn2)cc1 ZINC000147387430 GG On-Demand Anodyne MRGPRX1 48 45 Cc1ccc(F)c(C2=CCNCC2)c1F ZINC000147387440 BF For-Sale Anodyne QDPR 0 43 CC[C@H](NC(=O)C[C@@H](C)[C@@H]1CCCNC1)C(=O)O ZINC000147387463 CC For-Sale Anodyne CPN1 0 48 CN(C)C(=O)c1cccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)c1 ZINC000147387468 HE On-Demand Anodyne NOS2 72 33 Cc1cc(OC[C@@H]2CN(C)CCO2)ccc1S(N)(=O)=O ZINC000147387486 DC For-Sale Anodyne CHRNA10 48 32 CCNc1nc(Cl)nc(Oc2ccc3c(c2)OCO3)n1 ZINC000147387651 CE For-Sale Anodyne DYRK2 43 37 CCNc1nc(Cl)nc(Oc2ccc3c(c2)OCO3)n1 ZINC000147387651 CE For-Sale Anodyne PPX1 0 42 CC[C@H](NC(=O)C[C@H](C)[C@@H]1CCCNC1)C(=O)O ZINC000147387699 CC For-Sale Anodyne CPN1 0 48 Cc1cc(OC[C@H]2CN(C)CCO2)ccc1S(N)(=O)=O ZINC000147387709 DC For-Sale Anodyne CHRNA10 48 32 Cc1nc(-n2cc(-c3ccccc3)cn2)ccc1C(=O)O ZINC000147387746 CF For-Sale Anodyne EGLN1 0 42 CC[C@@H]1CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CCO1 ZINC000147387783 DF On-Demand Anodyne CACNA1I 41 32 COc1ccc(Nc2nc(-c3ccc4cnn(C)c4c3)cn3ccnc23)cc1OC ZINC000147387785 HI For-Sale Anodyne EPHB4 39 41 CCCC1CCC(CCc2cccc(F)c2)CC1 ZINC000147387794 BK For-Sale Anodyne SLC18A2 36 46 O=C(c1cc(F)ccc1[N+](=O)[O-])N1CCC[C@@H]1CCCBr ZINC000147387853 FH For-Sale Reactive HCRTR1 15 42 Cc1c(CN2CCSCC2)cccc1NC(=O)Cn1ccc(=O)[nH]c1=O ZINC000147387891 FD On-Demand Anodyne Q8II92_PLAF7 40 32 COc1ccc2c(c1)OC[C@H](C(=O)NCCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147387938 FF On-Demand Bother MTNR1A 71 41 COc1ccc2c(c1)OC[C@H](C(=O)NCCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147387938 FF On-Demand Bother MTNR1B 60 38 COc1ccc2c(c1)OC[C@H](C(=O)NCCc1ccc([N+](=O)[O-])cc1)C2 ZINC000147387938 FF On-Demand Bother ROCK2 28 41 CC[C@H](NC(=O)C[C@@H](C)[C@H]1CCCNC1)C(=O)O ZINC000147387963 CC For-Sale Anodyne CPN1 0 48 CCCCCCCCNS(=O)(=O)c1cccc(CO)c1 ZINC000147387975 CF For-Sale Mild TBXA2R 19 47 CCCCCCCCNS(=O)(=O)c1cccc(CO)c1 ZINC000147387975 CF For-Sale Mild FBP1 31 42 CCCCCCCCNS(=O)(=O)c1cccc(CO)c1 ZINC000147387975 CF For-Sale Mild ALOX15 53 44 CC[C@H]1CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CCO1 ZINC000147388007 DF On-Demand Anodyne CACNA1I 41 32 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(c2cnccn2)CC1 ZINC000147388028 DC On-Demand Anodyne P2RY12 177 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(c2cnccn2)CC1 ZINC000147388028 DC On-Demand Anodyne TGM2 18 42 Cc1ccc(SCc2cn3c(nc2=O)O[C@H]2[C@H](O)[C@@H](CO)O[C@H]23)cc1 ZINC000147388056 FC Annotated Anodyne SLC29A1 93 44 Cc1ccc(SCc2cn3c(nc2=O)O[C@H]2[C@H](O)[C@@H](CO)O[C@H]23)cc1 ZINC000147388056 FC Annotated Anodyne TK1 27 41 Cc1ccc(SCc2cn3c(nc2=O)O[C@H]2[C@H](O)[C@@H](CO)O[C@H]23)cc1 ZINC000147388056 FC Annotated Anodyne CDA 56 34 Cc1ccc(SCc2cn3c(nc2=O)O[C@H]2[C@H](O)[C@@H](CO)O[C@H]23)cc1 ZINC000147388056 FC Annotated Anodyne AK 0 43 Cc1ccc(SCc2cn3c(nc2=O)O[C@H]2[C@H](O)[C@@H](CO)O[C@H]23)cc1 ZINC000147388056 FC Annotated Anodyne FIMH 19 40 O=C(c1cc(F)ccc1[N+](=O)[O-])N1CCC[C@H]1CCCBr ZINC000147388076 FH For-Sale Reactive HCRTR1 15 42 CC[C@H](NC(=O)C[C@H](C)[C@H]1CCCNC1)C(=O)O ZINC000147388162 CC For-Sale Anodyne CPN1 0 48 CCNC(=O)CNC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147388225 ED For-Sale Anodyne F7 21 41 CCCCCCCCNS(=O)(=O)c1cc(CO)ccc1C ZINC000147388232 DG For-Sale Mild S1PR2 41 35 CC(C)(C)c1ccc(CCC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)cc1 ZINC000147388277 HJ On-Demand Anodyne TRPV1 33 49 CC(C)(C)c1ccc(CCC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)cc1 ZINC000147388277 HJ On-Demand Anodyne MLYCD 20 45 CC(C)(C)c1ccc(CCC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)cc1 ZINC000147388277 HJ On-Demand Anodyne L3MBTL3 54 37 CC(C)(C)c1ccc(CCC(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)cc1 ZINC000147388277 HJ On-Demand Anodyne HPGD 30 43 O=C(CCCc1ccccc1)N1CCC[C@@H]1CCCBr ZINC000147388301 EI For-Sale Reactive FKBP1A 59 47 O=C(CCCc1ccccc1)N1CCC[C@@H]1CCCBr ZINC000147388301 EI For-Sale Reactive SLC18A2 48 46 O=C(CCCc1ccccc1)N1CCC[C@@H]1CCCBr ZINC000147388301 EI For-Sale Reactive SIGMAR1 16 40 O=C(CCCc1ccccc1)N1CCC[C@@H]1CCCBr ZINC000147388301 EI For-Sale Reactive DPP4 20 47 O=C(CCCc1ccccc1)N1CCC[C@@H]1CCCBr ZINC000147388301 EI For-Sale Reactive PREP 111 59 O=C(CCCc1ccccc1)N1CCC[C@@H]1CCCBr ZINC000147388301 EI For-Sale Reactive FKBP12.6 0 43 O=C(CCCc1ccccc1)N1CCC[C@@H]1CCCBr ZINC000147388301 EI For-Sale Reactive FAP 0 44 O=C(O)C1(n2nnnc2CCCc2ccccc2)CCC1 ZINC000147388324 CD For-Sale Anodyne FAAH 24 51 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147388325 HE On-Demand Anodyne GHRHR 41 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147388325 HE On-Demand Anodyne P2RY12 179 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147388325 HE On-Demand Anodyne TRY2_BOVIN 52 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147388325 HE On-Demand Anodyne EPHX2 17 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147388325 HE On-Demand Anodyne MLYCD 18 41 CC(=O)Nc1cc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)ccc1C ZINC000147388349 HJ On-Demand Anodyne ROCK2 29 48 CC(=O)Nc1cc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)ccc1C ZINC000147388349 HJ On-Demand Anodyne MET 42 44 CC(=O)Nc1cc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)ccc1C ZINC000147388349 HJ On-Demand Anodyne NAMPT 51 46 CC[C@H](NC(=O)[C@@H]1CCNc2ccccc21)C(=O)O ZINC000147388361 CD For-Sale Anodyne ACE2 69 33 CCOC(=O)c1cnn(-c2ccc(C(=O)O)c(C)n2)c1 ZINC000147388378 CD For-Sale Anodyne EGLN1 0 44 C#Cc1nc(C)c(C(=O)NCc2ccccc2)s1 ZINC000147388387 CE For-Sale Anodyne CHRM4 37 52 C#Cc1nc(C)c(C(=O)NCc2ccccc2)s1 ZINC000147388387 CE For-Sale Anodyne SCD1 55 60 C#Cc1nc(C)c(C(=O)NCc2ccccc2)s1 ZINC000147388387 CE For-Sale Anodyne SCD 50 58 C#Cc1nc(C)c(C(=O)NCc2ccccc2)s1 ZINC000147388387 CE For-Sale Anodyne NAMPT 40 38 CCCCCCCCNS(=O)(=O)c1[nH]ncc1CO ZINC000147388418 CD For-Sale Mild ALOX15 28 41 CCCCCCCCNS(=O)(=O)c1[nH]ncc1CO ZINC000147388418 CD For-Sale Mild ASAH1 44 38 CCNC(=O)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147388437 CD On-Demand Anodyne CACNA1I 41 35 O=C(CCCc1ccccc1)N1CCC[C@H]1CCCBr ZINC000147388459 EI For-Sale Reactive FKBP1A 59 47 O=C(CCCc1ccccc1)N1CCC[C@H]1CCCBr ZINC000147388459 EI For-Sale Reactive SLC18A2 48 46 O=C(CCCc1ccccc1)N1CCC[C@H]1CCCBr ZINC000147388459 EI For-Sale Reactive SIGMAR1 16 40 O=C(CCCc1ccccc1)N1CCC[C@H]1CCCBr ZINC000147388459 EI For-Sale Reactive DPP4 20 47 O=C(CCCc1ccccc1)N1CCC[C@H]1CCCBr ZINC000147388459 EI For-Sale Reactive PREP 111 59 O=C(CCCc1ccccc1)N1CCC[C@H]1CCCBr ZINC000147388459 EI For-Sale Reactive FKBP12.6 0 43 O=C(CCCc1ccccc1)N1CCC[C@H]1CCCBr ZINC000147388459 EI For-Sale Reactive FAP 0 44 CC[C@H](NC(=O)[C@H]1CCNc2ccccc21)C(=O)O ZINC000147388540 CD For-Sale Anodyne ACE2 69 33 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cc(-c2ccccc2)n[nH]1 ZINC000147388558 GI On-Demand Anodyne HTR2C 15 43 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cc(-c2ccccc2)n[nH]1 ZINC000147388558 GI On-Demand Anodyne TACR3 16 44 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cc(-c2ccccc2)n[nH]1 ZINC000147388558 GI On-Demand Anodyne FLT3 22 40 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cc(-c2ccccc2)n[nH]1 ZINC000147388558 GI On-Demand Anodyne MRGPRX1 46 49 CCC[C@@H](NC(N)=O)C(=O)Nc1ncc(Cc2cccc(CC)c2)s1 ZINC000147388591 FG On-Demand Anodyne SCD1 37 41 CCC[C@@H](NC(N)=O)C(=O)Nc1ncc(Cc2cccc(CC)c2)s1 ZINC000147388591 FG On-Demand Anodyne SCD 31 41 CCCCC1CCC(NC(=O)Nc2ccc(C)c(NC(C)=O)c2)CC1 ZINC000147388646 EJ On-Demand Anodyne EPHX2 49 47 COc1cccc(OC)c1Oc1ccc(C(=O)O)c(C)n1 ZINC000147388656 CF For-Sale Anodyne ALS 95 46 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(CC)cc2)CC1 ZINC000147388767 FD On-Demand Anodyne GHRHR 42 34 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(CC)cc2)CC1 ZINC000147388767 FD On-Demand Anodyne P2RY12 181 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(CC)cc2)CC1 ZINC000147388767 FD On-Demand Anodyne TRY2_BOVIN 76 37 CC(=O)c1c[nH]c(C(=O)Nc2cccc(CN3CCSCC3)c2C)c1 ZINC000147388792 FG On-Demand Anodyne MRGPRX1 32 41 Cc1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)cc1C(F)(F)F ZINC000147388798 GH On-Demand Anodyne EPHX2 15 42 Cc1c(-c2csc(-c3cnccc3C(F)(F)F)n2)sc2ccc(Cl)cc12 ZINC000147388831 HK Annotated Anodyne ROCK1 22 46 COCCCOc1ccccc1NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147388860 FG On-Demand Anodyne ROCK2 42 51 CC[C@@H]1CN(S(=O)(=O)c2cc(F)ccc2F)CC[C@@H]1N ZINC000147388862 DD On-Demand Anodyne DPP4 15 44 CC(=O)Nc1cc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)ccc1C ZINC000147388869 GI On-Demand Anodyne LDLR 0 45 Cc1nc(Oc2ccccc2C(F)(F)F)ccc1C(=O)O ZINC000147388888 CH For-Sale Anodyne RBP4 76 43 Cc1nc(Oc2ccccc2C(F)(F)F)ccc1C(=O)O ZINC000147388888 CH For-Sale Anodyne ALS 41 45 O=C(c1cc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)c[nH]1)N1CCCC1 ZINC000147388897 HE On-Demand Anodyne NOS2 40 30 Cc1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)cc1C(F)(F)F ZINC000147388985 GH On-Demand Anodyne EPHX2 15 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(CC)cc2)CC1 ZINC000147388995 FD On-Demand Anodyne GHRHR 42 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(CC)cc2)CC1 ZINC000147388995 FD On-Demand Anodyne P2RY12 181 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(CC)cc2)CC1 ZINC000147388995 FD On-Demand Anodyne TRY2_BOVIN 76 37 CC(C)NC(=O)CNC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147389021 FD For-Sale Anodyne F7 30 47 CC[C@H](CNS(=O)(=O)c1ccccc1Cl)CC(=O)O ZINC000147389032 DE On-Demand Anodyne ITGAV 33 45 CCNc1ncc(F)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147389052 CF For-Sale Anodyne CLK4 44 38 BrCCN(c1ccnc2ccccc12)C1CCCCC1 ZINC000147389056 EJ For-Sale Reactive HNMT 40 44 CCN(CC)C(=O)[C@@H]1CCCN(S(=O)(=O)c2ccccc2C#N)C1 ZINC000147389069 ED Annotated Mild AKR1C3 19 40 CC(=O)Nc1cc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)ccc1C ZINC000147389070 GI On-Demand Anodyne LDLR 0 45 CC[C@H]1CN(S(=O)(=O)c2cc(F)ccc2F)CC[C@@H]1N ZINC000147389073 DD On-Demand Anodyne DPP4 15 44 Cc1cc(Cl)cc(C)c1Oc1ccc(C(=O)O)c(C)n1 ZINC000147389151 CI For-Sale Anodyne PRS 46 42 CCc1ncc(C(=O)N(C)Cc2ccc3cc(OC)ccc3c2)s1 ZINC000147389195 EI On-Demand Anodyne HSD17B2 38 50 CN1CCC[C@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389229 CD On-Demand Anodyne CHRM2 18 43 CN1CCC[C@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389229 CD On-Demand Anodyne DRD2 30 41 CN1CCC[C@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389229 CD On-Demand Anodyne DRD4 56 42 CN1CCC[C@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389229 CD On-Demand Anodyne ACHE 40 42 CN1CCC[C@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389229 CD On-Demand Anodyne SLC6A4 19 44 CN1CCC[C@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389229 CD On-Demand Anodyne DRD3 28 43 CN1CCC[C@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389229 CD On-Demand Anodyne HRH3 28 45 CN1CCC[C@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389229 CD On-Demand Anodyne SIGMAR1 99 51 CN1CCC[C@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389229 CD On-Demand Anodyne SLC18A3 25 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(F)c(F)c2)CC1 ZINC000147389246 GD On-Demand Anodyne P2RY12 190 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(F)c(F)c2)CC1 ZINC000147389246 GD On-Demand Anodyne TRY2_BOVIN 67 37 CC(=O)Nc1cc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)ccc1C ZINC000147389253 GI On-Demand Anodyne LDLR 0 45 CC[C@@H](CNS(=O)(=O)c1ccccc1Cl)CC(=O)O ZINC000147389256 DE On-Demand Anodyne ITGAV 33 45 CC(C)NC(=O)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147389261 DD On-Demand Anodyne CCKBR 45 36 CC(C)NC(=O)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147389261 DD On-Demand Anodyne F7 30 42 CC(C)NC(=O)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147389261 DD On-Demand Anodyne CACNA1I 42 35 CC(=O)Nc1cccc(-c2cnc3ccc(NCc4ccc(F)cc4)nn23)c1 ZINC000147389263 GI Annotated Anodyne IKBKB 31 46 CC(=O)Nc1cccc(-c2cnc3ccc(NCc4ccc(F)cc4)nn23)c1 ZINC000147389263 GI Annotated Anodyne HDAC10 18 42 CC(=O)Nc1cccc(-c2cnc3ccc(NCc4ccc(F)cc4)nn23)c1 ZINC000147389263 GI Annotated Anodyne HDAC3 20 42 CC(=O)Nc1cccc(-c2cnc3ccc(NCc4ccc(F)cc4)nn23)c1 ZINC000147389263 GI Annotated Anodyne HDAC6 15 42 CC(=O)Nc1cccc(-c2cnc3ccc(NCc4ccc(F)cc4)nn23)c1 ZINC000147389263 GI Annotated Anodyne BRAF 47 38 CC[C@H](NC(=O)c1cc(N)cc(Cl)c1)C(=O)O ZINC000147389267 CD For-Sale Anodyne CA2 22 43 CC[C@H](NC(=O)c1cc(N)cc(Cl)c1)C(=O)O ZINC000147389267 CD For-Sale Anodyne CCKAR 0 44 CC[C@H](NC(=O)c1cc(N)cc(Cl)c1)C(=O)O ZINC000147389267 CD For-Sale Anodyne CCKBR 23 41 CC(C)CCCCNCc1c(O)ccc2ccccc12 ZINC000147389268 CI For-Sale Clean METG 40 34 CC(C)CCCCNCc1c(O)ccc2ccccc12 ZINC000147389268 CI For-Sale Clean LMGT2 0 55 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cnn(Cc2ccccc2)c1 ZINC000147389283 HI On-Demand Anodyne ACHE 20 41 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cnn(Cc2ccccc2)c1 ZINC000147389283 HI On-Demand Anodyne SIGMAR1 20 41 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cnn(Cc2ccccc2)c1 ZINC000147389283 HI On-Demand Anodyne MRGPRX1 49 47 CCN(CC)C(=O)[C@H]1CCCN(S(=O)(=O)c2ccccc2C#N)C1 ZINC000147389293 ED Annotated Mild AKR1C3 19 40 Cc1nc(Oc2ccccc2C(C)(C)C)ccc1C(=O)O ZINC000147389388 CI For-Sale Anodyne P2RY1 34 41 Cc1nc(Oc2ccccc2C(C)(C)C)ccc1C(=O)O ZINC000147389388 CI For-Sale Anodyne ALS 57 41 CC(=O)Nc1cc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)ccc1C ZINC000147389441 GI On-Demand Anodyne LDLR 0 45 CC[C@H](CNS(=O)(=O)c1ccc(C)c(C)c1)CC(=O)O ZINC000147389446 CE On-Demand Anodyne LEF 58 40 CC[C@@H]1CN(S(=O)(=O)c2cccs2)CC[C@@H]1N ZINC000147389453 CD On-Demand Anodyne GCKR 41 42 CN1CCC[C@@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389457 CD On-Demand Anodyne CHRM2 18 43 CN1CCC[C@@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389457 CD On-Demand Anodyne DRD2 30 41 CN1CCC[C@@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389457 CD On-Demand Anodyne DRD4 56 42 CN1CCC[C@@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389457 CD On-Demand Anodyne ACHE 40 42 CN1CCC[C@@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389457 CD On-Demand Anodyne SLC6A4 19 44 CN1CCC[C@@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389457 CD On-Demand Anodyne DRD3 28 43 CN1CCC[C@@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389457 CD On-Demand Anodyne HRH3 28 45 CN1CCC[C@@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389457 CD On-Demand Anodyne SIGMAR1 99 51 CN1CCC[C@@H](N2CCN(Cc3ccccc3)CC2)C1 ZINC000147389457 CD On-Demand Anodyne SLC18A3 25 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(F)c(F)c2)CC1 ZINC000147389461 GD On-Demand Anodyne P2RY12 190 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccc(F)c(F)c2)CC1 ZINC000147389461 GD On-Demand Anodyne TRY2_BOVIN 67 37 CCc1c(NC)ncnc1Oc1ccc2c(c1)OCO2 ZINC000147389498 CF For-Sale Anodyne DYRK1A 44 39 CCc1c(NC)ncnc1Oc1ccc2c(c1)OCO2 ZINC000147389498 CF For-Sale Anodyne CLK1 46 39 CCc1c(NC)ncnc1Oc1ccc2c(c1)OCO2 ZINC000147389498 CF For-Sale Anodyne CLK2 49 39 CCc1c(NC)ncnc1Oc1ccc2c(c1)OCO2 ZINC000147389498 CF For-Sale Anodyne CLK4 67 39 CC(C)CCCCN[C@@H](C)c1cccc2ccccc12 ZINC000147389514 CK For-Sale Anodyne CACNA2D1 0 43 C[C@]1(C(=O)N(CC(=O)O)Cc2ccc(Cl)cc2)CCN1C(=O)Cc1coc2ccccc12 ZINC000147389576 JH Annotated Anodyne FFAR2 157 72 CCOc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147389595 CG For-Sale Anodyne CACNA2D1 40 35 CC(C)[C@H]1CC[C@@H](C)C[C@H]1NCC(F)F ZINC000147389613 BG On-Demand Anodyne TRPM8 15 40 CC[C@H]1CN(S(=O)(=O)c2cccs2)CC[C@@H]1N ZINC000147389645 CD On-Demand Anodyne GCKR 24 41 CC[C@@H](CNS(=O)(=O)c1ccc(C)c(C)c1)CC(=O)O ZINC000147389649 CE On-Demand Anodyne LEF 58 40 Cc1cc(OCCN2CCCCC2)cc(C)c1S(N)(=O)=O ZINC000147389667 DD For-Sale Anodyne ESR1 75 39 Cc1cc(OCCN2CCCCC2)cc(C)c1S(N)(=O)=O ZINC000147389667 DD For-Sale Anodyne ESR2 54 39 Cc1cc(OCCN2CCCCC2)cc(C)c1S(N)(=O)=O ZINC000147389667 DD For-Sale Anodyne LTA4H 45 43 Cc1cc(OCCN2CCCCC2)cc(C)c1S(N)(=O)=O ZINC000147389667 DD For-Sale Anodyne HRH3 61 52 Cc1cc(OCCN2CCCCC2)cc(C)c1S(N)(=O)=O ZINC000147389667 DD For-Sale Anodyne PSMB2 46 45 Cc1cc(OCCN2CCCCC2)cc(C)c1S(N)(=O)=O ZINC000147389667 DD For-Sale Anodyne PSMB1 51 46 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2cc(OC)cc(OC)c2)CC1 ZINC000147389682 HD On-Demand Anodyne P2RY12 194 45 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2cc(OC)cc(OC)c2)CC1 ZINC000147389682 HD On-Demand Anodyne TRY2_BOVIN 72 35 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2cc(OC)cc(OC)c2)CC1 ZINC000147389682 HD On-Demand Anodyne CCKAR 15 40 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2cc(OC)cc(OC)c2)CC1 ZINC000147389682 HD On-Demand Anodyne CCKBR 23 40 O=C(CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1)NC1CC1 ZINC000147389708 DD On-Demand Anodyne EPHX2 27 49 O=C(CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1)NC1CC1 ZINC000147389708 DD On-Demand Anodyne CACNA1I 55 36 Nc1nc2ccccc2n1-c1ccc(Cl)cc1Br ZINC000147389727 DI For-Sale Anodyne Q581W1_TRYB2 0 41 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(NC(N)=O)c1 ZINC000147389729 GG On-Demand Anodyne CCR3 23 43 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(NC(N)=O)c1 ZINC000147389729 GG On-Demand Anodyne MRGPRX1 43 40 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(NC(N)=O)c1 ZINC000147389729 GG On-Demand Anodyne KCNK3 86 38 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cccc(NC(N)=O)c1 ZINC000147389729 GG On-Demand Anodyne KCNK9 47 38 CC(C)CCCCN[C@H](C)c1cccc2ccccc12 ZINC000147389742 CK For-Sale Anodyne CACNA2D1 0 43 CCCCCCCCNS(=O)(=O)c1cc(CO)n(CC)c1 ZINC000147389749 DF For-Sale Mild ASAH1 70 33 CNc1ncnc(Oc2ccc3c(c2)OCO3)c1C(C)C ZINC000147389751 CG For-Sale Anodyne CLK4 45 35 C[C@@]1(C(=O)N(CC(=O)O)Cc2ccc(Cl)cc2)CCN1C(=O)Cc1coc2ccccc12 ZINC000147389802 JH Annotated Anodyne FFAR2 157 72 Cc1nn(-c2ccccc2)c(C)c1NC(=O)[C@@H](C)Cc1cccc(F)c1 ZINC000147389813 FI On-Demand Anodyne P2RX7 28 55 Cc1nn(-c2ccccc2)c(C)c1NC(=O)[C@@H](C)Cc1cccc(F)c1 ZINC000147389813 FI On-Demand Anodyne CARM1 51 37 COc1cc(C#N)ccc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147389863 CF For-Sale Mild ALS 40 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2cc(OC)cc(OC)c2)CC1 ZINC000147389871 HD On-Demand Anodyne P2RY12 194 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2cc(OC)cc(OC)c2)CC1 ZINC000147389871 HD On-Demand Anodyne TRY2_BOVIN 72 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2cc(OC)cc(OC)c2)CC1 ZINC000147389871 HD On-Demand Anodyne CCKAR 15 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2cc(OC)cc(OC)c2)CC1 ZINC000147389871 HD On-Demand Anodyne CCKBR 23 40 CC(C)CNCc1cnccc1Oc1ccc(Cl)c(F)c1 ZINC000147389879 DI For-Sale Anodyne SLC6A4 15 50 CCOC[C@H](C)NC(=O)Nc1cc(NC(=O)c2ccccc2)ccc1C ZINC000147389911 FH On-Demand Anodyne MAPK14 24 48 CCOC[C@H](C)NC(=O)Nc1cc(NC(=O)c2ccccc2)ccc1C ZINC000147389911 FH On-Demand Anodyne PYGL 21 41 CCOC[C@H](C)NC(=O)Nc1cc(NC(=O)c2ccccc2)ccc1C ZINC000147389911 FH On-Demand Anodyne PRNP 50 37 CCOC[C@H](C)NC(=O)Nc1cc(NC(=O)c2ccccc2)ccc1C ZINC000147389911 FH On-Demand Anodyne SMO 24 43 CCOC[C@H](C)NC(=O)Nc1cc(NC(=O)c2ccccc2)ccc1C ZINC000147389911 FH On-Demand Anodyne KCNK3 87 41 CCOC[C@H](C)NC(=O)Nc1cc(NC(=O)c2ccccc2)ccc1C ZINC000147389911 FH On-Demand Anodyne KCNK9 69 40 CCCCCCCCNS(=O)(=O)c1cccc(CO)c1C ZINC000147390003 DG For-Sale Mild ALOX15 24 41 Cc1nn(-c2ccccc2)c(C)c1NC(=O)[C@H](C)Cc1cccc(F)c1 ZINC000147390006 FI On-Demand Anodyne P2RX7 28 55 Cc1nn(-c2ccccc2)c(C)c1NC(=O)[C@H](C)Cc1cccc(F)c1 ZINC000147390006 FI On-Demand Anodyne CARM1 51 37 CC(C)[C@@H]1CC[C@@H](C)C[C@H]1NCC(F)F ZINC000147390016 BG On-Demand Anodyne TRPM8 15 40 O=C(c1ccc2c(c1)COC2)N(Cc1ccccc1)C[C@H]1CCCO1 ZINC000147390068 EH On-Demand Anodyne OXTR 38 67 O=C(c1ccc2c(c1)COC2)N(Cc1ccccc1)C[C@H]1CCCO1 ZINC000147390068 EH On-Demand Anodyne AVPR1A 26 67 CCCC[C@H](NC(N)=O)C(=O)N1CCc2[nH]c3ccc(F)cc3c2C1 ZINC000147390082 EE On-Demand Anodyne P2RY12 47 33 Cc1nc(Oc2ccc(C(C)C)cc2)ccc1C(=O)O ZINC000147390095 CI For-Sale Anodyne ACACA 42 36 O=C(O)c1csc(Nc2c(Cl)cccc2Cl)n1 ZINC000147390118 CH For-Sale Anodyne PTGER1 42 49 O=C(O)c1csc(Nc2c(Cl)cccc2Cl)n1 ZINC000147390118 CH For-Sale Anodyne CXCL8 45 42 O=C(O)c1csc(Nc2c(Cl)cccc2Cl)n1 ZINC000147390118 CH For-Sale Anodyne TRPC6 71 41 O=C(O)c1csc(Nc2c(Cl)cccc2Cl)n1 ZINC000147390118 CH For-Sale Anodyne TRPC3 52 41 Cc1cnc(N)nc1Oc1ccc2c(c1)OCO2 ZINC000147390185 BD For-Sale Anodyne FOLA 21 46 CCCCCCCCNS(=O)(=O)CCCCO ZINC000147390215 CE For-Sale Mild RELA 27 61 NC(=O)[C@@H](NO)c1ccccc1 ZINC000147390229 AC For-Sale Anodyne CSNK1G1 19 45 NC(=O)[C@@H](NO)c1ccccc1 ZINC000147390229 AC For-Sale Anodyne KYNU 40 29 CCCC[C@@H](NC(N)=O)C(=O)N1CCc2[nH]c3ccc(F)cc3c2C1 ZINC000147390249 EE On-Demand Anodyne P2RY12 47 33 CS(=O)(=O)c1cc(C(=O)NCC(=O)Nc2ccccc2)cc([N+](=O)[O-])c1 ZINC000147390291 GD On-Demand Bother CA2 40 42 COc1ccc2c(c1)nc(CCCl)n2CCNC(N)=O ZINC000147390400 CD For-Sale Reactive DRD4 40 31 COc1ccc2c(c1)nc(CCCl)n2CCNC(N)=O ZINC000147390400 CD For-Sale Reactive NQO2 33 41 COc1ccc2c(c1)nc(CCCl)n2CCNC(N)=O ZINC000147390400 CD For-Sale Reactive MTNR1A 64 45 COc1ccc2c(c1)nc(CCCl)n2CCNC(N)=O ZINC000147390400 CD For-Sale Reactive MTNR1B 51 41 COc1ccc2c(c1)nc(CCCl)n2CCNC(N)=O ZINC000147390400 CD For-Sale Reactive PROKR1 63 35 C#CCOc1ccccc1CNCC(F)F ZINC000147390450 BE On-Demand Mild PHES 0 43 CCCCCCCCNS(=O)(=O)c1ccc(F)c(CO)c1 ZINC000147390485 DF For-Sale Mild ALOX15 53 45 CCCCCCCCNS(=O)(=O)c1ccc(F)c(CO)c1 ZINC000147390485 DF For-Sale Mild LEF 51 40 CCCCCCCCNS(=O)(=O)c1ccc(F)c(CO)c1 ZINC000147390485 DF For-Sale Mild ASAH1 51 31 CCOC[C@H](C)NC(=O)Nc1cc(C(=O)NCC(F)(F)F)ccc1C ZINC000147390505 FF On-Demand Anodyne MAPK14 26 40 Nc1ccc(C(=O)O)cc1Nc1ccccc1 ZINC000147390511 BF For-Sale Anodyne SRD5A2 34 40 Nc1ccc(C(=O)O)cc1Nc1ccccc1 ZINC000147390511 BF For-Sale Anodyne HDAC1 29 43 Nc1ccc(C(=O)O)cc1Nc1ccccc1 ZINC000147390511 BF For-Sale Anodyne HDAC2 24 40 Nc1ccc(C(=O)O)cc1Nc1ccccc1 ZINC000147390511 BF For-Sale Anodyne HDAC3 0 42 Nc1ccc(C(=O)O)cc1Nc1ccccc1 ZINC000147390511 BF For-Sale Anodyne NEU3 0 40 Nc1ccc(C(=O)O)cc1Nc1ccccc1 ZINC000147390511 BF For-Sale Anodyne AKR1C3 74 56 Nc1ccc(C(=O)O)cc1Nc1ccccc1 ZINC000147390511 BF For-Sale Anodyne AKR1C4 0 42 Nc1ccc(C(=O)O)cc1Nc1ccccc1 ZINC000147390511 BF For-Sale Anodyne AKR1C2 93 49 Nc1ccc(C(=O)O)cc1Nc1ccccc1 ZINC000147390511 BF For-Sale Anodyne MBTD1 0 41 Nc1ccc(C(=O)O)cc1Nc1ccccc1 ZINC000147390511 BF For-Sale Anodyne TRPM4 0 40 Nc1ccc(C(=O)O)cc1Nc1ccccc1 ZINC000147390511 BF For-Sale Anodyne KCNK3 43 35 COc1ccc2c(c1)nc([C@H](C)Cl)n2CCNC(N)=O ZINC000147390597 CE For-Sale Reactive DRD4 40 30 COc1ccc2c(c1)nc([C@H](C)Cl)n2CCNC(N)=O ZINC000147390597 CE For-Sale Reactive MTNR1A 43 42 COc1ccc2c(c1)nc([C@H](C)Cl)n2CCNC(N)=O ZINC000147390597 CE For-Sale Reactive MTNR1B 33 40 COc1ccc2c(c1)nc([C@H](C)Cl)n2CCNC(N)=O ZINC000147390597 CE For-Sale Reactive PROKR1 65 35 Cc1nc(Oc2cccc(C(C)C)c2)ccc1C(=O)O ZINC000147390636 CI For-Sale Anodyne TRY1_BOVIN 25 43 Cc1nc(Oc2cccc(C(C)C)c2)ccc1C(=O)O ZINC000147390636 CI For-Sale Anodyne ALS 67 32 CNS(=O)(=O)c1ccc(C(=O)Nc2cccc(CN3CCSCC3)c2C)cc1 ZINC000147390683 HF On-Demand Anodyne MRGPRX1 45 42 FC(F)CN[C@H]1CCCCc2ccccc21 ZINC000147390700 BG For-Sale Anodyne KCNN3 15 44 CC[C@@H]1CN(S(=O)(=O)c2ccccc2C)CC[C@@H]1N ZINC000147390716 CD On-Demand Anodyne EPHX2 21 45 COc1ccc(Nc2nc(-c3ccc4[nH]ccc4c3)cn3ccnc23)cc1OC ZINC000147390743 GJ For-Sale Anodyne PRKCQ 16 41 COc1ccc(Nc2nc(-c3ccc4[nH]ccc4c3)cn3ccnc23)cc1OC ZINC000147390743 GJ For-Sale Anodyne EPHB4 27 41 COc1ccc(Nc2nc(-c3ccc4[nH]ccc4c3)cn3ccnc23)cc1OC ZINC000147390743 GJ For-Sale Anodyne ENPP1 51 32 COc1ccc2c(c1)nc([C@@H](C)Cl)n2CCNC(N)=O ZINC000147390808 CE For-Sale Reactive DRD4 40 30 COc1ccc2c(c1)nc([C@@H](C)Cl)n2CCNC(N)=O ZINC000147390808 CE For-Sale Reactive MTNR1A 43 42 COc1ccc2c(c1)nc([C@@H](C)Cl)n2CCNC(N)=O ZINC000147390808 CE For-Sale Reactive MTNR1B 33 40 COc1ccc2c(c1)nc([C@@H](C)Cl)n2CCNC(N)=O ZINC000147390808 CE For-Sale Reactive PROKR1 65 35 CCOc1ccccc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147390845 CG For-Sale Anodyne GRM2 15 42 CCOc1ccccc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147390845 CG For-Sale Anodyne ALS 48 44 CCOc1ccccc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147390845 CG For-Sale Anodyne HCN1 47 32 CCOc1ccccc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147390845 CG For-Sale Anodyne HCN4 40 31 Cc1cc(OCC(=O)NC2CC2)cc(C)c1S(N)(=O)=O ZINC000147390854 CC For-Sale Anodyne CA7 20 42 Cc1cc(OCC(=O)NC2CC2)cc(C)c1S(N)(=O)=O ZINC000147390854 CC For-Sale Anodyne LUXN 0 43 Cc1cc(OCC(=O)NC2CC2)cc(C)c1S(N)(=O)=O ZINC000147390854 CC For-Sale Anodyne ADIPOR1 0 41 Cc1cc(OCC(=O)NC2CC2)cc(C)c1S(N)(=O)=O ZINC000147390854 CC For-Sale Anodyne ADIPOR2 0 41 FC(F)CN[C@@H]1CCCCc2ccccc21 ZINC000147390901 BG For-Sale Anodyne KCNN3 15 44 CC[C@H]1CN(S(=O)(=O)c2ccccc2C)CC[C@@H]1N ZINC000147390922 CD On-Demand Anodyne EPHX2 21 45 CCNC(=O)COc1cccc(NC(=O)CNC(=O)OCC)c1 ZINC000147390926 DC On-Demand Anodyne MTNR1A 24 40 CCNC(=O)COc1cccc(NC(=O)CNC(=O)OCC)c1 ZINC000147390926 DC On-Demand Anodyne MTNR1B 20 40 CCNC(=O)COc1cccc(NC(=O)CNC(=O)OCC)c1 ZINC000147390926 DC On-Demand Anodyne PDS 40 33 CCCCCCCCNS(=O)(=O)c1ccc(CO)cn1 ZINC000147390934 DE For-Sale Mild S1PR2 50 37 CCCCCCCCNS(=O)(=O)c1ccc(CO)cn1 ZINC000147390934 DE For-Sale Mild ALOX15 40 38 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)Nc1ccc(Cl)cc1)C2 ZINC000147390943 FF On-Demand Anodyne MTNR1A 41 43 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)Nc1ccc(Cl)cc1)C2 ZINC000147390943 FF On-Demand Anodyne ROCK2 27 48 CS(=O)(=O)NCCC(=O)Nc1ccc(-c2cnco2)cc1 ZINC000147390980 DD On-Demand Anodyne IMPDH2 0 49 CCNc1nc(OC)nc(Oc2ccc3c(c2)OCO3)n1 ZINC000147391107 CD For-Sale Anodyne EDNRB 46 37 CCNc1nc(OC)nc(Oc2ccc3c(c2)OCO3)n1 ZINC000147391107 CD For-Sale Anodyne EDNRA 45 37 CCNc1nc(OC)nc(Oc2ccc3c(c2)OCO3)n1 ZINC000147391107 CD For-Sale Anodyne DYRK2 44 37 NCCc1ccccc1C(=O)NN1CCCCC1 ZINC000147391116 BD For-Sale Anodyne CNR1 50 31 CCCNC(=O)c1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1Cl ZINC000147391161 GJ On-Demand Anodyne SLC6A9 46 34 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(-n2cnnn2)cc1 ZINC000147391171 GF On-Demand Anodyne MRGPRX1 46 44 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(-n2cnnn2)cc1 ZINC000147391171 GF On-Demand Anodyne KCNJ1 45 37 CC(C)CCCCNCc1ccc(OC(F)(F)F)cc1 ZINC000147391177 CJ For-Sale Anodyne LEF 88 41 NCC(=O)c1cccc(OCC2CC2)c1 ZINC000147391200 BD For-Sale Anodyne CHRNA10 53 35 COc1cc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)ccc1NC(C)=O ZINC000147391274 HF On-Demand Anodyne ADRB2 20 40 COc1cc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)ccc1NC(C)=O ZINC000147391274 HF On-Demand Anodyne ADRB1 58 39 COc1cc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)ccc1NC(C)=O ZINC000147391274 HF On-Demand Anodyne TSHR 40 31 Cc1cc(Oc2ccc(C(=O)O)c(C)n2)ccc1C(C)C ZINC000147391336 CI For-Sale Anodyne THRA 51 39 Cc1cc(Oc2ccc(C(=O)O)c(C)n2)ccc1C(C)C ZINC000147391336 CI For-Sale Anodyne THRB 53 42 Cc1cc(C(=O)NCCSc2ccccc2)cc([N+](=O)[O-])c1 ZINC000147391366 DG On-Demand Bother MCL1 16 40 CCCNC(=O)c1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1Cl ZINC000147391371 GJ On-Demand Anodyne SLC6A9 46 34 CC(C)c1nc(CC2CCCCC2)no1 ZINC000147391394 BG On-Demand Anodyne BMP1 40 37 Cc1c(CN2CCSCC2)cccc1NC(=O)C[C@@H](C)NC(=O)c1ccccc1 ZINC000147391395 HH On-Demand Anodyne MRGPRX1 41 43 CCCCCCCCNS(=O)(=O)c1ccc(CO)cc1Br ZINC000147391440 GH For-Sale Mild LPAR2 43 38 CCCCCCCCNS(=O)(=O)c1ccc(CO)cc1Br ZINC000147391440 GH For-Sale Mild S1PR2 41 38 COc1ccc(CNCC(F)F)cc1O ZINC000147391446 BD On-Demand Anodyne INHA 40 33 COc1ccc(CNCC(F)F)cc1O ZINC000147391446 BD On-Demand Anodyne SLC6A13 0 58 COc1ccc(CNCC(F)F)cc1O ZINC000147391446 BD On-Demand Anodyne TTR 0 40 COc1ccc(CNCC(F)F)cc1O ZINC000147391446 BD On-Demand Anodyne MT-ND1 16 42 COc1ccc(CNCC(F)F)cc1O ZINC000147391446 BD On-Demand Anodyne CDK4 23 42 COc1ccc(CNCC(F)F)cc1O ZINC000147391446 BD On-Demand Anodyne DRTS_TRYCR 45 34 COc1ccc(CNCC(F)F)cc1O ZINC000147391446 BD On-Demand Anodyne CAN2 0 40 COc1cc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)ccc1NC(C)=O ZINC000147391462 HF On-Demand Anodyne ADRB2 20 40 COc1cc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)ccc1NC(C)=O ZINC000147391462 HF On-Demand Anodyne ADRB1 58 39 COc1cc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)ccc1NC(C)=O ZINC000147391462 HF On-Demand Anodyne TSHR 40 31 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OCC(=O)NCC)cc1 ZINC000147391469 FD On-Demand Anodyne SCN2A 18 41 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OCC(=O)NCC)cc1 ZINC000147391469 FD On-Demand Anodyne MMP3 27 44 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OCC(=O)NCC)cc1 ZINC000147391469 FD On-Demand Anodyne PLA2G4B 47 32 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OCC(=O)NCC)cc1 ZINC000147391469 FD On-Demand Anodyne ACR 18 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OCC(=O)NCC)cc1 ZINC000147391469 FD On-Demand Anodyne POLG_WNV 55 38 CC[C@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147391478 FE On-Demand Anodyne IDO1 23 40 CC[C@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147391478 FE On-Demand Anodyne Q9JN24_ECOLX 0 40 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000147391480 HG On-Demand Anodyne MAOB 23 41 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000147391480 HG On-Demand Anodyne COLA 33 42 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000147391480 HG On-Demand Anodyne CPT1A 31 42 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000147391480 HG On-Demand Anodyne ROCK1 20 40 CCCOc1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147391487 GG On-Demand Anodyne CYP2C19 18 42 CNc1cc(Oc2ccc3c(c2)OCO3)ncn1 ZINC000147391539 BE For-Sale Anodyne CLK1 51 38 CNc1cc(Oc2ccc3c(c2)OCO3)ncn1 ZINC000147391539 BE For-Sale Anodyne CLK4 52 34 CNc1cc(Oc2ccc3c(c2)OCO3)ncn1 ZINC000147391539 BE For-Sale Anodyne DYRK2 60 38 Cc1nc(Oc2ccc(C(C)(C)C)cc2)ccc1C(=O)O ZINC000147391549 CI For-Sale Anodyne MT-ND1 18 41 Cc1nc(Oc2ccc(C(C)(C)C)cc2)ccc1C(=O)O ZINC000147391549 CI For-Sale Anodyne AKR1C2 26 43 Cc1c(CN2CCSCC2)cccc1NC(=O)C[C@H](C)NC(=O)c1ccccc1 ZINC000147391588 HH On-Demand Anodyne MRGPRX1 41 43 COC(=O)[C@H](CN)N[C@@H](CC(C)C)C(=O)OC ZINC000147391608 BB For-Sale Anodyne FOLH1 44 43 COC(=O)[C@H](CN)N[C@@H](CC(C)C)C(=O)OC ZINC000147391608 BB For-Sale Anodyne NPR 17 45 CCC(CC)N(C)C(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147391613 EH For-Sale Anodyne NPY5R 27 43 CC(=O)c1c(C)[nH]c(C(=O)Nc2nc3ccc(OC(F)(F)F)cc3s2)c1C ZINC000147391622 GJ On-Demand Anodyne CSNK1D 50 50 CCCNC(=O)c1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1Cl ZINC000147391639 GJ On-Demand Anodyne SLC6A9 46 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OCC(=O)NCC)cc1 ZINC000147391661 FD On-Demand Anodyne SCN2A 18 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OCC(=O)NCC)cc1 ZINC000147391661 FD On-Demand Anodyne MMP3 27 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OCC(=O)NCC)cc1 ZINC000147391661 FD On-Demand Anodyne PLA2G4B 47 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OCC(=O)NCC)cc1 ZINC000147391661 FD On-Demand Anodyne ACR 18 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OCC(=O)NCC)cc1 ZINC000147391661 FD On-Demand Anodyne POLG_WNV 55 38 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000147391675 HG On-Demand Anodyne CPT1A 31 42 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2nc(-c3ccccc3)cs2)C1 ZINC000147391675 HG On-Demand Anodyne ROCK1 20 40 CC[C@@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147391676 FE On-Demand Anodyne IDO1 23 40 CC[C@@H](CNS(=O)(=O)c1ccc(Br)cc1)CC(=O)O ZINC000147391676 FE On-Demand Anodyne Q9JN24_ECOLX 0 40 Oc1ccc(CNCC(F)F)c(O)c1 ZINC000147391684 BD For-Sale Clean TYR 26 48 CCNc1ncc(Br)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147391771 EG For-Sale Anodyne DYRK1A 23 40 CCNc1ncc(Br)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147391771 EG For-Sale Anodyne CLK1 32 40 CCNc1ncc(Br)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147391771 EG For-Sale Anodyne CLK2 32 40 CCNc1ncc(Br)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147391771 EG For-Sale Anodyne CLK4 38 40 CCNc1ncc(Br)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147391771 EG For-Sale Anodyne DYRK1B 18 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccnc1N1CCOCC1)C2 ZINC000147391835 FE On-Demand Anodyne ROCK2 35 45 CCC(CC)N(C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147391849 CH For-Sale Anodyne NPY5R 27 43 NC(=O)NCCNS(=O)(=O)c1cccc(/C=C/C(=O)O)c1 ZINC000147391877 DB For-Sale Anodyne AKR1C3 19 43 CC[C@H](CNS(=O)(=O)c1ccc(OC)c(C)c1)CC(=O)O ZINC000147391893 DD On-Demand Anodyne LEF 41 39 COc1cc(CNCCCCC(C)C)cc(OC)c1O ZINC000147391945 CG For-Sale Anodyne LPAR2 51 40 COc1cc(CNCCCCC(C)C)cc(OC)c1O ZINC000147391945 CG For-Sale Anodyne S1PR2 50 39 COc1cc(CNCCCCC(C)C)cc(OC)c1O ZINC000147391945 CG For-Sale Anodyne SLC6A13 0 47 COc1cc(CNCCCCC(C)C)cc(OC)c1O ZINC000147391945 CG For-Sale Anodyne LEF 73 37 COc1cc(CNCCCCC(C)C)cc(OC)c1O ZINC000147391945 CG For-Sale Anodyne GPM3 0 40 O=S(=O)(NCc1ccc(-n2ccnc2)c(F)c1)N1CCOCC1 ZINC000147391954 EC On-Demand Anodyne NOS2 50 33 CCN(CC)[C@@H](C)CNC(=O)CCNS(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000147391987 GD On-Demand Bother COLA 29 41 Cc1nc(Oc2cccc3ccccc23)ccc1C(=O)O ZINC000147392017 CI For-Sale Anodyne ALB 24 43 Cc1nc(Oc2cccc3ccccc23)ccc1C(=O)O ZINC000147392017 CI For-Sale Anodyne ALS 58 37 Cc1nc(Oc2cccc3ccccc23)ccc1C(=O)O ZINC000147392017 CI For-Sale Anodyne MCL1 48 43 CCCNC(=O)c1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1Cl ZINC000147392066 HH On-Demand Anodyne ROCK2 25 47 COc1cc(NC(=O)NCc2ccc(-n3ccnc3C)c(F)c2)ccc1NC(C)=O ZINC000147392083 HH On-Demand Anodyne ROCK2 21 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive FKBP1A 23 42 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive CASP3 69 38 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive MMP13 36 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive MMP3 38 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive MMP8 15 44 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive EPHX2 38 41 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive CASP7 81 38 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive TGM2 59 42 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive MMP7 47 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive MMP1 43 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive F13A1 93 42 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive AKR1C3 23 56 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147392090 GF For-Sale Reactive NAMPT 25 46 CC[C@@H](CNS(=O)(=O)c1ccc(OC)c(C)c1)CC(=O)O ZINC000147392107 DD On-Demand Anodyne LEF 41 39 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccccc1NS(C)(=O)=O ZINC000147392115 HG On-Demand Anodyne CCR8 59 34 CC(C)CCCCNC(=O)CCl ZINC000147392149 AE For-Sale Reactive DNPEP 51 34 Cc1cc(N)c(OCCN2CCN(C(=O)OC(C)(C)C)CC2)cc1Cl ZINC000147392162 FG For-Sale Anodyne HTR4 46 38 Cc1cc(N)c(OCCN2CCN(C(=O)OC(C)(C)C)CC2)cc1Cl ZINC000147392162 FG For-Sale Anodyne THRB 15 40 CCN(CC)[C@H](C)CNC(=O)CCNS(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000147392178 GD On-Demand Bother COLA 29 41 CCCNc1ncc(F)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147392194 CF For-Sale Anodyne CLK4 42 38 CCCNc1ncc(F)c(Oc2ccc3c(c2)OCO3)n1 ZINC000147392194 CF For-Sale Anodyne DYRK2 40 37 CSCC(=O)Nc1ccc(-c2cnco2)cc1 ZINC000147392202 BF On-Demand Anodyne IMPDH2 0 54 Cc1nc(Oc2ccc3ccccc3c2)ccc1C(=O)O ZINC000147392237 CI For-Sale Anodyne PYGL 21 40 Cc1nc(Oc2ccc3ccccc3c2)ccc1C(=O)O ZINC000147392237 CI For-Sale Anodyne PYGM 28 40 Cc1nc(Oc2ccc3ccccc3c2)ccc1C(=O)O ZINC000147392237 CI For-Sale Anodyne AKR1C2 46 35 O=Cc1ccc(OC[C@@H](O)CCl)cc1 ZINC000147392280 BD For-Sale Reactive ADRB2 23 41 CCCCCCCCNS(=O)(=O)c1cc(CO)n(C)c1 ZINC000147392314 DE For-Sale Mild ASAH1 67 34 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive FKBP1A 23 42 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive CASP3 69 38 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive MMP13 36 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive MMP3 38 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive MMP8 15 44 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive EPHX2 38 41 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive CASP7 81 38 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive TGM2 59 42 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive MMP7 47 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive MMP1 43 45 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive F13A1 93 42 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive AKR1C3 23 56 CC(=O)Nc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147392324 GF For-Sale Reactive NAMPT 25 46 c1ccc([C@@H]2C[C@H](c3ccccc3)CCN2)cc1 ZINC000147392333 BH For-Sale Anodyne PRCP 18 40 CNc1ccc(C(=O)Nc2cccc(CN3CCSCC3)c2C)cc1[N+](=O)[O-] ZINC000147392335 HH On-Demand Bother SLC9A1 41 37 CNc1ccc(C(=O)Nc2cccc(CN3CCSCC3)c2C)cc1[N+](=O)[O-] ZINC000147392335 HH On-Demand Bother BCL2 40 32 CNc1ccc(C(=O)Nc2cccc(CN3CCSCC3)c2C)cc1[N+](=O)[O-] ZINC000147392335 HH On-Demand Bother TAAR1 21 40 CNc1ccc(C(=O)Nc2cccc(CN3CCSCC3)c2C)cc1[N+](=O)[O-] ZINC000147392335 HH On-Demand Bother MRGPRX1 43 40 COc1ccc(C(=O)NCC2(C(=O)O)CCC2)cc1 ZINC000147392342 CD On-Demand Anodyne MT-ND1 16 40 COc1ccc(C(=O)NCC2(C(=O)O)CCC2)cc1 ZINC000147392342 CD On-Demand Anodyne H9B8T9_CAPHI 15 50 CC[C@H](C)NC(=O)c1ccc(NC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147392370 GI On-Demand Anodyne AVPR2 40 37 CC[C@H](C)NC(=O)c1ccc(NC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147392370 GI On-Demand Anodyne PRNP 73 38 CC[C@H](C)NC(=O)c1ccc(NC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147392370 GI On-Demand Anodyne MAPK10 15 40 CC[C@H](C)NC(=O)c1ccc(NC(=O)c2cnn(-c3ccccc3Cl)c2)cc1 ZINC000147392370 GI On-Demand Anodyne NOD2 40 34 O=C(CN1CCCCCC1=O)Nc1ccc(-c2cnco2)cc1 ZINC000147392389 DF On-Demand Anodyne CHRNA7 20 41 O=C(CN1CCCCCC1=O)Nc1ccc(-c2cnco2)cc1 ZINC000147392389 DF On-Demand Anodyne IMPDH2 0 43 COc1cc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)ccc1NC(C)=O ZINC000147392414 GH On-Demand Anodyne TSHR 48 31 Cc1nn(C(F)F)c(C)c1CC(=O)Nc1ccccc1-n1ccnc1 ZINC000147392463 EG On-Demand Anodyne KCNQ2 52 37 O=Cc1ccc(OC[C@H](O)CCl)cc1 ZINC000147392495 BD For-Sale Reactive ADRB2 23 41 Cc1nc(Oc2ccccc2C(C)C)ccc1C(=O)O ZINC000147392498 CI For-Sale Anodyne ALS 49 33 Cc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1C ZINC000147392558 CE On-Demand Anodyne HCN1 53 33 Cc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1C ZINC000147392558 CE On-Demand Anodyne HCN4 51 33 Cc1cc(C)n(-c2ccc(NC(=O)C(=O)NCC(C)(C)N3CCC[C@H](C)C3)cn2)n1 ZINC000147392569 HE On-Demand Anodyne DGAT1 19 40 COc1cc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)ccc1NC(C)=O ZINC000147392597 GH On-Demand Anodyne TSHR 48 31 CCCNc1cc(Oc2ccc3c(c2)OCO3)nc(C)n1 ZINC000147392614 CG For-Sale Anodyne EDNRB 21 42 CCCNc1cc(Oc2ccc3c(c2)OCO3)nc(C)n1 ZINC000147392614 CG For-Sale Anodyne EDNRA 21 42 CCCNc1cc(Oc2ccc3c(c2)OCO3)nc(C)n1 ZINC000147392614 CG For-Sale Anodyne DYRK1A 19 41 CCCNc1cc(Oc2ccc3c(c2)OCO3)nc(C)n1 ZINC000147392614 CG For-Sale Anodyne CLK1 30 41 CCCNc1cc(Oc2ccc3c(c2)OCO3)nc(C)n1 ZINC000147392614 CG For-Sale Anodyne DYRK2 49 41 COc1ccc2nc(CCCl)n(CCNC(N)=O)c2c1 ZINC000147392622 CD For-Sale Reactive DRD4 42 32 COc1ccc2nc(CCCl)n(CCNC(N)=O)c2c1 ZINC000147392622 CD For-Sale Reactive NQO2 33 40 COc1ccc2nc(CCCl)n(CCNC(N)=O)c2c1 ZINC000147392622 CD For-Sale Reactive MTNR1A 60 44 COc1ccc2nc(CCCl)n(CCNC(N)=O)c2c1 ZINC000147392622 CD For-Sale Reactive MTNR1B 47 40 COc1ccc2nc(CCCl)n(CCNC(N)=O)c2c1 ZINC000147392622 CD For-Sale Reactive SCD 17 41 COc1ccc2nc(CCCl)n(CCNC(N)=O)c2c1 ZINC000147392622 CD For-Sale Reactive PROKR1 62 35 Cc1c(CN2CCSCC2)cccc1NC(=O)[C@H](C)NC(=O)Nc1ccccc1 ZINC000147392637 HH On-Demand Anodyne CCR3 26 45 CC[C@H](C)NC(=O)c1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147392705 EG On-Demand Anodyne PRNP 59 36 CC[C@H](C)NC(=O)c1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147392705 EG On-Demand Anodyne F3 72 34 CC[C@H](C)NC(=O)c1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147392705 EG On-Demand Anodyne NOD2 40 34 CC[C@H](CNS(=O)(=O)Cc1ccc(F)cc1)CC(=O)O ZINC000147392740 DD On-Demand Anodyne HMGCR 40 33 Cc1cc(C)n(-c2ccc(NC(=O)C(=O)NCC(C)(C)N3CCC[C@@H](C)C3)cn2)n1 ZINC000147392751 HE On-Demand Anodyne DGAT1 19 40 CCCCCCCCNS(=O)(=O)c1ccc(CO)cc1F ZINC000147392785 DF For-Sale Mild ASAH1 51 31 CCNc1cc(Oc2ccc3c(c2)OCO3)nc(C)n1 ZINC000147392814 CF For-Sale Anodyne DYRK2 54 39 COc1cc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)ccc1NC(C)=O ZINC000147392816 GH On-Demand Anodyne TSHR 48 31 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)NCc1ccc(-n3ccnc3)c(F)c1)C(=O)C2 ZINC000147392843 HF On-Demand Anodyne CA5B 29 56 CC1(C)[C@H]2CC[C@@]1(CS(=O)(=O)NCc1ccc(-n3ccnc3)c(F)c1)C(=O)C2 ZINC000147392843 HF On-Demand Anodyne CA5A 32 56 CS(=O)(=O)c1cc(C(=O)N2CCN(CC3CC3)CC2)cc([N+](=O)[O-])c1 ZINC000147392862 FD On-Demand Bother SLC6A9 16 40 CCCCCc1ccc(N[C@@H]2CCO[C@@H]2C)cc1 ZINC000147392893 BI For-Sale Anodyne SPHK1 19 45 O=C(Nc1cccnc1N1CCOCC1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147392894 FG On-Demand Anodyne SCN10A 19 40 O=C(Nc1cccnc1N1CCOCC1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147392894 FG On-Demand Anodyne G2YM83_BOTF4 45 32 CC[C@@H](CNS(=O)(=O)Cc1ccc(F)cc1)CC(=O)O ZINC000147392933 DD On-Demand Anodyne HMGCR 40 33 Oc1cccc(CNCC(F)F)c1 ZINC000147392973 AD On-Demand Anodyne KYNU 40 28 Oc1cccc(CNCC(F)F)c1 ZINC000147392973 AD On-Demand Anodyne SLC6A13 0 51 Cc1cc(C(=O)NCC2(C(=O)O)CCC2)ccc1F ZINC000147393007 CE On-Demand Anodyne LEF 42 32 CC[C@@H]1CN(S(=O)(=O)c2ccc(F)c(F)c2)CC[C@@H]1N ZINC000147393015 DD On-Demand Anodyne GCKR 61 31 COc1cc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)ccc1NC(C)=O ZINC000147393056 GH On-Demand Anodyne TSHR 48 31 CC[C@H](NC(=O)[C@@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393070 BD For-Sale Anodyne LTA4H 41 35 CC[C@H](NC(=O)[C@@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393070 BD For-Sale Anodyne HLA-A 45 40 CC[C@H](NC(=O)[C@@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393070 BD For-Sale Anodyne ENPEP 72 38 CC[C@H](NC(=O)[C@@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393070 BD For-Sale Anodyne ACE2 58 35 CC[C@H](NC(=O)[C@@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393070 BD For-Sale Anodyne GNPAT 0 43 CC[C@H](NC(=O)[C@@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393070 BD For-Sale Anodyne GSP 0 41 CC[C@H](NC(=O)[C@@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393070 BD For-Sale Anodyne SLC15A2 0 46 CC[C@H](NC(=O)[C@@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393070 BD For-Sale Anodyne NOD1 102 44 COc1ccccc1CN(C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1)C1CC1 ZINC000147393097 HF On-Demand Bother COLA 43 35 COc1ccccc1CN(C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1)C1CC1 ZINC000147393097 HF On-Demand Bother MBTPS1 54 37 CCCCCc1ccc(N[C@H]2CCO[C@@H]2C)cc1 ZINC000147393101 BI For-Sale Anodyne SPHK1 19 45 CNC(=O)c1cccc([N+](=O)[O-])c1F ZINC000147393108 AD For-Sale Bother COLA 53 32 CNC(=O)c1cccc([N+](=O)[O-])c1F ZINC000147393108 AD For-Sale Bother KCNMA1 18 46 Cc1c(CN2CCSCC2)cccc1NC(=O)CNC(=O)Cc1ccccc1 ZINC000147393113 GF On-Demand Anodyne KCNQ2 32 41 Cc1c(CN2CCSCC2)cccc1NC(=O)CNC(=O)Cc1ccccc1 ZINC000147393113 GF On-Demand Anodyne SIGMAR1 19 42 Cc1c(CN2CCSCC2)cccc1NC(=O)CNC(=O)Cc1ccccc1 ZINC000147393113 GF On-Demand Anodyne CCR3 29 43 Cc1c(CN2CCSCC2)cccc1NC(=O)CNC(=O)Cc1ccccc1 ZINC000147393113 GF On-Demand Anodyne MRGPRX1 28 40 Cc1c(CN2CCSCC2)cccc1NC(=O)CNC(=O)Cc1ccccc1 ZINC000147393113 GF On-Demand Anodyne NPFFR1 56 39 CC(=O)Nc1ccccc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147393126 CF For-Sale Anodyne PYGL 23 44 CC(=O)Nc1ccccc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147393126 CF For-Sale Anodyne PYGM 29 44 O=C(Nc1cccnc1N1CCOCC1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147393129 FG On-Demand Anodyne SCN10A 19 40 O=C(Nc1cccnc1N1CCOCC1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147393129 FG On-Demand Anodyne G2YM83_BOTF4 45 32 CC(=O)N1CCC[C@H](C(=O)Nc2ccc(-c3cnco3)cc2)C1 ZINC000147393131 DF On-Demand Anodyne IMPDH2 0 47 CC(=O)N1CCC[C@H](C(=O)Nc2ccc(-c3cnco3)cc2)C1 ZINC000147393131 DF On-Demand Anodyne RHOA 0 52 Cn1nccc1CNC(=O)[C@@H]1CCC(=O)N(Cc2ccccc2)[C@@H]1c1ccccc1 ZINC000147393133 HG On-Demand Anodyne P2RX7 35 45 CC[C@H]1CN(S(=O)(=O)c2ccc(F)c(F)c2)CC[C@@H]1N ZINC000147393204 DD On-Demand Anodyne GCKR 61 31 CCCCCCCCNS(=O)(=O)c1ccc(C)c(CO)c1 ZINC000147393209 DG For-Sale Mild ALOX15 56 46 FC(F)CNCc1ccc(OC(F)F)cc1OC(F)F ZINC000147393218 DG For-Sale Anodyne PHES 0 41 COc1ccc(OC)c(NC(=O)CN2CCC(c3ccccn3)CC2)c1 ZINC000147393234 FF On-Demand Anodyne DRD4 31 66 COc1ccc(OC)c(NC(=O)CN2CCC(c3ccccn3)CC2)c1 ZINC000147393234 FF On-Demand Anodyne HCRTR1 21 40 COc1ccc(OC)c(NC(=O)CN2CCC(c3ccccn3)CC2)c1 ZINC000147393234 FF On-Demand Anodyne NPY2R 23 40 COc1ccc(OC)c(NC(=O)CN2CCC(c3ccccn3)CC2)c1 ZINC000147393234 FF On-Demand Anodyne ACOX1 47 37 COc1ccc(OC)c(NC(=O)CN2CCC(c3ccccn3)CC2)c1 ZINC000147393234 FF On-Demand Anodyne ALK 18 41 CCc1cccc(Oc2ccc(NC(=O)N[C@@H]3CCCN(S(C)(=O)=O)C3)cn2)c1 ZINC000147393282 HF On-Demand Anodyne CHRNA7 19 40 CCc1cccc(Oc2ccc(NC(=O)N[C@@H]3CCCN(S(C)(=O)=O)C3)cn2)c1 ZINC000147393282 HF On-Demand Anodyne EPHX2 39 41 CC[C@H](NC(=O)[C@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393290 BD For-Sale Anodyne LTA4H 41 35 CC[C@H](NC(=O)[C@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393290 BD For-Sale Anodyne HLA-A 45 40 CC[C@H](NC(=O)[C@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393290 BD For-Sale Anodyne ENPEP 72 38 CC[C@H](NC(=O)[C@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393290 BD For-Sale Anodyne ACE2 58 35 CC[C@H](NC(=O)[C@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393290 BD For-Sale Anodyne GNPAT 0 43 CC[C@H](NC(=O)[C@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393290 BD For-Sale Anodyne GSP 0 41 CC[C@H](NC(=O)[C@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393290 BD For-Sale Anodyne SLC15A2 0 46 CC[C@H](NC(=O)[C@H](C)CCC[C@H](C)N)C(=O)O ZINC000147393290 BD For-Sale Anodyne NOD1 102 44 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1CC ZINC000147393295 CF For-Sale Anodyne Q9XSW7_PIG 0 40 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1CC ZINC000147393295 CF For-Sale Anodyne DYRK1A 49 41 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1CC ZINC000147393295 CF For-Sale Anodyne CLK1 58 41 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1CC ZINC000147393295 CF For-Sale Anodyne CLK2 51 41 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1CC ZINC000147393295 CF For-Sale Anodyne CLK3 36 41 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1CC ZINC000147393295 CF For-Sale Anodyne CLK4 78 41 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1CC ZINC000147393295 CF For-Sale Anodyne DYRK2 52 38 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1CC ZINC000147393295 CF For-Sale Anodyne DYRK1B 39 40 CCCCCc1ccc(N[C@@H]2CCO[C@H]2C)cc1 ZINC000147393319 BI For-Sale Anodyne SPHK1 19 45 O=C(Nc1cccnc1N1CCOCC1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147393323 FG On-Demand Anodyne SCN10A 19 40 O=C(Nc1cccnc1N1CCOCC1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147393323 FG On-Demand Anodyne G2YM83_BOTF4 45 32 C[C@H](Cl)c1nc2ccccc2n1CCNC(N)=O ZINC000147393350 CE For-Sale Reactive HRH1 27 43 C[C@H](Cl)c1nc2ccccc2n1CCNC(N)=O ZINC000147393350 CE For-Sale Reactive PDE6D 67 38 COc1cc(C)ccc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147393351 CG For-Sale Anodyne ALS 66 38 Cc1c(CN2CCSCC2)cccc1NC(=O)[C@@H](C)NC(=O)c1ccccc1 ZINC000147393352 GG On-Demand Anodyne MRGPRX1 41 43 CC(=O)N1CCC[C@@H](C(=O)Nc2ccc(-c3cnco3)cc2)C1 ZINC000147393353 DF On-Demand Anodyne IMPDH2 0 47 CC(=O)N1CCC[C@@H](C(=O)Nc2ccc(-c3cnco3)cc2)C1 ZINC000147393353 DF On-Demand Anodyne RHOA 0 52 Cn1nccc1CNC(=O)[C@H]1CCC(=O)N(Cc2ccccc2)[C@@H]1c1ccccc1 ZINC000147393368 HG On-Demand Anodyne P2RX7 35 45 O=C(O)c1ccc(-c2ccsc2Cl)cc1 ZINC000147393369 BH For-Sale Anodyne SRD5A2 27 46 FC(F)CNCc1ccc2ccccc2c1 ZINC000147393471 BG On-Demand Anodyne CYP2A5 0 45 CCc1cccc(Oc2ccc(NC(=O)N[C@H]3CCCN(S(C)(=O)=O)C3)cn2)c1 ZINC000147393494 HF On-Demand Anodyne CHRNA7 19 40 CCc1cccc(Oc2ccc(NC(=O)N[C@H]3CCCN(S(C)(=O)=O)C3)cn2)c1 ZINC000147393494 HF On-Demand Anodyne EPHX2 39 41 CCCCCc1ccc(N[C@H]2CCO[C@H]2C)cc1 ZINC000147393495 BI For-Sale Anodyne SPHK1 19 45 CCCNc1ncnc(Oc2ccc3c(c2)OCO3)c1C ZINC000147393504 CG For-Sale Anodyne CLK1 45 39 CCCNc1ncnc(Oc2ccc3c(c2)OCO3)c1C ZINC000147393504 CG For-Sale Anodyne CLK4 56 39 CCCNc1ncnc(Oc2ccc3c(c2)OCO3)c1C ZINC000147393504 CG For-Sale Anodyne DYRK2 43 38 O=S(=O)(NCc1ccc(-n2ccnc2)c(F)c1)c1ccc(Cl)s1 ZINC000147393509 FG On-Demand Anodyne CCR4 57 38 CC(C)CCCCNC(=O)CCCCCl ZINC000147393556 BG For-Sale Reactive NOD1 29 43 C[C@@H](Cl)c1nc2ccccc2n1CCNC(N)=O ZINC000147393568 CE For-Sale Reactive HRH1 27 43 C[C@@H](Cl)c1nc2ccccc2n1CCNC(N)=O ZINC000147393568 CE For-Sale Reactive PDE6D 67 38 Cn1nccc1CNC(=O)[C@@H]1CCC(=O)N(Cc2ccccc2)[C@H]1c1ccccc1 ZINC000147393576 HG On-Demand Anodyne P2RX7 35 45 Cc1nc(Oc2cc(Cl)c(Cl)cc2Cl)ccc1C(=O)O ZINC000147393610 EJ For-Sale Anodyne ALS 45 37 Cc1nc(Oc2cc(Cl)c(Cl)cc2Cl)ccc1C(=O)O ZINC000147393610 EJ For-Sale Anodyne AKR1C2 47 36 Cc1nc(Oc2cc(Cl)c(Cl)cc2Cl)ccc1C(=O)O ZINC000147393610 EJ For-Sale Anodyne AKR1C1 48 36 CCCOc1cccc(CNCC(F)F)c1 ZINC000147393634 BF On-Demand Anodyne PDS 49 36 CCCCCCCCNS(=O)(=O)c1c[nH]c(CO)c1 ZINC000147393643 CE For-Sale Mild ALOX15 41 44 CCCCCCCCNS(=O)(=O)c1c[nH]c(CO)c1 ZINC000147393643 CE For-Sale Mild ASAH1 52 34 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1C ZINC000147393711 CF For-Sale Anodyne DYRK1A 46 41 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1C ZINC000147393711 CF For-Sale Anodyne CLK1 54 41 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1C ZINC000147393711 CF For-Sale Anodyne CLK2 48 41 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1C ZINC000147393711 CF For-Sale Anodyne CLK3 35 40 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1C ZINC000147393711 CF For-Sale Anodyne CLK4 73 41 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1C ZINC000147393711 CF For-Sale Anodyne DYRK2 51 37 CCNc1ncnc(Oc2ccc3c(c2)OCO3)c1C ZINC000147393711 CF For-Sale Anodyne DYRK1B 38 41 CCC(=O)Nc1ccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147393730 HG On-Demand Anodyne ROCK2 23 40 CC(C)CCCCNC(=O)CCCCl ZINC000147393776 BF For-Sale Reactive NOD1 28 41 CC[C@@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147393782 DH On-Demand Anodyne CACNA1H 39 40 CC[C@@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147393782 DH On-Demand Anodyne CACNA1I 64 39 Cn1nccc1CNC(=O)[C@H]1CCC(=O)N(Cc2ccccc2)[C@H]1c1ccccc1 ZINC000147393785 HG On-Demand Anodyne P2RX7 35 45 CCCCc1ccc(N[C@@H]2CCO[C@@H]2C)cc1 ZINC000147393830 BH On-Demand Anodyne SPHK1 15 40 CCCOc1ccccc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147393831 CH For-Sale Anodyne GRM2 22 42 CCCOc1ccccc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147393831 CH For-Sale Anodyne ALS 44 43 CCCOc1ccccc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147393831 CH For-Sale Anodyne MCL1 41 37 CC[C@@H](N)[C@@H]1CCCN(C(C)=O)C1 ZINC000147393865 AC For-Sale Anodyne DPP8 18 40 CCC(=O)Nc1ccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147393914 HG On-Demand Anodyne ROCK2 23 40 CC[C@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147393977 DH On-Demand Anodyne CACNA1H 39 40 CC[C@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147393977 DH On-Demand Anodyne CACNA1I 64 39 O=S(=O)(c1cccc2cnccc12)N1CCCC[C@@H]1CBr ZINC000147394024 FG For-Sale Reactive P2RX7 43 41 O=S(=O)(c1cccc2cnccc12)N1CCCC[C@@H]1CBr ZINC000147394024 FG For-Sale Reactive Q95J97_RABIT 0 53 O=C(NCC1(C(=O)O)CCC1)c1cccc(F)c1Cl ZINC000147394028 CE On-Demand Anodyne HCN1 49 30 O=C(NCC1(C(=O)O)CCC1)c1cccc(F)c1Cl ZINC000147394028 CE On-Demand Anodyne HCN4 46 30 CC[C@H](N)[C@@H]1CCCN(C(C)=O)C1 ZINC000147394048 AC For-Sale Anodyne DPP8 18 40 Cn1nccc1CNC(=O)c1ccccc1Oc1ccc(Cl)cc1Cl ZINC000147394049 GI On-Demand Anodyne P2RX7 19 53 Cn1nccc1CNC(=O)c1ccccc1Oc1ccc(Cl)cc1Cl ZINC000147394049 GI On-Demand Anodyne HCN1 60 32 CCCCCCCCNS(=O)(=O)Cc1ccc(CO)cc1 ZINC000147394091 DF For-Sale Mild S1PR2 69 39 CCCCCCCCNS(=O)(=O)Cc1ccc(CO)cc1 ZINC000147394091 DF For-Sale Mild RELA 18 41 CCCCCCCCNS(=O)(=O)Cc1ccc(CO)cc1 ZINC000147394091 DF For-Sale Mild ASAH1 46 32 Cc1nc(OCCOc2ccccc2)ccc1C(=O)O ZINC000147394124 CF For-Sale Anodyne PPARG 66 40 Cc1nc(OCCOc2ccccc2)ccc1C(=O)O ZINC000147394124 CF For-Sale Anodyne PPARA 66 40 Cc1nc(OCCOc2ccccc2)ccc1C(=O)O ZINC000147394124 CF For-Sale Anodyne GRM2 0 42 Cc1nc(OCCOc2ccccc2)ccc1C(=O)O ZINC000147394124 CF For-Sale Anodyne PLA2G4B 40 33 CNc1nccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147394139 BE For-Sale Anodyne DYRK1A 23 42 CNc1nccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147394139 BE For-Sale Anodyne CLK1 24 42 CNc1nccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147394139 BE For-Sale Anodyne CLK4 40 42 CNc1nccc(Oc2ccc3c(c2)OCO3)n1 ZINC000147394139 BE For-Sale Anodyne DYRK1B 22 42 COC(=O)CNC(C)(C)c1cccc(F)c1 ZINC000147394202 BD On-Demand Anodyne KCNN4 0 44 CCCCc1ccc(N[C@@H]2CCO[C@H]2C)cc1 ZINC000147394211 BH On-Demand Anodyne SPHK1 15 40 C[C@@]1(C(=O)N(CCCC(=O)O)Cc2cccc(Cl)c2)CCN1C(=O)c1csc2ccccc12 ZINC000147394221 JK Annotated Anodyne C5AR1 27 43 O=C(NCC1(C(=O)O)CCC1)c1ccc(Br)cc1Cl ZINC000147394232 EG On-Demand Anodyne P2RX7 0 43 O=S(=O)(c1cccc2cnccc12)N1CCCC[C@H]1CBr ZINC000147394241 FG For-Sale Reactive P2RX7 43 41 O=S(=O)(c1cccc2cnccc12)N1CCCC[C@H]1CBr ZINC000147394241 FG For-Sale Reactive Q95J97_RABIT 0 53 CC[C@@H](N)[C@H]1CCCN(C(C)=O)C1 ZINC000147394256 AC For-Sale Anodyne DPP8 18 40 O=C(Nc1ccccc1OCCn1ccnc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147394262 GI On-Demand Anodyne TBXAS1 35 41 Cc1ccc(C(=O)CCC(=O)Nc2cccc(CN3CCSCC3)c2C)cc1 ZINC000147394269 GI On-Demand Anodyne MRGPRX1 40 39 N#CCOc1ccccc1CNCC(F)F ZINC000147394359 BD For-Sale Mild PHES 0 57 CCCCc1ccc(N[C@H]2CCO[C@H]2C)cc1 ZINC000147394437 BH On-Demand Anodyne SPHK1 15 40 CC[C@H](N)[C@H]1CCCN(C(C)=O)C1 ZINC000147394447 AC For-Sale Anodyne DPP8 18 40 Cc1nc(O[C@@H]2C[C@H](C)CC[C@@H]2C(C)C)ccc1C(=O)O ZINC000147394452 CH For-Sale Anodyne SERPINE1 40 39 CO/C=C1/CCc2ccccc2C1=O ZINC000147394460 AE For-Sale Mild CYP27A1 0 47 O=C(Nc1ccccc1OCCn1ccnc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147394470 GI On-Demand Anodyne TBXAS1 35 41 CCCCCCCCNS(=O)(=O)c1ccc(Cl)c(CO)c1 ZINC000147394549 EG For-Sale Mild TBXA2R 42 33 CCCCCCCCNS(=O)(=O)c1ccc(Cl)c(CO)c1 ZINC000147394549 EG For-Sale Mild ALOX15 60 45 O=C(O)c1cc(Cl)cc(NC(=O)N2CCC[C@H](CO)C2)c1 ZINC000147394658 DE On-Demand Anodyne CACNA1I 45 35 C[C@H]1OCC[C@H]1Nc1ccc(N2CCOCC2)cc1 ZINC000147394667 CE On-Demand Anodyne AKR1C3 0 40 O=C(Nc1ccccc1OCCn1ccnc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147394677 GI On-Demand Anodyne TBXAS1 35 41 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNC(C)(C)Cc2ccccc2)cc(N2CCCC2=O)c1 ZINC000147394749 KJ Annotated Anodyne CTSD 70 78 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNC(C)(C)Cc2ccccc2)cc(N2CCCC2=O)c1 ZINC000147394749 KJ Annotated Anodyne BACE2 75 77 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNC(C)(C)Cc2ccccc2)cc(N2CCCC2=O)c1 ZINC000147394749 KJ Annotated Anodyne BACE1 88 87 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNC(C)(C)Cc2ccccc2)cc(N2CCCC2=O)c1 ZINC000147394749 KJ Annotated Anodyne PLM1_PLAFA 62 51 CCNc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNC(C)(C)Cc2ccccc2)cc(N2CCCC2=O)c1 ZINC000147394749 KJ Annotated Anodyne PLM2_PLAFA 45 51 CS(=O)(=O)c1cc(C(=O)N(Cc2ccccc2)C2CCCCC2)cc([N+](=O)[O-])c1 ZINC000147394761 HH On-Demand Bother ACE 38 40 CS(=O)(=O)c1cc(C(=O)N(Cc2ccccc2)C2CCCCC2)cc([N+](=O)[O-])c1 ZINC000147394761 HH On-Demand Bother LIMK2 42 35 CCCCCCCCNS(=O)(=O)c1cnn(CCO)c1 ZINC000147394778 DD For-Sale Mild ASAH1 75 33 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2o1 ZINC000147394799 FJ On-Demand Anodyne MAOB 19 40 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2o1 ZINC000147394799 FJ On-Demand Anodyne HPSE 27 41 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2o1 ZINC000147394799 FJ On-Demand Anodyne AGPAT2 46 41 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2o1 ZINC000147394799 FJ On-Demand Anodyne TAAR1 18 42 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2o1 ZINC000147394799 FJ On-Demand Anodyne SHH 49 35 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2o1 ZINC000147394799 FJ On-Demand Anodyne IMDH_CRYPV 43 38 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2o1 ZINC000147394799 FJ On-Demand Anodyne KCNK3 54 37 Cc1ccc(Cc2cnc(NC(=O)COc3ccc(C(N)=O)cc3)s2)cc1C ZINC000147394849 GG On-Demand Anodyne SCD1 43 46 Cc1ccc(Cc2cnc(NC(=O)COc3ccc(C(N)=O)cc3)s2)cc1C ZINC000147394849 GG On-Demand Anodyne SCD 38 46 COCc1nc(C(=O)NCc2ccc(CN3CCOCC3)cc2)cs1 ZINC000147394863 FE On-Demand Anodyne DPOL_VZVD 25 44 C[C@@H]1OCC[C@H]1Nc1ccc(N2CCOCC2)cc1 ZINC000147394870 CE On-Demand Anodyne AKR1C3 0 40 Cc1nc(O[C@@H]2C[C@@H](C)CC[C@@H]2C(C)C)ccc1C(=O)O ZINC000147394875 CH For-Sale Anodyne SERPINE1 40 39 O=C(O)c1cc(Cl)cc(NC(=O)N2CCC[C@@H](CO)C2)c1 ZINC000147394876 DE On-Demand Anodyne CACNA1I 45 35 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1OCCn1ccnc1)C2 ZINC000147394883 GG On-Demand Anodyne TBXAS1 27 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1OCCn1ccnc1)C2 ZINC000147394883 GG On-Demand Anodyne ROCK2 46 51 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1OCCn1ccnc1)C2 ZINC000147394883 GG On-Demand Anodyne QPCT 27 42 CC[C@H](NC(=O)[C@H]1Cc2ccccc2N1)C(=O)O ZINC000147394933 BD For-Sale Anodyne ACE 54 42 CC[C@H](NC(=O)[C@H]1Cc2ccccc2N1)C(=O)O ZINC000147394933 BD For-Sale Anodyne MME 40 42 CC[C@H](NC(=O)[C@H]1Cc2ccccc2N1)C(=O)O ZINC000147394933 BD For-Sale Anodyne TRHR 46 38 CC[C@H](NC(=O)[C@H]1Cc2ccccc2N1)C(=O)O ZINC000147394933 BD For-Sale Anodyne GZMB 41 34 CCCc1c(NC)ncnc1Oc1ccc2c(c1)OCO2 ZINC000147394954 CF For-Sale Anodyne CLK4 49 37 Cc1ncoc1-c1nnc(SCCCN2C[C@@H]3C[C@@]3(c3ccc(OC(F)(F)F)cc3)C2)n1C ZINC000147394959 JI Annotated Anodyne DRD3 23 79 Cc1ncoc1-c1nnc(SCCCN2C[C@@H]3C[C@@]3(c3ccc(OC(F)(F)F)cc3)C2)n1C ZINC000147394959 JI Annotated Anodyne CYP2D6 0 77 Cc1ncoc1-c1nnc(SCCCN2C[C@@H]3C[C@@]3(c3ccc(OC(F)(F)F)cc3)C2)n1C ZINC000147394959 JI Annotated Anodyne CYP1A2 0 83 Cc1ncoc1-c1nnc(SCCCN2C[C@@H]3C[C@@]3(c3ccc(OC(F)(F)F)cc3)C2)n1C ZINC000147394959 JI Annotated Anodyne CYP2C19 0 75 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCCc3ccccc3)c2)c1 ZINC000147394965 GI On-Demand Bother HRH2 17 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCCc3ccccc3)c2)c1 ZINC000147394965 GI On-Demand Bother MAOB 15 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCCc3ccccc3)c2)c1 ZINC000147394965 GI On-Demand Bother PTGER3 16 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCCc3ccccc3)c2)c1 ZINC000147394965 GI On-Demand Bother MMP13 20 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCCc3ccccc3)c2)c1 ZINC000147394965 GI On-Demand Bother MTNR1B 37 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCCc3ccccc3)c2)c1 ZINC000147394965 GI On-Demand Bother TAAR1 42 56 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCCc3ccccc3)c2)c1 ZINC000147394965 GI On-Demand Bother AKR1C3 24 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCCc3ccccc3)c2)c1 ZINC000147394965 GI On-Demand Bother AKR1C2 41 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCCc3ccccc3)c2)c1 ZINC000147394965 GI On-Demand Bother KCNK3 76 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(OCCc3ccccc3)c2)c1 ZINC000147394965 GI On-Demand Bother KCNK9 59 41 C[C@H](OC[C@@H]1CCCO1)C(=O)NCc1ccccc1Cn1cccn1 ZINC000147394988 EE On-Demand Anodyne PANC 47 37 CCCCCCCCNS(=O)(=O)c1cnn(CCCO)c1 ZINC000147395000 DD For-Sale Mild ASAH1 67 34 C[C@H]1OCC[C@@H]1Nc1ccc(N2CCOCC2)cc1 ZINC000147395078 CE On-Demand Anodyne AKR1C3 0 40 CCNc1nc(C)nc(Oc2ccc3c(c2)OCO3)c1C ZINC000147395167 CG For-Sale Anodyne CLK4 48 34 CCNc1nc(C)nc(Oc2ccc3c(c2)OCO3)c1C ZINC000147395167 CG For-Sale Anodyne DYRK2 48 37 C[C@@H](CC(=O)NN1CCCCC1)[C@@H]1CCCNC1 ZINC000147395183 CD For-Sale Anodyne CPN1 0 43 C[C@@H](OC[C@@H]1CCCO1)C(=O)NCc1ccccc1Cn1cccn1 ZINC000147395195 EE On-Demand Anodyne PANC 47 37 CCCCCCCCNS(=O)(=O)c1ccccc1CO ZINC000147395220 CF For-Sale Mild ALOX15 41 45 CCCCCCCCNS(=O)(=O)c1ccccc1CO ZINC000147395220 CF For-Sale Mild ASAH1 52 35 CCC[C@@H](NC(N)=O)C(=O)Nc1ncc(Cc2ccc(C)c(C)c2)s1 ZINC000147395294 FG On-Demand Anodyne SCD1 38 40 C[C@@H]1OCC[C@@H]1Nc1ccc(N2CCOCC2)cc1 ZINC000147395312 CE On-Demand Anodyne AKR1C3 0 40 Cc1nc(OCc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147395384 CE For-Sale Anodyne EDNRB 48 43 Cc1nc(OCc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147395384 CE For-Sale Anodyne EDNRA 53 43 Cc1nc(OCc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147395384 CE For-Sale Anodyne BMP1 49 38 Cc1nc(OCc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147395384 CE For-Sale Anodyne NOS2 90 33 Cc1nc(OCc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147395384 CE For-Sale Anodyne SSTR3 91 32 Cc1nc(OCc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147395384 CE For-Sale Anodyne SLC5A5 0 42 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(Cl)cc1[N+](=O)[O-] ZINC000147395386 HI On-Demand Bother F10 17 50 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(Cl)cc1[N+](=O)[O-] ZINC000147395386 HI On-Demand Bother KCNMA1 41 36 Cc1cc(OCCN2CCOCC2)cc(C)c1S(N)(=O)=O ZINC000147395390 DC For-Sale Anodyne LTA4H 26 44 Cc1cc(OCCN2CCOCC2)cc(C)c1S(N)(=O)=O ZINC000147395390 DC For-Sale Anodyne THRB 0 52 C[C@H](OC[C@H]1CCCO1)C(=O)NCc1ccccc1Cn1cccn1 ZINC000147395404 EE On-Demand Anodyne PANC 47 37 C[C@H](CC(=O)NN1CCCCC1)[C@@H]1CCCNC1 ZINC000147395411 CD For-Sale Anodyne CPN1 0 43 CCOC(=O)[C@H]1CCCN(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)C1 ZINC000147395433 HD On-Demand Anodyne NOS2 65 34 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild CA2 24 45 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild TBXA2R 47 36 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild TBXAS1 40 37 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild CA1 22 45 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild CPT1A 25 40 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild S1PR4 37 40 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild ALOX15B 0 43 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild S1PR2 64 43 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild ALOX15 79 57 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild S1PR1 16 40 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild CA12 15 46 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild TPSAB1 15 40 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild CA9 19 46 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild CA 0 46 CCCCCCCCNS(=O)(=O)c1ccc(CCO)cc1 ZINC000147395434 DF For-Sale Mild A6YCJ1_9METZ 23 44 C[C@@]1(O)O[C@H](CO)[C@H](O)[C@@H]1O ZINC000147395437 AA For-Sale Anodyne PYGL 24 41 CC(C)CCCCNCc1ccc2c(c1)OCCCO2 ZINC000147395580 CH For-Sale Anodyne NOS2 17 43 CC(C)CCCCNCc1ccc2c(c1)OCCCO2 ZINC000147395580 CH For-Sale Anodyne LEF 60 35 O=S(=O)(c1ccccc1C(F)(F)F)N1CCCC[C@@H]1CBr ZINC000147395592 GH For-Sale Reactive RBP4 40 35 O=S(=O)(c1ccccc1C(F)(F)F)N1CCCC[C@@H]1CBr ZINC000147395592 GH For-Sale Reactive SFRP1 122 37 O=S(=O)(c1ccccc1C(F)(F)F)N1CCCC[C@@H]1CBr ZINC000147395592 GH For-Sale Reactive WNT3 86 35 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(N)c([N+](=O)[O-])c1 ZINC000147395602 GG On-Demand Bother SLC9A1 42 38 Cc1c(CN2CCSCC2)cccc1NC(=O)c1ccc(N)c([N+](=O)[O-])c1 ZINC000147395602 GG On-Demand Bother MRGPRX1 42 39 C[C@@H](OC[C@H]1CCCO1)C(=O)NCc1ccccc1Cn1cccn1 ZINC000147395619 EE On-Demand Anodyne PANC 47 37 C[C@@H](CC(=O)NN1CCCCC1)[C@H]1CCCNC1 ZINC000147395628 CD For-Sale Anodyne CPN1 0 43 Cc1cc(OCCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147395645 DD For-Sale Anodyne ACHE 16 41 Cc1cc(OCCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147395645 DD For-Sale Anodyne KCNH2 0 47 Cc1cc(OCCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147395645 DD For-Sale Anodyne LTA4H 30 40 Cc1cc(OCCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147395645 DD For-Sale Anodyne HRH3 88 60 Cc1cc(OCCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147395645 DD For-Sale Anodyne SIGMAR1 16 43 Cc1cc(OCCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147395645 DD For-Sale Anodyne PSMB1 41 37 O=S(=O)(NCc1ccc(-n2ccnc2)c(F)c1)c1ccc(Cl)cc1 ZINC000147395715 FG On-Demand Anodyne TBXA2R 50 38 O=S(=O)(NCc1ccc(-n2ccnc2)c(F)c1)c1ccc(Cl)cc1 ZINC000147395715 FG On-Demand Anodyne TBXAS1 28 46 O=S(=O)(NCc1ccc(-n2ccnc2)c(F)c1)c1ccc(Cl)cc1 ZINC000147395715 FG On-Demand Anodyne CYP17A1 15 40 CC1(C)CN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CCO1 ZINC000147395737 DF On-Demand Anodyne EPHX2 26 44 C[C@H](CC(=O)NN1CCCCC1)[C@H]1CCCNC1 ZINC000147395798 CD For-Sale Anodyne CPN1 0 43 O=S(=O)(c1ccccc1C(F)(F)F)N1CCCC[C@H]1CBr ZINC000147395830 GH For-Sale Reactive RBP4 40 35 O=S(=O)(c1ccccc1C(F)(F)F)N1CCCC[C@H]1CBr ZINC000147395830 GH For-Sale Reactive SFRP1 122 37 O=S(=O)(c1ccccc1C(F)(F)F)N1CCCC[C@H]1CBr ZINC000147395830 GH For-Sale Reactive WNT3 86 35 Cc1c(C(=O)NCC2(C(=O)O)CCC2)cnn1C ZINC000147395919 CC On-Demand Anodyne HCN1 52 32 Cc1c(C(=O)NCC2(C(=O)O)CCC2)cnn1C ZINC000147395919 CC On-Demand Anodyne HCN4 50 32 NC(=O)c1ccc(OCC(=O)N2CCC(C(=O)Nc3nccs3)CC2)cc1 ZINC000147395939 GD On-Demand Anodyne MAP1 112 41 NC(=O)c1ccc(OCC(=O)N2CCC(C(=O)Nc3nccs3)CC2)cc1 ZINC000147395939 GD On-Demand Anodyne CPT1A 60 43 NC(=O)c1ccc(OCC(=O)N2CCC(C(=O)Nc3nccs3)CC2)cc1 ZINC000147395939 GD On-Demand Anodyne GCK 23 40 O=C(Nc1cc(Br)cc(C(=O)O)c1)NC1CCOCC1 ZINC000147395943 EE For-Sale Anodyne EPHX2 44 40 CCS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3ccc(F)cc3)no2)CC1 ZINC000147396010 GF Annotated Anodyne NPY2R 0 50 COc1ccc(C(=O)NN2CCCCC2)c(N)c1 ZINC000147396033 BD For-Sale Anodyne DRD4 40 31 COc1ccc(C(=O)NN2CCCCC2)c(N)c1 ZINC000147396033 BD For-Sale Anodyne AKR1C2 53 39 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1ccccc1Cn1cccn1 ZINC000147396053 FH On-Demand Anodyne ANPEP 20 42 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1ccccc1Cn1cccn1 ZINC000147396053 FH On-Demand Anodyne AMP1_PLAFQ 44 33 C[C@@H](Cc1cccc(F)c1)C(=O)NCc1ccccc1Cn1cccn1 ZINC000147396053 FH On-Demand Anodyne CARM1 78 33 O=C(Nc1cc(Cl)cc(C(=O)O)c1)NC1CCOCC1 ZINC000147396155 CE On-Demand Anodyne EPHX2 47 51 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne HTR4 39 40 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne CHRM5 19 41 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne GRIN2B 57 40 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne MMP13 30 46 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne CTSK 25 43 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne CAPNS1 67 36 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne MMP2 24 48 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne MMP3 30 48 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne TGM1 25 44 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne CAPN1 81 40 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne CAPN2 89 40 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne EPHX2 24 43 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne TGM2 80 53 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne MMP1 26 48 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne NPR 55 33 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne F13A1 83 53 C[C@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396164 HF On-Demand Anodyne NAMPT 32 41 O=C(NCC[C@H](O)CO)[C@@H]1N[C@H](CCc2ccsc2)[C@]2(C(=O)Nc3cc(Cl)c(F)cc32)[C@H]1c1cccc(Cl)c1 ZINC000147396167 KI Annotated Anodyne MDM2 57 74 O=C(Nc1ccc(-c2cnco2)cc1)c1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147396168 HH On-Demand Anodyne LPL 46 37 O=C(Nc1ccc(-c2cnco2)cc1)c1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147396168 HH On-Demand Anodyne CHRNA7 25 44 O=C(Nc1ccc(-c2cnco2)cc1)c1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147396168 HH On-Demand Anodyne F13A1 42 38 O=C(Nc1ccc(-c2cnco2)cc1)c1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147396168 HH On-Demand Anodyne NR2E3 68 36 O=C(Nc1ccc(-c2cnco2)cc1)c1ccccc1S(=O)(=O)N1CCCCC1 ZINC000147396168 HH On-Demand Anodyne SMO 23 42 Cc1nc(Oc2ccccc2C(N)=O)ccc1C(=O)O ZINC000147396184 CD For-Sale Anodyne ALS 45 33 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild CNR1 32 75 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild CNR2 20 52 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild PLA2G4C 0 50 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild FABP4 23 63 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild TRPV1 0 55 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild LPAR1 41 46 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild LPAR2 20 45 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild PRKCE 25 45 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild PLA2G4B 80 50 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild FAAH 33 60 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild PRKCA 35 56 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild EPHX2 36 55 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild LPAR3 81 52 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild FABP3 60 63 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild FABP5 17 54 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild LOX1.1 16 63 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild MGLL 0 58 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild TLR2 0 47 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild ENPP2 34 52 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild FABP1 18 54 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild LPAR4 0 52 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild LPAR5 0 52 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild ACAT 0 46 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild FBA1 29 45 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild NOD1 47 43 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild OXER1 21 44 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild CQSS 55 35 CCCCC/C=C\C/C=C\CCCCCCCC(=O)OCCCCCCCCCCCCC ZINC000147396188 JK Annotated Mild LPAR6 0 52 C[C@H](Cc1cccc(F)c1)C(=O)NCc1ccccc1Cn1cccn1 ZINC000147396268 FH On-Demand Anodyne ANPEP 20 42 C[C@H](Cc1cccc(F)c1)C(=O)NCc1ccccc1Cn1cccn1 ZINC000147396268 FH On-Demand Anodyne AMP1_PLAFQ 44 33 C[C@H](Cc1cccc(F)c1)C(=O)NCc1ccccc1Cn1cccn1 ZINC000147396268 FH On-Demand Anodyne CARM1 78 33 CC(C)CCCCNC1CCN(c2ccncc2)CC1 ZINC000147396270 CG For-Sale Anodyne HRH4 37 44 O=S(=O)(NCc1ccc(-n2ccnc2)c(F)c1)c1ccc2ccccc2c1 ZINC000147396329 GH On-Demand Anodyne NPY1R 21 45 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne HTR4 39 40 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne CHRM5 19 41 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne GRIN2B 57 40 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne MMP13 30 46 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne CTSK 25 43 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne CAPNS1 67 36 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne MMP2 24 48 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne MMP3 30 48 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne TGM1 25 44 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne CAPN1 81 40 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne CAPN2 89 40 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne EPHX2 24 43 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne TGM2 80 53 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne MMP1 26 48 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne NPR 55 33 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne F13A1 83 53 C[C@@H](OCc1ccccc1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147396366 HF On-Demand Anodyne NAMPT 32 41 Cc1nc(Oc2ccc(Cl)cc2[N+](=O)[O-])ccc1C(=O)O ZINC000147396444 DG For-Sale Bother S1PR4 25 43 Cc1nc(Oc2ccc(Cl)cc2[N+](=O)[O-])ccc1C(=O)O ZINC000147396444 DG For-Sale Bother ENR 0 43 CCS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3ccccc3)no2)CC1 ZINC000147396451 FF Annotated Anodyne NPY2R 30 46 COc1cccc(-c2nnnn2C2(C(=O)O)CCC2)c1 ZINC000147396496 CD For-Sale Anodyne DHODH 18 40 CC[C@H](CNS(=O)(=O)c1ccccc1OC)CC(=O)O ZINC000147396497 DD On-Demand Anodyne ITGAV 34 49 CCCCCCCCNS(=O)(=O)c1cc(C)c(CO)s1 ZINC000147396555 DG For-Sale Mild FBP1 0 44 CNc1cn2ccnc2c(Oc2ccc3c(c2)CCC3)n1 ZINC000147396618 CG For-Sale Anodyne HIVRT 0 41 Cc1nc(Oc2ccc(C(N)=O)cc2)ccc1C(=O)O ZINC000147396676 CD For-Sale Anodyne TRY1_BOVIN 24 41 COCc1nc(C(=O)N2CCC[C@@H]2c2cc(OC)ccc2OC)cs1 ZINC000147396733 FG On-Demand Anodyne CPT1A 24 40 COCc1nc(C(=O)N2CCC[C@@H]2c2cc(OC)ccc2OC)cs1 ZINC000147396733 FG On-Demand Anodyne TRPC6 55 39 COCc1nc(C(=O)N2CCC[C@@H]2c2cc(OC)ccc2OC)cs1 ZINC000147396733 FG On-Demand Anodyne TRPC3 44 39 O=S1(=O)N=C(N(CCBr)C2CCCCC2)c2ccccc21 ZINC000147396735 FG For-Sale Reactive KCNA3 47 60 CC[C@@H](CNS(=O)(=O)c1ccccc1OC)CC(=O)O ZINC000147396750 DD On-Demand Anodyne ITGAV 34 49 CCOc1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147396865 GF On-Demand Anodyne ALPI 15 42 Cc1nc(Oc2cccc(C(N)=O)c2)ccc1C(=O)O ZINC000147396898 CD For-Sale Anodyne F10 17 65 Cc1nc(Oc2cccc(C(N)=O)c2)ccc1C(=O)O ZINC000147396898 CD For-Sale Anodyne TRY1_BOVIN 52 59 Cc1nc(Oc2cccc(C(N)=O)c2)ccc1C(=O)O ZINC000147396898 CD For-Sale Anodyne CHEK2 22 43 Cc1nc(Oc2cccc(C(N)=O)c2)ccc1C(=O)O ZINC000147396898 CD For-Sale Anodyne ALS 43 31 Cc1nc(Oc2cccc(C(N)=O)c2)ccc1C(=O)O ZINC000147396898 CD For-Sale Anodyne FABH 0 40 Cc1nc(Oc2cccc(C(N)=O)c2)ccc1C(=O)O ZINC000147396898 CD For-Sale Anodyne AKR1C3 17 43 COc1ccc2nc(CCCl)n(CCNC(N)=O)c2n1 ZINC000147396905 CC For-Sale Reactive PDE10A 25 45 COCc1nc(C(=O)N2CCC[C@H]2c2cc(OC)ccc2OC)cs1 ZINC000147396939 FG On-Demand Anodyne CPT1A 24 40 COCc1nc(C(=O)N2CCC[C@H]2c2cc(OC)ccc2OC)cs1 ZINC000147396939 FG On-Demand Anodyne TRPC6 55 39 COCc1nc(C(=O)N2CCC[C@H]2c2cc(OC)ccc2OC)cs1 ZINC000147396939 FG On-Demand Anodyne TRPC3 44 39 COc1ccccc1[C@@H](NC(=O)N(C)Cc1cscn1)c1nccn1C ZINC000147397041 FF On-Demand Anodyne CYP3A4 18 40 COCCNC(=O)COc1cc(C)c(S(N)(=O)=O)c(C)c1 ZINC000147397061 DC For-Sale Anodyne CA9 17 40 COCCNC(=O)COc1cc(C)c(S(N)(=O)=O)c(C)c1 ZINC000147397061 DC For-Sale Anodyne CAN2 0 40 Cc1ccc(Oc2ccc(NC(=O)N[C@@H]3CCCN(S(C)(=O)=O)C3)cn2)cc1 ZINC000147397118 HF On-Demand Anodyne EPHX2 44 45 COc1ccc2nc([C@H](C)Cl)n(CCNC(N)=O)c2n1 ZINC000147397127 CD For-Sale Reactive PDE10A 34 40 COc1ccc2nc([C@H](C)Cl)n(CCNC(N)=O)c2n1 ZINC000147397127 CD For-Sale Reactive PROKR1 41 32 COc1cccc(COc2ccc(C(=O)O)c(C)n2)c1 ZINC000147397164 CF For-Sale Anodyne PLG 0 40 COc1cccc(COc2ccc(C(=O)O)c(C)n2)c1 ZINC000147397164 CF For-Sale Anodyne MAOB 24 44 COc1cccc(COc2ccc(C(=O)O)c(C)n2)c1 ZINC000147397164 CF For-Sale Anodyne GRM2 20 41 COc1cccc(COc2ccc(C(=O)O)c(C)n2)c1 ZINC000147397164 CF For-Sale Anodyne MTNR1A 32 41 COc1cccc(COc2ccc(C(=O)O)c(C)n2)c1 ZINC000147397164 CF For-Sale Anodyne MTNR1B 35 40 COc1cccc(COc2ccc(C(=O)O)c(C)n2)c1 ZINC000147397164 CF For-Sale Anodyne ALS 84 34 COc1cccc(COc2ccc(C(=O)O)c(C)n2)c1 ZINC000147397164 CF For-Sale Anodyne FFAR1 63 47 COc1cccc(COc2ccc(C(=O)O)c(C)n2)c1 ZINC000147397164 CF For-Sale Anodyne AKR1C3 24 42 COc1cccc(COc2ccc(C(=O)O)c(C)n2)c1 ZINC000147397164 CF For-Sale Anodyne AKR1C2 53 39 COc1cccc(COc2ccc(C(=O)O)c(C)n2)c1 ZINC000147397164 CF For-Sale Anodyne SLC5A5 0 40 COc1ccccc1[C@H](NC(=O)N(C)Cc1cscn1)c1nccn1C ZINC000147397192 FF On-Demand Anodyne CYP3A4 18 40 COc1ccc(C(=O)/C=C\c2ccc(OC)c(F)c2)cc1 ZINC000147397217 CH On-Demand Mild MAOB 0 64 COc1ccc(C(=O)/C=C\c2ccc(OC)c(F)c2)cc1 ZINC000147397217 CH On-Demand Mild PTGS2 0 42 CC[C@@H]1COCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147397241 DF On-Demand Anodyne CACNA1I 44 32 CCCCCCCCNS(=O)(=O)CCCNCCC ZINC000147397293 CF For-Sale Mild ADH1A 0 41 CCCCCCCCNS(=O)(=O)CCCNCCC ZINC000147397293 CF For-Sale Mild ADH7 0 41 CCCCCCCCNS(=O)(=O)CCCNCCC ZINC000147397293 CF For-Sale Mild S1PR3 22 46 CCCCCCCCNS(=O)(=O)CCCNCCC ZINC000147397293 CF For-Sale Mild S1PR2 37 46 CCCCCCCCNS(=O)(=O)CCCNCCC ZINC000147397293 CF For-Sale Mild ADH1B 0 41 CCCCCCCCNS(=O)(=O)CCCNCCC ZINC000147397293 CF For-Sale Mild RELA 31 71 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@@H]1CBr ZINC000147397296 GH For-Sale Reactive CASP3 94 38 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@@H]1CBr ZINC000147397296 GH For-Sale Reactive CACNA1B 59 41 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@@H]1CBr ZINC000147397296 GH For-Sale Reactive BDKRB1 32 52 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@@H]1CBr ZINC000147397296 GH For-Sale Reactive CASP7 106 41 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@@H]1CBr ZINC000147397296 GH For-Sale Reactive SFRP1 52 32 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@@H]1CBr ZINC000147397296 GH For-Sale Reactive WNT3 40 31 COc1ccc2nc([C@@H](C)Cl)n(CCNC(N)=O)c2n1 ZINC000147397325 CD For-Sale Reactive PDE10A 34 40 COc1ccc2nc([C@@H](C)Cl)n(CCNC(N)=O)c2n1 ZINC000147397325 CD For-Sale Reactive PROKR1 41 32 Cc1ccc(Oc2ccc(NC(=O)N[C@H]3CCCN(S(C)(=O)=O)C3)cn2)cc1 ZINC000147397336 HF On-Demand Anodyne EPHX2 44 45 C[C@H](Cl)c1nc2ccccc2n1-c1ccc(Cl)cc1Br ZINC000147397412 FK For-Sale Reactive ALOX5AP 26 40 CC[C@H]1COCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147397420 DF On-Demand Anodyne CACNA1I 44 32 Cc1nc(Oc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147397423 CH For-Sale Anodyne TRY1_BOVIN 28 42 Cc1nc(Oc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147397423 CH For-Sale Anodyne SORT1 25 45 Cc1nc(Oc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147397423 CH For-Sale Anodyne ALS 44 31 Cc1nc(Oc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147397423 CH For-Sale Anodyne AKR1C2 21 45 Cc1nc(Oc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147397423 CH For-Sale Anodyne TRPM4 0 40 Cc1nc(Oc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147397423 CH For-Sale Anodyne HAO2 17 40 Cc1nc(Oc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147397423 CH For-Sale Anodyne PDS 42 37 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne MME 43 40 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne ANPEP 43 40 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne PAPA1_CARPA 51 38 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne CTSK 19 40 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne CTSL 23 43 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne SLC15A1 48 33 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne CA5B 32 40 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne CA5A 37 40 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne SLC1A6 50 33 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne PAM 0 44 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne SLC1A7 50 33 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne CPA3 53 32 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne POL 0 49 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne NPR 41 33 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne AMP1_PLAFQ 47 36 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne HDA106 0 40 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne PLC 47 32 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne Q9JN24_ECOLX 0 43 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne PDS 48 36 COC(=O)NC(=O)Cc1ccccc1 ZINC000147397454 AD For-Sale Anodyne H9B8T9_CAPHI 24 53 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@H]1CBr ZINC000147397495 GH For-Sale Reactive CASP3 94 38 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@H]1CBr ZINC000147397495 GH For-Sale Reactive CACNA1B 59 41 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@H]1CBr ZINC000147397495 GH For-Sale Reactive BDKRB1 32 52 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@H]1CBr ZINC000147397495 GH For-Sale Reactive CASP7 106 41 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@H]1CBr ZINC000147397495 GH For-Sale Reactive SFRP1 52 32 O=S(=O)(c1cccc(C(F)(F)F)c1)N1CCCC[C@H]1CBr ZINC000147397495 GH For-Sale Reactive WNT3 40 31 N#Cc1cccc(S(=O)(=O)CCN2CCC(O)CC2)c1 ZINC000147397516 CC On-Demand Mild MEN1 50 35 CCCc1ccc(S(=O)(=O)N2CC[C@H](N)[C@H](CC)C2)cc1 ZINC000147397585 DE On-Demand Anodyne MMP7 23 42 C[C@@H](Cl)c1nc2ccccc2n1-c1ccc(Cl)cc1Br ZINC000147397636 FK For-Sale Reactive ALOX5AP 26 40 Cc1nc(Oc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147397675 CF For-Sale Anodyne EDNRB 67 39 Cc1nc(Oc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147397675 CF For-Sale Anodyne EDNRA 65 39 Cc1nc(Oc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147397675 CF For-Sale Anodyne BMP1 41 37 COC(=O)[C@@H]1CCCN(C(=O)c2c(Cl)cccc2Cl)C1 ZINC000147397738 DG On-Demand Anodyne SLC6A1 47 36 COC(=O)[C@@H]1CCCN(C(=O)c2c(Cl)cccc2Cl)C1 ZINC000147397738 DG On-Demand Anodyne CCR5 15 41 COC(=O)[C@@H]1CCCN(C(=O)c2c(Cl)cccc2Cl)C1 ZINC000147397738 DG On-Demand Anodyne PREP 28 45 COC(=O)[C@@H]1CCCN(C(=O)c2c(Cl)cccc2Cl)C1 ZINC000147397738 DG On-Demand Anodyne RHOA 0 43 COC(=O)[C@@H]1CCCN(C(=O)c2c(Cl)cccc2Cl)C1 ZINC000147397738 DG On-Demand Anodyne L3MBTL3 52 36 CCCc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147397785 FH For-Sale Reactive FKBP1A 32 46 CCCc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147397785 FH For-Sale Reactive CASP3 87 40 CCCc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147397785 FH For-Sale Reactive MMP13 19 41 CCCc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147397785 FH For-Sale Reactive MMP3 16 40 CCCc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147397785 FH For-Sale Reactive CASP7 104 40 CCCc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147397785 FH For-Sale Reactive MMP7 30 47 CCCc1ccc(S(=O)(=O)N2CCCC[C@@H]2CBr)cc1 ZINC000147397785 FH For-Sale Reactive AKR1C3 0 42 CCCc1ccc(S(=O)(=O)N2CC[C@@H](N)[C@H](CC)C2)cc1 ZINC000147397829 DE On-Demand Anodyne MMP7 23 42 COc1ccc(COc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147397919 CF For-Sale Anodyne PPARG 41 32 COc1ccc(COc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147397919 CF For-Sale Anodyne PPARA 40 32 COc1ccc(COc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147397919 CF For-Sale Anodyne P2RX1 23 44 COc1ccc(COc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147397919 CF For-Sale Anodyne POBA 0 40 COc1ccc(COc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147397919 CF For-Sale Anodyne FFAR1 34 44 COc1ccc(COc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147397919 CF For-Sale Anodyne AKR1C3 18 40 COc1ccc(COc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147397919 CF For-Sale Anodyne AKR1C2 52 40 COC(=O)[C@H]1CCCN(C(=O)c2c(Cl)cccc2Cl)C1 ZINC000147397957 DG On-Demand Anodyne SLC6A1 47 36 COC(=O)[C@H]1CCCN(C(=O)c2c(Cl)cccc2Cl)C1 ZINC000147397957 DG On-Demand Anodyne CCR5 15 41 COC(=O)[C@H]1CCCN(C(=O)c2c(Cl)cccc2Cl)C1 ZINC000147397957 DG On-Demand Anodyne PREP 28 45 COC(=O)[C@H]1CCCN(C(=O)c2c(Cl)cccc2Cl)C1 ZINC000147397957 DG On-Demand Anodyne RHOA 0 43 COC(=O)[C@H]1CCCN(C(=O)c2c(Cl)cccc2Cl)C1 ZINC000147397957 DG On-Demand Anodyne L3MBTL3 52 36 CCCCCCCCNS(=O)(=O)c1cc(CN)ccc1F ZINC000147397964 DF For-Sale Mild ASAH1 55 31 Cc1cc(OCCn2ccnc2)cc(C)c1S(N)(=O)=O ZINC000147398010 CD For-Sale Anodyne TBXAS1 39 52 Cc1cc(OCCn2ccnc2)cc(C)c1S(N)(=O)=O ZINC000147398010 CD For-Sale Anodyne HMOX2 19 40 CCCc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147398019 FH For-Sale Reactive FKBP1A 32 46 CCCc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147398019 FH For-Sale Reactive CASP3 87 40 CCCc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147398019 FH For-Sale Reactive MMP13 19 41 CCCc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147398019 FH For-Sale Reactive MMP3 16 40 CCCc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147398019 FH For-Sale Reactive CASP7 104 40 CCCc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147398019 FH For-Sale Reactive MMP7 30 47 CCCc1ccc(S(=O)(=O)N2CCCC[C@H]2CBr)cc1 ZINC000147398019 FH For-Sale Reactive AKR1C3 0 42 Cc1nc(-c2ccc(NC(=O)C(=O)NCC(C)(C)N3CCC[C@H](C)C3)cc2)cs1 ZINC000147398196 HH On-Demand Anodyne MTOR 48 35 CC[C@H](CNS(=O)(=O)c1ccc(C)c(F)c1)CC(=O)O ZINC000147398211 DD On-Demand Anodyne TBXA2R 42 34 CC[C@H](CNS(=O)(=O)c1ccc(C)c(F)c1)CC(=O)O ZINC000147398211 DD On-Demand Anodyne LEF 62 43 CC(C)S(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3ccccc3)no2)CC1 ZINC000147398232 GG Annotated Anodyne NPY5R 22 44 CCOC[C@H](C)NC(=O)Nc1ccc(Oc2ccc(C)cc2)nc1 ZINC000147398282 EH On-Demand Anodyne ACACA 76 44 CCOC[C@H](C)NC(=O)Nc1ccc(Oc2ccc(C)cc2)nc1 ZINC000147398282 EH On-Demand Anodyne ACACB 43 44 OCCNc1ccc(-c2nc(-c3cncs3)no2)cc1 ZINC000147398302 CE For-Sale Anodyne CD38 26 43 Cn1ccc(NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147398306 CE For-Sale Anodyne PPIA 15 42 O=C(NN1CCCCC1)[C@H]1NCCc2ccccc21 ZINC000147398365 CD For-Sale Anodyne PRCP 48 41 CC[C@@H](CNS(=O)(=O)c1ccc(C)c(F)c1)CC(=O)O ZINC000147398393 DD On-Demand Anodyne TBXA2R 42 34 CC[C@@H](CNS(=O)(=O)c1ccc(C)c(F)c1)CC(=O)O ZINC000147398393 DD On-Demand Anodyne LEF 62 43 Cc1nc(Oc2cccc3cccnc23)ccc1C(=O)O ZINC000147398414 CG For-Sale Anodyne ALS 47 35 Cc1nc(Oc2cccc3cccnc23)ccc1C(=O)O ZINC000147398414 CG For-Sale Anodyne FTO 0 40 Cc1nc(-c2ccc(NC(=O)C(=O)NCC(C)(C)N3CCC[C@@H](C)C3)cc2)cs1 ZINC000147398422 HH On-Demand Anodyne MTOR 48 35 OCCCN1CC(O)(c2ccccc2)C1 ZINC000147398426 BC On-Demand Anodyne OPRL1 15 43 OCCCN1CC(O)(c2ccccc2)C1 ZINC000147398426 BC On-Demand Anodyne CCR1 46 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398437 EE On-Demand Anodyne PRSS1 15 46 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398437 EE On-Demand Anodyne TRY2_BOVIN 61 35 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398437 EE On-Demand Anodyne HDAC10 45 38 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398437 EE On-Demand Anodyne CCKBR 17 42 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398437 EE On-Demand Anodyne HDAC11 45 38 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398437 EE On-Demand Anodyne ST14 54 39 C[C@H](c1ccccc1)N1CC[C@H](NC(=O)c2ccc3c(c2)COC3)C1 ZINC000147398438 EG On-Demand Anodyne DRD4 16 64 CCC(C)(C)NC(=O)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1 ZINC000147398491 GI On-Demand Anodyne PRNP 48 32 Cc1cc(OCCCn2ccnc2)cc(C)c1S(N)(=O)=O ZINC000147398493 DD For-Sale Anodyne TBXAS1 43 49 Cc1cc(OCCCn2ccnc2)cc(C)c1S(N)(=O)=O ZINC000147398493 DD For-Sale Anodyne HMOX2 50 45 CC(C)c1ccc(-c2nc(=O)n(C(C)C)c3ccccc23)cc1 ZINC000147398537 DJ For-Sale Anodyne CASR 35 57 Cc1noc(C)c1S(=O)(=O)NCc1ccc(-n2ccnc2)c(F)c1 ZINC000147398560 FE On-Demand Anodyne NR3C2 17 53 O=C(NN1CCCCC1)[C@@H]1NCCc2ccccc21 ZINC000147398569 CD For-Sale Anodyne PRCP 48 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398632 EE On-Demand Anodyne PRSS1 15 46 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398632 EE On-Demand Anodyne TRY2_BOVIN 61 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398632 EE On-Demand Anodyne CCKAR 30 46 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398632 EE On-Demand Anodyne HDAC10 45 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398632 EE On-Demand Anodyne CCKBR 34 46 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398632 EE On-Demand Anodyne HDAC11 45 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(C(=O)N2CCCC2)c1 ZINC000147398632 EE On-Demand Anodyne ST14 54 39 CC(C)(CO)c1cccc(C#N)c1 ZINC000147398744 AD For-Sale Mild GRM5 18 41 CCCCCCCCNS(=O)(=O)c1ccccc1CNC ZINC000147398817 DG For-Sale Mild LPAR2 41 35 CCCCCCCCNS(=O)(=O)c1ccccc1CNC ZINC000147398817 DG For-Sale Mild S1PR2 56 35 CCCCCCCCNS(=O)(=O)c1ccccc1CNC ZINC000147398817 DG For-Sale Mild ALOX15 32 42 CCCOc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147398879 CH For-Sale Anodyne PPARG 41 36 CCCOc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147398879 CH For-Sale Anodyne PPARA 47 36 CCCOc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147398879 CH For-Sale Anodyne ACACA 47 44 CCCOc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147398879 CH For-Sale Anodyne ACACB 26 44 CCCOc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147398879 CH For-Sale Anodyne PLA2G4B 80 37 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@H]1C[C@H]1c1ccccc1 ZINC000147398953 HI On-Demand Anodyne PTK2 20 40 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@H]1C[C@H]1c1ccccc1 ZINC000147398953 HI On-Demand Anodyne SCN5A 17 40 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@H]1C[C@H]1c1ccccc1 ZINC000147398953 HI On-Demand Anodyne EPHX2 29 50 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@H]1C[C@H]1c1ccccc1 ZINC000147398953 HI On-Demand Anodyne RBP4 45 32 CN1CC[C@H](CNC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147398959 FE For-Sale Anodyne CCR3 46 38 CN1CC[C@H](CNC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147398959 FE For-Sale Anodyne CACNA1I 75 37 Cn1c(CNCC(F)F)nc2ccccc21 ZINC000147399053 BD On-Demand Anodyne GRM2 0 44 CCCCCCCCNS(=O)(=O)N(C)CCCNCC ZINC000147399054 DE For-Sale Mild RELA 18 41 CS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3cccc(F)c3)no2)CC1 ZINC000147399106 FE Annotated Anodyne NPY2R 27 48 CS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3cccc(F)c3)no2)CC1 ZINC000147399106 FE Annotated Anodyne GRM5 0 41 CS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3cccc(F)c3)no2)CC1 ZINC000147399106 FE Annotated Anodyne GPR39 0 40 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne ACE 57 46 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne OPRM1 45 46 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne OPRD1 44 46 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne FOLH1 56 39 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne MME 162 54 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne LTA4H 19 47 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne ANPEP 126 43 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CTSD 17 41 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne FCER2 85 41 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne RNPEP 48 44 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne PFDN6 0 41 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne KLK3 77 38 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CTSB 56 43 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne PAPA1_CARPA 62 40 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CYSP_TRYCR 51 35 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CTSL 51 43 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CPA1 63 39 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne SLC15A1 0 45 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne PGA 45 34 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne F2R 26 40 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne NPFFR2 59 41 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne C3AR1 71 39 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CTRB1 37 44 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CAPNS1 67 37 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne MMP2 42 46 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne MMP3 66 44 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne MMP8 40 45 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne GRIA1 62 43 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne ECE1 18 45 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne HLA-DRB1 74 42 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne PAM 0 43 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne FURIN 68 39 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CTSS 20 40 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne DNPEP 0 53 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CAPN1 97 40 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne MMP9 37 46 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CAPN2 110 40 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne ACE2 62 35 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne LAP3 82 53 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne MMP7 33 41 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne GNPAT 0 40 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CPA3 0 40 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne MMP1 58 42 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne FPR1 71 45 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne CTRB_BOVIN 45 32 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne POL 0 46 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne NPR 92 48 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne AMP1_PLAFQ 68 45 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne HDA106 0 41 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne SIRT1 33 40 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne SLC15A2 0 44 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne KISS1R 74 35 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne POLG_WNV 79 37 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne QRFPR 61 40 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne NPFFR1 83 41 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne TMPRSS6 42 33 CC(C)CCCCNC(=O)[C@H](CN)Cc1ccccc1 ZINC000147399116 CF For-Sale Anodyne VM1B1_BOTAS 0 43 Nc1cc(Oc2ccc3c(c2)CCC3)ncn1 ZINC000147399134 BE For-Sale Anodyne HRH3 15 45 Cc1cc(-c2cnc3c(NCCC(F)(F)F)cc(C(F)(F)c4cccc(F)c4)nn23)ccc1C(=O)NC1CC1 ZINC000147399156 KK For-Sale Anodyne PDE4B 51 32 Cc1cc(-c2cnc3c(NCCC(F)(F)F)cc(C(F)(F)c4cccc(F)c4)nn23)ccc1C(=O)NC1CC1 ZINC000147399156 KK For-Sale Anodyne TTK 17 73 CCc1cc(C(=O)O)c(OC)cc1N ZINC000147399174 AD For-Sale Anodyne HTR4 80 43 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147399180 HI On-Demand Anodyne PTK2 20 40 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147399180 HI On-Demand Anodyne EPHX2 29 50 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147399180 HI On-Demand Anodyne RBP4 45 32 CC[C@@H]1CN(S(=O)(=O)c2ccc(C)c(C)c2)CC[C@@H]1N ZINC000147399185 CE On-Demand Anodyne AKR1C3 0 40 CC[C@H](NC(=O)c1ccc(S(=O)(=O)Nc2nccs2)cc1)c1ccccc1 ZINC000147399220 HH On-Demand Anodyne MAP1 106 39 CC[C@H](NC(=O)c1ccc(S(=O)(=O)Nc2nccs2)cc1)c1ccccc1 ZINC000147399220 HH On-Demand Anodyne TACR3 54 41 CC[C@H](NC(=O)c1ccc(S(=O)(=O)Nc2nccs2)cc1)c1ccccc1 ZINC000147399220 HH On-Demand Anodyne LIMK2 43 34 CN1CC[C@@H](CNC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147399230 FE For-Sale Anodyne CCR3 46 38 CN1CC[C@@H](CNC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147399230 FE For-Sale Anodyne CACNA1I 75 37 COC(=O)[C@@H]1CN(C(=O)C#Cc2ccccc2)CCO1 ZINC000147399273 CC On-Demand Mild GRM5 20 42 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne ACE 57 46 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne OPRM1 45 46 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne OPRD1 44 46 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne FOLH1 56 39 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne MME 162 54 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne LTA4H 19 47 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne ANPEP 126 43 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CTSD 17 41 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne FCER2 85 41 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne RNPEP 48 44 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne PFDN6 0 41 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne KLK3 77 38 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CTSB 56 43 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne PAPA1_CARPA 62 40 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CYSP_TRYCR 51 35 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CTSL 51 43 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CPA1 63 39 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne SLC15A1 0 45 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne PGA 45 34 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne F2R 26 40 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne NPFFR2 59 41 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne C3AR1 71 39 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CTRB1 37 44 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CAPNS1 67 37 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne MMP2 42 46 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne MMP3 66 44 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne MMP8 40 45 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne GRIA1 62 43 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne ECE1 18 45 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne HLA-DRB1 74 42 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne PAM 0 43 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne FURIN 68 39 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CTSS 20 40 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne DNPEP 0 53 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CAPN1 97 40 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne MMP9 37 46 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CAPN2 110 40 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne ACE2 62 35 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne LAP3 82 53 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne MMP7 33 41 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne GNPAT 0 40 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CPA3 0 40 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne MMP1 58 42 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne FPR1 71 45 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne CTRB_BOVIN 45 32 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne POL 0 46 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne NPR 92 48 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne AMP1_PLAFQ 68 45 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne HDA106 0 41 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne SIRT1 33 40 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne SLC15A2 0 44 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne KISS1R 74 35 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne POLG_WNV 79 37 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne QRFPR 61 40 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne NPFFR1 83 41 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne TMPRSS6 42 33 CC(C)CCCCNC(=O)[C@@H](CN)Cc1ccccc1 ZINC000147399301 CF For-Sale Anodyne VM1B1_BOTAS 0 43 CCCCCCCCNS(=O)(=O)CCCNC1CC1 ZINC000147399302 CE For-Sale Mild RELA 23 51 CC(=O)Nc1ccc(CCCN(C)C)cc1 ZINC000147399324 BE For-Sale Anodyne THRA 15 44 CC(=O)Nc1ccc(CCCN(C)C)cc1 ZINC000147399324 BE For-Sale Anodyne INHA 27 46 CC(=O)Nc1ccc(CCCN(C)C)cc1 ZINC000147399324 BE For-Sale Anodyne ALOX15 16 40 CC(=O)Nc1ccc(CCCN(C)C)cc1 ZINC000147399324 BE For-Sale Anodyne SPHK1 21 40 CC(=O)Nc1ccc(CCCN(C)C)cc1 ZINC000147399324 BE For-Sale Anodyne NAMPT 15 46 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(Cl)c1Oc1cccnc1)C2 ZINC000147399361 HJ On-Demand Anodyne ROCK2 37 46 CCC(C)(C)NC(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147399387 HI On-Demand Bother TAAR1 28 46 CCC(C)(C)NC(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147399387 HI On-Demand Bother AKR1C2 47 38 CCC(C)(C)NC(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147399387 HI On-Demand Bother USP7 27 40 CCC(C)(C)NC(=O)c1ccc(NC(=O)c2cc(OC)ccc2[N+](=O)[O-])cc1Cl ZINC000147399387 HI On-Demand Bother USP47 34 40 CC[C@H]1CN(S(=O)(=O)c2ccc(C)c(C)c2)CC[C@@H]1N ZINC000147399416 CE On-Demand Anodyne AKR1C3 0 40 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147399419 HI On-Demand Anodyne PTK2 20 40 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147399419 HI On-Demand Anodyne SCN5A 17 40 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147399419 HI On-Demand Anodyne EPHX2 29 50 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147399419 HI On-Demand Anodyne RBP4 45 32 CCCC[C@H](N)C(=O)NN1[C@@H](C)CCC[C@H]1C ZINC000147399444 BD For-Sale Anodyne DPP7 45 48 CCCC[C@H](N)C(=O)NN1[C@@H](C)CCC[C@H]1C ZINC000147399444 BD For-Sale Anodyne DPP8 37 40 CCCC[C@H](N)C(=O)NN1[C@@H](C)CCC[C@H]1C ZINC000147399444 BD For-Sale Anodyne DPP9 31 40 CN1CC[C@H](CNC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147399477 DE For-Sale Anodyne CACNA1H 28 48 CN1CC[C@H](CNC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147399477 DE For-Sale Anodyne CCR3 40 39 CN1CC[C@H](CNC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147399477 DE For-Sale Anodyne CACNA1I 80 49 COC(=O)[C@H]1CN(C(=O)C#Cc2ccccc2)CCO1 ZINC000147399485 CC On-Demand Mild GRM5 20 42 CCCCCCCCNS(=O)(=O)CCCNCC ZINC000147399550 CE For-Sale Mild RELA 29 66 Cc1cc(OCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147399566 CD For-Sale Anodyne ESR1 70 38 Cc1cc(OCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147399566 CD For-Sale Anodyne ESR2 50 38 Cc1cc(OCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147399566 CD For-Sale Anodyne LTA4H 46 44 Cc1cc(OCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147399566 CD For-Sale Anodyne HRH3 53 51 Cc1cc(OCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147399566 CD For-Sale Anodyne PSMB2 55 43 Cc1cc(OCCN2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147399566 CD For-Sale Anodyne PSMB1 49 43 CCOC(=O)c1ccc(-c2cccc(Cl)n2)cc1 ZINC000147399570 CH For-Sale Anodyne ACR 15 41 CCOC(=O)c1ccc(-c2cccc(Cl)n2)cc1 ZINC000147399570 CH For-Sale Anodyne ADORA3 32 41 CCOC(=O)c1ccc(-c2cccc(Cl)n2)cc1 ZINC000147399570 CH For-Sale Anodyne F2RL3 21 44 C[C@@H](CC(=O)O)CN1C(=O)c2cccnc2C1=O ZINC000147399596 BC For-Sale Anodyne J7HAW4_RAPRA 0 40 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147399603 HF On-Demand Anodyne PLD1 15 41 CC[C@@H](CN)C(=O)NCCCCC(C)C ZINC000147399617 BD For-Sale Anodyne DPP7 18 44 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147399645 HI On-Demand Anodyne PTK2 20 40 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147399645 HI On-Demand Anodyne EPHX2 29 50 O=C(Nc1ccc(N2CCOCC2)cc1C(F)(F)F)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147399645 HI On-Demand Anodyne RBP4 45 32 CCCC[C@@H](N)C(=O)NN1[C@@H](C)CCC[C@H]1C ZINC000147399652 BD For-Sale Anodyne DPP7 45 48 CCCC[C@@H](N)C(=O)NN1[C@@H](C)CCC[C@H]1C ZINC000147399652 BD For-Sale Anodyne DPP8 37 40 CCCC[C@@H](N)C(=O)NN1[C@@H](C)CCC[C@H]1C ZINC000147399652 BD For-Sale Anodyne DPP9 31 40 CC[C@@H]1CN(S(=O)(=O)c2ccc(F)cc2C)CC[C@@H]1N ZINC000147399688 DD On-Demand Anodyne EPHX2 20 50 CN1CC[C@@H](CNC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147399700 DE For-Sale Anodyne CACNA1H 28 48 CN1CC[C@@H](CNC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147399700 DE For-Sale Anodyne CCR3 40 39 CN1CC[C@@H](CNC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147399700 DE For-Sale Anodyne CACNA1I 80 49 CCN1CCN(c2ccc(NC(=O)Nc3cc(C)nn3-c3ccccn3)c(C)c2)CC1 ZINC000147399724 HH On-Demand Anodyne TNF 41 36 CCN1CCN(c2ccc(NC(=O)Nc3cc(C)nn3-c3ccccn3)c(C)c2)CC1 ZINC000147399724 HH On-Demand Anodyne PRNP 40 44 CCCCCCCCNS(=O)(=O)c1ccc(C)c(CN)c1 ZINC000147399744 DG For-Sale Mild ALOX15 52 44 CCCCCCCCNS(=O)(=O)c1ccc(C)c(CN)c1 ZINC000147399744 DG For-Sale Mild RELA 17 40 CC[C@H](CN)C(=O)NCCCCC(C)C ZINC000147399813 BD For-Sale Anodyne DPP7 18 44 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@H]1C[C@@H]1c1cccc(Br)c1 ZINC000147399814 HF On-Demand Anodyne PLD1 15 41 C[C@H](CC(=O)O)CN1C(=O)c2cccnc2C1=O ZINC000147399828 BC For-Sale Anodyne J7HAW4_RAPRA 0 40 O=C(Nc1ccc(-c2cnco2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147399851 FH On-Demand Anodyne DRTS_PLAFK 19 40 O=C(Nc1ccc(-c2cnco2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147399851 FH On-Demand Anodyne NR2E3 60 33 O=C(Nc1ccc(-c2cnco2)cc1)c1cccn(Cc2ccccc2)c1=O ZINC000147399851 FH On-Demand Anodyne SMO 23 42 CCCC[C@H](N)C(=O)NN1[C@@H](C)CCC[C@@H]1C ZINC000147399852 BD For-Sale Anodyne DPP7 45 48 CCCC[C@H](N)C(=O)NN1[C@@H](C)CCC[C@@H]1C ZINC000147399852 BD For-Sale Anodyne DPP8 37 40 CCCC[C@H](N)C(=O)NN1[C@@H](C)CCC[C@@H]1C ZINC000147399852 BD For-Sale Anodyne DPP9 31 40 CCO[C@@H]1CCCN(C(=O)Nc2ccc(N3CCOCC3)cc2C(F)(F)F)C1 ZINC000147399865 HH On-Demand Anodyne RBP4 60 36 CCO[C@@H]1CCCN(C(=O)Nc2ccc(N3CCOCC3)cc2C(F)(F)F)C1 ZINC000147399865 HH On-Demand Anodyne TTK 22 40 CC[C@H]1CN(S(=O)(=O)c2ccc(F)cc2C)CC[C@@H]1N ZINC000147399914 DD On-Demand Anodyne EPHX2 20 50 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne CA2 45 52 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne CA6 21 47 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne CA1 45 52 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne CA7 26 47 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne CA4 34 48 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne CA12 28 47 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne CA9 38 52 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne CAH_METTE 24 47 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne CYNT 19 47 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne NCE103 15 47 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne ALPI 15 46 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne CA15 17 47 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne MTCA1 19 47 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne P96878_MYCTU 24 40 NS(=O)(=O)c1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3)c(F)c2)cc1 ZINC000147400013 HD On-Demand Anodyne A6YCJ1_9METZ 25 47 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@@H]1C[C@H]1c1cccc(Br)c1 ZINC000147400021 HF On-Demand Anodyne PLD1 15 41 O=C(NCC1(C(=O)O)CCC1)c1cccnc1 ZINC000147400045 BD On-Demand Anodyne TBXAS1 48 39 CCO[C@H]1CCCN(C(=O)Nc2ccc(N3CCOCC3)cc2C(F)(F)F)C1 ZINC000147400049 HH On-Demand Anodyne RBP4 60 36 CCO[C@H]1CCCN(C(=O)Nc2ccc(N3CCOCC3)cc2C(F)(F)F)C1 ZINC000147400049 HH On-Demand Anodyne TTK 22 40 CCCOCC(=O)NCc1cccc(Cn2ccnc2)c1 ZINC000147400140 CD On-Demand Anodyne CYP19A1 36 42 CCCOCC(=O)NCc1cccc(Cn2ccnc2)c1 ZINC000147400140 CD On-Demand Anodyne CYP11B1 59 48 CCCOCC(=O)NCc1cccc(Cn2ccnc2)c1 ZINC000147400140 CD On-Demand Anodyne TBXAS1 57 44 CCCOCC(=O)NCc1cccc(Cn2ccnc2)c1 ZINC000147400140 CD On-Demand Anodyne AGTR2 15 48 CCCOCC(=O)NCc1cccc(Cn2ccnc2)c1 ZINC000147400140 CD On-Demand Anodyne CYP11B2 60 48 CCCOCC(=O)NCc1cccc(Cn2ccnc2)c1 ZINC000147400140 CD On-Demand Anodyne NOS2 75 33 CCCOCC(=O)NCc1cccc(Cn2ccnc2)c1 ZINC000147400140 CD On-Demand Anodyne CYP17A1 17 40 CC[C@@H]1CN(S(=O)(=O)c2cc(F)ccc2C)CC[C@@H]1N ZINC000147400160 DD On-Demand Anodyne EPHX2 17 42 CCCCCCCCNS(=O)(=O)c1cc(CNCC)cs1 ZINC000147400171 EG For-Sale Mild LPAR2 52 33 CCCCCCCCNS(=O)(=O)c1cc(CNCC)cs1 ZINC000147400171 EG For-Sale Mild S1PR2 67 33 CCN1CCN(c2ccc(NC(=O)Nc3nc(C)cs3)c(C)c2)CC1 ZINC000147400194 FH On-Demand Anodyne PRNP 29 42 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@H]1C[C@H]1c1cccc(Br)c1 ZINC000147400209 HF On-Demand Anodyne PLD1 15 41 Cc1ccncc1CNCCCCC(C)C ZINC000147400266 BG On-Demand Anodyne FDFT1 0 46 Cc1ccncc1CNCCCCC(C)C ZINC000147400266 BG On-Demand Anodyne GPM3 0 44 Cc1nc(OC/C=C/c2ccccc2)ccc1C(=O)O ZINC000147400274 CG For-Sale Anodyne CACNA1B 55 41 CN(C)C1(Cn2cnc3cc(C(=O)O)ccc32)CCCC1 ZINC000147400297 CF For-Sale Anodyne TBXA2R 18 44 CN(C)C1(Cn2cnc3cc(C(=O)O)ccc32)CCCC1 ZINC000147400297 CF For-Sale Anodyne HPGD 51 47 O=C(/C=C/c1ccccc1)NCC1(C(=O)O)CCC1 ZINC000147400300 CE On-Demand Anodyne HDAC8 52 40 O=C(/C=C/c1ccccc1)NCC1(C(=O)O)CCC1 ZINC000147400300 CE On-Demand Anodyne MMP2 0 50 O=C(/C=C/c1ccccc1)NCC1(C(=O)O)CCC1 ZINC000147400300 CE On-Demand Anodyne HDAC6 39 50 O=C(/C=C/c1ccccc1)NCC1(C(=O)O)CCC1 ZINC000147400300 CE On-Demand Anodyne MMP9 0 43 O=C(/C=C/c1ccccc1)NCC1(C(=O)O)CCC1 ZINC000147400300 CE On-Demand Anodyne MMP1 0 46 O=C(/C=C/c1ccccc1)NCC1(C(=O)O)CCC1 ZINC000147400300 CE On-Demand Anodyne IMA1 0 42 CC[C@H]1CN(S(=O)(=O)c2cc(F)ccc2C)CC[C@@H]1N ZINC000147400352 DD On-Demand Anodyne EPHX2 17 42 O=C1CC(=O)c2cc(O)ccc21 ZINC000147400404 AD In-Stock Clean ESR1 0 41 O=C1CC(=O)c2cc(O)ccc21 ZINC000147400404 AD In-Stock Clean ESR2 0 41 COc1ccc2c(c1)OC[C@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400436 GD On-Demand Anodyne HTR1A 15 45 COc1ccc2c(c1)OC[C@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400436 GD On-Demand Anodyne DRD4 43 35 COc1ccc2c(c1)OC[C@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400436 GD On-Demand Anodyne NQO2 33 41 COc1ccc2c(c1)OC[C@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400436 GD On-Demand Anodyne MTNR1A 76 45 COc1ccc2c(c1)OC[C@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400436 GD On-Demand Anodyne MTNR1B 64 45 COc1ccc2c(c1)OC[C@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400436 GD On-Demand Anodyne ROCK2 30 42 CCCCCCCCNS(=O)(=O)CCCNC ZINC000147400584 CD For-Sale Mild RELA 26 58 COc1ccc2c(c1)OC[C@@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400659 GD On-Demand Anodyne HTR1A 15 45 COc1ccc2c(c1)OC[C@@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400659 GD On-Demand Anodyne DRD4 43 35 COc1ccc2c(c1)OC[C@@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400659 GD On-Demand Anodyne NQO2 33 41 COc1ccc2c(c1)OC[C@@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400659 GD On-Demand Anodyne MTNR1A 76 45 COc1ccc2c(c1)OC[C@@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400659 GD On-Demand Anodyne MTNR1B 64 45 COc1ccc2c(c1)OC[C@@H](C(=O)NCCN1C(=O)c3ccccc3C1=O)C2 ZINC000147400659 GD On-Demand Anodyne ROCK2 30 42 O=c1c(-c2ccc(O)cc2)coc2c([C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c(O[C@@H]3OC[C@@H](O)[C@H](O)[C@H]3O)ccc12 ZINC000147400661 KA Annotated Anodyne ALDH2 98 57 O=c1c(-c2ccc(O)cc2)coc2c([C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c(O[C@@H]3OC[C@@H](O)[C@H](O)[C@H]3O)ccc12 ZINC000147400661 KA Annotated Anodyne IL2 32 49 O=c1c(-c2ccc(O)cc2)coc2c([C@@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@H]3O)c(O[C@@H]3OC[C@@H](O)[C@H](O)[C@H]3O)ccc12 ZINC000147400661 KA Annotated Anodyne FIMH 76 36 CCCCC[C@](C)(O)/C=C/[C@@H]1CC[C@H](O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147400757 FI For-Sale Anodyne PTGFR 55 48 CCCCC[C@](C)(O)/C=C/[C@@H]1CC[C@H](O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147400757 FI For-Sale Anodyne PTGER2 33 43 CCCCC[C@](C)(O)/C=C/[C@@H]1CC[C@H](O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147400757 FI For-Sale Anodyne TBXA2R 21 48 CCCCC[C@](C)(O)/C=C/[C@@H]1CC[C@H](O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147400757 FI For-Sale Anodyne PTGDR 25 47 CCCCC[C@](C)(O)/C=C/[C@@H]1CC[C@H](O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147400757 FI For-Sale Anodyne FABP3 33 40 CCCCC[C@](C)(O)/C=C/[C@@H]1CC[C@H](O)[C@@H]1C/C=C\CCCC(=O)O ZINC000147400757 FI For-Sale Anodyne SLCO2A1 46 47 Cc1ccc(Br)c(C(=O)NCCCOc2ccccc2)c1 ZINC000147400786 EH On-Demand Anodyne DRD4 22 49 Cc1ccc(Br)c(C(=O)NCCCOc2ccccc2)c1 ZINC000147400786 EH On-Demand Anodyne HTR2C 17 40 Cc1ccc(Br)c(C(=O)NCCCOc2ccccc2)c1 ZINC000147400786 EH On-Demand Anodyne DRD3 25 49 Cc1ccc(Br)c(C(=O)NCCCOc2ccccc2)c1 ZINC000147400786 EH On-Demand Anodyne LTA4H 15 40 Cc1ccc(Br)c(C(=O)NCCCOc2ccccc2)c1 ZINC000147400786 EH On-Demand Anodyne CASR 18 42 Cc1ccc(Br)c(C(=O)NCCCOc2ccccc2)c1 ZINC000147400786 EH On-Demand Anodyne MTNR1A 21 40 Cc1ccc(Br)c(C(=O)NCCCOc2ccccc2)c1 ZINC000147400786 EH On-Demand Anodyne MTNR1B 20 40 CCCCCCCCNS(=O)(=O)c1ccc(CNC)cn1 ZINC000147400792 DE For-Sale Mild LPAR2 61 38 CCCCCCCCNS(=O)(=O)c1ccc(CNC)cn1 ZINC000147400792 DE For-Sale Mild S1PR2 77 38 O=C(NCCC1CCCC1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147400797 FH For-Sale Anodyne PRMT3 26 47 O=C(NCCN1C(=O)c2ccccc2C1=O)c1cnn(-c2ccccc2Cl)c1 ZINC000147400860 GF On-Demand Anodyne DRD3 26 41 CCS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3ccc(F)cc3F)no2)CC1 ZINC000147400924 HF Annotated Anodyne NPY2R 0 43 CN(C)C1(Cn2cnc3ccc(C(=O)O)cc32)CCCC1 ZINC000147400925 CF For-Sale Anodyne TBXA2R 18 41 O=C(NCCC1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147401007 DH For-Sale Anodyne CACNA1H 26 41 O=C(NCCC1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147401007 DH For-Sale Anodyne CCR3 37 41 O=C(NCCC1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147401007 DH For-Sale Anodyne CACNA1I 61 42 O=C(NCCC1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147401007 DH For-Sale Anodyne PRMT3 26 47 CCCCCCCCCC[C@@H](CCCCCCCC)COC(=O)[C@H]1CCC(=O)N1 ZINC000147401057 HK For-Sale Mild DAGLA 15 52 Cc1cc(N2CCCC2)ccc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@H](C)C1 ZINC000147401086 HG On-Demand Anodyne HRH3 23 45 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147401090 FF On-Demand Anodyne PLD1 15 41 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147401090 FF On-Demand Anodyne MDM2 47 32 CCCNCCC[C@@H](C)Oc1ccc(Cl)c(F)c1 ZINC000147401096 CI For-Sale Anodyne LEF 41 35 CCC[C@@H](NC(N)=O)C(=O)Nc1ccc(-c2cnco2)cc1 ZINC000147401132 DE On-Demand Anodyne IMPDH2 0 47 CCCCCCCCCC[C@H](CCCCCCCC)COC(=O)[C@H]1CCC(=O)N1 ZINC000147401198 HK For-Sale Mild DAGLA 15 52 Cc1nc(Oc2ccc(C(F)(F)F)cc2)ccc1C(=O)O ZINC000147401221 CH For-Sale Anodyne PPARD 53 41 Cc1nc(Oc2ccc(C(F)(F)F)cc2)ccc1C(=O)O ZINC000147401221 CH For-Sale Anodyne LIPE 26 42 Cc1nc(Oc2ccc(C(F)(F)F)cc2)ccc1C(=O)O ZINC000147401221 CH For-Sale Anodyne SORT1 16 43 O=C(NCC1(C(=O)O)CCC1)c1cccc(F)c1 ZINC000147401255 CD On-Demand Anodyne ELOVL6 0 41 O=C(NCC1(C(=O)O)CCC1)c1cccc(F)c1 ZINC000147401255 CD On-Demand Anodyne KCNK3 71 52 O=C(NCC1(C(=O)O)CCC1)c1cccc(F)c1 ZINC000147401255 CD On-Demand Anodyne KCNK9 29 46 CCCCCCC[C@@H](C)[C@@H](N)c1ccccc1 ZINC000147401269 BJ For-Sale Mild SOAT1 28 42 CCCCCCC[C@@H](C)[C@@H](N)c1ccccc1 ZINC000147401269 BJ For-Sale Mild ACER2 0 43 CCCNCCC[C@H](C)Oc1ccc(Cl)c(F)c1 ZINC000147401270 CI For-Sale Anodyne LEF 41 35 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147401273 FF On-Demand Anodyne PLD1 15 41 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147401273 FF On-Demand Anodyne MDM2 47 32 Cc1cc(N2CCCC2)ccc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@@H](C)C1 ZINC000147401289 HG On-Demand Anodyne HRH3 23 45 CCN1CCN(c2ccc(NC(=O)Nc3nc(C)c(C)s3)c(C)c2)CC1 ZINC000147401300 FH On-Demand Anodyne SLC27A1 29 55 CCCCCCCCNS(=O)(=O)c1c[nH]c(CNC)c1 ZINC000147401301 DE For-Sale Mild ALOX15 40 43 COc1ccc(CNCC(F)F)cc1F ZINC000147401336 BE On-Demand Anodyne SLC6A13 0 40 COc1ccc(CNCC(F)F)cc1F ZINC000147401336 BE On-Demand Anodyne MT-ND1 15 40 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147401460 FF On-Demand Anodyne PLD1 15 41 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147401460 FF On-Demand Anodyne MDM2 47 32 CCCCCCC[C@H](C)[C@@H](N)c1ccccc1 ZINC000147401481 BJ For-Sale Mild SOAT1 28 42 CCCCCCC[C@H](C)[C@@H](N)c1ccccc1 ZINC000147401481 BJ For-Sale Mild ACER2 0 43 O=S(=O)(NC[C@@H]1OCC[C@@]2(S(=O)(=O)c3ccc(Cl)cc3)c3c(F)ccc(F)c3OC[C@@H]12)C(F)(F)F ZINC000147401495 KH Annotated Anodyne PSEN2 126 73 O=S(=O)(NC[C@@H]1OCC[C@@]2(S(=O)(=O)c3ccc(Cl)cc3)c3c(F)ccc(F)c3OC[C@@H]12)C(F)(F)F ZINC000147401495 KH Annotated Anodyne PSEN1 99 73 O=C(N[C@H]1CCC[C@@H]1c1ccccc1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147401510 II On-Demand Anodyne MAP1 52 34 COc1cc(C(F)(F)F)cc(SC)c1C(=O)N[C@@H]1COCC[C@H]1N[C@H](C)C1CC1 ZINC000147401574 IH Annotated Anodyne SLC6A9 0 42 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147401663 FF On-Demand Anodyne PLD1 15 41 O=C(NCCN1C(=O)c2ccccc2C1=O)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147401663 FF On-Demand Anodyne MDM2 47 32 CCCCCCC[C@@H](C)[C@H](N)c1ccccc1 ZINC000147401680 BJ For-Sale Mild SOAT1 28 42 CCCCCCC[C@@H](C)[C@H](N)c1ccccc1 ZINC000147401680 BJ For-Sale Mild ACER2 0 43 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne CA2 36 50 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne KCNQ2 17 50 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne CA1 34 50 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne CA7 16 50 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne CSNK1D 28 45 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne CA5B 50 50 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne CA4 38 48 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne CA5A 57 50 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne SLC1A1 24 43 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne SLC1A3 18 43 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne EPHX2 15 41 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne CA12 22 50 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne SLC1A2 40 43 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne CA9 25 50 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne AKR1C3 18 42 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne IDO1 33 41 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne LIMK2 59 44 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne RORC 40 48 O=C(Cc1cccc(C(F)(F)F)c1)Nc1ccc(S(=O)(=O)Nc2ccccc2)cc1 ZINC000147401717 IJ On-Demand Anodyne NAMPT 27 47 O=C(NCC1(C(=O)O)CCC1)c1cccc(Cl)c1Cl ZINC000147401725 DF On-Demand Anodyne P2RX7 27 57 O=C(NCC1(C(=O)O)CCC1)c1cccc(Cl)c1Cl ZINC000147401725 DF On-Demand Anodyne HCN1 50 31 O=C(NCC1(C(=O)O)CCC1)c1cccc(Cl)c1Cl ZINC000147401725 DF On-Demand Anodyne HCN4 48 31 CCCCCCCCNS(=O)(=O)CCNCCC ZINC000147401727 CE For-Sale Mild S1PR2 31 43 CCCCCCCCNS(=O)(=O)CCNCCC ZINC000147401727 CE For-Sale Mild RELA 28 63 Cc1nc(Oc2cccc(C(C)(C)C)c2)ccc1C(=O)O ZINC000147401738 CI For-Sale Anodyne TRY1_BOVIN 26 44 Cc1nc(Oc2cccc(C(C)(C)C)c2)ccc1C(=O)O ZINC000147401738 CI For-Sale Anodyne ALS 49 32 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@H]1c1cccnc1 ZINC000147401758 FI On-Demand Anodyne CHRNA2 45 46 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@H]1c1cccnc1 ZINC000147401758 FI On-Demand Anodyne CHRNA7 19 46 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@H]1c1cccnc1 ZINC000147401758 FI On-Demand Anodyne GRM5 15 46 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@H]1c1cccnc1 ZINC000147401758 FI On-Demand Anodyne GPBAR1 0 43 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@H]1c1cccnc1 ZINC000147401758 FI On-Demand Anodyne CRTY 0 46 CCN1CCN(c2ccc(NC(=O)Nc3cccc(C(=O)N(C)C)c3)c(C)c2)CC1 ZINC000147401775 HG On-Demand Anodyne DRD4 42 36 CCN1CCN(c2ccc(NC(=O)Nc3cccc(C(=O)N(C)C)c3)c(C)c2)CC1 ZINC000147401775 HG On-Demand Anodyne PRNP 35 41 CN(C)C(=O)NCCn1cnc2cc(C(=O)O)ccc21 ZINC000147401798 CD For-Sale Anodyne TBXA2R 17 42 CN(C)C(=O)NCCn1cnc2cc(C(=O)O)ccc21 ZINC000147401798 CD For-Sale Anodyne NR1I2 46 35 CN(C)C(=O)NCCn1cnc2cc(C(=O)O)ccc21 ZINC000147401798 CD For-Sale Anodyne HPGD 45 47 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne ACE 57 44 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne MME 118 47 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne LTA4H 43 33 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne ANPEP 67 38 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne CTSB 30 44 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne CTSL 21 42 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne CPA1 40 44 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne GRIA1 53 39 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne PAM 0 40 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne FURIN 60 37 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne CAPN1 51 44 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne CAPN2 89 44 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne ACE2 90 44 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne NPR 64 39 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne SLC15A2 0 48 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne BLA1_STEMA 47 38 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne POLG_WNV 50 33 CC[C@H](NC(=O)Cc1ccccc1CN)C(=O)O ZINC000147401834 CC For-Sale Anodyne PDS 47 33 Nc1cc(/C=C/C(=O)O)ccc1O ZINC000147401852 AD For-Sale Anodyne AKR1B1 15 57 Nc1cc(/C=C/C(=O)O)ccc1O ZINC000147401852 AD For-Sale Anodyne CA7 17 60 Nc1cc(/C=C/C(=O)O)ccc1O ZINC000147401852 AD For-Sale Anodyne APP 42 41 Nc1cc(/C=C/C(=O)O)ccc1O ZINC000147401852 AD For-Sale Anodyne MMP2 18 72 Nc1cc(/C=C/C(=O)O)ccc1O ZINC000147401852 AD For-Sale Anodyne MMP9 18 72 Nc1cc(/C=C/C(=O)O)ccc1O ZINC000147401852 AD For-Sale Anodyne MMP1 21 72 Nc1cc(/C=C/C(=O)O)ccc1O ZINC000147401852 AD For-Sale Anodyne AKR1C3 38 47 CCCCCCC[C@H](C)[C@H](N)c1ccccc1 ZINC000147401867 BJ For-Sale Mild SOAT1 28 42 CCCCCCC[C@H](C)[C@H](N)c1ccccc1 ZINC000147401867 BJ For-Sale Mild ACER2 0 43 CS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3ccc(F)cc3)no2)CC1 ZINC000147401868 FE Annotated Anodyne NPY2R 0 59 CCNc1nc(Cl)nc(Oc2ccc3c(c2)CCC3)n1 ZINC000147401876 CG For-Sale Anodyne Q31945_CHEAL 0 40 CCNc1nc(Cl)nc(Oc2ccc3c(c2)CCC3)n1 ZINC000147401876 CG For-Sale Anodyne PPX1 0 43 O=C(NCCN1C(=O)c2ccccc2C1=O)c1ccc2c(c1)COC2 ZINC000147401882 ED On-Demand Anodyne DRD4 42 33 O=C(NCCN1C(=O)c2ccccc2C1=O)c1ccc2c(c1)COC2 ZINC000147401882 ED On-Demand Anodyne PLD2 62 37 Cc1cc(OCCc2cccnc2)cc(C)c1S(N)(=O)=O ZINC000147401896 DD For-Sale Anodyne ISPH 0 40 CC(C)CCCCNC(=O)c1cccc2[nH]ccc12 ZINC000147401913 CH For-Sale Anodyne KISS1R 49 33 CC(C)CCCCNC(=O)c1cccc2[nH]ccc12 ZINC000147401913 CH For-Sale Anodyne HPGDS 15 44 CCCCCCCCNS(=O)(=O)CCCCNCC ZINC000147401929 CF For-Sale Mild ADH1A 0 41 CCCCCCCCNS(=O)(=O)CCCCNCC ZINC000147401929 CF For-Sale Mild ADH7 0 41 CCCCCCCCNS(=O)(=O)CCCCNCC ZINC000147401929 CF For-Sale Mild ADH1B 0 41 CCCCCCCCNS(=O)(=O)CCCCNCC ZINC000147401929 CF For-Sale Mild RELA 31 71 COCCc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147401943 CG For-Sale Anodyne ACACA 0 41 COCCc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147401943 CG For-Sale Anodyne P2RX1 24 42 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@@H]1c1cccnc1 ZINC000147401960 FI On-Demand Anodyne CHRNA2 45 46 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@@H]1c1cccnc1 ZINC000147401960 FI On-Demand Anodyne CHRNA7 19 46 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@@H]1c1cccnc1 ZINC000147401960 FI On-Demand Anodyne GRM5 15 46 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@@H]1c1cccnc1 ZINC000147401960 FI On-Demand Anodyne GPBAR1 0 43 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@@H]1c1cccnc1 ZINC000147401960 FI On-Demand Anodyne CRTY 0 46 CN(C)C(=O)NCCn1cnc2ccc(C(=O)O)cc21 ZINC000147402035 CD For-Sale Anodyne TBXA2R 0 42 CCCCCCCOc1c(F)cc(CNCCC)cc1F ZINC000147402070 CJ For-Sale Mild LPAR2 80 54 CCCCCCCOc1c(F)cc(CNCCC)cc1F ZINC000147402070 CJ For-Sale Mild S1PR3 27 53 CCCCCCCOc1c(F)cc(CNCCC)cc1F ZINC000147402070 CJ For-Sale Mild S1PR2 86 53 CCCCCCCOc1c(F)cc(CNCCC)cc1F ZINC000147402070 CJ For-Sale Mild S1PR1 17 54 CC(C)CNCCCCCOc1ccc(Cl)c(F)c1 ZINC000147402100 CI For-Sale Anodyne DRD4 19 43 CC(=O)/C=C(/C)c1ccc(C(C)(C)C)cc1 ZINC000147402106 BH For-Sale Mild MT-ND1 18 41 CCCCCCCCCOc1ccc(CNCC)nc1 ZINC000147402129 CI For-Sale Mild LPAR2 53 44 CCCCCCCCCOc1ccc(CNCC)nc1 ZINC000147402129 CI For-Sale Mild S1PR3 27 44 CCCCCCCCCOc1ccc(CNCC)nc1 ZINC000147402129 CI For-Sale Mild PLA2G4B 93 40 CCCCCCCCCOc1ccc(CNCC)nc1 ZINC000147402129 CI For-Sale Mild FAAH 23 40 CCCCCCCCCOc1ccc(CNCC)nc1 ZINC000147402129 CI For-Sale Mild S1PR2 52 44 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(C(=O)N3CCOCC3)c1C)C2 ZINC000147402157 HF On-Demand Anodyne ROCK2 29 44 CCCCCCCCNS(=O)(=O)c1c[nH]c(CN)c1 ZINC000147402171 CE For-Sale Mild ALOX15 42 44 CCCCCCCCNS(=O)(=O)c1c[nH]c(CN)c1 ZINC000147402171 CE For-Sale Mild RELA 17 40 Cc1ccc(Br)c(C(=O)N2CCC[C@@H]2c2cccnc2)c1 ZINC000147402177 EI On-Demand Anodyne HCRTR1 41 37 Cc1ccc(Br)c(C(=O)N2CCC[C@@H]2c2cccnc2)c1 ZINC000147402177 EI On-Demand Anodyne CHRNA2 48 49 Cc1ccc(Br)c(C(=O)N2CCC[C@@H]2c2cccnc2)c1 ZINC000147402177 EI On-Demand Anodyne GPBAR1 0 47 Cc1ccc(Br)c(C(=O)N2CCC[C@@H]2c2cccnc2)c1 ZINC000147402177 EI On-Demand Anodyne CRTY 0 49 COc1ccc2cc(/C=C\[C@@H](C)O)ccc2c1 ZINC000147402218 BG For-Sale Anodyne CYP1B1 53 47 COc1ccc2cc(/C=C\[C@@H](C)O)ccc2c1 ZINC000147402218 BG For-Sale Anodyne AHR 39 46 COc1ccc2cc(/C=C\[C@@H](C)O)ccc2c1 ZINC000147402218 BG For-Sale Anodyne CYP11B2 21 45 COc1ccc2cc(/C=C\[C@@H](C)O)ccc2c1 ZINC000147402218 BG For-Sale Anodyne CYP1A1 50 47 COc1ccc2cc(/C=C\[C@@H](C)O)ccc2c1 ZINC000147402218 BG For-Sale Anodyne TUBB1 23 42 COc1ccc2cc(/C=C\[C@@H](C)O)ccc2c1 ZINC000147402218 BG For-Sale Anodyne CYP1A2 15 40 COc1ccc(S(=O)(=O)NCc2ccc(-n3ccnc3C)c(F)c2)cc1F ZINC000147402223 GF On-Demand Anodyne SCN9A 0 47 CCC(CC)(CN)C(=O)Nc1ccc(Br)c(OC)c1 ZINC000147402243 EG On-Demand Anodyne ENPP1 55 32 Cc1nc2cc(C(=O)O)ccc2n1CCNC(=O)N(C)C ZINC000147402268 CD For-Sale Anodyne HPD 41 31 Cc1ccc(Br)c(C(=O)N2CCC[C@H]2c2cccnc2)c1 ZINC000147402360 EI On-Demand Anodyne HCRTR1 41 37 Cc1ccc(Br)c(C(=O)N2CCC[C@H]2c2cccnc2)c1 ZINC000147402360 EI On-Demand Anodyne CHRNA2 48 49 Cc1ccc(Br)c(C(=O)N2CCC[C@H]2c2cccnc2)c1 ZINC000147402360 EI On-Demand Anodyne GPBAR1 0 47 Cc1ccc(Br)c(C(=O)N2CCC[C@H]2c2cccnc2)c1 ZINC000147402360 EI On-Demand Anodyne CRTY 0 49 CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(C)cc(C)c3)[nH]2)cc1 ZINC000147402371 GI Annotated Anodyne ADORA2B 43 39 CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(C)cc(C)c3)[nH]2)cc1 ZINC000147402371 GI Annotated Anodyne SCN10A 40 47 CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(C)cc(C)c3)[nH]2)cc1 ZINC000147402371 GI Annotated Anodyne ENPP1 83 41 CCc1cc(Oc2ccc(C(=O)O)c(C)n2)ccc1Cl ZINC000147402400 CI For-Sale Anodyne AKR1C2 45 33 CCc1cc(Oc2ccc(C(=O)O)c(C)n2)ccc1Cl ZINC000147402400 CI For-Sale Anodyne AKR1C1 41 33 CCCCCCCCNS(=O)(=O)c1cc(CNC)cs1 ZINC000147402401 DG For-Sale Mild S1PR2 44 31 CCCCCCCCCOC(=O)[C@H]1CCC(=O)N1 ZINC000147402417 CF For-Sale Mild LASR 45 34 COc1ccc2cc(/C=C\[C@H](C)O)ccc2c1 ZINC000147402437 BG For-Sale Anodyne CYP1B1 53 47 COc1ccc2cc(/C=C\[C@H](C)O)ccc2c1 ZINC000147402437 BG For-Sale Anodyne AHR 39 46 COc1ccc2cc(/C=C\[C@H](C)O)ccc2c1 ZINC000147402437 BG For-Sale Anodyne CYP11B2 21 45 COc1ccc2cc(/C=C\[C@H](C)O)ccc2c1 ZINC000147402437 BG For-Sale Anodyne CYP1A1 50 47 COc1ccc2cc(/C=C\[C@H](C)O)ccc2c1 ZINC000147402437 BG For-Sale Anodyne TUBB1 23 42 COc1ccc2cc(/C=C\[C@H](C)O)ccc2c1 ZINC000147402437 BG For-Sale Anodyne CYP1A2 15 40 COc1cc(NC(=O)C2(C)CCNCC2)ccc1Br ZINC000147402465 EF For-Sale Anodyne ENPP1 59 32 CCCCCCCCCCCCNC(=O)c1ccc(C(=O)OC)cc1 ZINC000147402475 EK For-Sale Mild FOLH1 30 51 CCCCCCCCCCCCNC(=O)c1ccc(C(=O)OC)cc1 ZINC000147402475 EK For-Sale Mild LPAR2 41 42 CCCCCCCCCCCCNC(=O)c1ccc(C(=O)OC)cc1 ZINC000147402475 EK For-Sale Mild PLA2G4B 51 36 CCCCCCCCCCCCNC(=O)c1ccc(C(=O)OC)cc1 ZINC000147402475 EK For-Sale Mild HDAC6 15 47 CCCCCCCCCCCCNC(=O)c1ccc(C(=O)OC)cc1 ZINC000147402475 EK For-Sale Mild FAAH 18 59 CCCCCCCCCCCCNC(=O)c1ccc(C(=O)OC)cc1 ZINC000147402475 EK For-Sale Mild S1PR2 63 42 CCCCCCCCCCCCNC(=O)c1ccc(C(=O)OC)cc1 ZINC000147402475 EK For-Sale Mild EPHX2 22 43 CCCCCCCCCCCCNC(=O)c1ccc(C(=O)OC)cc1 ZINC000147402475 EK For-Sale Mild HDAC9 18 40 CCCCCCCCCCCCNC(=O)c1ccc(C(=O)OC)cc1 ZINC000147402475 EK For-Sale Mild ASAH1 104 40 CCN1CCN(c2ccc(NC(=O)Nc3ccc(=O)n(C)c3)c(C)c2)CC1 ZINC000147402591 FE On-Demand Anodyne PRNP 29 41 CCCCCCCCNS(=O)(=O)c1cnn(CCN)c1 ZINC000147402609 DD For-Sale Mild ASAH1 60 33 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(OCC(F)(F)F)c2)C1 ZINC000147402610 HG On-Demand Anodyne EPHX2 22 41 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(OCC(F)(F)F)c2)C1 ZINC000147402610 HG On-Demand Anodyne TAAR1 31 43 Cc1cccc(NC(=O)[C@@H]2CCCN(C(=O)CN3CCCCCC3=O)C2)n1 ZINC000147402635 FD On-Demand Anodyne F10 17 42 CC(=O)N1CCCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147402665 FF On-Demand Anodyne L3MBTL1 0 41 CC(=O)N1CCCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147402665 FF On-Demand Anodyne L3MBTL3 54 38 CC(=O)N1CCCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147402665 FF On-Demand Anodyne MBTD1 0 41 CC(=O)N1CCCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147402665 FF On-Demand Anodyne HPGD 41 38 COc1cc(OC)cc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147402693 CF For-Sale Anodyne ALS 84 36 COc1cc(OC)cc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147402693 CF For-Sale Anodyne AKR1C3 23 42 COc1cc(OC)cc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147402693 CF For-Sale Anodyne AKR1C2 55 42 COCCOc1cc(C)ccc1NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147402742 HF On-Demand Bother PYGL 19 45 CCCCC1CCC(NC(=O)Nc2ccc(CC(=O)N(C)C)cc2)CC1 ZINC000147402744 FI On-Demand Anodyne EPHX2 49 43 O=C(NCCCC(F)(F)F)c1cccc2[nH]ccc12 ZINC000147402828 CG On-Demand Anodyne HPGDS 18 42 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(OCC(F)(F)F)c2)C1 ZINC000147402830 HG On-Demand Anodyne EPHX2 22 41 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(OCC(F)(F)F)c2)C1 ZINC000147402830 HG On-Demand Anodyne TAAR1 31 43 Cc1cccc(NC(=O)[C@H]2CCCN(C(=O)CN3CCCCCC3=O)C2)n1 ZINC000147402843 FD On-Demand Anodyne F10 17 42 CCCCCCCCNS(=O)(=O)c1ccsc1CNC ZINC000147402850 DG For-Sale Mild S1PR2 42 33 C[C@@H]1CCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147402906 CG On-Demand Anodyne HRH3 29 43 C[C@@H]1CCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147402906 CG On-Demand Anodyne CACNA1I 47 35 Cc1nc(Oc2cccc(F)c2C#N)ccc1C(=O)O ZINC000147402927 CF For-Sale Mild ALS 47 39 N#Cc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147402993 CD On-Demand Mild KCNK3 51 32 CCN1CCN(c2ccc(NC(=O)Nc3ccc(S(C)(=O)=O)nc3)c(C)c2)CC1 ZINC000147403046 HF On-Demand Anodyne PRNP 30 41 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@H]1CC[C@@H](C)O1 ZINC000147403099 DC On-Demand Anodyne CA2 41 42 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@H]1CC[C@@H](C)O1 ZINC000147403099 DC On-Demand Anodyne CA1 43 40 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@H]1CC[C@@H](C)O1 ZINC000147403099 DC On-Demand Anodyne CA7 43 42 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@H]1CC[C@@H](C)O1 ZINC000147403099 DC On-Demand Anodyne CA4 42 37 C[C@H]1CCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147403116 CG On-Demand Anodyne HRH3 29 43 C[C@H]1CCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147403116 CG On-Demand Anodyne CACNA1I 47 35 C[C@H](NCC(F)F)[C@@H]1CCCN(C(=O)OC(C)(C)C)C1 ZINC000147403132 CF On-Demand Anodyne GPR119 29 41 Cc1nc(Oc2cccc(F)c2C(N)=O)ccc1C(=O)O ZINC000147403143 CE For-Sale Anodyne ALS 63 48 CCS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3ccc(F)c(F)c3)no2)CC1 ZINC000147403163 HF Annotated Anodyne NPY2R 0 41 O=C(NCC1(C(=O)O)CCC1)c1ccc(Cl)cc1F ZINC000147403279 CE On-Demand Anodyne P2RX7 0 44 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@H]1CC[C@H](C)O1 ZINC000147403313 DC On-Demand Anodyne CA2 41 42 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@H]1CC[C@H](C)O1 ZINC000147403313 DC On-Demand Anodyne CA1 43 40 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@H]1CC[C@H](C)O1 ZINC000147403313 DC On-Demand Anodyne CA7 43 42 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@H]1CC[C@H](C)O1 ZINC000147403313 DC On-Demand Anodyne CA4 42 37 C[C@@H](NCC(F)F)[C@@H]1CCCN(C(=O)OC(C)(C)C)C1 ZINC000147403345 CF On-Demand Anodyne GPR119 29 41 Cc1nc(Oc2ccc(S(C)(=O)=O)cc2)ccc1C(=O)O ZINC000147403383 DE For-Sale Anodyne PTGS2 27 40 Cc1nc(Oc2ccc(S(C)(=O)=O)cc2)ccc1C(=O)O ZINC000147403383 DE For-Sale Anodyne MT-CO2 34 41 CNC(=O)C1CCN(C(=O)C(F)(F)c2cccc(Cl)c2)CC1 ZINC000147403406 EE On-Demand Anodyne FDFT1 15 42 CCN1CCN(c2ccc(NC(=O)Nc3cc(C(=O)OC)ccc3C)c(C)c2)CC1 ZINC000147403472 HH On-Demand Anodyne PRNP 34 41 Cc1c(Br)cccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147403483 EF On-Demand Anodyne HCN1 52 32 Cc1c(Br)cccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147403483 EF On-Demand Anodyne HCN4 50 32 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@@H]1CC[C@@H](C)O1 ZINC000147403534 DC On-Demand Anodyne CA2 41 42 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@@H]1CC[C@@H](C)O1 ZINC000147403534 DC On-Demand Anodyne CA1 43 40 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@@H]1CC[C@@H](C)O1 ZINC000147403534 DC On-Demand Anodyne CA7 43 42 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@@H]1CC[C@@H](C)O1 ZINC000147403534 DC On-Demand Anodyne CA4 42 37 C[C@H](NCC(F)F)[C@H]1CCCN(C(=O)OC(C)(C)C)C1 ZINC000147403553 CF On-Demand Anodyne GPR119 29 41 Cc1nc2ccc(C(=O)O)cc2n1CCNC(=O)N(C)C ZINC000147403560 CD For-Sale Anodyne HPD 44 32 CC[C@H](N)C(=O)O[C@@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000147403562 BF For-Sale Anodyne TRPM8 0 41 Cc1nc(Oc2cccc(S(C)(=O)=O)c2)ccc1C(=O)O ZINC000147403630 DE For-Sale Anodyne TRY1_BOVIN 27 42 Cc1nc(Oc2cccc(S(C)(=O)=O)c2)ccc1C(=O)O ZINC000147403630 DE For-Sale Anodyne NR1H3 40 37 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)c1ccccc1 ZINC000147403643 CD For-Sale Anodyne XIAP 53 37 CCCCO[C@H](C)C(=O)N1CCN([C@@H](C)c2nc(-c3ccc(C)cc3)no2)CC1 ZINC000147403659 HG On-Demand Anodyne PLA2G2A 25 43 CCCCO[C@H](C)C(=O)N1CCN([C@@H](C)c2nc(-c3ccc(C)cc3)no2)CC1 ZINC000147403659 HG On-Demand Anodyne DPP7 22 42 O=C(Nc1nc(-c2ccc(Cl)cc2)cs1)[C@H]1CCCCN1C(=O)c1cccs1 ZINC000147403709 IK On-Demand Anodyne MPL 49 43 O=C(Nc1nc(-c2ccc(Cl)cc2)cs1)[C@H]1CCCCN1C(=O)c1cccs1 ZINC000147403709 IK On-Demand Anodyne SPHK2 24 43 O=C(Nc1nc(-c2ccc(Cl)cc2)cs1)[C@H]1CCCCN1C(=O)c1cccs1 ZINC000147403709 IK On-Demand Anodyne SPHK1 31 43 O=C(Nc1nc(-c2ccc(Cl)cc2)cs1)[C@H]1CCCCN1C(=O)c1cccs1 ZINC000147403709 IK On-Demand Anodyne TRPC6 44 36 O=C(Nc1nc(-c2ccc(Cl)cc2)cs1)[C@H]1CCCCN1C(=O)c1cccs1 ZINC000147403709 IK On-Demand Anodyne TRPC3 43 36 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@@H]1CC[C@H](C)O1 ZINC000147403749 DC On-Demand Anodyne CA2 41 42 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@@H]1CC[C@H](C)O1 ZINC000147403749 DC On-Demand Anodyne CA1 43 40 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@@H]1CC[C@H](C)O1 ZINC000147403749 DC On-Demand Anodyne CA7 43 42 COc1ccc(S(N)(=O)=O)cc1NC(=O)[C@@H]1CC[C@H](C)O1 ZINC000147403749 DC On-Demand Anodyne CA4 42 37 CC[C@H](N)C(=O)O[C@H]1C[C@@H](C)CC[C@@H]1C(C)C ZINC000147403753 BF For-Sale Anodyne TRPM8 0 41 CC[C@@H]1CCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147403791 CG On-Demand Anodyne CACNA1I 52 35 Cc1cc(OCCC(=O)NC2CC2)cc(C)c1S(N)(=O)=O ZINC000147403806 DC For-Sale Anodyne CA7 24 44 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)c1ccccc1 ZINC000147403858 CD For-Sale Anodyne XIAP 53 37 CCCCO[C@@H](C)C(=O)N1CCN([C@H](C)c2nc(-c3ccc(C)cc3)no2)CC1 ZINC000147403900 HG On-Demand Anodyne PLA2G2A 25 43 CCCCO[C@@H](C)C(=O)N1CCN([C@H](C)c2nc(-c3ccc(C)cc3)no2)CC1 ZINC000147403900 HG On-Demand Anodyne DPP7 22 42 c1ccc2c(c1)CCN[C@@H]2c1nc(-c2cncs2)no1 ZINC000147403913 CE For-Sale Anodyne PRCP 49 41 O=C(Nc1nc(-c2ccc(Cl)cc2)cs1)[C@@H]1CCCCN1C(=O)c1cccs1 ZINC000147403951 IK On-Demand Anodyne MPL 49 43 O=C(Nc1nc(-c2ccc(Cl)cc2)cs1)[C@@H]1CCCCN1C(=O)c1cccs1 ZINC000147403951 IK On-Demand Anodyne SPHK2 24 43 O=C(Nc1nc(-c2ccc(Cl)cc2)cs1)[C@@H]1CCCCN1C(=O)c1cccs1 ZINC000147403951 IK On-Demand Anodyne SPHK1 31 43 O=C(Nc1nc(-c2ccc(Cl)cc2)cs1)[C@@H]1CCCCN1C(=O)c1cccs1 ZINC000147403951 IK On-Demand Anodyne TRPC6 44 36 O=C(Nc1nc(-c2ccc(Cl)cc2)cs1)[C@@H]1CCCCN1C(=O)c1cccs1 ZINC000147403951 IK On-Demand Anodyne TRPC3 43 36 Cc1ccc(Br)c(C(=O)NCc2ccc(C)c(F)c2)c1 ZINC000147403959 EI On-Demand Anodyne LEF 90 39 CC[C@H]1CCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147403984 CG On-Demand Anodyne CACNA1I 52 35 Cc1cc(OCC(=O)N2CCCC2)cc(C)c1S(N)(=O)=O ZINC000147404000 DC For-Sale Anodyne GPR183 0 45 CN(C)c1ccccc1NC(=O)c1ccc(O)cc1O ZINC000147404064 CE On-Demand Anodyne KCNMA1 36 41 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)c1ccccc1 ZINC000147404069 CD For-Sale Anodyne XIAP 53 37 CCCCO[C@H](C)C(=O)N1CCN([C@H](C)c2nc(-c3ccc(C)cc3)no2)CC1 ZINC000147404095 HG On-Demand Anodyne PLA2G2A 25 43 CCCCO[C@H](C)C(=O)N1CCN([C@H](C)c2nc(-c3ccc(C)cc3)no2)CC1 ZINC000147404095 HG On-Demand Anodyne DPP7 22 42 c1ccc2c(c1)CCN[C@H]2c1nc(-c2cncs2)no1 ZINC000147404100 CE For-Sale Anodyne PRCP 49 41 CNC(=O)C1CCN(C(=O)[C@@H](C)Cc2cccc(F)c2)CC1 ZINC000147404110 DD On-Demand Anodyne F2 30 42 CNC(=O)C1CCN(C(=O)[C@@H](C)Cc2cccc(F)c2)CC1 ZINC000147404110 DD On-Demand Anodyne PLG 40 44 CNC(=O)C1CCN(C(=O)[C@@H](C)Cc2cccc(F)c2)CC1 ZINC000147404110 DD On-Demand Anodyne TRY2_BOVIN 97 54 CNC(=O)C1CCN(C(=O)[C@@H](C)Cc2cccc(F)c2)CC1 ZINC000147404110 DD On-Demand Anodyne CCR1 30 46 CNC(=O)C1CCN(C(=O)[C@@H](C)Cc2cccc(F)c2)CC1 ZINC000147404110 DD On-Demand Anodyne DPP4 15 42 CNC(=O)C1CCN(C(=O)[C@@H](C)Cc2cccc(F)c2)CC1 ZINC000147404110 DD On-Demand Anodyne MLNR 20 41 CNC(=O)C1CCN(C(=O)[C@@H](C)Cc2cccc(F)c2)CC1 ZINC000147404110 DD On-Demand Anodyne ST14 112 42 CNC(=O)C1CCN(C(=O)[C@@H](C)Cc2cccc(F)c2)CC1 ZINC000147404110 DD On-Demand Anodyne CACNA1G 33 45 CNC(=O)C1CCN(C(=O)[C@@H](C)Cc2cccc(F)c2)CC1 ZINC000147404110 DD On-Demand Anodyne TMPRSS6 66 35 Cc1nc(Oc2ccc([N+](=O)[O-])cc2)ccc1C(=O)O ZINC000147404134 CF For-Sale Bother AKR1C2 27 46 Clc1cc(NCc2ccccc2)n2ncnc2n1 ZINC000147404184 CE For-Sale Anodyne DHOD 0 52 Clc1cc(NCc2ccccc2)n2ncnc2n1 ZINC000147404184 CE For-Sale Anodyne ISPD 0 46 CCc1nc2c(C(=O)O)cccc2n1CCNC(N)=O ZINC000147404204 CC For-Sale Anodyne AGTR1 36 41 CCc1nc2c(C(=O)O)cccc2n1CCNC(N)=O ZINC000147404204 CC For-Sale Anodyne AGTR1B 25 41 CCc1nc2c(C(=O)O)cccc2n1CCNC(N)=O ZINC000147404204 CC For-Sale Anodyne PARP1 0 40 COc1ccc(NC(C)=O)c(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147404280 FI On-Demand Anodyne AKR1C2 31 42 CNC(=O)C1CCN(C(=O)[C@H](C)Cc2cccc(F)c2)CC1 ZINC000147404359 DD On-Demand Anodyne F2 30 42 CNC(=O)C1CCN(C(=O)[C@H](C)Cc2cccc(F)c2)CC1 ZINC000147404359 DD On-Demand Anodyne PLG 40 44 CNC(=O)C1CCN(C(=O)[C@H](C)Cc2cccc(F)c2)CC1 ZINC000147404359 DD On-Demand Anodyne TRY2_BOVIN 97 54 CNC(=O)C1CCN(C(=O)[C@H](C)Cc2cccc(F)c2)CC1 ZINC000147404359 DD On-Demand Anodyne CCKAR 16 41 CNC(=O)C1CCN(C(=O)[C@H](C)Cc2cccc(F)c2)CC1 ZINC000147404359 DD On-Demand Anodyne CCR1 30 46 CNC(=O)C1CCN(C(=O)[C@H](C)Cc2cccc(F)c2)CC1 ZINC000147404359 DD On-Demand Anodyne DPP4 15 42 CNC(=O)C1CCN(C(=O)[C@H](C)Cc2cccc(F)c2)CC1 ZINC000147404359 DD On-Demand Anodyne MLNR 20 41 CNC(=O)C1CCN(C(=O)[C@H](C)Cc2cccc(F)c2)CC1 ZINC000147404359 DD On-Demand Anodyne ST14 112 42 CNC(=O)C1CCN(C(=O)[C@H](C)Cc2cccc(F)c2)CC1 ZINC000147404359 DD On-Demand Anodyne CACNA1G 33 45 CNC(=O)C1CCN(C(=O)[C@H](C)Cc2cccc(F)c2)CC1 ZINC000147404359 DD On-Demand Anodyne TMPRSS6 66 35 Cc1nc(Oc2cccc([N+](=O)[O-])c2)ccc1C(=O)O ZINC000147404366 CF For-Sale Bother CACNA1C 56 38 Cc1nc(Oc2cccc([N+](=O)[O-])c2)ccc1C(=O)O ZINC000147404366 CF For-Sale Bother TRY1_BOVIN 24 42 Cc1nc(Oc2cccc([N+](=O)[O-])c2)ccc1C(=O)O ZINC000147404366 CF For-Sale Bother CACNA1D 83 38 Cc1nc(Oc2cccc([N+](=O)[O-])c2)ccc1C(=O)O ZINC000147404366 CF For-Sale Bother PYGL 34 45 Cc1nc(Oc2cccc([N+](=O)[O-])c2)ccc1C(=O)O ZINC000147404366 CF For-Sale Bother PYGM 27 40 Cc1nc(Oc2cccc([N+](=O)[O-])c2)ccc1C(=O)O ZINC000147404366 CF For-Sale Bother PLAU 0 45 Cc1nc(Oc2cccc([N+](=O)[O-])c2)ccc1C(=O)O ZINC000147404366 CF For-Sale Bother ALS 62 33 Cc1nc(Oc2cccc([N+](=O)[O-])c2)ccc1C(=O)O ZINC000147404366 CF For-Sale Bother APR 0 40 Cc1nc(Oc2cccc([N+](=O)[O-])c2)ccc1C(=O)O ZINC000147404366 CF For-Sale Bother ATSA 0 46 Cc1nc(Oc2cccc([N+](=O)[O-])c2)ccc1C(=O)O ZINC000147404366 CF For-Sale Bother AKR1C2 28 46 COc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1F ZINC000147404445 HG On-Demand Anodyne BMP1 40 43 COc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1F ZINC000147404445 HG On-Demand Anodyne ROCK2 18 50 COc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1F ZINC000147404445 HG On-Demand Anodyne MMP12 28 41 COc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1F ZINC000147404445 HG On-Demand Anodyne CA9 15 41 COc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1F ZINC000147404445 HG On-Demand Anodyne PRMT3 18 41 COc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1F ZINC000147404445 HG On-Demand Anodyne MTCA1 15 40 COc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1F ZINC000147404445 HG On-Demand Anodyne NAMPT 44 40 CN(CC1CC1)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147404447 CF On-Demand Anodyne CACNA1I 57 40 COc1ccc(NC(C)=O)c(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)c1 ZINC000147404495 FI On-Demand Anodyne AKR1C2 31 42 Cc1cccc(NC(=O)[C@@H]2CCCN(C(=O)c3ccccc3OCCN(C)C)C2)n1 ZINC000147404547 HF On-Demand Anodyne SLC6A1 40 32 Cc1nc(Oc2ccccc2[N+](=O)[O-])ccc1C(=O)O ZINC000147404600 CF For-Sale Bother ALS 38 46 COc1ccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1F ZINC000147404674 FF On-Demand Anodyne HTR1D 26 43 CCc1nc2ccc(C(=O)O)cc2n1CCNC(N)=O ZINC000147404682 CC For-Sale Anodyne CDPK1 0 41 CC(C)C(NCCCc1ccccc1)C(C)C ZINC000147404683 BH For-Sale Anodyne SIGMAR1 25 57 CC(C)C(NCCCc1ccccc1)C(C)C ZINC000147404683 BH For-Sale Anodyne AMP1_PLAFQ 28 44 COc1ccc(NC(C)=O)c(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)c1 ZINC000147404727 FI On-Demand Anodyne AKR1C2 31 42 Cc1cccc(NC(=O)[C@H]2CCCN(C(=O)c3ccccc3OCCN(C)C)C2)n1 ZINC000147404750 HF On-Demand Anodyne SLC6A1 40 32 Cc1nccn1-c1ccc(CNS(=O)(=O)C[C@@]23CC[C@@H](CC2=O)C3(C)C)cc1F ZINC000147404779 HG On-Demand Anodyne CA5B 28 55 Cc1nccn1-c1ccc(CNS(=O)(=O)C[C@@]23CC[C@@H](CC2=O)C3(C)C)cc1F ZINC000147404779 HG On-Demand Anodyne CA5A 31 55 Cc1nccn1-c1ccc(CNS(=O)(=O)C[C@@]23CC[C@@H](CC2=O)C3(C)C)cc1F ZINC000147404779 HG On-Demand Anodyne CXCR3 40 38 Cc1ccc([N+](=O)[O-])c(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147404846 CG For-Sale Bother ALS 17 40 O=C(Nc1cc2c(cc1Cl)OCO2)c1ccc(Br)c(Cl)c1 ZINC000147404895 GJ On-Demand Anodyne CCR2 0 44 O=C(Nc1cc2c(cc1Cl)OCO2)c1ccc(Br)c(Cl)c1 ZINC000147404895 GJ On-Demand Anodyne GPR35 16 43 CCC[C@@H](CN)C(=O)NCCCCC(C)C ZINC000147404900 BE For-Sale Anodyne DPP7 0 46 CCCCCCCCNS(=O)(=O)[C@@H](C)CNCC ZINC000147404935 CE For-Sale Mild RELA 17 40 CCCNCc1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147404940 DJ For-Sale Anodyne MCHR1 0 53 C[C@H]1CCC[C@@H](C)N1NC(=O)CNC1CCCC1 ZINC000147404960 CD For-Sale Anodyne DPP7 15 41 O=C(CC(=O)N1CCc2ccccc21)Nc1ccccc1 ZINC000147405030 CF For-Sale Anodyne ACE 17 41 O=C(CC(=O)N1CCc2ccccc21)Nc1ccccc1 ZINC000147405030 CF For-Sale Anodyne AVPR2 83 54 O=C(CC(=O)N1CCc2ccccc21)Nc1ccccc1 ZINC000147405030 CF For-Sale Anodyne AVPR1A 45 51 O=C(CC(=O)N1CCc2ccccc21)Nc1ccccc1 ZINC000147405030 CF For-Sale Anodyne HSD17B3 15 41 COc1ccc(NC(C)=O)c(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147405062 FF On-Demand Anodyne MTNR1A 31 47 COc1ccc(NC(C)=O)c(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)c1 ZINC000147405062 FF On-Demand Anodyne ROCK2 41 55 COc1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405072 HG On-Demand Anodyne ADRB2 23 42 COc1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405072 HG On-Demand Anodyne ADRB1 55 41 COc1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405072 HG On-Demand Anodyne HTR2A 16 41 COc1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405072 HG On-Demand Anodyne ADRB3 23 43 COc1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405072 HG On-Demand Anodyne P2RY1 17 43 COc1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405072 HG On-Demand Anodyne RAF1 42 41 COc1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405072 HG On-Demand Anodyne ACR 18 40 COc1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405072 HG On-Demand Anodyne TEK 44 35 COc1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405072 HG On-Demand Anodyne Q8MMZ8_EIMTE 43 41 COc1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405072 HG On-Demand Anodyne RIPK1 51 32 COc1ccc(NC(=O)NC[C@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405072 HG On-Demand Anodyne PDS 55 46 O=C(NC[C@@H]1COCCO1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147405086 DD On-Demand Anodyne CACNA1I 42 34 CCC[C@H](CN)C(=O)NCCCCC(C)C ZINC000147405095 BE For-Sale Anodyne DPP7 0 46 Cc1ccc(CCC(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147405122 EI For-Sale Reactive PREP 48 39 Cc1ccc(CCC(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147405122 EI For-Sale Reactive FAP 0 40 NC(=O)NCCn1c(C2CC2)nc2c(C(=O)O)cccc21 ZINC000147405123 CD For-Sale Anodyne PARP1 28 51 CC(C)CNCCCOc1ccc(Cl)c(F)c1 ZINC000147405145 CG For-Sale Anodyne DRD4 21 48 CCCCCCCCNS(=O)(=O)[C@H](C)CNCC ZINC000147405147 CE For-Sale Mild RELA 17 40 CCCCCCc1ccc2c(c1)c1ccccc1c(=O)n2CCCC ZINC000147405155 EK Annotated Bother CNR1 27 48 CCCCCCc1ccc2c(c1)c1ccccc1c(=O)n2CCCC ZINC000147405155 EK Annotated Bother INHA 88 39 CCCCCCc1ccc2c(c1)c1ccccc1c(=O)n2CCCC ZINC000147405155 EK Annotated Bother CNR2 30 48 CCCCCCc1ccc2c(c1)c1ccccc1c(=O)n2CCCC ZINC000147405155 EK Annotated Bother RORC 0 59 CCCCCCc1ccc2c(c1)c1ccccc1c(=O)n2CCCC ZINC000147405155 EK Annotated Bother OXER1 43 37 CCCCCCc1ccc2c(c1)c1ccccc1c(=O)n2CCCC ZINC000147405155 EK Annotated Bother RORB 0 80 C[C@H]1CCC[C@H](C)N1NC(=O)CNC1CCCC1 ZINC000147405181 CD For-Sale Anodyne DPP7 15 41 Cc1nc(Oc2ccc([N+](=O)[O-])cc2Cl)ccc1C(=O)O ZINC000147405227 DG For-Sale Bother ENR 0 48 Cc1nc(Oc2ccc([N+](=O)[O-])cc2Cl)ccc1C(=O)O ZINC000147405227 DG For-Sale Bother PPXII 0 40 COc1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405283 HG On-Demand Anodyne ADRB2 23 42 COc1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405283 HG On-Demand Anodyne ADRB1 55 41 COc1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405283 HG On-Demand Anodyne HTR2A 16 41 COc1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405283 HG On-Demand Anodyne ADRB3 23 43 COc1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405283 HG On-Demand Anodyne P2RY1 17 43 COc1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405283 HG On-Demand Anodyne RAF1 42 41 COc1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405283 HG On-Demand Anodyne ACR 18 40 COc1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405283 HG On-Demand Anodyne TEK 44 35 COc1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405283 HG On-Demand Anodyne RIPK1 51 32 COc1ccc(NC(=O)NC[C@@H](O)COc2cccc(C(F)(F)F)c2)cc1F ZINC000147405283 HG On-Demand Anodyne PDS 55 46 O=C(NC[C@H]1COCCO1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147405289 DD On-Demand Anodyne CACNA1I 42 34 Cc1ccc(CCC(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147405342 EI For-Sale Reactive PREP 48 39 Cc1ccc(CCC(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147405342 EI For-Sale Reactive FAP 0 40 Cc1cccc(NC(=O)[C@@H]2CCCN(C(=O)COc3ccc(C(N)=O)cc3)C2)n1 ZINC000147405354 GD On-Demand Anodyne CPT1A 101 42 CC(C)CNCCCCCCOc1ccc(Cl)c(F)c1 ZINC000147405356 DJ For-Sale Anodyne DRD4 19 43 C[C@@H]1CCC[C@@H](C)N1NC(=O)CNC1CCCC1 ZINC000147405383 CD For-Sale Anodyne DPP7 15 41 CCCC[C@H](NC(N)=O)C(=O)Nc1cc(C(=O)NC)ccc1C ZINC000147405386 DD On-Demand Anodyne MAPK14 23 44 CCCC[C@H](NC(N)=O)C(=O)Nc1cc(C(=O)NC)ccc1C ZINC000147405386 DD On-Demand Anodyne PCSK5 40 33 CCCC[C@H](NC(N)=O)C(=O)Nc1cc(C(=O)NC)ccc1C ZINC000147405386 DD On-Demand Anodyne FURIN 53 33 CCCC[C@H](NC(N)=O)C(=O)Nc1cc(C(=O)NC)ccc1C ZINC000147405386 DD On-Demand Anodyne ERAP2 51 39 Cc1nc(Oc2cc(F)ccc2[N+](=O)[O-])ccc1C(=O)O ZINC000147405442 CF For-Sale Bother ALS 25 41 COc1cc(CNC(=O)c2cc(C)cc([N+](=O)[O-])c2)ccc1OC(F)F ZINC000147405500 FG On-Demand Bother MT-ND1 24 44 Cc1cccc(NC(=O)[C@H]2CCCN(C(=O)COc3ccc(C(N)=O)cc3)C2)n1 ZINC000147405542 GD On-Demand Anodyne CPT1A 101 42 CC(C)CCCCNCc1ccn(C)c1 ZINC000147405555 BF On-Demand Anodyne LEF 49 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1cc(C(=O)NC)ccc1C ZINC000147405571 DD On-Demand Anodyne MAPK14 23 44 CCCC[C@@H](NC(N)=O)C(=O)Nc1cc(C(=O)NC)ccc1C ZINC000147405571 DD On-Demand Anodyne PCSK5 40 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1cc(C(=O)NC)ccc1C ZINC000147405571 DD On-Demand Anodyne FURIN 53 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1cc(C(=O)NC)ccc1C ZINC000147405571 DD On-Demand Anodyne ERAP2 51 39 CCCOc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147405630 FI For-Sale Reactive PLA2G4B 35 40 CCCOc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147405630 FI For-Sale Reactive CFTR 41 41 CCCOc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147405630 FI For-Sale Reactive CHRNA10 61 39 COc1ccc(NC(=O)N2CCO[C@H](c3ccc(Br)cc3)C2)cc1F ZINC000147405653 HI On-Demand Anodyne HTR1D 19 41 CC(C)(C)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147405658 CG For-Sale Anodyne CACNA1I 53 39 CC(C)(C)CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147405658 CG For-Sale Anodyne HCAR1 0 41 Cc1nc(Oc2cccc([N+](=O)[O-])c2C)ccc1C(=O)O ZINC000147405675 CG For-Sale Bother ALS 45 47 FC(F)CNCc1c[nH]c2ncccc12 ZINC000147405682 BD For-Sale Anodyne CDC7 46 34 CCc1ncc(C(=O)NCc2ccc(OC(F)F)c(OC)c2)s1 ZINC000147405683 EG On-Demand Anodyne MT-ND1 22 40 CCc1ncc(C(=O)NCc2ccc(OC(F)F)c(OC)c2)s1 ZINC000147405683 EG On-Demand Anodyne HCRTR2 15 41 CCc1ncc(C(=O)NCc2ccc(OC(F)F)c(OC)c2)s1 ZINC000147405683 EG On-Demand Anodyne DRTS_TRYCR 44 30 O[C@@H]1CN(Cc2ccccc2)C[C@@H]2C[C@@H]12 ZINC000147405737 BD For-Sale Anodyne DRD2 16 41 C[C@H](c1ccco1)N(C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)C1CC1 ZINC000147405747 EJ On-Demand Anodyne MDM2 62 33 C[C@@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147405762 EJ On-Demand Anodyne PPARA 17 41 C[C@@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147405762 EJ On-Demand Anodyne TACR1 32 51 C[C@@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147405762 EJ On-Demand Anodyne TRPV1 22 40 C[C@@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147405762 EJ On-Demand Anodyne CSNK1D 26 40 C[C@@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147405762 EJ On-Demand Anodyne CCR5 16 45 C[C@@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147405762 EJ On-Demand Anodyne PPARD 27 43 C[C@@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147405762 EJ On-Demand Anodyne SLC6A9 15 48 C[C@@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147405762 EJ On-Demand Anodyne MTTP 67 41 C[C@@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147405762 EJ On-Demand Anodyne EPHX2 16 44 CCN(CC)C(=O)c1cccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)c1 ZINC000147405790 HF On-Demand Anodyne OPRD1 30 40 CCCOc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147405862 FI For-Sale Reactive PLA2G4B 35 40 CCCOc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147405862 FI For-Sale Reactive CFTR 41 41 CCCOc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147405862 FI For-Sale Reactive CHRNA10 61 39 COc1ccc(NC(=O)N2CCO[C@@H](c3ccc(Br)cc3)C2)cc1F ZINC000147405865 HI On-Demand Anodyne HTR1D 19 41 Cc1ccc([N+](=O)[O-])cc1Oc1ccc(C(=O)O)c(C)n1 ZINC000147405901 CG For-Sale Bother AKR1C2 23 40 Cc1cc(OCCc2ccncc2)cc(C)c1S(N)(=O)=O ZINC000147405939 DD For-Sale Anodyne CA7 17 43 CCCCCCCCNS(=O)(=O)CCCCNC(C)C ZINC000147405955 DG For-Sale Mild RELA 26 58 C[C@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147406007 EJ On-Demand Anodyne PPARA 17 41 C[C@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147406007 EJ On-Demand Anodyne TACR1 32 51 C[C@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147406007 EJ On-Demand Anodyne TRPV1 22 40 C[C@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147406007 EJ On-Demand Anodyne CSNK1D 26 40 C[C@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147406007 EJ On-Demand Anodyne CCR5 16 45 C[C@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147406007 EJ On-Demand Anodyne PPARD 27 43 C[C@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147406007 EJ On-Demand Anodyne SLC6A9 15 48 C[C@H](CCNC(=O)Cc1ccc(C(F)(F)F)cc1)c1ccccc1 ZINC000147406007 EJ On-Demand Anodyne MTTP 67 41 CCN(CC)C(=O)c1cccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)c1 ZINC000147406012 HF On-Demand Anodyne OPRD1 30 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCc2sccc2[C@@H]1c1cccs1 ZINC000147406043 GK On-Demand Anodyne TRPM8 19 45 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406113 FI On-Demand Anodyne TSHR 49 35 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406113 FI On-Demand Anodyne IGF1R 16 40 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406113 FI On-Demand Anodyne KDR 15 40 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406113 FI On-Demand Anodyne ROCK2 15 40 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406113 FI On-Demand Anodyne MET 60 40 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406113 FI On-Demand Anodyne QRFPR 41 39 Cc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1[N+](=O)[O-] ZINC000147406114 CG For-Sale Bother ALS 47 40 O=C(O)c1cccc2oc(-c3ccc4c(c3)OCO4)nc12 ZINC000147406115 CF For-Sale Anodyne EDNRB 33 41 O=C(O)c1cccc2oc(-c3ccc4c(c3)OCO4)nc12 ZINC000147406115 CF For-Sale Anodyne EDNRA 34 41 O=C(O)c1cccc2oc(-c3ccc4c(c3)OCO4)nc12 ZINC000147406115 CF For-Sale Anodyne GSK3A 25 40 O=C(O)c1cccc2oc(-c3ccc4c(c3)OCO4)nc12 ZINC000147406115 CF For-Sale Anodyne TGFBR1 33 41 COc1cccc(F)c1C(=O)N1CCC[C@@H]1CCCBr ZINC000147406120 EH For-Sale Reactive HCRTR1 20 44 COc1cccc(F)c1C(=O)N1CCC[C@@H]1CCCBr ZINC000147406120 EH For-Sale Reactive HCRTR2 19 44 COc1cccc(F)c1C(=O)N1CCC[C@@H]1CCCBr ZINC000147406120 EH For-Sale Reactive ACKR3 68 35 CCCCCCCCNS(=O)(=O)CCCCNC ZINC000147406166 CE For-Sale Mild RELA 28 63 NC(=O)C(F)(F)c1cccc([N+](=O)[O-])c1 ZINC000147406197 BD For-Sale Bother CACNA1C 44 38 NC(=O)C(F)(F)c1cccc([N+](=O)[O-])c1 ZINC000147406197 BD For-Sale Bother CACNA1D 73 38 C[C@H](c1ccco1)N(C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)C1CC1 ZINC000147406200 EJ On-Demand Anodyne MDM2 62 33 N#CCNC(=O)Cc1nnc(Cc2nc3c(-c4ccccc4)cccc3s2)o1 ZINC000147406201 GG Annotated Mild CTSV 46 35 CC(C)c1nc2ccc(C(=O)O)cc2n1CCNC(N)=O ZINC000147406222 CD For-Sale Anodyne CDPK1 0 43 C[C@H](Cc1cccc(F)c1)C(=O)N1CCc2sccc2[C@@H]1c1cccs1 ZINC000147406223 GK On-Demand Anodyne TRPM8 19 45 O=C(N[C@H]1C[C@H]1c1ccccc1)N[C@@H]1CCOc2c(Cl)cccc21 ZINC000147406298 EI On-Demand Anodyne EPHX2 21 46 C[C@H](NC(=O)[C@]1(C)CCCS1)c1nc2ccccc2[nH]1 ZINC000147406312 CG For-Sale Anodyne PTPN1 29 42 COc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406326 FI On-Demand Anodyne TSHR 49 35 COc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406326 FI On-Demand Anodyne IGF1R 16 40 COc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406326 FI On-Demand Anodyne KDR 15 40 COc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406326 FI On-Demand Anodyne ROCK2 15 40 COc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406326 FI On-Demand Anodyne MET 60 40 COc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1F ZINC000147406326 FI On-Demand Anodyne QRFPR 41 39 COc1cccc(F)c1C(=O)N1CCC[C@H]1CCCBr ZINC000147406347 EH For-Sale Reactive HCRTR1 20 44 COc1cccc(F)c1C(=O)N1CCC[C@H]1CCCBr ZINC000147406347 EH For-Sale Reactive HCRTR2 19 44 COc1cccc(F)c1C(=O)N1CCC[C@H]1CCCBr ZINC000147406347 EH For-Sale Reactive ACKR3 68 35 CCCCCCCCNS(=O)(=O)c1ccc(Cl)c(CN)c1 ZINC000147406362 EG For-Sale Mild ALOX15 53 42 COC(=O)c1ccc(-c2noc(-c3sccc3Cl)n2)cc1 ZINC000147406363 DH On-Demand Anodyne CASP3 16 66 CN1CCC[C@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147406366 DE On-Demand Anodyne CACNA1H 26 47 CN1CCC[C@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147406366 DE On-Demand Anodyne EPHX2 43 50 CN1CCC[C@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147406366 DE On-Demand Anodyne CACNA1I 57 37 NCCc1ccccc1COc1ccc(Cl)c(F)c1 ZINC000147406376 CH For-Sale Anodyne TAAR1 38 47 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCc2sccc2[C@H]1c1cccs1 ZINC000147406416 GK On-Demand Anodyne TRPM8 19 45 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne NPY1R 22 40 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne KLK3 50 40 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne CTSK 17 46 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne CTSL 28 41 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne NPFFR2 42 38 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne GRIA1 55 34 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne PCSK5 62 40 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne FURIN 69 42 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne AMP1_PLAFQ 29 41 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne POLG_WNV 76 35 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne QRFPR 46 41 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406417 EE On-Demand Anodyne NPFFR1 57 38 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc(F)cc1Br)C2 ZINC000147406448 GG On-Demand Anodyne P2RX7 21 47 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc(F)cc1Br)C2 ZINC000147406448 GG On-Demand Anodyne MTNR1A 23 40 COc1ccc2c(c1)OC[C@H](C(=O)NCc1ccc(F)cc1Br)C2 ZINC000147406448 GG On-Demand Anodyne ROCK2 23 40 CN(C(=O)Nc1ccc(-c2ccc(Cl)s2)nc1)C1CCN(S(C)(=O)=O)CC1 ZINC000147406514 IG On-Demand Anodyne NPY2R 15 45 C[C@@H](NC(=O)[C@]1(C)CCCS1)c1nc2ccccc2[nH]1 ZINC000147406520 CG For-Sale Anodyne PTPN1 29 42 O=C(N[C@H]1C[C@@H]1c1ccccc1)N[C@@H]1CCOc2c(Cl)cccc21 ZINC000147406529 EI On-Demand Anodyne EPHX2 21 46 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406557 FI On-Demand Anodyne TSHR 49 35 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406557 FI On-Demand Anodyne IGF1R 16 40 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406557 FI On-Demand Anodyne KDR 15 40 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406557 FI On-Demand Anodyne ROCK2 15 40 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406557 FI On-Demand Anodyne MET 60 40 COc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406557 FI On-Demand Anodyne QRFPR 41 39 CCCC(=O)[C@@H](CC)SC ZINC000147406564 AE For-Sale Anodyne CQSS 55 34 CN1CCC[C@@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147406591 DE On-Demand Anodyne CACNA1H 26 47 CN1CCC[C@@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147406591 DE On-Demand Anodyne EPHX2 43 50 CN1CCC[C@@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147406591 DE On-Demand Anodyne CACNA1I 57 37 CCN(CC)CCOc1cc(C)c(S(N)(=O)=O)c(C)c1 ZINC000147406614 DD For-Sale Anodyne ERG2 16 41 CCOC(=O)C1CCC(c2cccc(F)c2Cl)CC1 ZINC000147406621 CI For-Sale Anodyne FDFT1 21 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne NPY1R 22 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne KLK3 50 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne CTSK 17 46 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne CTSL 28 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne NPFFR2 42 38 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne GRIA1 55 34 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne PCSK5 62 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne FURIN 69 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne AMP1_PLAFQ 29 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne POLG_WNV 76 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne QRFPR 46 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(Br)c1 ZINC000147406645 EE On-Demand Anodyne NPFFR1 57 38 CCCc1nc2cc(C(=O)O)ccc2n1CCNC(N)=O ZINC000147406671 CD For-Sale Anodyne AGTR1 31 42 CCCc1nc2cc(C(=O)O)ccc2n1CCNC(N)=O ZINC000147406671 CD For-Sale Anodyne HDAC10 24 43 CCCc1nc2cc(C(=O)O)ccc2n1CCNC(N)=O ZINC000147406671 CD For-Sale Anodyne HDAC1 15 45 CCCc1nc2cc(C(=O)O)ccc2n1CCNC(N)=O ZINC000147406671 CD For-Sale Anodyne HDAC4 27 43 CCCc1nc2cc(C(=O)O)ccc2n1CCNC(N)=O ZINC000147406671 CD For-Sale Anodyne HDAC5 35 43 CCCc1nc2cc(C(=O)O)ccc2n1CCNC(N)=O ZINC000147406671 CD For-Sale Anodyne HDAC9 29 43 CCCc1nc2cc(C(=O)O)ccc2n1CCNC(N)=O ZINC000147406671 CD For-Sale Anodyne HDAC11 26 43 CCCc1nc2cc(C(=O)O)ccc2n1CCNC(N)=O ZINC000147406671 CD For-Sale Anodyne HDAC7 35 43 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(F)cc1Br)C2 ZINC000147406679 GG On-Demand Anodyne P2RX7 21 47 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(F)cc1Br)C2 ZINC000147406679 GG On-Demand Anodyne MTNR1A 23 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(F)cc1Br)C2 ZINC000147406679 GG On-Demand Anodyne ROCK2 23 40 Nc1c(C(=O)O)ccc2c1CCC2 ZINC000147406682 AD For-Sale Anodyne HAAO 41 33 CC(C)CCCCNCc1ccc(Cl)cc1 ZINC000147406691 BI For-Sale Anodyne FDFT1 0 41 CC(C)CCCCNCc1ccc(Cl)cc1 ZINC000147406691 BI For-Sale Anodyne S1PR2 34 41 CC(C)CCCCNCc1ccc(Cl)cc1 ZINC000147406691 BI For-Sale Anodyne DPP7 31 41 CC(C)CCCCNCc1ccc(Cl)cc1 ZINC000147406691 BI For-Sale Anodyne LEF 89 50 C[C@H](NC(=O)[C@@]1(C)CCCS1)c1nc2ccccc2[nH]1 ZINC000147406721 CG For-Sale Anodyne PTPN1 29 42 O=C(N[C@@H]1CCOc2c(Cl)cccc21)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147406743 EI On-Demand Anodyne EPHX2 21 46 Cc1nc(Oc2cccc(N(C)C)c2)ccc1C(=O)O ZINC000147406745 CF For-Sale Anodyne PLG 0 42 Cc1nc(Oc2cccc(N(C)C)c2)ccc1C(=O)O ZINC000147406745 CF For-Sale Anodyne TRY1_BOVIN 36 52 Cc1nc(Oc2cccc(N(C)C)c2)ccc1C(=O)O ZINC000147406745 CF For-Sale Anodyne ALS 43 31 C[C@@H](CC(=O)O)CN1C(=O)C[C@H](c2ccccc2)C1=O ZINC000147406771 CD For-Sale Anodyne HSD17B2 65 33 COc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406776 FI On-Demand Anodyne TSHR 49 35 COc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406776 FI On-Demand Anodyne IGF1R 16 40 COc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406776 FI On-Demand Anodyne KDR 15 40 COc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406776 FI On-Demand Anodyne ROCK2 15 40 COc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406776 FI On-Demand Anodyne MET 60 40 COc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1F ZINC000147406776 FI On-Demand Anodyne QRFPR 41 39 CCCC(=O)[C@H](CC)SC ZINC000147406803 AE For-Sale Anodyne CQSS 55 34 CCCCCCCCNS(=O)(=O)c1cccc(CNC)c1 ZINC000147406813 DG For-Sale Mild S1PR2 51 33 CCCCCCCCNS(=O)(=O)c1cccc(CNC)c1 ZINC000147406813 DG For-Sale Mild ALOX15 52 43 C[C@@H](NC(=O)[C@@]1(C)CCCS1)c1nc2ccccc2[nH]1 ZINC000147406904 CG For-Sale Anodyne PTPN1 29 42 CCN(CC)CCNC(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147406916 DG On-Demand Anodyne CACNA1H 22 43 O=C(N[C@@H]1CCOc2c(Cl)cccc21)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147406967 EI On-Demand Anodyne EPHX2 21 46 Cc1ccc(Oc2ccc(C(=O)O)c(C)n2)c([N+](=O)[O-])c1 ZINC000147406974 CG For-Sale Bother ALS 17 40 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne CA2 26 48 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne ADRB2 43 45 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne ADRB1 30 45 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne ADRB3 54 45 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne TBXAS1 15 42 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne BMP1 62 37 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne CA1 25 48 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne MMP13 35 40 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne MAP1 80 38 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne CA4 15 46 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne CA14 17 47 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne MMP3 21 40 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne MMP8 17 40 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne MMP9 29 40 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne CA12 17 48 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne CA9 31 48 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne CYNT 18 44 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne LIMK2 35 41 COc1ccc(CCNC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cc1 ZINC000147406998 HF On-Demand Anodyne A6YCJ1_9METZ 15 46 C[C@H](CC(=O)O)CN1C(=O)C[C@H](c2ccccc2)C1=O ZINC000147407001 CD For-Sale Anodyne HSD17B2 65 33 COc1cc(NC(=O)c2ccc3[nH]ncc3c2)ccc1Cl ZINC000147407012 DG On-Demand Anodyne COLA 77 41 COc1cc(NC(=O)c2ccc3[nH]ncc3c2)ccc1Cl ZINC000147407012 DG On-Demand Anodyne ROCK1 26 52 COc1cc(NC(=O)c2ccc3[nH]ncc3c2)ccc1Cl ZINC000147407012 DG On-Demand Anodyne DYRK1A 23 41 COc1cc(NC(=O)c2ccc3[nH]ncc3c2)ccc1Cl ZINC000147407012 DG On-Demand Anodyne AKT1 15 48 CCCCCCCCNS(=O)(=O)c1c[nH]c(CNCC)c1 ZINC000147407024 DF For-Sale Mild ALOX15 37 42 CCCCCCCCNS(=O)(=O)c1c[nH]c(CNCC)c1 ZINC000147407024 DF For-Sale Mild ASAH1 43 30 NC(=O)c1cc2c(Cl)ncnc2s1 ZINC000147407051 BD For-Sale Anodyne SELE 64 41 NC(=O)c1cc2c(Cl)ncnc2s1 ZINC000147407051 BD For-Sale Anodyne ICAM1 45 40 NC(=O)c1cc2c(Cl)ncnc2s1 ZINC000147407051 BD For-Sale Anodyne VCAM1 43 38 NC(=O)c1cc2c(Cl)ncnc2s1 ZINC000147407051 BD For-Sale Anodyne SIRT3 40 32 Cc1ccccc1C(=O)NNC(=O)Nc1cccc(CN2CCC[C@@H]2C(N)=O)c1 ZINC000147407154 GD On-Demand Reactive CCR3 44 37 Cc1ccccc1C(=O)NNC(=O)Nc1cccc(CN2CCC[C@@H]2C(N)=O)c1 ZINC000147407154 GD On-Demand Reactive CCR8 54 34 O=S(=O)(Nc1ccc(Cl)cc1Br)c1ccc(Br)cc1 ZINC000147407190 IJ For-Sale Anodyne CA2 15 45 O=S(=O)(Nc1ccc(Cl)cc1Br)c1ccc(Br)cc1 ZINC000147407190 IJ For-Sale Anodyne CA4 20 44 O=S(=O)(Nc1ccc(Cl)cc1Br)c1ccc(Br)cc1 ZINC000147407190 IJ For-Sale Anodyne IDO1 26 41 C[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147407208 CF On-Demand Anodyne CACNA1H 41 35 C[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147407208 CF On-Demand Anodyne EPHX2 17 44 C[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147407208 CF On-Demand Anodyne CACNA1I 49 36 C[C@@H](CC(=O)O)CN1C(=O)C[C@@H](c2ccccc2)C1=O ZINC000147407222 CD For-Sale Anodyne HSD17B2 65 33 COc1ccc(OC)c(CCNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147407229 HH On-Demand Anodyne NQO2 31 45 COc1ccc(OC)c(CCNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147407229 HH On-Demand Anodyne MTNR1A 94 45 COc1ccc(OC)c(CCNC(=O)[C@@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147407229 HH On-Demand Anodyne MTNR1B 76 46 O=C(NCC1(C(=O)O)CCC1)c1ccccc1Cl ZINC000147407232 CE On-Demand Anodyne P2RX7 24 55 O=C(NCC1(C(=O)O)CCC1)c1ccccc1Cl ZINC000147407232 CE On-Demand Anodyne SLC6A9 53 44 O=C(NCC1(C(=O)O)CCC1)c1ccccc1Cl ZINC000147407232 CE On-Demand Anodyne NR2E3 44 33 O=C(NCC1(C(=O)O)CCC1)c1ccccc1Cl ZINC000147407232 CE On-Demand Anodyne SMO 0 41 O=C(NCC1(C(=O)O)CCC1)c1ccccc1Cl ZINC000147407232 CE On-Demand Anodyne HCN1 64 36 O=C(NCC1(C(=O)O)CCC1)c1ccccc1Cl ZINC000147407232 CE On-Demand Anodyne HCN4 53 34 Cc1cccc(NC(=O)[C@@H]2CCCN(C(=O)c3ccc(Oc4cccnc4)cc3)C2)n1 ZINC000147407245 HI On-Demand Anodyne SLC18A3 16 42 Cc1cccc(NC(=O)[C@@H]2CCCN(C(=O)c3ccc(Oc4cccnc4)cc3)C2)n1 ZINC000147407245 HI On-Demand Anodyne GRM5 19 52 C[C@@H](OC(N)=O)[C@H](N)C(=O)O ZINC000147407248 AA For-Sale Anodyne SLC1A6 45 29 C[C@@H](OC(N)=O)[C@H](N)C(=O)O ZINC000147407248 AA For-Sale Anodyne SLC1A7 45 29 Cc1ccccc1C(=O)NNC(=O)Nc1cccc(CN2CCC[C@H]2C(N)=O)c1 ZINC000147407345 GD On-Demand Reactive CCR3 44 37 Cc1ccccc1C(=O)NNC(=O)Nc1cccc(CN2CCC[C@H]2C(N)=O)c1 ZINC000147407345 GD On-Demand Reactive CCR8 54 34 CCCc1nc2ccc(C(=O)O)cc2n1CCNC(N)=O ZINC000147407403 CD For-Sale Anodyne AGTR1 38 42 CCCc1nc2ccc(C(=O)O)cc2n1CCNC(N)=O ZINC000147407403 CD For-Sale Anodyne AGTR1B 21 40 O=C(Cc1c(F)cccc1Cl)N1CCC[C@@H]1CCCBr ZINC000147407418 FI For-Sale Reactive OPRK1 19 42 COc1ccc(OC)c(CCNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147407455 HH On-Demand Anodyne NQO2 31 45 COc1ccc(OC)c(CCNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147407455 HH On-Demand Anodyne MTNR1A 94 45 COc1ccc(OC)c(CCNC(=O)[C@H]2C[C@@H]2c2cccc(Br)c2)c1 ZINC000147407455 HH On-Demand Anodyne MTNR1B 76 46 C[C@H](CC(=O)O)CN1C(=O)C[C@@H](c2ccccc2)C1=O ZINC000147407456 CD For-Sale Anodyne HSD17B2 65 33 COc1ccc2ccccc2c1CNCCCCC(C)C ZINC000147407461 CJ For-Sale Anodyne SLC2A1 23 67 COc1ccc2ccccc2c1CNCCCCC(C)C ZINC000147407461 CJ For-Sale Anodyne XIAP 47 35 COc1ccc2ccccc2c1CNCCCCC(C)C ZINC000147407461 CJ For-Sale Anodyne HT1 0 67 COc1ccc2ccccc2c1CNCCCCC(C)C ZINC000147407461 CJ For-Sale Anodyne GPM3 0 43 COc1ccc2ccccc2c1CNCCCCC(C)C ZINC000147407461 CJ For-Sale Anodyne LMGT2 0 67 Cc1cccc(NC(=O)[C@H]2CCCN(C(=O)c3ccc(Oc4cccnc4)cc3)C2)n1 ZINC000147407462 HI On-Demand Anodyne SLC18A3 16 42 Cc1cccc(NC(=O)[C@H]2CCCN(C(=O)c3ccc(Oc4cccnc4)cc3)C2)n1 ZINC000147407462 HI On-Demand Anodyne GRM5 19 52 C[C@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147407478 CF On-Demand Anodyne CACNA1H 41 35 C[C@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147407478 CF On-Demand Anodyne EPHX2 17 44 C[C@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147407478 CF On-Demand Anodyne CACNA1I 49 36 Cc1nc(Oc2ccc([N+](=O)[O-])c(F)c2)ccc1C(=O)O ZINC000147407517 CF For-Sale Bother PPXII 0 40 CC[C@@H]1CN(S(=O)(=O)c2ccc3c(c2)CCC3)CC[C@@H]1N ZINC000147407552 DD On-Demand Anodyne CASP7 50 34 CNC(=O)C1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147407617 FF On-Demand Anodyne EPHX2 27 47 CNC(=O)C1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147407617 FF On-Demand Anodyne L3MBTL1 0 45 CNC(=O)C1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147407617 FF On-Demand Anodyne L3MBTL3 78 42 CNC(=O)C1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147407617 FF On-Demand Anodyne MBTD1 0 45 CNC(=O)C1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147407617 FF On-Demand Anodyne TP53BP1 0 42 O=C(Cc1c(F)cccc1Cl)N1CCC[C@H]1CCCBr ZINC000147407625 FI For-Sale Reactive OPRK1 19 42 NC(=O)NCCn1c(C2CC2)nc2ccc(C(=O)O)cc21 ZINC000147407639 CD For-Sale Anodyne CDPK1 0 43 COc1ccc(OC)c(CCNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147407661 HH On-Demand Anodyne NQO2 31 45 COc1ccc(OC)c(CCNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147407661 HH On-Demand Anodyne MTNR1A 94 45 COc1ccc(OC)c(CCNC(=O)[C@@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147407661 HH On-Demand Anodyne MTNR1B 76 46 Cc1nc(OCCCc2ccccc2)ccc1C(=O)O ZINC000147407723 CG For-Sale Anodyne ALOX5 15 45 Cc1nc(OCCCc2ccccc2)ccc1C(=O)O ZINC000147407723 CG For-Sale Anodyne PPARG 51 42 Cc1nc(OCCCc2ccccc2)ccc1C(=O)O ZINC000147407723 CG For-Sale Anodyne PPARA 51 42 Cc1nc(OCCCc2ccccc2)ccc1C(=O)O ZINC000147407723 CG For-Sale Anodyne P2RX1 31 42 Cc1nc(OCCCc2ccccc2)ccc1C(=O)O ZINC000147407723 CG For-Sale Anodyne LTB4R 57 36 Cc1nc(OCCCc2ccccc2)ccc1C(=O)O ZINC000147407723 CG For-Sale Anodyne FAAH 65 37 Cc1nc(OCCCc2ccccc2)ccc1C(=O)O ZINC000147407723 CG For-Sale Anodyne CES1 64 37 Cc1nc(OCCCc2ccccc2)ccc1C(=O)O ZINC000147407723 CG For-Sale Anodyne TSPAN17 0 42 Cc1nc(OCCCc2ccccc2)ccc1C(=O)O ZINC000147407723 CG For-Sale Anodyne MCL1 50 38 Cc1nc(OCCCc2ccccc2)ccc1C(=O)O ZINC000147407723 CG For-Sale Anodyne SLC16A3 0 40 CC[C@H]1CN(S(=O)(=O)c2ccc3c(c2)CCC3)CC[C@@H]1N ZINC000147407773 DD On-Demand Anodyne CASP7 50 34 Cc1c(CN2CCSCC2)cccc1NC(=O)c1cc2c(F)cccc2[nH]1 ZINC000147407793 GI On-Demand Anodyne CCKAR 21 46 CNC(=O)C1CCN(C(=O)c2cc(C)ccc2Br)CC1 ZINC000147407827 EE On-Demand Anodyne EPHX2 31 44 CNC(=O)C1CCN(C(=O)c2cc(C)ccc2Br)CC1 ZINC000147407827 EE On-Demand Anodyne L3MBTL1 0 41 CNC(=O)C1CCN(C(=O)c2cc(C)ccc2Br)CC1 ZINC000147407827 EE On-Demand Anodyne L3MBTL3 49 40 CNC(=O)C1CCN(C(=O)c2cc(C)ccc2Br)CC1 ZINC000147407827 EE On-Demand Anodyne MBTD1 0 41 CN(CC(F)(F)F)C(=O)[C@H]1CCCCN1C(=O)OC(C)(C)C ZINC000147407853 DF On-Demand Anodyne PREP 20 53 COc1ccc(OC)c(CCNC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147407859 HH On-Demand Anodyne NQO2 31 45 COc1ccc(OC)c(CCNC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147407859 HH On-Demand Anodyne MTNR1A 94 45 COc1ccc(OC)c(CCNC(=O)[C@H]2C[C@H]2c2cccc(Br)c2)c1 ZINC000147407859 HH On-Demand Anodyne MTNR1B 76 46 O=C(O)c1cc(Cl)cc(NC(=O)N(CCO)CCO)c1 ZINC000147407897 DC For-Sale Anodyne HCAR1 0 41 O=C(NCC1(C(=O)O)CCC1)c1cccc(I)c1 ZINC000147407937 FE On-Demand Anodyne KCNK3 62 34 Cc1nc(Oc2ccc([N+](=O)[O-])c(Cl)c2)ccc1C(=O)O ZINC000147407938 DG For-Sale Bother PPXII 0 45 CC(C)S(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3cccc(F)c3)no2)CC1 ZINC000147407953 GG Annotated Anodyne NPY5R 21 44 CSc1ncc(Cl)c(C(=O)Nc2cccc(CN3CCSCC3)c2C)n1 ZINC000147408003 HH On-Demand Anodyne MRGPRX1 44 37 COc1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1O ZINC000147408033 EG For-Sale Reactive ACKR3 67 36 COc1ccc(OC)c(CCNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147408067 FF On-Demand Anodyne NQO2 41 49 COc1ccc(OC)c(CCNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147408067 FF On-Demand Anodyne MTNR1A 122 49 COc1ccc(OC)c(CCNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147408067 FF On-Demand Anodyne MTNR1B 103 47 COc1ccc(OC)c(CCNC(=O)[C@H]2COc3cc(OC)ccc3C2)c1 ZINC000147408067 FF On-Demand Anodyne ROCK2 29 44 CN1CCN([C@@H](CN)c2ccc(Cl)cc2F)CC1 ZINC000147408102 CD For-Sale Anodyne MC4R 35 57 Cc1ccc(Br)c(C(=O)Nc2ccc3sccc3c2)c1 ZINC000147408154 EK For-Sale Anodyne KCNK3 64 35 Cc1ccc(Br)c(C(=O)Nc2ccc3sccc3c2)c1 ZINC000147408154 EK For-Sale Anodyne KCNK9 58 35 Cc1nc(Oc2cc(Cl)ccc2[N+](=O)[O-])ccc1C(=O)O ZINC000147408200 DG For-Sale Bother ENR 0 40 COc1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1O ZINC000147408266 EG For-Sale Reactive ACKR3 67 36 CN1CCN([C@H](CN)c2ccc(Cl)cc2F)CC1 ZINC000147408279 CD For-Sale Anodyne MC4R 35 57 O=C(NCC1(c2ccc(Cl)cc2)CCOCC1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147408335 GI On-Demand Anodyne EPHX2 27 42 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H]1CCCOc3ccc(F)cc31)C2 ZINC000147408338 FG On-Demand Anodyne ROCK2 23 40 CC(C)Oc1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147408355 GI On-Demand Anodyne HRH2 25 42 CC(C)Oc1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147408355 GI On-Demand Anodyne EPHX2 21 43 CCS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3cccc(F)c3)no2)CC1 ZINC000147408370 GF Annotated Anodyne NPY2R 0 40 CCS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3cccc(F)c3)no2)CC1 ZINC000147408370 GF Annotated Anodyne GRM5 0 40 CCS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3cccc(F)c3)no2)CC1 ZINC000147408370 GF Annotated Anodyne GPR39 0 41 CCOc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147408432 CG For-Sale Anodyne PPARG 26 40 CCOc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147408432 CG For-Sale Anodyne DHODH 18 40 CCOc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147408432 CG For-Sale Anodyne P2RX3 16 40 CCOc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147408432 CG For-Sale Anodyne ACACA 0 40 CCOc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147408432 CG For-Sale Anodyne TRY1_BOVIN 38 51 CCOc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147408432 CG For-Sale Anodyne CCKAR 56 37 CCOc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147408432 CG For-Sale Anodyne ALS 55 40 CCOc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147408432 CG For-Sale Anodyne PDS 42 34 Cc1[nH]c2ccc(C(=O)Nc3cccc(CN4CCSCC4)c3C)cc2c1C ZINC000147408490 GJ On-Demand Anodyne MRGPRX1 45 42 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H]1CCCOc3ccc(F)cc31)C2 ZINC000147408493 FG On-Demand Anodyne ROCK2 23 40 CCOc1ccccc1-c1nnnn1C1(C(=O)O)CCC1 ZINC000147408510 CD For-Sale Anodyne HCN1 49 34 CCOc1ccccc1-c1nnnn1C1(C(=O)O)CCC1 ZINC000147408510 CD For-Sale Anodyne HCN4 42 33 O=C(NCC1(c2ccc(Cl)cc2)CCOCC1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147408527 GI On-Demand Anodyne EPHX2 27 42 CCCc1nc2c(C(=O)O)cccc2n1CCNC(N)=O ZINC000147408553 CD For-Sale Anodyne AGTR1 53 43 CCCc1nc2c(C(=O)O)cccc2n1CCNC(N)=O ZINC000147408553 CD For-Sale Anodyne AGTR2 25 43 CCCc1nc2c(C(=O)O)cccc2n1CCNC(N)=O ZINC000147408553 CD For-Sale Anodyne AGTR1B 36 41 CC(C)Oc1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147408558 GI On-Demand Anodyne HRH2 25 42 CC(C)Oc1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147408558 GI On-Demand Anodyne EPHX2 21 43 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2[nH]1 ZINC000147408594 FJ On-Demand Anodyne MAOB 22 50 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2[nH]1 ZINC000147408594 FJ On-Demand Anodyne HPSE 18 42 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2[nH]1 ZINC000147408594 FJ On-Demand Anodyne TAAR1 19 42 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2[nH]1 ZINC000147408594 FJ On-Demand Anodyne NR2E3 82 47 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2[nH]1 ZINC000147408594 FJ On-Demand Anodyne SHH 55 44 Cc1nc2cc(NC(=O)c3ccc(Br)c(Cl)c3)ccc2[nH]1 ZINC000147408594 FJ On-Demand Anodyne KCNK3 57 37 CN(CC(F)(F)F)C(=O)[C@@H]1CCCCN1C(=O)OC(C)(C)C ZINC000147408619 DF On-Demand Anodyne PREP 20 53 Cc1nc(Oc2ccc(F)cc2[N+](=O)[O-])ccc1C(=O)O ZINC000147408681 CF For-Sale Bother ALS 25 41 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H]1CCCOc3ccc(F)cc31)C2 ZINC000147408701 FG On-Demand Anodyne ROCK2 23 40 O=C(NCC1(c2ccc(Cl)cc2)CCOCC1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147408709 GI On-Demand Anodyne EPHX2 27 42 c1cnc(Cn2ccnc2)cn1 ZINC000147408714 AC For-Sale Anodyne CYP19A1 31 47 c1cnc(Cn2ccnc2)cn1 ZINC000147408714 AC For-Sale Anodyne CYP11B1 62 54 c1cnc(Cn2ccnc2)cn1 ZINC000147408714 AC For-Sale Anodyne TBXAS1 37 47 c1cnc(Cn2ccnc2)cn1 ZINC000147408714 AC For-Sale Anodyne CYP11B2 30 47 c1cnc(Cn2ccnc2)cn1 ZINC000147408714 AC For-Sale Anodyne CYP17A1 15 44 Cc1nn(C)c(C)c1[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147408724 HE On-Demand Anodyne CHRM5 16 40 Cc1nn(C)c(C)c1[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147408724 HE On-Demand Anodyne TGM2 49 41 Cc1nn(C)c(C)c1[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147408724 HE On-Demand Anodyne F13A1 43 41 Cc1ccc(Br)c(C(=O)Nc2ccc3[nH]c(C)nc3c2)c1 ZINC000147408830 EI On-Demand Anodyne HPSE 15 46 Cc1ccc(Br)c(C(=O)Nc2ccc3[nH]c(C)nc3c2)c1 ZINC000147408830 EI On-Demand Anodyne NR2E3 79 45 Cc1ccc(Br)c(C(=O)Nc2ccc3[nH]c(C)nc3c2)c1 ZINC000147408830 EI On-Demand Anodyne KCNK3 54 33 Cc1ccc(Br)c(C(=O)Nc2ccc3[nH]c(C)nc3c2)c1 ZINC000147408830 EI On-Demand Anodyne KCNK9 48 33 O=S(=O)(c1ccc2c(c1)CCC2)N1CCCC[C@@H]1CBr ZINC000147408853 FG For-Sale Reactive CASP3 121 44 O=S(=O)(c1ccc2c(c1)CCC2)N1CCCC[C@@H]1CBr ZINC000147408853 FG For-Sale Reactive CASP7 121 43 O=S(=O)(c1ccc2c(c1)CCC2)N1CCCC[C@@H]1CBr ZINC000147408853 FG For-Sale Reactive AKR1C3 28 40 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(N3CCCC3=O)cc2)C1 ZINC000147408885 HE On-Demand Anodyne AKR1C3 24 46 O=C(C[C@@H]1CNc2ccccc21)NCc1c[nH]cn1 ZINC000147408917 CD For-Sale Anodyne HRAS 45 30 O=C(C[C@@H]1CNc2ccccc21)NCc1c[nH]cn1 ZINC000147408917 CD For-Sale Anodyne HRH3 35 41 C=CCCO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147408924 GE On-Demand Mild TGM2 91 49 C=CCCO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147408924 GE On-Demand Mild F13A1 98 49 CCCc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147408952 CH For-Sale Anodyne P2RX3 15 40 CCCc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147408952 CH For-Sale Anodyne P2RX1 24 40 O=S(=O)(c1ccc2c(c1)CCC2)N1CCCC[C@H]1CBr ZINC000147409064 FG For-Sale Reactive CASP3 121 44 O=S(=O)(c1ccc2c(c1)CCC2)N1CCCC[C@H]1CBr ZINC000147409064 FG For-Sale Reactive CASP7 121 43 O=S(=O)(c1ccc2c(c1)CCC2)N1CCCC[C@H]1CBr ZINC000147409064 FG For-Sale Reactive AKR1C3 28 40 CC(C)CCCCNCc1ccc(-c2ccccc2)cc1 ZINC000147409084 CK For-Sale Anodyne SLC15A1 0 40 CC(C)CCCCNCc1ccc(-c2ccccc2)cc1 ZINC000147409084 CK For-Sale Anodyne LPAR2 26 41 CC(C)CCCCNCc1ccc(-c2ccccc2)cc1 ZINC000147409084 CK For-Sale Anodyne S1PR2 31 41 CC(C)CCCCNCc1ccc(-c2ccccc2)cc1 ZINC000147409084 CK For-Sale Anodyne LEF 77 39 CC(C)CCCCNCc1ccc(-c2ccccc2)cc1 ZINC000147409084 CK For-Sale Anodyne GPM3 0 53 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(N3CCCC3=O)cc2)C1 ZINC000147409089 HE On-Demand Anodyne AKR1C3 24 46 C=CCCO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147409119 GE On-Demand Mild TGM2 91 49 C=CCCO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147409119 GE On-Demand Mild F13A1 98 49 O=C(C[C@H]1CNc2ccccc21)NCc1c[nH]cn1 ZINC000147409135 CD For-Sale Anodyne HRAS 45 30 O=C(C[C@H]1CNc2ccccc21)NCc1c[nH]cn1 ZINC000147409135 CD For-Sale Anodyne HRH3 35 41 CC(=C/C(=O)O)/C=C/[C@H]1CC=CCC1 ZINC000147409170 AF For-Sale Anodyne RXRG 29 40 CC(=C/C(=O)O)/C=C/[C@H]1CC=CCC1 ZINC000147409170 AF For-Sale Anodyne RXRA 26 40 CC(=C/C(=O)O)/C=C/[C@H]1CC=CCC1 ZINC000147409170 AF For-Sale Anodyne RXRB 30 40 Cc1ccc(Br)c(C(=O)N[C@@H](c2ccccc2)C2CC2)c1 ZINC000147409193 EJ On-Demand Anodyne TACR3 17 43 Cc1cccnc1NC(=O)C1CCN(C(=O)COc2ccc(C(N)=O)cc2)CC1 ZINC000147409244 GD On-Demand Anodyne CPT1A 72 39 COc1cc(N)cc(-c2ccccc2)c1 ZINC000147409283 AF In-Stock Anodyne DFR1 25 42 COc1cc(N)cc(-c2ccccc2)c1 ZINC000147409283 AF In-Stock Anodyne DFRA 0 42 NCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147409299 CD For-Sale Anodyne HCAR1 0 41 CC(=C/C(=O)O)/C=C/[C@@H]1CC=CCC1 ZINC000147409356 AF For-Sale Anodyne RXRG 29 40 CC(=C/C(=O)O)/C=C/[C@@H]1CC=CCC1 ZINC000147409356 AF For-Sale Anodyne RXRA 26 40 CC(=C/C(=O)O)/C=C/[C@@H]1CC=CCC1 ZINC000147409356 AF For-Sale Anodyne RXRB 30 40 Cc1ccc(Br)c(C(=O)N[C@H](c2ccccc2)C2CC2)c1 ZINC000147409389 EJ On-Demand Anodyne TACR3 17 43 CC(C)CC(C)(C)C[C@H]1N[C@@H](C(=O)NCC[C@H](O)CO)[C@H](c2cccc(Cl)c2)[C@@]12C(=O)Nc1cc(F)c(F)cc12 ZINC000147409475 KI Annotated Anodyne MDM2 79 79 O=C(Nc1cc(Br)cc(C(=O)O)c1)NC1CCNCC1 ZINC000147409528 EE For-Sale Anodyne EPHX2 43 40 Cc1cc(C)n([C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1 ZINC000147409553 HE On-Demand Anodyne CHRM5 20 40 Cc1cc(C)n([C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1 ZINC000147409553 HE On-Demand Anodyne EPHX2 27 40 Cc1cc(C)n([C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1 ZINC000147409553 HE On-Demand Anodyne TGM2 67 43 Cc1cc(C)n([C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1 ZINC000147409553 HE On-Demand Anodyne F13A1 67 43 C[C@@H]1CN(c2ccc(C(F)(F)F)c(F)c2)C[C@@H](C)N1 ZINC000147409554 CG For-Sale Anodyne GHSR 39 42 CCCCCCCCNS(=O)(=O)[C@@H](C)CNCCC ZINC000147409572 CF For-Sale Mild RELA 17 40 CCCCCCCCNS(=O)(=O)[C@@H](C)CNCCC ZINC000147409572 CF For-Sale Mild Q8WS26_TRYCR 40 45 CCCCCCCCNS(=O)(=O)[C@@H](C)CNCCC ZINC000147409572 CF For-Sale Mild FPPS 0 45 CCCCCCCCNS(=O)(=O)[C@@H](C)CNCCC ZINC000147409572 CF For-Sale Mild SPPS 0 45 CC(C)Oc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147409637 HH On-Demand Anodyne CA2 28 53 CC(C)Oc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147409637 HH On-Demand Anodyne BMP1 42 48 CC(C)Oc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147409637 HH On-Demand Anodyne CA1 56 39 CC(C)Oc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147409637 HH On-Demand Anodyne CA4 15 46 CC(C)Oc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147409637 HH On-Demand Anodyne MMP3 15 45 CC(C)Oc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147409637 HH On-Demand Anodyne CA12 37 53 CC(C)Oc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147409637 HH On-Demand Anodyne CA9 42 53 CC(C)Oc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147409637 HH On-Demand Anodyne NCE103 32 49 CC(C)Oc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147409637 HH On-Demand Anodyne PRMT3 17 40 CC(C)Oc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147409637 HH On-Demand Anodyne P96878_MYCTU 41 37 CC(C)Oc1ccc(NC(=O)NCc2ccc(S(=O)(=O)N(C)C(C)C)cc2)cc1 ZINC000147409637 HH On-Demand Anodyne NAMPT 51 45 NS(=O)(=O)c1cc(F)cc(F)c1OCCN1CCCCC1 ZINC000147409667 DD For-Sale Anodyne LTA4H 31 42 NS(=O)(=O)c1cc(F)cc(F)c1OCCN1CCCCC1 ZINC000147409667 DD For-Sale Anodyne HRH3 20 44 NS(=O)(=O)c1cc(F)cc(F)c1OCCN1CCCCC1 ZINC000147409667 DD For-Sale Anodyne PSMB2 47 38 NS(=O)(=O)c1cc(F)cc(F)c1OCCN1CCCCC1 ZINC000147409667 DD For-Sale Anodyne PSMB1 41 38 Cc1cc(-c2nc(-c3cncs3)no2)ccc1N ZINC000147409736 CF For-Sale Anodyne CD38 47 31 Cc1cc(C)n([C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1 ZINC000147409751 HE On-Demand Anodyne CHRM5 20 40 Cc1cc(C)n([C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1 ZINC000147409751 HE On-Demand Anodyne EPHX2 27 40 Cc1cc(C)n([C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1 ZINC000147409751 HE On-Demand Anodyne TGM2 67 43 Cc1cc(C)n([C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1 ZINC000147409751 HE On-Demand Anodyne F13A1 67 43 COCc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147409753 CG For-Sale Anodyne P2RX3 16 44 COCc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147409753 CG For-Sale Anodyne TRY1_BOVIN 28 44 COCc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147409753 CG For-Sale Anodyne ALS 66 33 COCc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147409753 CG For-Sale Anodyne CRTM 43 31 COCc1cccc(Oc2ccc(C(=O)O)c(C)n2)c1 ZINC000147409753 CG For-Sale Anodyne HAO2 29 41 O=C(Nc1cc(Cl)cc(C(=O)O)c1)NC1CCNCC1 ZINC000147409764 CD For-Sale Anodyne EPHX2 46 51 CN(C)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cn1 ZINC000147409771 FH On-Demand Anodyne MAOB 18 40 CN(C)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cn1 ZINC000147409771 FH On-Demand Anodyne CSF1R 21 43 CN(C)c1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cn1 ZINC000147409771 FH On-Demand Anodyne TAAR1 19 44 C[C@H]1CN(c2ccc(C(F)(F)F)c(F)c2)C[C@H](C)N1 ZINC000147409781 CG For-Sale Anodyne GHSR 39 42 CCCCCCCCNS(=O)(=O)[C@H](C)CNCCC ZINC000147409805 CF For-Sale Mild RELA 17 40 CCCCCCCCNS(=O)(=O)[C@H](C)CNCCC ZINC000147409805 CF For-Sale Mild Q8WS26_TRYCR 40 45 CCCCCCCCNS(=O)(=O)[C@H](C)CNCCC ZINC000147409805 CF For-Sale Mild FPPS 0 45 CCCCCCCCNS(=O)(=O)[C@H](C)CNCCC ZINC000147409805 CF For-Sale Mild SPPS 0 45 CC(C)Oc1ccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147409890 FG On-Demand Anodyne PDGFRB 24 42 CC(C)Oc1ccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147409890 FG On-Demand Anodyne EPHX2 47 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc2c1OCCO2 ZINC000147409985 HE On-Demand Anodyne HTR4 66 61 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc2c1OCCO2 ZINC000147409985 HE On-Demand Anodyne PKM 31 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc2c1OCCO2 ZINC000147409985 HE On-Demand Anodyne TGM2 54 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc2c1OCCO2 ZINC000147409985 HE On-Demand Anodyne F13A1 41 42 CC(C)Oc1ccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147410073 DI On-Demand Anodyne CA1 42 36 CC(C)Oc1ccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147410073 DI On-Demand Anodyne EPHX2 58 44 CC(C)Oc1ccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147410073 DI On-Demand Anodyne KDM1A 45 40 O=S(=O)(c1c(F)cc(F)cc1F)N1CCCC[C@@H]1CBr ZINC000147410103 FG For-Sale Reactive CASP7 48 35 CCCCCCCCNCCCCC(C)C ZINC000147410117 BJ For-Sale Mild ADH1A 0 47 CCCCCCCCNCCCCC(C)C ZINC000147410117 BJ For-Sale Mild ADH7 0 44 CCCCCCCCNCCCCC(C)C ZINC000147410117 BJ For-Sale Mild S1PR3 21 50 CCCCCCCCNCCCCC(C)C ZINC000147410117 BJ For-Sale Mild S1PR2 47 50 CCCCCCCCNCCCCC(C)C ZINC000147410117 BJ For-Sale Mild ADH1B 0 47 CCCCCCCCNCCCCC(C)C ZINC000147410117 BJ For-Sale Mild ADH1C 0 47 CCCCCCCCNCCCCC(C)C ZINC000147410117 BJ For-Sale Mild Q8WS26_TRYCR 41 42 CCCCCCCCNCCCCC(C)C ZINC000147410117 BJ For-Sale Mild FPPS 0 42 CCCCCCCCNCCCCC(C)C ZINC000147410117 BJ For-Sale Mild SPPS 0 42 O=C(NCC1(C(=O)O)CCC1)c1cc(C2CC2)on1 ZINC000147410132 CD On-Demand Anodyne S1PR3 23 47 Fc1cc(OCc2ccc(CNC3CC3)o2)ccc1Cl ZINC000147410190 CH For-Sale Anodyne ENV 43 34 NC1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147410195 CD For-Sale Anodyne CACNA1H 42 36 NC1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147410195 CD For-Sale Anodyne EPHX2 17 41 NC1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147410195 CD For-Sale Anodyne CACNA1I 59 38 COc1c(Br)cc(Cl)cc1NC(=O)c1cc(C)ccc1Br ZINC000147410208 IK On-Demand Anodyne KCNMA1 35 47 COc1c(Br)cc(Cl)cc1NC(=O)c1cc(C)ccc1Br ZINC000147410208 IK On-Demand Anodyne GPR35 42 36 CC(C)Oc1ccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147410259 DI On-Demand Anodyne CA1 42 36 CC(C)Oc1ccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147410259 DI On-Demand Anodyne EPHX2 58 44 CC(C)Oc1ccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)cc1 ZINC000147410259 DI On-Demand Anodyne KDM1A 45 40 O=S(=O)(c1c(F)cc(F)cc1F)N1CCCC[C@H]1CBr ZINC000147410335 FG For-Sale Reactive CASP7 48 35 Cn1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1C1CC1 ZINC000147410434 HE On-Demand Anodyne HTR4 67 39 Cn1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1C1CC1 ZINC000147410434 HE On-Demand Anodyne TGM2 62 42 Cn1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1C1CC1 ZINC000147410434 HE On-Demand Anodyne CACNA1I 58 37 Cn1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1C1CC1 ZINC000147410434 HE On-Demand Anodyne F13A1 55 42 Cn1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1C1CC1 ZINC000147410434 HE On-Demand Anodyne NAMPT 40 38 O=C(O)C1(n2nnnc2C2(c3ccccc3)CC2)CCC1 ZINC000147410460 CD For-Sale Anodyne HSD11B1 15 42 CC(C)Oc1ccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147410469 DI On-Demand Anodyne CA1 42 36 CC(C)Oc1ccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147410469 DI On-Demand Anodyne EPHX2 58 44 CC(C)Oc1ccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)cc1 ZINC000147410469 DI On-Demand Anodyne KDM1A 45 40 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@H](C(F)(F)F)C1 ZINC000147410477 FJ On-Demand Anodyne RHOA 0 41 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@H](C(F)(F)F)C1 ZINC000147410477 FJ On-Demand Anodyne L3MBTL3 56 39 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@H](C(F)(F)F)C1 ZINC000147410477 FJ On-Demand Anodyne HPGD 28 49 Cc1cc(C#N)cc(C)c1Oc1ccc(C(=O)O)c(C)n1 ZINC000147410594 CG For-Sale Mild HIVRT 0 43 CC(C)Oc1ccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147410616 DI On-Demand Anodyne CA1 42 36 CC(C)Oc1ccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147410616 DI On-Demand Anodyne EPHX2 58 44 CC(C)Oc1ccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)cc1 ZINC000147410616 DI On-Demand Anodyne KDM1A 45 40 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@@H](C(F)(F)F)C1 ZINC000147410683 FJ On-Demand Anodyne RHOA 0 41 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@@H](C(F)(F)F)C1 ZINC000147410683 FJ On-Demand Anodyne L3MBTL3 56 39 O=C(c1ccc(Br)c(Cl)c1)N1CCC[C@@H](C(F)(F)F)C1 ZINC000147410683 FJ On-Demand Anodyne HPGD 28 49 Cc1cccc2cc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)oc12 ZINC000147410695 HH On-Demand Anodyne HTR4 53 36 Cc1cccc2cc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)oc12 ZINC000147410695 HH On-Demand Anodyne EPHX2 31 41 Cc1cccc2cc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)oc12 ZINC000147410695 HH On-Demand Anodyne TGM2 54 42 Cc1cccc2cc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)oc12 ZINC000147410695 HH On-Demand Anodyne CACNA1I 58 36 Cc1cccc2cc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)oc12 ZINC000147410695 HH On-Demand Anodyne F13A1 43 42 Cc1cccc2cc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)oc12 ZINC000147410695 HH On-Demand Anodyne NAMPT 44 40 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2ncccc2C)CC1 ZINC000147410727 FD On-Demand Anodyne P2RY12 166 37 Cc1nc2cccc(Cl)c2n1[C@@H]1CCNC1 ZINC000147410744 BF For-Sale Anodyne JAK1 25 44 Cc1ccc(C(=O)N2CC[C@@H](NC(N)=O)C2)cn1 ZINC000147410827 BC On-Demand Anodyne L3MBTL3 48 36 Cc1nc2cccc(Cl)c2n1[C@H]1CCNC1 ZINC000147410860 BF For-Sale Anodyne JAK1 25 44 CNCc1coc(COc2ccc(Cl)c(F)c2)c1 ZINC000147410866 CG For-Sale Anodyne DAO 15 44 Cc1nn(C(F)F)c(C)c1CC(=O)N1CCc2[nH]c3ccc(F)cc3c2C1 ZINC000147410878 GH On-Demand Anodyne P2RX7 23 40 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147410890 HD On-Demand Anodyne HTR4 43 36 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147410890 HD On-Demand Anodyne GRIN2B 28 43 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147410890 HD On-Demand Anodyne EPHX2 16 43 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147410890 HD On-Demand Anodyne TGM2 65 44 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147410890 HD On-Demand Anodyne CACNA1I 61 38 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147410890 HD On-Demand Anodyne F13A1 56 44 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147410890 HD On-Demand Anodyne NAMPT 55 46 CNc1cc(Oc2cccc3cccnc23)nc(C)n1 ZINC000147410898 CG For-Sale Anodyne C0L093_TOBAC 55 33 COC(=O)Cc1ccc(C)c(Cl)c1 ZINC000147410919 AE For-Sale Anodyne NCE103 32 50 COC(=O)Cc1ccc(C)c(Cl)c1 ZINC000147410919 AE For-Sale Anodyne PFK 0 42 COC(=O)Cc1ccc(C)c(Cl)c1 ZINC000147410919 AE For-Sale Anodyne P96878_MYCTU 19 43 COC(=O)Cc1ccc(C)c(Cl)c1 ZINC000147410919 AE For-Sale Anodyne CAN2 0 50 N[C@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147410939 CD For-Sale Anodyne CACNA1I 56 39 N#Cc1ncccc1/C=C/C(=O)O ZINC000147411007 AD For-Sale Anodyne PTGER2 36 44 N#Cc1ncccc1/C=C/C(=O)O ZINC000147411007 AD For-Sale Anodyne PTGER4 20 44 N#Cc1ncccc1/C=C/C(=O)O ZINC000147411007 AD For-Sale Anodyne PTGER3 19 44 Cc1cc(C(=O)N2CCC(C(=O)Nc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147411034 FG On-Demand Bother CCKAR 0 42 Cc1cc(C(=O)N2CCC(C(=O)Nc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147411034 FG On-Demand Bother NPY2R 17 42 Cc1cc(C(=O)N2CCC(C(=O)Nc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147411034 FG On-Demand Bother EPHX2 36 48 Cc1cc(C(=O)N2CCC(C(=O)Nc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147411034 FG On-Demand Bother LIMK2 17 40 Cc1cc(C(=O)N2CCC(C(=O)Nc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147411034 FG On-Demand Bother L3MBTL3 60 34 Cc1nccn1-c1ccc(CNC(=O)Nc2ccc(OC(C)C)cc2)cc1F ZINC000147411042 GI On-Demand Anodyne ROCK2 17 41 COc1cc(Br)c(Oc2ccc(C(=O)O)c(C)n2)cc1Br ZINC000147411058 HI For-Sale Anodyne ALS 81 40 CCCCCCCCCCCCCCCCc1c(C)n(O)c2ccccc2[n+]1=O ZINC000147411064 HK In-Stock Mild OXER1 48 37 N[C@@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147411118 CD For-Sale Anodyne CACNA1I 56 39 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(C)c(OC)c1)C2 ZINC000147411200 EF On-Demand Anodyne MTNR1A 36 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCc1ccc(C)c(OC)c1)C2 ZINC000147411200 EF On-Demand Anodyne ROCK2 31 44 O=C1C[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147411231 FC On-Demand Anodyne FKBP1A 15 41 O=C1C[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147411231 FC On-Demand Anodyne EPHX2 38 46 O=C1C[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147411231 FC On-Demand Anodyne TGM2 62 44 O=C1C[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147411231 FC On-Demand Anodyne F13A1 66 44 CC(C)Oc1ccc(NC(=O)N2CCO[C@H](c3ccc(Br)cc3)C2)cc1 ZINC000147411264 HJ On-Demand Anodyne PDGFRB 18 40 Nc1ccccc1NC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147411326 FG For-Sale Anodyne HDAC1 36 45 Nc1ccccc1NC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147411326 FG For-Sale Anodyne HDAC2 21 45 Nc1ccccc1NC(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147411326 FG For-Sale Anodyne HDAC3 0 48 O=C1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147411372 FC On-Demand Anodyne FKBP1A 15 41 O=C1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147411372 FC On-Demand Anodyne EPHX2 38 46 O=C1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147411372 FC On-Demand Anodyne TGM2 62 44 O=C1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147411372 FC On-Demand Anodyne F13A1 66 44 CC(C)Oc1ccc(NC(=O)N2CCO[C@@H](c3ccc(Br)cc3)C2)cc1 ZINC000147411417 HJ On-Demand Anodyne PDGFRB 18 40 COc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147411491 CD On-Demand Anodyne DRD4 59 45 COc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147411491 CD On-Demand Anodyne MTNR1A 48 38 COc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147411491 CD On-Demand Anodyne MTNR1B 38 45 COc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147411491 CD On-Demand Anodyne TAAR1 35 43 COc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147411491 CD On-Demand Anodyne AKR1C3 26 41 COc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147411491 CD On-Demand Anodyne KCNK3 76 55 COc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147411491 CD On-Demand Anodyne KCNK9 53 35 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)N3CCOCC3)c(Cl)c2)c1 ZINC000147411498 HF On-Demand Bother AVPR2 39 45 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)N3CCOCC3)c(Cl)c2)c1 ZINC000147411498 HF On-Demand Bother PTK6 29 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)N3CCOCC3)c(Cl)c2)c1 ZINC000147411498 HF On-Demand Bother TAAR1 26 49 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)N3CCOCC3)c(Cl)c2)c1 ZINC000147411498 HF On-Demand Bother AKR1C2 44 38 Nc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147411563 DG For-Sale Anodyne PPIA 27 48 Nc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147411563 DG For-Sale Anodyne LPL 44 33 Nc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147411563 DG For-Sale Anodyne PTGER3 25 40 Nc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147411563 DG For-Sale Anodyne HDAC1 39 45 Nc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147411563 DG For-Sale Anodyne HDAC2 23 45 Nc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147411563 DG For-Sale Anodyne HDAC3 0 48 Nc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147411563 DG For-Sale Anodyne AKR1C3 28 41 Nc1ccccc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147411563 DG For-Sale Anodyne DDX3X 0 40 Cc1ccnc(NC(=O)C2CCN(C(=O)C(=O)c3ccc4c(c3)CCC4)CC2)c1 ZINC000147411628 GF On-Demand Anodyne TYK2 45 36 O=C(Nc1cccc2cn[nH]c12)c1ccc(Br)c(Cl)c1 ZINC000147411709 FI On-Demand Anodyne MAOB 19 45 CC(C)CCCCNS(=O)(=O)CCCCN ZINC000147411787 CD For-Sale Anodyne RELA 24 54 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)N(C)c3ccccc3)c2)c1 ZINC000147411893 HI On-Demand Bother PYGL 24 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)N(C)c3ccccc3)c2)c1 ZINC000147411893 HI On-Demand Bother MTNR1B 17 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)N(C)c3ccccc3)c2)c1 ZINC000147411893 HI On-Demand Bother HSD17B2 19 47 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)N(C)c3ccccc3)c2)c1 ZINC000147411893 HI On-Demand Bother TAAR1 36 51 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)N(C)c3ccccc3)c2)c1 ZINC000147411893 HI On-Demand Bother AKR1C3 38 52 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)N(C)c3ccccc3)c2)c1 ZINC000147411893 HI On-Demand Bother AKR1C2 57 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)N(C)c3ccccc3)c2)c1 ZINC000147411893 HI On-Demand Bother KCNK3 110 47 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)N(C)c3ccccc3)c2)c1 ZINC000147411893 HI On-Demand Bother KCNK9 75 39 CCCC[C@H](NC(N)=O)C(=O)N1CCc2[nH]c3ccc(C)cc3c2C1 ZINC000147411901 EF On-Demand Anodyne P2RY12 55 33 CCCC[C@H](NC(N)=O)C(=O)N1CCc2[nH]c3ccc(C)cc3c2C1 ZINC000147411901 EF On-Demand Anodyne TRY2_BOVIN 41 31 CNCCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147411958 CD For-Sale Anodyne CACNA1H 24 40 CC(C)Oc1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147411997 FJ On-Demand Anodyne EPHX2 16 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCc2[nH]c3ccc(C)cc3c2C1 ZINC000147412028 EF On-Demand Anodyne P2RY12 55 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCc2[nH]c3ccc(C)cc3c2C1 ZINC000147412028 EF On-Demand Anodyne TRY2_BOVIN 41 31 CCOc1ccccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147412112 FJ On-Demand Anodyne FABH 0 47 CCOc1ccccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147412112 FJ On-Demand Anodyne TAAR1 19 41 CCOc1ccccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147412112 FJ On-Demand Anodyne KCNK3 46 43 CCOc1ccccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147412112 FJ On-Demand Anodyne KCNK9 46 43 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2cc(C)ccn2)CC1 ZINC000147412141 FD On-Demand Anodyne P2RY12 135 35 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2cc(C)ccn2)CC1 ZINC000147412141 FD On-Demand Anodyne MAPK10 15 40 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2cc(C)ccn2)CC1 ZINC000147412141 FD On-Demand Anodyne TYK2 40 35 CCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)Nc2cc(C)ccn2)CC1 ZINC000147412141 FD On-Demand Anodyne ST14 44 34 CC(C)Oc1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147412143 FJ On-Demand Anodyne EPHX2 16 44 CCc1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147412182 GF On-Demand Anodyne HTR4 50 38 CCc1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147412182 GF On-Demand Anodyne EPHX2 16 43 CCc1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147412182 GF On-Demand Anodyne TGM2 63 42 CCc1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147412182 GF On-Demand Anodyne CACNA1I 56 34 CCc1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147412182 GF On-Demand Anodyne F13A1 51 42 CCc1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147412182 GF On-Demand Anodyne SIRT3 41 33 CCc1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147412182 GF On-Demand Anodyne SIRT1 41 33 CCc1ncc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147412182 GF On-Demand Anodyne NAMPT 45 40 CC(C)Oc1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147412273 FJ On-Demand Anodyne EPHX2 16 44 Cc1nc(Oc2ccc(C(N)=O)c(F)c2)ccc1C(=O)O ZINC000147412310 CE For-Sale Anodyne TRY1_BOVIN 27 41 O=C(NCC1(C(=O)O)CCC1)c1ccccc1I ZINC000147412314 FE On-Demand Anodyne KCNA3 40 41 O=C(NCC1(C(=O)O)CCC1)c1ccccc1I ZINC000147412314 FE On-Demand Anodyne HCN1 63 36 O=C(NCC1(C(=O)O)CCC1)c1ccccc1I ZINC000147412314 FE On-Demand Anodyne HCN4 53 34 CS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3cccc(Cl)c3)no2)CC1 ZINC000147412325 GF Annotated Anodyne NPY2R 32 41 CS(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3cccc(Cl)c3)no2)CC1 ZINC000147412325 GF Annotated Anodyne GRM5 22 41 O=C(Nc1ccccc1OC(F)F)c1ccc(Br)c(Cl)c1 ZINC000147412352 GJ On-Demand Anodyne FABH 0 45 O=C(Nc1ccccc1OC(F)F)c1ccc(Br)c(Cl)c1 ZINC000147412352 GJ On-Demand Anodyne TAAR1 23 41 CCCOCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147412364 FD On-Demand Anodyne CHRM5 28 40 CCCOCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147412364 FD On-Demand Anodyne EPHX2 29 40 CCCOCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147412364 FD On-Demand Anodyne TGM2 64 45 CCCOCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147412364 FD On-Demand Anodyne CACNA1I 47 35 CCCOCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147412364 FD On-Demand Anodyne F13A1 71 45 CC(C)CCCCN[C@@H](C)c1ccc(OC(C)C)cc1 ZINC000147412383 CJ For-Sale Anodyne ACACA 0 40 Cc1ccc(NC(=O)C2CC2)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@H](C)C1 ZINC000147412410 HF On-Demand Anodyne HRH3 26 43 CCNCCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147412413 CE For-Sale Anodyne CACNA1H 24 41 CC(C)Oc1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147412428 FJ On-Demand Anodyne EPHX2 16 44 CC(C)CCCCN[C@H](C)c1ccc(OC(C)C)cc1 ZINC000147412535 CJ For-Sale Anodyne ACACA 0 40 CCCCCCCCNS(=O)(=O)c1cnn(CCCN)c1 ZINC000147412564 DD For-Sale Mild ASAH1 46 32 COc1ccc(N/C(=C/[N+](=O)[O-])NCCCn2cncc2C)c(OC)c1 ZINC000147412580 FE Annotated Anodyne QPCT 103 64 Cc1ccc(NC(=O)C2CC2)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@@H](C)C1 ZINC000147412611 HF On-Demand Anodyne HRH3 26 43 Cc1ccccc1-n1nc(C(=O)NCc2cccc(Cn3ccnc3)c2)c2c1CCC2 ZINC000147412619 HH On-Demand Anodyne CYP11B1 28 43 Cc1ccccc1-n1nc(C(=O)NCc2cccc(Cn3ccnc3)c2)c2c1CCC2 ZINC000147412619 HH On-Demand Anodyne TBXAS1 33 40 Cc1ccccc1-n1nc(C(=O)NCc2cccc(Cn3ccnc3)c2)c2c1CCC2 ZINC000147412619 HH On-Demand Anodyne CYP11B2 32 43 Cc1ccccc1-n1nc(C(=O)NCc2cccc(Cn3ccnc3)c2)c2c1CCC2 ZINC000147412619 HH On-Demand Anodyne NOS2 47 32 CCn1nc(C)c2c1CCN([C@@H](C(=O)NC)c1ccccc1)[C@H]2CCc1ccccc1F ZINC000147412663 II Annotated Anodyne HCRTR1 0 48 CCn1nc(C)c2c1CCN([C@@H](C(=O)NC)c1ccccc1)[C@H]2CCc1ccccc1F ZINC000147412663 II Annotated Anodyne HCRTR2 42 78 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne MAOB 26 68 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne HTR1F 19 41 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne CPT1A 59 38 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne PRNP 40 37 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne FLT1 20 43 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne GRM4 40 38 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne AGPAT2 27 40 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne RPS6KA3 44 39 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne CSF1R 26 44 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne TAAR1 37 49 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne SHH 63 38 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne RORC 26 42 Cn1ccc2cc(C(=O)Nc3ccc(Cl)c(Cl)c3)ccc21 ZINC000147412695 DJ Annotated Anodyne KCNK3 65 38 CCOC[C@H](C)NC(=O)Nc1c(C)cc(Br)cc1C ZINC000147412702 EH On-Demand Anodyne PYGL 15 41 CC(C)CCCCNS(=O)(=O)c1ccc(F)c(CN)c1 ZINC000147412754 DE For-Sale Anodyne LEF 45 36 C=C(C)C[C@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412770 DI For-Sale Anodyne ALOX5 20 54 C=C(C)C[C@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412770 DI For-Sale Anodyne MAOB 47 41 C=C(C)C[C@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412770 DI For-Sale Anodyne PTGER3 46 38 C=C(C)C[C@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412770 DI For-Sale Anodyne ACE2 17 42 C=C(C)C[C@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412770 DI For-Sale Anodyne FFAR1 61 43 C=C(C)C[C@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412770 DI For-Sale Anodyne PDS 74 40 O=C(Nc1ccc(F)cc1F)c1cccnc1Oc1cccc(Br)c1 ZINC000147412771 HK On-Demand Anodyne P2RY1 27 56 O=C(Nc1ccc(F)cc1F)c1cccnc1Oc1cccc(Br)c1 ZINC000147412771 HK On-Demand Anodyne G2YM83_BOTF4 43 31 O=C(NCCCNC1CC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147412800 DE For-Sale Anodyne CACNA1I 43 36 CC(C)(C)S(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3ccc(F)cn3)no2)CC1 ZINC000147412910 HF Annotated Anodyne HCAR2 22 40 C=C(C)C[C@@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412922 DI For-Sale Anodyne ALOX5 20 54 C=C(C)C[C@@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412922 DI For-Sale Anodyne MAOB 47 41 C=C(C)C[C@@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412922 DI For-Sale Anodyne PTGER3 46 38 C=C(C)C[C@@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412922 DI For-Sale Anodyne ACE2 17 42 C=C(C)C[C@@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412922 DI For-Sale Anodyne FFAR1 61 43 C=C(C)C[C@@H](C(=O)OC)c1cccc(OCc2ccccc2)c1 ZINC000147412922 DI For-Sale Anodyne PDS 74 40 O=C([C@@H]1C[C@H]1c1cccc(Cl)c1)N1CCO[C@H]2CCC[C@@H]21 ZINC000147412966 DG On-Demand Anodyne MDM2 49 32 CC(C)CCCCNS(=O)(=O)CCN ZINC000147413016 BC For-Sale Anodyne RELA 20 45 O=C([C@@H]1C[C@@H]1c1cccc(Cl)c1)N1CCO[C@H]2CCC[C@@H]21 ZINC000147413080 DG On-Demand Anodyne MDM2 49 32 Cc1nc(Oc2ccc(Br)cc2C(C)C)ccc1C(=O)O ZINC000147413132 FJ For-Sale Anodyne PRS 55 34 CC[C@@H]1CN([C@@H]2CCC[C@@H]2O)CC[C@@H]1N ZINC000147413168 BC For-Sale Anodyne SLC18A3 36 44 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc3c(c2)OCO3)C1 ZINC000147413264 FD On-Demand Anodyne NOS2 42 32 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc3c(c2)OCO3)C1 ZINC000147413264 FD On-Demand Anodyne DYRK2 43 34 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc3c(c2)OCO3)C1 ZINC000147413264 FD On-Demand Anodyne TRPC6 25 40 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc3c(c2)OCO3)C1 ZINC000147413264 FD On-Demand Anodyne TRPC3 29 40 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne F2 52 42 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne SSTR2 23 43 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne P2RY12 94 36 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne CHRM5 37 40 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne CTSK 57 46 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne NPFFR2 43 31 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne PCSK5 36 46 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne FURIN 55 46 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne CTSS 18 42 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne TGM2 55 42 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne ST14 49 32 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne F13A1 50 42 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne POLG_WNV 59 38 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne NPFFR1 42 32 CCCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413279 HD On-Demand Anodyne TMPRSS6 55 32 CCCCc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147413294 CI For-Sale Anodyne INHA 80 38 CCCCc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147413294 CI For-Sale Anodyne RARB 22 42 CCCCc1ccc(Oc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147413294 CI For-Sale Anodyne AGTR1B 44 37 Cc1cccc(S(=O)(=O)Nc2ccccc2C(=O)O)c1C ZINC000147413310 DF For-Sale Anodyne PRTN3 61 40 Cc1cccc(S(=O)(=O)Nc2ccccc2C(=O)O)c1C ZINC000147413310 DF For-Sale Anodyne POLG_HCV1 15 43 Cc1cccc(S(=O)(=O)Nc2ccccc2C(=O)O)c1C ZINC000147413310 DF For-Sale Anodyne CCR8 55 34 Cc1cccc(S(=O)(=O)Nc2ccccc2C(=O)O)c1C ZINC000147413310 DF For-Sale Anodyne MCL1 15 43 Cc1cccc(S(=O)(=O)Nc2ccccc2C(=O)O)c1C ZINC000147413310 DF For-Sale Anodyne AKR1C3 24 62 Cc1cccc(S(=O)(=O)Nc2ccccc2C(=O)O)c1C ZINC000147413310 DF For-Sale Anodyne AKR1C2 45 62 CC[C@H]1CN([C@@H]2CCC[C@@H]2O)CC[C@@H]1N ZINC000147413325 BC For-Sale Anodyne SLC18A3 36 44 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)[C@@H]2CCCO2)cc1 ZINC000147413414 FD On-Demand Anodyne HDAC10 45 39 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)[C@@H]2CCCO2)cc1 ZINC000147413414 FD On-Demand Anodyne HDAC11 45 36 CCOC(=O)c1ccc(NC(=O)[C@@H]2CSCCC2=O)cc1 ZINC000147413432 DE For-Sale Anodyne ACR 57 35 CCOC(=O)c1ccc(NC(=O)[C@@H]2CSCCC2=O)cc1 ZINC000147413432 DE For-Sale Anodyne NOD2 16 40 Cc1cc(Br)cc(C)c1NC(=O)NCc1ccc(-n2ccnc2)c(F)c1 ZINC000147413445 HJ On-Demand Anodyne NOS2 72 32 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc3c(c2)OCO3)C1 ZINC000147413463 FD On-Demand Anodyne NOS2 42 32 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc3c(c2)OCO3)C1 ZINC000147413463 FD On-Demand Anodyne DYRK2 43 34 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc3c(c2)OCO3)C1 ZINC000147413463 FD On-Demand Anodyne TRPC6 25 40 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc3c(c2)OCO3)C1 ZINC000147413463 FD On-Demand Anodyne TRPC3 29 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)[C@@H]2CCCO2)cc1 ZINC000147413548 FD On-Demand Anodyne HDAC10 45 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)[C@@H]2CCCO2)cc1 ZINC000147413548 FD On-Demand Anodyne HDAC11 45 36 CCOC(=O)c1ccc(NC(=O)[C@H]2CSCCC2=O)cc1 ZINC000147413587 DE For-Sale Anodyne ACR 57 35 CCOC(=O)c1ccc(NC(=O)[C@H]2CSCCC2=O)cc1 ZINC000147413587 DE For-Sale Anodyne NOD2 16 40 COc1ccc(-c2noc(-c3sccc3Cl)n2)cn1 ZINC000147413637 CH On-Demand Anodyne CASP3 17 71 CCOc1ccc([C@H]2CCCN2C(=O)c2cnc(CC)s2)cc1 ZINC000147413647 EI On-Demand Anodyne CPT1A 82 39 CC(C)CCO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413671 GF On-Demand Anodyne CHRM5 24 43 CC(C)CCO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413671 GF On-Demand Anodyne EPHX2 18 42 CC(C)CCO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413671 GF On-Demand Anodyne TGM2 62 43 CC(C)CCO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413671 GF On-Demand Anodyne F13A1 64 43 CC(C)CCCCNS(=O)(=O)c1ccc(CCN)cc1 ZINC000147413712 CE For-Sale Anodyne CA2 25 49 CC(C)CCCCNS(=O)(=O)c1ccc(CCN)cc1 ZINC000147413712 CE For-Sale Anodyne TBXAS1 39 42 CC(C)CCCCNS(=O)(=O)c1ccc(CCN)cc1 ZINC000147413712 CE For-Sale Anodyne CA1 25 49 CC(C)CCCCNS(=O)(=O)c1ccc(CCN)cc1 ZINC000147413712 CE For-Sale Anodyne ALOX15 49 41 CC(C)CCCCNS(=O)(=O)c1ccc(CCN)cc1 ZINC000147413712 CE For-Sale Anodyne CA12 17 49 CC(C)CCCCNS(=O)(=O)c1ccc(CCN)cc1 ZINC000147413712 CE For-Sale Anodyne CA9 22 49 CC(C)CCCCNS(=O)(=O)c1ccc(CCN)cc1 ZINC000147413712 CE For-Sale Anodyne CAH_METTE 15 45 CC(C)CCCCNS(=O)(=O)c1ccc(CCN)cc1 ZINC000147413712 CE For-Sale Anodyne CA15 15 49 CC(C)CCCCNS(=O)(=O)c1ccc(CCN)cc1 ZINC000147413712 CE For-Sale Anodyne CA 0 49 CC(C)CCCCNS(=O)(=O)c1ccc(CCN)cc1 ZINC000147413712 CE For-Sale Anodyne A6YCJ1_9METZ 25 49 CC(C)CCCCNS(=O)(=O)c1ccc(CCN)cc1 ZINC000147413712 CE For-Sale Anodyne Q5TU56_ANOGA 0 49 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)[C@H]2CCCO2)cc1 ZINC000147413727 FD On-Demand Anodyne HDAC10 45 39 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)[C@H]2CCCO2)cc1 ZINC000147413727 FD On-Demand Anodyne HDAC11 45 36 CCOc1ccc([C@@H]2CCCN2C(=O)c2cnc(CC)s2)cc1 ZINC000147413817 EI On-Demand Anodyne COLA 87 39 CCOc1ccc([C@@H]2CCCN2C(=O)c2cnc(CC)s2)cc1 ZINC000147413817 EI On-Demand Anodyne CPT1A 82 39 CC(C)CCO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413873 GF On-Demand Anodyne CHRM5 24 43 CC(C)CCO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413873 GF On-Demand Anodyne EPHX2 18 42 CC(C)CCO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413873 GF On-Demand Anodyne TGM2 62 43 CC(C)CCO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147413873 GF On-Demand Anodyne F13A1 64 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)[C@H]2CCCO2)cc1 ZINC000147413884 FD On-Demand Anodyne BDKRB2 29 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)[C@H]2CCCO2)cc1 ZINC000147413884 FD On-Demand Anodyne HDAC10 45 39 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(NC(=O)[C@H]2CCCO2)cc1 ZINC000147413884 FD On-Demand Anodyne HDAC11 45 36 COc1ccc2c(c1)[C@H](NCC(F)F)CC2 ZINC000147413928 BF For-Sale Anodyne NQO2 42 46 COc1ccc2c(c1)[C@H](NCC(F)F)CC2 ZINC000147413928 BF For-Sale Anodyne MTR1B_CHICK 0 47 COc1ccc2c(c1)[C@H](NCC(F)F)CC2 ZINC000147413928 BF For-Sale Anodyne MTNR1B 16 43 OC[C@H](O)COc1cccc(OC[C@H](O)CO)c1 ZINC000147413978 CB For-Sale Anodyne ADRB2 20 49 OC[C@H](O)COc1cccc(OC[C@H](O)CO)c1 ZINC000147413978 CB For-Sale Anodyne ADRB1 24 49 OC[C@H](O)COc1cccc(OC[C@H](O)CO)c1 ZINC000147413978 CB For-Sale Anodyne PDS 53 34 CCCCCCCCCCCC[C@@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414008 GK For-Sale Mild INHA 16 48 CCCCCCCCCCCC[C@@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414008 GK For-Sale Mild CACNA1C 29 40 CCCCCCCCCCCC[C@@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414008 GK For-Sale Mild TBXA2R 17 43 CCCCCCCCCCCC[C@@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414008 GK For-Sale Mild CACNA1D 40 40 CCCCCCCCCCCC[C@@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414008 GK For-Sale Mild PLA2G4B 49 37 CCCCCCCCCCCC[C@@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414008 GK For-Sale Mild SLC27A4 48 37 COc1ccc2c(c1)[C@@H](NCC(F)F)CC2 ZINC000147414059 BF For-Sale Anodyne NQO2 42 46 COc1ccc2c(c1)[C@@H](NCC(F)F)CC2 ZINC000147414059 BF For-Sale Anodyne MTR1B_CHICK 0 47 COc1ccc2c(c1)[C@@H](NCC(F)F)CC2 ZINC000147414059 BF For-Sale Anodyne MTNR1B 16 43 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H](C(=O)Nc3ccc(Cl)cn3)C2)cc1 ZINC000147414123 HE On-Demand Anodyne F10 36 43 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H](C(=O)Nc3ccc(Cl)cn3)C2)cc1 ZINC000147414123 HE On-Demand Anodyne CPT1A 86 43 OC[C@H](O)COc1cccc(OC[C@@H](O)CO)c1 ZINC000147414138 CB For-Sale Anodyne ADRB2 20 49 OC[C@H](O)COc1cccc(OC[C@@H](O)CO)c1 ZINC000147414138 CB For-Sale Anodyne ADRB1 24 49 OC[C@H](O)COc1cccc(OC[C@@H](O)CO)c1 ZINC000147414138 CB For-Sale Anodyne PDS 53 34 CCCCCCCCCCCC[C@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414148 GK For-Sale Mild INHA 16 48 CCCCCCCCCCCC[C@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414148 GK For-Sale Mild CACNA1C 29 40 CCCCCCCCCCCC[C@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414148 GK For-Sale Mild TBXA2R 17 43 CCCCCCCCCCCC[C@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414148 GK For-Sale Mild CACNA1D 40 40 CCCCCCCCCCCC[C@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414148 GK For-Sale Mild PLA2G4B 49 37 CCCCCCCCCCCC[C@H](Oc1ccc([N+](=O)[O-])cc1)C(=O)OCC ZINC000147414148 GK For-Sale Mild SLC27A4 48 37 COC(=O)c1ccc(N2CCC[C@H](C(=O)O)C2)nc1C ZINC000147414163 CD On-Demand Anodyne SLC6A1 123 37 COC(=O)c1ccc(N2CCC[C@H](C(=O)O)C2)nc1C ZINC000147414163 CD On-Demand Anodyne ALK 19 41 COC(=O)c1ccc(N2CCC[C@H](C(=O)O)C2)nc1C ZINC000147414163 CD On-Demand Anodyne GPBAR1 28 42 CCOC(=O)c1ccc(N[C@@H]2CCO[C@@H]2C)cc1 ZINC000147414254 BE For-Sale Anodyne ACR 44 36 OC[C@@H](O)COc1cccc(OC[C@H](O)CO)c1 ZINC000147414286 CB For-Sale Anodyne ADRB2 20 49 OC[C@@H](O)COc1cccc(OC[C@H](O)CO)c1 ZINC000147414286 CB For-Sale Anodyne ADRB1 24 49 OC[C@@H](O)COc1cccc(OC[C@H](O)CO)c1 ZINC000147414286 CB For-Sale Anodyne PDS 53 34 CNc1ccc(S(=O)(=O)NCCNC(N)=O)cc1[N+](=O)[O-] ZINC000147414300 DB For-Sale Bother BDKRB1 0 45 Cc1cc(C)n([C@@H](C)C(=O)N2CCC[C@H](C(=O)Nc3ccc(Cl)cn3)C2)n1 ZINC000147414347 GF On-Demand Anodyne F10 22 47 COC(=O)c1ccc(N2CCC[C@@H](C(=O)O)C2)nc1C ZINC000147414349 CD On-Demand Anodyne SLC6A1 123 37 COC(=O)c1ccc(N2CCC[C@@H](C(=O)O)C2)nc1C ZINC000147414349 CD On-Demand Anodyne ALK 19 41 COC(=O)c1ccc(N2CCC[C@@H](C(=O)O)C2)nc1C ZINC000147414349 CD On-Demand Anodyne GPBAR1 28 42 CCOc1c(Br)cc(Br)cc1CNCCCCC(C)C ZINC000147414385 HK For-Sale Anodyne METG 72 51 CC(C)C(=O)Oc1ccc([C@@H](O)CNC(C)(C)C)cc1OC(=O)C(C)C ZINC000147414410 FG Annotated Anodyne ADRB1 23 45 CCOC(=O)c1ccc(N[C@H]2CCO[C@@H]2C)cc1 ZINC000147414412 BE For-Sale Anodyne ACR 44 36 Sc1cn(Cc2ccccc2)nn1 ZINC000147414426 AD For-Sale Anodyne HSP90AB1 29 48 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147414427 HF On-Demand Bother EPHX2 32 41 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147414427 HF On-Demand Bother TGM2 63 42 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147414427 HF On-Demand Bother CACNA1I 75 42 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147414427 HF On-Demand Bother F13A1 59 42 Cc1cc(C(=O)NCCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147414465 CE On-Demand Bother ADRA2A 0 44 Cc1cc(C(=O)NCCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147414465 CE On-Demand Bother DRD4 43 34 Cc1cc(C(=O)NCCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147414465 CE On-Demand Bother ADRA1D 44 44 Cc1cc(C(=O)NCCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147414465 CE On-Demand Bother HTR1D 22 44 Cc1cc(C(=O)NCCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147414465 CE On-Demand Bother ADRA1A 44 43 Cc1cc(C(=O)NCCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147414465 CE On-Demand Bother ADRA1B 39 44 Cc1cc(C(=O)NCCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147414465 CE On-Demand Bother ADRA2B 22 44 Cc1cc(C(=O)NCCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147414465 CE On-Demand Bother ADRA2C 23 44 Cc1cc(C(=O)NCCCN2CCCC2)cc([N+](=O)[O-])c1 ZINC000147414465 CE On-Demand Bother HRP1_PLAFA 35 46 Cc1cc(C)n([C@H](C)C(=O)N2CCC[C@H](C(=O)Nc3ccc(Cl)cn3)C2)n1 ZINC000147414487 GF On-Demand Anodyne F10 22 47 Oc1ccccc1CNCC(F)F ZINC000147414497 AD On-Demand Clean PHES 91 36 O=c1[nH]c(-c2cccc(-c3cc4ccccc4o3)c2)ncc1O ZINC000147414503 DH For-Sale Anodyne DAO 21 43 O=c1[nH]c(-c2cccc(-c3cc4ccccc4o3)c2)ncc1O ZINC000147414503 DH For-Sale Anodyne TNKS 31 40 Cc1ccccc1C(=O)NNC(=O)Nc1nc(CN2CCCCC2)cs1 ZINC000147414545 FF On-Demand Reactive CCR8 45 33 COc1ccccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147414554 CD On-Demand Anodyne KCNA3 61 60 COc1ccccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147414554 CD On-Demand Anodyne HCN1 85 57 COc1ccccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147414554 CD On-Demand Anodyne HCN4 70 54 COc1ccccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147414554 CD On-Demand Anodyne KCNK3 67 51 COc1ccccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147414554 CD On-Demand Anodyne KCNK9 56 51 CNc1nc(C)cc(Oc2cccc3cccnc23)n1 ZINC000147414576 CG For-Sale Anodyne C0L093_TOBAC 57 35 CCOC(=O)c1ccc(N[C@@H]2CCO[C@H]2C)cc1 ZINC000147414584 BE For-Sale Anodyne ACR 44 36 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H]1CCCBr ZINC000147414616 FI For-Sale Reactive HCRTR1 20 46 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H]1CCCBr ZINC000147414616 FI For-Sale Reactive RBP4 59 39 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H]1CCCBr ZINC000147414616 FI For-Sale Reactive SFRP1 52 32 O=C(c1ccccc1C(F)(F)F)N1CCC[C@@H]1CCCBr ZINC000147414616 FI For-Sale Reactive WNT3 43 31 Cc1cc(C)n([C@@H](C)C(=O)N2CCC[C@@H](C(=O)Nc3ccc(Cl)cn3)C2)n1 ZINC000147414621 GF On-Demand Anodyne F10 22 47 CC[C@H](NC(=O)N1[C@H](C)CCC[C@H]1C)C(=O)O ZINC000147414633 BD On-Demand Anodyne EDNRB 41 44 CC[C@H](NC(=O)N1[C@H](C)CCC[C@H]1C)C(=O)O ZINC000147414633 BD On-Demand Anodyne EDNRA 41 45 CCOC(=O)c1ccc(N[C@H]2CCO[C@H]2C)cc1 ZINC000147414720 BE For-Sale Anodyne ACR 44 36 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H]1CCCBr ZINC000147414735 FI For-Sale Reactive HCRTR1 20 46 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H]1CCCBr ZINC000147414735 FI For-Sale Reactive RBP4 59 39 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H]1CCCBr ZINC000147414735 FI For-Sale Reactive SFRP1 52 32 O=C(c1ccccc1C(F)(F)F)N1CCC[C@H]1CCCBr ZINC000147414735 FI For-Sale Reactive WNT3 43 31 Cc1cc(C)n([C@H](C)C(=O)N2CCC[C@@H](C(=O)Nc3ccc(Cl)cn3)C2)n1 ZINC000147414736 GF On-Demand Anodyne F10 22 47 CCCCCCCCNS(=O)(=O)N(C)CCCNCCC ZINC000147414748 DF For-Sale Mild S1PR3 15 41 CCCCCCCCNS(=O)(=O)N(C)CCCNCCC ZINC000147414748 DF For-Sale Mild S1PR2 30 41 CCCCCCCCNS(=O)(=O)N(C)CCCNCCC ZINC000147414748 DF For-Sale Mild RELA 19 44 CCCCCCCCOc1ccc(Br)cc1C(F)(F)F ZINC000147414809 FK Annotated Mild S1PR4 20 43 CCCCCCCCOc1ccc(Br)cc1C(F)(F)F ZINC000147414809 FK Annotated Mild PLA2G4B 78 38 Nc1cc(Oc2cccc3cccnc23)cc([N+](=O)[O-])c1 ZINC000147414817 CH For-Sale Bother NFKBIA 0 41 O=C(O)c1cc(-c2ccc(F)cc2Cl)ccc1O ZINC000147414934 CH For-Sale Anodyne DHODH 40 37 O=C(O)c1cc(-c2ccc(F)cc2Cl)ccc1O ZINC000147414934 CH For-Sale Anodyne PYGL 22 43 O=C(O)c1cc(-c2ccc(F)cc2Cl)ccc1O ZINC000147414934 CH For-Sale Anodyne NR0B2 0 40 O=C(O)c1cc(-c2ccc(F)cc2Cl)ccc1O ZINC000147414934 CH For-Sale Anodyne SLC22A6 15 73 O=C(O)c1cc(-c2ccc(F)cc2Cl)ccc1O ZINC000147414934 CH For-Sale Anodyne AKR1C2 69 41 O=C(O)c1cc(-c2ccc(F)cc2Cl)ccc1O ZINC000147414934 CH For-Sale Anodyne AKR1C1 67 41 O=C(O)c1cc(-c2ccc(F)cc2Cl)ccc1O ZINC000147414934 CH For-Sale Anodyne MGRA 0 40 O=C(C(=O)N1CCC[C@H](C(=O)Nc2ccc(Cl)cn2)C1)c1ccc2c(c1)CCC2 ZINC000147414965 HG On-Demand Anodyne F10 35 44 CCOC(=O)C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147414967 EG For-Sale Anodyne FKBP1A 29 40 CCOC(=O)C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147414967 EG For-Sale Anodyne GHRHR 61 40 CCOC(=O)C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147414967 EG For-Sale Anodyne GRIN2B 19 44 CCOC(=O)C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147414967 EG For-Sale Anodyne ELANE 15 41 CCOC(=O)C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147414967 EG For-Sale Anodyne TIMP3 40 33 CCOC(=O)C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147414967 EG For-Sale Anodyne F13A1 40 38 CCOC(=O)C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147414967 EG For-Sale Anodyne CCR8 33 41 CCOC(=O)C1CC2(CCN(C(=O)OCc3ccccc3)CC2)C1 ZINC000147414967 EG For-Sale Anodyne SLC12A5 79 42 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@@H]1CCCBr ZINC000147414973 FI For-Sale Reactive PREP 28 40 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@@H]1CCCBr ZINC000147414973 FI For-Sale Reactive FAP 0 42 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@@H]1CCCBr ZINC000147414973 FI For-Sale Reactive L3MBTL3 40 34 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne F2 34 42 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne TACR1 15 40 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne CTSB 31 40 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne TRY2_BOVIN 86 39 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne CTSK 18 40 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne CTSL 27 40 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne CACNA1B 27 42 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne CCR3 61 39 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne CTSS 20 40 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne CAPN1 45 40 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne EPHX2 26 41 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne ACE2 41 34 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne TGM2 56 44 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne BACE1 23 42 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne ST14 101 42 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne F13A1 51 44 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne BRCA1 42 29 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne NAMPT 27 48 C[C@@H](Cc1cccc(F)c1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415040 HG On-Demand Anodyne TMPRSS6 61 34 Nc1nccc(Oc2cccc3cccnc23)n1 ZINC000147415043 BE For-Sale Anodyne CCR1 0 41 Nc1nccc(Oc2cccc3cccnc23)n1 ZINC000147415043 BE For-Sale Anodyne METAP2 0 41 O=c1[nH]c2ccc(S(=O)(=O)Nc3ccc(OCC(F)(F)F)cc3)cc2[nH]1 ZINC000147415068 GF On-Demand Anodyne MGAT1 47 35 CCOc1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1S(=O)(=O)N(C)C ZINC000147415093 HF On-Demand Bother KCNK3 36 40 CCOc1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1S(=O)(=O)N(C)C ZINC000147415093 HF On-Demand Bother KCNK9 36 40 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@H]1CCCBr ZINC000147415122 FI For-Sale Reactive PREP 28 40 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@H]1CCCBr ZINC000147415122 FI For-Sale Reactive FAP 0 42 O=C(c1ccc(C(F)(F)F)cc1)N1CCC[C@H]1CCCBr ZINC000147415122 FI For-Sale Reactive L3MBTL3 40 34 O=C(C(=O)N1CCC[C@@H](C(=O)Nc2ccc(Cl)cn2)C1)c1ccc2c(c1)CCC2 ZINC000147415132 HG On-Demand Anodyne F10 35 44 O=C(NCC1(C(=O)O)CCC1)c1ccc(F)cc1Cl ZINC000147415179 CE On-Demand Anodyne P2RX7 53 45 O=C(NCC1(C(=O)O)CCC1)c1ccc(F)cc1Cl ZINC000147415179 CE On-Demand Anodyne PYGL 24 48 O=C(NCC1(C(=O)O)CCC1)c1ccc(F)cc1Cl ZINC000147415179 CE On-Demand Anodyne SLC6A9 57 48 CCCCCCCCNS(=O)(=O)CCCCNC1CC1 ZINC000147415196 DF For-Sale Mild RELA 24 55 CCCCCCCCNS(=O)(=O)CCCCNCCC ZINC000147415308 DG For-Sale Mild ADH1A 0 41 CCCCCCCCNS(=O)(=O)CCCCNCCC ZINC000147415308 DG For-Sale Mild ADH7 0 41 CCCCCCCCNS(=O)(=O)CCCCNCCC ZINC000147415308 DG For-Sale Mild S1PR3 17 46 CCCCCCCCNS(=O)(=O)CCCCNCCC ZINC000147415308 DG For-Sale Mild S1PR2 36 46 CCCCCCCCNS(=O)(=O)CCCCNCCC ZINC000147415308 DG For-Sale Mild ADH1B 0 41 CCCCCCCCNS(=O)(=O)CCCCNCCC ZINC000147415308 DG For-Sale Mild RELA 34 76 Clc1ccsc1-c1nc(-c2ccccc2)n[nH]1 ZINC000147415330 CH For-Sale Anodyne XDH 25 43 NS(=O)(=O)c1cc(F)cc(F)c1OCCCN1CCCC1 ZINC000147415417 DD For-Sale Anodyne HRH3 52 51 NS(=O)(=O)c1cc(F)cc(F)c1OCCCN1CCCC1 ZINC000147415417 DD For-Sale Anodyne HNMT 55 33 O=C(NCC1(C(=O)O)CCC1)c1c(F)cccc1Cl ZINC000147415448 CE On-Demand Anodyne TYK2 20 47 Cc1cc(C)n([C@@H](C)C(=O)N2CCC(C(=O)Nc3ccc(Cl)cn3)CC2)n1 ZINC000147415475 GF On-Demand Anodyne F10 40 52 Cc1cc(C)n([C@@H](C)C(=O)N2CCC(C(=O)Nc3ccc(Cl)cn3)CC2)n1 ZINC000147415475 GF On-Demand Anodyne CCR1 40 37 CC[C@@H]1CN([C@@H]2CCCC[C@@H]2O)CC[C@@H]1N ZINC000147415485 BD For-Sale Anodyne VACHT_TETCF 0 40 CC[C@@H]1CN([C@@H]2CCCC[C@@H]2O)CC[C@@H]1N ZINC000147415485 BD For-Sale Anodyne SLC18A3 30 46 O=C(NCC1(C(=O)O)CCC1)c1cc(Br)ccc1Cl ZINC000147415651 EG On-Demand Anodyne P2RX7 24 42 Cc1cc(C)n([C@H](C)C(=O)N2CCC(C(=O)Nc3ccc(Cl)cn3)CC2)n1 ZINC000147415652 GF On-Demand Anodyne F10 40 52 Cc1cc(C)n([C@H](C)C(=O)N2CCC(C(=O)Nc3ccc(Cl)cn3)CC2)n1 ZINC000147415652 GF On-Demand Anodyne CCR1 40 37 O=C(O)c1cc(Cl)cc(NC(=O)N2CCC[C@@H]2CO)c1 ZINC000147415671 CE On-Demand Anodyne CACNA1I 46 36 CC[C@H]1CN([C@@H]2CCCC[C@@H]2O)CC[C@@H]1N ZINC000147415686 BD For-Sale Anodyne VACHT_TETCF 0 40 CC[C@H]1CN([C@@H]2CCCC[C@@H]2O)CC[C@@H]1N ZINC000147415686 BD For-Sale Anodyne SLC18A3 30 46 Cc1cc(C(=O)Nc2nc(-c3ccc[nH]3)cs2)cc([N+](=O)[O-])c1 ZINC000147415704 EH On-Demand Bother MPL 53 40 CC(C)C[C@@H](C)CCC(=O)O ZINC000147415805 AF For-Sale Anodyne FOLH1 27 50 CC(C)C[C@@H](C)CCC(=O)O ZINC000147415805 AF For-Sale Anodyne Q6UB75_PIG 0 43 CC(C)CCCCN[C@@H](C)c1cccc(S(N)(=O)=O)c1 ZINC000147415833 CF For-Sale Anodyne CA2 26 42 CC(C)CCCCN[C@@H](C)c1cccc(S(N)(=O)=O)c1 ZINC000147415833 CF For-Sale Anodyne CA1 16 41 CCCCCCCCCCCCc1ccc2c(c1)c1ccccc1c(=O)n2CCCC ZINC000147415863 HK Annotated Mild CNR1 27 48 CCCCCCCCCCCCc1ccc2c(c1)c1ccccc1c(=O)n2CCCC ZINC000147415863 HK Annotated Mild INHA 88 39 CCCCCCCCCCCCc1ccc2c(c1)c1ccccc1c(=O)n2CCCC ZINC000147415863 HK Annotated Mild CNR2 27 46 CCCCCCCCCCCCc1ccc2c(c1)c1ccccc1c(=O)n2CCCC ZINC000147415863 HK Annotated Mild RORC 0 59 CCCCCCCCCCCCc1ccc2c(c1)c1ccccc1c(=O)n2CCCC ZINC000147415863 HK Annotated Mild RORB 0 80 O=C(C(=O)N1CCC(C(=O)Nc2ccc(Cl)cn2)CC1)c1ccc2c(c1)CCC2 ZINC000147415891 HG On-Demand Anodyne F10 40 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(-c3cnco3)c2)c1 ZINC000147415894 EH On-Demand Bother TAAR1 34 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(-c3cnco3)c2)c1 ZINC000147415894 EH On-Demand Bother AKR1C3 15 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(-c3cnco3)c2)c1 ZINC000147415894 EH On-Demand Bother AKR1C2 26 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(-c3cnco3)c2)c1 ZINC000147415894 EH On-Demand Bother KCNK3 38 40 O=C(O)c1cc(Cl)cc(NC(=O)N2CCC[C@H]2CO)c1 ZINC000147415905 CE On-Demand Anodyne CACNA1I 46 36 O=S(=O)(c1ccc(F)cc1)N1CCO[C@H](c2ccc(Br)cc2)C1 ZINC000147415909 HG On-Demand Anodyne PKM 19 42 CCOCCOCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415929 GD On-Demand Anodyne EPHX2 28 46 CCOCCOCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415929 GD On-Demand Anodyne TGM2 68 44 CCOCCOCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415929 GD On-Demand Anodyne CACNA1I 41 34 CCOCCOCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147415929 GD On-Demand Anodyne F13A1 70 44 CCNc1nc(Cl)nc(Oc2cccc3cccnc23)n1 ZINC000147415938 DG For-Sale Anodyne PPX1 0 43 COc1cccc(CNCC(F)F)c1OC ZINC000147416033 BE On-Demand Anodyne PHES 0 45 COc1cccc(CNCC(F)F)c1OC ZINC000147416033 BE On-Demand Anodyne KCNJ2 0 40 CC[C@@H]1CCCN(C(=O)c2cccn(Cc3ccccc3)c2=O)C1 ZINC000147416045 DG On-Demand Anodyne SLC6A1 41 32 CC(C)CCCCN[C@H](C)c1cccc(S(N)(=O)=O)c1 ZINC000147416056 CF For-Sale Anodyne CA2 26 42 CC(C)CCCCN[C@H](C)c1cccc(S(N)(=O)=O)c1 ZINC000147416056 CF For-Sale Anodyne CA1 16 41 CCCCCCCCn1cncc1CNCCOC ZINC000147416069 CF For-Sale Mild LPAR2 40 31 CCCCCCCCn1cncc1CNCCOC ZINC000147416069 CF For-Sale Mild S1PR2 42 32 O=C(NCC1(C(=O)O)CCC1)c1c(Cl)cccc1Cl ZINC000147416091 DF On-Demand Anodyne SLC6A9 19 40 C[C@H](NC(=O)CCn1ccc2ccccc21)c1cccc(C(F)(F)F)c1 ZINC000147416122 FJ On-Demand Anodyne PSMB1 15 41 C[C@H](NC(=O)CCn1ccc2ccccc21)c1cccc(C(F)(F)F)c1 ZINC000147416122 FJ On-Demand Anodyne RORC 20 41 C[C@H](NC(=O)CCn1ccc2ccccc21)c1cccc(C(F)(F)F)c1 ZINC000147416122 FJ On-Demand Anodyne SUCNR1 19 42 CN(C)c1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147416126 EH For-Sale Reactive HCRTR1 0 43 CN(C)c1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147416126 EH For-Sale Reactive PREP 36 41 C[C@@H](CCc1ccc(O)cc1)NC(=O)N(C)Cc1cscn1 ZINC000147416130 DG On-Demand Anodyne BMP1 55 35 C[C@@H](CCc1ccc(O)cc1)NC(=O)N(C)Cc1cscn1 ZINC000147416130 DG On-Demand Anodyne CYP3A4 20 47 COC(=O)c1ccc(Nc2ccc(C(=O)O)cc2)nc1C ZINC000147416151 CF For-Sale Anodyne PDE4D 0 45 COC(=O)c1ccc(Nc2ccc(C(=O)O)cc2)nc1C ZINC000147416151 CF For-Sale Anodyne AKR1C3 42 47 COC(=O)c1ccc(Nc2ccc(C(=O)O)cc2)nc1C ZINC000147416151 CF For-Sale Anodyne AKR1C2 62 47 CC(C)CCSCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147416153 GF On-Demand Anodyne CHRM5 15 42 CC(C)CCSCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147416153 GF On-Demand Anodyne EPHX2 16 42 CC(C)CCSCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147416153 GF On-Demand Anodyne TGM2 65 43 CC(C)CCSCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147416153 GF On-Demand Anodyne F13A1 68 43 COc1cc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)c(OC)cc1Cl ZINC000147416156 HF On-Demand Anodyne HTR4 35 46 CC[C@H]1CCCN(C(=O)c2cccn(Cc3ccccc3)c2=O)C1 ZINC000147416219 DG On-Demand Anodyne SLC6A1 41 32 CNc1ccc([N+](=O)[O-])cc1S(=O)(=O)NCCNC(N)=O ZINC000147416235 DB For-Sale Bother TBXA2R 33 45 COC(=O)[C@@](C)(N)CCOCc1ccccc1 ZINC000147416259 BD For-Sale Anodyne AMY2 56 34 COC(=O)[C@@](C)(N)CCOCc1ccccc1 ZINC000147416259 BD For-Sale Anodyne PTPRB 31 43 COC(=O)[C@@](C)(N)CCOCc1ccccc1 ZINC000147416259 BD For-Sale Anodyne GHSR 30 40 CCOc1ccccc1CNCC(F)F ZINC000147416262 BE On-Demand Anodyne PHES 0 41 C[C@H](CCc1ccc(O)cc1)NC(=O)N(C)Cc1cscn1 ZINC000147416314 DG On-Demand Anodyne BMP1 55 35 C[C@H](CCc1ccc(O)cc1)NC(=O)N(C)Cc1cscn1 ZINC000147416314 DG On-Demand Anodyne CYP3A4 20 47 Cc1ccccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147416338 BD On-Demand Anodyne KCNA3 41 41 Cc1ccccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147416338 BD On-Demand Anodyne ACAT 0 41 Cc1ccccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147416338 BD On-Demand Anodyne HCN1 68 38 Cc1ccccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147416338 BD On-Demand Anodyne HCN4 56 36 Cc1ccccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147416338 BD On-Demand Anodyne KCNK3 26 46 Cc1ccccc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147416338 BD On-Demand Anodyne KCNK9 22 40 CN(C)c1cccc(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147416360 EH For-Sale Reactive HCRTR1 0 43 CN(C)c1cccc(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147416360 EH For-Sale Reactive PREP 36 41 C[C@@H](NC(=O)CCn1ccc2ccccc21)c1cccc(C(F)(F)F)c1 ZINC000147416372 FJ On-Demand Anodyne PSMB1 15 41 C[C@@H](NC(=O)CCn1ccc2ccccc21)c1cccc(C(F)(F)F)c1 ZINC000147416372 FJ On-Demand Anodyne RORC 20 41 C[C@@H](NC(=O)CCn1ccc2ccccc21)c1cccc(C(F)(F)F)c1 ZINC000147416372 FJ On-Demand Anodyne SUCNR1 19 42 COc1cc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)c(OC)cc1Cl ZINC000147416377 HF On-Demand Anodyne HTR4 35 46 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne HTR1A 87 53 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne DRD2 70 53 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne DRD4 54 44 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne ADRA1D 33 42 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne HTR2A 62 43 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne HTR2C 42 43 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne SLC6A4 21 41 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne ADRA1A 32 42 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne HRH1 15 44 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne DRD3 78 49 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne HTR4 24 41 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne HTR7 90 44 CCCOCC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416379 DD On-Demand Anodyne SIGMAR1 15 52 COC(=O)c1ccc(Nc2cccc(C(=O)O)c2)nc1C ZINC000147416394 CF For-Sale Anodyne AKR1C3 65 54 COC(=O)c1ccc(Nc2cccc(C(=O)O)c2)nc1C ZINC000147416394 CF For-Sale Anodyne AKR1C2 67 41 COC(=O)c1ccc(Nc2cccc(C(=O)O)c2)nc1C ZINC000147416394 CF For-Sale Anodyne KCNK3 72 35 COC(=O)c1ccc(Nc2cccc(C(=O)O)c2)nc1C ZINC000147416394 CF For-Sale Anodyne KCNK9 43 33 C[C@@H](Cn1ccnc1)NC(=O)c1csc(-c2ccccc2F)n1 ZINC000147416397 EF On-Demand Anodyne TBXAS1 27 41 N#CC1(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCCCC1 ZINC000147416398 GF On-Demand Mild CTSB 15 42 N#CC1(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCCCC1 ZINC000147416398 GF On-Demand Mild CTSK 18 45 N#CC1(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCCCC1 ZINC000147416398 GF On-Demand Mild EPHX2 19 47 N#CC1(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCCCC1 ZINC000147416398 GF On-Demand Mild TGM2 58 45 N#CC1(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCCCC1 ZINC000147416398 GF On-Demand Mild F13A1 57 45 N#CC1(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCCCC1 ZINC000147416398 GF On-Demand Mild NAMPT 38 44 COc1ccc(S(=O)(=O)N2CCO[C@H](c3ccc(Br)cc3)C2)cc1 ZINC000147416412 HG On-Demand Anodyne MMP13 42 47 COc1ccc(S(=O)(=O)N2CCO[C@H](c3ccc(Br)cc3)C2)cc1 ZINC000147416412 HG On-Demand Anodyne MMP2 18 41 COc1ccc(S(=O)(=O)N2CCO[C@H](c3ccc(Br)cc3)C2)cc1 ZINC000147416412 HG On-Demand Anodyne MMP3 47 47 COc1ccc(S(=O)(=O)N2CCO[C@H](c3ccc(Br)cc3)C2)cc1 ZINC000147416412 HG On-Demand Anodyne MMP8 23 41 COc1ccc(S(=O)(=O)N2CCO[C@H](c3ccc(Br)cc3)C2)cc1 ZINC000147416412 HG On-Demand Anodyne MMP9 33 47 COc1ccc(S(=O)(=O)N2CCO[C@H](c3ccc(Br)cc3)C2)cc1 ZINC000147416412 HG On-Demand Anodyne PKM 15 51 COc1ccc(S(=O)(=O)N2CCO[C@H](c3ccc(Br)cc3)C2)cc1 ZINC000147416412 HG On-Demand Anodyne MMP7 47 41 COc1ccc(S(=O)(=O)N2CCO[C@H](c3ccc(Br)cc3)C2)cc1 ZINC000147416412 HG On-Demand Anodyne MMP1 46 47 COC(=O)[C@](C)(N)CCOCc1ccccc1 ZINC000147416477 BD For-Sale Anodyne AMY2 56 34 COC(=O)[C@](C)(N)CCOCc1ccccc1 ZINC000147416477 BD For-Sale Anodyne PTPRB 31 43 COC(=O)[C@](C)(N)CCOCc1ccccc1 ZINC000147416477 BD For-Sale Anodyne GHSR 30 40 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H]1CCCBr ZINC000147416578 FH For-Sale Reactive COLA 128 44 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H]1CCCBr ZINC000147416578 FH For-Sale Reactive CPT1A 109 43 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H]1CCCBr ZINC000147416578 FH For-Sale Reactive CPT2 48 42 O=C(COc1ccc(Cl)cc1)N1CCC[C@@H]1CCCBr ZINC000147416578 FH For-Sale Reactive CHRNA10 23 44 C[C@@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416593 ED On-Demand Anodyne CYP19A1 21 44 C[C@@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416593 ED On-Demand Anodyne DRTS_PLAFK 19 42 C[C@@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416593 ED On-Demand Anodyne CYP11B1 34 44 C[C@@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416593 ED On-Demand Anodyne TBXAS1 62 44 C[C@@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416593 ED On-Demand Anodyne AGTR2 36 43 C[C@@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416593 ED On-Demand Anodyne CYP11B2 41 44 C[C@@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416593 ED On-Demand Anodyne POLR1A 47 40 Cc1nn(C(F)F)c(C)c1CC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416660 GE On-Demand Anodyne HTR1A 79 51 Cc1nn(C(F)F)c(C)c1CC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416660 GE On-Demand Anodyne DRD2 65 51 Cc1nn(C(F)F)c(C)c1CC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416660 GE On-Demand Anodyne DRD4 50 41 Cc1nn(C(F)F)c(C)c1CC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416660 GE On-Demand Anodyne HTR2A 60 44 Cc1nn(C(F)F)c(C)c1CC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416660 GE On-Demand Anodyne HTR2C 51 42 Cc1nn(C(F)F)c(C)c1CC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416660 GE On-Demand Anodyne SLC6A4 23 44 Cc1nn(C(F)F)c(C)c1CC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416660 GE On-Demand Anodyne ADRA1A 33 45 Cc1nn(C(F)F)c(C)c1CC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416660 GE On-Demand Anodyne ADRA1B 18 45 Cc1nn(C(F)F)c(C)c1CC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416660 GE On-Demand Anodyne DRD3 92 46 Cc1nn(C(F)F)c(C)c1CC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416660 GE On-Demand Anodyne HTR7 77 44 Cc1nn(C(F)F)c(C)c1CC(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147416660 GE On-Demand Anodyne P2RX7 44 45 O=S(=O)(c1cccc(F)c1)N1CCO[C@H](c2ccc(Br)cc2)C1 ZINC000147416700 HG On-Demand Anodyne PKM 37 48 O=C(COc1ccc(Cl)cc1)N1CCC[C@H]1CCCBr ZINC000147416805 FH For-Sale Reactive COLA 128 44 O=C(COc1ccc(Cl)cc1)N1CCC[C@H]1CCCBr ZINC000147416805 FH For-Sale Reactive CPT1A 109 43 O=C(COc1ccc(Cl)cc1)N1CCC[C@H]1CCCBr ZINC000147416805 FH For-Sale Reactive CPT2 48 42 O=C(COc1ccc(Cl)cc1)N1CCC[C@H]1CCCBr ZINC000147416805 FH For-Sale Reactive CHRNA10 23 44 C[C@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416843 ED On-Demand Anodyne CYP19A1 21 44 C[C@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416843 ED On-Demand Anodyne DRTS_PLAFK 19 42 C[C@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416843 ED On-Demand Anodyne CYP11B1 34 44 C[C@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416843 ED On-Demand Anodyne TBXAS1 62 44 C[C@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416843 ED On-Demand Anodyne AGTR2 36 43 C[C@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416843 ED On-Demand Anodyne CYP11B2 41 44 C[C@H](Cn1ccnc1)NC(=O)c1cccn(Cc2ccccc2)c1=O ZINC000147416843 ED On-Demand Anodyne POLR1A 47 40 CCC1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147416850 DH On-Demand Anodyne CACNA1H 46 36 CCC1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147416850 DH On-Demand Anodyne EPHX2 28 46 CCC1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147416850 DH On-Demand Anodyne CACNA1I 73 41 CCCC[C@H](Nc1ccc(C(=O)OC)c(C)n1)C(=O)O ZINC000147416915 CE On-Demand Anodyne NOD1 41 33 CC(=O)c1ccc(NCC(=O)O)nc1 ZINC000147416980 AC On-Demand Anodyne P4HTM 40 35 CC(C)CCCCNCc1cccc(Cl)c1 ZINC000147416989 BI For-Sale Anodyne FDFT1 0 48 CC(C)CCCCNCc1cccc(Cl)c1 ZINC000147416989 BI For-Sale Anodyne LEF 77 39 CC(C)CCCCNCc1cccc(Cl)c1 ZINC000147416989 BI For-Sale Anodyne NAMPT 0 41 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H]1CCOc3ccc(Br)cc31)C2 ZINC000147416990 HH On-Demand Anodyne MTNR1A 15 41 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H]1CCOc3ccc(Br)cc31)C2 ZINC000147416990 HH On-Demand Anodyne ROCK2 22 41 Cc1cccc(C2(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)CC2)c1 ZINC000147417028 HG On-Demand Anodyne EPHX2 32 40 Cc1cccc(C2(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)CC2)c1 ZINC000147417028 HG On-Demand Anodyne TGM2 53 41 Cc1cccc(C2(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)CC2)c1 ZINC000147417028 HG On-Demand Anodyne F13A1 43 41 C[C@H]1CCC[C@@H](C)N1NC(=O)c1ccc2c(c1)CNCC2 ZINC000147417045 CE For-Sale Anodyne PNMT 19 41 COC(=O)[C@](C)(CC=O)NC(=O)OC(C)(C)C ZINC000147417081 BD For-Sale Mild CTSK 17 41 CCCC[C@@H](Nc1ccc(C(=O)OC)c(C)n1)C(=O)O ZINC000147417109 CE On-Demand Anodyne NOD1 41 33 CCCCCCCOc1ccc(CNCCC)nc1 ZINC000147417120 CH For-Sale Mild LPAR2 63 49 CCCCCCCOc1ccc(CNCCC)nc1 ZINC000147417120 CH For-Sale Mild S1PR3 28 49 CCCCCCCOc1ccc(CNCCC)nc1 ZINC000147417120 CH For-Sale Mild SLC2A1 0 43 CCCCCCCOc1ccc(CNCCC)nc1 ZINC000147417120 CH For-Sale Mild PLA2G4B 85 37 CCCCCCCOc1ccc(CNCCC)nc1 ZINC000147417120 CH For-Sale Mild S1PR2 68 49 CCCCCCCOc1ccc(CNCCC)nc1 ZINC000147417120 CH For-Sale Mild LMGT2 0 43 O=S(=O)(c1c(F)cccc1F)N1CCO[C@H](c2ccc(Br)cc2)C1 ZINC000147417204 HG On-Demand Anodyne PKM 29 49 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H]1CCOc3ccc(Br)cc31)C2 ZINC000147417214 HH On-Demand Anodyne MTNR1A 15 41 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H]1CCOc3ccc(Br)cc31)C2 ZINC000147417214 HH On-Demand Anodyne ROCK2 22 41 Cc1ccc(CNCC(F)F)c(C)c1 ZINC000147417216 AF On-Demand Anodyne CCR2 29 41 CCCOC(=O)c1ccc(N[C@@H]2CCO[C@@H]2C)cc1 ZINC000147417220 CF For-Sale Anodyne CNGA1 0 40 Nc1ccc([N+](=O)[O-])c(Oc2cccc3cccnc23)n1 ZINC000147417246 CF For-Sale Bother MCHR1 22 40 O=C(NCC1(C(=O)O)CCC1)c1ccccc1F ZINC000147417255 CD On-Demand Anodyne KCNA3 45 38 O=C(NCC1(C(=O)O)CCC1)c1ccccc1F ZINC000147417255 CD On-Demand Anodyne SLC6A9 24 42 O=C(NCC1(C(=O)O)CCC1)c1ccccc1F ZINC000147417255 CD On-Demand Anodyne HCN1 75 36 O=C(NCC1(C(=O)O)CCC1)c1ccccc1F ZINC000147417255 CD On-Demand Anodyne HCN4 53 34 CN(CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147417260 HE On-Demand Anodyne CHRM5 16 40 CN(CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147417260 HE On-Demand Anodyne EPHX2 20 44 CN(CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147417260 HE On-Demand Anodyne TGM2 70 45 CN(CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147417260 HE On-Demand Anodyne F13A1 64 45 C[C@H]1CCC[C@H](C)N1NC(=O)c1ccc2c(c1)CNCC2 ZINC000147417267 CE For-Sale Anodyne PNMT 19 41 O=C(CCN1C(=O)CCC1=O)N1CCN(S(=O)(=O)c2ccc3c(c2)OCCO3)CC1 ZINC000147417275 IB On-Demand Anodyne PKM 53 60 CCCNc1ccc(S(=O)(=O)NCCNC(N)=O)cc1 ZINC000147417290 DC For-Sale Anodyne CA2 34 44 CCCNc1ccc(S(=O)(=O)NCCNC(N)=O)cc1 ZINC000147417290 DC For-Sale Anodyne CA1 32 44 CCCNc1ccc(S(=O)(=O)NCCNC(N)=O)cc1 ZINC000147417290 DC For-Sale Anodyne CA4 29 44 CCCNc1ccc(S(=O)(=O)NCCNC(N)=O)cc1 ZINC000147417290 DC For-Sale Anodyne CA9 28 41 CCCNc1ccc(S(=O)(=O)NCCNC(N)=O)cc1 ZINC000147417290 DC For-Sale Anodyne CYNT 40 36 Cn1ncc2c1CCC[C@@H]2NC(=O)c1cccnc1Oc1ccc(Cl)cc1Cl ZINC000147417303 HJ On-Demand Anodyne UGCG 37 44 Cn1ncc2c1CCC[C@@H]2NC(=O)c1cccnc1Oc1ccc(Cl)cc1Cl ZINC000147417303 HJ On-Demand Anodyne GPBAR1 23 41 COc1ccc2c(c1)OC[C@H](C(=O)N[C@H]1CCOc3ccc(Br)cc31)C2 ZINC000147417436 HH On-Demand Anodyne MTNR1A 15 41 COc1ccc2c(c1)OC[C@H](C(=O)N[C@H]1CCOc3ccc(Br)cc31)C2 ZINC000147417436 HH On-Demand Anodyne ROCK2 22 41 CCCOC(=O)c1ccc(N[C@H]2CCO[C@@H]2C)cc1 ZINC000147417438 CF For-Sale Anodyne CNGA1 0 40 O=C(NCC1(C(=O)O)CCC1)c1ccc(Cl)c(Cl)c1 ZINC000147417464 DF On-Demand Anodyne KMO 0 41 C[C@@H]1CCC[C@@H](C)N1NC(=O)c1ccc2c(c1)CNCC2 ZINC000147417469 CE For-Sale Anodyne PNMT 19 41 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCN(C)CC3)cc2)cc([N+](=O)[O-])c1 ZINC000147417476 HE On-Demand Bother CPT1A 34 41 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCN(C)CC3)cc2)cc([N+](=O)[O-])c1 ZINC000147417476 HE On-Demand Bother TGM2 62 40 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCN(C)CC3)cc2)cc([N+](=O)[O-])c1 ZINC000147417476 HE On-Demand Bother F13A1 86 41 Cc1cc(C(=O)Nc2ccc(S(=O)(=O)N3CCN(C)CC3)cc2)cc([N+](=O)[O-])c1 ZINC000147417476 HE On-Demand Bother WDR5 34 40 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne F2 44 42 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne CHRM5 41 41 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne MMP13 16 41 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne CTSK 22 40 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne PCSK5 25 44 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne FURIN 29 44 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne CAPN1 37 40 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne CAPN2 40 39 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne TGM2 64 44 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne ST14 59 33 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne MMP1 15 40 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne F13A1 66 44 CCC[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147417558 GD On-Demand Anodyne TMPRSS6 52 33 CCNC(=O)CN1CCN(C(=O)C2(NC(=O)NCc3ccccc3)CCCC2)CC1 ZINC000147417587 HD On-Demand Anodyne NPFFR1 40 33 CCCOC(=O)c1ccc(N[C@@H]2CCO[C@H]2C)cc1 ZINC000147417629 CF For-Sale Anodyne CNGA1 0 40 NS(=O)(=O)c1cc(F)cc(F)c1OCCn1ccnc1 ZINC000147417651 DC For-Sale Anodyne TBXAS1 30 42 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H]1CCOc3ccc(Br)cc31)C2 ZINC000147417662 HH On-Demand Anodyne MTNR1A 15 41 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H]1CCOc3ccc(Br)cc31)C2 ZINC000147417662 HH On-Demand Anodyne ROCK2 22 41 CC(C)N1CCC(N(C)C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147417665 FI On-Demand Anodyne HRH3 0 46 CCc1ncc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)s1 ZINC000147417729 FF On-Demand Anodyne PREP 19 42 CCc1ncc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)s1 ZINC000147417729 FF On-Demand Anodyne EPHX2 27 46 CCc1ncc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)s1 ZINC000147417729 FF On-Demand Anodyne PTR1 49 35 CCc1ncc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)s1 ZINC000147417729 FF On-Demand Anodyne PDS 40 32 COC(=O)c1ccc(N2CCN(CC(=O)O)CC2)nc1C ZINC000147417780 CC For-Sale Anodyne SLC27A1 56 36 CCNC(=O)CN1CCN(C(=O)[C@@H]2CC=CC[C@@H]2c2nc3ccccc3s2)CC1 ZINC000147417785 HF On-Demand Anodyne SLC27A1 17 40 CCCOC(=O)c1ccc(N[C@H]2CCO[C@H]2C)cc1 ZINC000147417841 CF For-Sale Anodyne CNGA1 0 40 O=C(NCC1(C(=O)O)CCC1)c1cccc(F)c1F ZINC000147417894 CD On-Demand Anodyne HCN1 61 33 O=C(NCC1(C(=O)O)CCC1)c1cccc(F)c1F ZINC000147417894 CD On-Demand Anodyne HCN4 49 31 Cc1cc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147417914 GG On-Demand Bother TACR1 15 44 Cc1cc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147417914 GG On-Demand Bother EPHX2 33 52 Cc1cc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147417914 GG On-Demand Bother L3MBTL1 0 40 Cc1cc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147417914 GG On-Demand Bother L3MBTL3 48 40 Cc1cc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)cc([N+](=O)[O-])c1 ZINC000147417914 GG On-Demand Bother TP53BP1 0 40 COc1ccc(C[C@H](C)NCC(F)F)cc1 ZINC000147417920 BE On-Demand Anodyne ADRB2 15 58 COc1ccc(C[C@H](C)NCC(F)F)cc1 ZINC000147417920 BE On-Demand Anodyne ADRB1 20 48 O=C(O)c1cc(Cl)c2nc(-n3ccnc3)nc(N3CCOCC3)c2n1 ZINC000147417951 FD For-Sale Anodyne NOS2 55 33 CCNC(=O)CN1CCN(C(=O)[C@H]2CC=CC[C@@H]2c2nc3ccccc3s2)CC1 ZINC000147418015 HF On-Demand Anodyne SLC27A1 17 40 CCO[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147418036 HF On-Demand Anodyne CHRM5 19 45 CCO[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147418036 HF On-Demand Anodyne EPHX2 17 42 CCO[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147418036 HF On-Demand Anodyne TGM2 68 46 CCO[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147418036 HF On-Demand Anodyne F13A1 73 46 NS(=O)(=O)c1cc(F)cc(F)c1OCCCn1ccnc1 ZINC000147418065 DD For-Sale Anodyne TBXAS1 37 41 NS(=O)(=O)c1cc(F)cc(F)c1OCCCn1ccnc1 ZINC000147418065 DD For-Sale Anodyne HMOX2 40 38 COCc1nc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)cs1 ZINC000147418125 FE On-Demand Anodyne PREP 19 42 COCc1nc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)cs1 ZINC000147418125 FE On-Demand Anodyne EPHX2 20 46 COCc1nc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)cs1 ZINC000147418125 FE On-Demand Anodyne PTR1 47 34 COCc1nc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)cs1 ZINC000147418125 FE On-Demand Anodyne TRPC6 68 41 COCc1nc(C(=O)N2CCC(C(=O)NCc3ccccc3)CC2)cs1 ZINC000147418125 FE On-Demand Anodyne TRPC3 40 41 COc1ccc(C[C@@H](C)NCC(F)F)cc1 ZINC000147418133 BE On-Demand Anodyne ADRB2 15 58 COc1ccc(C[C@@H](C)NCC(F)F)cc1 ZINC000147418133 BE On-Demand Anodyne ADRB1 20 48 CCNC(=O)CN1CCN(C(=O)[C@@H]2CC=CC[C@H]2c2nc3ccccc3s2)CC1 ZINC000147418217 HF On-Demand Anodyne SLC27A1 17 40 CC(C)S(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3ccc(F)cn3)no2)CC1 ZINC000147418245 GF Annotated Anodyne NPY2R 31 43 CC(C)S(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3ccc(F)cn3)no2)CC1 ZINC000147418245 GF Annotated Anodyne NPY5R 19 43 CC(C)S(=O)(=O)NC[C@@H]1CC[C@@H](Nc2nc(-c3ccc(F)cn3)no2)CC1 ZINC000147418245 GF Annotated Anodyne HCAR2 24 41 Clc1ccc2c(N(CCBr)C3CCCCC3)ccnc2c1 ZINC000147418248 FK For-Sale Reactive HRP1_PLAFA 92 40 Clc1ccc2c(N(CCBr)C3CCCCC3)ccnc2c1 ZINC000147418248 FK For-Sale Reactive HNMT 58 38 CCO[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147418271 HF On-Demand Anodyne CHRM5 19 45 CCO[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147418271 HF On-Demand Anodyne EPHX2 17 42 CCO[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147418271 HF On-Demand Anodyne TGM2 68 46 CCO[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147418271 HF On-Demand Anodyne F13A1 73 46 Cc1cc(C(=O)NCCCN(C)Cc2ccccc2)cc([N+](=O)[O-])c1 ZINC000147418346 EG On-Demand Bother ACHE 23 50 COC(=O)c1cc([N+](=O)[O-])ccc1/C=C/c1ccc(F)cc1 ZINC000147418384 DH For-Sale Bother CACNA1C 58 38 COC(=O)c1cc([N+](=O)[O-])ccc1/C=C/c1ccc(F)cc1 ZINC000147418384 DH For-Sale Bother CACNA1D 90 38 CCNC(=O)CN1CCN(C(=O)[C@H]2CC=CC[C@H]2c2nc3ccccc3s2)CC1 ZINC000147418421 HF On-Demand Anodyne SLC27A1 17 40 CNC(=O)c1ccccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147418449 FH On-Demand Anodyne F10 22 46 CNC(=O)c1ccccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147418449 FH On-Demand Anodyne PPARD 0 41 CNC(=O)c1ccccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147418449 FH On-Demand Anodyne NR1H4 25 49 CNC(=O)c1ccccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147418449 FH On-Demand Anodyne FABH 0 50 CNC(=O)c1ccccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147418449 FH On-Demand Anodyne PAGA 0 45 O=C(CN1CCc2ccccc21)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147418509 HE On-Demand Anodyne APP 45 37 O=C(CN1CCc2ccccc21)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147418509 HE On-Demand Anodyne TGM2 59 43 O=C(CN1CCc2ccccc21)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147418509 HE On-Demand Anodyne F13A1 56 43 O=C(CN1CCc2ccccc21)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147418509 HE On-Demand Anodyne AKR1C3 59 38 N#Cc1cccc(S(=O)(=O)CCN2CCC(CO)CC2)c1 ZINC000147418542 DD On-Demand Mild CCR3 22 44 N#Cc1cccc(S(=O)(=O)CCN2CCC(CO)CC2)c1 ZINC000147418542 DD On-Demand Mild MEN1 49 34 CC(C)CCCCNS(=O)(=O)CCCN ZINC000147418577 BD For-Sale Anodyne RELA 23 51 CC(C)CNCCC[C@@H](C)Oc1ccc(Cl)c(F)c1 ZINC000147418587 CI For-Sale Anodyne LEF 40 35 O=S(=O)(c1cc(F)ccc1F)N1CCN(CCBr)CC1 ZINC000147418629 FD For-Sale Reactive HTR2A 15 51 CNC(=O)c1ccccc1NC(=O)c1cc(C)ccc1Br ZINC000147418637 EG On-Demand Anodyne PPARA 0 41 CNC(=O)c1ccccc1NC(=O)c1cc(C)ccc1Br ZINC000147418637 EG On-Demand Anodyne NR1H4 23 48 CNC(=O)c1ccccc1NC(=O)c1cc(C)ccc1Br ZINC000147418637 EG On-Demand Anodyne FABH 0 42 CNC(=O)c1ccccc1NC(=O)c1cc(C)ccc1Br ZINC000147418637 EG On-Demand Anodyne KCNK3 47 37 CNC(=O)c1ccccc1NC(=O)c1cc(C)ccc1Br ZINC000147418637 EG On-Demand Anodyne KCNK9 47 37 CCNC(=O)CN1CCN(C(=O)[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147418656 HD On-Demand Anodyne P2RY12 84 39 CCNC(=O)CN1CCN(C(=O)[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147418656 HD On-Demand Anodyne CCR1 18 41 CCNC(=O)CN1CCN(C(=O)[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147418656 HD On-Demand Anodyne MTTP 91 45 CCNC(=O)CN1CCN(C(=O)[C@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147418656 HD On-Demand Anodyne CCKBR 45 38 COC[C@@]1(CO)CCN(Cc2ccccc2)C1 ZINC000147418662 BD On-Demand Anodyne DRD3 16 41 COC[C@@]1(CO)CCN(Cc2ccccc2)C1 ZINC000147418662 BD On-Demand Anodyne SIGMAR1 75 43 COC[C@@]1(CO)CCN(Cc2ccccc2)C1 ZINC000147418662 BD On-Demand Anodyne NPFFR2 32 40 COC[C@@]1(CO)CCN(Cc2ccccc2)C1 ZINC000147418662 BD On-Demand Anodyne NPFFR1 56 41 COC[C@H](N)C(C)=O ZINC000147418698 AB For-Sale Anodyne GRIK3 37 41 COC[C@H](N)C(C)=O ZINC000147418698 AB For-Sale Anodyne GRIK2 23 41 COC[C@H](N)C(C)=O ZINC000147418698 AB For-Sale Anodyne GRIK1 49 41 CC(C)CNCCC[C@H](C)Oc1ccc(Cl)c(F)c1 ZINC000147418807 CI For-Sale Anodyne LEF 40 35 COC[C@]1(CO)CCN(Cc2ccccc2)C1 ZINC000147418869 BD On-Demand Anodyne DRD3 16 41 COC[C@]1(CO)CCN(Cc2ccccc2)C1 ZINC000147418869 BD On-Demand Anodyne SIGMAR1 75 43 COC[C@]1(CO)CCN(Cc2ccccc2)C1 ZINC000147418869 BD On-Demand Anodyne NPFFR2 32 40 COC[C@]1(CO)CCN(Cc2ccccc2)C1 ZINC000147418869 BD On-Demand Anodyne NPFFR1 56 41 CCNC(=O)CN1CCN(C(=O)[C@@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147418880 HD On-Demand Anodyne P2RY12 84 39 CCNC(=O)CN1CCN(C(=O)[C@@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147418880 HD On-Demand Anodyne CCR1 18 41 CCNC(=O)CN1CCN(C(=O)[C@@H](NC(=O)c2ccccc2)c2ccccc2)CC1 ZINC000147418880 HD On-Demand Anodyne MTTP 91 45 CCCS(=O)(=O)Nc1ccccc1C(=O)N[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147418922 GG On-Demand Bother CACNA1D 57 35 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1 ZINC000147418979 HI On-Demand Anodyne SCD1 41 55 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1 ZINC000147418979 HI On-Demand Anodyne SCD 40 55 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(CN3CCCCC3)c2)C1 ZINC000147418985 HG On-Demand Anodyne HRH2 52 43 O=C(NC1CCC(C(F)(F)F)CC1)c1ccc(Br)c(Cl)c1 ZINC000147419020 GJ On-Demand Anodyne MAPK14 43 37 O=C(NC1CCC(C(F)(F)F)CC1)c1ccc(Br)c(Cl)c1 ZINC000147419020 GJ On-Demand Anodyne MAPK13 63 37 CC(C)NCCCCCOc1ccc(Cl)c(F)c1 ZINC000147419035 CI For-Sale Anodyne HT1 0 40 NC(=O)c1csc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147419058 HD On-Demand Anodyne EPHX2 15 40 NC(=O)c1csc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147419058 HD On-Demand Anodyne TGM2 62 44 NC(=O)c1csc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147419058 HD On-Demand Anodyne ST14 47 32 NC(=O)c1csc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147419058 HD On-Demand Anodyne CACNA1I 59 34 NC(=O)c1csc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147419058 HD On-Demand Anodyne F13A1 50 44 NC(=O)c1csc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147419058 HD On-Demand Anodyne SIRT3 52 34 NC(=O)c1csc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147419058 HD On-Demand Anodyne SIRT2 52 34 NC(=O)c1csc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147419058 HD On-Demand Anodyne SIRT1 52 34 NC(=O)c1csc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147419058 HD On-Demand Anodyne AKR1C3 55 37 NC(=O)c1csc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147419058 HD On-Demand Anodyne NAMPT 32 40 Cc1cccc(CC(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147419065 CD On-Demand Anodyne KCNK9 43 39 CCc1nc(CN(C)C(=O)NC2CCN(S(C)(=O)=O)CC2)cs1 ZINC000147419089 FD On-Demand Anodyne NPY2R 18 46 NS(=O)(=O)c1cc(F)cc(F)c1OCCN1CCCC1 ZINC000147419092 DD For-Sale Anodyne LTA4H 29 43 NS(=O)(=O)c1cc(F)cc(F)c1OCCN1CCCC1 ZINC000147419092 DD For-Sale Anodyne PSMB2 44 35 CCCS(=O)(=O)Nc1ccccc1C(=O)N[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147419129 GG On-Demand Bother CACNA1D 57 35 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(CN3CCCCC3)c2)C1 ZINC000147419184 HG On-Demand Anodyne HRH2 52 43 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1 ZINC000147419208 HI On-Demand Anodyne SCD1 41 55 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1 ZINC000147419208 HI On-Demand Anodyne SCD 40 55 N#Cc1cccc(S(=O)(=O)CCN2CCCC[C@@H]2CO)c1 ZINC000147419216 DD On-Demand Mild CHRNA10 28 44 O=C(Nc1ccc2[nH]ccc2c1)c1ccc(Br)c(Cl)c1 ZINC000147419312 EJ On-Demand Anodyne MAOB 24 71 O=C(Nc1ccc2[nH]ccc2c1)c1ccc(Br)c(Cl)c1 ZINC000147419312 EJ On-Demand Anodyne TAAR1 19 42 O=C(Nc1ccc2[nH]ccc2c1)c1ccc(Br)c(Cl)c1 ZINC000147419312 EJ On-Demand Anodyne NR2E3 60 36 O=C(Nc1ccc2[nH]ccc2c1)c1ccc(Br)c(Cl)c1 ZINC000147419312 EJ On-Demand Anodyne KCNK3 44 35 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Br)c1)C(=O)NCc1ccccc1 ZINC000147419339 HG On-Demand Anodyne ANPEP 34 40 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Br)c1)C(=O)NCc1ccccc1 ZINC000147419339 HG On-Demand Anodyne AMP1_PLAFQ 51 40 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Br)c1)C(=O)NCc1ccccc1 ZINC000147419339 HG On-Demand Anodyne PDS 49 41 CCNC(=O)CN1CCN(C(=O)c2ccc(C(N)=O)cc2)CC1 ZINC000147419340 DB On-Demand Anodyne PLA2G2A 21 40 CCNC(=O)CN1CCN(C(=O)c2ccc(C(N)=O)cc2)CC1 ZINC000147419340 DB On-Demand Anodyne L3MBTL3 51 34 CC(C)N(Cc1ccccn1)C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147419356 GE On-Demand Bother COLA 65 36 CC1(C)Oc2ccc(NC(=O)NCc3cccc(NC(=O)[C@@H]4CCCO4)c3)cc2O1 ZINC000147419357 HH On-Demand Anodyne ROCK2 17 40 CCCCCCCCOc1ccc(CNCCC)nc1 ZINC000147419360 CI For-Sale Mild LPAR2 63 49 CCCCCCCCOc1ccc(CNCCC)nc1 ZINC000147419360 CI For-Sale Mild S1PR3 31 49 CCCCCCCCOc1ccc(CNCCC)nc1 ZINC000147419360 CI For-Sale Mild PLA2G4B 85 37 CCCCCCCCOc1ccc(CNCCC)nc1 ZINC000147419360 CI For-Sale Mild S1PR2 68 49 CCCCCCCCOc1ccc(CNCCC)nc1 ZINC000147419360 CI For-Sale Mild S1PR1 15 49 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1 ZINC000147419381 HI On-Demand Anodyne SCD1 49 56 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1 ZINC000147419381 HI On-Demand Anodyne SCD 40 55 N#Cc1cccc(S(=O)(=O)CCN2CCCC[C@H]2CO)c1 ZINC000147419415 DD On-Demand Mild CHRNA10 28 44 C[C@H](Oc1cccc(Cl)c1)C(=O)N1CCC[C@@H]1CCCBr ZINC000147419430 FI For-Sale Reactive CHRNA10 35 45 Cc1c(C(=O)O)cccc1S(=O)(=O)NCCc1ccc(Cl)cc1 ZINC000147419437 FF On-Demand Anodyne TBXA2R 18 42 Cc1c(C(=O)O)cccc1S(=O)(=O)NCCc1ccc(Cl)cc1 ZINC000147419437 FF On-Demand Anodyne TBXAS1 35 42 O=C(CCOCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147419542 HF On-Demand Anodyne GRIN2B 42 40 O=C(CCOCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147419542 HF On-Demand Anodyne SIGMAR1 15 53 O=C(CCOCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147419542 HF On-Demand Anodyne EPHX2 16 41 O=C(CCOCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147419542 HF On-Demand Anodyne TGM2 83 53 O=C(CCOCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147419542 HF On-Demand Anodyne F13A1 93 53 O=C(CCOCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147419542 HF On-Demand Anodyne NAMPT 33 41 Nc1nc(Br)c(-c2ccccc2)s1 ZINC000147419545 CG For-Sale Anodyne FBP1 17 43 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1 ZINC000147419571 HI On-Demand Anodyne SCD1 41 55 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1ncc(Cc2cccc(C(F)(F)F)c2)s1 ZINC000147419571 HI On-Demand Anodyne SCD 40 55 COc1cc(Br)cc(C)c1NC(=O)Nc1ccc2c(c1)n(C)c(=O)n2C ZINC000147419573 HH On-Demand Anodyne HTR2A 23 40 CC1(C)Oc2ccc(NC(=O)NCc3cccc(NC(=O)[C@H]4CCCO4)c3)cc2O1 ZINC000147419576 HH On-Demand Anodyne ROCK2 17 40 COc1nc(N)nc(Oc2ccc(Br)cc2Cl)n1 ZINC000147419599 EF For-Sale Anodyne AGPAT2 36 41 CC(=O)Nc1ccc(-c2noc(C(F)(F)F)n2)cc1 ZINC000147419628 CF On-Demand Anodyne IDO1 0 40 C[C@@H](Oc1cccc(Cl)c1)C(=O)N1CCC[C@@H]1CCCBr ZINC000147419660 FI For-Sale Reactive CHRNA10 35 45 CC(C)CN(CCS(=O)(=O)c1cccc(C#N)c1)C(C)C ZINC000147419661 DF On-Demand Mild NR1H2 15 45 COC(=O)c1ccc(N(CC(=O)O)C2CCCC2)nc1C ZINC000147419675 CE For-Sale Anodyne ACE 51 37 CCN(CC)C(=O)c1ccc(S(=O)(=O)N2C[C@H](C)O[C@H](c3ccccc3)C2)cc1 ZINC000147419678 HG On-Demand Anodyne OPRM1 21 41 CCN(CC)C(=O)c1ccc(S(=O)(=O)N2C[C@H](C)O[C@H](c3ccccc3)C2)cc1 ZINC000147419678 HG On-Demand Anodyne OPRD1 39 43 CCN(CC)C(=O)c1ccc(S(=O)(=O)N2C[C@H](C)O[C@H](c3ccccc3)C2)cc1 ZINC000147419678 HG On-Demand Anodyne LIMK2 18 40 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne MAPK14 34 48 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne CPT1A 76 39 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne CPT2 50 38 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne GRM4 23 54 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne CPT1B 53 39 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne PDGFRA 41 38 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne IMPDH2 0 47 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne TEK 43 33 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne TAAR1 43 57 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne ENPP1 49 33 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne SMO 22 44 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne GLMU 0 44 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne KCNK3 98 42 COc1cc(C(=O)Nc2ccc(C)c(Br)c2)ccc1F ZINC000147419691 EI On-Demand Anodyne KCNK9 71 42 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Br)c1)C(=O)NCc1ccccc1 ZINC000147419746 HG On-Demand Anodyne ANPEP 34 40 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Br)c1)C(=O)NCc1ccccc1 ZINC000147419746 HG On-Demand Anodyne AMP1_PLAFQ 51 40 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Br)c1)C(=O)NCc1ccccc1 ZINC000147419746 HG On-Demand Anodyne PDS 49 41 C/C=C(\C)CC/C=C(\C)C=O ZINC000147419756 AF For-Sale Reactive GGPS1 19 44 COCc1nc(C(=O)N2CCN(Cc3ccc4c(c3)OCCO4)CC2)cs1 ZINC000147419772 GE On-Demand Anodyne NOS2 54 34 COCc1nc(C(=O)N2CCN(Cc3ccc4c(c3)OCCO4)CC2)cs1 ZINC000147419772 GE On-Demand Anodyne MCHR1 23 40 COCc1nc(C(=O)N2CCN(Cc3ccc4c(c3)OCCO4)CC2)cs1 ZINC000147419772 GE On-Demand Anodyne TRPC6 55 40 COCc1nc(C(=O)N2CCN(Cc3ccc4c(c3)OCCO4)CC2)cs1 ZINC000147419772 GE On-Demand Anodyne TRPC3 39 40 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3ccc4c(c3)OC(C)(C)O4)c2)CCO1 ZINC000147419785 HH On-Demand Anodyne HRH2 20 40 CC[C@H](NC(=O)N1CCC[C@H]2CCCC[C@H]21)C(=O)O ZINC000147419789 CE For-Sale Anodyne ACE 41 40 CC[C@H](NC(=O)N1CCC[C@H]2CCCC[C@H]21)C(=O)O ZINC000147419789 CE For-Sale Anodyne SLC5A1 19 40 CC(C)[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(Cl)cc1 ZINC000147419801 EI On-Demand Anodyne CYP3A4 16 42 CC(C)[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(Cl)cc1 ZINC000147419801 EI On-Demand Anodyne UTS2 41 32 C[C@H](Oc1cccc(Cl)c1)C(=O)N1CCC[C@H]1CCCBr ZINC000147419863 FI For-Sale Reactive CHRNA10 35 45 C=C1CN(Cc2ccc(C(=O)Nc3ccccc3N)cc2)C(=O)c2ccccc21 ZINC000147419870 GI In-Stock Anodyne HDAC8 32 44 C=C1CN(Cc2ccc(C(=O)Nc3ccccc3N)cc2)C(=O)c2ccccc21 ZINC000147419870 GI In-Stock Anodyne HDAC1 116 78 C=C1CN(Cc2ccc(C(=O)Nc3ccccc3N)cc2)C(=O)c2ccccc21 ZINC000147419870 GI In-Stock Anodyne HDAC2 49 45 C=C1CN(Cc2ccc(C(=O)Nc3ccccc3N)cc2)C(=O)c2ccccc21 ZINC000147419870 GI In-Stock Anodyne HDAC3 37 48 C=C1CN(Cc2ccc(C(=O)Nc3ccccc3N)cc2)C(=O)c2ccccc21 ZINC000147419870 GI In-Stock Anodyne NOD2 41 35 CCN(CC)C(=O)c1ccc(S(=O)(=O)N2C[C@@H](C)O[C@H](c3ccccc3)C2)cc1 ZINC000147419896 HG On-Demand Anodyne OPRM1 21 41 CCN(CC)C(=O)c1ccc(S(=O)(=O)N2C[C@@H](C)O[C@H](c3ccccc3)C2)cc1 ZINC000147419896 HG On-Demand Anodyne OPRD1 39 43 CCN(CC)C(=O)c1ccc(S(=O)(=O)N2C[C@@H](C)O[C@H](c3ccccc3)C2)cc1 ZINC000147419896 HG On-Demand Anodyne LIMK2 18 40 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3ccc4c(c3)OC(C)(C)O4)c2)CCO1 ZINC000147419982 HH On-Demand Anodyne HRH2 20 40 Cc1ccc2oc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147419994 HH On-Demand Anodyne HTR4 56 38 Cc1ccc2oc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147419994 HH On-Demand Anodyne EPHX2 31 41 Cc1ccc2oc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147419994 HH On-Demand Anodyne TGM2 57 44 Cc1ccc2oc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147419994 HH On-Demand Anodyne CACNA1I 59 42 Cc1ccc2oc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147419994 HH On-Demand Anodyne F13A1 48 44 Cc1ccc2oc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147419994 HH On-Demand Anodyne NAMPT 50 46 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(-n4cccn4)c(F)c3)ccc21 ZINC000147419995 GF On-Demand Anodyne FPR2 42 36 CC[C@H](NC(=O)N1CCC[C@@H]2CCCC[C@H]21)C(=O)O ZINC000147420024 CE For-Sale Anodyne ACE 41 40 CC[C@H](NC(=O)N1CCC[C@@H]2CCCC[C@H]21)C(=O)O ZINC000147420024 CE For-Sale Anodyne SLC5A1 19 40 CC(C)[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(Cl)cc1 ZINC000147420044 EI On-Demand Anodyne CYP3A4 16 42 CC(C)[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(Cl)cc1 ZINC000147420044 EI On-Demand Anodyne UTS2 41 32 O=C(NCc1ccc(F)cc1Cl)c1c[nH]nn1 ZINC000147420073 CD In-Stock Anodyne P2RX7 91 52 O=C(NCc1ccc(F)cc1Cl)c1c[nH]nn1 ZINC000147420073 CD In-Stock Anodyne ALPL 54 33 C[C@@H](Oc1cccc(Cl)c1)C(=O)N1CCC[C@H]1CCCBr ZINC000147420076 FI For-Sale Reactive CHRNA10 35 45 Nc1ccc([N+](=O)[O-])cc1C(=O)Nc1ccc(Cl)cc1Br ZINC000147420086 FH For-Sale Bother F10 0 40 Nc1ccc([N+](=O)[O-])cc1C(=O)Nc1ccc(Cl)cc1Br ZINC000147420086 FH For-Sale Bother KCNMA1 47 54 Nc1ccc([N+](=O)[O-])cc1C(=O)Nc1ccc(Cl)cc1Br ZINC000147420086 FH For-Sale Bother WDR5 34 42 C/C=C(\C)CC/C=C(/C)C=O ZINC000147420163 AF For-Sale Reactive GGPS1 19 44 CCCCCCCCNCC(F)F ZINC000147420196 AG For-Sale Mild S1PR2 33 41 CCCCCCCCNCC(F)F ZINC000147420196 AG For-Sale Mild Q8WS26_TRYCR 45 52 C=CCNC(=O)c1cccc(S(=O)(=O)N2C[C@H](c3ccccc3)O[C@H](C)C2)c1 ZINC000147420217 HF On-Demand Mild TGM2 40 36 C=CCNC(=O)c1cccc(S(=O)(=O)N2C[C@H](c3ccccc3)O[C@H](C)C2)c1 ZINC000147420217 HF On-Demand Mild AKR1C3 56 39 CCNc1ncnc(Oc2ccc(Br)cc2Cl)c1[N+](=O)[O-] ZINC000147420230 FI For-Sale Bother S1PR4 17 47 COC(=O)c1ccc(C)c(NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)c1 ZINC000147420232 FF On-Demand Anodyne MAPK14 24 42 C/C=C(/C)CC/C=C(/C)C=O ZINC000147420314 AF For-Sale Reactive GGPS1 19 44 COc1cc(C(=O)N2CCC[C@@H]2CCCBr)ccc1C ZINC000147420341 EH For-Sale Reactive HCRTR1 0 47 COc1cc(C(=O)N2CCC[C@@H]2CCCBr)ccc1C ZINC000147420341 EH For-Sale Reactive ACKR3 69 36 CC(C)Oc1ccccc1CNCC(F)F ZINC000147420383 BF On-Demand Anodyne PHES 0 44 NC(=O)NNc1ccc(O)cc1 ZINC000147420388 AC For-Sale Reactive H9TVJ1_CHISP 40 30 C=CCNC(=O)c1cccc(S(=O)(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)c1 ZINC000147420418 HF On-Demand Mild TGM2 40 36 C=CCNC(=O)c1cccc(S(=O)(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)c1 ZINC000147420418 HF On-Demand Mild AKR1C3 56 39 COC(=O)c1ccc(N2CCCC[C@@H]2CC(=O)O)nc1C ZINC000147420426 CE On-Demand Anodyne NOS2 25 41 CCNCCCCCCOc1ccc(Cl)c(F)c1 ZINC000147420506 CI For-Sale Anodyne DRD4 20 45 O=C(O)c1cc(Cl)cc(NC(=O)N2CCC[C@H](O)C2)c1 ZINC000147420571 CE On-Demand Anodyne CACNA1I 45 34 COc1cc(C(=O)N2CCC[C@H]2CCCBr)ccc1C ZINC000147420576 EH For-Sale Reactive HCRTR1 0 47 COc1cc(C(=O)N2CCC[C@H]2CCCBr)ccc1C ZINC000147420576 EH For-Sale Reactive ACKR3 69 36 COC(=O)c1ccc(N2CCCC[C@H]2CC(=O)O)nc1C ZINC000147420630 CE On-Demand Anodyne NOS2 25 41 Cc1nc(-c2ccc(NC(=O)Nc3ccc4c(c3)n(C)c(=O)n4C)cc2)oc1C ZINC000147420657 GH On-Demand Anodyne LPL 50 33 Cc1nc(-c2ccc(NC(=O)Nc3ccc4c(c3)n(C)c(=O)n4C)cc2)oc1C ZINC000147420657 GH On-Demand Anodyne MTOR 42 37 CC[C@H](NC(=O)c1cccn(Cc2ccccc2)c1=O)c1ccccc1OC(F)F ZINC000147420703 HI On-Demand Anodyne CTSA 42 32 COc1ccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)cn1 ZINC000147420736 HD On-Demand Anodyne ROCK2 23 42 CC(C)NS(=O)(=O)Cc1ccc(CNC(=O)N(C)Cc2cscn2)cc1 ZINC000147420741 GE On-Demand Anodyne TMPRSS11D 57 35 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild CNR1 18 48 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild INHA 82 39 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild CNR2 20 42 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild LPAR2 58 36 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild S1PR3 43 38 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild MTNR1A 47 41 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild MTNR1B 45 43 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild GRIA1 41 37 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild PLA2G4B 88 38 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild SOAT1 41 38 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild FAAH 41 48 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild S1PR2 88 38 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild EPHX2 15 41 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild ASAH1 104 40 CCCCCCCCNC(=O)COc1ccccc1OCC(=O)NCCCCCCCC ZINC000147420767 IK For-Sale Mild LIPG 15 41 O=C(O)c1cc(Cl)cc(NC(=O)N2CCC[C@@H](O)C2)c1 ZINC000147420779 CE On-Demand Anodyne CACNA1I 45 34 Cc1cccc(CC(=O)NCC[C@H](C)c2ccccc2)c1 ZINC000147420813 CH On-Demand Anodyne MME 37 40 Cc1cccc(CC(=O)NCC[C@H](C)c2ccccc2)c1 ZINC000147420813 CH On-Demand Anodyne ANPEP 31 40 Cc1cccc(CC(=O)NCC[C@H](C)c2ccccc2)c1 ZINC000147420813 CH On-Demand Anodyne CMA1 17 44 Cc1cccc(CC(=O)NCC[C@H](C)c2ccccc2)c1 ZINC000147420813 CH On-Demand Anodyne CTSB 26 44 Cc1cccc(CC(=O)NCC[C@H](C)c2ccccc2)c1 ZINC000147420813 CH On-Demand Anodyne CTSL 28 44 Cc1cccc(CC(=O)NCC[C@H](C)c2ccccc2)c1 ZINC000147420813 CH On-Demand Anodyne C3AR1 44 32 Cc1cccc(CC(=O)NCC[C@H](C)c2ccccc2)c1 ZINC000147420813 CH On-Demand Anodyne NCE103 20 40 Cc1cccc(CC(=O)NCC[C@H](C)c2ccccc2)c1 ZINC000147420813 CH On-Demand Anodyne P96878_MYCTU 17 40 COc1cc(NC(=O)c2c[nH]c(-c3ccccc3)n2)cc(OC)c1OC ZINC000147420842 FG On-Demand Anodyne CPT1A 47 33 COc1cc(NC(=O)c2c[nH]c(-c3ccccc3)n2)cc(OC)c1OC ZINC000147420842 FG On-Demand Anodyne GRM4 21 44 COc1cc(NC(=O)c2c[nH]c(-c3ccccc3)n2)cc(OC)c1OC ZINC000147420842 FG On-Demand Anodyne PTK2 54 42 COc1cc(NC(=O)c2c[nH]c(-c3ccccc3)n2)cc(OC)c1OC ZINC000147420842 FG On-Demand Anodyne NR2E3 53 33 COc1cc(NC(=O)c2c[nH]c(-c3ccccc3)n2)cc(OC)c1OC ZINC000147420842 FG On-Demand Anodyne ENPP1 50 30 COc1cc(NC(=O)c2c[nH]c(-c3ccccc3)n2)cc(OC)c1OC ZINC000147420842 FG On-Demand Anodyne SMO 27 44 O=C(c1cc2ccccc2o1)N1CCC[C@@H]1CCCBr ZINC000147420868 EI For-Sale Reactive HCRTR1 17 40 O=C(c1cc2ccccc2o1)N1CCC[C@@H]1CCCBr ZINC000147420868 EI For-Sale Reactive PREP 40 34 CCOc1ccc([C@@H](C)NC(=O)[C@@H](C)OCCC(C)C)cc1 ZINC000147420917 DH On-Demand Anodyne ACACA 33 53 CCOc1ccc([C@@H](C)NC(=O)[C@@H](C)OCCC(C)C)cc1 ZINC000147420917 DH On-Demand Anodyne ACACB 36 56 C[C@H]1Cc2ccccc2C[C@@H]1c1ccccc1 ZINC000147420931 BI For-Sale Anodyne PRCP 19 42 O=C(NCc1cccc(C(=O)NC[C@@H]2CCCO2)c1)C(=O)Nc1cccnc1 ZINC000147420950 GD On-Demand Anodyne NAMPT 60 42 CN(Cc1cscn1)C(=O)N[C@@H](c1ccccc1)c1cc2ccccc2o1 ZINC000147420985 GJ On-Demand Anodyne CYP3A4 20 42 O=C(CC(F)(F)F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421009 FE On-Demand Anodyne CHRM5 18 40 O=C(CC(F)(F)F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421009 FE On-Demand Anodyne EPHX2 36 49 O=C(CC(F)(F)F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421009 FE On-Demand Anodyne TGM2 88 48 O=C(CC(F)(F)F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421009 FE On-Demand Anodyne CACNA1I 56 38 O=C(CC(F)(F)F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421009 FE On-Demand Anodyne F13A1 96 48 O=C(CC(F)(F)F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421009 FE On-Demand Anodyne AKR1C3 54 38 O=C(CC(F)(F)F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421009 FE On-Demand Anodyne SFRP1 108 45 O=C(CC(F)(F)F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421009 FE On-Demand Anodyne WNT3 65 33 O=C(CC(F)(F)F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421009 FE On-Demand Anodyne NAMPT 31 40 Cc1cccc(CC(=O)NCC[C@@H](C)c2ccccc2)c1 ZINC000147421020 CH On-Demand Anodyne MME 37 40 Cc1cccc(CC(=O)NCC[C@@H](C)c2ccccc2)c1 ZINC000147421020 CH On-Demand Anodyne ANPEP 31 40 Cc1cccc(CC(=O)NCC[C@@H](C)c2ccccc2)c1 ZINC000147421020 CH On-Demand Anodyne CMA1 17 44 Cc1cccc(CC(=O)NCC[C@@H](C)c2ccccc2)c1 ZINC000147421020 CH On-Demand Anodyne CTSB 26 44 Cc1cccc(CC(=O)NCC[C@@H](C)c2ccccc2)c1 ZINC000147421020 CH On-Demand Anodyne CTSL 28 44 Cc1cccc(CC(=O)NCC[C@@H](C)c2ccccc2)c1 ZINC000147421020 CH On-Demand Anodyne C3AR1 44 32 Cc1cccc(CC(=O)NCC[C@@H](C)c2ccccc2)c1 ZINC000147421020 CH On-Demand Anodyne NCE103 20 40 Cc1cccc(CC(=O)NCC[C@@H](C)c2ccccc2)c1 ZINC000147421020 CH On-Demand Anodyne P96878_MYCTU 17 40 O=C(c1cc2ccccc2o1)N1CCC[C@H]1CCCBr ZINC000147421072 EI For-Sale Reactive HCRTR1 17 40 O=C(c1cc2ccccc2o1)N1CCC[C@H]1CCCBr ZINC000147421072 EI For-Sale Reactive PREP 40 34 CCOc1ccc([C@H](C)NC(=O)[C@@H](C)OCCC(C)C)cc1 ZINC000147421127 DH On-Demand Anodyne ACACA 33 53 CCOc1ccc([C@H](C)NC(=O)[C@@H](C)OCCC(C)C)cc1 ZINC000147421127 DH On-Demand Anodyne ACACB 36 56 O=C(NCc1cccc(C(=O)NC[C@H]2CCCO2)c1)C(=O)Nc1cccnc1 ZINC000147421137 GD On-Demand Anodyne NAMPT 60 42 Oc1ccc(OCOCc2ccccc2)cc1 ZINC000147421147 BF For-Sale Anodyne ESR1 15 45 Oc1ccc(OCOCc2ccccc2)cc1 ZINC000147421147 BF For-Sale Anodyne MAOB 22 47 Oc1ccc(OCOCc2ccccc2)cc1 ZINC000147421147 BF For-Sale Anodyne IMPA1 21 43 Oc1ccc(OCOCc2ccccc2)cc1 ZINC000147421147 BF For-Sale Anodyne LTA4H 45 43 Oc1ccc(OCOCc2ccccc2)cc1 ZINC000147421147 BF For-Sale Anodyne ESRRG 47 36 Oc1ccc(OCOCc2ccccc2)cc1 ZINC000147421147 BF For-Sale Anodyne POBA 0 45 Oc1ccc(OCOCc2ccccc2)cc1 ZINC000147421147 BF For-Sale Anodyne TAAR1 26 46 Oc1ccc(OCOCc2ccccc2)cc1 ZINC000147421147 BF For-Sale Anodyne FFAR1 26 46 CC(C)CCCCNCc1cc(Cl)ccc1OC(F)F ZINC000147421168 DJ For-Sale Anodyne LEF 56 39 CN(Cc1cscn1)C(=O)N[C@H](c1ccccc1)c1cc2ccccc2o1 ZINC000147421180 GJ On-Demand Anodyne CYP3A4 20 42 CCNCc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147421202 CI For-Sale Anodyne MAOB 64 47 CCNCc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147421202 CI For-Sale Anodyne F9 0 41 CCNCc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147421202 CI For-Sale Anodyne GYS1 47 36 CCNCc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147421202 CI For-Sale Anodyne FFAR1 50 42 CCNCc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147421202 CI For-Sale Anodyne PDS 57 38 CCCN(CC1CC1)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147421213 DH On-Demand Anodyne CACNA1I 55 37 O=C(NCC1(C(=O)O)CCC1)c1ccccc1Br ZINC000147421300 DE On-Demand Anodyne KCNA3 38 41 O=C(NCC1(C(=O)O)CCC1)c1ccccc1Br ZINC000147421300 DE On-Demand Anodyne MAN2A1 0 41 O=C(NCC1(C(=O)O)CCC1)c1ccccc1Br ZINC000147421300 DE On-Demand Anodyne HCN1 55 34 O=C(NCC1(C(=O)O)CCC1)c1ccccc1Br ZINC000147421300 DE On-Demand Anodyne HCN4 53 34 CC(C)S(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421304 HD On-Demand Anodyne HTR4 45 38 CC(C)S(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421304 HD On-Demand Anodyne CHRM5 18 42 CC(C)S(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421304 HD On-Demand Anodyne MMP13 16 40 CC(C)S(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421304 HD On-Demand Anodyne MMP2 15 40 CC(C)S(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421304 HD On-Demand Anodyne EPHX2 27 40 CC(C)S(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421304 HD On-Demand Anodyne TGM2 73 45 CC(C)S(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421304 HD On-Demand Anodyne CACNA1I 53 35 CC(C)S(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421304 HD On-Demand Anodyne F13A1 77 45 CC(C)S(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421304 HD On-Demand Anodyne AKR1C3 45 33 CC(C)(C)c1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147421308 FJ For-Sale Reactive PREP 28 40 CC(C)(C)c1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147421308 FJ For-Sale Reactive L3MBTL3 48 35 CCOc1ccc([C@@H](C)NC(=O)[C@H](C)OCCC(C)C)cc1 ZINC000147421316 DH On-Demand Anodyne ACACA 33 53 CCOc1ccc([C@@H](C)NC(=O)[C@H](C)OCCC(C)C)cc1 ZINC000147421316 DH On-Demand Anodyne ACACB 36 56 NNC(=O)c1ccc(OCF)cc1 ZINC000147421331 AC For-Sale Reactive ACR 46 36 NNC(=O)c1ccc(OCF)cc1 ZINC000147421331 AC For-Sale Reactive AOC2 0 44 NNC(=O)c1ccc(OCF)cc1 ZINC000147421331 AC For-Sale Reactive AOC3 20 40 NNC(=O)c1ccc(OCF)cc1 ZINC000147421331 AC For-Sale Reactive H9B8T9_CAPHI 24 61 CC[C@@H](CC(=O)O)CN1C(=O)C[C@H](c2ccccc2)C1=O ZINC000147421335 CE For-Sale Anodyne HSD17B2 42 32 CCCOc1ccc(Br)cc1CNCCCCC(C)C ZINC000147421370 EK For-Sale Anodyne S1PR2 43 39 Fc1cc(OCc2cccc(CNC3CC3)c2)ccc1Cl ZINC000147421403 DI For-Sale Anodyne MAOB 48 38 Fc1cc(OCc2cccc(CNC3CC3)c2)ccc1Cl ZINC000147421403 DI For-Sale Anodyne GYS1 43 38 O=C(Nc1ccc2cn[nH]c2c1)c1ccc(Br)c(Cl)c1 ZINC000147421438 FI On-Demand Anodyne MAOB 26 63 O=C(Nc1ccc2cn[nH]c2c1)c1ccc(Br)c(Cl)c1 ZINC000147421438 FI On-Demand Anodyne ROCK1 21 42 O=C(Nc1ccc2cn[nH]c2c1)c1ccc(Br)c(Cl)c1 ZINC000147421438 FI On-Demand Anodyne CSF1R 20 42 O=C(Nc1ccc2cn[nH]c2c1)c1ccc(Br)c(Cl)c1 ZINC000147421438 FI On-Demand Anodyne TAAR1 15 43 O=C(Nc1ccc2cn[nH]c2c1)c1ccc(Br)c(Cl)c1 ZINC000147421438 FI On-Demand Anodyne NR2E3 45 35 O=C(Nc1ccc2cn[nH]c2c1)c1ccc(Br)c(Cl)c1 ZINC000147421438 FI On-Demand Anodyne PHLPP2 0 51 CCCCN(C(=O)Nc1cc(Br)cc(C(=O)O)c1)C1CC1 ZINC000147421447 FH For-Sale Anodyne PPARA 35 43 CN(Cc1cscn1)C(=O)NCC1(c2ccccc2)CCCC1 ZINC000147421449 EH On-Demand Anodyne KCNA3 44 37 CN(Cc1cscn1)C(=O)NCC1(c2ccccc2)CCCC1 ZINC000147421449 EH On-Demand Anodyne ACAT 0 48 CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(OC)cc(OC)c3)[nH]2)cc1 ZINC000147421459 HH Annotated Anodyne ADORA2B 44 36 CCOc1ccc(-c2nnc(SCC(=O)Nc3cc(OC)cc(OC)c3)[nH]2)cc1 ZINC000147421459 HH Annotated Anodyne ENPP1 90 44 CC1(C)Oc2ccc(NC(=O)NCc3ccc(Oc4cccnc4)c(F)c3)cc2O1 ZINC000147421477 HJ On-Demand Anodyne ROCK2 26 45 CC1(C)Oc2ccc(NC(=O)NCc3ccc(Oc4cccnc4)c(F)c3)cc2O1 ZINC000147421477 HJ On-Demand Anodyne MET 33 44 CC1(C)Oc2ccc(NC(=O)NCc3ccc(Oc4cccnc4)c(F)c3)cc2O1 ZINC000147421477 HJ On-Demand Anodyne NAMPT 51 45 CC(C)(C)c1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147421505 FJ For-Sale Reactive PREP 28 40 CC(C)(C)c1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147421505 FJ For-Sale Reactive L3MBTL3 48 35 CCOc1ccc([C@H](C)NC(=O)[C@H](C)OCCC(C)C)cc1 ZINC000147421507 DH On-Demand Anodyne ACACA 33 53 CCOc1ccc([C@H](C)NC(=O)[C@H](C)OCCC(C)C)cc1 ZINC000147421507 DH On-Demand Anodyne ACACB 36 56 Cc1cc(C)n([C@@H](C)C(=O)N2CCC[C@@H]2c2ccc(Cl)c(Cl)c2)n1 ZINC000147421514 FJ On-Demand Anodyne KCNA5 23 49 Cc1cc(C)n([C@@H](C)C(=O)N2CCC[C@@H]2c2ccc(Cl)c(Cl)c2)n1 ZINC000147421514 FJ On-Demand Anodyne ADAM17 45 38 O=C(Cc1cccs1)NCC1(C(=O)O)CCC1 ZINC000147421521 CD On-Demand Anodyne CA5B 35 44 O=C(Cc1cccs1)NCC1(C(=O)O)CCC1 ZINC000147421521 CD On-Demand Anodyne CA5A 34 44 Cc1nn(C(F)F)c(C)c1CC(=O)N[C@@H](C)c1cnn(C)c1C ZINC000147421522 EE On-Demand Anodyne P2RX7 27 41 FC(F)CNCc1ccc2ccccc2n1 ZINC000147421523 BF For-Sale Anodyne CYSLTR1 26 43 CC[C@H](CC(=O)O)CN1C(=O)C[C@H](c2ccccc2)C1=O ZINC000147421545 CE For-Sale Anodyne HSD17B2 42 32 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne HTR4 40 36 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne EDNRB 50 38 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne EDNRA 48 39 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne BMP1 68 44 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne NOS2 95 36 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne EPHX2 17 41 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne PKM 36 47 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne TGM2 68 44 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne MCHR1 24 47 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne CACNA1I 50 39 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne F13A1 66 44 O=C(Cc1ccc2c(c1)OCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147421604 HE On-Demand Anodyne NAMPT 44 38 Cc1ccc(Br)c(C(=O)Nc2ccc3cn[nH]c3c2)c1 ZINC000147421665 EH On-Demand Anodyne MAOB 18 43 Cc1ccc(Br)c(C(=O)Nc2ccc3cn[nH]c3c2)c1 ZINC000147421665 EH On-Demand Anodyne ROCK1 22 41 Cc1ccc(Br)c(C(=O)Nc2ccc3cn[nH]c3c2)c1 ZINC000147421665 EH On-Demand Anodyne PHLPP2 0 51 Cc1ccc(Br)c(C(=O)Nc2ccc3cn[nH]c3c2)c1 ZINC000147421665 EH On-Demand Anodyne KCNK3 49 33 CCCCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147421669 DH On-Demand Anodyne PPARA 35 46 CCCCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147421669 DH On-Demand Anodyne CACNA1I 42 33 CCc1nc(CN(C)C(=O)NCC2(c3ccccc3)CCCC2)cs1 ZINC000147421684 FI On-Demand Anodyne KCNA3 41 36 Cc1nn(C(F)F)c(C)c1CC(=O)N[C@H](C)c1cnn(C)c1C ZINC000147421718 EE On-Demand Anodyne P2RX7 27 41 COc1ccc(CC(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147421720 EG For-Sale Reactive FKBP1A 17 40 COc1ccc(CC(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147421720 EG For-Sale Reactive OPRK1 30 48 COc1ccc(CC(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147421720 EG For-Sale Reactive DPP4 17 45 COc1ccc(CC(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147421720 EG For-Sale Reactive FAP 0 45 Cc1cc(C)n([C@H](C)C(=O)N2CCC[C@@H]2c2ccc(Cl)c(Cl)c2)n1 ZINC000147421736 FJ On-Demand Anodyne KCNA5 23 49 Cc1cc(C)n([C@H](C)C(=O)N2CCC[C@@H]2c2ccc(Cl)c(Cl)c2)n1 ZINC000147421736 FJ On-Demand Anodyne ADAM17 45 38 CC[C@@H](CC(=O)O)CN1C(=O)C[C@@H](c2ccccc2)C1=O ZINC000147421767 CE For-Sale Anodyne HSD17B2 42 32 COc1ccc2c(O)c(C(C)=O)cnc2c1 ZINC000147421770 BE In-Stock Anodyne KDR 47 39 COc1ccc2c(O)c(C(C)=O)cnc2c1 ZINC000147421770 BE In-Stock Anodyne PDGFRA 45 38 COc1ccc2c(O)c(C(C)=O)cnc2c1 ZINC000147421770 BE In-Stock Anodyne CSF1R 47 43 CC1(C)Oc2ccc(NC(=O)NC[C@@H]3CCCO[C@@H]3c3ccccc3)cc2O1 ZINC000147421771 GI On-Demand Anodyne PRMT3 45 33 NC(=O)c1cc(-c2csc(NC(=O)c3ccc4[nH]c5c(c4c3)CCCC5)n2)c[nH]1 ZINC000147421816 HH On-Demand Anodyne MAPKAPK2 19 46 CCCc1c(NCC)ncnc1Oc1ccc(Br)cc1Cl ZINC000147421841 FK For-Sale Anodyne PDE6A 42 33 CCCc1c(NCC)ncnc1Oc1ccc(Br)cc1Cl ZINC000147421841 FK For-Sale Anodyne HTT 0 40 O=C(Nc1ccc2[nH]ncc2c1)c1ccc(Br)c(Cl)c1 ZINC000147421849 FI On-Demand Anodyne MAOB 33 74 O=C(Nc1ccc2[nH]ncc2c1)c1ccc(Br)c(Cl)c1 ZINC000147421849 FI On-Demand Anodyne ROCK1 24 49 O=C(Nc1ccc2[nH]ncc2c1)c1ccc(Br)c(Cl)c1 ZINC000147421849 FI On-Demand Anodyne ROCK2 23 45 O=C(Nc1ccc2[nH]ncc2c1)c1ccc(Br)c(Cl)c1 ZINC000147421849 FI On-Demand Anodyne CSF1R 21 42 O=C(Nc1ccc2[nH]ncc2c1)c1ccc(Br)c(Cl)c1 ZINC000147421849 FI On-Demand Anodyne TAAR1 15 43 O=C(Nc1ccc2[nH]ncc2c1)c1ccc(Br)c(Cl)c1 ZINC000147421849 FI On-Demand Anodyne PTPA 0 40 O=C(Nc1ccc2[nH]ncc2c1)c1ccc(Br)c(Cl)c1 ZINC000147421849 FI On-Demand Anodyne NR2E3 62 37 O=C(Nc1ccc2[nH]ncc2c1)c1ccc(Br)c(Cl)c1 ZINC000147421849 FI On-Demand Anodyne SHH 41 38 COc1ccc(CC(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147421898 EG For-Sale Reactive FKBP1A 17 40 COc1ccc(CC(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147421898 EG For-Sale Reactive OPRK1 30 48 COc1ccc(CC(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147421898 EG For-Sale Reactive DPP4 17 45 COc1ccc(CC(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147421898 EG For-Sale Reactive FAP 0 45 C[C@H](C(=O)Nc1ccccc1)c1cccs1 ZINC000147421932 BG On-Demand Anodyne EPHX1 0 42 C[C@H](C(=O)Nc1ccccc1)c1cccs1 ZINC000147421932 BG On-Demand Anodyne P95276_MYCTO 0 42 C[C@H](C(=O)Nc1ccccc1)c1cccs1 ZINC000147421932 BG On-Demand Anodyne KCNK9 19 40 CC[C@H](CC(=O)O)CN1C(=O)C[C@@H](c2ccccc2)C1=O ZINC000147421959 CE For-Sale Anodyne HSD17B2 42 32 Cc1cc(C)n([C@@H](C)C(=O)N2CCC[C@H]2c2ccc(Cl)c(Cl)c2)n1 ZINC000147421961 FJ On-Demand Anodyne KCNA5 23 49 Cc1cc(C)n([C@@H](C)C(=O)N2CCC[C@H]2c2ccc(Cl)c(Cl)c2)n1 ZINC000147421961 FJ On-Demand Anodyne ADAM17 45 38 CC(=O)Nc1cccc(C2CCN(CCCN)CC2)c1 ZINC000147421963 CE For-Sale Anodyne SCN9A 23 46 CC1(C)Oc2ccc(NC(=O)NC[C@H]3CCCO[C@@H]3c3ccccc3)cc2O1 ZINC000147422027 GI On-Demand Anodyne PRMT3 45 33 O=C(CCc1ccccc1)NCC1(C(=O)O)CCC1 ZINC000147422040 CD On-Demand Anodyne NPFFR2 33 40 O=C(CCc1ccccc1)NCC1(C(=O)O)CCC1 ZINC000147422040 CD On-Demand Anodyne NPFFR1 48 38 CC(C)CCCCNCc1cc(Br)c(Br)o1 ZINC000147422049 FJ For-Sale Anodyne LEF 47 31 Cc1cc(C)n([C@H](C)C(=O)N2CCC[C@H]2c2ccc(Cl)c(Cl)c2)n1 ZINC000147422086 FJ On-Demand Anodyne KCNA5 23 49 Cc1cc(C)n([C@H](C)C(=O)N2CCC[C@H]2c2ccc(Cl)c(Cl)c2)n1 ZINC000147422086 FJ On-Demand Anodyne ADAM17 45 38 C[C@@H](C(=O)Nc1ccccc1)c1cccs1 ZINC000147422132 BG On-Demand Anodyne EPHX1 0 42 C[C@@H](C(=O)Nc1ccccc1)c1cccs1 ZINC000147422132 BG On-Demand Anodyne P95276_MYCTO 0 42 C[C@@H](C(=O)Nc1ccccc1)c1cccs1 ZINC000147422132 BG On-Demand Anodyne KCNK9 19 40 CC[C@@H]1CN([C@@H]2CCCCC[C@@H]2O)CC[C@@H]1N ZINC000147422159 BD For-Sale Anodyne VACHT_TETCF 0 40 CC[C@@H]1CN([C@@H]2CCCCC[C@@H]2O)CC[C@@H]1N ZINC000147422159 BD For-Sale Anodyne SLC18A3 30 49 CN(Cc1cscn1)C(=O)N[C@@H](c1ccccc1)C1CC1 ZINC000147422160 DG On-Demand Anodyne CYP3A4 18 44 O=C(c1cc2ccccc2s1)N1CCC[C@@H]1CCCBr ZINC000147422184 FJ For-Sale Reactive HCRTR1 17 41 CC1(C)Oc2ccc(NC(=O)NC[C@@H]3CCCO[C@H]3c3ccccc3)cc2O1 ZINC000147422212 GI On-Demand Anodyne PRMT3 45 33 CNc1cn2ccnc2c(Oc2ccc(Br)cc2Cl)n1 ZINC000147422255 FH For-Sale Anodyne HIVRT 0 47 COC(=O)CNC(=O)c1ccc(NC(=O)c2cc(C)cc([N+](=O)[O-])c2)cc1 ZINC000147422274 FE On-Demand Bother KCNK3 58 36 CC[C@H]1CN([C@@H]2CCCCC[C@@H]2O)CC[C@@H]1N ZINC000147422300 BD For-Sale Anodyne VACHT_TETCF 0 40 CC[C@H]1CN([C@@H]2CCCCC[C@@H]2O)CC[C@@H]1N ZINC000147422300 BD For-Sale Anodyne SLC18A3 30 49 O=C(Cc1ccccc1Cl)NCC1(C(=O)O)CCC1 ZINC000147422310 CE On-Demand Anodyne P2RX7 23 42 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)C(=O)NCc1ccccc1 ZINC000147422331 FG On-Demand Anodyne ANPEP 22 43 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)C(=O)NCc1ccccc1 ZINC000147422331 FG On-Demand Anodyne MDM2 70 34 C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)C(=O)NCc1ccccc1 ZINC000147422331 FG On-Demand Anodyne PDS 57 41 CN(Cc1cscn1)C(=O)N[C@H](c1ccccc1)C1CC1 ZINC000147422385 DG On-Demand Anodyne CYP3A4 18 44 O=C(c1cc2ccccc2s1)N1CCC[C@H]1CCCBr ZINC000147422405 FJ For-Sale Reactive HCRTR1 17 41 CC1(C)Oc2ccc(NC(=O)NC[C@H]3CCCO[C@H]3c3ccccc3)cc2O1 ZINC000147422429 GI On-Demand Anodyne PRMT3 45 33 COC(=O)c1ccc(N[C@@H](CC(C)C)C(=O)OC)nc1C ZINC000147422458 CE For-Sale Anodyne FOLH1 41 34 CS(=O)(=O)c1ccc(N)c(S(=O)(=O)NCCNC(N)=O)c1 ZINC000147422533 EA For-Sale Anodyne MAPK8 25 44 CCSc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccn1 ZINC000147422567 HG On-Demand Anodyne EPHX2 18 40 CCSc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccn1 ZINC000147422567 HG On-Demand Anodyne TGM2 46 39 CCSc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccn1 ZINC000147422567 HG On-Demand Anodyne CACNA1I 63 40 CCSc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccn1 ZINC000147422567 HG On-Demand Anodyne NAMPT 42 40 O=C(O)c1ccccc1Nc1ccc(Cl)cc1/N=C/c1ccc(Cl)nc1 ZINC000147422591 GK For-Sale Anodyne AKR1C3 21 46 O=C(O)c1ccccc1Nc1ccc(Cl)cc1/N=C/c1ccc(Cl)nc1 ZINC000147422591 GK For-Sale Anodyne AKR1C2 52 46 CCOc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147422625 DG On-Demand Anodyne ACACA 27 47 CCOc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147422625 DG On-Demand Anodyne ACACB 31 49 CCOc1ccc([C@@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147422625 DG On-Demand Anodyne CYP3A4 15 44 CCO[C@@H]1CCCN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147422664 FE On-Demand Anodyne PIK3CA 27 43 CCO[C@@H]1CCCN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147422664 FE On-Demand Anodyne MTOR 56 43 CCO[C@@H]1CCCN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147422664 FE On-Demand Anodyne EPHX2 50 48 CCO[C@@H]1CCCN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147422664 FE On-Demand Anodyne PIK3CG 25 43 CCO[C@@H]1CCCN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147422664 FE On-Demand Anodyne L3MBTL3 57 37 COC(=O)c1ccc(N[C@H](CC(C)C)C(=O)OC)nc1C ZINC000147422672 CE For-Sale Anodyne FOLH1 41 34 CC(C)(c1ccccc1)N1CCC(N)CC1 ZINC000147422685 BE For-Sale Anodyne CHRM3 18 43 CCCNc1cc(Oc2ccc(Br)cc2Cl)nc(N)n1 ZINC000147422705 FI For-Sale Anodyne AGPAT2 67 47 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)C(=O)NCc1ccccc1 ZINC000147422740 FG On-Demand Anodyne ANPEP 22 43 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)C(=O)NCc1ccccc1 ZINC000147422740 FG On-Demand Anodyne MDM2 70 34 C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)C(=O)NCc1ccccc1 ZINC000147422740 FG On-Demand Anodyne PDS 57 41 Oc1ccc(CNCC(F)F)cc1Cl ZINC000147422750 BE For-Sale Anodyne NCE103 29 44 Oc1ccc(CNCC(F)F)cc1Cl ZINC000147422750 BE For-Sale Anodyne CAN2 0 45 CC(C)CO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147422799 GE On-Demand Anodyne CHRM5 22 44 CC(C)CO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147422799 GE On-Demand Anodyne MMP2 18 42 CC(C)CO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147422799 GE On-Demand Anodyne EPHX2 22 44 CC(C)CO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147422799 GE On-Demand Anodyne TGM2 65 45 CC(C)CO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147422799 GE On-Demand Anodyne F13A1 65 45 N#Cc1cccc(S(=O)(=O)CCN2CCC[C@@H]2CO)c1 ZINC000147422805 CC On-Demand Mild CHRNA10 35 47 O=C(NCC1(C(=O)O)CCC1)c1cc(Cl)ccc1F ZINC000147422813 CE On-Demand Anodyne P2RX7 0 46 CCOc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147422837 DG On-Demand Anodyne ACACA 27 47 CCOc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147422837 DG On-Demand Anodyne ACACB 31 49 CCOc1ccc([C@H](C)NC(=O)N(C)Cc2cscn2)cc1 ZINC000147422837 DG On-Demand Anodyne CYP3A4 15 44 COC(=O)c1ccc(N[C@@H](CC(C)C)C(=O)O)nc1C ZINC000147422878 CE On-Demand Anodyne FOLH1 52 36 COC(=O)c1ccc(N[C@@H](CC(C)C)C(=O)O)nc1C ZINC000147422878 CE On-Demand Anodyne FPR1 42 35 CCO[C@H]1CCCN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147422899 FE On-Demand Anodyne PIK3CA 27 43 CCO[C@H]1CCCN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147422899 FE On-Demand Anodyne MTOR 56 43 CCO[C@H]1CCCN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147422899 FE On-Demand Anodyne EPHX2 50 48 CCO[C@H]1CCCN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147422899 FE On-Demand Anodyne PIK3CG 25 43 CCO[C@H]1CCCN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147422899 FE On-Demand Anodyne L3MBTL3 57 37 CC(C)CO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423030 GE On-Demand Anodyne CHRM5 22 44 CC(C)CO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423030 GE On-Demand Anodyne MMP2 18 42 CC(C)CO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423030 GE On-Demand Anodyne EPHX2 22 44 CC(C)CO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423030 GE On-Demand Anodyne TGM2 65 45 CC(C)CO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423030 GE On-Demand Anodyne F13A1 65 45 COC(=O)c1ccc(N[C@H](CC(C)C)C(=O)O)nc1C ZINC000147423091 CE On-Demand Anodyne FOLH1 52 36 COC(=O)c1ccc(N[C@H](CC(C)C)C(=O)O)nc1C ZINC000147423091 CE On-Demand Anodyne FPR1 42 35 CN(Cc1ccccc1)C(=O)CNC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147423092 HD On-Demand Bother LIMK2 46 42 O=C(O)c1cccc(-c2nc(-c3cncs3)no2)c1 ZINC000147423103 CF For-Sale Anodyne S1PR1 33 40 O=C(O)c1cccc(-c2nc(-c3cncs3)no2)c1 ZINC000147423103 CF For-Sale Anodyne PLCG2 0 40 O=C(O)c1cccc(-c2nc(-c3cncs3)no2)c1 ZINC000147423103 CF For-Sale Anodyne CD38 74 34 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423126 FJ On-Demand Anodyne EPHX2 18 40 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423126 FJ On-Demand Anodyne ENV 48 37 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423126 FJ On-Demand Anodyne PRMT3 46 34 CC(C)Oc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147423180 FI For-Sale Reactive PREP 48 45 CC(C)Oc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147423180 FI For-Sale Reactive CFTR 43 40 CC(C)Oc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147423180 FI For-Sale Reactive FAP 0 42 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423209 FE On-Demand Anodyne MTNR1A 54 40 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423209 FE On-Demand Anodyne MTNR1B 45 38 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423209 FE On-Demand Anodyne ADAM9 40 35 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423209 FE On-Demand Anodyne PSMB8 51 38 C[C@@H]1CCCN(CCS(=O)(=O)c2cccc(C#N)c2)CC1 ZINC000147423221 DE On-Demand Mild CHRNA10 29 44 CN(C)Cc1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147423246 FI On-Demand Anodyne KLKB1 27 43 CN(C)Cc1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147423246 FI On-Demand Anodyne PDGFRA 0 42 CN(C)Cc1ccc(NC(=O)c2ccc(Br)c(Cl)c2)cc1 ZINC000147423246 FI On-Demand Anodyne TAAR1 20 46 COc1cccc(CCNC(=O)COc2ccc(C(N)=O)cc2)c1OC ZINC000147423254 FD On-Demand Anodyne NQO2 45 44 COc1cccc(CCNC(=O)COc2ccc(C(N)=O)cc2)c1OC ZINC000147423254 FD On-Demand Anodyne MTNR1A 90 48 COc1cccc(CCNC(=O)COc2ccc(C(N)=O)cc2)c1OC ZINC000147423254 FD On-Demand Anodyne MTNR1B 67 44 COC[C@H](C)N(C)C(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147423261 EF For-Sale Anodyne NPY5R 32 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1cc(C)sc1C ZINC000147423265 DF On-Demand Anodyne PCSK5 51 33 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1cc(C)sc1C ZINC000147423265 DF On-Demand Anodyne NOD1 46 33 CC(=O)NCC(=O)NCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423302 HB On-Demand Anodyne HTR4 45 33 CC(=O)NCC(=O)NCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423302 HB On-Demand Anodyne EPHX2 26 45 CC(=O)NCC(=O)NCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423302 HB On-Demand Anodyne TGM2 76 46 CC(=O)NCC(=O)NCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423302 HB On-Demand Anodyne CACNA1I 49 36 CC(=O)NCC(=O)NCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423302 HB On-Demand Anodyne F13A1 82 46 CN(C(=O)c1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1)c1ccccc1 ZINC000147423331 HJ On-Demand Anodyne MAPK10 17 43 CN(C(=O)c1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1)c1ccccc1 ZINC000147423331 HJ On-Demand Anodyne KCNK3 82 44 CN(C(=O)c1cccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1)c1ccccc1 ZINC000147423331 HJ On-Demand Anodyne KCNK9 40 39 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423332 FJ On-Demand Anodyne EPHX2 18 40 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423332 FJ On-Demand Anodyne ENV 48 37 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423332 FJ On-Demand Anodyne PRMT3 46 34 CC(C)Oc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147423398 FI For-Sale Reactive PREP 48 45 CC(C)Oc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147423398 FI For-Sale Reactive CFTR 43 40 CC(C)Oc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147423398 FI For-Sale Reactive FAP 0 42 CC[C@@H]1CN(Cc2nc3ccccc3c(=O)[nH]2)CC[C@@H]1N ZINC000147423401 CD On-Demand Anodyne PARP1 24 48 CC[C@@H]1CN(Cc2nc3ccccc3c(=O)[nH]2)CC[C@@H]1N ZINC000147423401 CD On-Demand Anodyne PDE9A 0 41 COc1ccc2c(c1)OC[C@H](C(=O)N[C@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423408 FE On-Demand Anodyne MTNR1A 54 40 COc1ccc2c(c1)OC[C@H](C(=O)N[C@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423408 FE On-Demand Anodyne MTNR1B 45 38 COc1ccc2c(c1)OC[C@H](C(=O)N[C@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423408 FE On-Demand Anodyne ADAM9 40 35 COc1ccc2c(c1)OC[C@H](C(=O)N[C@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423408 FE On-Demand Anodyne PSMB8 51 38 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(C(=O)C23CC4CC(CC(C4)C2)C3)CC1 ZINC000147423440 HH On-Demand Anodyne MC4R 34 41 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(C(=O)C23CC4CC(CC(C4)C2)C3)CC1 ZINC000147423440 HH On-Demand Anodyne TRY2_BOVIN 96 37 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(C(=O)C23CC4CC(CC(C4)C2)C3)CC1 ZINC000147423440 HH On-Demand Anodyne CCR1 18 43 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCN(C(=O)C23CC4CC(CC(C4)C2)C3)CC1 ZINC000147423440 HH On-Demand Anodyne ST14 57 36 C[C@H]1CCCN(CCS(=O)(=O)c2cccc(C#N)c2)CC1 ZINC000147423442 DE On-Demand Mild CHRNA10 29 44 Cc1c(C)n(CCNC(=O)N(C)C)c2ncnc(N)c12 ZINC000147423446 CC For-Sale Anodyne OXGR1 51 32 C[C@H](N)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147423451 BC For-Sale Anodyne ACE 17 40 C[C@H](N)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147423451 BC For-Sale Anodyne TPP2 53 36 COC[C@@H](C)N(C)C(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147423458 EF For-Sale Anodyne NPY5R 32 40 Cc1ccc(Br)c(C(=O)Nc2ccc(CN(C)C)cc2)c1 ZINC000147423474 EI On-Demand Anodyne KCNK3 53 33 Cc1ccc(Br)c(C(=O)Nc2ccc(CN(C)C)cc2)c1 ZINC000147423474 EI On-Demand Anodyne KCNK9 44 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1cc(C)sc1C ZINC000147423481 DF On-Demand Anodyne PCSK5 51 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1cc(C)sc1C ZINC000147423481 DF On-Demand Anodyne NOD1 46 33 CCOC(=O)[C@@H]1CC[C@@H](Oc2ccc(-c3ccc(C=O)cn3)cn2)CC1 ZINC000147423557 FG For-Sale Anodyne DGAT1 37 48 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423561 FJ On-Demand Anodyne EPHX2 18 40 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423561 FJ On-Demand Anodyne ENV 48 37 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423561 FJ On-Demand Anodyne PRMT3 46 34 Cc1ccc(C(=O)NCC2(C(=O)O)CCC2)cc1Cl ZINC000147423567 CF On-Demand Anodyne DRD4 40 32 Cc1cnn(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147423573 GD On-Demand Anodyne EPHX2 30 40 Cc1cnn(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147423573 GD On-Demand Anodyne TGM2 66 43 Cc1cnn(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147423573 GD On-Demand Anodyne CACNA1I 47 35 Cc1cnn(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147423573 GD On-Demand Anodyne F13A1 65 43 Cc1cnn(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147423573 GD On-Demand Anodyne NAMPT 40 38 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423608 FE On-Demand Anodyne MTNR1A 54 40 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423608 FE On-Demand Anodyne MTNR1B 45 38 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423608 FE On-Demand Anodyne ADAM9 40 35 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423608 FE On-Demand Anodyne PSMB8 51 38 CC[C@H]1CN(Cc2nc3ccccc3c(=O)[nH]2)CC[C@@H]1N ZINC000147423609 CD On-Demand Anodyne PARP1 24 48 CC[C@H]1CN(Cc2nc3ccccc3c(=O)[nH]2)CC[C@@H]1N ZINC000147423609 CD On-Demand Anodyne PDE9A 0 41 C[C@H](Cc1cccc(F)c1)C(=O)N1CCN(C(=O)C23CC4CC(CC(C4)C2)C3)CC1 ZINC000147423654 HH On-Demand Anodyne MC4R 34 41 C[C@H](Cc1cccc(F)c1)C(=O)N1CCN(C(=O)C23CC4CC(CC(C4)C2)C3)CC1 ZINC000147423654 HH On-Demand Anodyne TRY2_BOVIN 96 37 C[C@H](Cc1cccc(F)c1)C(=O)N1CCN(C(=O)C23CC4CC(CC(C4)C2)C3)CC1 ZINC000147423654 HH On-Demand Anodyne CCR1 18 43 C[C@H](Cc1cccc(F)c1)C(=O)N1CCN(C(=O)C23CC4CC(CC(C4)C2)C3)CC1 ZINC000147423654 HH On-Demand Anodyne ST14 57 36 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1cc(C)sc1C ZINC000147423660 DF On-Demand Anodyne PCSK5 51 33 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1cc(C)sc1C ZINC000147423660 DF On-Demand Anodyne NOD1 46 33 C[C@@H](N)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147423672 BC For-Sale Anodyne ACE 17 40 C[C@@H](N)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147423672 BC For-Sale Anodyne TPP2 53 36 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423734 FJ On-Demand Anodyne EPHX2 18 40 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423734 FJ On-Demand Anodyne ENV 48 37 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1ccc(Cl)c(F)c1 ZINC000147423734 FJ On-Demand Anodyne PRMT3 46 34 CCOCCO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423775 GD On-Demand Anodyne CHRM5 21 41 CCOCCO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423775 GD On-Demand Anodyne MMP13 15 41 CCOCCO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423775 GD On-Demand Anodyne TGM2 55 42 CCOCCO[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147423775 GD On-Demand Anodyne F13A1 53 42 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423802 FE On-Demand Anodyne MTNR1A 54 40 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423802 FE On-Demand Anodyne MTNR1B 45 38 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423802 FE On-Demand Anodyne ADAM9 40 35 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@H](C)C(=O)NCc1ccccc1)C2 ZINC000147423802 FE On-Demand Anodyne PSMB8 51 38 Fc1ccc(NCc2ccn(C3CCCC3)n2)cc1Cl ZINC000147423826 CI On-Demand Anodyne MAP3K8 108 44 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1cc(C)sc1C ZINC000147423838 DF On-Demand Anodyne PCSK5 51 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1cc(C)sc1C ZINC000147423838 DF On-Demand Anodyne NOD1 46 33 C[C@H](N)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147423880 BC For-Sale Anodyne ACE 17 40 C[C@H](N)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147423880 BC For-Sale Anodyne TPP2 53 36 CC[C@@H]1CN(CC(=O)Nc2ccc(C)cc2)CC[C@@H]1N ZINC000147423975 CD On-Demand Anodyne DRD4 0 47 CCOCCO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147424005 GD On-Demand Anodyne CHRM5 21 41 CCOCCO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147424005 GD On-Demand Anodyne MMP13 15 41 CCOCCO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147424005 GD On-Demand Anodyne TGM2 55 42 CCOCCO[C@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147424005 GD On-Demand Anodyne F13A1 53 42 C[C@@H](NC(=O)c1ccc2c(c1)COC2)C(=O)NCc1ccccc1 ZINC000147424018 DE On-Demand Anodyne MME 40 36 C[C@@H](NC(=O)c1ccc2c(c1)COC2)C(=O)NCc1ccccc1 ZINC000147424018 DE On-Demand Anodyne CTSB 18 42 C[C@@H](NC(=O)c1ccc2c(c1)COC2)C(=O)NCc1ccccc1 ZINC000147424018 DE On-Demand Anodyne FURIN 45 35 C[C@@H](NC(=O)c1ccc2c(c1)COC2)C(=O)NCc1ccccc1 ZINC000147424018 DE On-Demand Anodyne CAPN2 15 44 C[C@@H](NC(=O)c1ccc2c(c1)COC2)C(=O)NCc1ccccc1 ZINC000147424018 DE On-Demand Anodyne PROC 46 38 C[C@@H](NC(=O)c1ccc2c(c1)COC2)C(=O)NCc1ccccc1 ZINC000147424018 DE On-Demand Anodyne AMP1_PLAFQ 46 40 COCC[C@H](Nc1ccc(C(=O)OC)c(C)n1)C(=O)O ZINC000147424023 CD For-Sale Anodyne NPPA 45 38 CCCCCCCCOCCOCCOCCOCCOCCOCCOCCOCCOCCO ZINC000147424031 KE For-Sale Mild UGCG 15 41 CCCCCCCCOCCOCCOCCOCCOCCOCCOCCOCCOCCO ZINC000147424031 KE For-Sale Mild GBA 15 41 CCCCCCCCOCCOCCOCCOCCOCCOCCOCCOCCOCCO ZINC000147424031 KE For-Sale Mild GBA2 32 41 CCCCCCCCOCCOCCOCCOCCOCCOCCOCCOCCOCCO ZINC000147424031 KE For-Sale Mild LPAR3 18 41 CN(C)C(=O)NCCn1c(N)cc2ccccc2c1=O ZINC000147424102 CC For-Sale Anodyne POLR1A 60 34 C[C@@H](N)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147424104 BC For-Sale Anodyne ACE 17 40 C[C@@H](N)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147424104 BC For-Sale Anodyne TPP2 53 36 COCCN(C(=O)Nc1cc(Br)cc(C(=O)O)c1)C1CC1 ZINC000147424110 FF For-Sale Anodyne PPARA 26 41 CC(C)c1c(Br)cccc1[N+](=O)[O-] ZINC000147424168 BG For-Sale Anodyne COLA 91 36 CCOC[C@H](C)NC(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147424203 EG On-Demand Anodyne PPIA 26 40 CCOC[C@H](C)NC(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147424203 EG On-Demand Anodyne CCKAR 39 40 CCOC[C@H](C)NC(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147424203 EG On-Demand Anodyne F2R 16 45 CCOC[C@H](C)NC(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147424203 EG On-Demand Anodyne PRNP 52 43 CCOC[C@H](C)NC(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147424203 EG On-Demand Anodyne CCKBR 29 40 CCOC[C@H](C)NC(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147424203 EG On-Demand Anodyne KCNK3 109 50 CCOC[C@H](C)NC(=O)Nc1cccc(NC(=O)c2ccccc2)c1 ZINC000147424203 EG On-Demand Anodyne KCNK9 97 50 CC[C@H]1CN(CC(=O)Nc2ccc(C)cc2)CC[C@@H]1N ZINC000147424205 CD On-Demand Anodyne DRD4 0 47 COCC[C@@H](Nc1ccc(C(=O)OC)c(C)n1)C(=O)O ZINC000147424238 CD For-Sale Anodyne NPPA 45 38 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147424248 HH On-Demand Anodyne SLC6A3 26 41 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147424248 HH On-Demand Anodyne CHRM5 20 41 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147424248 HH On-Demand Anodyne EPHX2 19 40 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147424248 HH On-Demand Anodyne TGM2 62 42 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(F)cc1 ZINC000147424248 HH On-Demand Anodyne F13A1 60 42 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne CA2 15 43 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne ADRB3 49 39 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne CA1 15 43 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne CTSB 23 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne TRY2_BOVIN 61 34 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne CYSP_TRYCR 19 43 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne CTSK 26 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne CTSL 30 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne MMP2 23 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne MMP3 32 40 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne CCKBR 44 37 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne CTSS 24 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne CAPN1 22 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne MTNN 63 38 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne AKR1C3 17 50 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne LIMK2 54 43 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@@H](C)CCc3ccccc3)c2)cc1 ZINC000147424291 HJ In-Stock Anodyne KCNK3 43 34 COCCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147424329 DF For-Sale Anodyne GCGR 15 48 COCCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147424329 DF For-Sale Anodyne CACNA1I 54 37 COCCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147424329 DF For-Sale Anodyne GIPR 46 37 CNc1ccc(C(=O)NCC2(N(C)C)CCCC2)cc1C ZINC000147424341 CF For-Sale Anodyne SLC6A5 17 47 CS(=O)(=O)c1ccc(-c2cc3nccc(Oc4ccc([N+](=O)[O-])cc4F)c3s2)cc1 ZINC000147424355 IK For-Sale Bother MST1R 54 39 CS(=O)(=O)c1ccc(-c2cc3nccc(Oc4ccc([N+](=O)[O-])cc4F)c3s2)cc1 ZINC000147424355 IK For-Sale Bother MET 42 41 Cl[C@@H]1CCN2Cc3ccccc3N=C12 ZINC000147424401 BF For-Sale Reactive CCR3 0 41 O=S(=O)(c1ccc(Cl)c(Cl)c1)N1CCN(CCBr)CC1 ZINC000147424406 HF For-Sale Reactive ADORA2B 48 35 O=S(=O)(c1ccc(Cl)c(Cl)c1)N1CCN(CCBr)CC1 ZINC000147424406 HF For-Sale Reactive SIGMAR1 15 44 O=S(=O)(c1ccc(Cl)c(Cl)c1)N1CCN(CCBr)CC1 ZINC000147424406 HF For-Sale Reactive PKM 42 42 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424471 HE On-Demand Anodyne LPL 55 38 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424471 HE On-Demand Anodyne CCKAR 32 41 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424471 HE On-Demand Anodyne CCR3 44 39 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424471 HE On-Demand Anodyne PRNP 46 39 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424471 HE On-Demand Anodyne CCKBR 56 39 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424471 HE On-Demand Anodyne EPHX2 55 46 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424471 HE On-Demand Anodyne SMO 17 46 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424471 HE On-Demand Anodyne KCNK3 123 48 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424471 HE On-Demand Anodyne KCNK9 73 44 CCNC(=O)c1ccc(C)c(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)c1 ZINC000147424489 HE On-Demand Anodyne MAPK14 30 40 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne CA2 15 43 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne ADRB3 49 39 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne CA1 15 43 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne CTSB 23 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne TRY2_BOVIN 61 34 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne CYSP_TRYCR 19 43 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne CTSK 26 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne CTSL 30 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne MMP2 23 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne MMP3 32 40 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne CCKBR 44 37 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne CTSS 24 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne CAPN1 22 41 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne MTNN 63 38 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne AKR1C3 17 50 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne LIMK2 54 43 Cc1ccc(NS(=O)(=O)c2cccc(C(=O)N[C@H](C)CCc3ccccc3)c2)cc1 ZINC000147424491 HJ In-Stock Anodyne KCNK3 43 34 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1 ZINC000147424528 GF On-Demand Anodyne HTR4 63 41 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1 ZINC000147424528 GF On-Demand Anodyne CHRM5 19 40 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1 ZINC000147424528 GF On-Demand Anodyne ACACB 25 40 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1 ZINC000147424528 GF On-Demand Anodyne SLC6A9 48 38 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1 ZINC000147424528 GF On-Demand Anodyne EPHX2 32 40 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1 ZINC000147424528 GF On-Demand Anodyne TGM2 63 43 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1 ZINC000147424528 GF On-Demand Anodyne CACNA1I 57 35 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1 ZINC000147424528 GF On-Demand Anodyne F13A1 58 43 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1 ZINC000147424528 GF On-Demand Anodyne NAMPT 42 38 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)N2C[C@H](C)O[C@H](C)C2)CC1 ZINC000147424549 HB On-Demand Anodyne P2RY12 42 32 CNc1ccc(Cl)cc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147424569 DF For-Sale Anodyne P2RX7 18 43 CNc1ccc(Cl)cc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147424569 DF For-Sale Anodyne SLC6A9 45 34 CNc1ccc(Cl)cc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147424569 DF For-Sale Anodyne SLC6A5 15 42 N#Cc1cccc(S(=O)(=O)CCN2CCC(C#N)CC2)c1 ZINC000147424622 DD On-Demand Mild MEN1 44 33 Cl[C@H]1CCN2Cc3ccccc3N=C12 ZINC000147424648 BF For-Sale Reactive CCR3 0 41 CCCNCCCCCCOc1ccc(Cl)c(F)c1 ZINC000147424662 CI For-Sale Anodyne DRD4 21 48 CCCNCCCCCCOc1ccc(Cl)c(F)c1 ZINC000147424662 CI For-Sale Anodyne PLA2G4B 44 33 CCNC(=O)c1ccc(C)c(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)c1 ZINC000147424694 HE On-Demand Anodyne MAPK14 30 40 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424698 HE On-Demand Anodyne LPL 55 38 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424698 HE On-Demand Anodyne CCKAR 32 41 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424698 HE On-Demand Anodyne CCR3 44 39 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424698 HE On-Demand Anodyne PRNP 46 39 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424698 HE On-Demand Anodyne CCKBR 56 39 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424698 HE On-Demand Anodyne EPHX2 55 46 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424698 HE On-Demand Anodyne SMO 17 46 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424698 HE On-Demand Anodyne KCNK3 123 48 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C1 ZINC000147424698 HE On-Demand Anodyne KCNK9 73 44 O=C(NCc1cccc(C(=O)NC[C@H]2CCCO2)c1)C(=O)Nc1c(F)cccc1F ZINC000147424714 HE On-Demand Anodyne TNK2 15 40 O=C(NCCn1cccn1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147424730 DE On-Demand Anodyne CACNA1H 24 40 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147424739 FD On-Demand Anodyne HTR4 56 39 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147424739 FD On-Demand Anodyne CHRM5 20 40 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147424739 FD On-Demand Anodyne GRIN2B 32 42 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147424739 FD On-Demand Anodyne TGM2 58 42 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147424739 FD On-Demand Anodyne CACNA1I 50 37 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147424739 FD On-Demand Anodyne F13A1 59 42 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147424739 FD On-Demand Anodyne NAMPT 40 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)N2C[C@H](C)O[C@H](C)C2)CC1 ZINC000147424772 HB On-Demand Anodyne P2RY12 42 32 CCOC(=O)CCCNC(=O)[C@]1(C)CCCS1 ZINC000147424773 CD For-Sale Anodyne EPHX2 25 44 CNc1ncccc1C(=O)Nc1cc(Cl)ccc1Br ZINC000147424816 EH For-Sale Anodyne F10 32 41 CNc1ncccc1C(=O)Nc1cc(Cl)ccc1Br ZINC000147424816 EH For-Sale Anodyne GRM4 46 41 CNc1ncccc1C(=O)Nc1cc(Cl)ccc1Br ZINC000147424816 EH For-Sale Anodyne KCNMA1 25 45 CNc1ncccc1C(=O)Nc1cc(Cl)ccc1Br ZINC000147424816 EH For-Sale Anodyne G2YM83_BOTF4 75 39 CN(C)C1(CNC(=O)c2nc(N)ccc2Cl)CCCC1 ZINC000147424817 CD For-Sale Anodyne SLC6A5 15 42 C[C@H](N)CC(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147424823 CD For-Sale Anodyne TPP2 50 31 CCNCc1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147424898 CI For-Sale Anodyne MCHR1 0 41 O=C(NCCn1ccnc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147424945 FE For-Sale Anodyne TBXAS1 51 42 O=C(NCCn1ccnc1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147424945 FE For-Sale Anodyne QPCT 36 48 N#Cc1cccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)c1 ZINC000147424956 HD On-Demand Mild CCR3 16 40 C[C@@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@H](c2ccccc2)O1 ZINC000147424971 HJ On-Demand Anodyne PRNP 31 40 C[C@@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@H](c2ccccc2)O1 ZINC000147424971 HJ On-Demand Anodyne KCNK3 134 47 C[C@@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@H](c2ccccc2)O1 ZINC000147424971 HJ On-Demand Anodyne KCNK9 86 46 CCOC(=O)CCCNC(=O)[C@@]1(C)CCCS1 ZINC000147424975 CD For-Sale Anodyne EPHX2 25 44 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)N2C[C@@H](C)O[C@H](C)C2)CC1 ZINC000147424998 HB On-Demand Anodyne P2RY12 42 32 O=C(CSCc1ccncc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147425004 HF On-Demand Anodyne GRIN2B 21 42 O=C(CSCc1ccncc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147425004 HF On-Demand Anodyne TGM2 76 46 O=C(CSCc1ccncc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147425004 HF On-Demand Anodyne F13A1 80 46 O=C(CSCc1ccncc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147425004 HF On-Demand Anodyne NAMPT 69 41 CC(C)CCCCNCc1ccc(F)cc1C(F)(F)F ZINC000147425038 CJ For-Sale Anodyne LEF 72 34 C[C@@H](N)CC(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147425054 CD For-Sale Anodyne TPP2 50 31 CN(C)C1(CNC(=O)c2cc(Br)cnc2N)CCCC1 ZINC000147425110 EE For-Sale Anodyne SLC6A5 15 43 O=C(NCCn1ccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147425152 DE On-Demand Anodyne CACNA1H 24 40 O=C(NCCn1ccnc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147425152 DE On-Demand Anodyne QPCT 36 48 C[C@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@H](c2ccccc2)O1 ZINC000147425173 HJ On-Demand Anodyne PRNP 31 40 C[C@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@H](c2ccccc2)O1 ZINC000147425173 HJ On-Demand Anodyne KCNK3 134 47 C[C@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@H](c2ccccc2)O1 ZINC000147425173 HJ On-Demand Anodyne KCNK9 86 46 Cc1ccc2nc(COc3cccc(C(=O)Nc4ncc(C)s4)c3)cn2c1 ZINC000147425190 GI On-Demand Anodyne MAP3K5 40 37 Cc1ccc2nc(COc3cccc(C(=O)Nc4ncc(C)s4)c3)cn2c1 ZINC000147425190 GI On-Demand Anodyne SCD1 25 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc2[nH]cnc12 ZINC000147425206 HF On-Demand Anodyne HTR4 58 54 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc2[nH]cnc12 ZINC000147425206 HF On-Demand Anodyne CACNA1I 59 33 COc1ccc2c(c1)OC[C@@H](C(=O)NNC(=O)Cc1ccccc1OC)C2 ZINC000147425245 FD On-Demand Reactive ADRA2C 50 34 COc1ccc2c(c1)OC[C@@H](C(=O)NNC(=O)Cc1ccccc1OC)C2 ZINC000147425245 FD On-Demand Reactive EDNRB 41 37 COc1ccc2c(c1)OC[C@@H](C(=O)NNC(=O)Cc1ccccc1OC)C2 ZINC000147425245 FD On-Demand Reactive MTNR1A 49 39 COc1ccc2c(c1)OC[C@@H](C(=O)NNC(=O)Cc1ccccc1OC)C2 ZINC000147425245 FD On-Demand Reactive MTNR1B 45 36 COc1ccc2c(c1)OC[C@@H](C(=O)NNC(=O)Cc1ccccc1OC)C2 ZINC000147425245 FD On-Demand Reactive ROCK2 30 43 CCNS(=O)(=O)c1ccc(NC[C@@H](C)CC(=O)O)cc1 ZINC000147425273 DD For-Sale Anodyne CA2 16 40 C[C@H](N)CC(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147425287 CD For-Sale Anodyne TPP2 50 31 CC(C)CCCCNC(=O)c1cc2ccccc2c(Cl)n1 ZINC000147425314 DI For-Sale Anodyne DRD3 25 40 CC(C)CCCCNC(=O)c1cc2ccccc2c(Cl)n1 ZINC000147425314 DI For-Sale Anodyne PLA2G7 24 45 CCCN(CC(C)C)C(=O)c1ccc(C(F)(F)F)cc1 ZINC000147425328 CI On-Demand Anodyne MTTP 22 40 CCCN(CC(C)C)C(=O)c1ccc(C(F)(F)F)cc1 ZINC000147425328 CI On-Demand Anodyne PLM2_PLAFA 30 45 CCCN(CC(C)C)C(=O)c1ccc(C(F)(F)F)cc1 ZINC000147425328 CI On-Demand Anodyne MCHR1 21 46 CCCN(CC(C)C)C(=O)c1ccc(C(F)(F)F)cc1 ZINC000147425328 CI On-Demand Anodyne MLYCD 44 62 COc1ccc(OC(F)F)c(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)c1 ZINC000147425335 HF On-Demand Anodyne RORC 43 39 O=C(O)C[C@@H](O)CS(=O)(=O)c1ccccc1 ZINC000147425341 BC For-Sale Anodyne HMGCR 17 45 O=C(O)C[C@@H](O)CS(=O)(=O)c1ccccc1 ZINC000147425341 BC For-Sale Anodyne MMP12 15 44 CNc1cccc(C(=O)NCC2(N(C)C)CCCC2)n1 ZINC000147425349 CD For-Sale Anodyne SLC6A5 15 43 CNc1cccc(C(=O)NCC2(N(C)C)CCCC2)n1 ZINC000147425349 CD For-Sale Anodyne HCN1 40 31 CN1CC[C@H](NC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147425356 ED For-Sale Anodyne EPHX2 40 43 CN1CC[C@H](NC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147425356 ED For-Sale Anodyne CXCR3 15 42 C[C@@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@@H](c2ccccc2)O1 ZINC000147425400 HJ On-Demand Anodyne PRNP 31 40 C[C@@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@@H](c2ccccc2)O1 ZINC000147425400 HJ On-Demand Anodyne KCNK3 134 47 C[C@@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@@H](c2ccccc2)O1 ZINC000147425400 HJ On-Demand Anodyne KCNK9 86 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cn[nH]n1 ZINC000147425472 EC In-Stock Anodyne GRIN2B 26 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cn[nH]n1 ZINC000147425472 EC In-Stock Anodyne TGM2 61 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cn[nH]n1 ZINC000147425472 EC In-Stock Anodyne CACNA1I 46 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cn[nH]n1 ZINC000147425472 EC In-Stock Anodyne F13A1 64 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cn[nH]n1 ZINC000147425472 EC In-Stock Anodyne NAMPT 45 42 C[C@@H](N)CC(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147425504 CD For-Sale Anodyne TPP2 50 31 CCNS(=O)(=O)c1ccc(NC[C@H](C)CC(=O)O)cc1 ZINC000147425513 DD For-Sale Anodyne CA2 16 40 FC(F)(F)c1ccc(CN2CC[C@H](Br)C2)cc1 ZINC000147425551 DH For-Sale Reactive DRD4 15 47 FC(F)(F)c1ccc(CN2CC[C@H](Br)C2)cc1 ZINC000147425551 DH For-Sale Reactive SIGMAR1 27 49 FC(F)(F)c1ccc(CN2CC[C@H](Br)C2)cc1 ZINC000147425551 DH For-Sale Reactive CCR2 16 42 FC(F)(F)c1ccc(CN2CC[C@H](Br)C2)cc1 ZINC000147425551 DH For-Sale Reactive SLC6A5 29 41 FC(F)(F)c1ccc(CN2CC[C@H](Br)C2)cc1 ZINC000147425551 DH For-Sale Reactive CACNA1G 25 40 O=C(O)C[C@H](O)CS(=O)(=O)c1ccccc1 ZINC000147425566 BC For-Sale Anodyne HMGCR 17 45 CNc1ccc(Cl)c(C(=O)NCC2(N(C)C)CCCC2)n1 ZINC000147425596 DE For-Sale Anodyne P2RX7 20 41 CN1CC[C@@H](NC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147425606 ED For-Sale Anodyne EPHX2 40 43 CN1CC[C@@H](NC(=O)Nc2cc(Br)cc(C(=O)O)c2)C1 ZINC000147425606 ED For-Sale Anodyne CXCR3 15 42 COc1ccc(OC(F)F)c(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)c1 ZINC000147425608 HF On-Demand Anodyne RORC 43 39 COc1ccc(NC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cn1 ZINC000147425616 GF On-Demand Anodyne MAP1 105 39 COc1ccc(NC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cn1 ZINC000147425616 GF On-Demand Anodyne GRM4 23 42 COc1ccc(NC(=O)c2ccc(S(=O)(=O)Nc3nccs3)cc2)cn1 ZINC000147425616 GF On-Demand Anodyne GCK 22 41 C[C@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@@H](c2ccccc2)O1 ZINC000147425624 HJ On-Demand Anodyne PRNP 31 40 C[C@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@@H](c2ccccc2)O1 ZINC000147425624 HJ On-Demand Anodyne KCNK3 134 47 C[C@H]1CN(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2)C[C@@H](c2ccccc2)O1 ZINC000147425624 HJ On-Demand Anodyne KCNK9 86 46 O=C(O)c1ccc(-c2nc(-c3cncs3)no2)cc1 ZINC000147425701 CF For-Sale Anodyne KCNQ1 0 41 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ncc(Cc4cccc(F)c4)s3)ccc21 ZINC000147425733 HH On-Demand Anodyne SCD1 37 40 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ncc(Cc4cccc(F)c4)s3)ccc21 ZINC000147425733 HH On-Demand Anodyne SCD 34 42 FC(F)(F)c1ccc(CN2CC[C@@H](Br)C2)cc1 ZINC000147425751 DH For-Sale Reactive DRD4 15 47 FC(F)(F)c1ccc(CN2CC[C@@H](Br)C2)cc1 ZINC000147425751 DH For-Sale Reactive SIGMAR1 27 49 FC(F)(F)c1ccc(CN2CC[C@@H](Br)C2)cc1 ZINC000147425751 DH For-Sale Reactive CCR2 16 42 FC(F)(F)c1ccc(CN2CC[C@@H](Br)C2)cc1 ZINC000147425751 DH For-Sale Reactive SLC6A5 29 41 FC(F)(F)c1ccc(CN2CC[C@@H](Br)C2)cc1 ZINC000147425751 DH For-Sale Reactive CACNA1G 25 40 CN(C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc(F)c(F)c1 ZINC000147425761 DI On-Demand Anodyne MDM2 58 32 CNc1ccncc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147425799 CD For-Sale Anodyne HCN1 40 31 CC(C)CCCCNC(=O)c1cc(Cl)nc2ccccc12 ZINC000147425810 DI For-Sale Anodyne DRD3 23 41 CC(C)CCCCNC(=O)c1cc(Cl)nc2ccccc12 ZINC000147425810 DI For-Sale Anodyne TACR2 0 40 CC(C)CCCCNC(=O)c1cc(Cl)nc2ccccc12 ZINC000147425810 DI For-Sale Anodyne BCHE 56 36 CC(C)CCCCNC(=O)c1cc(Cl)nc2ccccc12 ZINC000147425810 DI For-Sale Anodyne ACACB 25 42 CC(C)CCCCNC(=O)c1cc(Cl)nc2ccccc12 ZINC000147425810 DI For-Sale Anodyne TACR3 40 44 CC(C)CCCCNC(=O)c1cc(Cl)nc2ccccc12 ZINC000147425810 DI For-Sale Anodyne POLR1A 62 37 CN1CC[C@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147425813 CD For-Sale Anodyne CACNA1H 25 44 CN1CC[C@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147425813 CD For-Sale Anodyne EPHX2 42 54 CN1CC[C@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147425813 CD For-Sale Anodyne CXCR3 15 44 CN1CC[C@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147425813 CD For-Sale Anodyne CACNA1I 60 38 COc1ccc2c(c1)C(=O)/C(=C\N(C)C)CC2 ZINC000147425823 BE For-Sale Mild CYP27A1 0 47 CCc1ncc(C(=O)N[C@@H](c2ccc(OC)cc2)C(C)C)s1 ZINC000147425862 DH On-Demand Anodyne ACACB 47 38 Cc1nonc1CNC(=O)C(C)C ZINC000147425907 AC On-Demand Anodyne CASP3 47 36 Cc1nonc1CNC(=O)C(C)C ZINC000147425907 AC On-Demand Anodyne CASP7 54 36 CN(C)/C=C1/C(=O)Nc2ccc3ncccc3c21 ZINC000147425960 BE For-Sale Anodyne CDK2 15 56 CN(C)/C=C1/C(=O)Nc2ccc3ncccc3c21 ZINC000147425960 BE For-Sale Anodyne CDK1 16 56 CN(C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc(F)c(F)c1 ZINC000147425996 DI On-Demand Anodyne MDM2 58 32 CN1CC[C@@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147426003 CD For-Sale Anodyne CACNA1H 25 44 CN1CC[C@@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147426003 CD For-Sale Anodyne EPHX2 42 54 CN1CC[C@@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147426003 CD For-Sale Anodyne CXCR3 15 44 CN1CC[C@@H](NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147426003 CD For-Sale Anodyne CACNA1I 60 38 CNc1ccc(C(=O)NCC2(N(C)C)CCCC2)nn1 ZINC000147426033 CD For-Sale Anodyne HCN1 50 32 CNc1ccc(C(=O)NCC2(N(C)C)CCCC2)nn1 ZINC000147426033 CD For-Sale Anodyne HCN4 47 32 O=C(Cc1csc(-c2cccs2)n1)Nc1ccc2oc3ccccc3c2c1 ZINC000147426043 GK On-Demand Anodyne IMDH_CRYPV 44 48 CCc1ncc(C(=O)N[C@H](c2ccc(OC)cc2)C(C)C)s1 ZINC000147426065 DH On-Demand Anodyne ACACB 47 38 CCOC[C@H](C)NC(=O)Nc1cccc(C(=O)N2CCOCC2)c1 ZINC000147426067 ED On-Demand Anodyne EPHX2 30 57 CCc1cccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)c1 ZINC000147426112 HE On-Demand Anodyne KCNK3 42 32 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne DRD2 19 41 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne DRD4 48 39 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne ACHE 15 42 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne DRD3 18 40 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne HTR4 62 40 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne F10 21 45 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne GRIN2B 27 43 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne MMP13 28 48 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne CCR3 41 40 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne EPHX2 28 43 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne TGM2 60 42 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne CACNA1I 70 46 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne F13A1 50 42 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne AKR1C3 60 40 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne NAMPT 39 40 CCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147426172 HF On-Demand Anodyne PDS 59 37 CC(C)NS(=O)(=O)c1ccccc1NC[C@@H](C)CC(=O)O ZINC000147426177 DD For-Sale Anodyne ITGAV 48 41 CN(C(=O)[C@H]1C[C@H]1c1cccc(Cl)c1)c1ccc(F)c(F)c1 ZINC000147426210 DI On-Demand Anodyne MDM2 58 32 CC(C)CNCCCCOc1ccc(Cl)c(F)c1 ZINC000147426226 CH For-Sale Anodyne DRD4 19 43 CC(C)CCCCNC(=O)c1cc(Cl)c2ccccc2n1 ZINC000147426242 DI For-Sale Anodyne DRD3 22 41 CC(C)CCCCNC(=O)c1cc(Cl)c2ccccc2n1 ZINC000147426242 DI For-Sale Anodyne PLA2G7 21 44 CC(C)CCCCNC(=O)c1cc(Cl)c2ccccc2n1 ZINC000147426242 DI For-Sale Anodyne TSPO 20 40 CC(C)CCCCNC(=O)c1cc(Cl)c2ccccc2n1 ZINC000147426242 DI For-Sale Anodyne BCHE 63 35 COCc1nc(C(=O)N[C@H](c2ccccc2)C(C)C)cs1 ZINC000147426260 DG On-Demand Anodyne TACR3 20 41 C[C@H](NCC(F)F)c1ccc(O)cc1 ZINC000147426302 BE For-Sale Anodyne NMUR2 0 44 CNc1ccc(C(=O)NCC2(N(C)C)CCCC2)cc1 ZINC000147426324 CE For-Sale Anodyne SLC6A5 17 49 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(C(=O)N3CCOCC3)c2)C1 ZINC000147426352 HC On-Demand Anodyne CNR2 16 40 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(C(=O)N3CCOCC3)c2)C1 ZINC000147426352 HC On-Demand Anodyne EPHX2 55 54 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2cccc(C(=O)N3CCOCC3)c2)C1 ZINC000147426352 HC On-Demand Anodyne BTK 34 41 CC(C)NS(=O)(=O)c1ccccc1NC[C@H](C)CC(=O)O ZINC000147426378 DD For-Sale Anodyne ITGAV 48 41 CC(C)CCCCNC(=O)c1ccc(F)c(C(F)(F)F)c1 ZINC000147426429 DI For-Sale Anodyne TAAR1 18 45 CC(C)CCCCNC(=O)c1ccc(F)c(C(F)(F)F)c1 ZINC000147426429 DI For-Sale Anodyne LEF 41 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnns1 ZINC000147426440 FD On-Demand Anodyne HTR4 45 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnns1 ZINC000147426440 FD On-Demand Anodyne EPHX2 16 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnns1 ZINC000147426440 FD On-Demand Anodyne TGM2 64 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnns1 ZINC000147426440 FD On-Demand Anodyne CACNA1I 46 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnns1 ZINC000147426440 FD On-Demand Anodyne F13A1 60 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnns1 ZINC000147426440 FD On-Demand Anodyne NAMPT 46 40 CC[C@@H]1CN([C@@H](C)C(=O)N2CCCCC2)CC[C@@H]1N ZINC000147426443 CD On-Demand Anodyne DPP7 45 38 CC(C)C[C@@H]1CN(Cc2ccccc2)C[C@H]1C(=O)O ZINC000147426447 CF In-Stock Anodyne DRD3 24 40 CC(C)C[C@@H]1CN(Cc2ccccc2)C[C@H]1C(=O)O ZINC000147426447 CF In-Stock Anodyne S1PR3 26 41 C[C@@H](NCC(F)F)c1ccc(O)cc1 ZINC000147426514 BE For-Sale Anodyne NMUR2 0 44 Cc1cccc(C)c1NC(=O)C(=O)NCc1cccc(C(=O)NC[C@H]2CCCO2)c1 ZINC000147426542 HE On-Demand Anodyne LCK 24 43 Cc1cccc(C)c1NC(=O)C(=O)NCc1cccc(C(=O)NC[C@H]2CCCO2)c1 ZINC000147426542 HE On-Demand Anodyne FYN 18 43 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(C(=O)N3CCOCC3)c2)C1 ZINC000147426585 HC On-Demand Anodyne CNR2 16 40 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(C(=O)N3CCOCC3)c2)C1 ZINC000147426585 HC On-Demand Anodyne EPHX2 55 54 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2cccc(C(=O)N3CCOCC3)c2)C1 ZINC000147426585 HC On-Demand Anodyne BTK 34 41 C[C@H](CNc1ccccc1S(=O)(=O)NC1CC1)CC(=O)O ZINC000147426587 DD For-Sale Anodyne CCR8 97 40 C[C@H](CNc1ccccc1S(=O)(=O)NC1CC1)CC(=O)O ZINC000147426587 DD For-Sale Anodyne SFRP1 108 36 C[C@H](CNc1ccccc1S(=O)(=O)NC1CC1)CC(=O)O ZINC000147426587 DD For-Sale Anodyne WNT3 71 36 CCNc1ncccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147426597 CE For-Sale Anodyne SLC6A9 19 43 CCNc1ncccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147426597 CE For-Sale Anodyne SLC6A5 15 43 CCNc1ncccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147426597 CE For-Sale Anodyne HCN1 80 39 CCNc1ncccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147426597 CE For-Sale Anodyne HCN4 57 39 O=C(NCC1(C(=O)O)CCC1)c1cc(Cl)ccc1Cl ZINC000147426605 DF On-Demand Anodyne P2RX7 26 57 Cn1c(=O)n(C)c2cc(NC(=O)Nc3nc(C(F)(F)F)cs3)ccc21 ZINC000147426646 FF On-Demand Anodyne MPL 60 38 CC[C@H]1CN([C@@H](C)C(=O)N2CCCCC2)CC[C@@H]1N ZINC000147426665 CD For-Sale Anodyne DPP7 53 38 COC(=O)CN(C)C(=O)c1cc(C)cc(Cl)c1 ZINC000147426679 CD On-Demand Anodyne ECR 34 41 CC[C@H](N)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147426680 CD For-Sale Anodyne TPP2 62 41 N#Cc1ccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)cc1 ZINC000147426741 HD On-Demand Mild ROCK2 15 53 C[C@@H](CNc1ccccc1S(=O)(=O)NC1CC1)CC(=O)O ZINC000147426807 DD For-Sale Anodyne CCR8 97 40 C[C@@H](CNc1ccccc1S(=O)(=O)NC1CC1)CC(=O)O ZINC000147426807 DD For-Sale Anodyne SFRP1 108 36 C[C@@H](CNc1ccccc1S(=O)(=O)NC1CC1)CC(=O)O ZINC000147426807 DD For-Sale Anodyne WNT3 71 36 CNc1ccc(C(=O)NCC2(N(C)C)CCCC2)cn1 ZINC000147426820 CD On-Demand Anodyne SLC6A5 18 51 CNc1ccc(C(=O)NCC2(N(C)C)CCCC2)cn1 ZINC000147426820 CD On-Demand Anodyne HCN1 49 31 CNc1ccc(C(=O)NCC2(N(C)C)CCCC2)cn1 ZINC000147426820 CD On-Demand Anodyne HCN4 47 31 C[C@@H]1CN(C(=O)Nc2cccc(C(=O)N3CCOCC3)c2)C[C@H](c2ccccc2)O1 ZINC000147426827 HG On-Demand Anodyne EPHX2 20 50 CC[C@H](N)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147426857 CD For-Sale Anodyne TPP2 62 41 CC(C)CCCCNC(=O)c1cc(C(F)(F)F)ccc1F ZINC000147426858 DI For-Sale Anodyne LEF 53 37 CC(C)CCCCNC(=O)c1cc(C(F)(F)F)ccc1F ZINC000147426858 DI For-Sale Anodyne LIPG 40 33 O=C(Cn1cnc([N+](=O)[O-])n1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147426942 HC On-Demand Bother TGM2 62 42 O=C(Cn1cnc([N+](=O)[O-])n1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147426942 HC On-Demand Bother F13A1 61 42 CNc1ncccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147427021 CD For-Sale Anodyne SLC6A9 19 44 CNc1ncccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147427021 CD For-Sale Anodyne SLC6A5 15 44 CNc1ncccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147427021 CD For-Sale Anodyne HCN1 79 38 CNc1ncccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147427021 CD For-Sale Anodyne HCN4 56 38 C[C@H]1CN(C(=O)Nc2cccc(C(=O)N3CCOCC3)c2)C[C@H](c2ccccc2)O1 ZINC000147427023 HG On-Demand Anodyne EPHX2 20 50 Nc1nc(Oc2ccc(Br)cc2Cl)c2ccccc2n1 ZINC000147427034 FI For-Sale Anodyne DHFR 15 40 Nc1nc(Oc2ccc(Br)cc2Cl)c2ccccc2n1 ZINC000147427034 FI For-Sale Anodyne FOLA 19 40 c1ccc(-c2ccc(-c3c4ccccc4cc4ccc(-c5ccccc5)cc34)cc2)cc1 ZINC000147427096 HK For-Sale Bother HSD17B1 17 47 Cc1cc(C(=O)N2CCN(Cc3ccc4c(c3)OCCO4)CC2)cc([N+](=O)[O-])c1 ZINC000147427101 GF On-Demand Bother MCHR1 18 48 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1noc2c1CCCC2 ZINC000147427138 HE On-Demand Anodyne HTR4 50 36 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1noc2c1CCCC2 ZINC000147427138 HE On-Demand Anodyne TGM2 56 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1noc2c1CCCC2 ZINC000147427138 HE On-Demand Anodyne CACNA1I 59 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1noc2c1CCCC2 ZINC000147427138 HE On-Demand Anodyne F13A1 47 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1noc2c1CCCC2 ZINC000147427138 HE On-Demand Anodyne PANC 58 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1noc2c1CCCC2 ZINC000147427138 HE On-Demand Anodyne NAMPT 43 37 CC(CCCC(=O)O)(CCCC(=O)O)c1ccccc1 ZINC000147427226 CG For-Sale Anodyne AMY2 58 34 CC(CCCC(=O)O)(CCCC(=O)O)c1ccccc1 ZINC000147427226 CG For-Sale Anodyne KIF11 22 42 CNc1cc(C)ncc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147427231 CE For-Sale Anodyne SLC6A5 15 44 C[C@@H]1CN(C(=O)Nc2cccc(C(=O)N3CCOCC3)c2)C[C@@H](c2ccccc2)O1 ZINC000147427239 HG On-Demand Anodyne EPHX2 20 50 COc1ccc(NC(C)=O)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@@H](C)C1 ZINC000147427283 HE On-Demand Anodyne TSHR 40 29 O=C(O)C1(n2nnnc2-c2ccc(Cl)cc2)CCC1 ZINC000147427335 CD For-Sale Anodyne HSD11B1 23 40 CC(C)(C)OC(=O)N1CC=C(OS(C)(=O)=O)CC1 ZINC000147427383 CD For-Sale Mild GPR119 37 40 Cc1cc(CNC(=O)Cc2cccc(OC(C)C)c2)ccc1F ZINC000147427387 DH On-Demand Anodyne TRPV1 17 41 Cc1cc(CNC(=O)Cc2cccc(OC(C)C)c2)ccc1F ZINC000147427387 DH On-Demand Anodyne P2RX7 32 41 Cc1cc(CNC(=O)Cc2cccc(OC(C)C)c2)ccc1F ZINC000147427387 DH On-Demand Anodyne LEF 65 46 Cc1cc(CNC(=O)Cc2cccc(OC(C)C)c2)ccc1F ZINC000147427387 DH On-Demand Anodyne PDS 64 38 C[C@H]1CN(C(=O)Nc2cccc(C(=O)N3CCOCC3)c2)C[C@@H](c2ccccc2)O1 ZINC000147427418 HG On-Demand Anodyne EPHX2 20 50 CN(C)C(=O)NCCn1c(CCl)nc2ccccc2c1=O ZINC000147427436 DD For-Sale Reactive AGTR1 21 40 CN(C)C(=O)NCCn1c(CCl)nc2ccccc2c1=O ZINC000147427436 DD For-Sale Reactive POLR1A 59 34 CC[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(Cl)cc1 ZINC000147427438 DI On-Demand Anodyne BMP1 43 38 CC[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(Cl)cc1 ZINC000147427438 DI On-Demand Anodyne UTS2 44 36 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427446 FF On-Demand Anodyne KLK3 44 34 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427446 FF On-Demand Anodyne CTSK 43 43 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427446 FF On-Demand Anodyne ACACB 25 40 CCCC[C@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427446 FF On-Demand Anodyne CTSS 26 41 CCc1ncncc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147427451 GD On-Demand Anodyne HTR4 59 38 CCc1ncncc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147427451 GD On-Demand Anodyne TGM2 66 42 CCc1ncncc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147427451 GD On-Demand Anodyne CACNA1I 48 33 CCc1ncncc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147427451 GD On-Demand Anodyne F13A1 58 42 CCc1ncncc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147427451 GD On-Demand Anodyne NAMPT 41 38 COc1ccc(NC(C)=O)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@H](C)C1 ZINC000147427471 HE On-Demand Anodyne TSHR 40 29 CCCc1cc(NC[C@@H](C)CC(=O)O)ncn1 ZINC000147427494 BD For-Sale Anodyne OXER1 41 32 CN(C)Cc1cccc(NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)c1 ZINC000147427592 FF On-Demand Anodyne NAMPT 23 51 CN(C)Cc1cccc(NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)c1 ZINC000147427592 FF On-Demand Anodyne KCNK3 50 35 CC[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(Cl)cc1 ZINC000147427626 DI On-Demand Anodyne BMP1 43 38 CC[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(Cl)cc1 ZINC000147427626 DI On-Demand Anodyne UTS2 44 36 Cc1cc(N)c(C(=O)NCC2(N(C)C)CCCC2)cn1 ZINC000147427643 CD For-Sale Anodyne SLC6A5 15 45 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427652 FF On-Demand Anodyne KLK3 44 34 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427652 FF On-Demand Anodyne CTSK 43 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427652 FF On-Demand Anodyne ACACB 25 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427652 FF On-Demand Anodyne CTSS 26 41 CCCc1cc(NC[C@H](C)CC(=O)O)ncn1 ZINC000147427696 BD For-Sale Anodyne OXER1 41 32 O=C(COC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147427748 GE On-Demand Anodyne FKBP1A 23 43 O=C(COC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147427748 GE On-Demand Anodyne EPHX2 22 50 O=C(COC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147427748 GE On-Demand Anodyne TGM2 79 48 O=C(COC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147427748 GE On-Demand Anodyne F13A1 88 48 O=C(COC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147427748 GE On-Demand Anodyne AKR1C3 44 36 O=C(COC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147427748 GE On-Demand Anodyne NAMPT 35 40 Cc1cc(C(=O)N2CCC(C(=O)N3CCCCCC3)CC2)cc([N+](=O)[O-])c1 ZINC000147427789 FG On-Demand Bother L3MBTL1 0 41 Cc1cc(C(=O)N2CCC(C(=O)N3CCCCCC3)CC2)cc([N+](=O)[O-])c1 ZINC000147427789 FG On-Demand Bother L3MBTL3 59 37 CCOc1ccc(-c2nnnn2C2(C(=O)O)CCC2)cc1 ZINC000147427801 CD For-Sale Anodyne CACNA2D1 45 36 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427824 FF On-Demand Anodyne ACACA 18 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427824 FF On-Demand Anodyne KLK3 49 36 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427824 FF On-Demand Anodyne CTSK 51 43 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427824 FF On-Demand Anodyne ACACB 18 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427824 FF On-Demand Anodyne HLA-DRB1 32 40 CCCC[C@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147427824 FF On-Demand Anodyne CTSS 23 41 CS(=O)(=O)Nc1ccc(-c2csc(NC(=O)c3ccc(-n4cncn4)cc3)n2)cc1 ZINC000147427832 IG On-Demand Anodyne MPL 60 46 CS(=O)(=O)Nc1ccc(-c2csc(NC(=O)c3ccc(-n4cncn4)cc3)n2)cc1 ZINC000147427832 IG On-Demand Anodyne ROCK1 18 43 Cc1ccnc(-c2ccc(Cl)cc2Cl)c1[N+](=O)[O-] ZINC000147427843 CI For-Sale Anodyne S1PR4 18 40 Cc1ccc(F)cc1NC(=O)C(=O)NCc1cccc(C(=O)NC[C@H]2CCCO2)c1 ZINC000147427854 HE On-Demand Anodyne MAPK14 16 45 CNCc1ccccc1OCCOc1ccc(Cl)c(F)c1 ZINC000147427858 DH For-Sale Anodyne SLC6A4 17 60 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147427871 FF On-Demand Anodyne PIK3CA 28 42 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147427871 FF On-Demand Anodyne MTOR 62 45 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147427871 FF On-Demand Anodyne EPHX2 62 54 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147427871 FF On-Demand Anodyne PIK3CG 30 42 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@H]1C[C@H]1c1ccccc1 ZINC000147427871 FF On-Demand Anodyne BTK 40 37 C[C@@H](C[C@@](C)(CCCC(=O)O)c1ccccc1)C(=O)O ZINC000147427891 CG For-Sale Anodyne AMY2 53 31 C[C@@H](C[C@@](C)(CCCC(=O)O)c1ccccc1)C(=O)O ZINC000147427891 CG For-Sale Anodyne KIF11 28 41 COCCc1cc(-c2c(C)nc3c(N4CCOCC4)nccn23)ccn1 ZINC000147427915 FE Annotated Anodyne PDE10A 32 70 Cn1c(=O)n(C)c2cc(NC(=O)Nc3nc(C4CC4)cs3)ccc21 ZINC000147428019 EF On-Demand Anodyne TRPC6 46 33 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147428027 FF On-Demand Anodyne ACACA 18 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147428027 FF On-Demand Anodyne KLK3 49 36 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147428027 FF On-Demand Anodyne CTSK 51 43 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147428027 FF On-Demand Anodyne ACACB 18 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147428027 FF On-Demand Anodyne HLA-DRB1 32 40 CCCC[C@@H](NC(N)=O)C(=O)N[C@H](C)c1ccc(OC(F)(F)F)cc1 ZINC000147428027 FF On-Demand Anodyne CTSS 23 41 CC[C@@H]1CN(CC(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147428054 CD On-Demand Anodyne DRD4 22 52 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147428086 FF On-Demand Anodyne PIK3CA 28 42 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147428086 FF On-Demand Anodyne MTOR 62 45 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147428086 FF On-Demand Anodyne EPHX2 62 54 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147428086 FF On-Demand Anodyne PIK3CG 30 42 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147428086 FF On-Demand Anodyne BTK 40 37 C[C@H](C[C@@](C)(CCCC(=O)O)c1ccccc1)C(=O)O ZINC000147428103 CG For-Sale Anodyne AMY2 53 31 C[C@H](C[C@@](C)(CCCC(=O)O)c1ccccc1)C(=O)O ZINC000147428103 CG For-Sale Anodyne KIF11 28 41 Cc1ccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)cc1F ZINC000147428109 HE On-Demand Anodyne ENV 40 31 C[C@]1(C(=O)N(CCCC(=O)O)Cc2ccc(Cl)cc2)CCN1C(=O)Cc1coc2ccccc12 ZINC000147428123 JJ Annotated Anodyne FFAR2 180 83 CNc1cc(Oc2ccc(Br)cc2Cl)cc([N+](=O)[O-])c1 ZINC000147428172 FJ For-Sale Bother PPOX1 15 47 Cc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147428202 BD On-Demand Anodyne CCKAR 0 42 Cc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147428202 BD On-Demand Anodyne ACAT 0 45 Cc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147428202 BD On-Demand Anodyne KCNK3 91 52 Cc1cccc(C(=O)NCC2(C(=O)O)CCC2)c1 ZINC000147428202 BD On-Demand Anodyne KCNK9 62 52 C[C@H](Cl)c1nc2ccccc2c(=O)n1CCNC(N)=O ZINC000147428253 CD For-Sale Reactive POLR1A 60 32 CC[C@H]1CN(CC(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147428258 CD On-Demand Anodyne DRD4 22 52 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147428291 FF On-Demand Anodyne PIK3CA 28 42 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147428291 FF On-Demand Anodyne MTOR 62 45 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147428291 FF On-Demand Anodyne EPHX2 62 54 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147428291 FF On-Demand Anodyne PIK3CG 30 42 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147428291 FF On-Demand Anodyne BTK 40 37 C[C@H](CNc1cc(C(N)=O)c2ccccc2n1)CC(=O)O ZINC000147428301 CD For-Sale Anodyne TACR2 0 40 C[C@H](CNc1cc(C(N)=O)c2ccccc2n1)CC(=O)O ZINC000147428301 CD For-Sale Anodyne TACR3 43 42 C[C@H](CNc1cc(C(N)=O)c2ccccc2n1)CC(=O)O ZINC000147428301 CD For-Sale Anodyne METG 82 35 C[C@@H](C[C@](C)(CCCC(=O)O)c1ccccc1)C(=O)O ZINC000147428305 CG For-Sale Anodyne AMY2 53 31 C[C@@H](C[C@](C)(CCCC(=O)O)c1ccccc1)C(=O)O ZINC000147428305 CG For-Sale Anodyne KIF11 28 41 C[C@@]1(C(=O)N(CCCC(=O)O)Cc2ccc(Cl)cc2)CCN1C(=O)Cc1coc2ccccc12 ZINC000147428314 JJ Annotated Anodyne FFAR2 180 83 Cc1ccc(C)c(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)c1 ZINC000147428353 HE On-Demand Anodyne MAPK14 17 42 CCc1ncc(C(=O)N2CCN(Cc3ccc(OC)c(OC)c3OC)CC2)s1 ZINC000147428371 HF On-Demand Anodyne SLC9A1 69 39 CCCOc1nc(N)nc(Oc2ccc(Br)cc2Cl)n1 ZINC000147428399 FG For-Sale Anodyne S1PR4 0 40 O=c1ccc2ccc3c(c2o1)CCO3 ZINC000147428447 AD Annotated Anodyne NTBBF1.1 63 37 C[C@@H](Cl)c1nc2ccccc2c(=O)n1CCNC(N)=O ZINC000147428466 CD For-Sale Reactive POLR1A 60 32 CN[C@@H](C)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147428470 CD For-Sale Anodyne XIAP 52 35 CN[C@@H](C)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147428470 CD For-Sale Anodyne BIRC2 48 32 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147428480 FF On-Demand Anodyne PIK3CA 28 42 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147428480 FF On-Demand Anodyne MTOR 62 45 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147428480 FF On-Demand Anodyne EPHX2 62 54 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147428480 FF On-Demand Anodyne PIK3CG 30 42 O=C(Nc1ccc(C(=O)N2CCOCC2)cc1)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147428480 FF On-Demand Anodyne BTK 40 37 C[C@H](C[C@](C)(CCCC(=O)O)c1ccccc1)C(=O)O ZINC000147428506 CG For-Sale Anodyne AMY2 53 31 C[C@H](C[C@](C)(CCCC(=O)O)c1ccccc1)C(=O)O ZINC000147428506 CG For-Sale Anodyne KIF11 28 41 C[C@@H](CNc1cc(C(N)=O)c2ccccc2n1)CC(=O)O ZINC000147428512 CD For-Sale Anodyne TACR2 0 40 C[C@@H](CNc1cc(C(N)=O)c2ccccc2n1)CC(=O)O ZINC000147428512 CD For-Sale Anodyne TACR3 43 42 C[C@@H](CNc1cc(C(N)=O)c2ccccc2n1)CC(=O)O ZINC000147428512 CD For-Sale Anodyne METG 82 35 COc1cc([C@H](C)NCC(F)F)ccc1O ZINC000147428514 BE For-Sale Anodyne PNLIP 0 53 COc1cc([C@H](C)NCC(F)F)ccc1O ZINC000147428514 BE For-Sale Anodyne FOLH1 25 43 COc1cc([C@H](C)NCC(F)F)ccc1O ZINC000147428514 BE For-Sale Anodyne TRPV1 0 50 COc1cc([C@H](C)NCC(F)F)ccc1O ZINC000147428514 BE For-Sale Anodyne N1L 0 54 COc1cc([C@H](C)NCC(F)F)ccc1O ZINC000147428514 BE For-Sale Anodyne CAN2 0 45 COc1cc([C@H](C)NCC(F)F)ccc1O ZINC000147428514 BE For-Sale Anodyne SLC22A3 0 60 CC(C)(C)NCc1coc(COc2ccc(Cl)c(F)c2)c1 ZINC000147428521 DJ For-Sale Anodyne DAO 15 43 CC[C@@H]1CN([C@@H](C)C(=O)N2CCCCCC2)CC[C@@H]1N ZINC000147428553 CD On-Demand Anodyne DPP7 45 38 COc1cccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)c1 ZINC000147428634 HD On-Demand Anodyne DRD4 47 36 COc1cccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)c1 ZINC000147428634 HD On-Demand Anodyne CCR3 18 43 COc1cccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)c1 ZINC000147428634 HD On-Demand Anodyne ROCK2 38 41 COc1cccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)c1 ZINC000147428634 HD On-Demand Anodyne TAAR1 42 40 COc1cccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)c1 ZINC000147428634 HD On-Demand Anodyne KCNK3 40 42 CN[C@H](C)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147428696 CD For-Sale Anodyne XIAP 52 35 CN[C@H](C)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147428696 CD For-Sale Anodyne BIRC2 48 32 COc1cc([C@@H](C)NCC(F)F)ccc1O ZINC000147428716 BE For-Sale Anodyne PNLIP 0 53 COc1cc([C@@H](C)NCC(F)F)ccc1O ZINC000147428716 BE For-Sale Anodyne FOLH1 25 43 COc1cc([C@@H](C)NCC(F)F)ccc1O ZINC000147428716 BE For-Sale Anodyne TRPV1 0 50 COc1cc([C@@H](C)NCC(F)F)ccc1O ZINC000147428716 BE For-Sale Anodyne N1L 0 54 COc1cc([C@@H](C)NCC(F)F)ccc1O ZINC000147428716 BE For-Sale Anodyne CAN2 0 45 COc1cc([C@@H](C)NCC(F)F)ccc1O ZINC000147428716 BE For-Sale Anodyne SLC22A3 0 60 CN(C)C1(CNC(=O)c2cc(F)c(N)c(F)c2)CCCC1 ZINC000147428722 CE For-Sale Anodyne SLC6A5 18 53 CCN(CC)C(=O)Cc1cscn1 ZINC000147428740 AD On-Demand Anodyne BMP1 42 33 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428742 HC On-Demand Anodyne PIK3CA 35 44 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428742 HC On-Demand Anodyne MTOR 84 44 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428742 HC On-Demand Anodyne EPHX2 58 50 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428742 HC On-Demand Anodyne PIK3CG 34 44 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428742 HC On-Demand Anodyne BTK 40 38 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428742 HC On-Demand Anodyne L3MBTL3 55 36 C[C@H](CNc1cnc2ccccc2n1)CC(=O)O ZINC000147428751 BE On-Demand Anodyne CCR1 49 39 C[C@H](CNc1cnc2ccccc2n1)CC(=O)O ZINC000147428751 BE On-Demand Anodyne CASP1 21 46 C[C@H](CNc1cnc2ccccc2n1)CC(=O)O ZINC000147428751 BE On-Demand Anodyne CAPN2 22 46 C[C@H](CNc1cnc2ccccc2n1)CC(=O)O ZINC000147428751 BE On-Demand Anodyne METG 41 32 C[C@H](CNc1cnc2ccccc2n1)CC(=O)O ZINC000147428751 BE On-Demand Anodyne RHOA 0 44 CC[C@H]1CN([C@@H](C)C(=O)N2CCCCCC2)CC[C@@H]1N ZINC000147428756 CD For-Sale Anodyne DPP7 53 38 CC(C)(C)C(=O)NCCC(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147428822 EE On-Demand Anodyne MAPK14 37 41 CC(C)(C)C(=O)NCCC(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147428822 EE On-Demand Anodyne CCR2 27 40 CC(C)(C)C(=O)NCCC(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147428822 EE On-Demand Anodyne EPHX2 16 41 CC(C)(C)C(=O)NCCC(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147428822 EE On-Demand Anodyne PLAU 15 41 CC(C)(C)C(=O)NCCC(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147428822 EE On-Demand Anodyne KCNK3 76 37 CC(C)(C)C(=O)NCCC(=O)Nc1cccc(C(=O)NC2CC2)c1 ZINC000147428822 EE On-Demand Anodyne KCNK9 54 37 COc1ccccc1NC(=O)C(=O)NCc1cccc(C(=O)NC[C@H]2CCCO2)c1 ZINC000147428835 HD On-Demand Anodyne DRD2 19 40 COc1ccccc1NC(=O)C(=O)NCc1cccc(C(=O)NC[C@H]2CCCO2)c1 ZINC000147428835 HD On-Demand Anodyne DRD3 21 40 COc1ccccc1NC(=O)C(=O)NCc1cccc(C(=O)NC[C@H]2CCCO2)c1 ZINC000147428835 HD On-Demand Anodyne ROCK2 15 43 Cc1[nH]nc2ncc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc12 ZINC000147428847 HE On-Demand Anodyne HTR4 51 37 Cc1[nH]nc2ncc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc12 ZINC000147428847 HE On-Demand Anodyne TGM2 44 38 Cc1[nH]nc2ncc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc12 ZINC000147428847 HE On-Demand Anodyne CACNA1I 61 38 Cc1[nH]nc2ncc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc12 ZINC000147428847 HE On-Demand Anodyne NAMPT 49 49 CN[C@@H](C)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147428893 CD For-Sale Anodyne XIAP 52 35 CN[C@@H](C)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147428893 CD For-Sale Anodyne BIRC2 48 32 Cc1ccc(C(=O)NCC2(N(C)C)CCCC2)c(N)c1 ZINC000147428931 CE For-Sale Anodyne SLC6A5 15 43 Cc1ccc(C(=O)NCC2(N(C)C)CCCC2)c(N)c1 ZINC000147428931 CE For-Sale Anodyne HCN1 57 35 Cc1ccc(C(=O)NCC2(N(C)C)CCCC2)c(N)c1 ZINC000147428931 CE For-Sale Anodyne HCN4 48 34 O=C(Nc1nc2c(s1)CCCCCC2)c1ccc2c(c1)COC2 ZINC000147428940 EI On-Demand Anodyne SLC27A1 29 41 CNCc1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147428954 CH For-Sale Anodyne MAOB 47 41 CNCc1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147428954 CH For-Sale Anodyne TAAR1 16 41 C[C@@H](CNc1cnc2ccccc2n1)CC(=O)O ZINC000147428959 BE On-Demand Anodyne CCR1 49 39 C[C@@H](CNc1cnc2ccccc2n1)CC(=O)O ZINC000147428959 BE On-Demand Anodyne CASP1 21 46 C[C@@H](CNc1cnc2ccccc2n1)CC(=O)O ZINC000147428959 BE On-Demand Anodyne CAPN2 22 46 C[C@@H](CNc1cnc2ccccc2n1)CC(=O)O ZINC000147428959 BE On-Demand Anodyne METG 41 32 C[C@@H](CNc1cnc2ccccc2n1)CC(=O)O ZINC000147428959 BE On-Demand Anodyne RHOA 0 44 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428978 HC On-Demand Anodyne PIK3CA 35 44 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428978 HC On-Demand Anodyne MTOR 84 44 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428978 HC On-Demand Anodyne EPHX2 58 50 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428978 HC On-Demand Anodyne PIK3CG 34 44 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428978 HC On-Demand Anodyne BTK 40 38 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C1 ZINC000147428978 HC On-Demand Anodyne L3MBTL3 55 36 CN(Cc1cscn1)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147429018 GE On-Demand Anodyne DRD4 18 41 CN(Cc1cscn1)C(=O)NC1CCN(CC(=O)Nc2ccccc2)CC1 ZINC000147429018 GE On-Demand Anodyne LTA4H 15 44 c1cncc(N2C[C@@H]3CCN[C@H]3C2)c1 ZINC000147429051 AC For-Sale Anodyne HRH4 18 40 c1cncc(N2C[C@@H]3CCN[C@H]3C2)c1 ZINC000147429051 AC For-Sale Anodyne CHRNA3 62 72 c1cncc(N2C[C@@H]3CCN[C@H]3C2)c1 ZINC000147429051 AC For-Sale Anodyne CHRNA4 67 76 C#CCCCCCNCc1ccccc1 ZINC000147429054 BF For-Sale Mild SLC6A13 0 40 C#CCCCCCNCc1ccccc1 ZINC000147429054 BF For-Sale Mild GPM3 0 69 COC(=O)c1ccc(N2C[C@@H](C(=O)O)[C@@H](C)C2)nc1C ZINC000147429056 CD For-Sale Anodyne SORD 49 35 CN[C@H](C)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147429099 CD For-Sale Anodyne XIAP 52 35 CN[C@H](C)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147429099 CD For-Sale Anodyne BIRC2 48 32 CCNc1cccc(C(=O)NCC2(N(C)C)CCCC2)n1 ZINC000147429143 CE For-Sale Anodyne SLC6A5 15 41 CCNc1cccc(C(=O)NCC2(N(C)C)CCCC2)n1 ZINC000147429143 CE For-Sale Anodyne HCN1 50 31 CCNc1cccc(C(=O)NCC2(N(C)C)CCCC2)n1 ZINC000147429143 CE For-Sale Anodyne HCN4 48 31 C[C@@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@H](c2ccccc2)O1 ZINC000147429199 HG On-Demand Anodyne PIK3CA 17 41 C[C@@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@H](c2ccccc2)O1 ZINC000147429199 HG On-Demand Anodyne MTOR 32 41 C[C@@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@H](c2ccccc2)O1 ZINC000147429199 HG On-Demand Anodyne EPHX2 25 57 C[C@@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@H](c2ccccc2)O1 ZINC000147429199 HG On-Demand Anodyne PIK3CG 16 41 Cc1ccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)cc1C ZINC000147429245 HE On-Demand Anodyne MAPK14 15 42 COC(=O)c1ccc(N2C[C@@H](C)[C@H](C(=O)O)C2)nc1C ZINC000147429257 CD On-Demand Anodyne SORD 49 35 Nc1nccc(-c2ccc(F)c3ccccc23)n1 ZINC000147429311 BG For-Sale Anodyne ROCK1 24 47 Nc1nccc(-c2ccc(F)c3ccccc23)n1 ZINC000147429311 BG For-Sale Anodyne CDK9 28 40 Nc1nccc(-c2ccc(F)c3ccccc23)n1 ZINC000147429311 BG For-Sale Anodyne DYRK1A 18 47 Nc1nccc(-c2ccc(F)c3ccccc23)n1 ZINC000147429311 BG For-Sale Anodyne CDC7 50 42 Nc1nccc(-c2ccc(F)c3ccccc23)n1 ZINC000147429311 BG For-Sale Anodyne MAP3K14 55 51 CCNc1ccncc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147429320 CE For-Sale Anodyne HCN1 59 35 CCNc1ccncc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147429320 CE For-Sale Anodyne HCN4 50 33 C[C@@H](CN)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147429322 CD For-Sale Anodyne ACE 18 41 CC1=CC(C)(C)Nc2ccc(N3CCOCC3)nc21 ZINC000147429382 CF For-Sale Anodyne PGA 59 37 COc1cc2c(cc1O)CCN1C[C@H](CC(C)C)[C@@H](O)C[C@H]21 ZINC000147429389 DF For-Sale Anodyne DRD1 28 48 COc1cc2c(cc1O)CCN1C[C@H](CC(C)C)[C@@H](O)C[C@H]21 ZINC000147429389 DF For-Sale Anodyne SLC18A2 94 85 COc1cc2c(cc1O)CCN1C[C@H](CC(C)C)[C@@H](O)C[C@H]21 ZINC000147429389 DF For-Sale Anodyne F3 30 48 COc1cc2c(cc1O)CCN1C[C@H](CC(C)C)[C@@H](O)C[C@H]21 ZINC000147429389 DF For-Sale Anodyne SLC2A1 17 48 C[C@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@H](c2ccccc2)O1 ZINC000147429438 HG On-Demand Anodyne PIK3CA 17 41 C[C@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@H](c2ccccc2)O1 ZINC000147429438 HG On-Demand Anodyne MTOR 32 41 C[C@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@H](c2ccccc2)O1 ZINC000147429438 HG On-Demand Anodyne EPHX2 25 57 C[C@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@H](c2ccccc2)O1 ZINC000147429438 HG On-Demand Anodyne PIK3CG 16 41 O=C(NCc1cccc(C(=O)NC[C@H]2CCCO2)c1)C(=O)Nc1ccccc1Cl ZINC000147429468 HF On-Demand Anodyne SSTR3 21 41 O=C(NCc1cccc(C(=O)NC[C@H]2CCCO2)c1)C(=O)Nc1ccccc1Cl ZINC000147429468 HF On-Demand Anodyne MAPK10 18 41 C[C@H](CN)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147429500 CD For-Sale Anodyne ACE 18 41 CC(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147429502 GE On-Demand Anodyne HTR4 55 42 CC(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147429502 GE On-Demand Anodyne CHRM5 21 40 CC(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147429502 GE On-Demand Anodyne GRIN2B 30 41 CC(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147429502 GE On-Demand Anodyne EPHX2 19 40 CC(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147429502 GE On-Demand Anodyne TGM2 55 41 CC(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147429502 GE On-Demand Anodyne CACNA1I 59 36 CC(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147429502 GE On-Demand Anodyne F13A1 44 41 CNc1cc(C(=O)NCC2(N(C)C)CCCC2)ccn1 ZINC000147429543 CD For-Sale Anodyne SLC6A5 17 49 O=C(NCC1(C(=O)O)CCC1)c1ccc(Cl)cc1Cl ZINC000147429553 DF On-Demand Anodyne P2RX7 38 46 O=C(NCC1(C(=O)O)CCC1)c1ccc(Cl)cc1Cl ZINC000147429553 DF On-Demand Anodyne SLC6A9 34 40 C[C@H](CNc1cccc(Cl)c1C#N)CC(=O)O ZINC000147429615 CF For-Sale Mild CXCL8 49 36 CC(C)(C(=O)NCc1ccc(S(N)(=O)=O)cc1)c1ccc(S(=O)(=O)/C=C/C#N)cc1 ZINC000147429621 ID For-Sale Reactive CA2 70 56 CC(C)(C(=O)NCc1ccc(S(N)(=O)=O)cc1)c1ccc(S(=O)(=O)/C=C/C#N)cc1 ZINC000147429621 ID For-Sale Reactive CA1 55 56 CC(C)(C(=O)NCc1ccc(S(N)(=O)=O)cc1)c1ccc(S(=O)(=O)/C=C/C#N)cc1 ZINC000147429621 ID For-Sale Reactive CA7 37 56 CC(C)(C(=O)NCc1ccc(S(N)(=O)=O)cc1)c1ccc(S(=O)(=O)/C=C/C#N)cc1 ZINC000147429621 ID For-Sale Reactive CA5B 29 41 CC(C)(C(=O)NCc1ccc(S(N)(=O)=O)cc1)c1ccc(S(=O)(=O)/C=C/C#N)cc1 ZINC000147429621 ID For-Sale Reactive CA4 40 41 CC(C)(C(=O)NCc1ccc(S(N)(=O)=O)cc1)c1ccc(S(=O)(=O)/C=C/C#N)cc1 ZINC000147429621 ID For-Sale Reactive CA5A 29 41 CC(C)(C(=O)NCc1ccc(S(N)(=O)=O)cc1)c1ccc(S(=O)(=O)/C=C/C#N)cc1 ZINC000147429621 ID For-Sale Reactive CA14 39 56 CC(C)(C(=O)NCc1ccc(S(N)(=O)=O)cc1)c1ccc(S(=O)(=O)/C=C/C#N)cc1 ZINC000147429621 ID For-Sale Reactive CA12 42 41 CC(C)(C(=O)NCc1ccc(S(N)(=O)=O)cc1)c1ccc(S(=O)(=O)/C=C/C#N)cc1 ZINC000147429621 ID For-Sale Reactive CA9 46 41 CC(C)(C(=O)NCc1ccc(S(N)(=O)=O)cc1)c1ccc(S(=O)(=O)/C=C/C#N)cc1 ZINC000147429621 ID For-Sale Reactive CYNT 41 52 CCc1ccccc1C(=O)NCCC#N ZINC000147429660 BD On-Demand Mild SLC6A5 49 38 C[C@@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@@H](c2ccccc2)O1 ZINC000147429662 HG On-Demand Anodyne PIK3CA 17 41 C[C@@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@@H](c2ccccc2)O1 ZINC000147429662 HG On-Demand Anodyne MTOR 32 41 C[C@@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@@H](c2ccccc2)O1 ZINC000147429662 HG On-Demand Anodyne EPHX2 25 57 C[C@@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@@H](c2ccccc2)O1 ZINC000147429662 HG On-Demand Anodyne PIK3CG 16 41 CCCCC[C@@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147429680 DI For-Sale Anodyne CCKAR 0 41 CCCCC[C@@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147429680 DI For-Sale Anodyne CCKBR 22 41 C[C@@H](CN)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147429691 CD For-Sale Anodyne ACE 18 41 COc1c(F)cc(C(=O)NN)cc1F ZINC000147429714 BC For-Sale Reactive METC 0 52 COc1c(F)cc(C(=O)NN)cc1F ZINC000147429714 BC For-Sale Reactive H9B8T9_CAPHI 15 50 COc1ccc([N+](=O)[O-])c(C(=O)N(Cc2ccccn2)C(C)C)c1 ZINC000147429719 EG On-Demand Bother COLA 82 39 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)nn1C(C)(C)C ZINC000147429730 HF On-Demand Anodyne HTR4 57 36 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)nn1C(C)(C)C ZINC000147429730 HF On-Demand Anodyne EPHX2 27 40 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)nn1C(C)(C)C ZINC000147429730 HF On-Demand Anodyne TGM2 60 42 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)nn1C(C)(C)C ZINC000147429730 HF On-Demand Anodyne CACNA1I 63 39 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)nn1C(C)(C)C ZINC000147429730 HF On-Demand Anodyne F13A1 53 42 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)nn1C(C)(C)C ZINC000147429730 HF On-Demand Anodyne SFRP1 45 38 C[C@H](C(=O)NN1[C@@H](C)CCC[C@H]1C)[C@H](N)c1ccccc1 ZINC000147429732 CF For-Sale Anodyne XIAP 50 38 C[C@@H](CNc1cccc(Cl)c1C#N)CC(=O)O ZINC000147429768 CF For-Sale Mild CXCL8 49 36 O=C(CSc1ccccc1)NCC1(C(=O)O)CCC1 ZINC000147429825 CE On-Demand Anodyne NPFFR1 50 34 O=C(CSc1ccccc1)NCC1(C(=O)O)CCC1 ZINC000147429825 CE On-Demand Anodyne FAS 36 40 C[C@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@@H](c2ccccc2)O1 ZINC000147429848 HG On-Demand Anodyne PIK3CA 17 41 C[C@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@@H](c2ccccc2)O1 ZINC000147429848 HG On-Demand Anodyne MTOR 32 41 C[C@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@@H](c2ccccc2)O1 ZINC000147429848 HG On-Demand Anodyne EPHX2 25 57 C[C@H]1CN(C(=O)Nc2ccc(C(=O)N3CCOCC3)cc2)C[C@@H](c2ccccc2)O1 ZINC000147429848 HG On-Demand Anodyne PIK3CG 16 41 C[C@H](CN)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147429886 CD For-Sale Anodyne ACE 18 41 CCCCC[C@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147429897 DI For-Sale Anodyne CCKAR 0 41 CCCCC[C@H](C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147429897 DI For-Sale Anodyne CCKBR 22 41 CNCc1cccc2c(F)cccc12 ZINC000147429917 AF For-Sale Anodyne IFNAR1 0 46 C[C@H](CNc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)CC(=O)O ZINC000147429977 DG On-Demand Bother AR 0 60 C[C@H](CNc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)CC(=O)O ZINC000147429977 DG On-Demand Bother AADAC 0 60 O=C(Nc1cccc(C(=O)N2CCCCC2)c1)c1ccn(-c2cccc(F)c2)n1 ZINC000147429998 GH On-Demand Anodyne TAAR1 24 40 O=C(Nc1cccc(C(=O)N2CCCCC2)c1)c1ccn(-c2cccc(F)c2)n1 ZINC000147429998 GH On-Demand Anodyne HPGD 49 42 O=C(Nc1cccc(C(=O)N2CCCCC2)c1)c1ccn(-c2cccc(F)c2)n1 ZINC000147429998 GH On-Demand Anodyne KCNK3 44 40 Cc1cc(N(CCBr)C2CCCCC2)n2ncnc2n1 ZINC000147430021 EF For-Sale Reactive DHOD 0 42 CC(C)[C@@H](CNC1CC1)Oc1ccc(Cl)c(F)c1 ZINC000147430030 CH For-Sale Anodyne ENV 41 32 Cc1ccccc1C(=O)NNC(=O)Nc1nc(C2CC2)cs1 ZINC000147430042 DF On-Demand Reactive ROCK1 17 42 Cc1ccccc1C(=O)NNC(=O)Nc1nc(C2CC2)cs1 ZINC000147430042 DF On-Demand Reactive CCR8 48 32 COc1ccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)cc1 ZINC000147430043 HD On-Demand Anodyne DRD4 43 33 COc1ccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)cc1 ZINC000147430043 HD On-Demand Anodyne MMP13 23 42 COc1ccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)cc1 ZINC000147430043 HD On-Demand Anodyne ROCK2 41 45 COc1ccc(NC(=O)C(=O)NCc2cccc(C(=O)NC[C@H]3CCCO3)c2)cc1 ZINC000147430043 HD On-Demand Anodyne MCHR1 15 41 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne CNR1 29 61 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne PLA2G4C 0 59 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne FABP2 0 50 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne FABP4 31 85 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne LPAR1 18 40 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne PLA2G4B 54 59 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne FAAH 20 59 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne EPHX2 15 56 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne CDC25C 0 50 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne PLCG1 0 42 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne Q6UB75_PIG 0 41 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne FABP3 65 82 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne FABP5 22 71 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne LOX1.1 18 82 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne FABP1 24 71 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne SLC22A20 0 52 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne ACAT 0 45 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne SAE1 0 42 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne OXER1 31 64 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne CQSS 51 31 CCCCC/C=C/C/C=C/C/C=C/C/C=C/C/C=C\CCC(=O)O ZINC000147430097 EK For-Sale Anodyne SLCO2A1 48 37 C[C@]1(C(=O)Nc2cccc(NS(N)(=O)=O)c2)CCCS1 ZINC000147430109 DD For-Sale Anodyne NCE103 22 41 C[C@H](C(=O)NN1[C@H](C)CCC[C@H]1C)[C@H](N)c1ccccc1 ZINC000147430129 CF For-Sale Anodyne XIAP 50 38 CC[C@H](NC(=O)N[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147430132 CD For-Sale Anodyne ACE 28 40 CC[C@H](NC(=O)N[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147430132 CD For-Sale Anodyne MME 34 40 CC[C@H](NC(=O)N[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147430132 CD For-Sale Anodyne EPHX2 24 52 CC[C@H](NC(=O)N[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147430132 CD For-Sale Anodyne ACE2 66 35 CC[C@H](NC(=O)N[C@@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147430132 CD For-Sale Anodyne KDM1A 44 36 C[C@@H](CNc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)CC(=O)O ZINC000147430199 DG On-Demand Bother AR 0 60 C[C@@H](CNc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)CC(=O)O ZINC000147430199 DG On-Demand Bother AADAC 0 60 CC(C)[C@H](CNC1CC1)Oc1ccc(Cl)c(F)c1 ZINC000147430216 CH For-Sale Anodyne ENV 41 32 O=C(Nc1ccc(C(=O)N2CCCCCC2)cc1)c1ccn(-c2cccc(F)c2)n1 ZINC000147430255 HI On-Demand Anodyne AVPR2 41 36 O=C(Nc1ccc(C(=O)N2CCCCCC2)cc1)c1ccn(-c2cccc(F)c2)n1 ZINC000147430255 HI On-Demand Anodyne HPGD 49 42 CNc1cc(C)ccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147430274 CF For-Sale Anodyne SLC6A5 15 43 CNc1cc(C)ccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147430274 CF For-Sale Anodyne HCN1 44 35 Cc1ccc(F)cc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147430307 CE On-Demand Anodyne HCN1 49 30 Cc1ccc(F)cc1C(=O)NCC1(C(=O)O)CCC1 ZINC000147430307 CE On-Demand Anodyne HCN4 46 30 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive ADORA2B 52 44 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive HTR7 21 43 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive HSD11B1 15 49 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive MMP13 57 47 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive HTR6 19 44 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive MMP2 30 47 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive MMP3 55 47 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive MMP8 32 47 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive MMP9 48 47 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive PKM 34 71 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive MMP7 50 47 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive MMP1 56 47 COc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147430312 FD For-Sale Reactive F13A1 45 36 CCC(CC)C(=O)CCCN ZINC000147430316 AD For-Sale Anodyne CQSS 63 42 CC[C@H](NC(=O)N[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147430325 CD For-Sale Anodyne ACE 28 40 CC[C@H](NC(=O)N[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147430325 CD For-Sale Anodyne MME 34 40 CC[C@H](NC(=O)N[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147430325 CD For-Sale Anodyne EPHX2 24 52 CC[C@H](NC(=O)N[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147430325 CD For-Sale Anodyne ACE2 66 35 CC[C@H](NC(=O)N[C@H]1C[C@H]1c1ccccc1)C(=O)O ZINC000147430325 CD For-Sale Anodyne KDM1A 44 36 C[C@@]1(C(=O)Nc2cccc(NS(N)(=O)=O)c2)CCCS1 ZINC000147430334 DD For-Sale Anodyne NCE103 22 41 N#Cc1cc(CC(=O)NN)ccc1O ZINC000147430336 AB For-Sale Reactive AOC2 0 41 N#Cc1cc(CC(=O)NN)ccc1O ZINC000147430336 AB For-Sale Reactive NCE103 29 41 N#Cc1cc(CC(=O)NN)ccc1O ZINC000147430336 AB For-Sale Reactive CAN2 0 41 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cnc(-c4ccccc4)nc3)ccc21 ZINC000147430349 FF On-Demand Anodyne MAPK14 15 43 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cnc(-c4ccccc4)nc3)ccc21 ZINC000147430349 FF On-Demand Anodyne IMPDH2 18 44 CCCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147430361 HG On-Demand Anodyne DRD2 15 41 CCCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147430361 HG On-Demand Anodyne DRD4 47 38 CCCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147430361 HG On-Demand Anodyne HTR4 49 38 CCCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147430361 HG On-Demand Anodyne F10 19 48 CCCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147430361 HG On-Demand Anodyne GRIN2B 26 44 CCCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147430361 HG On-Demand Anodyne MMP13 34 41 CCCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147430361 HG On-Demand Anodyne EPHX2 26 42 CCCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147430361 HG On-Demand Anodyne TGM2 56 41 CCCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147430361 HG On-Demand Anodyne CACNA1I 65 43 CCCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147430361 HG On-Demand Anodyne F13A1 43 41 CCCOc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147430361 HG On-Demand Anodyne AKR1C3 59 39 COc1ccc(/C=C/C(=O)N2CCC[C@@H]2CN2CCCC2)cc1 ZINC000147430417 DF On-Demand Anodyne OPRK1 29 47 Cc1nn(-c2ccccc2)c(C)c1NC(=O)Nc1ccc2c(c1)n(C)c(=O)n2C ZINC000147430554 GG On-Demand Anodyne FPR2 62 44 Cc1ccc(Br)c(C(=O)N(C)Cc2ccc(F)c(F)c2)c1 ZINC000147430558 FI On-Demand Anodyne HSP90AB1 36 48 COc1ccc(/C=C/C(=O)N2CCC[C@H]2CN2CCCC2)cc1 ZINC000147430631 DF On-Demand Anodyne OPRK1 29 47 O=C1CC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147430635 GC On-Demand Anodyne EPHX2 31 47 O=C1CC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147430635 GC On-Demand Anodyne TGM2 60 43 O=C1CC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147430635 GC On-Demand Anodyne F13A1 47 43 O=C1CC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147430635 GC On-Demand Anodyne SFRP1 54 38 CNCc1ccccc1COc1ccc(Cl)c(F)c1 ZINC000147430695 CH For-Sale Anodyne SLC6A4 15 57 CCNc1cc(Oc2ccc(Br)cc2Cl)cc([N+](=O)[O-])c1 ZINC000147430740 FK For-Sale Bother ENR 0 42 CCNc1cc(Oc2ccc(Br)cc2Cl)cc([N+](=O)[O-])c1 ZINC000147430740 FK For-Sale Bother PPOX1 15 44 CCNc1ccnc(C(=O)NCC2(N(C)C)CCCC2)c1 ZINC000147430752 CE For-Sale Anodyne SLC6A5 15 45 CCNc1ccnc(C(=O)NCC2(N(C)C)CCCC2)c1 ZINC000147430752 CE For-Sale Anodyne HCN1 49 31 CCNc1ccnc(C(=O)NCC2(N(C)C)CCCC2)c1 ZINC000147430752 CE For-Sale Anodyne HCN4 47 31 C[C@@H]1CCCN(Cc2csc(NC(=O)Nc3ccc4c(c3)n(C)c(=O)n4C)n2)C1 ZINC000147430776 HG On-Demand Anodyne CCR3 43 31 C[C@@H]1CCCN(Cc2csc(NC(=O)Nc3ccc4c(c3)n(C)c(=O)n4C)n2)C1 ZINC000147430776 HG On-Demand Anodyne TRPC6 47 34 C[C@@H]1CCCN(Cc2csc(NC(=O)Nc3ccc4c(c3)n(C)c(=O)n4C)n2)C1 ZINC000147430776 HG On-Demand Anodyne TRPC3 44 34 NS(=O)(=O)c1cccc(S(=O)(=O)Nc2cc3c(cc2Cl)OCCO3)c1 ZINC000147430784 HD On-Demand Anodyne CA2 23 44 NS(=O)(=O)c1cccc(S(=O)(=O)Nc2cc3c(cc2Cl)OCCO3)c1 ZINC000147430784 HD On-Demand Anodyne CA1 20 44 NS(=O)(=O)c1cccc(S(=O)(=O)Nc2cc3c(cc2Cl)OCCO3)c1 ZINC000147430784 HD On-Demand Anodyne CA4 30 43 NS(=O)(=O)c1cccc(S(=O)(=O)Nc2cc3c(cc2Cl)OCCO3)c1 ZINC000147430784 HD On-Demand Anodyne PKM 27 41 NS(=O)(=O)c1cccc(S(=O)(=O)Nc2cc3c(cc2Cl)OCCO3)c1 ZINC000147430784 HD On-Demand Anodyne CAH_METTE 27 40 NS(=O)(=O)c1cccc(S(=O)(=O)Nc2cc3c(cc2Cl)OCCO3)c1 ZINC000147430784 HD On-Demand Anodyne CYNT 26 41 NS(=O)(=O)c1cccc(S(=O)(=O)Nc2cc3c(cc2Cl)OCCO3)c1 ZINC000147430784 HD On-Demand Anodyne CA15 23 41 NS(=O)(=O)c1cccc(S(=O)(=O)Nc2cc3c(cc2Cl)OCCO3)c1 ZINC000147430784 HD On-Demand Anodyne A6YCJ1_9METZ 15 41 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@H](C)C1 ZINC000147430806 HE On-Demand Anodyne MAPK11 42 43 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@H](C)C1 ZINC000147430806 HE On-Demand Anodyne MAPK14 53 41 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@H](C)C1 ZINC000147430806 HE On-Demand Anodyne MAPK13 44 35 O=C1CC[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147430835 GC On-Demand Anodyne EPHX2 31 47 O=C1CC[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147430835 GC On-Demand Anodyne TGM2 60 43 O=C1CC[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147430835 GC On-Demand Anodyne F13A1 47 43 O=C1CC[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CN1 ZINC000147430835 GC On-Demand Anodyne SFRP1 54 38 CCCN(CCS(=O)(=O)c1cccc(C#N)c1)C1CC1 ZINC000147430859 CE On-Demand Mild HTR1A 23 41 CC[C@@H]1CN(CCCn2ccnc2)CC[C@@H]1N ZINC000147430906 BD For-Sale Anodyne TBXAS1 22 44 CC(C)NCc1ccc(COc2ccc(Cl)c(F)c2)cc1 ZINC000147430954 DJ For-Sale Anodyne MAOB 29 43 COC(=O)COc1ccc(S(=O)(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)cc1 ZINC000147430962 HE On-Demand Anodyne MMP13 68 44 COC(=O)COc1ccc(S(=O)(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)cc1 ZINC000147430962 HE On-Demand Anodyne ADAM17 57 39 COC(=O)COc1ccc(S(=O)(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)cc1 ZINC000147430962 HE On-Demand Anodyne MMP3 62 44 COC(=O)COc1ccc(S(=O)(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)cc1 ZINC000147430962 HE On-Demand Anodyne MMP9 38 44 COC(=O)COc1ccc(S(=O)(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)cc1 ZINC000147430962 HE On-Demand Anodyne MMP7 66 44 COC(=O)COc1ccc(S(=O)(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)cc1 ZINC000147430962 HE On-Demand Anodyne MMP1 68 44 C[C@H]1CCCN(Cc2csc(NC(=O)Nc3ccc4c(c3)n(C)c(=O)n4C)n2)C1 ZINC000147430965 HG On-Demand Anodyne CCR3 43 31 C[C@H]1CCCN(Cc2csc(NC(=O)Nc3ccc4c(c3)n(C)c(=O)n4C)n2)C1 ZINC000147430965 HG On-Demand Anodyne TRPC6 47 34 C[C@H]1CCCN(Cc2csc(NC(=O)Nc3ccc4c(c3)n(C)c(=O)n4C)n2)C1 ZINC000147430965 HG On-Demand Anodyne TRPC3 44 34 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@@H](C)C1 ZINC000147431000 HE On-Demand Anodyne MAPK11 42 43 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@@H](C)C1 ZINC000147431000 HE On-Demand Anodyne MAPK14 53 41 Cc1ccc(C(=O)NC2CC2)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@@H](C)C1 ZINC000147431000 HE On-Demand Anodyne MAPK13 44 35 CNc1ccnc(C(=O)NCC2(N(C)C)CCCC2)c1 ZINC000147431009 CD For-Sale Anodyne SLC6A5 15 44 Cc1nn(C(F)F)c(C)c1CC(=O)NC[C@@H](C)N1C[C@H](C)O[C@H](C)C1 ZINC000147431064 FE On-Demand Anodyne P2RX7 17 40 CC[C@H]1CN(CCCn2ccnc2)CC[C@@H]1N ZINC000147431083 BD For-Sale Anodyne TBXAS1 22 44 O=C(Cc1nc2ncccn2n1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147431117 HC On-Demand Anodyne TGM2 58 39 O=C(Cc1nc2ncccn2n1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147431117 HC On-Demand Anodyne F13A1 55 39 O=C(Cc1nc2ncccn2n1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147431117 HC On-Demand Anodyne NAMPT 42 36 CCNc1ccc(C(=O)NCC2(N(C)C)CCCC2)cn1 ZINC000147431213 CE For-Sale Anodyne SLC6A5 17 49 CCNc1ccc(C(=O)NCC2(N(C)C)CCCC2)cn1 ZINC000147431213 CE For-Sale Anodyne HCN1 50 32 CCNc1ccc(C(=O)NCC2(N(C)C)CCCC2)cn1 ZINC000147431213 CE For-Sale Anodyne HCN4 48 32 C[C@@H]1CN(S(=O)(=O)c2cc3c(cc2F)NC(=O)CC3)C[C@H](c2ccccc2)O1 ZINC000147431220 HF On-Demand Anodyne PKM 39 44 Cc1ccccc1NC(=O)CNc1ccc(Cl)cc1Br ZINC000147431282 FI On-Demand Anodyne CA1 17 41 Cc1ccccc1NC(=O)CNc1ccc(Cl)cc1Br ZINC000147431282 FI On-Demand Anodyne CA4 20 40 Cc1nn(C(F)F)c(C)c1CC(=O)NC[C@H](C)N1C[C@H](C)O[C@H](C)C1 ZINC000147431290 FE On-Demand Anodyne P2RX7 17 40 COC(=O)N(C)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147431331 GC On-Demand Anodyne CHRM5 17 41 COC(=O)N(C)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147431331 GC On-Demand Anodyne EPHX2 18 43 COC(=O)N(C)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147431331 GC On-Demand Anodyne TGM2 67 44 COC(=O)N(C)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147431331 GC On-Demand Anodyne F13A1 70 44 CC[C@H](C(=O)N1CCC[C@@H]1CCCBr)c1ccccc1 ZINC000147431380 EI For-Sale Reactive KCNQ2 50 42 CC[C@H](C(=O)N1CCC[C@@H]1CCCBr)c1ccccc1 ZINC000147431380 EI For-Sale Reactive KCNQ4 0 42 NC(=O)c1cccc(CNCC(F)F)c1 ZINC000147431387 BD On-Demand Anodyne F10 15 40 NC(=O)c1cccc(CNCC(F)F)c1 ZINC000147431387 BD On-Demand Anodyne TRY2_BOVIN 47 31 NC(=O)c1cccc(CNCC(F)F)c1 ZINC000147431387 BD On-Demand Anodyne MVFR 0 41 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(-c4nc5ccccc5o4)cc3)ccc21 ZINC000147431430 HI On-Demand Anodyne MTOR 56 36 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(-c4nc5ccccc5o4)cc3)ccc21 ZINC000147431430 HI On-Demand Anodyne PTPN11 44 36 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(-c4nc5ccccc5o4)cc3)ccc21 ZINC000147431430 HI On-Demand Anodyne HPSE 49 37 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(-c4nc5ccccc5o4)cc3)ccc21 ZINC000147431430 HI On-Demand Anodyne AGPAT2 40 44 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(-c4nc5ccccc5o4)cc3)ccc21 ZINC000147431430 HI On-Demand Anodyne NR2E3 43 32 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(-c4nc5ccccc5o4)cc3)ccc21 ZINC000147431430 HI On-Demand Anodyne IMDH_CRYPV 59 42 C[C@H]1CN(S(=O)(=O)c2cc3c(cc2F)NC(=O)CC3)C[C@H](c2ccccc2)O1 ZINC000147431460 HF On-Demand Anodyne PKM 39 44 NCC1(CC(=O)N2CCC[C@H](C(N)=O)C2)CCC1 ZINC000147431474 CC For-Sale Anodyne CACNA2D1 0 41 CN(Cc1cscn1)C(=O)NCc1ccccc1OC(F)F ZINC000147431489 EG On-Demand Anodyne BMP1 50 33 O=C(CNc1ccc(Cl)cc1Br)NCc1ccccc1 ZINC000147431517 FH On-Demand Anodyne CA5B 26 40 O=C(CNc1ccc(Cl)cc1Br)NCc1ccccc1 ZINC000147431517 FH On-Demand Anodyne CA5A 29 40 O=C(CNc1ccc(Cl)cc1Br)NCc1ccccc1 ZINC000147431517 FH On-Demand Anodyne AMP1_PLAFQ 31 42 O=C(CNc1ccc(Cl)cc1Br)NCc1ccccc1 ZINC000147431517 FH On-Demand Anodyne PDS 42 36 COc1ccc2c(C)ncnc2c1 ZINC000147431529 AD For-Sale Anodyne CYP1B1 40 36 COc1ccc2c(C)ncnc2c1 ZINC000147431529 AD For-Sale Anodyne PDE3B 57 39 CS[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147431559 FD On-Demand Anodyne CHRM5 22 42 CS[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147431559 FD On-Demand Anodyne TGM2 64 45 CS[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147431559 FD On-Demand Anodyne CACNA1I 40 32 CS[C@@H](C)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147431559 FD On-Demand Anodyne F13A1 72 45 CC[C@@H](C(=O)N1CCC[C@@H]1CCCBr)c1ccccc1 ZINC000147431588 EI For-Sale Reactive KCNQ2 50 42 CC[C@@H](C(=O)N1CCC[C@@H]1CCCBr)c1ccccc1 ZINC000147431588 EI For-Sale Reactive KCNQ4 0 42 N#Cc1cccc(S(=O)(=O)CCN2CCC[C@H]2CO)c1 ZINC000147431592 CC On-Demand Mild CHRNA10 35 47 CCc1ncc(C(=O)Nc2ccccc2N2CCCC2=O)s1 ZINC000147431619 DG On-Demand Anodyne KCNQ2 72 34 CCOC(=O)COc1cccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)c1 ZINC000147431645 HE On-Demand Anodyne TAAR1 23 40 NCC1(CC(=O)N2CCC[C@@H](C(N)=O)C2)CCC1 ZINC000147431679 CC For-Sale Anodyne CACNA2D1 0 41 O=C(O)[C@H](O)C(=O)N1CCCCC1 ZINC000147431745 AB For-Sale Anodyne DPP7 45 39 O=C(O)c1ccccc1-c1nc(-c2cncs2)no1 ZINC000147431766 CF For-Sale Anodyne LUCI_PHOPE 40 34 CC[C@H](C(=O)N1CCC[C@H]1CCCBr)c1ccccc1 ZINC000147431793 EI For-Sale Reactive KCNQ2 50 42 CC[C@H](C(=O)N1CCC[C@H]1CCCBr)c1ccccc1 ZINC000147431793 EI For-Sale Reactive KCNQ4 0 42 C[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147431799 GC On-Demand Anodyne HTR4 45 39 C[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147431799 GC On-Demand Anodyne CHRM5 22 43 C[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147431799 GC On-Demand Anodyne TGM2 66 46 C[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147431799 GC On-Demand Anodyne CACNA1I 41 33 C[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147431799 GC On-Demand Anodyne F13A1 75 46 CCOC(=O)COc1cccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)c1 ZINC000147431859 HE On-Demand Anodyne TAAR1 23 40 CCCNc1ncnc(Oc2ccc(Br)cc2Cl)c1CC ZINC000147431865 FK For-Sale Anodyne HTT 0 51 COc1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147431894 BE For-Sale Anodyne CA1 21 43 COc1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147431894 BE For-Sale Anodyne MTNR1A 56 43 COc1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147431894 BE For-Sale Anodyne MTNR1B 48 43 COc1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147431894 BE For-Sale Anodyne ACR 50 43 COc1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147431894 BE For-Sale Anodyne CA12 16 47 COc1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147431894 BE For-Sale Anodyne CA9 22 47 CCc1ccc(C(=O)NCC2(C(=O)O)CCC2)o1 ZINC000147431915 CD For-Sale Anodyne GNRHR 22 40 O=C(O)[C@@H](O)C(=O)N1CCCCC1 ZINC000147431939 AB For-Sale Anodyne DPP7 45 39 CC(C)CCCCNC(=O)[C@@H]1CCCN1C1CCNCC1 ZINC000147431947 CE For-Sale Anodyne TPP2 43 42 CC(C)CCCCNC(=O)[C@@H]1CCCN1C1CCNCC1 ZINC000147431947 CE For-Sale Anodyne GNAI1 0 41 CC(C)CCCCNC(=O)[C@@H]1CCCN1C1CCNCC1 ZINC000147431947 CE For-Sale Anodyne GNAI3 0 41 CC(C)CCCCNC(=O)[C@@H]1CCCN1C1CCNCC1 ZINC000147431947 CE For-Sale Anodyne GNAO1 0 41 CCNC(=O)CN(C)C(=O)c1ccccc1NS(=O)(=O)c1ccc(F)c(F)c1 ZINC000147431953 HD On-Demand Anodyne PRTN3 61 39 CCNC(=O)CN(C)C(=O)c1ccccc1NS(=O)(=O)c1ccc(F)c(F)c1 ZINC000147431953 HD On-Demand Anodyne LIMK2 26 44 Clc1nc(Nc2ccc3c(c2)CCC3)c2nc[nH]c2n1 ZINC000147432005 CG For-Sale Anodyne BRAF 0 52 Clc1nc(Nc2ccc3c(c2)CCC3)c2nc[nH]c2n1 ZINC000147432005 CG For-Sale Anodyne PRIM_HHV11 44 41 Clc1nc(Nc2ccc3c(c2)CCC3)c2nc[nH]c2n1 ZINC000147432005 CG For-Sale Anodyne AHK4 0 62 Clc1nc(Nc2ccc3c(c2)CCC3)c2nc[nH]c2n1 ZINC000147432005 CG For-Sale Anodyne AHK3 0 59 Clc1nc(Nc2ccc3c(c2)CCC3)c2nc[nH]c2n1 ZINC000147432005 CG For-Sale Anodyne CKX2 0 62 CC[C@@H](C(=O)N1CCC[C@H]1CCCBr)c1ccccc1 ZINC000147432009 EI For-Sale Reactive KCNQ2 50 42 CC[C@@H](C(=O)N1CCC[C@H]1CCCBr)c1ccccc1 ZINC000147432009 EI For-Sale Reactive KCNQ4 0 42 C[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147432037 GC On-Demand Anodyne HTR4 45 39 C[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147432037 GC On-Demand Anodyne CHRM5 22 43 C[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147432037 GC On-Demand Anodyne TGM2 66 46 C[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147432037 GC On-Demand Anodyne CACNA1I 41 33 C[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147432037 GC On-Demand Anodyne F13A1 75 46 C=CC(C)(C)c1cc(OC)c(O)cc1-c1coc2cc(O)cc(O)c2c1=O ZINC000147432055 FI Annotated Mild CYP1B1 25 40 C=CC(C)(C)c1cc(OC)c(O)cc1-c1coc2cc(O)cc(O)c2c1=O ZINC000147432055 FI Annotated Mild CYP1A1 16 40 C=CC(C)(C)c1cc(OC)c(O)cc1-c1coc2cc(O)cc(O)c2c1=O ZINC000147432055 FI Annotated Mild LYZ1 0 49 CCNc1ccc(C(=O)NCC2(N(C)C)CCCC2)nn1 ZINC000147432090 CD For-Sale Anodyne HCN1 51 32 CCNc1ccc(C(=O)NCC2(N(C)C)CCCC2)nn1 ZINC000147432090 CD For-Sale Anodyne HCN4 49 32 CC(C)CCCCNC(=O)[C@H]1CCCN1C1CCNCC1 ZINC000147432133 CE For-Sale Anodyne TPP2 43 42 CC(C)CCCCNC(=O)[C@H]1CCCN1C1CCNCC1 ZINC000147432133 CE For-Sale Anodyne GNAI1 0 41 CC(C)CCCCNC(=O)[C@H]1CCCN1C1CCNCC1 ZINC000147432133 CE For-Sale Anodyne GNAI3 0 41 CC(C)CCCCNC(=O)[C@H]1CCCN1C1CCNCC1 ZINC000147432133 CE For-Sale Anodyne GNAO1 0 41 C[C@H](CNc1ncc(C(F)(F)F)cc1Cl)CC(=O)O ZINC000147432183 CG For-Sale Anodyne TRPM8 40 37 C[C@H](CNc1ncc(C(F)(F)F)cc1Cl)CC(=O)O ZINC000147432183 CG For-Sale Anodyne H9BT73_9POAL 0 44 COc1ccc(C)cc1-n1ccc(C(=O)Nc2ccc3[nH]c(C)cc3c2)n1 ZINC000147432211 FI On-Demand Anodyne ENPP1 78 38 CCCCCCCCCC(=O)N1CCC[C@@H]1CCCBr ZINC000147432262 EK For-Sale Reactive PREP 22 41 CCCCCCCCCC(=O)N1CCC[C@@H]1CCCBr ZINC000147432262 EK For-Sale Reactive GNAI1 0 43 CCCCCCCCCC(=O)N1CCC[C@@H]1CCCBr ZINC000147432262 EK For-Sale Reactive GNAI3 0 44 CCCCCCCCCC(=O)N1CCC[C@@H]1CCCBr ZINC000147432262 EK For-Sale Reactive GNAO1 0 42 CCCCCCCCCC(=O)N1CCC[C@@H]1CCCBr ZINC000147432262 EK For-Sale Reactive CQSS 48 30 C[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)n1cccn1 ZINC000147432280 GD On-Demand Anodyne HTR4 35 41 C[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)n1cccn1 ZINC000147432280 GD On-Demand Anodyne CHRM5 19 42 C[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)n1cccn1 ZINC000147432280 GD On-Demand Anodyne EPHX2 17 42 C[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)n1cccn1 ZINC000147432280 GD On-Demand Anodyne TGM2 70 45 C[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)n1cccn1 ZINC000147432280 GD On-Demand Anodyne F13A1 71 45 Cc1ccc(F)c(-c2ccnc(N)n2)c1F ZINC000147432309 BE For-Sale Anodyne HRH4 0 41 Cc1ccc(F)c(-c2ccnc(N)n2)c1F ZINC000147432309 BE For-Sale Anodyne ROCK1 24 43 Cc1ccc(F)c(-c2ccnc(N)n2)c1F ZINC000147432309 BE For-Sale Anodyne MAP3K14 57 49 C[C@@H](CNc1ncc(C(F)(F)F)cc1Cl)CC(=O)O ZINC000147432399 CG For-Sale Anodyne TRPM8 40 37 C[C@@H](CNc1ncc(C(F)(F)F)cc1Cl)CC(=O)O ZINC000147432399 CG For-Sale Anodyne H9BT73_9POAL 0 44 COc1ccc(Br)c2c1CC[C@@]1(C2)NC(=O)NC1=O ZINC000147432426 ED For-Sale Anodyne PDE7A 20 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc2[nH]c(C)cc2c1 ZINC000147432465 DF On-Demand Anodyne HDAC10 42 35 COc1cc(OCC(=O)Nc2ccc(-c3cn4ccccc4n3)cc2)ccc1[N+](=O)[O-] ZINC000147432467 HH On-Demand Bother ADORA2B 40 38 CCCCCCCCCC(=O)N1CCC[C@H]1CCCBr ZINC000147432479 EK For-Sale Reactive PREP 22 41 CCCCCCCCCC(=O)N1CCC[C@H]1CCCBr ZINC000147432479 EK For-Sale Reactive GNAI1 0 43 CCCCCCCCCC(=O)N1CCC[C@H]1CCCBr ZINC000147432479 EK For-Sale Reactive GNAI3 0 44 CCCCCCCCCC(=O)N1CCC[C@H]1CCCBr ZINC000147432479 EK For-Sale Reactive GNAO1 0 42 CCCCCCCCCC(=O)N1CCC[C@H]1CCCBr ZINC000147432479 EK For-Sale Reactive CQSS 48 30 CC[C@H](NC(=O)N1CCC[C@H](C)[C@H]1C)C(=O)O ZINC000147432483 BD For-Sale Anodyne TRPC6 45 35 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(N4CCOCC4)nc3)ccc21 ZINC000147432571 GD On-Demand Anodyne PIK3CA 49 47 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(N4CCOCC4)nc3)ccc21 ZINC000147432571 GD On-Demand Anodyne MTOR 88 47 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(N4CCOCC4)nc3)ccc21 ZINC000147432571 GD On-Demand Anodyne PIK3CG 41 41 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(N4CCOCC4)nc3)ccc21 ZINC000147432571 GD On-Demand Anodyne PIK3CB 34 44 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(N4CCOCC4)nc3)ccc21 ZINC000147432571 GD On-Demand Anodyne DGAT1 45 48 O=C(CNC(=O)C1CC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147432596 GC On-Demand Anodyne EPHX2 40 54 O=C(CNC(=O)C1CC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147432596 GC On-Demand Anodyne TGM2 78 46 O=C(CNC(=O)C1CC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147432596 GC On-Demand Anodyne F13A1 76 46 O=C(CNC(=O)C1CC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147432596 GC On-Demand Anodyne SFRP1 41 39 O=C(CNC(=O)C1CC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147432596 GC On-Demand Anodyne NAMPT 31 41 C[C@H](CNc1ccc(C(N)=O)cc1)CC(=O)O ZINC000147432598 BD For-Sale Anodyne ACR 43 35 C[C@H](CNc1ccc(C(N)=O)cc1)CC(=O)O ZINC000147432598 BD For-Sale Anodyne PARP10 0 40 CCOC(=O)c1cc2cc(C(F)(F)F)ccc2o1 ZINC000147432628 CH For-Sale Anodyne PDGFRB 17 41 COc1ccc(Br)c2c1CC[C@]1(C2)NC(=O)NC1=O ZINC000147432653 ED For-Sale Anodyne PDE7A 20 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc2[nH]c(C)cc2c1 ZINC000147432682 DF On-Demand Anodyne HDAC10 42 35 CC[C@H](NC(=O)N1CCC[C@@H](C)[C@H]1C)C(=O)O ZINC000147432726 BD For-Sale Anodyne TRPC6 45 35 CNc1cc(Oc2ccc(Br)cc2Cl)nc(N)n1 ZINC000147432727 EG For-Sale Anodyne AGPAT2 64 43 CC(C)c1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147432760 EJ For-Sale Reactive UL80 15 42 CC(C)c1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147432760 EJ For-Sale Reactive L3MBTL3 43 34 N#CCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147432814 GF On-Demand Mild DRD4 40 32 N#CCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147432814 GF On-Demand Mild ACHE 15 41 N#CCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147432814 GF On-Demand Mild TRY2_BOVIN 44 38 N#CCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147432814 GF On-Demand Mild TGM2 61 45 N#CCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147432814 GF On-Demand Mild ST14 76 36 N#CCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147432814 GF On-Demand Mild CACNA1I 63 41 N#CCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147432814 GF On-Demand Mild F13A1 40 45 N#CCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147432814 GF On-Demand Mild AKR1C3 59 39 N#CCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147432814 GF On-Demand Mild NAMPT 40 41 N#CCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147432814 GF On-Demand Mild TMPRSS6 56 33 C[C@@H](CNc1ccc(C(N)=O)cc1)CC(=O)O ZINC000147432817 BD For-Sale Anodyne ACR 43 35 C[C@@H](CNc1ccc(C(N)=O)cc1)CC(=O)O ZINC000147432817 BD For-Sale Anodyne PARP10 0 40 CCNc1ccc(C(=O)NCC2(N(C)C)CCCC2)cc1 ZINC000147432830 CF For-Sale Anodyne SLC6A5 17 50 CCCC[C@@H](CC)C(=O)NCC1(C(=O)O)CCC1 ZINC000147432841 CF On-Demand Anodyne SLC22A20 0 45 Cc1cc(CNC(=O)[C@@H](C)Cc2cccc(F)c2)ccc1F ZINC000147432908 DH On-Demand Anodyne ANPEP 27 52 Cc1cc(CNC(=O)[C@@H](C)Cc2cccc(F)c2)ccc1F ZINC000147432908 DH On-Demand Anodyne PAPA1_CARPA 15 41 Cc1cc(CNC(=O)[C@@H](C)Cc2cccc(F)c2)ccc1F ZINC000147432908 DH On-Demand Anodyne CTSL 18 41 Cc1cc(CNC(=O)[C@@H](C)Cc2cccc(F)c2)ccc1F ZINC000147432908 DH On-Demand Anodyne CPA1 15 40 Cc1cc(CNC(=O)[C@@H](C)Cc2cccc(F)c2)ccc1F ZINC000147432908 DH On-Demand Anodyne CTSS 15 41 Cc1cc(CNC(=O)[C@@H](C)Cc2cccc(F)c2)ccc1F ZINC000147432908 DH On-Demand Anodyne ACE2 44 33 Cc1cc(CNC(=O)[C@@H](C)Cc2cccc(F)c2)ccc1F ZINC000147432908 DH On-Demand Anodyne LEF 115 47 Cc1cc(CNC(=O)[C@@H](C)Cc2cccc(F)c2)ccc1F ZINC000147432908 DH On-Demand Anodyne CARM1 51 35 CN(C(=O)CC1(CN)CCC1)c1ccccc1 ZINC000147432962 BE For-Sale Anodyne CACNA2D1 42 45 CC(C)c1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147432968 EJ For-Sale Reactive UL80 15 42 CC(C)c1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147432968 EJ For-Sale Reactive L3MBTL3 43 34 O=C(O)Cc1sc(-c2cncs2)nc1-c1ccccc1 ZINC000147433008 DH For-Sale Anodyne PTGDR2 58 49 CC(C)CS(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147433032 HD On-Demand Anodyne HTR4 41 39 CC(C)CS(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147433032 HD On-Demand Anodyne CHRM5 24 43 CC(C)CS(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147433032 HD On-Demand Anodyne MMP13 22 40 CC(C)CS(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147433032 HD On-Demand Anodyne CAPN1 22 40 CC(C)CS(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147433032 HD On-Demand Anodyne EPHX2 24 43 CC(C)CS(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147433032 HD On-Demand Anodyne TGM2 85 48 CC(C)CS(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147433032 HD On-Demand Anodyne MMP1 18 40 CC(C)CS(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147433032 HD On-Demand Anodyne CACNA1I 45 34 CC(C)CS(=O)(=O)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147433032 HD On-Demand Anodyne F13A1 100 48 CCCC[C@H](CC)C(=O)NCC1(C(=O)O)CCC1 ZINC000147433046 CF On-Demand Anodyne SLC22A20 0 45 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1c(Cl)cccc1Cl ZINC000147433057 EG On-Demand Anodyne CCKAR 49 50 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1c(Cl)cccc1Cl ZINC000147433057 EG On-Demand Anodyne CCR3 29 46 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1c(Cl)cccc1Cl ZINC000147433057 EG On-Demand Anodyne CDC25B 21 48 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1c(Cl)cccc1Cl ZINC000147433057 EG On-Demand Anodyne CCKBR 35 42 O=C(N[C@H](Cc1ccccc1)C(=O)O)c1c(Cl)cccc1Cl ZINC000147433057 EG On-Demand Anodyne SMO 15 41 Cc1cc(CNC(=O)[C@H](C)Cc2cccc(F)c2)ccc1F ZINC000147433141 DH On-Demand Anodyne ANPEP 27 52 Cc1cc(CNC(=O)[C@H](C)Cc2cccc(F)c2)ccc1F ZINC000147433141 DH On-Demand Anodyne PAPA1_CARPA 15 41 Cc1cc(CNC(=O)[C@H](C)Cc2cccc(F)c2)ccc1F ZINC000147433141 DH On-Demand Anodyne CTSL 18 41 Cc1cc(CNC(=O)[C@H](C)Cc2cccc(F)c2)ccc1F ZINC000147433141 DH On-Demand Anodyne CPA1 15 40 Cc1cc(CNC(=O)[C@H](C)Cc2cccc(F)c2)ccc1F ZINC000147433141 DH On-Demand Anodyne CTSS 15 41 Cc1cc(CNC(=O)[C@H](C)Cc2cccc(F)c2)ccc1F ZINC000147433141 DH On-Demand Anodyne ACE2 44 33 Cc1cc(CNC(=O)[C@H](C)Cc2cccc(F)c2)ccc1F ZINC000147433141 DH On-Demand Anodyne LEF 115 47 Cc1cc(CNC(=O)[C@H](C)Cc2cccc(F)c2)ccc1F ZINC000147433141 DH On-Demand Anodyne CARM1 51 35 CC[C@@H](N)C(=O)N1C[C@H](CC(=O)O)c2ccccc21 ZINC000147433143 CD For-Sale Anodyne TPP2 62 41 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433162 FE On-Demand Anodyne CTSK 18 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433162 FE On-Demand Anodyne F2R 17 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433162 FE On-Demand Anodyne ROCK2 27 41 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433162 FE On-Demand Anodyne HDAC1 22 42 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433162 FE On-Demand Anodyne HDAC2 20 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433162 FE On-Demand Anodyne HDAC11 49 35 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433162 FE On-Demand Anodyne KCNK3 117 51 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433162 FE On-Demand Anodyne KCNK9 74 38 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne HTR2A 17 42 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne P2RY12 37 41 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne KIT 16 42 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne LCK 33 43 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne RAF1 20 41 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne KDR 38 42 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne NPY5R 18 44 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne MST1R 57 47 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne MET 49 39 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne MTTP 43 35 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne CSF1R 15 40 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne BTK 28 43 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne BRAF 32 41 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne SCD1 19 41 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne SCD 23 41 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne ENPP1 71 35 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne KCNK3 62 44 CCOc1ccc(NC(=O)c2cnn(-c3cccc(C(F)(F)F)c3)c2C)cc1OC ZINC000147433181 HJ On-Demand Anodyne KCNK9 51 44 O=C(CNc1ccc(Cl)cc1Br)Nc1ccccc1Cl ZINC000147433187 FJ On-Demand Anodyne CA2 18 40 O=C(CNc1ccc(Cl)cc1Br)Nc1ccccc1Cl ZINC000147433187 FJ On-Demand Anodyne CXCL8 23 41 O=C(CNc1ccc(Cl)cc1Br)Nc1ccccc1Cl ZINC000147433187 FJ On-Demand Anodyne CA1 20 42 O=C(CNc1ccc(Cl)cc1Br)Nc1ccccc1Cl ZINC000147433187 FJ On-Demand Anodyne CA5B 22 40 O=C(CNc1ccc(Cl)cc1Br)Nc1ccccc1Cl ZINC000147433187 FJ On-Demand Anodyne CA4 24 40 O=C(CNc1ccc(Cl)cc1Br)Nc1ccccc1Cl ZINC000147433187 FJ On-Demand Anodyne CA5A 25 40 C[C@H](F)c1ccccc1C[C@H](N)C(=O)O ZINC000147433228 BD For-Sale Anodyne IDO1 17 48 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(C(=O)N3CCCC3)c2)C1 ZINC000147433233 HE On-Demand Anodyne L3MBTL3 42 38 O=c1cc(-c2ccccc2)nc(-c2cncs2)[nH]1 ZINC000147433242 CF For-Sale Anodyne XDH 27 52 Cc1cc(C(=O)Nc2nc3c(s2)CCC3)cc([N+](=O)[O-])c1 ZINC000147433250 DG On-Demand Bother SLC27A1 23 41 CNc1ccc(C)cc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147433272 CF For-Sale Anodyne SLC6A5 15 43 CNc1ccc(C)cc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147433272 CF For-Sale Anodyne HCN1 44 35 COc1cccc(CC(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147433298 EG For-Sale Reactive FKBP1A 45 43 COc1cccc(CC(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147433298 EG For-Sale Reactive OPRM1 0 44 COc1cccc(CC(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147433298 EG For-Sale Reactive OPRK1 35 42 COc1cccc(CC(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147433298 EG For-Sale Reactive SLC18A2 24 43 COc1cccc(CC(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147433298 EG For-Sale Reactive SIGMAR1 16 47 COc1cccc(CC(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147433298 EG For-Sale Reactive CHRNA10 43 42 COc1cccc(CC(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147433298 EG For-Sale Reactive FAP 0 44 COc1cccc(CC(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147433298 EG For-Sale Reactive ACKR3 62 32 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@@H]1[N+](=O)[O-] ZINC000147433302 FC On-Demand Bother MMP3 16 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@@H]1[N+](=O)[O-] ZINC000147433302 FC On-Demand Bother EPHX2 19 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@@H]1[N+](=O)[O-] ZINC000147433302 FC On-Demand Bother TGM2 67 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@@H]1[N+](=O)[O-] ZINC000147433302 FC On-Demand Bother MMP7 23 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@@H]1[N+](=O)[O-] ZINC000147433302 FC On-Demand Bother F13A1 90 46 C[C@H]1CN(C(=O)CC2(CN)CCC2)C[C@@H](C)O1 ZINC000147433315 BD For-Sale Anodyne CACNA2D1 33 42 Cc1cnc(-c2ccn3c(-c4cccc(NC(=O)NCC(F)(F)F)c4)cnc3c2)nc1 ZINC000147433341 II Annotated Anodyne GYRB 0 41 CC[C@@H](N)C(=O)N1C[C@@H](CC(=O)O)c2ccccc21 ZINC000147433384 CD For-Sale Anodyne TPP2 62 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433391 FE On-Demand Anodyne CTSK 18 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433391 FE On-Demand Anodyne F2R 17 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433391 FE On-Demand Anodyne ROCK2 27 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433391 FE On-Demand Anodyne HDAC1 22 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433391 FE On-Demand Anodyne HDAC2 20 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433391 FE On-Demand Anodyne HDAC11 49 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433391 FE On-Demand Anodyne KCNK3 117 51 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(NC(=O)c2ccncc2)c1 ZINC000147433391 FE On-Demand Anodyne KCNK9 74 38 C[C@@H](F)c1ccccc1C[C@H](N)C(=O)O ZINC000147433432 BD For-Sale Anodyne IDO1 17 48 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne PTGS2 23 44 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne F10 16 43 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne CA1 17 44 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne CETP 0 47 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne S1PR4 15 40 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne MTNR1B 15 41 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne CA12 15 44 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne CA9 27 44 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne AKR1C3 26 41 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne AKR1C2 42 41 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne ENPP1 60 34 COc1ccc(NC(=O)CNc2ccc(Cl)cc2Br)cc1 ZINC000147433436 FI On-Demand Anodyne PSBA 0 40 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(C(=O)N3CCCC3)c2)C1 ZINC000147433464 HE On-Demand Anodyne L3MBTL3 42 38 COc1cccc(CC(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147433467 EG For-Sale Reactive FKBP1A 45 43 COc1cccc(CC(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147433467 EG For-Sale Reactive OPRM1 0 44 COc1cccc(CC(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147433467 EG For-Sale Reactive OPRK1 35 42 COc1cccc(CC(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147433467 EG For-Sale Reactive SLC18A2 24 43 COc1cccc(CC(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147433467 EG For-Sale Reactive SIGMAR1 16 47 COc1cccc(CC(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147433467 EG For-Sale Reactive CHRNA10 43 42 COc1cccc(CC(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147433467 EG For-Sale Reactive FAP 0 44 COc1cccc(CC(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147433467 EG For-Sale Reactive ACKR3 62 32 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive CYP19A1 25 56 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive CYP11B1 20 46 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive MAOA 61 39 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive MAOB 57 59 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive CA7 20 49 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive CYP11B2 16 46 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive CA14 15 55 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive MTNR1A 42 38 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive HSD17B3 24 49 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive CA12 15 55 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive KDM1A 15 40 COc1ccc2c(CCBr)cc(=O)oc2c1 ZINC000147433481 CF For-Sale Reactive SLC22A12 20 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@@H]1[N+](=O)[O-] ZINC000147433531 FC On-Demand Bother MMP3 16 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@@H]1[N+](=O)[O-] ZINC000147433531 FC On-Demand Bother EPHX2 19 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@@H]1[N+](=O)[O-] ZINC000147433531 FC On-Demand Bother TGM2 67 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@@H]1[N+](=O)[O-] ZINC000147433531 FC On-Demand Bother MMP7 23 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@@H]1[N+](=O)[O-] ZINC000147433531 FC On-Demand Bother F13A1 90 46 C[C@H]1CN(C(=O)CC2(CN)CCC2)C[C@H](C)O1 ZINC000147433570 BD For-Sale Anodyne CACNA2D1 33 42 C[C@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433608 BD For-Sale Anodyne CACNA2D1 61 51 C[C@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433608 BD For-Sale Anodyne MME 47 35 C[C@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433608 BD For-Sale Anodyne ANPEP 73 36 C[C@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433608 BD For-Sale Anodyne TPH1 63 35 C[C@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433608 BD For-Sale Anodyne ACE2 56 35 C[C@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433608 BD For-Sale Anodyne GRIK1 46 37 C[C@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433608 BD For-Sale Anodyne LAP3 42 36 C[C@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433608 BD For-Sale Anodyne KIF11 41 41 C[C@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433608 BD For-Sale Anodyne IDO1 17 48 CNC[C@@H](O)c1c(F)ccc(C)c1F ZINC000147433640 BD For-Sale Anodyne NMUR2 0 42 CCCNC(=O)c1cccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)c1 ZINC000147433650 HE On-Demand Anodyne DRD4 42 32 O=C(CNc1ccc(Cl)cc1Br)Nc1ccccc1F ZINC000147433652 FI On-Demand Anodyne CA1 20 41 O=C(CNc1ccc(Cl)cc1Br)Nc1ccccc1F ZINC000147433652 FI On-Demand Anodyne CA4 23 40 COCCNC(=O)c1ccc(NC(=O)c2ccccc2OCCN(C)C)cc1Cl ZINC000147433662 HF On-Demand Anodyne GRM4 42 43 COCCNC(=O)c1ccc(NC(=O)c2ccccc2OCCN(C)C)cc1Cl ZINC000147433662 HF On-Demand Anodyne BRAF 19 41 COCCNC(=O)c1ccc(NC(=O)c2ccccc2OCCN(C)C)cc1Cl ZINC000147433662 HF On-Demand Anodyne NR2E3 52 34 COCCNC(=O)c1ccc(NC(=O)c2ccccc2OCCN(C)C)cc1Cl ZINC000147433662 HF On-Demand Anodyne KCNK3 58 44 COCCNC(=O)c1ccc(NC(=O)c2ccccc2OCCN(C)C)cc1Cl ZINC000147433662 HF On-Demand Anodyne KCNK9 58 44 CCNc1ncnc(Oc2ccc(Br)cc2Cl)c1CC ZINC000147433671 FJ For-Sale Anodyne PDE6A 42 34 O=c1[nH]c(-c2cncs2)nc2c1CCCCC2 ZINC000147433679 BE For-Sale Anodyne TNKS2 20 50 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@H]1[N+](=O)[O-] ZINC000147433711 FC On-Demand Bother MMP3 16 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@H]1[N+](=O)[O-] ZINC000147433711 FC On-Demand Bother EPHX2 19 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@H]1[N+](=O)[O-] ZINC000147433711 FC On-Demand Bother TGM2 67 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@H]1[N+](=O)[O-] ZINC000147433711 FC On-Demand Bother MMP7 23 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@H]1[N+](=O)[O-] ZINC000147433711 FC On-Demand Bother F13A1 90 46 C[C@@H]1CN(C(=O)CC2(CN)CCC2)C[C@@H](C)O1 ZINC000147433747 BD For-Sale Anodyne CACNA2D1 33 42 O=S(=O)(c1cc(Cl)ccc1Cl)N1CCN(CCBr)CC1 ZINC000147433786 HF For-Sale Reactive HRP1_PLAFA 65 34 CNC[C@H](O)c1c(F)ccc(C)c1F ZINC000147433830 BD For-Sale Anodyne NMUR2 0 42 CCCNC(=O)c1cccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)c1 ZINC000147433856 HE On-Demand Anodyne DRD4 42 32 C[C@@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433857 BD For-Sale Anodyne CACNA2D1 61 51 C[C@@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433857 BD For-Sale Anodyne KIF11 41 41 C[C@@H](F)c1ccccc1C[C@@H](N)C(=O)O ZINC000147433857 BD For-Sale Anodyne IDO1 17 48 CC(C)NC(=O)c1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147433862 HE On-Demand Bother CA2 16 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@H]1[N+](=O)[O-] ZINC000147433905 FC On-Demand Bother MMP3 16 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@H]1[N+](=O)[O-] ZINC000147433905 FC On-Demand Bother EPHX2 19 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@H]1[N+](=O)[O-] ZINC000147433905 FC On-Demand Bother TGM2 67 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@H]1[N+](=O)[O-] ZINC000147433905 FC On-Demand Bother MMP7 23 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@H]1[N+](=O)[O-] ZINC000147433905 FC On-Demand Bother F13A1 90 46 CCCNc1ncnc(Oc2ccc(Br)cc2Cl)c1C ZINC000147433912 FJ For-Sale Anodyne HTT 0 51 Cc1cc(C)c(O)c(C(=O)O)c1O ZINC000147434058 AD For-Sale Anodyne AKR1C2 52 34 Cc1cc(C)c(O)c(C(=O)O)c1O ZINC000147434058 AD For-Sale Anodyne AKR1C1 56 34 C[C@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434083 BD For-Sale Anodyne OPRM1 32 48 C[C@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434083 BD For-Sale Anodyne OPRD1 37 41 C[C@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434083 BD For-Sale Anodyne CACNA2D1 65 57 C[C@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434083 BD For-Sale Anodyne MME 25 49 C[C@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434083 BD For-Sale Anodyne ANPEP 64 33 C[C@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434083 BD For-Sale Anodyne TPH1 88 39 C[C@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434083 BD For-Sale Anodyne YARS 34 41 C[C@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434083 BD For-Sale Anodyne LAP3 43 39 C[C@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434083 BD For-Sale Anodyne CTSC 15 40 C[C@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434083 BD For-Sale Anodyne SLC1A2 44 35 C[C@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434083 BD For-Sale Anodyne AMP1_PLAFQ 40 35 O=C(NCC1(C(=O)O)CCC1)c1cc(Cl)ccn1 ZINC000147434090 CD On-Demand Anodyne GRM4 19 40 CC(C)NC(=O)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1 ZINC000147434110 FG On-Demand Anodyne PRNP 55 35 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cnn1C(C)(C)C ZINC000147434137 HF On-Demand Anodyne HTR4 62 38 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cnn1C(C)(C)C ZINC000147434137 HF On-Demand Anodyne ACACB 25 40 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cnn1C(C)(C)C ZINC000147434137 HF On-Demand Anodyne TGM2 64 42 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cnn1C(C)(C)C ZINC000147434137 HF On-Demand Anodyne CACNA1I 60 37 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cnn1C(C)(C)C ZINC000147434137 HF On-Demand Anodyne F13A1 57 42 Nc1ncc(Cl)c(Oc2ccc(Br)cc2Cl)n1 ZINC000147434159 EH For-Sale Anodyne P2RX2 40 36 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2CCc2ccccc2)cc1 ZINC000147434211 FF On-Demand Anodyne F2 15 40 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2CCc2ccccc2)cc1 ZINC000147434211 FF On-Demand Anodyne FKBP1A 43 39 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2CCc2ccccc2)cc1 ZINC000147434211 FF On-Demand Anodyne SLC18A2 55 42 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2CCc2ccccc2)cc1 ZINC000147434211 FF On-Demand Anodyne CHEK2 38 45 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2CCc2ccccc2)cc1 ZINC000147434211 FF On-Demand Anodyne CPT1A 129 52 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2CCc2ccccc2)cc1 ZINC000147434211 FF On-Demand Anodyne CPT2 52 40 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2CCc2ccccc2)cc1 ZINC000147434211 FF On-Demand Anodyne PREP 74 40 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2CCc2ccccc2)cc1 ZINC000147434211 FF On-Demand Anodyne PLA2G4B 31 41 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2CCc2ccccc2)cc1 ZINC000147434211 FF On-Demand Anodyne TMPRSS11D 52 33 NC(=O)c1ccc(OCC(=O)N2CCC[C@H]2CCc2ccccc2)cc1 ZINC000147434211 FF On-Demand Anodyne ACKR3 46 35 O=C(c1ccc(S(=O)(=O)Nc2nccs2)cc1)N1CCC[C@H](Oc2ccccc2)C1 ZINC000147434212 IH On-Demand Anodyne GCK 20 42 O=C(c1ccc(S(=O)(=O)Nc2nccs2)cc1)N1CCC[C@H](Oc2ccccc2)C1 ZINC000147434212 IH On-Demand Anodyne SFRP1 55 36 CNc1ncc(Br)cc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147434254 FE For-Sale Anodyne SLC6A5 15 43 COc1cc(C(=O)N2CCC3(CC2)OCCO3)ccc1F ZINC000147434294 CD On-Demand Anodyne CHRM5 0 40 COc1cc(C(=O)N2CCC3(CC2)OCCO3)ccc1F ZINC000147434294 CD On-Demand Anodyne SCN9A 0 44 COc1cc(C(=O)N2CCC3(CC2)OCCO3)ccc1F ZINC000147434294 CD On-Demand Anodyne SCN5A 24 44 COc1cc(C(=O)N2CCC3(CC2)OCCO3)ccc1F ZINC000147434294 CD On-Demand Anodyne CCR8 25 40 C[C@@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434299 BD For-Sale Anodyne OPRM1 32 48 C[C@@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434299 BD For-Sale Anodyne OPRD1 37 41 C[C@@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434299 BD For-Sale Anodyne CACNA2D1 65 57 C[C@@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434299 BD For-Sale Anodyne MME 25 49 C[C@@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434299 BD For-Sale Anodyne ANPEP 64 33 C[C@@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434299 BD For-Sale Anodyne TPH1 88 39 C[C@@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434299 BD For-Sale Anodyne YARS 34 41 C[C@@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434299 BD For-Sale Anodyne LAP3 43 39 C[C@@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434299 BD For-Sale Anodyne CTSC 15 40 C[C@@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434299 BD For-Sale Anodyne SLC1A2 44 35 C[C@@H](F)c1cccc(C[C@H](N)C(=O)O)c1 ZINC000147434299 BD For-Sale Anodyne AMP1_PLAFQ 40 35 O=C(C[C@@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434372 FD On-Demand Anodyne OXTR 27 41 O=C(C[C@@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434372 FD On-Demand Anodyne EPHX2 18 45 O=C(C[C@@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434372 FD On-Demand Anodyne TGM2 61 43 O=C(C[C@@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434372 FD On-Demand Anodyne F13A1 67 43 C[C@H](CNc1ccnc2ccccc12)CC(=O)O ZINC000147434378 BF On-Demand Anodyne DNMT1 32 42 C[C@H](CNc1ccnc2ccccc12)CC(=O)O ZINC000147434378 BF On-Demand Anodyne KCNN3 24 42 C[C@H](CNc1ccnc2ccccc12)CC(=O)O ZINC000147434378 BF On-Demand Anodyne HNMT 45 42 O=C(NCC1(C(=O)O)CCC1)c1ccc(Cl)cc1 ZINC000147434386 CE On-Demand Anodyne SLC6A9 21 44 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2CCc2ccccc2)cc1 ZINC000147434397 FF On-Demand Anodyne F2 15 40 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2CCc2ccccc2)cc1 ZINC000147434397 FF On-Demand Anodyne FKBP1A 43 39 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2CCc2ccccc2)cc1 ZINC000147434397 FF On-Demand Anodyne SLC18A2 55 42 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2CCc2ccccc2)cc1 ZINC000147434397 FF On-Demand Anodyne CHEK2 38 45 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2CCc2ccccc2)cc1 ZINC000147434397 FF On-Demand Anodyne COLA 154 57 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2CCc2ccccc2)cc1 ZINC000147434397 FF On-Demand Anodyne CPT1A 129 52 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2CCc2ccccc2)cc1 ZINC000147434397 FF On-Demand Anodyne CPT2 52 40 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2CCc2ccccc2)cc1 ZINC000147434397 FF On-Demand Anodyne PREP 74 40 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2CCc2ccccc2)cc1 ZINC000147434397 FF On-Demand Anodyne PLA2G4B 31 41 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2CCc2ccccc2)cc1 ZINC000147434397 FF On-Demand Anodyne TMPRSS11D 52 33 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H]2CCc2ccccc2)cc1 ZINC000147434397 FF On-Demand Anodyne ACKR3 46 35 O=C(c1ccc(S(=O)(=O)Nc2nccs2)cc1)N1CCC[C@@H](Oc2ccccc2)C1 ZINC000147434429 IH On-Demand Anodyne GCK 20 42 O=C(c1ccc(S(=O)(=O)Nc2nccs2)cc1)N1CCC[C@@H](Oc2ccccc2)C1 ZINC000147434429 IH On-Demand Anodyne SFRP1 55 36 COc1ccc2c(c1)OC[C@H](C(=O)NCC1(c3ccc(F)cc3)CCOCC1)C2 ZINC000147434465 GG On-Demand Anodyne MTNR1A 23 42 COc1ccc2c(c1)OC[C@H](C(=O)NCC1(c3ccc(F)cc3)CCOCC1)C2 ZINC000147434465 GG On-Demand Anodyne MTNR1B 18 42 C[C@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434472 BD For-Sale Anodyne OPRM1 32 48 C[C@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434472 BD For-Sale Anodyne OPRD1 37 41 C[C@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434472 BD For-Sale Anodyne CACNA2D1 65 57 C[C@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434472 BD For-Sale Anodyne MME 25 49 C[C@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434472 BD For-Sale Anodyne ANPEP 64 33 C[C@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434472 BD For-Sale Anodyne TPH1 88 39 C[C@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434472 BD For-Sale Anodyne YARS 34 41 C[C@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434472 BD For-Sale Anodyne LAP3 43 39 C[C@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434472 BD For-Sale Anodyne CTSC 15 40 C[C@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434472 BD For-Sale Anodyne SLC1A2 44 35 C[C@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434472 BD For-Sale Anodyne AMP1_PLAFQ 40 35 O=c1[nH]c(-c2cncs2)nc(-c2ccccc2)c1I ZINC000147434500 GG For-Sale Anodyne RAF1 24 40 CCN(CC)CCNC(=O)CC1(CN)CCC1 ZINC000147434560 BC For-Sale Anodyne CACNA2D1 0 41 CN(C)C(=O)c1cccc(NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)c1 ZINC000147434572 FE On-Demand Anodyne EPHX2 22 44 CN(C)C(=O)c1cccc(NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)c1 ZINC000147434572 FE On-Demand Anodyne KCNK3 88 43 O=C(C[C@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434581 FD On-Demand Anodyne OXTR 27 41 O=C(C[C@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434581 FD On-Demand Anodyne EPHX2 18 45 O=C(C[C@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434581 FD On-Demand Anodyne TGM2 61 43 O=C(C[C@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434581 FD On-Demand Anodyne F13A1 67 43 C[C@@H](CNc1ccnc2ccccc12)CC(=O)O ZINC000147434589 BF On-Demand Anodyne DNMT1 32 42 C[C@@H](CNc1ccnc2ccccc12)CC(=O)O ZINC000147434589 BF On-Demand Anodyne KCNN3 24 42 C[C@@H](CNc1ccnc2ccccc12)CC(=O)O ZINC000147434589 BF On-Demand Anodyne HNMT 45 42 C[C@@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434670 BD For-Sale Anodyne OPRM1 32 48 C[C@@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434670 BD For-Sale Anodyne OPRD1 37 41 C[C@@H](F)c1cccc(C[C@@H](N)C(=O)O)c1 ZINC000147434670 BD For-Sale Anodyne CACNA2D1 65 57 COc1ccc2c(c1)OC[C@@H](C(=O)NCC1(c3ccc(F)cc3)CCOCC1)C2 ZINC000147434672 GG On-Demand Anodyne MTNR1A 23 42 COc1ccc2c(c1)OC[C@@H](C(=O)NCC1(c3ccc(F)cc3)CCOCC1)C2 ZINC000147434672 GG On-Demand Anodyne MTNR1B 18 42 Cc1ncsc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434796 GE On-Demand Anodyne HTR4 51 36 Cc1ncsc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434796 GE On-Demand Anodyne TGM2 56 42 Cc1ncsc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434796 GE On-Demand Anodyne CACNA1I 47 35 Cc1ncsc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147434796 GE On-Demand Anodyne F13A1 57 42 C[C@H](NC(=O)CC1(CN)CCC1)c1ccccc1 ZINC000147434834 BE For-Sale Anodyne CACNA2D1 32 41 C[C@H](NC(=O)CC1(CN)CCC1)c1ccccc1 ZINC000147434834 BE For-Sale Anodyne CTSK 39 52 C[C@H](NC(=O)CC1(CN)CCC1)c1ccccc1 ZINC000147434834 BE For-Sale Anodyne F7 16 42 Cc1ccc(F)c([C@H](O)CNC(C)C)c1F ZINC000147434846 BE For-Sale Anodyne ADRB2 24 41 Cc1ccc(F)c([C@H](O)CNC(C)C)c1F ZINC000147434846 BE For-Sale Anodyne ADRB1 0 49 CCCCCCCC(=O)NCC1(C(=O)O)CCC1 ZINC000147434944 CF On-Demand Mild FABP2 0 40 CCCCCCCC(=O)NCC1(C(=O)O)CCC1 ZINC000147434944 CF On-Demand Mild FABP4 15 40 CCCCCCCC(=O)NCC1(C(=O)O)CCC1 ZINC000147434944 CF On-Demand Mild DNM1 0 44 CCCCCCCC(=O)NCC1(C(=O)O)CCC1 ZINC000147434944 CF On-Demand Mild FAAH 0 51 CCCCCCCC(=O)NCC1(C(=O)O)CCC1 ZINC000147434944 CF On-Demand Mild EPHX2 22 43 CCCCCCCC(=O)NCC1(C(=O)O)CCC1 ZINC000147434944 CF On-Demand Mild SLC22A20 0 40 CCCCCCCC(=O)NCC1(C(=O)O)CCC1 ZINC000147434944 CF On-Demand Mild LASR 40 35 CCCCCCCC(=O)NCC1(C(=O)O)CCC1 ZINC000147434944 CF On-Demand Mild NOD1 55 38 CCCCCCCC(=O)NCC1(C(=O)O)CCC1 ZINC000147434944 CF On-Demand Mild CQSS 53 33 C[C@@H](NC(=O)CC1(CN)CCC1)c1ccccc1 ZINC000147435007 BE For-Sale Anodyne CACNA2D1 32 41 C[C@@H](NC(=O)CC1(CN)CCC1)c1ccccc1 ZINC000147435007 BE For-Sale Anodyne CTSK 39 52 C[C@@H](NC(=O)CC1(CN)CCC1)c1ccccc1 ZINC000147435007 BE For-Sale Anodyne F7 16 42 Cc1ccc(F)c([C@@H](O)CNC(C)C)c1F ZINC000147435028 BE For-Sale Anodyne ADRB2 24 41 Cc1ccc(F)c([C@@H](O)CNC(C)C)c1F ZINC000147435028 BE For-Sale Anodyne ADRB1 0 49 CCc1ccccc1CN1CCC1 ZINC000147435045 AE For-Sale Anodyne SIGMAR1 21 43 COc1cc(OC)c(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)cc1Cl ZINC000147435242 HF On-Demand Anodyne HTR4 38 48 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne POLA1 40 51 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne P2RY6 206 87 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne POLB 41 34 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne P2RX4 38 43 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne P2RX1 52 44 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne P2RY4 211 98 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne P2RY1 34 73 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne ITPR1 33 55 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne P2RY2 243 98 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne FIMH 51 33 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne RNASE1 78 54 O=c1ccn([C@@H]2O[C@H](CO[P@@](=O)(O)O[P@@](=O)(O)O[C@H]3O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]3O)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147435262 KA For-Sale Anodyne GPR17 60 39 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)N3CCC(C)CC3)cc2C)c1 ZINC000147435314 HI On-Demand Bother TAAR1 24 47 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)N3CCC(C)CC3)cc2C)c1 ZINC000147435314 HI On-Demand Bother L3MBTL3 44 43 COc1cc(OC)c(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)cc1Cl ZINC000147435419 HF On-Demand Anodyne HTR4 38 48 CNc1c(F)cccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147435468 CE For-Sale Anodyne SLC6A5 15 42 CNc1c(F)cccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147435468 CE For-Sale Anodyne HCN1 74 37 CNc1c(F)cccc1C(=O)NCC1(N(C)C)CCCC1 ZINC000147435468 CE For-Sale Anodyne HCN4 52 35 CCN(CC)[C@@H](C)CNC(=O)CNC(=O)c1c[nH]c2ccccc2c1=O ZINC000147435514 FD On-Demand Anodyne CFTR 43 51 C[C@H](CNc1nc2ccccc2s1)CC(=O)O ZINC000147435565 CF On-Demand Anodyne CSNK1D 26 51 C[C@H](CNc1nc2ccccc2s1)CC(=O)O ZINC000147435565 CF On-Demand Anodyne FABK 0 40 C[C@H](CNc1nc2ccccc2s1)CC(=O)O ZINC000147435565 CF On-Demand Anodyne TMPRSS6 51 36 CCc1ccc(C(=O)NCC2(C(=O)O)CCC2)cc1 ZINC000147435652 CE On-Demand Anodyne ECR 26 43 CCc1ccc(C(=O)NCC2(C(=O)O)CCC2)cc1 ZINC000147435652 CE On-Demand Anodyne E3UJZ5_SPOLI 22 46 CCN(CC)[C@H](C)CNC(=O)CNC(=O)c1c[nH]c2ccccc2c1=O ZINC000147435710 FD On-Demand Anodyne CFTR 36 42 COc1cc(OC)cc(C(=O)NCC(=O)N2CCN(CC(=O)NC(C)C)CC2)c1 ZINC000147435738 HC On-Demand Anodyne DRD4 50 39 C[C@@H](CNc1nc2ccccc2s1)CC(=O)O ZINC000147435796 CF On-Demand Anodyne CSNK1D 26 51 C[C@@H](CNc1nc2ccccc2s1)CC(=O)O ZINC000147435796 CF On-Demand Anodyne FABK 0 40 C[C@@H](CNc1nc2ccccc2s1)CC(=O)O ZINC000147435796 CF On-Demand Anodyne TMPRSS6 51 36 CCNc1cn2ccnc2c(Oc2ccc(Br)cc2Cl)n1 ZINC000147435800 FI For-Sale Anodyne HIVRT 0 44 Cc1cc(C)cc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147435966 CG For-Sale Anodyne ADRB2 51 45 Cc1cc(C)cc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147435966 CG For-Sale Anodyne ADRB1 53 45 Cc1cc(C)cc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147435966 CG For-Sale Anodyne ADRB3 42 43 C[C@@H]1CCCCCN1CCS(=O)(=O)c1cccc(C#N)c1 ZINC000147436030 DF On-Demand Mild HRH3 51 45 O=S(=O)(c1ccc(F)cc1F)N1CCN(CCBr)CC1 ZINC000147436046 FD For-Sale Reactive HTR2A 21 54 O=S(=O)(c1ccc(F)cc1F)N1CCN(CCBr)CC1 ZINC000147436046 FD For-Sale Reactive PKM 22 52 O=S(=O)(c1ccc(F)cc1F)N1CCN(CCBr)CC1 ZINC000147436046 FD For-Sale Reactive TRPV4 15 41 NC(=O)c1cc(NC(=O)c2ccc(Br)c(Cl)c2)ccc1Cl ZINC000147436064 GI On-Demand Anodyne MAOB 20 43 NC(=O)c1cc(NC(=O)c2ccc(Br)c(Cl)c2)ccc1Cl ZINC000147436064 GI On-Demand Anodyne PLAU 20 42 NC(=O)c1cc(NC(=O)c2ccc(Br)c(Cl)c2)ccc1Cl ZINC000147436064 GI On-Demand Anodyne CSF1R 21 50 NC(=O)c1cc(NC(=O)c2ccc(Br)c(Cl)c2)ccc1Cl ZINC000147436064 GI On-Demand Anodyne TAAR1 22 49 NC(=O)c1cc(NC(=O)c2ccc(Br)c(Cl)c2)ccc1Cl ZINC000147436064 GI On-Demand Anodyne SHH 48 40 NC(=O)c1cc(NC(=O)c2ccc(Br)c(Cl)c2)ccc1Cl ZINC000147436064 GI On-Demand Anodyne IMDH_CRYPV 19 41 NC(=O)c1cc(NC(=O)c2ccc(Br)c(Cl)c2)ccc1Cl ZINC000147436064 GI On-Demand Anodyne SENP1 0 40 NC(=O)c1cc(NC(=O)c2ccc(Br)c(Cl)c2)ccc1Cl ZINC000147436064 GI On-Demand Anodyne KCNK3 74 40 CCc1cccc(C)c1NC(=O)C1(N)CCC1 ZINC000147436100 BE For-Sale Anodyne S1PR4 0 41 CCc1cccc(C)c1NC(=O)C1(N)CCC1 ZINC000147436100 BE For-Sale Anodyne ACAT 0 42 CN(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccn1 ZINC000147436103 HD On-Demand Anodyne HTR4 46 35 CN(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccn1 ZINC000147436103 HD On-Demand Anodyne EPHX2 24 42 CN(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccn1 ZINC000147436103 HD On-Demand Anodyne TGM2 58 41 CN(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccn1 ZINC000147436103 HD On-Demand Anodyne CACNA1I 65 42 CN(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccn1 ZINC000147436103 HD On-Demand Anodyne F13A1 45 41 CN(C)c1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccn1 ZINC000147436103 HD On-Demand Anodyne NAMPT 52 41 NS(=O)(=O)c1cc(F)c(OCCN2CCCCC2)c(F)c1 ZINC000147436123 DD For-Sale Anodyne LTA4H 33 40 NS(=O)(=O)c1cc(F)c(OCCN2CCCCC2)c(F)c1 ZINC000147436123 DD For-Sale Anodyne HRH3 25 52 NS(=O)(=O)c1cc(F)c(OCCN2CCCCC2)c(F)c1 ZINC000147436123 DD For-Sale Anodyne PSMB2 49 39 NS(=O)(=O)c1cc(F)c(OCCN2CCCCC2)c(F)c1 ZINC000147436123 DD For-Sale Anodyne PSMB1 42 39 Cc1cc(C)cc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147436162 CG For-Sale Anodyne ADRB2 51 45 Cc1cc(C)cc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147436162 CG For-Sale Anodyne ADRB1 53 45 Cc1cc(C)cc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147436162 CG For-Sale Anodyne ADRB3 42 43 Oc1ccc(-c2nc(-c3ccc(Oc4ccc(C(F)(F)F)cc4)cc3)no2)cc1 ZINC000147436167 GK Annotated Anodyne S1PR1 20 40 C[C@H]1CCCCCN1CCS(=O)(=O)c1cccc(C#N)c1 ZINC000147436250 DF On-Demand Mild HRH3 51 45 CCNc1cc(Oc2ccc(C(N)=O)cc2)nc(N)n1 ZINC000147436258 CD For-Sale Anodyne TRY1_BOVIN 18 40 CCNc1cc(Oc2ccc(C(N)=O)cc2)nc(N)n1 ZINC000147436258 CD For-Sale Anodyne AGPAT2 19 43 Cc1ccc(Br)c(C(=O)Nc2ccc(Cl)c(C(N)=O)c2)c1 ZINC000147436283 FH On-Demand Anodyne F12 0 41 Cc1ccc(Br)c(C(=O)Nc2ccc(Cl)c(C(N)=O)c2)c1 ZINC000147436283 FH On-Demand Anodyne CSF1R 21 44 Cc1ccc(Br)c(C(=O)Nc2ccc(Cl)c(C(N)=O)c2)c1 ZINC000147436283 FH On-Demand Anodyne SHH 46 41 Cc1ccc(Br)c(C(=O)Nc2ccc(Cl)c(C(N)=O)c2)c1 ZINC000147436283 FH On-Demand Anodyne IMDH_CRYPV 17 41 Cc1ccc(Br)c(C(=O)Nc2ccc(Cl)c(C(N)=O)c2)c1 ZINC000147436283 FH On-Demand Anodyne KCNK3 57 42 Cc1ccc(Br)c(C(=O)Nc2ccc(Cl)c(C(N)=O)c2)c1 ZINC000147436283 FH On-Demand Anodyne KCNK9 60 37 CN(CC1CC1)C(=O)c1ccccc1NS(=O)(=O)c1ccc(F)c(F)c1 ZINC000147436284 GG On-Demand Anodyne PRTN3 60 38 CN(CC1CC1)C(=O)c1ccccc1NS(=O)(=O)c1ccc(F)c(F)c1 ZINC000147436284 GG On-Demand Anodyne LEF 48 37 CN(CC1CC1)C(=O)c1ccccc1NS(=O)(=O)c1ccc(F)c(F)c1 ZINC000147436284 GG On-Demand Anodyne LIMK2 36 44 CN(CC1CC1)C(=O)c1ccccc1NS(=O)(=O)c1ccc(F)c(F)c1 ZINC000147436284 GG On-Demand Anodyne WNT3 40 33 O=C([C@H]1Cc2ccccc2O1)N1CCC[C@@H]1CCCBr ZINC000147436345 EG For-Sale Reactive PREP 48 35 C[C@H](CNc1ncccc1C(N)=O)CC(=O)O ZINC000147436387 BC For-Sale Anodyne PARP1 0 40 CC(C)CCCCNC(=O)[C@H](N)CC(N)=O ZINC000147436402 BC For-Sale Anodyne GRIA1 41 38 CC(C)CCCCNC(=O)[C@H](N)CC(N)=O ZINC000147436402 BC For-Sale Anodyne DNPEP 0 40 CC(C)(C)c1cc(NC(=O)[C@@H]2C[C@@H](O)CN2CC2CCOCC2)on1 ZINC000147436415 FD Annotated Anodyne CNR2 16 51 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne ACE 29 58 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne SSTR2 32 44 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne OPRM1 17 54 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MME 49 56 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne EDNRB 62 46 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne EDNRA 48 56 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne TACR1 36 56 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MC4R 57 47 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne CTSB 25 47 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne CCKAR 133 52 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne CTSL 36 46 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne BRS3 36 59 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne TIMP3 15 54 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne NMBR 52 55 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MC3R 76 47 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MC5R 72 41 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MMP2 38 58 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MMP8 58 55 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne GRIA1 47 41 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MMP14 28 52 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne GRPR 84 42 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne ECE1 75 56 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne LNPEP 22 43 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne SSTR3 21 41 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MMP11 101 42 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne CCKBR 95 49 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne GHSR 68 52 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne CAPN1 21 52 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MMP9 37 55 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne CAPN2 22 41 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MC1R 110 47 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MMP7 29 55 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne MMP1 34 55 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne FPR1 28 49 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne NPR 58 54 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne ADAM12 17 52 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne KISS1R 91 43 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne ERAP2 47 43 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne PSMB8 29 44 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne TMPRSS6 17 43 CCN(CC)[C@@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436488 GF On-Demand Anodyne HPN 21 42 CNc1cccc(Oc2ccc(C(N)=O)cc2)c1[N+](=O)[O-] ZINC000147436490 CF For-Sale Bother SIRT2 38 42 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc2c(c1)n(C)c(=O)n2C ZINC000147436524 HF On-Demand Anodyne LCK 21 41 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc2c(c1)n(C)c(=O)n2C ZINC000147436524 HF On-Demand Anodyne PRNP 41 42 Cc1cc(N2CCN(C)CC2)ccc1NC(=O)Nc1ccc2c(c1)n(C)c(=O)n2C ZINC000147436524 HF On-Demand Anodyne FLT3 16 44 O=C([C@@H]1Cc2ccccc2O1)N1CCC[C@@H]1CCCBr ZINC000147436558 EG For-Sale Reactive PREP 48 35 C[C@@H](CNc1ncccc1C(N)=O)CC(=O)O ZINC000147436599 BC For-Sale Anodyne PARP1 0 40 CC(C)CCCCNC(=O)[C@@H](N)CC(N)=O ZINC000147436614 BC For-Sale Anodyne GRIA1 41 38 CC(C)CCCCNC(=O)[C@@H](N)CC(N)=O ZINC000147436614 BC For-Sale Anodyne DNPEP 0 40 O[C@@H](CNCCCn1cnc2ccccc21)COc1ccccc1 ZINC000147436628 EE On-Demand Anodyne ADRB2 59 49 O[C@@H](CNCCCn1cnc2ccccc21)COc1ccccc1 ZINC000147436628 EE On-Demand Anodyne ADRB1 63 46 O[C@@H](CNCCCn1cnc2ccccc21)COc1ccccc1 ZINC000147436628 EE On-Demand Anodyne GRIN1 15 40 O[C@@H](CNCCCn1cnc2ccccc21)COc1ccccc1 ZINC000147436628 EE On-Demand Anodyne ADRB3 58 46 CC[C@H](NC(=O)N1CCCN2CCC[C@H]2C1)C(=O)O ZINC000147436683 CC For-Sale Anodyne RIR1_HHV11 48 31 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne ACE 29 58 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne SSTR2 32 44 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne OPRM1 17 54 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MME 49 56 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne EDNRB 62 46 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne EDNRA 54 53 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne TACR1 36 56 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MC4R 57 47 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne CTSB 25 47 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne CCKAR 133 52 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne CTSL 42 46 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne BRS3 36 59 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne TIMP3 20 54 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne NMBR 52 55 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MC3R 76 47 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MC5R 72 41 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MMP2 38 58 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MMP8 58 55 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne GRIA1 49 41 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MMP14 28 52 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne GRPR 84 42 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne ECE1 75 56 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne REN 17 43 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne REN1 17 42 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne LNPEP 26 40 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne SSTR3 27 41 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MMP11 101 42 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne CCKBR 95 49 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne GHSR 72 52 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne CAPN1 21 52 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MMP9 37 55 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne CAPN2 22 41 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MC1R 110 47 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne ADAM9 51 52 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne CTSC 15 48 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MMP7 29 55 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne MMP1 34 55 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne FPR1 28 49 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne NPR 62 54 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne ADAM12 17 52 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne KISS1R 91 43 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne ERAP2 47 43 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne PSMB8 29 44 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne TMPRSS6 17 43 CCN(CC)[C@H](C)CNC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436691 GF On-Demand Anodyne HPN 21 42 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne NPY1R 22 41 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne KLK3 49 38 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne CTSK 32 48 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne NPFFR2 41 38 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne C3AR1 52 32 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne GRIA1 45 33 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne PCSK5 54 37 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne FURIN 59 37 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne CTSS 17 48 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne CTRB_BOVIN 46 34 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne POLG_WNV 75 34 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne QRFPR 42 40 CCCC[C@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436714 DE On-Demand Anodyne NPFFR1 56 38 Cc1ccc(F)c(CN2CCNCC2)c1F ZINC000147436729 BD For-Sale Anodyne CXCR4 21 41 O=C([C@H]1Cc2ccccc2O1)N1CCC[C@H]1CCCBr ZINC000147436772 EG For-Sale Reactive PREP 48 35 C[C@H](CNc1c([N+](=O)[O-])ccc(F)c1F)CC(=O)O ZINC000147436811 CE For-Sale Bother COLA 46 31 O[C@H](CNCCCn1cnc2ccccc21)COc1ccccc1 ZINC000147436815 EE On-Demand Anodyne ADRB2 59 49 O[C@H](CNCCCn1cnc2ccccc21)COc1ccccc1 ZINC000147436815 EE On-Demand Anodyne ADRB1 63 46 O[C@H](CNCCCn1cnc2ccccc21)COc1ccccc1 ZINC000147436815 EE On-Demand Anodyne GRIN1 15 40 O[C@H](CNCCCn1cnc2ccccc21)COc1ccccc1 ZINC000147436815 EE On-Demand Anodyne ADRB3 58 46 NS(=O)(=O)c1cc(F)c(OCC(=O)NC2CC2)c(F)c1 ZINC000147436817 DC For-Sale Anodyne CA2 20 40 NS(=O)(=O)c1cc(F)c(OCC(=O)NC2CC2)c(F)c1 ZINC000147436817 DC For-Sale Anodyne CA1 16 40 NS(=O)(=O)c1cc(F)c(OCC(=O)NC2CC2)c(F)c1 ZINC000147436817 DC For-Sale Anodyne CA7 29 40 NS(=O)(=O)c1cc(F)c(OCC(=O)NC2CC2)c(F)c1 ZINC000147436817 DC For-Sale Anodyne CA12 16 40 CC(C)CCCCNC(=O)c1ccc2nc(N)sc2c1 ZINC000147436824 CG For-Sale Anodyne LCK 26 42 CC(C)CCCCNC(=O)c1ccc2nc(N)sc2c1 ZINC000147436824 CG For-Sale Anodyne NMT1 18 43 CC(C)CCCCNC(=O)c1ccc2nc(N)sc2c1 ZINC000147436824 CG For-Sale Anodyne TMPRSS6 44 32 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne ACE 29 58 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne SSTR2 32 44 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne OPRM1 17 54 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MME 49 56 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne EDNRB 62 46 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne EDNRA 48 56 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne TACR1 36 56 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MC4R 57 47 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne CTSB 25 47 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne CCKAR 133 52 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne CTSL 36 46 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne BRS3 36 59 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne TIMP3 15 54 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne NMBR 52 55 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MC3R 76 47 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MC5R 72 41 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MMP2 38 58 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MMP8 58 55 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne GRIA1 47 41 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MMP14 28 52 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne GRPR 84 42 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne ECE1 75 56 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne LNPEP 22 43 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne SSTR3 21 41 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MMP11 101 42 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne CCKBR 95 49 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne GHSR 68 52 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne CAPN1 21 52 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MMP9 37 55 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne CAPN2 22 41 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MC1R 110 47 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MMP7 29 55 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne MMP1 34 55 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne FPR1 28 49 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne NPR 58 54 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne ADAM12 17 52 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne KISS1R 91 43 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne ERAP2 47 43 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne PSMB8 29 44 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne TMPRSS6 17 43 CCN(CC)[C@@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147436883 GF On-Demand Anodyne HPN 21 42 CC(C)(C)NS(=O)(=O)Cc1cccc(NC(=O)c2ccc3c(c2)COC3)c1 ZINC000147436908 GG On-Demand Anodyne TAAR1 44 39 CC(C)(C)NS(=O)(=O)Cc1cccc(NC(=O)c2ccc3c(c2)COC3)c1 ZINC000147436908 GG On-Demand Anodyne KCNK3 94 41 CC(C)(C)NS(=O)(=O)Cc1cccc(NC(=O)c2ccc3c(c2)COC3)c1 ZINC000147436908 GG On-Demand Anodyne KCNK9 47 38 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne NPY1R 22 41 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne KLK3 49 38 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne CTSK 32 48 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne NPFFR2 41 38 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne C3AR1 52 32 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne GRIA1 45 33 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne PCSK5 54 37 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne FURIN 59 37 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne CTSS 17 48 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne CTRB_BOVIN 46 34 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne POLG_WNV 75 34 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne QRFPR 42 40 CCCC[C@@H](NC(N)=O)C(=O)NCC(C)(C)c1ccccc1 ZINC000147436939 DE On-Demand Anodyne NPFFR1 56 38 Cn1c(=O)n(C)c2cc(NC(=O)Nc3nc(CN4CCOCC4)cs3)ccc21 ZINC000147436940 HD On-Demand Anodyne MTOR 70 35 CNc1cn2ccnc2c(Oc2ccc(C(N)=O)cc2)n1 ZINC000147436951 CD For-Sale Anodyne SYK 22 44 CNc1cn2ccnc2c(Oc2ccc(C(N)=O)cc2)n1 ZINC000147436951 CD For-Sale Anodyne HIVRT 0 40 Cc1c(O)cccc1C(=O)N1CCNCC1 ZINC000147436966 BC For-Sale Anodyne REN 43 42 COc1cccc(NC(=O)CNc2ccc(Cl)cc2Br)c1 ZINC000147436969 FI On-Demand Anodyne DRD4 40 33 COc1cccc(NC(=O)CNc2ccc(Cl)cc2Br)c1 ZINC000147436969 FI On-Demand Anodyne PTGS2 0 42 COc1cccc(NC(=O)CNc2ccc(Cl)cc2Br)c1 ZINC000147436969 FI On-Demand Anodyne PTGER3 20 45 COc1cccc(NC(=O)CNc2ccc(Cl)cc2Br)c1 ZINC000147436969 FI On-Demand Anodyne MTNR1A 27 46 COc1cccc(NC(=O)CNc2ccc(Cl)cc2Br)c1 ZINC000147436969 FI On-Demand Anodyne MTNR1B 32 48 COc1cccc(NC(=O)CNc2ccc(Cl)cc2Br)c1 ZINC000147436969 FI On-Demand Anodyne TAAR1 35 52 COc1cccc(NC(=O)CNc2ccc(Cl)cc2Br)c1 ZINC000147436969 FI On-Demand Anodyne AKR1C3 26 41 COc1cccc(NC(=O)CNc2ccc(Cl)cc2Br)c1 ZINC000147436969 FI On-Demand Anodyne AKR1C2 36 41 COc1cccc(NC(=O)CNc2ccc(Cl)cc2Br)c1 ZINC000147436969 FI On-Demand Anodyne PSBA 0 45 COc1cccc(NC(=O)CNc2ccc(Cl)cc2Br)c1 ZINC000147436969 FI On-Demand Anodyne KCNK3 42 35 O=C([C@@H]1Cc2ccccc2O1)N1CCC[C@H]1CCCBr ZINC000147436976 EG For-Sale Reactive PREP 48 35 NC1(C(=O)Nc2cccc3ccccc23)CCC1 ZINC000147436986 BF For-Sale Anodyne TRPV1 36 43 CC(C)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147437018 DC For-Sale Anodyne CA2 47 42 CC(C)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147437018 DC For-Sale Anodyne CA1 32 40 CC(C)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147437018 DC For-Sale Anodyne CA4 43 40 C[C@@H](CNc1c([N+](=O)[O-])ccc(F)c1F)CC(=O)O ZINC000147437030 CE For-Sale Bother COLA 46 31 CCc1cccc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147437036 CG For-Sale Anodyne ADRB2 66 49 CCc1cccc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147437036 CG For-Sale Anodyne ADRB1 91 45 CCc1cccc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147437036 CG For-Sale Anodyne GRIN1 28 45 CCc1cccc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147437036 CG For-Sale Anodyne ADRB3 64 45 CCc1cccc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147437036 CG For-Sale Anodyne ABCB1 15 45 CCc1cccc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147437036 CG For-Sale Anodyne PDS 61 34 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne ACE 29 58 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne SSTR2 32 44 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne OPRM1 17 54 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MME 49 56 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne EDNRB 62 46 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne EDNRA 54 53 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne TACR1 36 56 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MC4R 57 47 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne CTSB 25 47 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne CCKAR 133 52 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne CTSL 42 46 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne BRS3 36 59 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne TIMP3 20 54 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne NMBR 52 55 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MC3R 76 47 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MC5R 72 41 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MMP2 38 58 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MMP8 58 55 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne GRIA1 49 41 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MMP14 28 52 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne GRPR 84 42 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne ECE1 75 56 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne REN 17 43 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne REN1 17 42 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne LNPEP 26 40 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne SSTR3 27 41 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MMP11 101 42 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne CCKBR 95 49 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne GHSR 72 52 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne CAPN1 21 52 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MMP9 37 55 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne CAPN2 22 41 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MC1R 110 47 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne ADAM9 51 52 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne CTSC 15 48 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MMP7 29 55 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne MMP1 34 55 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne FPR1 28 49 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne NPR 62 54 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne ADAM12 17 52 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne KISS1R 91 43 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne ERAP2 47 43 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne PSMB8 29 44 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne TMPRSS6 17 43 CCN(CC)[C@H](C)CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)C(C)C ZINC000147437097 GF On-Demand Anodyne HPN 21 42 CCNc1ncc(Cl)c(Oc2ccc(C(N)=O)cc2)n1 ZINC000147437157 CE For-Sale Anodyne CHEK2 50 39 O=C(CCNC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)NC1CCCCC1 ZINC000147437164 EG On-Demand Anodyne EPHX2 25 55 O=C(c1cccc2cccnc12)N1CCC[C@@H]1CCCBr ZINC000147437210 EI For-Sale Reactive HCRTR1 36 53 O=C(c1cccc2cccnc12)N1CCC[C@@H]1CCCBr ZINC000147437210 EI For-Sale Reactive HCRTR2 38 53 O=C(c1cccc2cccnc12)N1CCC[C@@H]1CCCBr ZINC000147437210 EI For-Sale Reactive FAP 0 50 Cc1ccc([N+](=O)[O-])c(NC[C@@H](C)CC(=O)O)c1 ZINC000147437250 CE On-Demand Bother COLA 40 33 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CC(=O)N(C)c3ccccc3)cc2)c1 ZINC000147437260 HI On-Demand Bother NPY5R 26 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CC(=O)N(C)c3ccccc3)cc2)c1 ZINC000147437260 HI On-Demand Bother TAAR1 24 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CC(=O)N(C)c3ccccc3)cc2)c1 ZINC000147437260 HI On-Demand Bother AKR1C3 20 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(CC(=O)N(C)c3ccccc3)cc2)c1 ZINC000147437260 HI On-Demand Bother AKR1C2 50 41 Cc1nc(=O)c(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)[nH]1 ZINC000147437268 HD On-Demand Anodyne TGM2 57 40 Cc1nc(=O)c(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)[nH]1 ZINC000147437268 HD On-Demand Anodyne F13A1 51 40 O=C(Nc1n[nH]c2ccccc12)c1cccc(Cl)c1F ZINC000147437276 CH On-Demand Anodyne GSK3B 0 42 O=C(Nc1n[nH]c2ccccc12)c1cccc(Cl)c1F ZINC000147437276 CH On-Demand Anodyne GSK3A 35 41 O=C(Nc1n[nH]c2ccccc12)c1cccc(Cl)c1F ZINC000147437276 CH On-Demand Anodyne CDC7 18 41 O=C(Nc1n[nH]c2ccccc12)c1cccc(Cl)c1F ZINC000147437276 CH On-Demand Anodyne NR2E3 61 35 CCc1cccc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147437293 CG For-Sale Anodyne ADRB2 66 49 CCc1cccc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147437293 CG For-Sale Anodyne ADRB1 91 45 CCc1cccc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147437293 CG For-Sale Anodyne GRIN1 28 45 CCc1cccc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147437293 CG For-Sale Anodyne ADRB3 64 45 CCc1cccc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147437293 CG For-Sale Anodyne ABCB1 15 45 CCc1cccc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147437293 CG For-Sale Anodyne PDS 61 34 O=C(CCNC(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1)NC1CCCCC1 ZINC000147437379 EG On-Demand Anodyne EPHX2 25 55 O=C(c1cccc2cccnc12)N1CCC[C@H]1CCCBr ZINC000147437398 EI For-Sale Reactive HCRTR1 36 53 O=C(c1cccc2cccnc12)N1CCC[C@H]1CCCBr ZINC000147437398 EI For-Sale Reactive HCRTR2 38 53 O=C(c1cccc2cccnc12)N1CCC[C@H]1CCCBr ZINC000147437398 EI For-Sale Reactive FAP 0 50 CCCNc1cc(Oc2ccc(C(N)=O)cc2)nc(N)n1 ZINC000147437404 CD For-Sale Anodyne AGPAT2 25 44 CC(=O)N1c2ccc(S(=O)(=O)N3C[C@H](C)O[C@H](c4ccccc4)C3)cc2C[C@@H]1C ZINC000147437412 HG On-Demand Anodyne NOD2 20 42 Cc1ccc([N+](=O)[O-])c(NC[C@H](C)CC(=O)O)c1 ZINC000147437429 CE On-Demand Bother COLA 40 33 C#CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147437484 DB For-Sale Mild CA2 36 45 C#CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147437484 DB For-Sale Mild CA1 27 40 C#CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147437484 DB For-Sale Mild CA4 34 40 C#CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147437484 DB For-Sale Mild CA14 16 45 C#CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147437484 DB For-Sale Mild CA12 19 45 COc1cc(C(=O)Nc2n[nH]c3ccccc23)ccc1F ZINC000147437520 CF On-Demand Anodyne GSK3B 0 40 COc1cc(C(=O)Nc2n[nH]c3ccccc23)ccc1F ZINC000147437520 CF On-Demand Anodyne COLA 36 48 COc1cc(C(=O)Nc2n[nH]c3ccccc23)ccc1F ZINC000147437520 CF On-Demand Anodyne CPT1A 47 33 COc1cc(C(=O)Nc2n[nH]c3ccccc23)ccc1F ZINC000147437520 CF On-Demand Anodyne AURKB 41 39 COc1cc(C(=O)Nc2n[nH]c3ccccc23)ccc1F ZINC000147437520 CF On-Demand Anodyne CDK2 0 44 COc1cc(C(=O)Nc2n[nH]c3ccccc23)ccc1F ZINC000147437520 CF On-Demand Anodyne FABH 0 40 COc1cc(C(=O)Nc2n[nH]c3ccccc23)ccc1F ZINC000147437520 CF On-Demand Anodyne CDC7 19 42 COc1cc(C(=O)Nc2n[nH]c3ccccc23)ccc1F ZINC000147437520 CF On-Demand Anodyne TAAR1 18 43 COc1cc(C(=O)Nc2n[nH]c3ccccc23)ccc1F ZINC000147437520 CF On-Demand Anodyne GLMU 0 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2cc[nH]c2c1 ZINC000147437538 GF On-Demand Anodyne HTR4 45 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2cc[nH]c2c1 ZINC000147437538 GF On-Demand Anodyne F10 17 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2cc[nH]c2c1 ZINC000147437538 GF On-Demand Anodyne GRIN2B 46 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2cc[nH]c2c1 ZINC000147437538 GF On-Demand Anodyne EPHX2 15 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2cc[nH]c2c1 ZINC000147437538 GF On-Demand Anodyne PLD2 40 35 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2cc[nH]c2c1 ZINC000147437538 GF On-Demand Anodyne TGM2 61 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2cc[nH]c2c1 ZINC000147437538 GF On-Demand Anodyne CACNA1I 64 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2cc[nH]c2c1 ZINC000147437538 GF On-Demand Anodyne F13A1 51 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2cc[nH]c2c1 ZINC000147437538 GF On-Demand Anodyne AKR1C3 51 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2cc[nH]c2c1 ZINC000147437538 GF On-Demand Anodyne NAMPT 42 43 CC(C)CCCCNC(=O)CNC(=O)CN ZINC000147437569 BC For-Sale Anodyne UREB 0 45 O=C(CCNC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)NC1CCCCC1 ZINC000147437570 EG On-Demand Anodyne EPHX2 25 55 CC(C)CCO[C@@H](C)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437582 EF On-Demand Anodyne DRD4 20 44 CC(C)CCO[C@@H](C)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437582 EF On-Demand Anodyne P2RY12 105 36 CC(C)CCO[C@@H](C)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437582 EF On-Demand Anodyne SIGMAR1 16 43 CC(C)CCO[C@@H](C)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437582 EF On-Demand Anodyne CCR1 34 42 CC(C)CCO[C@@H](C)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437582 EF On-Demand Anodyne MCHR1 18 44 O=C(Nc1cccc(S(=O)(=O)NC2=NCCC2)c1)c1cnccn1 ZINC000147437585 ED On-Demand Anodyne GRM4 48 42 Cc1ccccc1CCC(=O)N1CCC[C@@H]1CCCBr ZINC000147437629 EI For-Sale Reactive PREP 57 38 Cc1ccccc1CCC(=O)N1CCC[C@@H]1CCCBr ZINC000147437629 EI For-Sale Reactive FAP 0 42 Cc1nccc(-c2cccc(NC(=O)C(=O)NCC(C)(C)N3CCC[C@H](C)C3)c2)n1 ZINC000147437683 HG On-Demand Anodyne PRKD1 58 33 Cc1cc(Cl)cc(C(=O)Nc2n[nH]c3ccccc23)c1 ZINC000147437762 CH On-Demand Anodyne GSK3B 15 44 Cc1cc(Cl)cc(C(=O)Nc2n[nH]c3ccccc23)c1 ZINC000147437762 CH On-Demand Anodyne GSK3A 37 40 Cc1cc(Cl)cc(C(=O)Nc2n[nH]c3ccccc23)c1 ZINC000147437762 CH On-Demand Anodyne CDK2 0 41 Cc1cc(Cl)cc(C(=O)Nc2n[nH]c3ccccc23)c1 ZINC000147437762 CH On-Demand Anodyne CDC7 21 48 Cc1cc(Cl)cc(C(=O)Nc2n[nH]c3ccccc23)c1 ZINC000147437762 CH On-Demand Anodyne KCNK3 49 35 Cc1cc(Cl)cc(C(=O)Nc2n[nH]c3ccccc23)c1 ZINC000147437762 CH On-Demand Anodyne KCNK9 28 40 O=C(CCNC(=O)[C@H]1C[C@@H]1c1cccc(Br)c1)NC1CCCCC1 ZINC000147437802 GH On-Demand Anodyne EPHX2 22 41 COc1ccc([N+](=O)[O-])cc1CNCCCCC(C)C ZINC000147437803 CH For-Sale Bother GNRHR 0 42 COc1ccc([N+](=O)[O-])cc1CNCCCCC(C)C ZINC000147437803 CH For-Sale Bother GPM3 0 43 CC(C)CCO[C@H](C)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437804 EF On-Demand Anodyne DRD4 20 44 CC(C)CCO[C@H](C)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437804 EF On-Demand Anodyne P2RY12 105 36 CC(C)CCO[C@H](C)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437804 EF On-Demand Anodyne SIGMAR1 16 43 CC(C)CCO[C@H](C)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437804 EF On-Demand Anodyne CCR1 34 42 CC(C)CCO[C@H](C)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437804 EF On-Demand Anodyne MCHR1 18 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1COCCO1 ZINC000147437827 FC On-Demand Anodyne TGM2 54 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1COCCO1 ZINC000147437827 FC On-Demand Anodyne F13A1 56 43 Cc1ccccc1CCC(=O)N1CCC[C@H]1CCCBr ZINC000147437833 EI For-Sale Reactive PREP 57 38 Cc1ccccc1CCC(=O)N1CCC[C@H]1CCCBr ZINC000147437833 EI For-Sale Reactive FAP 0 42 COC[C@@H]1CCN(CCS(=O)(=O)c2cccc(C#N)c2)C1 ZINC000147437881 DD On-Demand Mild CCR3 16 41 COC[C@@H]1CCN(CCS(=O)(=O)c2cccc(C#N)c2)C1 ZINC000147437881 DD On-Demand Mild CHRNA10 15 41 CCN1CCN(c2ccccc2NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)CC1 ZINC000147437889 HF On-Demand Anodyne HTR1A 54 41 CCN1CCN(c2ccccc2NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)CC1 ZINC000147437889 HF On-Demand Anodyne DRD2 39 40 CCN1CCN(c2ccccc2NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)CC1 ZINC000147437889 HF On-Demand Anodyne HTR1D 18 41 CCN1CCN(c2ccccc2NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)CC1 ZINC000147437889 HF On-Demand Anodyne HTR1B 29 41 CCN1CCN(c2ccccc2NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)CC1 ZINC000147437889 HF On-Demand Anodyne DRD3 41 40 CCN1CCN(c2ccccc2NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)CC1 ZINC000147437889 HF On-Demand Anodyne HTR7 34 40 CCN1CCN(c2ccccc2NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)CC1 ZINC000147437889 HF On-Demand Anodyne KCNQ2 80 40 CCN1CCN(c2ccccc2NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)CC1 ZINC000147437889 HF On-Demand Anodyne NPY2R 76 37 CCN1CCN(c2ccccc2NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)CC1 ZINC000147437889 HF On-Demand Anodyne P2RY1 59 38 CCN1CCN(c2ccccc2NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)CC1 ZINC000147437889 HF On-Demand Anodyne PRNP 41 44 Cc1nccc(-c2cccc(NC(=O)C(=O)NCC(C)(C)N3CCC[C@@H](C)C3)c2)n1 ZINC000147437901 HG On-Demand Anodyne PRKD1 58 33 C[C@@H](CCN(C)C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147437944 DE On-Demand Anodyne UTS2 48 37 COCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147437954 BD For-Sale Anodyne DNPEP 0 41 COCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147437954 BD For-Sale Anodyne SIRT1 28 40 Cc1cn([C@H]2C[C@H](O)[C@@H](CN(N=O)C(=O)NCCCl)O2)c(=O)[nH]c1=O ZINC000147437958 GB Annotated Reactive TYMS 0 43 Cc1cn([C@H]2C[C@H](O)[C@@H](CN(N=O)C(=O)NCCCl)O2)c(=O)[nH]c1=O ZINC000147437958 GB Annotated Reactive POLA1 23 43 Cc1cn([C@H]2C[C@H](O)[C@@H](CN(N=O)C(=O)NCCCl)O2)c(=O)[nH]c1=O ZINC000147437958 GB Annotated Reactive TK 58 56 Cc1cn([C@H]2C[C@H](O)[C@@H](CN(N=O)C(=O)NCCCl)O2)c(=O)[nH]c1=O ZINC000147437958 GB Annotated Reactive TK1 50 56 Cc1cn([C@H]2C[C@H](O)[C@@H](CN(N=O)C(=O)NCCCl)O2)c(=O)[nH]c1=O ZINC000147437958 GB Annotated Reactive POLB 15 46 Cc1cn([C@H]2C[C@H](O)[C@@H](CN(N=O)C(=O)NCCCl)O2)c(=O)[nH]c1=O ZINC000147437958 GB Annotated Reactive TMK 32 47 Cc1cn([C@H]2C[C@H](O)[C@@H](CN(N=O)C(=O)NCCCl)O2)c(=O)[nH]c1=O ZINC000147437958 GB Annotated Reactive DNK 0 41 Cc1cn([C@H]2C[C@H](O)[C@@H](CN(N=O)C(=O)NCCCl)O2)c(=O)[nH]c1=O ZINC000147437958 GB Annotated Reactive TK2 61 45 Cc1cn([C@H]2C[C@H](O)[C@@H](CN(N=O)C(=O)NCCCl)O2)c(=O)[nH]c1=O ZINC000147437958 GB Annotated Reactive UL23 0 43 Cc1cn([C@H]2C[C@H](O)[C@@H](CN(N=O)C(=O)NCCCl)O2)c(=O)[nH]c1=O ZINC000147437958 GB Annotated Reactive THYX 0 40 Cc1cn([C@H]2C[C@H](O)[C@@H](CN(N=O)C(=O)NCCCl)O2)c(=O)[nH]c1=O ZINC000147437958 GB Annotated Reactive THYA 0 41 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437994 FD On-Demand Anodyne DRD4 15 40 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437994 FD On-Demand Anodyne CCR1 35 41 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147437994 FD On-Demand Anodyne SHH 33 40 O=C(CCNC(=O)[C@@H]1C[C@H]1c1cccc(Br)c1)NC1CCCCC1 ZINC000147437996 GH On-Demand Anodyne EPHX2 22 41 COc1cc(OC)cc(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147438032 FG For-Sale Reactive HCRTR1 0 43 COC[C@H]1CCN(CCS(=O)(=O)c2cccc(C#N)c2)C1 ZINC000147438052 DD On-Demand Mild CCR3 16 41 COC[C@H]1CCN(CCS(=O)(=O)c2cccc(C#N)c2)C1 ZINC000147438052 DD On-Demand Mild CHRNA10 15 41 O=C(CCCNC(=O)C1CC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438069 HD On-Demand Anodyne FKBP1A 15 48 O=C(CCCNC(=O)C1CC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438069 HD On-Demand Anodyne EPHX2 39 45 O=C(CCCNC(=O)C1CC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438069 HD On-Demand Anodyne TGM2 86 46 O=C(CCCNC(=O)C1CC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438069 HD On-Demand Anodyne F13A1 93 46 CC(C)[C@@H](c1ccccn1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147438086 KK Annotated Anodyne TP53 42 66 CC(C)[C@@H](c1ccccn1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147438086 KK Annotated Anodyne MDM2 252 68 CCCNc1ncc(Cl)c(Oc2ccc(C(N)=O)cc2)n1 ZINC000147438107 DF For-Sale Anodyne CHEK2 40 40 C[C@H](CCN(C)C)NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147438155 DE On-Demand Anodyne UTS2 48 37 COCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147438172 BD For-Sale Anodyne DNPEP 0 41 COCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147438172 BD For-Sale Anodyne SIRT1 28 40 C[C@@H](OC[C@@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147438191 FD On-Demand Anodyne DRD4 15 40 C[C@@H](OC[C@@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147438191 FD On-Demand Anodyne CCR1 35 41 C[C@@H](OC[C@@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147438191 FD On-Demand Anodyne SHH 33 40 COc1cc(OC)cc(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147438220 FG For-Sale Reactive HCRTR1 0 43 O=C(CCNC(=O)[C@@H]1C[C@@H]1c1cccc(Br)c1)NC1CCCCC1 ZINC000147438250 GH On-Demand Anodyne EPHX2 22 41 Cc1ccc(NC(=O)CC2(CN)CCC2)c(Br)c1 ZINC000147438271 DG For-Sale Anodyne CA4 19 42 N#Cc1cccc(S(=O)(=O)CCN2CC[C@H](CO)C2)c1 ZINC000147438307 CC On-Demand Mild ITGA4 47 30 Nc1ncccc1S(=O)(=O)Nc1ccc(Cl)c(Br)c1 ZINC000147438309 FF For-Sale Anodyne GRM4 21 41 Nc1ncccc1S(=O)(=O)Nc1ccc(Cl)c(Br)c1 ZINC000147438309 FF For-Sale Anodyne SGK1 73 42 CCCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147438327 DC For-Sale Anodyne CA2 52 41 CCCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147438327 DC For-Sale Anodyne CA1 39 41 CCCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147438327 DC For-Sale Anodyne CA4 45 41 CCCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147438327 DC For-Sale Anodyne CA12 26 40 C[C@H](OC[C@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147438359 FD On-Demand Anodyne DRD4 15 40 C[C@H](OC[C@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147438359 FD On-Demand Anodyne CCR1 35 41 C[C@H](OC[C@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147438359 FD On-Demand Anodyne SHH 33 40 O=C(Nc1n[nH]c2ccccc12)c1ccc(Br)c(Cl)c1 ZINC000147438386 FI On-Demand Anodyne KCNJ11 25 40 O=C(Nc1n[nH]c2ccccc12)c1ccc(Br)c(Cl)c1 ZINC000147438386 FI On-Demand Anodyne CDC7 21 46 C[C@H](CNc1ccc(C(F)(F)F)cc1)CC(=O)O ZINC000147438392 CG For-Sale Anodyne DHODH 29 43 C[C@H](CNc1ccc(C(F)(F)F)cc1)CC(=O)O ZINC000147438392 CG For-Sale Anodyne EPHX2 16 45 C[C@H](CNc1ccc(C(F)(F)F)cc1)CC(=O)O ZINC000147438392 CG For-Sale Anodyne FPR2 23 46 COc1ccc(Cl)cc1C(=O)N1CCC[C@@H]1CCCBr ZINC000147438424 FI For-Sale Reactive ACKR3 62 32 CCOC(=O)NCCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438491 GD On-Demand Anodyne F2 15 41 CCOC(=O)NCCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438491 GD On-Demand Anodyne CHRM4 16 44 CCOC(=O)NCCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438491 GD On-Demand Anodyne CHRM5 15 42 CCOC(=O)NCCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438491 GD On-Demand Anodyne EPHX2 21 42 CCOC(=O)NCCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438491 GD On-Demand Anodyne TGM2 73 49 CCOC(=O)NCCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438491 GD On-Demand Anodyne F13A1 80 49 CCCCCCCOc1ccc(CNC2CC2)nc1 ZINC000147438503 CH For-Sale Mild PLA2G4B 71 35 N#Cc1cccc(S(=O)(=O)CCN2CC[C@@H](CO)C2)c1 ZINC000147438531 CC On-Demand Mild ITGA4 47 30 CNc1cncc(Oc2ccc(C(N)=O)cc2)n1 ZINC000147438562 BD For-Sale Anodyne CHEK2 30 40 CNc1cncc(Oc2ccc(C(N)=O)cc2)n1 ZINC000147438562 BD For-Sale Anodyne SELE 48 31 CNc1cncc(Oc2ccc(C(N)=O)cc2)n1 ZINC000147438562 BD For-Sale Anodyne ICAM1 43 31 CN(C)C(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147438563 CC For-Sale Anodyne CA2 20 40 CN(C)C(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147438563 CC For-Sale Anodyne CA4 22 40 C[C@@H](OC[C@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147438570 FD On-Demand Anodyne DRD4 15 40 C[C@@H](OC[C@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147438570 FD On-Demand Anodyne CCR1 35 41 C[C@@H](OC[C@H]1CCCO1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147438570 FD On-Demand Anodyne SHH 33 40 Clc1cc(-c2ccccc2)nc(-c2cncs2)n1 ZINC000147438609 CH For-Sale Anodyne CD38 48 36 C[C@@H](CNc1ccc(C(F)(F)F)cc1)CC(=O)O ZINC000147438622 CG For-Sale Anodyne DHODH 29 43 C[C@@H](CNc1ccc(C(F)(F)F)cc1)CC(=O)O ZINC000147438622 CG For-Sale Anodyne EPHX2 16 45 C[C@@H](CNc1ccc(C(F)(F)F)cc1)CC(=O)O ZINC000147438622 CG For-Sale Anodyne FPR2 23 46 Cc1ccc(Br)c(C(=O)Nc2n[nH]c3ccccc23)c1 ZINC000147438653 EH On-Demand Anodyne GSK3B 22 43 Cc1ccc(Br)c(C(=O)Nc2n[nH]c3ccccc23)c1 ZINC000147438653 EH On-Demand Anodyne GSK3A 45 40 Cc1ccc(Br)c(C(=O)Nc2n[nH]c3ccccc23)c1 ZINC000147438653 EH On-Demand Anodyne CDK2 0 41 COc1ccc(Cl)cc1C(=O)N1CCC[C@H]1CCCBr ZINC000147438663 FI For-Sale Reactive ACKR3 62 32 O=S(=O)(NCCc1c[nH]c2ccccc12)c1cccc(Cl)c1Cl ZINC000147438667 FH On-Demand Anodyne ALOX15 40 59 CN(C)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147438730 HD On-Demand Anodyne HTR4 48 36 CN(C)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147438730 HD On-Demand Anodyne GRIN2B 25 40 CN(C)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147438730 HD On-Demand Anodyne EPHX2 19 42 CN(C)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147438730 HD On-Demand Anodyne TGM2 59 43 CN(C)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147438730 HD On-Demand Anodyne CACNA1I 62 40 CN(C)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147438730 HD On-Demand Anodyne F13A1 43 41 CN(C)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147438730 HD On-Demand Anodyne SFRP1 19 43 CN(C)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147438730 HD On-Demand Anodyne NAMPT 49 43 CCN(CC)[C@@H](C)CNC(=O)c1cc2ccc(Cl)cc2[nH]1 ZINC000147438732 DG On-Demand Anodyne CCKAR 22 42 CCCNc1nc(C)cc(Oc2ccc(C(N)=O)cc2)n1 ZINC000147438766 CE For-Sale Anodyne TRY1_BOVIN 18 41 NC(=O)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147438782 DB For-Sale Anodyne CA2 37 42 NC(=O)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147438782 DB For-Sale Anodyne CA1 31 42 NC(=O)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147438782 DB For-Sale Anodyne CA4 40 42 NC(=O)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147438782 DB For-Sale Anodyne CA5A 40 38 CO[C@@H]1CCN(C(=O)c2ccncc2/N=C(\O)c2nc(C3CC3)ccc2Nc2cncnc2)C1 ZINC000147438897 JG Annotated Mild PDE10A 0 51 Cc1cccc(CCC(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147438913 EI For-Sale Reactive PREP 61 39 CCN(CC)[C@H](C)CNC(=O)c1cc2ccc(Cl)cc2[nH]1 ZINC000147438942 DG On-Demand Anodyne CCKAR 22 42 CCN(CC)[C@H](C)CNC(=O)c1cc2ccc(Cl)cc2[nH]1 ZINC000147438942 DG On-Demand Anodyne PYGL 98 51 CCN(CC)[C@H](C)CNC(=O)c1cc2ccc(Cl)cc2[nH]1 ZINC000147438942 DG On-Demand Anodyne PYGM 17 41 CCN(CC)[C@H](C)CNC(=O)c1cc2ccc(Cl)cc2[nH]1 ZINC000147438942 DG On-Demand Anodyne ALPL 45 47 CCOc1ccc(NC(=O)C2(N)CCC2)cc1 ZINC000147438967 BD On-Demand Anodyne SCN2A 26 40 CCOc1ccc(NC(=O)C2(N)CCC2)cc1 ZINC000147438967 BD On-Demand Anodyne TIMP3 40 32 CCOc1ccc(NC(=O)C2(N)CCC2)cc1 ZINC000147438967 BD On-Demand Anodyne ACR 42 33 CCOc1ccc(NC(=O)C2(N)CCC2)cc1 ZINC000147438967 BD On-Demand Anodyne CA9 15 40 CCOc1ccc(NC(=O)C2(N)CCC2)cc1 ZINC000147438967 BD On-Demand Anodyne NCE103 15 40 CCOc1ccc(NC(=O)C2(N)CCC2)cc1 ZINC000147438967 BD On-Demand Anodyne NOD2 24 41 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne PPIA 15 48 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne F10 27 45 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne ECR 42 34 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne NR1H4 25 46 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne KCNMA1 28 40 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne CSF1R 15 42 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne FABH 0 40 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne ACPS 0 41 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne AKR1C3 20 42 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne PAGA 0 44 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne KCNK3 101 47 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne KCNK9 63 47 CC(=O)c1ccccc1NC(=O)c1cc(C)cc(Cl)c1 ZINC000147438984 CI On-Demand Anodyne G2YM83_BOTF4 44 33 COCc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438986 HF On-Demand Anodyne HTR4 62 40 COCc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438986 HF On-Demand Anodyne MMP13 17 45 COCc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438986 HF On-Demand Anodyne EPHX2 19 42 COCc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438986 HF On-Demand Anodyne TGM2 65 46 COCc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438986 HF On-Demand Anodyne CACNA1I 58 34 COCc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147438986 HF On-Demand Anodyne F13A1 64 46 CNc1nc(OC)nc(Oc2ccc(C(N)=O)cc2)n1 ZINC000147439012 CC For-Sale Anodyne CHEK2 27 41 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne PLG 41 37 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne CHRM1 16 43 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne DRD2 21 50 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne DRD4 40 31 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne F10 17 44 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne SIGMAR1 23 47 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne SSTR5 45 38 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne TRY2_BOVIN 81 35 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne CCR3 36 40 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne C3AR1 48 41 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne SLC6A5 36 41 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne EPHX2 37 43 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne ST14 98 39 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne AMP1_PLAFQ 26 40 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne MCHR1 35 48 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne CCR8 62 44 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne SHH 22 40 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne BIRC2 31 44 CC(C)Oc1cccc(CC(=O)N2CCC(NC(=O)c3ccccc3)CC2)c1 ZINC000147439013 GG On-Demand Anodyne TMPRSS6 40 33 O=C1CCCC[C@@H](C(C(=O)OCc2ccccc2)C(=O)OCc2ccccc2)C1 ZINC000147439068 GI For-Sale Anodyne AMY2 46 32 O=C1CCCC[C@@H](C(C(=O)OCc2ccccc2)C(=O)OCc2ccccc2)C1 ZINC000147439068 GI For-Sale Anodyne SLC12A5 58 40 Cc1cccc(CCC(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147439134 EI For-Sale Reactive PREP 61 39 CO[C@H]1CCN(C(=O)c2ccncc2/N=C(\O)c2nc(C3CC3)ccc2Nc2cncnc2)C1 ZINC000147439146 JG Annotated Mild PDE10A 0 51 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cc(C4CC4)nn3-c3ccccc3)ccc21 ZINC000147439196 HH On-Demand Anodyne FPR2 42 34 CCOc1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147439201 CF For-Sale Anodyne LTA4H 25 43 O=C(Cn1cccnc1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147439223 GC On-Demand Anodyne TGM2 61 42 O=C(Cn1cccnc1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147439223 GC On-Demand Anodyne F13A1 58 42 NC(=O)c1ccc(Oc2cc(N)ncn2)cc1 ZINC000147439241 BC For-Sale Anodyne CHEK2 37 40 CNc1ccc(Cl)cc1C(=O)NCCNC(=O)N(C)C ZINC000147439275 CD For-Sale Anodyne F10 32 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147439422 HD On-Demand Anodyne HTR4 45 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147439422 HD On-Demand Anodyne GRIN2B 39 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147439422 HD On-Demand Anodyne PLD1 62 36 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147439422 HD On-Demand Anodyne EPHX2 17 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147439422 HD On-Demand Anodyne PLD2 47 36 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147439422 HD On-Demand Anodyne TGM2 62 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147439422 HD On-Demand Anodyne CACNA1I 64 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147439422 HD On-Demand Anodyne F13A1 52 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147439422 HD On-Demand Anodyne AKR1C3 52 35 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2[nH]c(=O)[nH]c2c1 ZINC000147439422 HD On-Demand Anodyne NAMPT 42 42 C[C@@H]1CCCN(CCS(=O)(=O)c2cccc(C#N)c2)[C@@H]1C ZINC000147439424 DE On-Demand Mild CHRNA10 28 44 COc1ccc(CCNC(=O)C2(N)CCC2)cc1OC ZINC000147439428 CD On-Demand Anodyne TRPV1 21 42 COc1ccc(CCNC(=O)C2(N)CCC2)cc1OC ZINC000147439428 CD On-Demand Anodyne MTNR1A 41 35 COc1ccc(CCNC(=O)C2(N)CCC2)cc1OC ZINC000147439428 CD On-Demand Anodyne MTNR1B 43 46 COc1ccc(CCNC(=O)C2(N)CCC2)cc1OC ZINC000147439428 CD On-Demand Anodyne MT-ND1 26 41 COc1ccc(CCNC(=O)C2(N)CCC2)cc1OC ZINC000147439428 CD On-Demand Anodyne NCE103 25 55 COc1ccc(CCNC(=O)C2(N)CCC2)cc1OC ZINC000147439428 CD On-Demand Anodyne ABCG2 23 47 COc1ccc(CCNC(=O)C2(N)CCC2)cc1OC ZINC000147439428 CD On-Demand Anodyne P96878_MYCTU 18 55 COc1ccc(CCNC(=O)C2(N)CCC2)cc1OC ZINC000147439428 CD On-Demand Anodyne SCMU_MYCTU 0 41 COc1ccc(CCNC(=O)C2(N)CCC2)cc1OC ZINC000147439428 CD On-Demand Anodyne CAN2 0 55 Cc1cc(C(=O)Nc2cccc(S(C)(=O)=O)c2)cc([N+](=O)[O-])c1 ZINC000147439477 EF On-Demand Bother DDX3X 0 40 NC(=O)c1ccc(Oc2cc(N)nc(N)n2)cc1 ZINC000147439479 BC For-Sale Anodyne CHEK2 50 43 NC(=O)c1ccc(Oc2cc(N)nc(N)n2)cc1 ZINC000147439479 BC For-Sale Anodyne ST14 15 41 CCCNc1cc(C(=O)NCCNC(=O)N(C)C)ccn1 ZINC000147439530 CC For-Sale Anodyne KDM4E 23 40 CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147439607 CC For-Sale Anodyne CA2 60 48 CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147439607 CC For-Sale Anodyne CA1 42 41 CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147439607 CC For-Sale Anodyne CA7 41 38 CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147439607 CC For-Sale Anodyne CA5B 43 38 CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147439607 CC For-Sale Anodyne CA4 53 41 CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147439607 CC For-Sale Anodyne CA5A 45 38 CCN(CC)[C@@H](C)CNC(=O)c1ccc(OCc2ccncc2)cc1 ZINC000147439642 EG On-Demand Anodyne CYP3A4 16 49 CCN(CC)[C@@H](C)CNC(=O)c1ccc(OCc2ccncc2)cc1 ZINC000147439642 EG On-Demand Anodyne CYP26A1 31 41 C[C@H]1CCCN(CCS(=O)(=O)c2cccc(C#N)c2)[C@@H]1C ZINC000147439652 DE On-Demand Mild CHRNA10 28 44 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cccnc3N3CCCC3)ccc21 ZINC000147439670 FF On-Demand Anodyne KCNQ2 54 32 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cccnc3N3CCCC3)ccc21 ZINC000147439670 FF On-Demand Anodyne TRPV1 26 40 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cccnc3N3CCCC3)ccc21 ZINC000147439670 FF On-Demand Anodyne P2RY1 52 43 Cc1cc(C(=O)N2CCN(S(=O)(=O)c3ccc(C#N)cc3)CC2)cc([N+](=O)[O-])c1 ZINC000147439698 HD On-Demand Mild SLC6A9 15 42 COc1ccccc1CNC(=O)C1(N)CCC1 ZINC000147439704 BD On-Demand Anodyne TACR1 0 42 COc1ccccc1CNC(=O)C1(N)CCC1 ZINC000147439704 BD On-Demand Anodyne GPM3 0 48 COc1ccccc1CNC(=O)C1(N)CCC1 ZINC000147439704 BD On-Demand Anodyne MBTPS1 41 35 COc1ccc(NC(C)=O)cc1S(=O)(=O)N1C[C@H](c2ccccc2)O[C@H](C)C1 ZINC000147439711 HF On-Demand Anodyne TSHR 68 34 COc1ccc(NC(C)=O)cc1S(=O)(=O)N1C[C@H](c2ccccc2)O[C@H](C)C1 ZINC000147439711 HF On-Demand Anodyne CPT1A 59 40 COc1ccc(NC(C)=O)cc1S(=O)(=O)N1C[C@H](c2ccccc2)O[C@H](C)C1 ZINC000147439711 HF On-Demand Anodyne CPT2 45 40 COc1ccc(NC(C)=O)cc1S(=O)(=O)N1C[C@H](c2ccccc2)O[C@H](C)C1 ZINC000147439711 HF On-Demand Anodyne CPT1B 44 36 COC(=O)[C@@H](CO)NC(=O)CNC(=O)OC(C)(C)C ZINC000147439774 CB On-Demand Anodyne PAPA1_CARPA 50 39 N#CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147439808 DB For-Sale Mild CA2 34 40 N#CCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147439808 DB For-Sale Mild CA1 27 40 Cc1cc(Br)sc1C(=O)NCc1ccccc1 ZINC000147439850 DH For-Sale Anodyne CHRM4 29 45 Cc1cc(Br)sc1C(=O)NCc1ccccc1 ZINC000147439850 DH For-Sale Anodyne ANPEP 31 42 Cc1cc(Br)sc1C(=O)NCc1ccccc1 ZINC000147439850 DH For-Sale Anodyne MMP13 15 45 Cc1cc(Br)sc1C(=O)NCc1ccccc1 ZINC000147439850 DH For-Sale Anodyne AMP1_PLAFQ 55 42 Cc1cc(Br)sc1C(=O)NCc1ccccc1 ZINC000147439850 DH For-Sale Anodyne SCD1 33 46 Cc1cc(Br)sc1C(=O)NCc1ccccc1 ZINC000147439850 DH For-Sale Anodyne SCD 29 50 Cc1cc(Br)sc1C(=O)NCc1ccccc1 ZINC000147439850 DH For-Sale Anodyne PDS 50 37 CCN(CC)[C@H](C)CNC(=O)c1ccc(OCc2ccncc2)cc1 ZINC000147439853 EG On-Demand Anodyne CYP3A4 16 49 CCN(CC)[C@H](C)CNC(=O)c1ccc(OCc2ccncc2)cc1 ZINC000147439853 EG On-Demand Anodyne CYP26A1 31 41 COc1ccc(NC(C)=O)cc1S(=O)(=O)N1C[C@H](C)O[C@@H](c2ccccc2)C1 ZINC000147439933 HF On-Demand Anodyne TSHR 68 34 COc1ccc(NC(C)=O)cc1S(=O)(=O)N1C[C@H](C)O[C@@H](c2ccccc2)C1 ZINC000147439933 HF On-Demand Anodyne CPT1A 59 40 COc1ccc(NC(C)=O)cc1S(=O)(=O)N1C[C@H](C)O[C@@H](c2ccccc2)C1 ZINC000147439933 HF On-Demand Anodyne CPT2 45 40 COc1ccc(NC(C)=O)cc1S(=O)(=O)N1C[C@H](C)O[C@@H](c2ccccc2)C1 ZINC000147439933 HF On-Demand Anodyne CPT1B 44 36 COc1ccccc1CNC(=O)CC1(CN)CCC1 ZINC000147439938 CD For-Sale Anodyne TACR1 28 41 O=C(Nc1ncc(Cc2ccc(F)c(F)c2)s1)c1ccc[nH]c1=O ZINC000147439978 EF On-Demand Anodyne SCD1 40 44 O=C(Nc1ncc(Cc2ccc(F)c(F)c2)s1)c1ccc[nH]c1=O ZINC000147439978 EF On-Demand Anodyne SCD 30 52 COC(=O)[C@H](CO)NC(=O)CNC(=O)OC(C)(C)C ZINC000147439996 CB On-Demand Anodyne PAPA1_CARPA 50 39 CN1[C@H](C(=O)O)C[C@@H]2CCCC[C@H]21 ZINC000147440050 AD For-Sale Anodyne ACE 30 55 O=C(CC[C@@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440083 GE On-Demand Anodyne EPHX2 16 43 O=C(CC[C@@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440083 GE On-Demand Anodyne TGM2 71 42 O=C(CC[C@@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440083 GE On-Demand Anodyne F13A1 75 42 O=C(CC[C@@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440083 GE On-Demand Anodyne AKR1C3 42 35 CC(C)n1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147440128 CD For-Sale Anodyne CASP3 97 42 CC(C)n1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147440128 CD For-Sale Anodyne CASP8 70 42 CC(C)n1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147440128 CD For-Sale Anodyne CASP1 56 38 CC(C)n1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147440128 CD For-Sale Anodyne CASP7 68 42 NS(=O)(=O)c1cc(F)c(OCCCN2CCCC2)c(F)c1 ZINC000147440251 DD For-Sale Anodyne HRH3 59 60 NS(=O)(=O)c1cc(F)c(OCCCN2CCCC2)c(F)c1 ZINC000147440251 DD For-Sale Anodyne HNMT 53 33 O=C(CC[C@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440295 GE On-Demand Anodyne EPHX2 16 43 O=C(CC[C@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440295 GE On-Demand Anodyne TGM2 71 42 O=C(CC[C@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440295 GE On-Demand Anodyne F13A1 75 42 O=C(CC[C@H]1CCCO1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440295 GE On-Demand Anodyne AKR1C3 42 35 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne F2 38 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne PLG 50 42 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne PRSS1 21 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne CHRM1 19 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne ACE 41 42 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne DRD4 23 54 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne F10 22 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne CHRM3 17 42 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne TACR1 19 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne SIGMAR1 25 52 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne SSTR5 42 37 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne CTSB 18 41 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne TRY2_BOVIN 109 43 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne TRY1_BOVIN 17 43 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne CCKAR 0 50 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne NPY2R 37 43 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne CCR1 32 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne CCR3 53 42 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne C3AR1 44 37 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne DPP4 20 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne MLNR 25 43 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne CCKBR 47 41 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne EPHX2 28 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne ACE2 44 32 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne ST14 124 44 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne MCHR1 33 46 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne CCR8 41 41 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne BRCA1 43 32 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne TMPRSS6 70 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440333 FG On-Demand Anodyne DERP1 0 44 CC(C)n1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147440338 CD For-Sale Anodyne CASP3 97 42 CC(C)n1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147440338 CD For-Sale Anodyne CASP8 70 42 CC(C)n1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147440338 CD For-Sale Anodyne CASP1 56 38 CC(C)n1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147440338 CD For-Sale Anodyne CASP7 62 42 O=C(NCc1ccc(Cn2ccccc2=O)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147440341 HH On-Demand Anodyne NOX4 40 31 O=C(NCc1ccc(Cn2ccccc2=O)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147440341 HH On-Demand Anodyne NOX1 42 31 O=C(NCc1ccc(Cn2ccccc2=O)cc1)c1cnn(-c2ccccc2Cl)c1 ZINC000147440341 HH On-Demand Anodyne NAMPT 42 39 O=C(O)[C@@H]1CCCN1C(=O)C[C@@H]1CCc2ccccc21 ZINC000147440348 CE On-Demand Anodyne F2 20 50 O=C(O)[C@@H]1CCCN1C(=O)C[C@@H]1CCc2ccccc21 ZINC000147440348 CE On-Demand Anodyne ACE 84 49 O=C(O)[C@@H]1CCCN1C(=O)C[C@@H]1CCc2ccccc21 ZINC000147440348 CE On-Demand Anodyne SLC6A1 53 33 O=C(O)[C@@H]1CCCN1C(=O)C[C@@H]1CCc2ccccc21 ZINC000147440348 CE On-Demand Anodyne MME 24 43 O=C(O)[C@@H]1CCCN1C(=O)C[C@@H]1CCc2ccccc21 ZINC000147440348 CE On-Demand Anodyne CPT1A 17 42 O=C(O)[C@@H]1CCCN1C(=O)C[C@@H]1CCc2ccccc21 ZINC000147440348 CE On-Demand Anodyne CPT2 43 40 O=C(O)[C@@H]1CCCN1C(=O)C[C@@H]1CCc2ccccc21 ZINC000147440348 CE On-Demand Anodyne DPP4 15 43 O=C(O)[C@@H]1CCCN1C(=O)C[C@@H]1CCc2ccccc21 ZINC000147440348 CE On-Demand Anodyne PREP 135 51 CCCOCC(=O)Nc1ccc(NS(C)(=O)=O)c(OC)c1 ZINC000147440353 DD On-Demand Anodyne TRPV1 15 41 CCCOCC(=O)Nc1ccc(NS(C)(=O)=O)c(OC)c1 ZINC000147440353 DD On-Demand Anodyne ENPP1 59 35 CCN(CC)[C@H](C)CNC(=O)c1cc2cc(C)ccc2[nH]1 ZINC000147440359 CF On-Demand Anodyne AKR1C3 23 41 NC(=O)c1ccc(Oc2cc(N)cc([N+](=O)[O-])c2)cc1 ZINC000147440401 CE For-Sale Bother CHEK2 28 50 NC(=O)c1ccc(Oc2cc(N)cc([N+](=O)[O-])c2)cc1 ZINC000147440401 CE For-Sale Bother PLAU 24 49 Nc1c(C(=O)Nc2ccc(Cl)cn2)oc2ccc(O)cc12 ZINC000147440413 DG For-Sale Anodyne F10 54 36 Cc1ccc(C(C)C)c(OCC(=O)Nc2ccc(Cl)c(C#N)c2)c1 ZINC000147440425 EJ On-Demand Mild CETP 31 40 Cc1ccc(C(C)C)c(OCC(=O)Nc2ccc(Cl)c(C#N)c2)c1 ZINC000147440425 EJ On-Demand Mild IMDH_CRYPV 16 43 COc1ncccc1OC[C@@H]1CCCN1C ZINC000147440495 BD Annotated Anodyne CHRNA3 36 44 COc1ncccc1OC[C@@H]1CCCN1C ZINC000147440495 BD Annotated Anodyne CHRNA4 17 44 COc1ncccc1OC[C@@H]1CCCN1C ZINC000147440495 BD Annotated Anodyne CHRNA10 83 64 COc1ncccc1OC[C@@H]1CCCN1C ZINC000147440495 BD Annotated Anodyne ACKR3 74 37 CN(CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147440516 HC On-Demand Anodyne CHRM5 19 40 CN(CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147440516 HC On-Demand Anodyne EPHX2 20 44 CN(CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147440516 HC On-Demand Anodyne TGM2 67 45 CN(CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147440516 HC On-Demand Anodyne CACNA1I 57 35 CN(CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)S(C)(=O)=O ZINC000147440516 HC On-Demand Anodyne F13A1 71 45 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne F2 38 44 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne PLG 50 42 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne PRSS1 21 44 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne CHRM1 19 44 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne ACE 41 42 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne DRD4 23 54 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne F10 22 40 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne CHRM3 17 42 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne TACR1 19 40 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne SIGMAR1 25 52 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne SSTR5 42 37 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne CTSB 18 41 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne TRY2_BOVIN 109 43 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne TRY1_BOVIN 17 43 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne CCKAR 0 50 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne NPY2R 37 43 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne CCR1 32 44 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne CCR3 53 42 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne C3AR1 44 37 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne DPP4 20 40 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne MLNR 25 43 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne CCKBR 47 41 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne EPHX2 28 44 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne ACE2 44 32 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne ST14 124 44 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne MCHR1 33 46 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne CCR8 41 41 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne BRCA1 43 32 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne TMPRSS6 70 40 C[C@H](Cc1cccc(F)c1)C(=O)N1CCC(NC(=O)c2ccccc2)CC1 ZINC000147440517 FG On-Demand Anodyne DERP1 0 44 O=C(O)[C@@H]1CCCN1C(=O)C[C@H]1CCc2ccccc21 ZINC000147440530 CE On-Demand Anodyne F2 20 50 O=C(O)[C@@H]1CCCN1C(=O)C[C@H]1CCc2ccccc21 ZINC000147440530 CE On-Demand Anodyne ACE 84 49 O=C(O)[C@@H]1CCCN1C(=O)C[C@H]1CCc2ccccc21 ZINC000147440530 CE On-Demand Anodyne SLC6A1 53 33 O=C(O)[C@@H]1CCCN1C(=O)C[C@H]1CCc2ccccc21 ZINC000147440530 CE On-Demand Anodyne MME 24 43 O=C(O)[C@@H]1CCCN1C(=O)C[C@H]1CCc2ccccc21 ZINC000147440530 CE On-Demand Anodyne CPT1A 17 42 O=C(O)[C@@H]1CCCN1C(=O)C[C@H]1CCc2ccccc21 ZINC000147440530 CE On-Demand Anodyne CPT2 43 40 O=C(O)[C@@H]1CCCN1C(=O)C[C@H]1CCc2ccccc21 ZINC000147440530 CE On-Demand Anodyne DPP4 15 43 O=C(O)[C@@H]1CCCN1C(=O)C[C@H]1CCc2ccccc21 ZINC000147440530 CE On-Demand Anodyne PREP 135 51 Cc1c(O)cccc1C(=O)N1CCC(N)CC1 ZINC000147440559 BD For-Sale Anodyne CHRM2 0 41 Cc1c(O)cccc1C(=O)N1CCC(N)CC1 ZINC000147440559 BD For-Sale Anodyne L3MBTL1 0 44 Cc1c(O)cccc1C(=O)N1CCC(N)CC1 ZINC000147440559 BD For-Sale Anodyne L3MBTL3 51 44 Cc1c(O)cccc1C(=O)N1CCC(N)CC1 ZINC000147440559 BD For-Sale Anodyne TP53BP1 0 44 Cc1cc(OC(C)C)ccc1NC(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147440568 GG On-Demand Bother GCK 30 45 CCCCO[C@@H](C)C(=O)Nc1ccc(NS(C)(=O)=O)c(OC)c1 ZINC000147440577 EE On-Demand Anodyne TRPV1 55 39 O=C(NCc1ccc(Cn2ccccc2=O)cc1)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147440578 GH On-Demand Anodyne PLD1 15 43 CCN(CC)[C@H](C)CNC(=O)c1cc2cc(Cl)ccc2[nH]1 ZINC000147440595 DG On-Demand Anodyne CYP51A1 22 40 CCN(CC)[C@H](C)CNC(=O)c1cc2cc(Cl)ccc2[nH]1 ZINC000147440595 DG On-Demand Anodyne PYGL 112 62 CCN(CC)[C@H](C)CNC(=O)c1cc2cc(Cl)ccc2[nH]1 ZINC000147440595 DG On-Demand Anodyne PYGM 24 41 CCN(CC)[C@H](C)CNC(=O)c1cc2cc(Cl)ccc2[nH]1 ZINC000147440595 DG On-Demand Anodyne ALPL 45 47 CCN(CC)[C@H](C)CNC(=O)c1cc2cc(Cl)ccc2[nH]1 ZINC000147440595 DG On-Demand Anodyne PYK 23 41 CC[C@@H]1CN(C[C@H](O)c2ccccc2)CC[C@@H]1N ZINC000147440605 BD For-Sale Anodyne OPRK1 29 51 CC[C@@H]1CN(C[C@H](O)c2ccccc2)CC[C@@H]1N ZINC000147440605 BD For-Sale Anodyne IGF1R 0 44 CC[C@@H]1CN(C[C@H](O)c2ccccc2)CC[C@@H]1N ZINC000147440605 BD For-Sale Anodyne CCR5 37 40 CC[C@@H]1CN(C[C@H](O)c2ccccc2)CC[C@@H]1N ZINC000147440605 BD For-Sale Anodyne SLC18A3 23 41 C[C@@H]1CCc2ccccc2N1C(=O)C1(N)CCC1 ZINC000147440637 BE For-Sale Anodyne ACE 24 42 C[C@@H]1CCc2ccccc2N1C(=O)C1(N)CCC1 ZINC000147440637 BE For-Sale Anodyne DRD4 26 42 CCOC(=O)[C@@H]1CCCN(S(=O)(=O)N2C[C@H](C)O[C@H](c3ccccc3)C2)C1 ZINC000147440673 GD On-Demand Anodyne SLC6A1 57 34 COc1cc(OCC(=O)N2CCC(NC(=O)c3ccccc3)CC2)ccc1[N+](=O)[O-] ZINC000147440711 HE On-Demand Bother DRD4 25 42 COc1cc(OCC(=O)N2CCC(NC(=O)c3ccccc3)CC2)ccc1[N+](=O)[O-] ZINC000147440711 HE On-Demand Bother HTR1D 15 40 COc1cc(OCC(=O)N2CCC(NC(=O)c3ccccc3)CC2)ccc1[N+](=O)[O-] ZINC000147440711 HE On-Demand Bother SSTR5 39 40 COc1cc(OCC(=O)N2CCC(NC(=O)c3ccccc3)CC2)ccc1[N+](=O)[O-] ZINC000147440711 HE On-Demand Bother KCNA3 15 41 COc1cc(OCC(=O)N2CCC(NC(=O)c3ccccc3)CC2)ccc1[N+](=O)[O-] ZINC000147440711 HE On-Demand Bother CPT1A 35 40 COc1cc(OCC(=O)N2CCC(NC(=O)c3ccccc3)CC2)ccc1[N+](=O)[O-] ZINC000147440711 HE On-Demand Bother CPT2 41 37 COc1cc(OCC(=O)N2CCC(NC(=O)c3ccccc3)CC2)ccc1[N+](=O)[O-] ZINC000147440711 HE On-Demand Bother MCHR1 20 43 COc1cc(OCC(=O)N2CCC(NC(=O)c3ccccc3)CC2)ccc1[N+](=O)[O-] ZINC000147440711 HE On-Demand Bother SHH 22 41 CCC(CC)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440727 FF On-Demand Anodyne HTR4 58 38 CCC(CC)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440727 FF On-Demand Anodyne CHRM5 27 44 CCC(CC)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440727 FF On-Demand Anodyne MMP13 27 42 CCC(CC)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440727 FF On-Demand Anodyne TGM2 68 47 CCC(CC)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440727 FF On-Demand Anodyne MMP1 21 42 CCC(CC)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440727 FF On-Demand Anodyne CACNA1I 55 38 CCC(CC)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440727 FF On-Demand Anodyne F13A1 81 47 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc(C#N)cc3)CC2)s1 ZINC000147440731 GD On-Demand Mild TGM2 60 35 CCc1ncc(C(=O)N2CCN(S(=O)(=O)c3ccc(C#N)cc3)CC2)s1 ZINC000147440731 GD On-Demand Mild F13A1 60 35 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3cccc(-n4cccn4)c3)c2)CCO1 ZINC000147440782 HG On-Demand Anodyne HRH2 40 35 C[C@@H]1CN(Cc2cccc(CNC(=O)Nc3cccc(-n4cccn4)c3)c2)CCO1 ZINC000147440782 HG On-Demand Anodyne CCR3 28 41 O=C(NCc1ccc(Cn2ccccc2=O)cc1)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147440795 GH On-Demand Anodyne PLD1 15 43 CCCCO[C@H](C)C(=O)Nc1ccc(NS(C)(=O)=O)c(OC)c1 ZINC000147440805 EE On-Demand Anodyne TRPV1 55 39 CCCOc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1Cl ZINC000147440819 HH On-Demand Bother USP7 43 36 CCCOc1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1Cl ZINC000147440819 HH On-Demand Bother USP47 53 36 CCN(CC)[C@@H](C)CNC(=O)c1cc2cc(Br)ccc2[nH]1 ZINC000147440826 FG On-Demand Anodyne PYGL 73 50 CCN(CC)[C@@H](C)CNC(=O)c1cc2cc(Br)ccc2[nH]1 ZINC000147440826 FG On-Demand Anodyne PYGM 15 41 CCN(CC)[C@@H](C)CNC(=O)c1cc2cc(Br)ccc2[nH]1 ZINC000147440826 FG On-Demand Anodyne PYK 69 49 C[C@H]1CCc2ccccc2N1C(=O)C1(N)CCC1 ZINC000147440845 BE For-Sale Anodyne ACE 24 42 C[C@H]1CCc2ccccc2N1C(=O)C1(N)CCC1 ZINC000147440845 BE For-Sale Anodyne DRD4 26 42 NC(=O)c1ccc(Oc2nc(N)nc3ccccc23)cc1 ZINC000147440897 CE For-Sale Anodyne CHEK2 46 43 N#CCSCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440983 FD On-Demand Mild TGM2 62 44 N#CCSCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147440983 FD On-Demand Mild F13A1 69 44 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3cccc(-n4cccn4)c3)c2)CCO1 ZINC000147440999 HG On-Demand Anodyne HRH2 40 35 C[C@H]1CN(Cc2cccc(CNC(=O)Nc3cccc(-n4cccn4)c3)c2)CCO1 ZINC000147440999 HG On-Demand Anodyne CCR3 28 41 O=C(NCc1ccc(Cn2ccccc2=O)cc1)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147441000 GH On-Demand Anodyne PLD1 15 43 CCN(CC)[C@H](C)CNC(=O)c1cc2cc(Br)ccc2[nH]1 ZINC000147441038 FG On-Demand Anodyne PYGL 85 50 CCN(CC)[C@H](C)CNC(=O)c1cc2cc(Br)ccc2[nH]1 ZINC000147441038 FG On-Demand Anodyne PYGM 18 41 CCN(CC)[C@H](C)CNC(=O)c1cc2cc(Br)ccc2[nH]1 ZINC000147441038 FG On-Demand Anodyne PYK 69 49 C[C@@H]1CCc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147441076 CF For-Sale Anodyne ACE 19 41 C[C@@H]1CCc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147441076 CF For-Sale Anodyne DRD4 24 41 C[C@@H]1CCc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147441076 CF For-Sale Anodyne CACNA2D1 47 39 C[C@@H]1CCc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147441076 CF For-Sale Anodyne TPP2 55 37 Cc1csc(NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)n1 ZINC000147441091 DE On-Demand Anodyne GCK 20 41 Cc1csc(NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)n1 ZINC000147441091 DE On-Demand Anodyne TRPC6 45 33 O=C(NCc1cn[nH]c1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147441135 EE For-Sale Anodyne ROCK2 21 47 O=C(NCc1ccc(Cn2ccccc2=O)cc1)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147441140 GH On-Demand Anodyne PLD1 15 43 O=C(CNc1ccc2cc(Br)ccc2c1)N1CCOCC1 ZINC000147441157 EF On-Demand Anodyne AKR1C3 24 41 COCCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147441161 DB For-Sale Anodyne CA2 52 42 COCCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147441161 DB For-Sale Anodyne CA1 35 42 COCCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147441161 DB For-Sale Anodyne CA4 42 42 COCCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147441161 DB For-Sale Anodyne CA12 23 42 COCCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147441161 DB For-Sale Anodyne CA9 31 42 COCCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147441161 DB For-Sale Anodyne NCE103 16 40 CN1CC[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441192 GD On-Demand Anodyne CHRM5 18 40 CN1CC[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441192 GD On-Demand Anodyne EPHX2 41 47 CN1CC[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441192 GD On-Demand Anodyne TGM2 62 43 CN1CC[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441192 GD On-Demand Anodyne F13A1 61 43 C[C@@H]1CCCN1CCS(=O)(=O)c1cccc(C#N)c1 ZINC000147441283 CD On-Demand Mild KCNH2 0 47 C[C@H]1CCc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147441293 CF For-Sale Anodyne ACE 19 41 C[C@H]1CCc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147441293 CF For-Sale Anodyne DRD4 24 41 C[C@H]1CCc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147441293 CF For-Sale Anodyne CACNA2D1 47 39 C[C@H]1CCc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147441293 CF For-Sale Anodyne TPP2 55 37 COC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147441300 BC For-Sale Anodyne SIRT1 26 40 COc1cc(NC(=O)Cc2c(C)nn(C(F)F)c2C)ccc1NS(C)(=O)=O ZINC000147441304 HE On-Demand Anodyne ENPP1 69 34 O=C(c1ccccc1OC(F)F)N1CCC[C@@H]1CCCBr ZINC000147441307 FI For-Sale Reactive HCRTR1 19 45 O=C(NCc1cn[nH]c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147441321 CE For-Sale Anodyne ROCK2 22 50 COC(=O)c1cc(NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)cc(C(=O)OC)c1 ZINC000147441330 HE On-Demand Anodyne EPHX2 17 40 CO[C@H]1O[C@H](CBr)[C@@H](O)[C@H](O)[C@@H]1O ZINC000147441371 CA Annotated Reactive FIMH 64 42 CC[C@@H](C)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147441379 DC For-Sale Anodyne CA2 36 45 CN1CC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441384 GD On-Demand Anodyne CHRM5 18 40 CN1CC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441384 GD On-Demand Anodyne EPHX2 41 47 CN1CC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441384 GD On-Demand Anodyne TGM2 62 43 CN1CC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441384 GD On-Demand Anodyne F13A1 61 43 CCNc1nc(C)cc(Oc2ccc(C(N)=O)cc2)n1 ZINC000147441401 CE For-Sale Anodyne CHEK2 39 40 NC1(C(=O)NC23CC4CC(CC(C4)C2)C3)CCC1 ZINC000147441507 BD For-Sale Anodyne P95276_MYCTO 0 45 C[C@H]1CCCN1CCS(=O)(=O)c1cccc(C#N)c1 ZINC000147441510 CD On-Demand Mild KCNH2 0 47 O=C(c1ccccc1OC(F)F)N1CCC[C@H]1CCCBr ZINC000147441528 FI For-Sale Reactive HCRTR1 19 45 COC[C@H](N)C(=O)NCCCCC(C)C ZINC000147441549 BC For-Sale Anodyne SIRT1 26 40 CC[C@H](C)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147441577 DC For-Sale Anodyne CA2 36 45 CN1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441581 GC On-Demand Anodyne FKBP1A 24 40 CN1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441581 GC On-Demand Anodyne CHRM5 18 40 CN1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441581 GC On-Demand Anodyne P2RX7 15 47 CN1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441581 GC On-Demand Anodyne EPHX2 38 44 CN1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441581 GC On-Demand Anodyne TGM2 63 43 CN1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147441581 GC On-Demand Anodyne F13A1 64 43 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)C1 ZINC000147441642 HH On-Demand Anodyne RAF1 25 42 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)C1 ZINC000147441642 HH On-Demand Anodyne ENV 43 33 NC(=O)c1ccc(Oc2nc(N)nc(Cl)n2)cc1 ZINC000147441669 CC For-Sale Anodyne CHEK2 36 42 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2c2ccc(Cl)cc2)no1 ZINC000147441671 EI Annotated Anodyne FLT3 48 39 NCC1(CC(=O)NC23CC4CC(CC(C4)C2)C3)CCC1 ZINC000147441757 CF For-Sale Anodyne CACNA2D1 38 43 NCC1(CC(=O)NC23CC4CC(CC(C4)C2)C3)CCC1 ZINC000147441757 CF For-Sale Anodyne EPHX2 60 46 NCC1(CC(=O)NC23CC4CC(CC(C4)C2)C3)CCC1 ZINC000147441757 CF For-Sale Anodyne P95276_MYCTO 0 40 CCNC(=O)CN(C)C(=O)c1ccccc1Nc1ccc(OC(F)F)cc1 ZINC000147441803 GG On-Demand Anodyne AKR1C3 16 42 CCNC(=O)CN(C)C(=O)c1ccccc1Nc1ccc(OC(F)F)cc1 ZINC000147441803 GG On-Demand Anodyne AKR1C2 39 42 CCOC(=O)c1csc(-c2ccccc2[N+](=O)[O-])n1 ZINC000147441810 CF On-Demand Bother GSTM2 24 41 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)C1 ZINC000147441830 HH On-Demand Anodyne RAF1 25 42 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)C1 ZINC000147441830 HH On-Demand Anodyne ENV 43 33 NS(=O)(=O)c1cc(F)c(OCC(=O)NCC2CC2)c(F)c1 ZINC000147441833 DC For-Sale Anodyne CA2 26 42 Cc1cc(S(=O)(=O)NCCc2cnn(-c3ccccc3)c2)ccc1Br ZINC000147441851 HG On-Demand Anodyne TBXA2R 41 34 Cc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)c(C)c1 ZINC000147441857 FE For-Sale Reactive EPHX2 32 50 CCNc1nc(Cl)nc(Oc2ccc(C(N)=O)cc2)n1 ZINC000147441902 CD For-Sale Anodyne PPX1 0 44 CC(C)CCCCNC[C@H](O)COc1ccc(Cl)c(Cl)c1 ZINC000147441981 EI For-Sale Anodyne ADRB2 65 47 CC(C)CCCCNC[C@H](O)COc1ccc(Cl)c(Cl)c1 ZINC000147441981 EI For-Sale Anodyne ADRB1 76 45 CC(C)CCCCNC[C@H](O)COc1ccc(Cl)c(Cl)c1 ZINC000147441981 EI For-Sale Anodyne GRIN1 43 52 CC(C)CCCCNC[C@H](O)COc1ccc(Cl)c(Cl)c1 ZINC000147441981 EI For-Sale Anodyne ADRB3 55 45 NCC1(CC(=O)NCc2ccccc2)CCC1 ZINC000147441986 BD For-Sale Anodyne CACNA2D1 37 46 NCC1(CC(=O)NCc2ccccc2)CCC1 ZINC000147441986 BD For-Sale Anodyne SLC12A5 54 37 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(F)c3)c2)c1 ZINC000147441987 HI On-Demand Bother PYGL 27 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(F)c3)c2)c1 ZINC000147441987 HI On-Demand Bother BTK 24 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(F)c3)c2)c1 ZINC000147441987 HI On-Demand Bother TAAR1 58 63 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(F)c3)c2)c1 ZINC000147441987 HI On-Demand Bother AKR1C3 30 53 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(F)c3)c2)c1 ZINC000147441987 HI On-Demand Bother AKR1C2 42 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(F)c3)c2)c1 ZINC000147441987 HI On-Demand Bother KCNK3 130 53 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(F)c3)c2)c1 ZINC000147441987 HI On-Demand Bother KCNK9 89 47 CCN1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147442008 GD On-Demand Anodyne CHRM5 20 41 CCN1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147442008 GD On-Demand Anodyne EPHX2 37 45 CCN1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147442008 GD On-Demand Anodyne TGM2 54 42 CCN1C[C@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1=O ZINC000147442008 GD On-Demand Anodyne F13A1 53 42 NS(=O)(=O)c1cc(F)c(OCCn2ccnc2)c(F)c1 ZINC000147442087 DC For-Sale Anodyne CYP11B1 0 44 NS(=O)(=O)c1cc(F)c(OCCn2ccnc2)c(F)c1 ZINC000147442087 DC For-Sale Anodyne TBXAS1 38 45 CNc1cc(Oc2ccc(C(N)=O)cc2)cc([N+](=O)[O-])c1 ZINC000147442091 CF For-Sale Bother CHEK2 21 44 CNc1cc(Oc2ccc(C(N)=O)cc2)cc([N+](=O)[O-])c1 ZINC000147442091 CF For-Sale Bother PLAU 25 43 CNc1cc(Oc2ccc(C(N)=O)cc2)cc([N+](=O)[O-])c1 ZINC000147442091 CF For-Sale Bother ERO1A 0 40 Cc1ccc([C@@]2(C)NC(=O)N(Cc3nc(-c4ccccc4)oc3C)C2=O)cc1 ZINC000147442093 GH On-Demand Anodyne PPARG 72 39 Cc1ccc([C@@]2(C)NC(=O)N(Cc3nc(-c4ccccc4)oc3C)C2=O)cc1 ZINC000147442093 GH On-Demand Anodyne PPARA 78 39 Cc1ccc([C@@]2(C)NC(=O)N(Cc3nc(-c4ccccc4)oc3C)C2=O)cc1 ZINC000147442093 GH On-Demand Anodyne PDE8B 67 39 CC(C)CCCCNC[C@@H](O)COc1ccc(Cl)c(Cl)c1 ZINC000147442169 EI For-Sale Anodyne ADRB2 65 47 CC(C)CCCCNC[C@@H](O)COc1ccc(Cl)c(Cl)c1 ZINC000147442169 EI For-Sale Anodyne ADRB1 76 45 CC(C)CCCCNC[C@@H](O)COc1ccc(Cl)c(Cl)c1 ZINC000147442169 EI For-Sale Anodyne GRIN1 43 52 CC(C)CCCCNC[C@@H](O)COc1ccc(Cl)c(Cl)c1 ZINC000147442169 EI For-Sale Anodyne ADRB3 55 45 O=C(O)Cc1csc(Nc2cc(Cl)ccc2Br)n1 ZINC000147442183 EH For-Sale Anodyne CXCL8 17 40 O=C(O)Cc1csc(Nc2cc(Cl)ccc2Br)n1 ZINC000147442183 EH For-Sale Anodyne COLA 0 43 O=C(O)Cc1csc(Nc2cc(Cl)ccc2Br)n1 ZINC000147442183 EH For-Sale Anodyne CPT1A 30 43 O=C(O)Cc1csc(Nc2cc(Cl)ccc2Br)n1 ZINC000147442183 EH For-Sale Anodyne CPT1B 41 39 Cc1ccc([C@]2(C)NC(=O)N(Cc3nc(-c4ccccc4)oc3C)C2=O)cc1 ZINC000147442269 GH On-Demand Anodyne PPARG 72 39 Cc1ccc([C@]2(C)NC(=O)N(Cc3nc(-c4ccccc4)oc3C)C2=O)cc1 ZINC000147442269 GH On-Demand Anodyne PPARA 78 39 Cc1ccc([C@]2(C)NC(=O)N(Cc3nc(-c4ccccc4)oc3C)C2=O)cc1 ZINC000147442269 GH On-Demand Anodyne PDE8B 67 39 C[C@H](OC[C@@H]1CCCO1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147442278 HD On-Demand Anodyne CCR8 79 36 COc1cc(Cl)c(C)cc1NC(=O)Nc1ccc2c(c1)n(C)c(=O)n2C ZINC000147442283 FG On-Demand Anodyne HTR2A 33 40 COc1cc(Cl)c(C)cc1NC(=O)Nc1ccc2c(c1)n(C)c(=O)n2C ZINC000147442283 FG On-Demand Anodyne RAF1 19 40 COc1ccc(NC(=O)C2(N)CCC2)c(OC)c1 ZINC000147442284 CD For-Sale Anodyne CYP1B1 39 55 COc1ccc(NC(=O)C2(N)CCC2)c(OC)c1 ZINC000147442284 CD For-Sale Anodyne LUCI_LUCLA 15 40 COc1ccc(NC(=O)C2(N)CCC2)c(OC)c1 ZINC000147442284 CD For-Sale Anodyne AKR1C2 45 34 COc1ccc(NC(=O)C2(N)CCC2)c(OC)c1 ZINC000147442284 CD For-Sale Anodyne ACAT 0 44 CC(C)CCCCNCCCC(=O)O ZINC000147442405 BE For-Sale Anodyne Q6UB75_PIG 0 40 C[C@@H](OC[C@@H]1CCCO1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147442479 HD On-Demand Anodyne CCR8 79 36 COc1ccc(NC(=O)CC2(CN)CCC2)c(OC)c1 ZINC000147442487 CE For-Sale Anodyne MTNR1A 68 41 COc1ccc(NC(=O)CC2(CN)CCC2)c(OC)c1 ZINC000147442487 CE For-Sale Anodyne MTNR1B 63 41 COc1ccc(NC(=O)CC2(CN)CCC2)c(OC)c1 ZINC000147442487 CE For-Sale Anodyne ACAT 0 47 NS(=O)(=O)c1cc(F)c(OCCCn2ccnc2)c(F)c1 ZINC000147442496 DD For-Sale Anodyne TBXAS1 43 43 NS(=O)(=O)c1cc(F)c(OCCCn2ccnc2)c(F)c1 ZINC000147442496 DD For-Sale Anodyne HMOX2 49 40 COc1ccc(NC(=O)NC[C@@H](O)COc2c(C)cccc2C)c(C(F)(F)F)c1 ZINC000147442499 HH On-Demand Anodyne ADRB2 19 40 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild GRIN2B 48 50 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild SIGMAR1 30 41 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild TRY1_BOVIN 18 41 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild CCR5 16 41 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild HDAC8 44 39 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild HDAC10 46 39 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild PREP 55 47 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild MMP2 67 33 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild MMP3 24 40 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild HDAC1 39 60 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild HDAC2 34 60 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild FAAH 26 43 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild MMP1 17 40 O=C(CCCC1CCN(C(=O)CCCc2ccccc2)CC1)NO ZINC000147442514 EF For-Sale Mild AMP1_PLAFQ 34 42 COc1cc(Cl)c(C)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@H](C)C1 ZINC000147442524 GG On-Demand Anodyne HTR4 20 44 CC[C@@H]1CN(CC(=O)NCC2CC2)CC[C@@H]1N ZINC000147442545 BC On-Demand Anodyne CACNA1I 48 36 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442602 GF On-Demand Anodyne OPRM1 28 41 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442602 GF On-Demand Anodyne OPRD1 34 41 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442602 GF On-Demand Anodyne CTSB 15 40 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442602 GF On-Demand Anodyne TIMP3 62 38 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442602 GF On-Demand Anodyne MTNR1A 35 40 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442602 GF On-Demand Anodyne CAPN1 58 40 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442602 GF On-Demand Anodyne CAPN2 25 40 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442602 GF On-Demand Anodyne CTRB_BOVIN 40 39 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442602 GF On-Demand Anodyne FFAR1 20 42 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442602 GF On-Demand Anodyne PSMB8 61 37 C[C@H](OC[C@H]1CCCO1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147442667 HD On-Demand Anodyne CCR8 79 36 COc1ccc([N+](=O)[O-])c(NC[C@@H](C)CC(=O)O)c1 ZINC000147442681 CE On-Demand Bother AKR1C3 19 42 COc1ccc([N+](=O)[O-])c(NC[C@@H](C)CC(=O)O)c1 ZINC000147442681 CE On-Demand Bother AKR1C2 50 44 C=CCOc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147442695 HG On-Demand Mild HTR4 44 37 C=CCOc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147442695 HG On-Demand Mild KCNA3 44 39 C=CCOc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147442695 HG On-Demand Mild TGM2 94 49 C=CCOc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147442695 HG On-Demand Mild CACNA1I 41 31 C=CCOc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147442695 HG On-Demand Mild F13A1 98 49 C=CCOc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147442695 HG On-Demand Mild HCN1 77 37 C=CCOc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147442695 HG On-Demand Mild HCN4 54 36 COc1ccc(NC(=O)NC[C@H](O)COc2c(C)cccc2C)c(C(F)(F)F)c1 ZINC000147442708 HH On-Demand Anodyne ADRB2 19 40 Cc1ccc(Cl)c(NC(=O)C2(N)CCC2)c1Cl ZINC000147442711 CG For-Sale Anodyne FABP2 0 41 CC(C)(C)c1cc(NC(=O)[C@]2(C)CCCN2c2ccc(C(F)(F)F)cc2)no1 ZINC000147442712 GJ Annotated Anodyne FLT3 44 38 COc1cc(Cl)c(C)cc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@@H](C)C1 ZINC000147442751 GG On-Demand Anodyne HTR4 20 44 CC[C@H]1CN(CC(=O)NCC2CC2)CC[C@@H]1N ZINC000147442765 BC On-Demand Anodyne CACNA1I 48 36 C[C@@H](OC[C@H]1CCCO1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147442829 HD On-Demand Anodyne CCR8 79 36 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442831 GF On-Demand Anodyne OPRM1 28 41 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442831 GF On-Demand Anodyne OPRD1 34 41 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442831 GF On-Demand Anodyne CTSB 15 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442831 GF On-Demand Anodyne TIMP3 62 38 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442831 GF On-Demand Anodyne MTNR1A 35 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442831 GF On-Demand Anodyne CAPN1 58 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442831 GF On-Demand Anodyne CAPN2 25 40 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442831 GF On-Demand Anodyne CTRB_BOVIN 40 39 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442831 GF On-Demand Anodyne FFAR1 20 42 CCOC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147442831 GF On-Demand Anodyne PSMB8 61 37 CC(C)CCCCNC(=O)c1ccc2c(c1)CCCN2 ZINC000147442884 CH For-Sale Anodyne HDAC9 15 46 COc1ccc([N+](=O)[O-])c(NC[C@H](C)CC(=O)O)c1 ZINC000147442886 CE On-Demand Bother AKR1C3 19 42 COc1ccc([N+](=O)[O-])c(NC[C@H](C)CC(=O)O)c1 ZINC000147442886 CE On-Demand Bother AKR1C2 50 44 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne PLG 24 40 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne PRSS1 24 40 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne DRD4 41 33 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne HTR4 54 36 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne F10 37 42 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne EPHX2 23 44 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne TGM2 70 46 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne ST14 87 35 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne CACNA1I 67 44 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne F13A1 67 46 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne AKR1C3 62 42 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne SFRP1 23 40 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne NAMPT 42 42 NC(=O)c1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147442927 HD On-Demand Anodyne TMPRSS6 66 33 Cc1cc(-c2ccncc2NC(=O)c2nc(-c3c(F)cccc3F)ccc2N)cc(N)n1 ZINC000147442952 II Annotated Anodyne PIM1 36 46 Cc1cc(-c2ccncc2NC(=O)c2nc(-c3c(F)cccc3F)ccc2N)cc(N)n1 ZINC000147442952 II Annotated Anodyne PIM2 17 46 Cc1cc(-c2ccncc2NC(=O)c2nc(-c3c(F)cccc3F)ccc2N)cc(N)n1 ZINC000147442952 II Annotated Anodyne PIM3 24 46 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147443029 GF On-Demand Anodyne OPRM1 28 41 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147443029 GF On-Demand Anodyne OPRD1 34 41 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147443029 GF On-Demand Anodyne CTSB 15 40 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147443029 GF On-Demand Anodyne TIMP3 62 38 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147443029 GF On-Demand Anodyne MTNR1A 35 40 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147443029 GF On-Demand Anodyne CAPN1 58 40 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147443029 GF On-Demand Anodyne CAPN2 25 40 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147443029 GF On-Demand Anodyne CTRB_BOVIN 40 39 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147443029 GF On-Demand Anodyne FFAR1 20 42 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@@H]1COc2cc(OC)ccc2C1 ZINC000147443029 GF On-Demand Anodyne PSMB8 61 37 O=C(O)c1nc(-c2ccccc2)cnc1O ZINC000147443043 BD For-Sale Anodyne PRKDC 25 50 O=C(O)c1nc(-c2ccccc2)cnc1O ZINC000147443043 BD For-Sale Anodyne ATR 59 50 COc1ccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147443112 FI On-Demand Anodyne MTNR1A 17 41 COc1ccc(NC(=O)N[C@@H]2C[C@@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147443112 FI On-Demand Anodyne EPHX2 31 47 COc1ccc(NC(=O)C2(N)CCC2)cc1Cl ZINC000147443131 CE On-Demand Anodyne QRFPR 40 35 COc1ccc(NC(=O)C2(N)CCC2)cc1Cl ZINC000147443131 CE On-Demand Anodyne ENPP1 40 31 CCCCC[C@@H](CN)NCC(F)F ZINC000147443146 AD For-Sale Anodyne Q6UB75_PIG 0 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(C2CC2)[nH]n1 ZINC000147443181 GE On-Demand Anodyne GRIN2B 27 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(C2CC2)[nH]n1 ZINC000147443181 GE On-Demand Anodyne EPHX2 16 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(C2CC2)[nH]n1 ZINC000147443181 GE On-Demand Anodyne TGM2 56 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(C2CC2)[nH]n1 ZINC000147443181 GE On-Demand Anodyne CACNA1I 59 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(C2CC2)[nH]n1 ZINC000147443181 GE On-Demand Anodyne F13A1 43 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(C2CC2)[nH]n1 ZINC000147443181 GE On-Demand Anodyne NAMPT 36 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(C2CC2)[nH]n1 ZINC000147443181 GE On-Demand Anodyne PKNB 56 42 Cc1cc(NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)n(-c2ccccn2)n1 ZINC000147443184 GE On-Demand Anodyne SLC11A2 49 37 COc1ccc(N2CCOCC2)c2sc(NC(=O)N3CCC(N4CCCCC4)CC3)nc12 ZINC000147443204 JH For-Sale Clean ADORA2B 17 43 COc1ccc(N2CCOCC2)c2sc(NC(=O)N3CCC(N4CCCCC4)CC3)nc12 ZINC000147443204 JH For-Sale Clean MTOR 21 44 COc1ccc(N2CCOCC2)c2sc(NC(=O)N3CCC(N4CCCCC4)CC3)nc12 ZINC000147443204 JH For-Sale Clean L3MBTL3 74 38 CN(C)C(=O)NCCNC(=O)c1ccc([N+](=O)[O-])c(N)c1 ZINC000147443208 CC For-Sale Bother GSTM2 42 40 CCCc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147443232 GE For-Sale Reactive ADORA2B 56 39 CCCc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147443232 GE For-Sale Reactive PKM 19 42 CCCc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147443232 GE For-Sale Reactive TGM2 27 42 CCCc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1 ZINC000147443232 GE For-Sale Reactive F13A1 33 42 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne ACE 41 37 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne MME 66 37 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne ANPEP 66 37 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne TACR1 15 45 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne CTRA_BOVIN 48 38 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne CTSB 58 38 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne PAPA1_CARPA 50 42 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne CYSP_TRYCR 50 38 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne CTSL 38 42 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne CCR3 25 67 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne TIMP3 65 34 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne CAPNS1 54 34 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne HLA-DRB1 46 36 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne LNPEP 31 41 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne CTSS 28 42 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne CAPN1 56 44 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne MMP9 22 45 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne CAPN2 45 40 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne ACE2 68 37 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne PIN1 35 40 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne MMP1 16 45 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne CTRB_BOVIN 72 46 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne NPR 41 41 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne BLA1_STEMA 53 39 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne ERAP2 53 41 CCOC(=O)[C@@H](Cc1ccccc1)NC(=O)c1ccc2c(c1)COC2 ZINC000147443265 EF On-Demand Anodyne PSMB8 42 36 Clc1cccc(-c2c(Cl)nc(-c3cncs3)nc2Cl)c1 ZINC000147443287 EK For-Sale Anodyne CD38 24 40 COc1ccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147443298 FI On-Demand Anodyne MTNR1A 17 41 COc1ccc(NC(=O)N[C@H]2C[C@@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147443298 FI On-Demand Anodyne EPHX2 31 47 CCc1cc2cccc(Br)c2o1 ZINC000147443344 BH For-Sale Anodyne SLC22A12 35 40 CCCCC[C@H](CN)NCC(F)F ZINC000147443349 AD For-Sale Anodyne Q6UB75_PIG 0 41 COc1ccc(NC(=O)CC2(CN)CCC2)cc1Cl ZINC000147443357 CF For-Sale Anodyne GRM4 15 46 COc1ccc(NC(=O)CC2(CN)CCC2)cc1Cl ZINC000147443357 CF For-Sale Anodyne QRFPR 40 35 COc1ccc(NC(=O)CC2(CN)CCC2)cc1Cl ZINC000147443357 CF For-Sale Anodyne ENPP1 73 37 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(C#N)c3)c2)c1 ZINC000147443358 HH On-Demand Mild TAAR1 49 57 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(C#N)c3)c2)c1 ZINC000147443358 HH On-Demand Mild AKR1C3 25 50 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(C#N)c3)c2)c1 ZINC000147443358 HH On-Demand Mild AKR1C2 37 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(C#N)c3)c2)c1 ZINC000147443358 HH On-Demand Mild KCNK3 116 50 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(C(=O)Nc3cccc(C#N)c3)c2)c1 ZINC000147443358 HH On-Demand Mild KCNK9 77 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443371 GC On-Demand Anodyne F2 37 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443371 GC On-Demand Anodyne P2RY12 182 37 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443371 GC On-Demand Anodyne TRY2_BOVIN 84 39 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443371 GC On-Demand Anodyne TGM2 67 36 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443371 GC On-Demand Anodyne ST14 70 39 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443371 GC On-Demand Anodyne F13A1 59 36 CCCC[C@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443371 GC On-Demand Anodyne TMPRSS6 40 31 Cc1nc(N)cc(Oc2ccc(C(N)=O)cc2)n1 ZINC000147443429 BD For-Sale Anodyne TRY1_BOVIN 19 42 CCCC[C@H](O)[C@@H]1Cc2ccccc2O1 ZINC000147443431 BF For-Sale Anodyne MT-ND1 44 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1CCCc2ccccc21 ZINC000147443480 HG On-Demand Anodyne EPHX2 22 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1CCCc2ccccc21 ZINC000147443480 HG On-Demand Anodyne TGM2 56 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1CCCc2ccccc21 ZINC000147443480 HG On-Demand Anodyne F13A1 52 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1CCCc2ccccc21 ZINC000147443480 HG On-Demand Anodyne AKR1C3 61 39 COc1ccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147443489 FI On-Demand Anodyne MTNR1A 17 41 COc1ccc(NC(=O)N[C@@H]2C[C@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147443489 FI On-Demand Anodyne EPHX2 31 47 COC(=O)c1cccc(-c2cscn2)c1 ZINC000147443491 BF On-Demand Anodyne KDM3A 0 48 COC(=O)c1cccc(-c2cscn2)c1 ZINC000147443491 BF On-Demand Anodyne KDM5C 0 48 C[C@H](CNc1nc2ccccc2o1)CC(=O)O ZINC000147443531 BE On-Demand Anodyne ELANE 18 41 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147443533 HG On-Demand Anodyne F2 34 41 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147443533 HG On-Demand Anodyne TRY2_BOVIN 98 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147443533 HG On-Demand Anodyne MLNR 15 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147443533 HG On-Demand Anodyne ST14 112 41 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147443533 HG On-Demand Anodyne CCR8 73 40 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147443533 HG On-Demand Anodyne SFRP1 107 35 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147443533 HG On-Demand Anodyne WNT3 73 35 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCC(NS(=O)(=O)c2cccs2)CC1 ZINC000147443533 HG On-Demand Anodyne TMPRSS6 65 34 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cc(Cl)ccc1OC[C@@H]1CCCO1)C2 ZINC000147443556 HI On-Demand Anodyne ROCK2 30 45 NC1(C(=O)Nc2cccc3cccnc23)CCC1 ZINC000147443572 BE For-Sale Anodyne NFKBIA 0 40 NC1(C(=O)Nc2cccc3cccnc23)CCC1 ZINC000147443572 BE For-Sale Anodyne WNT3 15 42 NC1(C(=O)Nc2cccc3cccnc23)CCC1 ZINC000147443572 BE For-Sale Anodyne METAP2 0 43 NC1(C(=O)Nc2cccc3cccnc23)CCC1 ZINC000147443572 BE For-Sale Anodyne G2YM83_BOTF4 51 33 CCOCc1cccc2cccnc12 ZINC000147443590 AF For-Sale Anodyne CCR1 17 45 CCOCc1cccc2cccnc12 ZINC000147443590 AF For-Sale Anodyne METAP2 17 44 NS(=O)(=O)c1cc(F)c(OCCN2CCCC2)c(F)c1 ZINC000147443601 DD For-Sale Anodyne LTA4H 33 41 NS(=O)(=O)c1cc(F)c(OCCN2CCCC2)c(F)c1 ZINC000147443601 DD For-Sale Anodyne HRH3 17 51 NS(=O)(=O)c1cc(F)c(OCCN2CCCC2)c(F)c1 ZINC000147443601 DD For-Sale Anodyne PSMB2 46 37 NS(=O)(=O)c1cc(F)c(OCCN2CCCC2)c(F)c1 ZINC000147443601 DD For-Sale Anodyne PSMB1 40 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443606 GC On-Demand Anodyne F2 37 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443606 GC On-Demand Anodyne P2RY12 182 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443606 GC On-Demand Anodyne TRY2_BOVIN 84 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443606 GC On-Demand Anodyne TGM2 67 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443606 GC On-Demand Anodyne ST14 70 39 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443606 GC On-Demand Anodyne F13A1 59 36 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(S(=O)(=O)c2cccnc2)CC1 ZINC000147443606 GC On-Demand Anodyne TMPRSS6 40 31 O=C(OCc1ccccc1)c1cc(CN2CCOCC2)on1 ZINC000147443617 DD For-Sale Anodyne CASR 52 44 O=C(OCc1ccccc1)c1cc(CN2CCOCC2)on1 ZINC000147443617 DD For-Sale Anodyne PREP 25 43 O=C(OCc1ccccc1)c1cc(CN2CCOCC2)on1 ZINC000147443617 DD For-Sale Anodyne SLC12A5 50 32 Cc1nn(C)c(C)c1S(=O)(=O)N1CCN(CCBr)CC1 ZINC000147443628 FC For-Sale Reactive NMT1 35 41 CCCC[C@@H](O)[C@@H]1Cc2ccccc2O1 ZINC000147443647 BF For-Sale Anodyne MT-ND1 44 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1CCCc2ccccc21 ZINC000147443682 HG On-Demand Anodyne EPHX2 22 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1CCCc2ccccc21 ZINC000147443682 HG On-Demand Anodyne TGM2 56 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1CCCc2ccccc21 ZINC000147443682 HG On-Demand Anodyne F13A1 52 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1CCCc2ccccc21 ZINC000147443682 HG On-Demand Anodyne AKR1C3 61 39 COc1ccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147443683 FI On-Demand Anodyne MTNR1A 17 41 COc1ccc(NC(=O)N[C@H]2C[C@H]2c2ccccc2)c(C(F)(F)F)c1 ZINC000147443683 FI On-Demand Anodyne EPHX2 31 47 C[C@@H](CNc1nc2ccccc2o1)CC(=O)O ZINC000147443760 BE On-Demand Anodyne ELANE 18 41 O=C(NC1CCN(C(=O)c2csc(-c3ccccn3)n2)CC1)c1ccccc1 ZINC000147443801 GG On-Demand Anodyne DRD4 15 42 O=C(NC1CCN(C(=O)c2csc(-c3ccccn3)n2)CC1)c1ccccc1 ZINC000147443801 GG On-Demand Anodyne EPHX2 15 53 O=C(NC1CCN(C(=O)c2csc(-c3ccccn3)n2)CC1)c1ccccc1 ZINC000147443801 GG On-Demand Anodyne SFRP1 30 41 O=C(NC1CCN(C(=O)c2csc(-c3ccccn3)n2)CC1)c1ccccc1 ZINC000147443801 GG On-Demand Anodyne TRPC6 66 37 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cc(Cl)ccc1OC[C@@H]1CCCO1)C2 ZINC000147443802 HI On-Demand Anodyne ROCK2 30 45 CCCC[C@H](O)[C@H]1Cc2ccccc2O1 ZINC000147443818 BF For-Sale Anodyne MT-ND1 44 38 NCC1(CC(=O)Nc2cccc3cccnc23)CCC1 ZINC000147443830 CF For-Sale Anodyne WNT3 19 41 NCC1(CC(=O)Nc2cccc3cccnc23)CCC1 ZINC000147443830 CF For-Sale Anodyne TNKS 19 41 CNC(=O)CCCOc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147443831 DC For-Sale Anodyne CA2 38 43 CNC(=O)CCCOc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147443831 DC For-Sale Anodyne CA1 31 43 CNC(=O)CCCOc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147443831 DC For-Sale Anodyne CA4 36 43 Cc1cnc(NC(=O)Nc2ccc3c(c2)n(C)c(=O)n3C)s1 ZINC000147443852 DE On-Demand Anodyne CDK5 25 40 CCOc1ccccc1OCCNCCCCC(C)C ZINC000147443872 CH For-Sale Anodyne DRD4 20 41 CCOc1ccccc1OCCNCCCCC(C)C ZINC000147443872 CH For-Sale Anodyne ADRA1B 15 59 CCOc1ccccc1OCCNCCCCC(C)C ZINC000147443872 CH For-Sale Anodyne LMGT2 0 42 CC(C)(C)c1cc(NC(=O)[C@H]2CCCN2c2ccc(Cl)cc2)no1 ZINC000147443877 EI Annotated Anodyne CNR2 18 78 CC(C)(C)c1cc(NC(=O)[C@H]2CCCN2c2ccc(Cl)cc2)no1 ZINC000147443877 EI Annotated Anodyne FLT3 48 39 Cn1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1=O ZINC000147443899 GD On-Demand Anodyne HTR4 58 36 Cn1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1=O ZINC000147443899 GD On-Demand Anodyne EPHX2 29 43 Cn1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1=O ZINC000147443899 GD On-Demand Anodyne TGM2 63 44 Cn1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1=O ZINC000147443899 GD On-Demand Anodyne CACNA1I 68 43 Cn1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1=O ZINC000147443899 GD On-Demand Anodyne F13A1 53 42 Cn1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1=O ZINC000147443899 GD On-Demand Anodyne AKR1C3 44 36 COc1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147443900 GE On-Demand Anodyne EPHX2 52 42 COc1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147443900 GE On-Demand Anodyne RBP4 30 40 COc1ccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147443900 GE On-Demand Anodyne SFRP1 51 31 COc1cc(NC[C@@H](C)CC(=O)O)nc(C)n1 ZINC000147443997 BD For-Sale Anodyne ALS 53 32 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cc(Cl)ccc1OC[C@H]1CCCO1)C2 ZINC000147444003 HI On-Demand Anodyne ROCK2 30 45 CCCC[C@@H](O)[C@H]1Cc2ccccc2O1 ZINC000147444029 BF For-Sale Anodyne MT-ND1 44 38 COc1cccc([C@H](CNC(=O)C2(N)CCC2)N(C)C)c1 ZINC000147444042 CD On-Demand Anodyne OPRK1 0 43 CC(C)CCCCNC(=O)c1csc(N)n1 ZINC000147444103 BE For-Sale Anodyne HDAC3 15 45 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2C(=O)N2CCS(=O)(=O)CC2)no1 ZINC000147444108 GD Annotated Anodyne FLT3 42 36 O=C(NC1(CON2C(=O)c3ccccc3C2=O)CC1)OCc1ccccc1 ZINC000147444128 FF For-Sale Anodyne PAPA1_CARPA 44 35 O=C(NC1(CON2C(=O)c3ccccc3C2=O)CC1)OCc1ccccc1 ZINC000147444128 FF For-Sale Anodyne CTSK 17 42 O=C(NC1(CON2C(=O)c3ccccc3C2=O)CC1)OCc1ccccc1 ZINC000147444128 FF For-Sale Anodyne CAPNS1 51 32 O=C(NC1(CON2C(=O)c3ccccc3C2=O)CC1)OCc1ccccc1 ZINC000147444128 FF For-Sale Anodyne NPR 51 32 O=C(NC1(CON2C(=O)c3ccccc3C2=O)CC1)OCc1ccccc1 ZINC000147444128 FF For-Sale Anodyne SLC12A5 61 38 COc1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147444133 GE On-Demand Anodyne EPHX2 52 42 COc1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147444133 GE On-Demand Anodyne RBP4 30 40 COc1ccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c(C(F)(F)F)c1 ZINC000147444133 GE On-Demand Anodyne SFRP1 51 31 O=C(CCc1ccccc1O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444160 HF On-Demand Anodyne EPHX2 17 44 O=C(CCc1ccccc1O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444160 HF On-Demand Anodyne TGM2 77 45 O=C(CCc1ccccc1O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444160 HF On-Demand Anodyne F13A1 82 45 COc1cc(NC[C@H](C)CC(=O)O)nc(C)n1 ZINC000147444206 BD For-Sale Anodyne ALS 53 32 O=C(Nc1ccc2c(c1)CCO2)c1ccc(Br)c(Cl)c1 ZINC000147444238 FI On-Demand Anodyne PLAU 15 43 O=C(Nc1ccc2c(c1)CCO2)c1ccc(Br)c(Cl)c1 ZINC000147444238 FI On-Demand Anodyne TAAR1 28 40 C[C@H]1CN(S(=O)(=O)c2ccc(N3CCCC3=O)cc2)C[C@H](c2ccccc2)O1 ZINC000147444248 HF On-Demand Anodyne AKR1C3 40 57 COc1cccc([C@@H](CNC(=O)C2(N)CCC2)N(C)C)c1 ZINC000147444261 CD On-Demand Anodyne OPRK1 0 43 Cc1cc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)ccc1Br ZINC000147444281 HG On-Demand Anodyne DHODH 15 42 CC(C)CCCCNC[C@H](O)c1ccc(C(C)C)cc1 ZINC000147444315 CI For-Sale Anodyne ADRB2 31 40 CC(C)CCCCNC[C@H](O)c1ccc(C(C)C)cc1 ZINC000147444315 CI For-Sale Anodyne ADRB1 18 40 NS(=O)(=O)c1cc(F)c(OCCc2cccnc2)c(F)c1 ZINC000147444325 DD For-Sale Anodyne CA2 18 43 NS(=O)(=O)c1cc(F)c(OCCc2cccnc2)c(F)c1 ZINC000147444325 DD For-Sale Anodyne CA7 20 43 NS(=O)(=O)c1cc(F)c(OCCc2cccnc2)c(F)c1 ZINC000147444325 DD For-Sale Anodyne ISPH 0 40 CCO[C@@H]1CCCN(C(=O)Nc2ccc(OC)cc2C(F)(F)F)C1 ZINC000147444347 EH On-Demand Anodyne RBP4 63 39 CCO[C@@H]1CCCN(C(=O)Nc2ccc(OC)cc2C(F)(F)F)C1 ZINC000147444347 EH On-Demand Anodyne SFRP1 43 33 CCO[C@@H]1CCCN(C(=O)Nc2ccc(OC)cc2C(F)(F)F)C1 ZINC000147444347 EH On-Demand Anodyne WNT3 43 33 CS(=O)(=O)NCCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444417 HC On-Demand Anodyne HTR4 38 43 CS(=O)(=O)NCCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444417 HC On-Demand Anodyne EPHX2 21 44 CS(=O)(=O)NCCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444417 HC On-Demand Anodyne TGM2 79 45 CS(=O)(=O)NCCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444417 HC On-Demand Anodyne CACNA1I 41 35 CS(=O)(=O)NCCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444417 HC On-Demand Anodyne F13A1 83 45 O=S(=O)(c1ccc(F)c(F)c1)N1CCN(CCBr)CC1 ZINC000147444438 FD For-Sale Reactive PKM 52 43 Cc1cc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)ccc1Br ZINC000147444475 HG On-Demand Anodyne DHODH 15 42 Cc1ccc(Br)c(C(=O)Nc2ccc3c(c2)CCO3)c1 ZINC000147444483 EH On-Demand Anodyne KCNK3 51 33 CCOc1ccccc1NC(=O)C1(N)CCC1 ZINC000147444492 BD For-Sale Anodyne HCN1 48 37 CCOc1ccccc1NC(=O)C1(N)CCC1 ZINC000147444492 BD For-Sale Anodyne HCN4 48 37 CC(C)CCCCNC[C@@H](O)c1ccc(C(C)C)cc1 ZINC000147444495 CI For-Sale Anodyne ADRB2 31 40 CC(C)CCCCNC[C@@H](O)c1ccc(C(C)C)cc1 ZINC000147444495 CI For-Sale Anodyne ADRB1 18 40 CCO[C@H]1CCCN(C(=O)Nc2ccc(OC)cc2C(F)(F)F)C1 ZINC000147444520 EH On-Demand Anodyne RBP4 63 39 CCO[C@H]1CCCN(C(=O)Nc2ccc(OC)cc2C(F)(F)F)C1 ZINC000147444520 EH On-Demand Anodyne SFRP1 43 33 CCO[C@H]1CCCN(C(=O)Nc2ccc(OC)cc2C(F)(F)F)C1 ZINC000147444520 EH On-Demand Anodyne WNT3 43 33 CC(=O)N1CCCc2cc(S(=O)(=O)N3C[C@H](C)O[C@@H](c4ccccc4)C3)ccc21 ZINC000147444529 HG On-Demand Anodyne AKR1C3 54 34 C[C@@H](COc1c(F)cc(S(N)(=O)=O)cc1F)C(N)=O ZINC000147444559 CC For-Sale Anodyne CA2 25 41 C[C@@H](COc1c(F)cc(S(N)(=O)=O)cc1F)C(N)=O ZINC000147444559 CC For-Sale Anodyne CA4 22 40 CNc1cccc(Oc2ccc(C(N)=O)cc2)n1 ZINC000147444565 BE For-Sale Anodyne TRY1_BOVIN 25 41 CCOc1ccccc1NC(=O)CC1(CN)CCC1 ZINC000147444661 CF For-Sale Anodyne HCN1 52 36 CCOc1ccccc1NC(=O)CC1(CN)CCC1 ZINC000147444661 CF For-Sale Anodyne HCN4 45 35 COc1ccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c(C(F)(F)F)c1 ZINC000147444686 HI On-Demand Anodyne NOS2 69 38 COc1ccc(NC(=O)NCc2ccc(-n3ccnc3)c(F)c2)c(C(F)(F)F)c1 ZINC000147444686 HI On-Demand Anodyne ROCK2 15 45 CCNc1ccc(Cl)cc1C(=O)NCCNC(=O)N(C)C ZINC000147444691 DD On-Demand Anodyne F10 23 42 C[C@@]1(C(=O)Nc2ccc(C(F)(F)F)cn2)CCCN1c1ccc(C(F)(F)F)cn1 ZINC000147444707 HJ For-Sale Anodyne CNR2 17 75 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(Cl)c(C(N)=O)c3)ccc21 ZINC000147444719 FE On-Demand Anodyne IMDH_CRYPV 26 45 CC(=O)N1CCc2cc(S(=O)(=O)N3C[C@H](c4ccccc4)O[C@H](C)C3)ccc21 ZINC000147444751 HF On-Demand Anodyne HSD17B3 44 31 CC(=O)N1CCc2cc(S(=O)(=O)N3C[C@H](c4ccccc4)O[C@H](C)C3)ccc21 ZINC000147444751 HF On-Demand Anodyne AKR1C3 54 35 C[C@H](COc1c(F)cc(S(N)(=O)=O)cc1F)C(N)=O ZINC000147444764 CC For-Sale Anodyne CA2 25 41 C[C@H](COc1c(F)cc(S(N)(=O)=O)cc1F)C(N)=O ZINC000147444764 CC For-Sale Anodyne CA4 22 40 O=C(Cc1ccc(F)c(F)c1)N1CCC[C@@H]1CCCBr ZINC000147444828 EH For-Sale Reactive OPRK1 32 47 COc1ccc(NC(=O)N2C[C@H](c3ccccc3)O[C@H](C)C2)c(C(F)(F)F)c1 ZINC000147444870 GJ On-Demand Anodyne RBP4 80 42 NC1(C(=O)NCCc2ccc(F)cc2)CCC1 ZINC000147444911 BD On-Demand Anodyne CA12 15 49 NC1(C(=O)NCCc2ccc(F)cc2)CCC1 ZINC000147444911 BD On-Demand Anodyne Q76353_9HIV1 0 42 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne F2 84 52 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne PLG 24 48 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne PRSS1 25 51 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne ACE 40 37 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne FKBP1A 48 45 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne CELA1 50 42 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne CHRM4 20 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne ELANE 70 40 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne MMP13 44 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne TRY1_BOVIN 87 40 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne ADAM17 38 40 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne DPP4 15 40 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne ITGA4 31 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne PREP 88 36 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne CAPNS1 21 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne MMP2 22 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne MMP3 52 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne MMP8 25 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne LGMN 72 37 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne CAPN1 20 44 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne MMP9 29 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne EPHX2 29 43 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne TGM2 65 43 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne MMP7 56 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne MMP1 50 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne XIAP 58 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne F13A1 66 43 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne SFRP1 57 37 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne WNT3 62 41 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne BRCA1 61 34 CC(=O)N1CCC[C@H]1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147444949 GD On-Demand Anodyne TMPRSS11D 68 38 CC(=O)N1CCc2cc(S(=O)(=O)N3C[C@H](C)O[C@@H](c4ccccc4)C3)ccc21 ZINC000147444969 HF On-Demand Anodyne HSD17B3 44 31 CC(=O)N1CCc2cc(S(=O)(=O)N3C[C@H](C)O[C@@H](c4ccccc4)C3)ccc21 ZINC000147444969 HF On-Demand Anodyne AKR1C3 54 35 O=C(Cc1ccc(F)c(F)c1)N1CCC[C@H]1CCCBr ZINC000147445023 EH For-Sale Reactive OPRK1 32 47 COc1ccc(NC(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)c(C(F)(F)F)c1 ZINC000147445048 GJ On-Demand Anodyne RBP4 80 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(Cl)c1OC)C2 ZINC000147445053 EH On-Demand Anodyne MTNR1A 39 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(Cl)c1OC)C2 ZINC000147445053 EH On-Demand Anodyne ROCK2 42 49 COc1ccc(NC(=O)N2C[C@@H](C)O[C@H](c3ccccc3)C2)c(C(F)(F)F)c1 ZINC000147445183 GJ On-Demand Anodyne RBP4 80 42 O=C(c1cncs1)c1ccccc1OC(F)(F)F ZINC000147445192 CG For-Sale Anodyne KCNK3 15 40 O=C(c1cncs1)c1ccccc1OC(F)(F)F ZINC000147445192 CG For-Sale Anodyne KCNK9 22 40 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147445208 FA For-Sale Anodyne TOP1 58 39 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147445208 FA For-Sale Anodyne ADORA1 27 41 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147445208 FA For-Sale Anodyne SLC29A1 76 35 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147445208 FA For-Sale Anodyne P2RY6 63 63 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147445208 FA For-Sale Anodyne TK1 49 47 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147445208 FA For-Sale Anodyne CDA 76 46 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147445208 FA For-Sale Anodyne P2RY4 49 39 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147445208 FA For-Sale Anodyne P2RY2 51 39 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147445208 FA For-Sale Anodyne P2RY14 68 40 O=c1cc(I)n([C@@H]2O[C@H](CO)[C@@H](O)[C@@H]2O)c(=O)[nH]1 ZINC000147445208 FA For-Sale Anodyne RNASE1 15 45 COc1ccc(NC[C@@H](C)CC(=O)O)c([N+](=O)[O-])c1 ZINC000147445237 CE For-Sale Bother TAAR1 21 46 COc1ccc(NC[C@@H](C)CC(=O)O)c([N+](=O)[O-])c1 ZINC000147445237 CE For-Sale Bother AKR1C3 20 52 COc1ccc(NC[C@@H](C)CC(=O)O)c([N+](=O)[O-])c1 ZINC000147445237 CE For-Sale Bother AKR1C2 49 52 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2C2CCOCC2)no1 ZINC000147445238 DF Annotated Anodyne CNR2 15 84 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2C2CCOCC2)no1 ZINC000147445238 DF Annotated Anodyne FLT3 46 38 Cc1ccc2oc(C(=O)N3CCC[C@@H]3CCCBr)cc2c1 ZINC000147445243 FJ For-Sale Reactive FAP 0 41 O=c1nc(NCC2CCN(Cc3ccccc3)CC2)[nH]c2ccccc12 ZINC000147445282 EG On-Demand Anodyne DRD2 26 43 O=c1nc(NCC2CCN(Cc3ccccc3)CC2)[nH]c2ccccc12 ZINC000147445282 EG On-Demand Anodyne ACHE 44 53 O=c1nc(NCC2CCN(Cc3ccccc3)CC2)[nH]c2ccccc12 ZINC000147445282 EG On-Demand Anodyne DRD3 31 42 O=c1nc(NCC2CCN(Cc3ccccc3)CC2)[nH]c2ccccc12 ZINC000147445282 EG On-Demand Anodyne GRIN2B 55 39 O=c1nc(NCC2CCN(Cc3ccccc3)CC2)[nH]c2ccccc12 ZINC000147445282 EG On-Demand Anodyne SIGMAR1 61 45 O=c1nc(NCC2CCN(Cc3ccccc3)CC2)[nH]c2ccccc12 ZINC000147445282 EG On-Demand Anodyne SSTR5 46 34 O=c1nc(NCC2CCN(Cc3ccccc3)CC2)[nH]c2ccccc12 ZINC000147445282 EG On-Demand Anodyne BCHE 0 56 O=c1nc(NCC2CCN(Cc3ccccc3)CC2)[nH]c2ccccc12 ZINC000147445282 EG On-Demand Anodyne VCP 42 33 CC(C)CCO[C@@H](C)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147445285 FF On-Demand Anodyne ST14 45 33 O=C(Cn1cc([N+](=O)[O-])cn1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147445287 HD On-Demand Bother TGM2 65 42 O=C(Cn1cc([N+](=O)[O-])cn1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147445287 HD On-Demand Bother F13A1 64 42 O=C(Cn1cc([N+](=O)[O-])cn1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147445287 HD On-Demand Bother NAMPT 41 36 COc1ccc(NC(=O)N2C[C@H](C)O[C@H](c3ccccc3)C2)c(C(F)(F)F)c1 ZINC000147445314 GJ On-Demand Anodyne RBP4 80 42 COc1ccc(NC[C@H](C)CC(=O)O)c([N+](=O)[O-])c1 ZINC000147445375 CE For-Sale Bother TAAR1 21 46 COc1ccc(NC[C@H](C)CC(=O)O)c([N+](=O)[O-])c1 ZINC000147445375 CE For-Sale Bother AKR1C3 20 52 COc1ccc(NC[C@H](C)CC(=O)O)c([N+](=O)[O-])c1 ZINC000147445375 CE For-Sale Bother AKR1C2 49 52 Cc1ccc2oc(C(=O)N3CCC[C@H]3CCCBr)cc2c1 ZINC000147445387 FJ For-Sale Reactive FAP 0 41 Cc1ccc(NC(=O)C[C@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445403 GD On-Demand Anodyne CA2 60 39 Cc1ccc(NC(=O)C[C@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445403 GD On-Demand Anodyne CA1 49 39 Cc1ccc(NC(=O)C[C@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445403 GD On-Demand Anodyne CA4 65 39 Cc1ccc(NC(=O)C[C@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445403 GD On-Demand Anodyne CA5A 45 38 Cc1ccc(NC(=O)C[C@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445403 GD On-Demand Anodyne SLC1A1 53 36 Cc1ccc(NC(=O)C[C@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445403 GD On-Demand Anodyne SLC1A3 56 35 Cc1ccc(NC(=O)C[C@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445403 GD On-Demand Anodyne SLC1A2 79 38 CCc1cccc(CC)c1NC(=O)C1(N)CCC1 ZINC000147445419 BF For-Sale Anodyne ACAT 0 49 CC(C)CCO[C@H](C)C(=O)Nc1cccc(S(=O)(=O)NC2CC2)c1 ZINC000147445443 FF On-Demand Anodyne ST14 45 33 CCc1ccc(OC[C@H](O)CNCCCCC(C)C)cc1 ZINC000147445531 CG For-Sale Anodyne ADRB2 75 57 CCc1ccc(OC[C@H](O)CNCCCCC(C)C)cc1 ZINC000147445531 CG For-Sale Anodyne ADRB1 93 61 CCc1ccc(OC[C@H](O)CNCCCCC(C)C)cc1 ZINC000147445531 CG For-Sale Anodyne GRIN1 30 47 CCc1ccc(OC[C@H](O)CNCCCCC(C)C)cc1 ZINC000147445531 CG For-Sale Anodyne ADRB3 69 55 Cc1nn(C(F)F)c(C)c1CC(=O)NCc1ccccc1Cn1cncn1 ZINC000147445550 FE On-Demand Anodyne P2RX7 60 50 Cc1nn(C(F)F)c(C)c1CC(=O)NCc1ccccc1Cn1cncn1 ZINC000147445550 FE On-Demand Anodyne HIS3 60 37 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc3ccccc23)c1 ZINC000147445552 FH On-Demand Bother CASR 21 42 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc3ccccc23)c1 ZINC000147445552 FH On-Demand Bother NQO2 22 42 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc3ccccc23)c1 ZINC000147445552 FH On-Demand Bother MTNR1A 58 38 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc3ccccc23)c1 ZINC000147445552 FH On-Demand Bother MTNR1B 50 35 COc1ccc([N+](=O)[O-])c(C(=O)NCCOc2cccc3ccccc23)c1 ZINC000147445552 FH On-Demand Bother AKR1C2 33 43 Cc1ccc(NC(=O)C[C@@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445612 GD On-Demand Anodyne CA2 60 39 Cc1ccc(NC(=O)C[C@@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445612 GD On-Demand Anodyne CA1 49 39 Cc1ccc(NC(=O)C[C@@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445612 GD On-Demand Anodyne CA4 65 39 Cc1ccc(NC(=O)C[C@@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445612 GD On-Demand Anodyne CA5A 45 38 Cc1ccc(NC(=O)C[C@@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445612 GD On-Demand Anodyne SLC1A1 53 36 Cc1ccc(NC(=O)C[C@@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445612 GD On-Demand Anodyne SLC1A3 56 35 Cc1ccc(NC(=O)C[C@@H](NC(N)=O)c2ccccc2)cc1S(N)(=O)=O ZINC000147445612 GD On-Demand Anodyne SLC1A2 79 38 NS(=O)(=O)c1cc(F)c(OCc2ncccn2)c(F)c1 ZINC000147445650 DC For-Sale Anodyne CA2 22 41 NS(=O)(=O)c1cc(F)c(OCc2ncccn2)c(F)c1 ZINC000147445650 DC For-Sale Anodyne CA4 20 41 NS(=O)(=O)c1cc(F)c(OCc2ncccn2)c(F)c1 ZINC000147445650 DC For-Sale Anodyne CA9 15 41 CCc1cccc(CC)c1NC(=O)CC1(CN)CCC1 ZINC000147445653 CG For-Sale Anodyne ACAT 0 45 CCc1ccc(OC[C@@H](O)CNCCCCC(C)C)cc1 ZINC000147445684 CG For-Sale Anodyne ADRB2 75 57 CCc1ccc(OC[C@@H](O)CNCCCCC(C)C)cc1 ZINC000147445684 CG For-Sale Anodyne ADRB1 93 61 CCc1ccc(OC[C@@H](O)CNCCCCC(C)C)cc1 ZINC000147445684 CG For-Sale Anodyne GRIN1 30 47 CCc1ccc(OC[C@@H](O)CNCCCCC(C)C)cc1 ZINC000147445684 CG For-Sale Anodyne ADRB3 69 55 O=C(NCCNC(=O)[C@H]1C[C@H]1c1cccc(Cl)c1)c1ccc(F)cc1 ZINC000147445698 FG On-Demand Anodyne PLD2 42 41 Cc1ccc2[nH]c(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147445757 HG On-Demand Anodyne HTR4 44 39 Cc1ccc2[nH]c(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147445757 HG On-Demand Anodyne GRIN2B 48 41 Cc1ccc2[nH]c(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147445757 HG On-Demand Anodyne PYGL 90 44 Cc1ccc2[nH]c(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147445757 HG On-Demand Anodyne PYGM 30 44 Cc1ccc2[nH]c(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147445757 HG On-Demand Anodyne EPHX2 28 43 Cc1ccc2[nH]c(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147445757 HG On-Demand Anodyne TGM2 48 40 Cc1ccc2[nH]c(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147445757 HG On-Demand Anodyne CACNA1I 53 38 Cc1ccc2[nH]c(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147445757 HG On-Demand Anodyne F13A1 35 40 Cc1ccc2[nH]c(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147445757 HG On-Demand Anodyne AKR1C3 37 50 Cc1ccc2[nH]c(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc2c1 ZINC000147445757 HG On-Demand Anodyne NAMPT 33 42 NC(=O)c1ccc(Oc2nc(N)ccc2[N+](=O)[O-])cc1 ZINC000147445766 CD For-Sale Bother GSTM2 31 40 NC(=O)c1ccc(Oc2nc(N)ccc2[N+](=O)[O-])cc1 ZINC000147445766 CD For-Sale Bother CHEK2 21 41 NS(=O)(=O)c1cc(F)c(OCCC(=O)NC2CC2)c(F)c1 ZINC000147445827 DC For-Sale Anodyne CA2 18 44 NS(=O)(=O)c1cc(F)c(OCCC(=O)NC2CC2)c(F)c1 ZINC000147445827 DC For-Sale Anodyne CA1 15 44 NS(=O)(=O)c1cc(F)c(OCCC(=O)NC2CC2)c(F)c1 ZINC000147445827 DC For-Sale Anodyne CA7 25 44 CC(C)CCCCNC(=O)c1ccc2c(c1)CCN2 ZINC000147445871 CG For-Sale Anodyne HDAC9 15 47 NC1(C(=O)Nc2ccccc2Oc2ccccc2)CCC1 ZINC000147445899 CG For-Sale Anodyne PYGM 18 43 O=C(NCCNC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc(F)cc1 ZINC000147445913 FG On-Demand Anodyne PLD2 42 41 Clc1nc(-c2cccnc2)sc1Br ZINC000147445967 CH For-Sale Anodyne CYP11B2 25 41 Clc1nc(-c2cccnc2)sc1Br ZINC000147445967 CH For-Sale Anodyne CYP2E1 47 37 Clc1nc(-c2cccnc2)sc1Br ZINC000147445967 CH For-Sale Anodyne CYP2A6 48 38 Cc1ccccc1N(CC(C)C)S(=O)(=O)c1ccc(Br)cc1 ZINC000147445977 GJ For-Sale Anodyne MMP13 15 43 Cc1ccccc1N(CC(C)C)S(=O)(=O)c1ccc(Br)cc1 ZINC000147445977 GJ For-Sale Anodyne RORC 27 44 CNc1cc(Oc2ccc(C(N)=O)cc2)ncn1 ZINC000147445982 BD For-Sale Anodyne CDKL2 41 43 O=c1ccc2ccc(-c3ccccc3)oc-2c1 ZINC000147445998 BG Annotated Anodyne CYP1B1 40 42 O=c1ccc2ccc(-c3ccccc3)oc-2c1 ZINC000147445998 BG Annotated Anodyne CYP1A1 35 42 O=c1ccc2ccc(-c3ccccc3)oc-2c1 ZINC000147445998 BG Annotated Anodyne CYP1A2 27 42 O=c1ccc2ccc(-c3ccccc3)oc-2c1 ZINC000147445998 BG Annotated Anodyne TNKS 44 47 O=c1ccc2ccc(-c3ccccc3)oc-2c1 ZINC000147445998 BG Annotated Anodyne TNKS2 15 47 Cc1ccccc1N(CC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1)S(=O)(=O)c1ccccc1 ZINC000147446022 KG In-Stock Anodyne EDNRA 15 40 Cc1ccccc1N(CC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1)S(=O)(=O)c1ccccc1 ZINC000147446022 KG In-Stock Anodyne BMP1 66 49 Cc1ccccc1N(CC(=O)N1CCN(Cc2ccc3c(c2)OCO3)CC1)S(=O)(=O)c1ccccc1 ZINC000147446022 KG In-Stock Anodyne MCHR1 22 44 O=C(NCCNC(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1)c1ccc(F)cc1 ZINC000147446057 FG On-Demand Anodyne PLD2 42 41 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2CC2CCOCC2)no1 ZINC000147446065 EF Annotated Anodyne CNR2 25 94 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2CC2CCOCC2)no1 ZINC000147446065 EF Annotated Anodyne FLT3 45 38 O=C(C[C@@H]1NC(=O)NC1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147446111 GB On-Demand Anodyne EPHX2 18 42 O=C(C[C@@H]1NC(=O)NC1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147446111 GB On-Demand Anodyne TGM2 61 43 O=C(C[C@@H]1NC(=O)NC1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147446111 GB On-Demand Anodyne F13A1 62 43 C[C@H](CNc1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147446116 BE On-Demand Bother PGR 17 40 C[C@H](CNc1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147446116 BE On-Demand Bother AR 0 45 C[C@H](CNc1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147446116 BE On-Demand Bother AKR1C2 15 40 CCCCNC(=O)CNCCCCC(C)C ZINC000147446137 BE For-Sale Anodyne ASAH1 64 35 CCCCNC(=O)CNCCCCC(C)C ZINC000147446137 BE For-Sale Anodyne NOD1 62 45 O=C(NCc1ccn2ccnc2c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000147446161 FI On-Demand Anodyne LTA4H 38 40 O=C(NCc1ccn2ccnc2c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000147446161 FI On-Demand Anodyne CA1 34 40 O=C(NCc1ccn2ccnc2c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000147446161 FI On-Demand Anodyne RAF1 35 41 O=C(NCc1ccn2ccnc2c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000147446161 FI On-Demand Anodyne KDR 18 46 O=C(NCc1ccn2ccnc2c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000147446161 FI On-Demand Anodyne ROCK2 24 45 O=C(NCc1ccn2ccnc2c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000147446161 FI On-Demand Anodyne FAAH 17 45 O=C(NCc1ccn2ccnc2c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000147446161 FI On-Demand Anodyne PDGFRA 48 38 O=C(NCc1ccn2ccnc2c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000147446161 FI On-Demand Anodyne NCE103 18 45 O=C(NCc1ccn2ccnc2c1)Nc1ccc(Oc2ccccc2)cc1 ZINC000147446161 FI On-Demand Anodyne NAMPT 53 59 CN1C(=O)OC(C)(C)[C@H]1c1ccccc1 ZINC000147446162 BF For-Sale Anodyne TNKS 57 42 O=C(c1ccc(Br)c(Cl)c1)N1CCN(C2CCCC2)CC1 ZINC000147446190 FH On-Demand Anodyne HRH3 29 43 O=C(c1ccc(Br)c(Cl)c1)N1CCN(C2CCCC2)CC1 ZINC000147446190 FH On-Demand Anodyne CCR3 24 42 O=C(c1ccc(Br)c(Cl)c1)N1CCN(C2CCCC2)CC1 ZINC000147446190 FH On-Demand Anodyne L3MBTL1 0 60 O=C(c1ccc(Br)c(Cl)c1)N1CCN(C2CCCC2)CC1 ZINC000147446190 FH On-Demand Anodyne L3MBTL3 95 53 O=C(c1ccc(Br)c(Cl)c1)N1CCN(C2CCCC2)CC1 ZINC000147446190 FH On-Demand Anodyne L3MBTL4 0 45 O=C(c1ccc(Br)c(Cl)c1)N1CCN(C2CCCC2)CC1 ZINC000147446190 FH On-Demand Anodyne MBTD1 0 56 O=C(c1ccc(Br)c(Cl)c1)N1CCN(C2CCCC2)CC1 ZINC000147446190 FH On-Demand Anodyne TP53BP1 0 53 O=C(NCCNC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)c1ccc(F)cc1 ZINC000147446199 FG On-Demand Anodyne PLD2 42 41 O=C(O)c1ccc(N2CCC3(CCCC3)C2)cc1 ZINC000147446219 BG For-Sale Anodyne RARA 42 33 O=C(O)c1ccc(N2CCC3(CCCC3)C2)cc1 ZINC000147446219 BG For-Sale Anodyne RARG 40 35 O=C(O)c1ccc(N2CCC3(CCCC3)C2)cc1 ZINC000147446219 BG For-Sale Anodyne RXRG 49 32 O=C(O)c1ccc(N2CCC3(CCCC3)C2)cc1 ZINC000147446219 BG For-Sale Anodyne RXRB 52 33 O=C(NCC1(C(=O)O)CCC1)c1cc(Cl)cc(Cl)c1 ZINC000147446253 DF On-Demand Anodyne CACNA1I 49 38 C[C@@H](CNc1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147446279 BE On-Demand Bother PGR 17 40 C[C@@H](CNc1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147446279 BE On-Demand Bother AR 0 45 C[C@@H](CNc1ccc([N+](=O)[O-])cc1)CC(=O)O ZINC000147446279 BE On-Demand Bother AKR1C2 15 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc2cn[nH]c12 ZINC000147446349 GE On-Demand Anodyne HTR4 45 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc2cn[nH]c12 ZINC000147446349 GE On-Demand Anodyne CHRM5 21 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc2cn[nH]c12 ZINC000147446349 GE On-Demand Anodyne GRIN2B 21 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc2cn[nH]c12 ZINC000147446349 GE On-Demand Anodyne TGM2 54 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc2cn[nH]c12 ZINC000147446349 GE On-Demand Anodyne F13A1 41 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc2cn[nH]c12 ZINC000147446349 GE On-Demand Anodyne NAMPT 47 49 CC[C@H](NC(=O)N1CCC[C@H]2CCC[C@H]21)C(=O)O ZINC000147446354 CD For-Sale Anodyne SLC5A1 18 40 CC(C)CNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147446433 DC For-Sale Anodyne CA2 46 44 Cc1ccc(Br)c(C(=O)N2CCN(C3CCCC3)CC2)c1 ZINC000147446456 FG On-Demand Anodyne L3MBTL1 0 50 Cc1ccc(Br)c(C(=O)N2CCN(C3CCCC3)CC2)c1 ZINC000147446456 FG On-Demand Anodyne L3MBTL3 82 50 Cc1ccc(Br)c(C(=O)N2CCN(C3CCCC3)CC2)c1 ZINC000147446456 FG On-Demand Anodyne MBTD1 0 50 Cc1ccc(Br)c(C(=O)N2CCN(C3CCCC3)CC2)c1 ZINC000147446456 FG On-Demand Anodyne TP53BP1 0 46 Fc1cc(OCc2cc(CNC3CC3)co2)ccc1Cl ZINC000147446463 CH For-Sale Anodyne DAO 15 41 CC(C)CCCCNC[C@H](O)c1cccc(C(F)(F)F)c1 ZINC000147446477 DI For-Sale Anodyne ADRB3 45 38 CC(C)CCCCNC[C@H](O)c1cccc(C(F)(F)F)c1 ZINC000147446477 DI For-Sale Anodyne PHES 0 58 CC[C@H](NC(=O)N1CCC[C@@H]2CCC[C@H]21)C(=O)O ZINC000147446480 CD For-Sale Anodyne SLC5A1 18 40 O=C(/C=C/c1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147446558 GE On-Demand Anodyne GRIN2B 20 42 O=C(/C=C/c1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147446558 GE On-Demand Anodyne CHRNA7 30 46 O=C(/C=C/c1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147446558 GE On-Demand Anodyne C3AR1 18 42 O=C(/C=C/c1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147446558 GE On-Demand Anodyne TGM2 93 47 O=C(/C=C/c1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147446558 GE On-Demand Anodyne F13A1 101 47 O=C(/C=C/c1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147446558 GE On-Demand Anodyne NAMPT 76 55 CC(C)CCCCNC[C@@H](O)c1cccc(C(F)(F)F)c1 ZINC000147446619 DI For-Sale Anodyne ADRB3 45 38 CC(C)CCCCNC[C@@H](O)c1cccc(C(F)(F)F)c1 ZINC000147446619 DI For-Sale Anodyne PHES 0 58 CCCNc1ncc(F)c(Oc2ccc(C(N)=O)cc2)n1 ZINC000147446668 CE For-Sale Anodyne SYK 20 40 CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000147446711 JJ Annotated Anodyne PTGS2 56 43 CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000147446711 JJ Annotated Anodyne MMP13 21 56 CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000147446711 JJ Annotated Anodyne MMP2 27 56 CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000147446711 JJ Annotated Anodyne MMP3 24 56 CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000147446711 JJ Annotated Anodyne MMP8 34 56 CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000147446711 JJ Annotated Anodyne MMP9 26 56 CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000147446711 JJ Annotated Anodyne MMP12 19 42 CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000147446711 JJ Annotated Anodyne ADAMTS4 33 46 CC(C)CN(Cc1ccccc1)S(=O)(=O)c1ccc(-c2ccc(S(C)(=O)=O)cc2)cc1 ZINC000147446711 JJ Annotated Anodyne MMP1 19 44 CCNCCCCCOc1ccc(Cl)c(F)c1 ZINC000147446762 CH For-Sale Anodyne DRD4 20 45 NC1(C(=O)Nc2ccccc2C(F)(F)F)CCC1 ZINC000147446814 CF For-Sale Anodyne RBP4 59 38 CC(C)(C)OC(=O)NNCCN ZINC000147446850 AB For-Sale Reactive CTSK 0 43 CCNC(=O)CCOc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147446875 DC For-Sale Anodyne CA2 43 46 CCNC(=O)CCOc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147446875 DC For-Sale Anodyne CA1 32 40 CCNC(=O)CCOc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147446875 DC For-Sale Anodyne CA4 39 40 CSCSC[C@@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000147446979 CE For-Sale Anodyne PAPA1_CARPA 52 49 CSCSC[C@@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000147446979 CE For-Sale Anodyne CTSK 18 49 CSCSC[C@@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000147446979 CE For-Sale Anodyne POLG_HCV1 23 40 CSCSC[C@@H](NC(=O)OC(C)(C)C)C(=O)O ZINC000147446979 CE For-Sale Anodyne FPR1 53 46 NCC1(CC(=O)Nc2ccccc2C(F)(F)F)CCC1 ZINC000147446995 CG For-Sale Anodyne KCNJ11 44 35 CC(C)(O)C(=O)Nc1ccc(C#N)c(Cl)c1 ZINC000147447004 BD For-Sale Mild BLM 0 49 CNS(=O)(=O)c1ccc(NC[C@@H](C)CC(=O)O)cc1 ZINC000147447007 CD For-Sale Anodyne CA2 21 42 Cc1noc2ncc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc12 ZINC000147447031 HE On-Demand Anodyne HTR4 53 37 Cc1noc2ncc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc12 ZINC000147447031 HE On-Demand Anodyne EPHX2 25 42 Cc1noc2ncc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc12 ZINC000147447031 HE On-Demand Anodyne TGM2 48 39 Cc1noc2ncc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc12 ZINC000147447031 HE On-Demand Anodyne CACNA1I 62 38 Cc1noc2ncc(C(=O)NCC3CCN(S(=O)(=O)c4ccccc4)CC3)cc12 ZINC000147447031 HE On-Demand Anodyne NAMPT 50 47 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean TH 0 45 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean OPRM1 67 62 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean OPRD1 83 62 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean NTSR1 43 34 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean NTSR2 41 31 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean SLC15A1 0 41 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean PDYN 0 41 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean GRIA1 99 39 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean YARS 63 35 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean DNPEP 0 43 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean ALOX15 35 59 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean LEF 96 37 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean SLC15A2 0 45 CC(C)CCCCNC(=O)[C@@H](N)Cc1ccc(O)c(O)c1 ZINC000147447066 CD For-Sale Clean VM1B1_BOTAS 0 40 CNS(=O)(=O)c1ccc(NC[C@H](C)CC(=O)O)cc1 ZINC000147447118 CD For-Sale Anodyne CA2 21 42 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne HTR1A 81 52 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne DRD2 60 48 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne DRD4 47 38 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne ADRA1D 24 41 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne HTR2A 54 49 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne HTR2C 34 42 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne SLC6A4 15 41 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne ADRA1A 31 50 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne ADRA1B 19 50 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne DRD3 81 46 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne HTR4 19 41 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne P2RY12 89 38 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne HTR7 89 45 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne KLK3 61 36 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne CTSK 43 43 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne NPFFR2 51 34 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne C3AR1 51 32 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne MMP3 18 42 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne GRIA1 43 31 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne REN 17 40 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne PCSK5 54 36 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne FURIN 78 36 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne POLG_WNV 73 33 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne NPFFR1 74 34 CCCC[C@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447127 FD On-Demand Anodyne NOD1 41 31 CCCCNC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147447148 DC For-Sale Anodyne CA2 47 42 CCCNc1cc(Oc2ccc(C(N)=O)cc2)nc(C)n1 ZINC000147447150 CE For-Sale Anodyne TRY1_BOVIN 19 40 NC1(C(=O)Nc2cccc(C(F)(F)F)c2)CCC1 ZINC000147447213 CF On-Demand Anodyne TRPM4 0 43 COC(=O)Cc1csc(-c2ccc(OC)c(F)c2)n1 ZINC000147447256 CF For-Sale Anodyne DCK 46 42 COC(=O)Cc1csc(-c2ccc(OC)c(F)c2)n1 ZINC000147447256 CF For-Sale Anodyne PPARD 17 40 O=C(NCCNC(=O)c1ccc2c(c1)COC2)c1ccc(F)cc1 ZINC000147447260 EE On-Demand Anodyne PLD2 40 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(F)cccc2[nH]1 ZINC000147447270 HG On-Demand Anodyne HTR4 50 39 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(F)cccc2[nH]1 ZINC000147447270 HG On-Demand Anodyne GRIN2B 39 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(F)cccc2[nH]1 ZINC000147447270 HG On-Demand Anodyne PLD1 49 36 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(F)cccc2[nH]1 ZINC000147447270 HG On-Demand Anodyne TGM2 49 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(F)cccc2[nH]1 ZINC000147447270 HG On-Demand Anodyne CACNA1I 45 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(F)cccc2[nH]1 ZINC000147447270 HG On-Demand Anodyne F13A1 33 40 Cc1c(C(=O)N2CCC[C@@H]2CCCBr)cccc1[N+](=O)[O-] ZINC000147447271 FH For-Sale Reactive HCRTR1 15 41 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(OC(F)(F)F)c2)C1 ZINC000147447285 HG On-Demand Anodyne EPHX2 36 49 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(OC(F)(F)F)c2)C1 ZINC000147447285 HG On-Demand Anodyne TAAR1 31 46 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne HTR1A 81 52 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne DRD2 60 48 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne DRD4 47 38 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne ADRA1D 24 41 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne HTR2A 54 49 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne HTR2C 34 42 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne SLC6A4 15 41 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne ADRA1A 31 50 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne ADRA1B 19 50 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne DRD3 81 46 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne HTR4 19 41 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne P2RY12 89 38 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne HTR7 89 45 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne KLK3 61 36 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne CTSK 43 43 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne NPFFR2 51 34 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne C3AR1 51 32 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne MMP3 18 42 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne GRIA1 43 31 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne REN 17 40 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne PCSK5 54 36 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne FURIN 78 36 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne POLG_WNV 73 33 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne NPFFR1 74 34 CCCC[C@@H](NC(N)=O)C(=O)NCCN1CCN(c2ccccc2)CC1 ZINC000147447319 FD On-Demand Anodyne NOD1 41 31 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2CC2CC2)no1 ZINC000147447343 CF Annotated Anodyne CNR2 15 93 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2CC2CC2)no1 ZINC000147447343 CF Annotated Anodyne HSD11B1 37 40 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2CC2CC2)no1 ZINC000147447343 CF Annotated Anodyne FLT3 48 41 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2CC2CC2)no1 ZINC000147447343 CF Annotated Anodyne CSF1R 16 41 CCNc1cc(Oc2ccc(C(N)=O)cc2)nc(C)n1 ZINC000147447350 CE For-Sale Anodyne CHEK2 43 39 CCCCC1CCC(NS(=O)(=O)c2ccc3[nH]c(=O)c(=O)[nH]c3c2)CC1 ZINC000147447372 GE On-Demand Anodyne BRD4 17 40 CCCNc1ccc(C(=O)NCCNC(=O)N(C)C)cc1 ZINC000147447374 CD For-Sale Anodyne KCNQ1 0 41 CCCNc1ccc(C(=O)NCCNC(=O)N(C)C)cc1 ZINC000147447374 CD For-Sale Anodyne CNGA1 0 42 Cc1c(C(=O)N2CCC[C@H]2CCCBr)cccc1[N+](=O)[O-] ZINC000147447409 FH For-Sale Reactive HCRTR1 15 41 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(OC(F)(F)F)c2)C1 ZINC000147447439 HG On-Demand Anodyne EPHX2 36 49 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2cccc(OC(F)(F)F)c2)C1 ZINC000147447439 HG On-Demand Anodyne TAAR1 31 46 NCC1(CC(=O)Nc2cccc(C(F)(F)F)c2)CCC1 ZINC000147447443 CG For-Sale Anodyne SLC1A1 25 42 NCC1(CC(=O)Nc2cccc(C(F)(F)F)c2)CCC1 ZINC000147447443 CG For-Sale Anodyne SLC1A3 23 42 NCC1(CC(=O)Nc2cccc(C(F)(F)F)c2)CCC1 ZINC000147447443 CG For-Sale Anodyne EPHX2 15 48 NCC1(CC(=O)Nc2cccc(C(F)(F)F)c2)CCC1 ZINC000147447443 CG For-Sale Anodyne SLC1A2 36 42 NCC1(CC(=O)Nc2cccc(C(F)(F)F)c2)CCC1 ZINC000147447443 CG For-Sale Anodyne RIPK1 29 40 NCC1(CC(=O)Nc2cccc(C(F)(F)F)c2)CCC1 ZINC000147447443 CG For-Sale Anodyne TRPM4 0 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1CC(=O)N(C2CC2)C1 ZINC000147447576 HD On-Demand Anodyne INHA 22 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1CC(=O)N(C2CC2)C1 ZINC000147447576 HD On-Demand Anodyne EPHX2 26 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1CC(=O)N(C2CC2)C1 ZINC000147447576 HD On-Demand Anodyne TGM2 55 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1CC(=O)N(C2CC2)C1 ZINC000147447576 HD On-Demand Anodyne F13A1 46 42 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447603 CD For-Sale Anodyne OPRM1 98 56 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447603 CD For-Sale Anodyne OPRD1 87 45 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447603 CD For-Sale Anodyne NTSR1 45 33 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447603 CD For-Sale Anodyne HLA-A 49 35 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447603 CD For-Sale Anodyne GRIA1 51 38 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447603 CD For-Sale Anodyne YARS 111 51 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447603 CD For-Sale Anodyne MARS 41 31 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447603 CD For-Sale Anodyne SLC15A2 0 50 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc([N+](=O)[O-])cc3)ccc21 ZINC000147447608 EE On-Demand Bother EPHX2 16 45 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc([N+](=O)[O-])cc3)ccc21 ZINC000147447608 EE On-Demand Bother F2RL3 47 34 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc([N+](=O)[O-])cc3)ccc21 ZINC000147447608 EE On-Demand Bother MTCA1 23 44 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc([N+](=O)[O-])cc3)ccc21 ZINC000147447608 EE On-Demand Bother P96878_MYCTU 30 44 COc1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1OC ZINC000147447621 FG For-Sale Reactive HCRTR1 0 48 COc1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1OC ZINC000147447621 FG For-Sale Reactive FAP 0 43 COc1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1OC ZINC000147447621 FG For-Sale Reactive ACKR3 76 42 CCc1nc2cc(N)ccc2n1CCNC(=O)N(C)C ZINC000147447623 CD For-Sale Anodyne HDAC1 20 40 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2C2CCC2)no1 ZINC000147447654 CF Annotated Anodyne CNR2 15 93 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2C2CCC2)no1 ZINC000147447654 CF Annotated Anodyne FLT3 48 41 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2C2CCC2)no1 ZINC000147447654 CF Annotated Anodyne CSF1R 17 41 NC1(C(=O)Nc2nc3ccc(Cl)cc3s2)CCC1 ZINC000147447656 CF For-Sale Anodyne LCK 28 45 NC1(C(=O)Nc2nc3ccc(Cl)cc3s2)CCC1 ZINC000147447656 CF For-Sale Anodyne CSNK1D 49 49 NC1(C(=O)Nc2nc3ccc(Cl)cc3s2)CCC1 ZINC000147447656 CF For-Sale Anodyne PIK3CA 19 40 NC1(C(=O)Nc2nc3ccc(Cl)cc3s2)CCC1 ZINC000147447656 CF For-Sale Anodyne PORCN 0 41 C[C@H](CNc1ccccc1C(N)=O)CC(=O)O ZINC000147447657 BD For-Sale Anodyne PAGA 0 43 CN[C@@H]1CCN(OCc2ccccc2)C1=O ZINC000147447775 BC For-Sale Anodyne FKBP1A 18 40 CN[C@@H]1CCN(OCc2ccccc2)C1=O ZINC000147447775 BC For-Sale Anodyne GRIN2A 15 42 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447809 CD For-Sale Anodyne OPRM1 98 56 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447809 CD For-Sale Anodyne OPRD1 87 45 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447809 CD For-Sale Anodyne NTSR1 45 33 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447809 CD For-Sale Anodyne HLA-A 49 35 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447809 CD For-Sale Anodyne GRIA1 51 38 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447809 CD For-Sale Anodyne YARS 111 51 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447809 CD For-Sale Anodyne MARS 41 31 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447809 CD For-Sale Anodyne SLC15A2 0 50 COc1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1OC ZINC000147447811 FG For-Sale Reactive HCRTR1 0 48 COc1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1OC ZINC000147447811 FG For-Sale Reactive FAP 0 43 COc1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1OC ZINC000147447811 FG For-Sale Reactive ACKR3 76 42 CCCCC1CCC(NS(=O)(=O)c2ccc(C(N)=O)cc2)CC1 ZINC000147447812 EF On-Demand Anodyne SFRP1 47 31 C[C@@H](CNc1ccccc1C(N)=O)CC(=O)O ZINC000147447832 BD For-Sale Anodyne PAGA 0 43 N#CCCN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147447847 DF For-Sale Mild MCHR1 26 40 O=c1cc(OCc2ccccc2)ccn1-c1ccc(N2CC3(CCNCC3)C2)nc1 ZINC000147447882 HG For-Sale Anodyne KCNH2 21 47 O=c1cc(OCc2ccccc2)ccn1-c1ccc(N2CC3(CCNCC3)C2)nc1 ZINC000147447882 HG For-Sale Anodyne MCHR1 19 63 O=c1cc(OCc2ccccc2)ccn1-c1ccc(N2CC3(CCNCC3)C2)nc1 ZINC000147447882 HG For-Sale Anodyne DPP8 17 55 O=c1cc(OCc2ccccc2)ccn1-c1ccc(N2CC3(CCNCC3)C2)nc1 ZINC000147447882 HG For-Sale Anodyne DPP9 15 55 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2C2CCCC2)no1 ZINC000147447884 DG Annotated Anodyne CNR2 15 98 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2C2CCCC2)no1 ZINC000147447884 DG Annotated Anodyne FLT3 47 39 NS(=O)(=O)c1cc(F)c(OCCc2ccncc2)c(F)c1 ZINC000147447899 DD For-Sale Anodyne CA2 31 42 NS(=O)(=O)c1cc(F)c(OCCc2ccncc2)c(F)c1 ZINC000147447899 DD For-Sale Anodyne CA1 30 43 NS(=O)(=O)c1cc(F)c(OCCc2ccncc2)c(F)c1 ZINC000147447899 DD For-Sale Anodyne CA7 25 43 NS(=O)(=O)c1cc(F)c(OCCc2ccncc2)c(F)c1 ZINC000147447899 DD For-Sale Anodyne CA5B 17 41 NS(=O)(=O)c1cc(F)c(OCCc2ccncc2)c(F)c1 ZINC000147447899 DD For-Sale Anodyne CA4 24 41 NS(=O)(=O)c1cc(F)c(OCCc2ccncc2)c(F)c1 ZINC000147447899 DD For-Sale Anodyne CA5A 20 41 NS(=O)(=O)c1cc(F)c(OCCc2ccncc2)c(F)c1 ZINC000147447899 DD For-Sale Anodyne CA12 17 43 NS(=O)(=O)c1cc(F)c(OCCc2ccncc2)c(F)c1 ZINC000147447899 DD For-Sale Anodyne CA9 22 43 NCC1(CC(=O)Nc2nc3ccc(Cl)cc3s2)CCC1 ZINC000147447912 DG For-Sale Anodyne LCK 27 41 NCC1(CC(=O)Nc2nc3ccc(Cl)cc3s2)CCC1 ZINC000147447912 DG For-Sale Anodyne CSNK1D 51 51 NCC1(CC(=O)Nc2nc3ccc(Cl)cc3s2)CCC1 ZINC000147447912 DG For-Sale Anodyne PIK3CA 0 40 NCC1(CC(=O)Nc2nc3ccc(Cl)cc3s2)CCC1 ZINC000147447912 DG For-Sale Anodyne HSD17B1 0 42 NCC1(CC(=O)Nc2nc3ccc(Cl)cc3s2)CCC1 ZINC000147447912 DG For-Sale Anodyne PORCN 0 46 CN[C@H]1CCN(OCc2ccccc2)C1=O ZINC000147447933 BC For-Sale Anodyne FKBP1A 18 40 CN[C@H]1CCN(OCc2ccccc2)C1=O ZINC000147447933 BC For-Sale Anodyne GRIN2A 15 42 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447943 CD For-Sale Anodyne OPRM1 98 56 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447943 CD For-Sale Anodyne OPRD1 87 45 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447943 CD For-Sale Anodyne NTSR1 45 33 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447943 CD For-Sale Anodyne HLA-A 49 35 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447943 CD For-Sale Anodyne GRIA1 51 38 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447943 CD For-Sale Anodyne YARS 111 51 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447943 CD For-Sale Anodyne MARS 41 31 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccc(O)cc1 ZINC000147447943 CD For-Sale Anodyne SLC15A2 0 50 CCCc1nc2cc(N)ccc2n1CCNC(=O)N(C)C ZINC000147447945 CD For-Sale Anodyne HDAC10 26 46 CCCc1nc2cc(N)ccc2n1CCNC(=O)N(C)C ZINC000147447945 CD For-Sale Anodyne HDAC1 17 48 CCCc1nc2cc(N)ccc2n1CCNC(=O)N(C)C ZINC000147447945 CD For-Sale Anodyne HDAC4 28 46 CCCc1nc2cc(N)ccc2n1CCNC(=O)N(C)C ZINC000147447945 CD For-Sale Anodyne HDAC5 37 46 CCCc1nc2cc(N)ccc2n1CCNC(=O)N(C)C ZINC000147447945 CD For-Sale Anodyne HDAC9 31 46 CCCc1nc2cc(N)ccc2n1CCNC(=O)N(C)C ZINC000147447945 CD For-Sale Anodyne HDAC11 28 46 CCCc1nc2cc(N)ccc2n1CCNC(=O)N(C)C ZINC000147447945 CD For-Sale Anodyne HDAC7 38 46 COc1cc(C(=O)N[C@@H](C)c2cccc(Br)c2)ccc1F ZINC000147447963 FI On-Demand Anodyne TAAR1 16 42 CCCCC1CCC(NS(=O)(=O)c2cc(NC(C)=O)ccc2OC)CC1 ZINC000147447995 GH On-Demand Anodyne ADRA1D 22 42 CCCCC1CCC(NS(=O)(=O)c2cc(NC(C)=O)ccc2OC)CC1 ZINC000147447995 GH On-Demand Anodyne ADRA1A 15 42 CCCCC1CCC(NS(=O)(=O)c2cc(NC(C)=O)ccc2OC)CC1 ZINC000147447995 GH On-Demand Anodyne ADRA1B 27 42 CCCCC1CCC(NS(=O)(=O)c2cc(NC(C)=O)ccc2OC)CC1 ZINC000147447995 GH On-Demand Anodyne CCR8 72 36 CCc1c[nH]c2c(N3CCCC3=O)cc(C(=O)N[C@@H](Cc3ccccc3)[C@@H](O)CNC(C)(C)CCCC(C)C)cc12 ZINC000147448015 KK Annotated Anodyne CTSD 56 62 CCc1c[nH]c2c(N3CCCC3=O)cc(C(=O)N[C@@H](Cc3ccccc3)[C@@H](O)CNC(C)(C)CCCC(C)C)cc12 ZINC000147448015 KK Annotated Anodyne BACE2 69 62 CCc1c[nH]c2c(N3CCCC3=O)cc(C(=O)N[C@@H](Cc3ccccc3)[C@@H](O)CNC(C)(C)CCCC(C)C)cc12 ZINC000147448015 KK Annotated Anodyne BACE1 67 68 CCc1c[nH]c2c(N3CCCC3=O)cc(C(=O)N[C@@H](Cc3ccccc3)[C@@H](O)CNC(C)(C)CCCC(C)C)cc12 ZINC000147448015 KK Annotated Anodyne PLM1_PLAFA 59 42 CCc1c[nH]c2c(N3CCCC3=O)cc(C(=O)N[C@@H](Cc3ccccc3)[C@@H](O)CNC(C)(C)CCCC(C)C)cc12 ZINC000147448015 KK Annotated Anodyne PLM2_PLAFA 34 42 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccccc2N2CCCCC2)C1 ZINC000147448019 HG On-Demand Anodyne KCNQ2 88 43 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccccc2N2CCCCC2)C1 ZINC000147448019 HG On-Demand Anodyne CSF1R 22 45 CCc1ncc(C(=O)N[C@H](CC(C)C)c2nc3ccccc3[nH]2)s1 ZINC000147448072 EI On-Demand Anodyne MMP7 22 52 COc1cc(C(=O)N[C@H](C)c2cccc(Br)c2)ccc1F ZINC000147448086 FI On-Demand Anodyne TAAR1 16 42 CNC(=O)c1cccc(NC(=O)C(=O)N2CC=C(c3c(C)[nH]c4ccccc34)CC2)c1 ZINC000147448099 HG On-Demand Anodyne KCNK3 48 33 COc1cc(NC(=O)C2(N)CCC2)cc(OC)c1OC ZINC000147448108 CD On-Demand Anodyne TUBB1 52 37 CC(C)C[C@H](CS)NC(=O)OC(C)(C)C ZINC000147448130 BF For-Sale Mild CTSD 22 40 CC(C)C[C@H](CS)NC(=O)OC(C)(C)C ZINC000147448130 BF For-Sale Mild PAPA1_CARPA 43 36 CC(C)C[C@H](CS)NC(=O)OC(C)(C)C ZINC000147448130 BF For-Sale Mild CTSK 22 57 CC(C)C[C@H](CS)NC(=O)OC(C)(C)C ZINC000147448130 BF For-Sale Mild PGA 17 40 CC(C)C[C@H](CS)NC(=O)OC(C)(C)C ZINC000147448130 BF For-Sale Mild ECE1 32 40 CC(C)C[C@H](CS)NC(=O)OC(C)(C)C ZINC000147448130 BF For-Sale Mild PGA5 44 40 CC(C)C[C@H](CS)NC(=O)OC(C)(C)C ZINC000147448130 BF For-Sale Mild POLG_HCV1 24 40 CC(C)C[C@H](CS)NC(=O)OC(C)(C)C ZINC000147448130 BF For-Sale Mild FPR1 47 40 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2C2CCCCC2)no1 ZINC000147448149 DH Annotated Anodyne CNR2 19 98 CC(C)(C)c1cc(NC(=O)[C@@H]2CCCN2C2CCCCC2)no1 ZINC000147448149 DH Annotated Anodyne FLT3 46 39 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(-c2ccco2)on1 ZINC000147448164 HF On-Demand Anodyne HTR4 44 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(-c2ccco2)on1 ZINC000147448164 HF On-Demand Anodyne TGM2 48 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(-c2ccco2)on1 ZINC000147448164 HF On-Demand Anodyne CACNA1I 42 35 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(-c2ccco2)on1 ZINC000147448164 HF On-Demand Anodyne F13A1 29 40 O=C(Nc1cc(Cl)cc(Cl)c1)Nc1cc(NC(=O)Nc2cc(Cl)cc(Cl)c2)cc(C(=O)O)c1 ZINC000147448168 KK For-Sale Anodyne PPIA 24 58 O=C(Nc1cc(Cl)cc(Cl)c1)Nc1cc(NC(=O)Nc2cc(Cl)cc(Cl)c2)cc(C(=O)O)c1 ZINC000147448168 KK For-Sale Anodyne AKR1C3 25 46 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCN(C)CC3)cc1)C2 ZINC000147448171 HE On-Demand Anodyne MTNR1A 18 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCN(C)CC3)cc1)C2 ZINC000147448171 HE On-Demand Anodyne MTNR1B 20 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCN(C)CC3)cc1)C2 ZINC000147448171 HE On-Demand Anodyne ROCK2 32 51 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N3CCN(C)CC3)cc1)C2 ZINC000147448171 HE On-Demand Anodyne MTOR 18 43 Cc1c(NC[C@@H](C)CC(=O)O)cccc1[N+](=O)[O-] ZINC000147448191 CE For-Sale Bother COLA 109 38 NS(=O)(=O)c1cc(F)c(OCCc2ccccn2)c(F)c1 ZINC000147448195 DD For-Sale Anodyne CA2 18 44 NS(=O)(=O)c1cc(F)c(OCCc2ccccn2)c(F)c1 ZINC000147448195 DD For-Sale Anodyne CA1 18 43 NS(=O)(=O)c1cc(F)c(OCCc2ccccn2)c(F)c1 ZINC000147448195 DD For-Sale Anodyne CA7 18 42 NS(=O)(=O)c1cc(F)c(OCCc2ccccn2)c(F)c1 ZINC000147448195 DD For-Sale Anodyne CA4 16 44 NS(=O)(=O)c1cc(F)c(OCCc2ccccn2)c(F)c1 ZINC000147448195 DD For-Sale Anodyne CA5A 15 42 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccccc2N2CCCCC2)C1 ZINC000147448202 HG On-Demand Anodyne KCNQ2 88 43 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne CA2 126 59 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne PTGS2 34 41 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne CA6 28 45 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne CA1 98 59 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne CA7 63 53 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne CA13 37 42 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne CA4 86 59 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne CA5A 40 35 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne CA14 52 49 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne CA12 68 53 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne ALPL 15 42 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne CA9 74 56 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne CYNT 49 53 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne NCE103 41 53 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne ALPI 15 42 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne UTS2 46 40 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne MTCA1 68 35 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne P96878_MYCTU 74 44 Cc1ccc(C(NC(=O)c2ccc(S(N)(=O)=O)cc2)c2ccc(C)cc2)cc1 ZINC000147448280 GG For-Sale Anodyne A6YCJ1_9METZ 23 53 CC(C)(C)c1ccc(NC(=O)C2(N)CCC2)cc1 ZINC000147448320 BF On-Demand Anodyne TRPV1 28 44 CC(C)(C)c1ccc(NC(=O)C2(N)CCC2)cc1 ZINC000147448320 BF On-Demand Anodyne CYNT 42 43 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cccc([N+](=O)[O-])c3)ccc21 ZINC000147448326 EE On-Demand Bother PPIA 17 43 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cccc([N+](=O)[O-])c3)ccc21 ZINC000147448326 EE On-Demand Bother EPHX2 18 42 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cccc([N+](=O)[O-])c3)ccc21 ZINC000147448326 EE On-Demand Bother F2RL3 48 35 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cccc([N+](=O)[O-])c3)ccc21 ZINC000147448326 EE On-Demand Bother TRPM8 19 42 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cccc([N+](=O)[O-])c3)ccc21 ZINC000147448326 EE On-Demand Bother AKR1C2 15 41 Cn1c(=O)n(C)c2cc(NC(=O)Nc3cccc([N+](=O)[O-])c3)ccc21 ZINC000147448326 EE On-Demand Bother KCNK3 45 31 Cc1c(NC[C@H](C)CC(=O)O)cccc1[N+](=O)[O-] ZINC000147448342 CE For-Sale Bother COLA 109 38 CCON(C)C(=O)[C@@H]1CCCN1C(=O)OC(C)(C)C ZINC000147448343 CD On-Demand Anodyne PREP 27 56 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1cccc(-n2cccn2)c1 ZINC000147448401 HJ On-Demand Anodyne ROCK2 21 43 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1cccc(-n2cccn2)c1 ZINC000147448401 HJ On-Demand Anodyne MET 47 43 O=C(NCc1ccc(Oc2cccnc2)c(F)c1)Nc1cccc(-n2cccn2)c1 ZINC000147448401 HJ On-Demand Anodyne NAMPT 44 43 Cc1ccc(C(=O)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147448410 HE On-Demand Anodyne EPHX2 36 42 Cc1ccc(C(=O)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147448410 HE On-Demand Anodyne TGM2 67 45 Cc1ccc(C(=O)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147448410 HE On-Demand Anodyne CACNA1I 54 40 Cc1ccc(C(=O)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147448410 HE On-Demand Anodyne F13A1 65 45 Cc1ccc(C(=O)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147448410 HE On-Demand Anodyne AKR1C3 45 37 CC(C)(C)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147448428 DC For-Sale Anodyne CA2 34 40 CC(C)(C)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147448428 DC For-Sale Anodyne CA1 27 40 CC(C)(C)NC(=O)COc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147448428 DC For-Sale Anodyne CA4 30 40 NC(=O)c1ccc(Oc2nc(N)ncc2Cl)cc1 ZINC000147448429 CD For-Sale Anodyne CHEK2 72 44 CC(C)(C)c1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147448522 CG For-Sale Anodyne CACNA2D1 0 40 CC(C)(C)c1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147448522 CG For-Sale Anodyne TRPV1 25 40 CC(C)(C)c1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147448522 CG For-Sale Anodyne CYNT 39 40 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne CA2 139 55 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne LPL 43 32 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne CA1 125 55 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne CA7 68 47 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne CA5B 42 42 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne CA4 97 55 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne CA5A 48 42 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne CA14 59 47 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne CA12 107 57 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne CA9 115 57 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne CYNT 45 49 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne NCE103 62 42 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne MTCA1 69 57 Cn1c(=O)n(C)c2cc(NC(=O)Nc3ccc(S(N)(=O)=O)cc3)ccc21 ZINC000147448544 GD On-Demand Anodyne P96878_MYCTU 86 57 O=S(=O)(NC[C@@H]1CCCO[C@@H]1c1ccccc1)c1cccnc1 ZINC000147448554 EF On-Demand Anodyne NPY2R 35 40 CNc1nccc(Oc2ccc(C(N)=O)cc2)n1 ZINC000147448632 BD For-Sale Anodyne CHEK2 32 40 O=S(=O)(NC[C@@H]1CCCO[C@H]1c1ccccc1)c1cccnc1 ZINC000147448672 EF On-Demand Anodyne NPY2R 35 40 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne EPHX1 0 49 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne SRD5A2 0 40 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne LTA4H 58 47 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne CA1 44 50 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne MMP13 25 40 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne RAF1 22 42 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne MMP2 24 40 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne NPY5R 26 42 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne MMP9 23 40 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne EPHX2 18 49 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne CA12 18 50 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne CA9 20 50 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne Q8MMZ8_EIMTE 24 42 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne F13A1 24 48 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne NCE103 22 40 NC1(C(=O)Nc2ccc(Oc3ccccc3)cc2)CCC1 ZINC000147448753 CG For-Sale Anodyne UPPS 0 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1C[C@@H]2CCC[C@H](C1)C2=O ZINC000147448761 HF On-Demand Anodyne FKBP1A 17 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1C[C@@H]2CCC[C@H](C1)C2=O ZINC000147448761 HF On-Demand Anodyne EPHX2 35 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1C[C@@H]2CCC[C@H](C1)C2=O ZINC000147448761 HF On-Demand Anodyne TGM2 71 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1C[C@@H]2CCC[C@H](C1)C2=O ZINC000147448761 HF On-Demand Anodyne F13A1 76 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1C[C@@H]2CCC[C@H](C1)C2=O ZINC000147448761 HF On-Demand Anodyne NAMPT 32 40 O=C(NCC1(C(=O)O)CCC1)c1cccc(Cl)c1 ZINC000147448771 CE On-Demand Anodyne CCKBR 44 42 O=C(NCC1(C(=O)O)CCC1)c1cccc(Cl)c1 ZINC000147448771 CE On-Demand Anodyne CACNA1I 26 41 O=C(NCC1(C(=O)O)CCC1)c1cccc(Cl)c1 ZINC000147448771 CE On-Demand Anodyne KCNK3 66 52 O=C(NCC1(C(=O)O)CCC1)c1cccc(Cl)c1 ZINC000147448771 CE On-Demand Anodyne KCNK9 29 46 COCc1nc(C(=O)Nc2cccc(C(=O)NC3CC3)c2)cs1 ZINC000147448798 EE On-Demand Anodyne MAPK14 35 40 COCc1nc(C(=O)Nc2cccc(C(=O)NC3CC3)c2)cs1 ZINC000147448798 EE On-Demand Anodyne KCNK3 74 37 COCc1nc(C(=O)Nc2cccc(C(=O)NC3CC3)c2)cs1 ZINC000147448798 EE On-Demand Anodyne KCNK9 59 35 O=S(=O)(NC[C@H]1CCCO[C@@H]1c1ccccc1)c1cccnc1 ZINC000147448809 EF On-Demand Anodyne NPY2R 35 40 O=C(NC[C@@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(-n2cccn2)c1 ZINC000147448819 GI On-Demand Anodyne PRMT3 45 33 CC(C)CN(C(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147448842 DH On-Demand Anodyne CACNA1I 47 35 C[C@H](CNc1ccc([N+](=O)[O-])c2nonc12)CC(=O)O ZINC000147448868 CD For-Sale Bother GSTM2 135 47 C[C@H](CNc1ccc([N+](=O)[O-])c2nonc12)CC(=O)O ZINC000147448868 CD For-Sale Bother GSTP1 84 47 C[C@H](CNc1ccc([N+](=O)[O-])c2nonc12)CC(=O)O ZINC000147448868 CD For-Sale Bother MYC 0 46 CCOCCOC(=O)c1ccc(CNC)cc1 ZINC000147448872 BD For-Sale Anodyne LPAR2 19 49 O=S(=O)(NC[C@H]1CCCO[C@H]1c1ccccc1)c1cccnc1 ZINC000147448936 EF On-Demand Anodyne NPY2R 35 40 CCOc1nc(N)nc(Oc2ccc(C(N)=O)cc2)n1 ZINC000147448984 CC For-Sale Anodyne CHEK2 41 43 O=C(NC[C@@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(-n2cccn2)c1 ZINC000147449026 GI On-Demand Anodyne PRMT3 45 33 C[C@@H](CNc1ccc([N+](=O)[O-])c2nonc12)CC(=O)O ZINC000147449055 CD For-Sale Bother GSTM2 135 47 C[C@@H](CNc1ccc([N+](=O)[O-])c2nonc12)CC(=O)O ZINC000147449055 CD For-Sale Bother GSTP1 84 47 C[C@@H](CNc1ccc([N+](=O)[O-])c2nonc12)CC(=O)O ZINC000147449055 CD For-Sale Bother MYC 0 46 NC[C@H]1CCCN1C[C@H](O)CO ZINC000147449102 AA For-Sale Anodyne SLC18A2 52 40 O=C(NC[C@H]1CCCO[C@@H]1c1ccccc1)Nc1cccc(-n2cccn2)c1 ZINC000147449235 GI On-Demand Anodyne PRMT3 45 33 NC[C@@H]1CCCN1C[C@H](O)CO ZINC000147449298 AA For-Sale Anodyne SLC18A2 52 40 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne BMP1 101 42 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne MMP13 66 42 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne MMP2 51 63 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne MMP3 49 51 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne MMP8 32 48 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne MMP14 21 42 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne MMP9 53 63 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne MMP12 35 50 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne MMP10 15 51 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne MMP7 45 51 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne ADAMTS4 58 35 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne MMP1 56 51 CCN(CC)[C@@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449305 FD On-Demand Anodyne LEF 22 51 C[C@H](CNc1ccc([N+](=O)[O-])c(N)n1)CC(=O)O ZINC000147449310 CD For-Sale Bother GSTM2 40 35 O=C(Cc1ccc2c(c1)CCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147449341 HE On-Demand Anodyne CHRM5 22 40 O=C(Cc1ccc2c(c1)CCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147449341 HE On-Demand Anodyne PKM 33 44 O=C(Cc1ccc2c(c1)CCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147449341 HE On-Demand Anodyne TGM2 58 42 O=C(Cc1ccc2c(c1)CCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147449341 HE On-Demand Anodyne F13A1 49 42 O=C(Cc1ccc2c(c1)CCO2)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147449341 HE On-Demand Anodyne AKR1C3 46 33 O=C(NC[C@H]1CCCO[C@H]1c1ccccc1)Nc1cccc(-n2cccn2)c1 ZINC000147449457 GI On-Demand Anodyne PRMT3 45 33 CC(C)NC(=O)CCOc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147449458 DC For-Sale Anodyne CA2 39 40 COc1cc(N)cc(C(=O)Nc2ccncc2Br)c1 ZINC000147449475 DF For-Sale Anodyne TAAR1 24 40 COc1cc(N)cc(C(=O)Nc2ccncc2Br)c1 ZINC000147449475 DF For-Sale Anodyne SIRT2 22 42 COc1cc(N)cc(C(=O)Nc2ccncc2Br)c1 ZINC000147449475 DF For-Sale Anodyne GPR35 41 35 CC[C@@H](C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147449503 CG On-Demand Anodyne HCAR1 0 42 C[C@@H](CNc1ccc([N+](=O)[O-])c(N)n1)CC(=O)O ZINC000147449509 CD For-Sale Bother GSTM2 40 35 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne BMP1 101 42 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne MMP13 66 42 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne MMP2 51 63 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne MMP3 49 51 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne MMP8 32 48 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne MMP14 21 42 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne MMP9 53 63 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne MMP12 35 50 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne MMP10 15 51 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne MMP7 45 51 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne ADAMTS4 58 35 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne MMP1 56 51 CCN(CC)[C@H](C)CNC(=O)[C@H](C)NS(=O)(=O)c1ccc(OC)cc1 ZINC000147449515 FD On-Demand Anodyne LEF 22 51 CCNc1cc(C(=O)NCCNC(=O)N(C)C)ccn1 ZINC000147449572 CC For-Sale Anodyne KDM4E 24 41 Cc1ccc(C)c(S(=O)(=O)N2CCN(CCBr)CC2)c1 ZINC000147449626 FE For-Sale Reactive EPHX2 24 40 CNC(=O)CCOc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147449667 CC For-Sale Anodyne CA2 40 44 CNC(=O)CCOc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147449667 CC For-Sale Anodyne CA1 32 44 CNC(=O)CCOc1c(F)cc(S(N)(=O)=O)cc1F ZINC000147449667 CC For-Sale Anodyne CA4 41 44 CC[C@H](C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147449706 CG On-Demand Anodyne HCAR1 0 42 Nc1cccc(Cl)c1C(=O)Nc1ccncc1Br ZINC000147449721 EG For-Sale Anodyne JAK1 0 64 Nc1cccc(Cl)c1C(=O)Nc1ccncc1Br ZINC000147449721 EG For-Sale Anodyne HDAC1 0 42 Nc1cccc(Cl)c1C(=O)Nc1ccncc1Br ZINC000147449721 EG For-Sale Anodyne TYK2 64 40 CCN(CC)[C@H](C)CNC(=O)CCC(=O)c1ccc2ccccc2c1 ZINC000147449743 EH On-Demand Anodyne CCR2 16 40 COC(=O)Cc1csc(-c2ccc(O)c(Cl)c2)n1 ZINC000147449754 CF For-Sale Anodyne PDK1 43 33 COC(=O)Cc1csc(-c2ccc(O)c(Cl)c2)n1 ZINC000147449754 CF For-Sale Anodyne NCE103 26 40 COC(=O)Cc1csc(-c2ccc(O)c(Cl)c2)n1 ZINC000147449754 CF For-Sale Anodyne CAN2 0 40 Cc1c(Br)cc(C(=O)O)c(N)c1O ZINC000147449756 BD For-Sale Anodyne AKR1C2 50 44 Cc1c(Br)cc(C(=O)O)c(N)c1O ZINC000147449756 BD For-Sale Anodyne AKR1C1 53 44 CC[C@@H](C)[C@H](NC(=O)c1cc(C)ccc1Br)C(=O)OC ZINC000147449765 EG On-Demand Anodyne PAPA1_CARPA 45 34 CS(=O)(=O)c1cc(C(=O)N2CCC[C@@H]2c2ccccc2Cl)cc([N+](=O)[O-])c1 ZINC000147449800 HH On-Demand Bother SFRP1 42 33 CS(=O)(=O)c1cc(C(=O)N2CCC[C@@H]2c2ccccc2Cl)cc([N+](=O)[O-])c1 ZINC000147449800 HH On-Demand Bother WNT3 40 33 NC(=O)c1ccc(Oc2nc(N)cn3ccnc23)cc1 ZINC000147449820 CD For-Sale Anodyne SYK 15 42 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)s1 ZINC000147449921 CH On-Demand Anodyne CPT1A 0 47 CCOc1ccc(C(=O)Nc2ccncc2Br)cc1N ZINC000147449959 EG For-Sale Anodyne ROCK2 40 38 CCOc1ccc(C(=O)Nc2ccncc2Br)cc1N ZINC000147449959 EG For-Sale Anodyne HDAC1 42 38 CC[C@H](C)[C@H](NC(=O)c1cc(C)ccc1Br)C(=O)OC ZINC000147449960 EG On-Demand Anodyne PAPA1_CARPA 45 34 CS(=O)(=O)c1cc(C(=O)N2CCC[C@H]2c2ccccc2Cl)cc([N+](=O)[O-])c1 ZINC000147450002 HH On-Demand Bother SFRP1 42 33 CS(=O)(=O)c1cc(C(=O)N2CCC[C@H]2c2ccccc2Cl)cc([N+](=O)[O-])c1 ZINC000147450002 HH On-Demand Bother WNT3 40 33 CC(C)(C)c1nc2cc(N)ccc2n1CCNC(N)=O ZINC000147450095 CD For-Sale Anodyne CNR2 17 41 Cc1cc(C(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)cc([N+](=O)[O-])c1 ZINC000147450142 GG On-Demand Bother L3MBTL3 42 35 CCCOC(=O)c1ccc(OC(=O)c2ccccc2C(=O)Oc2ccc(C(=O)OCCC)cc2)cc1 ZINC000147450152 JK For-Sale Anodyne PRSS1 20 50 CCCOC(=O)c1ccc(OC(=O)c2ccccc2C(=O)Oc2ccc(C(=O)OCCC)cc2)cc1 ZINC000147450152 JK For-Sale Anodyne ACR 93 50 CC[C@@H](C)[C@@H](NC(=O)c1cc(C)ccc1Br)C(=O)OC ZINC000147450168 EG On-Demand Anodyne PAPA1_CARPA 45 34 O=C(/C=C/c1ccco1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147450169 CG On-Demand Anodyne MMP9 0 43 O=C(/C=C/c1ccco1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147450169 CG On-Demand Anodyne MMP1 0 46 C[C@H](CNc1ccccc1C(F)(F)F)CC(=O)O ZINC000147450183 CG For-Sale Anodyne ANPEP 16 50 C[C@H](CNc1ccccc1C(F)(F)F)CC(=O)O ZINC000147450183 CG For-Sale Anodyne RBP4 52 36 Cc1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)cc1Cl ZINC000147450201 FG On-Demand Anodyne NPY2R 40 36 Cc1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)cc1Cl ZINC000147450201 FG On-Demand Anodyne ENV 40 31 CN1CC[C@]23CC(=O)CC[C@@]2(O)[C@H]1Cc1ccc(C(=O)NCCc2ccc(-c4cnc(=O)[nH]c4)cc2)c(O)c13 ZINC000147450209 KE Annotated Anodyne OPRM1 31 53 CN1CC[C@]23CC(=O)CC[C@@]2(O)[C@H]1Cc1ccc(C(=O)NCCc2ccc(-c4cnc(=O)[nH]c4)cc2)c(O)c13 ZINC000147450209 KE Annotated Anodyne OPRD1 33 48 CN1CC[C@]23CC(=O)CC[C@@]2(O)[C@H]1Cc1ccc(C(=O)NCCc2ccc(-c4cnc(=O)[nH]c4)cc2)c(O)c13 ZINC000147450209 KE Annotated Anodyne OPRK1 29 53 COc1ccc(Cl)cc1CC(=O)c1cncs1 ZINC000147450252 CG For-Sale Anodyne PDE4D 15 42 NC(=O)c1ccc(OCC(=O)N2CCC[C@H](C(=O)Nc3nccs3)C2)cc1 ZINC000147450283 GD On-Demand Anodyne MAP1 105 42 NC(=O)c1ccc(OCC(=O)N2CCC[C@H](C(=O)Nc3nccs3)C2)cc1 ZINC000147450283 GD On-Demand Anodyne CPT1A 63 43 NC(=O)c1ccc(OCC(=O)N2CCC[C@H](C(=O)Nc3nccs3)C2)cc1 ZINC000147450283 GD On-Demand Anodyne GCK 22 41 CC[C@H](C)[C@@H](NC(=O)c1cc(C)ccc1Br)C(=O)OC ZINC000147450373 EG On-Demand Anodyne PAPA1_CARPA 45 34 O=C(NCC1(CO)CC1)Nc1ccc([N+](=O)[O-])cc1 ZINC000147450376 CD On-Demand Bother NADE 0 42 O=C(NCC1(CO)CC1)Nc1ccc([N+](=O)[O-])cc1 ZINC000147450376 CD On-Demand Bother NMBR 74 42 O=C(NCC1(CO)CC1)Nc1ccc([N+](=O)[O-])cc1 ZINC000147450376 CD On-Demand Bother GRPR 37 42 O=C(NCC1(CO)CC1)Nc1ccc([N+](=O)[O-])cc1 ZINC000147450376 CD On-Demand Bother NCE103 23 46 O=C(NCC1(CO)CC1)Nc1ccc([N+](=O)[O-])cc1 ZINC000147450376 CD On-Demand Bother ACAT 0 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne EPHX1 0 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne RARA 16 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne PPIA 22 56 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne ECR 44 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne CPT1A 48 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne PRNP 52 61 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne PPARD 0 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne GRM4 39 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne NR1H4 23 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne GRM5 16 48 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne LUCI_LUCLA 34 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne TAAR1 27 49 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne AKR1C3 47 53 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne PTPA 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne SHH 37 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne CYA 0 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne SMO 25 53 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne HCAR1 0 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne GPR35 19 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne SENP1 0 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne PARP15 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne E3UJZ5_SPOLI 28 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne KCNK3 120 62 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne KCNK9 62 47 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2)c1 ZINC000147450378 CG On-Demand Anodyne PARP10 0 40 CCCCCCCCOc1c(F)cc(CBr)cc1F ZINC000147450404 EK For-Sale Reactive LPAR2 48 39 CCCCCCCCOc1c(F)cc(CBr)cc1F ZINC000147450404 EK For-Sale Reactive PLA2G4B 47 31 CCCCCCCCOc1c(F)cc(CBr)cc1F ZINC000147450404 EK For-Sale Reactive S1PR2 48 39 C[C@@H](CNc1ccccc1C(F)(F)F)CC(=O)O ZINC000147450408 CG For-Sale Anodyne ANPEP 16 50 C[C@@H](CNc1ccccc1C(F)(F)F)CC(=O)O ZINC000147450408 CG For-Sale Anodyne RBP4 52 36 Cc1ccc(Sc2ccccc2C2=CCNCC2)cc1C ZINC000147450410 CJ For-Sale Anodyne HTR3A 18 52 CN(C)c1c(Cl)cccc1NC(=O)NCc1ccc(-n2ccnc2)c(F)c1 ZINC000147450414 GI On-Demand Anodyne NOS2 78 35 COC(=O)Cc1csc(-c2ccc(OC)c(Br)c2)n1 ZINC000147450415 EG For-Sale Anodyne DCK 43 40 COC(=O)Cc1csc(-c2ccc(OC)c(Br)c2)n1 ZINC000147450415 EG For-Sale Anodyne PPARD 20 42 COc1cc(NC(=O)C2(N)CCC2)c(OC)cc1Cl ZINC000147450420 CE For-Sale Anodyne HTR4 35 40 Cc1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)cc1Cl ZINC000147450432 FG On-Demand Anodyne NPY2R 40 36 Cc1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)cc1Cl ZINC000147450432 FG On-Demand Anodyne ENV 40 31 CNC(=O)COc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147450443 FD On-Demand Bother ROCK1 29 42 CNC(=O)COc1cccc(CNC(=O)c2cc(OC)ccc2[N+](=O)[O-])c1 ZINC000147450443 FD On-Demand Bother ROCK2 32 42 NCC[C@@H]1CCCCN1C[C@H](O)CO ZINC000147450450 BB For-Sale Anodyne SLC18A2 56 40 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H](C(=O)Nc3nccs3)C2)cc1 ZINC000147450503 GD On-Demand Anodyne MAP1 105 42 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H](C(=O)Nc3nccs3)C2)cc1 ZINC000147450503 GD On-Demand Anodyne CPT1A 63 43 NC(=O)c1ccc(OCC(=O)N2CCC[C@@H](C(=O)Nc3nccs3)C2)cc1 ZINC000147450503 GD On-Demand Anodyne GCK 22 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1(c2ccccc2)CCC1 ZINC000147450508 HG On-Demand Anodyne EPHX2 17 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1(c2ccccc2)CCC1 ZINC000147450508 HG On-Demand Anodyne TGM2 68 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1(c2ccccc2)CCC1 ZINC000147450508 HG On-Demand Anodyne CACNA1I 19 47 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1(c2ccccc2)CCC1 ZINC000147450508 HG On-Demand Anodyne F13A1 71 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1(c2ccccc2)CCC1 ZINC000147450508 HG On-Demand Anodyne NAMPT 39 42 CC(C)N(CC1CC1)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147450515 DH For-Sale Anodyne CACNA1I 53 38 CC(C)(C)CC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147450594 CG On-Demand Anodyne CACNA1H 15 41 CC(C)(C)CC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147450594 CG On-Demand Anodyne CACNA1I 48 37 CC(C)(C)CC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147450594 CG On-Demand Anodyne HCAR1 0 43 C[C@@H]1CN(C(=O)Nc2cccc(Cl)c2N(C)C)C[C@H](c2ccccc2)O1 ZINC000147450624 FI On-Demand Anodyne SMO 24 40 COC(=O)[C@H]1CCCN1C(=O)c1ccc(F)c(OC)c1 ZINC000147450653 CD On-Demand Anodyne FKBP12.6 0 40 NCC[C@H]1CCCCN1C[C@H](O)CO ZINC000147450661 BB For-Sale Anodyne SLC18A2 56 40 CCCc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147450769 GE On-Demand Anodyne HTR4 46 36 CCCc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147450769 GE On-Demand Anodyne GRIN2B 28 40 CCCc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147450769 GE On-Demand Anodyne TGM2 47 40 CCCc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147450769 GE On-Demand Anodyne CACNA1I 57 35 CCCc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n[nH]1 ZINC000147450769 GE On-Demand Anodyne F13A1 28 40 COCCOCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147450833 CD On-Demand Anodyne CACNA1I 46 34 COCCOCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147450833 CD On-Demand Anodyne HCAR1 0 41 C[C@H]1CN(C(=O)Nc2cccc(Cl)c2N(C)C)C[C@H](c2ccccc2)O1 ZINC000147450840 FI On-Demand Anodyne SMO 24 40 COC(=O)[C@@H]1CCCN1C(=O)c1ccc(F)c(OC)c1 ZINC000147450866 CD On-Demand Anodyne FKBP12.6 0 40 O=S(=O)(c1ccc2c(c1)CCC2)N1CCN(CCBr)CC1 ZINC000147450884 FD For-Sale Reactive AKR1C3 55 34 CNc1cn2ccnc2c(Oc2cc(C)cc(C)c2C)n1 ZINC000147450956 CG For-Sale Anodyne HIVRT 0 55 CC[C@@H](C)Oc1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147450966 DI On-Demand Anodyne PLG 19 40 CC[C@@H](C)Oc1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147450966 DI On-Demand Anodyne PRSS1 20 41 CC[C@@H](C)Oc1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147450966 DI On-Demand Anodyne NPR1 40 33 CC[C@@H](C)Oc1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147450966 DI On-Demand Anodyne PRNP 44 33 CC[C@@H](C)Oc1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147450966 DI On-Demand Anodyne F3 53 35 CC[C@@H](C)Oc1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147450966 DI On-Demand Anodyne PLAU 21 41 CC[C@@H](C)Oc1ccc(NC(=O)c2ccc3c(c2)COC3)cc1 ZINC000147450966 DI On-Demand Anodyne ACR 45 35 Cc1c(O)cccc1C(=O)N1CCC[C@@H]1C(=O)O ZINC000147450994 BD For-Sale Anodyne ACE 48 43 Cc1c(O)cccc1C(=O)N1CCC[C@@H]1C(=O)O ZINC000147450994 BD For-Sale Anodyne SLC6A1 40 33 Cc1c(O)cccc1C(=O)N1CCC[C@@H]1C(=O)O ZINC000147450994 BD For-Sale Anodyne PREP 75 40 Cc1c(O)cccc1C(=O)N1CCC[C@@H]1C(=O)O ZINC000147450994 BD For-Sale Anodyne DAPE 0 40 Nc1cc(Br)cc(C(=O)Nc2ccncc2Br)c1 ZINC000147451027 FG For-Sale Anodyne HDAC1 0 41 C[C@@H]1CN(C(=O)Nc2cccc(Cl)c2N(C)C)C[C@@H](c2ccccc2)O1 ZINC000147451045 FI On-Demand Anodyne SMO 24 40 C[C@@H]1C[C@@H]1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147451071 CF On-Demand Anodyne CACNA1I 41 33 C[C@@H]1C[C@@H]1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147451071 CF On-Demand Anodyne HCAR1 0 41 CCc1ncc(C(=O)Nc2ccccc2C(=O)N2CCCC2)s1 ZINC000147451095 EG On-Demand Anodyne NPSR1 15 51 CC(C)(C)CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147451194 FF On-Demand Anodyne NPY2R 17 40 Cc1ccc(Br)c(C(=O)NCc2ccc(F)c(F)c2)c1 ZINC000147451205 EH On-Demand Anodyne LEF 56 37 Cc1c(O)cccc1C(=O)N1CCC[C@H]1C(=O)O ZINC000147451216 BD For-Sale Anodyne ACE 48 43 Cc1c(O)cccc1C(=O)N1CCC[C@H]1C(=O)O ZINC000147451216 BD For-Sale Anodyne SLC6A1 40 33 Cc1c(O)cccc1C(=O)N1CCC[C@H]1C(=O)O ZINC000147451216 BD For-Sale Anodyne PREP 75 40 Cc1c(O)cccc1C(=O)N1CCC[C@H]1C(=O)O ZINC000147451216 BD For-Sale Anodyne DAPE 0 40 C=CCN(CC=C)C(=O)c1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147451217 HH On-Demand Mild ROCK2 36 52 C[C@H]1C[C@@H]1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147451259 CF On-Demand Anodyne CACNA1I 41 33 C[C@H]1C[C@@H]1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147451259 CF On-Demand Anodyne HCAR1 0 41 C[C@H]1CN(C(=O)Nc2cccc(Cl)c2N(C)C)C[C@@H](c2ccccc2)O1 ZINC000147451267 FI On-Demand Anodyne SMO 24 40 Cc1cc(C(=O)Nc2ccccc2C(=O)N2CCCC2)cc([N+](=O)[O-])c1 ZINC000147451320 FG On-Demand Bother PYGL 23 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(N3CCCC3)c(F)c2)c1 ZINC000147451394 FH On-Demand Bother NPY2R 82 43 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(N3CCCC3)c(F)c2)c1 ZINC000147451394 FH On-Demand Bother TAAR1 47 59 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(N3CCCC3)c(F)c2)c1 ZINC000147451394 FH On-Demand Bother AKR1C3 17 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(N3CCCC3)c(F)c2)c1 ZINC000147451394 FH On-Demand Bother AKR1C2 50 38 O=C(c1ccc2ccccc2c1)N1CCC[C@@H]1CCCBr ZINC000147451408 EJ For-Sale Reactive HCRTR1 15 45 O=C(c1ccc2ccccc2c1)N1CCC[C@@H]1CCCBr ZINC000147451408 EJ For-Sale Reactive PREP 47 39 O=C(c1ccc2ccccc2c1)N1CCC[C@@H]1CCCBr ZINC000147451408 EJ For-Sale Reactive FAP 0 46 O=C(c1ccc2ccccc2c1)N1CCC[C@@H]1CCCBr ZINC000147451408 EJ For-Sale Reactive L3MBTL1 0 41 O=C(c1ccc2ccccc2c1)N1CCC[C@@H]1CCCBr ZINC000147451408 EJ For-Sale Reactive L3MBTL3 45 41 CCOC(=O)c1ccc(CNC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147451478 FF On-Demand Anodyne MTNR1A 27 40 C[C@@H]1C[C@H]1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147451503 CF On-Demand Anodyne CACNA1I 41 33 C[C@@H]1C[C@H]1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147451503 CF On-Demand Anodyne HCAR1 0 41 Cc1ccc(Br)c(C(=O)NCc2cccc(Br)c2)c1 ZINC000147451529 GI On-Demand Anodyne ANPEP 28 43 N#Cc1ccc(C[S@](=O)c2ccc3c(c2)OCCO3)cc1 ZINC000147451535 CF On-Demand Mild GSK3A 22 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@@H]1c1ccc(F)cc1 ZINC000147451541 HG On-Demand Anodyne EPHX2 29 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@@H]1c1ccc(F)cc1 ZINC000147451541 HG On-Demand Anodyne TGM2 66 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@@H]1c1ccc(F)cc1 ZINC000147451541 HG On-Demand Anodyne F13A1 71 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@@H]1c1ccc(F)cc1 ZINC000147451541 HG On-Demand Anodyne NAMPT 45 39 COc1ccc(S(=O)(=O)N2CCN(C(=O)CN(C)CC(=O)N(C)C)CC2)cc1 ZINC000147451542 HB On-Demand Anodyne MMP13 61 45 COc1ccc(S(=O)(=O)N2CCN(C(=O)CN(C)CC(=O)N(C)C)CC2)cc1 ZINC000147451542 HB On-Demand Anodyne MMP2 31 45 COc1ccc(S(=O)(=O)N2CCN(C(=O)CN(C)CC(=O)N(C)C)CC2)cc1 ZINC000147451542 HB On-Demand Anodyne MMP3 60 45 COc1ccc(S(=O)(=O)N2CCN(C(=O)CN(C)CC(=O)N(C)C)CC2)cc1 ZINC000147451542 HB On-Demand Anodyne MMP8 39 45 COc1ccc(S(=O)(=O)N2CCN(C(=O)CN(C)CC(=O)N(C)C)CC2)cc1 ZINC000147451542 HB On-Demand Anodyne MMP9 52 45 COc1ccc(S(=O)(=O)N2CCN(C(=O)CN(C)CC(=O)N(C)C)CC2)cc1 ZINC000147451542 HB On-Demand Anodyne PKM 21 57 COc1ccc(S(=O)(=O)N2CCN(C(=O)CN(C)CC(=O)N(C)C)CC2)cc1 ZINC000147451542 HB On-Demand Anodyne TGM2 58 40 COc1ccc(S(=O)(=O)N2CCN(C(=O)CN(C)CC(=O)N(C)C)CC2)cc1 ZINC000147451542 HB On-Demand Anodyne MMP7 51 45 COc1ccc(S(=O)(=O)N2CCN(C(=O)CN(C)CC(=O)N(C)C)CC2)cc1 ZINC000147451542 HB On-Demand Anodyne MMP1 61 45 COc1ccc(S(=O)(=O)N2CCN(C(=O)CN(C)CC(=O)N(C)C)CC2)cc1 ZINC000147451542 HB On-Demand Anodyne F13A1 68 40 Cc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147451575 CE On-Demand Anodyne LCK 29 45 Cc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147451575 CE On-Demand Anodyne CSNK1D 39 48 Cc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147451575 CE On-Demand Anodyne PIK3CA 0 43 Cc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147451575 CE On-Demand Anodyne FABK 0 48 Cc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147451575 CE On-Demand Anodyne PORCN 0 41 Cc1ccccc1[C@@H]1CCCN1C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147451602 GG On-Demand Bother SFRP1 42 33 Cc1ccccc1[C@@H]1CCCN1C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147451602 GG On-Demand Bother WNT3 42 33 O=C(c1ccc2ccccc2c1)N1CCC[C@H]1CCCBr ZINC000147451603 EJ For-Sale Reactive HCRTR1 15 45 O=C(c1ccc2ccccc2c1)N1CCC[C@H]1CCCBr ZINC000147451603 EJ For-Sale Reactive PREP 47 39 O=C(c1ccc2ccccc2c1)N1CCC[C@H]1CCCBr ZINC000147451603 EJ For-Sale Reactive FAP 0 46 O=C(c1ccc2ccccc2c1)N1CCC[C@H]1CCCBr ZINC000147451603 EJ For-Sale Reactive L3MBTL1 0 41 O=C(c1ccc2ccccc2c1)N1CCC[C@H]1CCCBr ZINC000147451603 EJ For-Sale Reactive L3MBTL3 45 41 C[C@H]1C[C@H]1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147451694 CF On-Demand Anodyne CACNA1I 41 33 C[C@H]1C[C@H]1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147451694 CF On-Demand Anodyne HCAR1 0 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C)cc1OC[C@@H]1CCCO1)C2 ZINC000147451705 GH On-Demand Anodyne ROCK2 34 47 Cc1ccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147451778 EJ On-Demand Anodyne SDH1 0 49 Cc1ccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147451778 EJ On-Demand Anodyne ACACA 46 35 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@@H]1c1ccc(F)cc1 ZINC000147451789 HG On-Demand Anodyne EPHX2 29 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@@H]1c1ccc(F)cc1 ZINC000147451789 HG On-Demand Anodyne TGM2 66 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@@H]1c1ccc(F)cc1 ZINC000147451789 HG On-Demand Anodyne F13A1 71 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1C[C@@H]1c1ccc(F)cc1 ZINC000147451789 HG On-Demand Anodyne NAMPT 45 39 Cc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147451809 CG For-Sale Anodyne LCK 30 43 Cc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147451809 CG For-Sale Anodyne CSNK1D 50 53 Cc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147451809 CG For-Sale Anodyne PIK3CA 19 42 Cc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147451809 CG For-Sale Anodyne FABK 0 46 Cc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147451809 CG For-Sale Anodyne PORCN 0 46 Cc1ccccc1[C@H]1CCCN1C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147451810 GG On-Demand Bother SFRP1 42 33 Cc1ccccc1[C@H]1CCCN1C(=O)c1cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 ZINC000147451810 GG On-Demand Bother WNT3 42 33 COc1cccc(OC)c1C(=O)N1CCC[C@@H]1CCCBr ZINC000147451857 FG For-Sale Reactive HTR1A 18 48 COc1cccc(OC)c1C(=O)N1CCC[C@@H]1CCCBr ZINC000147451857 FG For-Sale Reactive HCRTR1 24 43 COc1cccc(OC)c1C(=O)N1CCC[C@@H]1CCCBr ZINC000147451857 FG For-Sale Reactive HCRTR2 21 43 COc1cccc(OC)c1C(=O)N1CCC[C@@H]1CCCBr ZINC000147451857 FG For-Sale Reactive ACKR3 65 33 CC(C)(C)CC(=O)N1CCC(NC(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147451881 FH For-Sale Anodyne MAPK13 43 31 CC(C)(C)CC(=O)N1CCC(NC(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147451881 FH For-Sale Anodyne CCR2 43 37 CC(C)(C)CC(=O)N1CCC(NC(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147451881 FH For-Sale Anodyne SLC6A5 42 52 CC(C)(C)CC(=O)N1CCC(NC(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147451881 FH For-Sale Anodyne EPHX2 45 60 CC(C)(C)CC(=O)N1CCC(NC(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147451881 FH For-Sale Anodyne MCHR1 42 44 CC(C)(C)CC(=O)N1CCC(NC(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147451881 FH For-Sale Anodyne LIPG 51 36 CC(C)(C)CC(=O)N1CCC(NC(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147451881 FH For-Sale Anodyne SFRP1 91 42 CC(C)(C)CC(=O)N1CCC(NC(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147451881 FH For-Sale Anodyne WNT3 69 38 CC(C)(C)CC(=O)N1CCC(NC(=O)c2ccc(C(F)(F)F)cc2)CC1 ZINC000147451881 FH For-Sale Anodyne HPGDS 33 40 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne RARA 29 45 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne MAOB 0 43 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne PTGS2 26 51 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne PPIA 15 46 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne F10 0 51 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne RARG 25 45 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne RARB 30 45 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne UL80 17 42 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne ATF1 53 36 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne COLA 78 40 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne CPT1A 84 42 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne CPT2 49 38 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne PRNP 38 46 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne NR1H4 20 49 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne NFKB1 49 36 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne CPT1B 56 38 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne SCN10A 37 42 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne MCHR1 15 42 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne LUCI_LUCLA 29 40 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne TAAR1 48 47 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne AKR1C3 60 48 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne AKR1C2 61 44 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne NOD1 27 44 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne NOD2 41 44 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne GPR35 49 52 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne Q25615_ONCVO 30 40 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne SENP1 0 41 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne KCNK3 86 47 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147451901 DG On-Demand Anodyne KCNK9 41 38 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C)cc1OC[C@H]1CCCO1)C2 ZINC000147451908 GH On-Demand Anodyne ROCK2 34 47 NS(=O)(=O)c1cc(Br)c(OCCN2CCCCC2)cc1F ZINC000147451910 GE For-Sale Anodyne LTA4H 28 42 NS(=O)(=O)c1cc(Br)c(OCCN2CCCCC2)cc1F ZINC000147451910 GE For-Sale Anodyne HRH3 15 42 NS(=O)(=O)c1cc(Br)c(OCCN2CCCCC2)cc1F ZINC000147451910 GE For-Sale Anodyne PSMB2 45 36 NS(=O)(=O)c1cc(Br)c(OCCN2CCCCC2)cc1F ZINC000147451910 GE For-Sale Anodyne PSMB1 40 37 Cc1ccc([C@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452010 EJ On-Demand Anodyne SDH1 0 49 Cc1ccc([C@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452010 EJ On-Demand Anodyne ACACA 46 35 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@H]1c1ccc(F)cc1 ZINC000147452011 HG On-Demand Anodyne EPHX2 29 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@H]1c1ccc(F)cc1 ZINC000147452011 HG On-Demand Anodyne TGM2 66 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@H]1c1ccc(F)cc1 ZINC000147452011 HG On-Demand Anodyne F13A1 71 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@@H]1C[C@H]1c1ccc(F)cc1 ZINC000147452011 HG On-Demand Anodyne NAMPT 45 39 C[C@@H](Cc1cccc(F)c1)C(=O)N1CCO[C@H](C)C1 ZINC000147452037 CE On-Demand Anodyne TRY2_BOVIN 69 37 COc1cccc(OC)c1C(=O)N1CCC[C@H]1CCCBr ZINC000147452103 FG For-Sale Reactive HTR1A 18 48 COc1cccc(OC)c1C(=O)N1CCC[C@H]1CCCBr ZINC000147452103 FG For-Sale Reactive HCRTR1 24 43 COc1cccc(OC)c1C(=O)N1CCC[C@H]1CCCBr ZINC000147452103 FG For-Sale Reactive HCRTR2 21 43 COc1cccc(OC)c1C(=O)N1CCC[C@H]1CCCBr ZINC000147452103 FG For-Sale Reactive ACKR3 65 33 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C)cc1OC[C@@H]1CCCO1)C2 ZINC000147452113 GH On-Demand Anodyne ROCK2 34 47 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne AVPR2 31 41 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne AVPR1A 16 41 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne JUN 19 41 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne ECR 45 44 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne ATF1 54 37 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne NR1H4 17 44 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne MTTP 45 37 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne NFKB1 49 37 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne CSF1R 17 42 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne AKR1C3 45 43 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne AKR1C2 29 40 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne SMO 31 40 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne E3UJZ5_SPOLI 24 43 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne KCNK3 118 49 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne KCNK9 83 43 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1C ZINC000147452129 DH On-Demand Anodyne TMPRSS4 0 43 CN(C)c1ccc(C(=O)Nc2ccncc2Br)cc1N ZINC000147452159 EF For-Sale Anodyne HDAC1 28 43 C[C@H]1CN(C(=O)[C@@H](C)Cc2cccc(F)c2)CCO1 ZINC000147452199 CE On-Demand Anodyne TRY2_BOVIN 69 37 CC[C@H](NC(=O)c1cc(C)ccc1Br)c1ccccc1 ZINC000147452213 EJ On-Demand Anodyne TACR2 0 54 CC[C@H](NC(=O)c1cc(C)ccc1Br)c1ccccc1 ZINC000147452213 EJ On-Demand Anodyne PTGER3 54 37 CC[C@H](NC(=O)c1cc(C)ccc1Br)c1ccccc1 ZINC000147452213 EJ On-Demand Anodyne TACR3 60 54 CC[C@H](NC(=O)c1cc(C)ccc1Br)c1ccccc1 ZINC000147452213 EJ On-Demand Anodyne UTS2 58 39 Cc1nn(C)c(C)c1CCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147452225 HE On-Demand Anodyne TGM2 62 40 Cc1nn(C)c(C)c1CCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147452225 HE On-Demand Anodyne F13A1 61 40 Nc1ccccc1C(=O)CO ZINC000147452241 AC For-Sale Anodyne KYNU 0 56 CCN(CC)[C@@H](C)CNC(=O)CCNS(=O)(=O)c1ccc2ccccc2c1 ZINC000147452250 GE On-Demand Anodyne F2 20 41 CCN(CC)[C@@H](C)CNC(=O)CCNS(=O)(=O)c1ccc2ccccc2c1 ZINC000147452250 GE On-Demand Anodyne TRY2_BOVIN 67 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C)cc1OC[C@H]1CCCO1)C2 ZINC000147452314 GH On-Demand Anodyne ROCK2 34 47 CCCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147452341 CH On-Demand Anodyne CNR1 0 41 CCCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147452341 CH On-Demand Anodyne FABP4 18 42 CCCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147452341 CH On-Demand Anodyne HDAC3 18 43 CCCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147452341 CH On-Demand Anodyne MSR1 0 43 CCCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147452341 CH On-Demand Anodyne ENPP2 31 43 CCCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147452341 CH On-Demand Anodyne ACAT 0 51 CCCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147452341 CH On-Demand Anodyne HCAR1 0 40 CCCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147452341 CH On-Demand Anodyne NOD1 43 35 CC[C@H](NC(=O)N1CCN2CCCC[C@H]2C1)C(=O)O ZINC000147452392 CC For-Sale Anodyne L3MBTL1 0 40 CC[C@H](NC(=O)N1CCN2CCCC[C@H]2C1)C(=O)O ZINC000147452392 CC For-Sale Anodyne L3MBTL3 59 37 CC[C@@H](NC(=O)c1cc(C)ccc1Br)c1ccccc1 ZINC000147452397 EJ On-Demand Anodyne TACR2 0 54 CC[C@@H](NC(=O)c1cc(C)ccc1Br)c1ccccc1 ZINC000147452397 EJ On-Demand Anodyne PTGER3 54 37 CC[C@@H](NC(=O)c1cc(C)ccc1Br)c1ccccc1 ZINC000147452397 EJ On-Demand Anodyne TACR3 60 54 CC[C@@H](NC(=O)c1cc(C)ccc1Br)c1ccccc1 ZINC000147452397 EJ On-Demand Anodyne UTS2 58 39 Cc1cc(NC[C@@H](C)CC(=O)O)c2ccccc2n1 ZINC000147452415 CG On-Demand Anodyne ADAM17 61 36 C[C@H]1CN(C(=O)[C@H](C)Cc2cccc(F)c2)CCO1 ZINC000147452424 CE On-Demand Anodyne TRY2_BOVIN 69 37 CCCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147452427 BE For-Sale Anodyne NOS1 0 45 CCCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147452427 BE For-Sale Anodyne S1PR2 20 48 CCCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147452427 BE For-Sale Anodyne NOS3 15 43 CCCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147452427 BE For-Sale Anodyne DNPEP 0 44 CCCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147452427 BE For-Sale Anodyne DPP7 19 49 CCCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147452427 BE For-Sale Anodyne DPP8 0 47 CCCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147452427 BE For-Sale Anodyne DPP9 0 47 CCCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147452427 BE For-Sale Anodyne SIRT1 24 42 CCCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147452427 BE For-Sale Anodyne METAP2 0 43 CCCC[C@H](N)C(=O)NCCCCC(C)C ZINC000147452427 BE For-Sale Anodyne NOD1 87 52 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne PLG 21 44 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne CA2 22 47 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne HTR4 41 34 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne F10 21 40 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne GRIN2B 25 42 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne LPL 42 33 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne TGM1 15 46 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne EPHX2 31 47 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne TGM2 99 55 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne ST14 72 36 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne CACNA1I 62 38 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne F13A1 111 55 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne SFRP1 17 41 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne NOD2 40 34 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne NAMPT 59 45 NC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147452434 HE On-Demand Anodyne TMPRSS6 44 31 CCN(CC)[C@H](C)CNC(=O)CCNS(=O)(=O)c1ccc2ccccc2c1 ZINC000147452462 GE On-Demand Anodyne F2 20 41 CCN(CC)[C@H](C)CNC(=O)CCNS(=O)(=O)c1ccc2ccccc2c1 ZINC000147452462 GE On-Demand Anodyne TRY2_BOVIN 67 41 Cc1cc(C(=O)NCc2c(C)nn(Cc3ccccc3)c2C)cc([N+](=O)[O-])c1 ZINC000147452475 GH On-Demand Bother P2RX7 31 48 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)s2)c1 ZINC000147452580 DI On-Demand Anodyne PPIA 15 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)s2)c1 ZINC000147452580 DI On-Demand Anodyne HCAR1 0 40 O=C(NC1CCN(Cc2ccc(F)cc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147452616 GG On-Demand Anodyne DRD2 22 48 O=C(NC1CCN(Cc2ccc(F)cc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147452616 GG On-Demand Anodyne DRD4 33 48 O=C(NC1CCN(Cc2ccc(F)cc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147452616 GG On-Demand Anodyne ACHE 21 49 O=C(NC1CCN(Cc2ccc(F)cc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147452616 GG On-Demand Anodyne HTR2A 20 46 O=C(NC1CCN(Cc2ccc(F)cc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147452616 GG On-Demand Anodyne KCNH2 19 46 O=C(NC1CCN(Cc2ccc(F)cc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147452616 GG On-Demand Anodyne SIGMAR1 42 54 O=C(NC1CCN(Cc2ccc(F)cc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147452616 GG On-Demand Anodyne SSTR5 53 43 O=C(NC1CCN(Cc2ccc(F)cc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147452616 GG On-Demand Anodyne CCR3 87 55 O=C(NC1CCN(Cc2ccc(F)cc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147452616 GG On-Demand Anodyne MLNR 49 37 O=C(NC1CCN(Cc2ccc(F)cc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147452616 GG On-Demand Anodyne MCHR1 62 52 O=C(NC1CCN(Cc2ccc(F)cc2)CC1)C(=O)c1ccc2c(c1)CCC2 ZINC000147452616 GG On-Demand Anodyne CACNA1G 40 48 CCCCCCCOc1ccc(CNC(C)(C)C)nc1 ZINC000147452644 CI For-Sale Mild KCNQ1 0 41 CCCCCCCOc1ccc(CNC(C)(C)C)nc1 ZINC000147452644 CI For-Sale Mild PLA2G4B 87 40 Cc1cc(NC[C@H](C)CC(=O)O)c2ccccc2n1 ZINC000147452648 CG On-Demand Anodyne ADAM17 61 36 COc1ccc([C@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452661 EI On-Demand Anodyne SDH1 0 43 COc1ccc([C@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452661 EI On-Demand Anodyne MMP13 15 40 COc1ccc([C@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452661 EI On-Demand Anodyne ACACB 26 42 COc1ccc([C@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452661 EI On-Demand Anodyne MMP9 23 40 COc1ccc([C@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452661 EI On-Demand Anodyne MMP1 21 40 COc1ccc([C@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452661 EI On-Demand Anodyne DXR 23 42 CCCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147452669 BE For-Sale Anodyne NOS1 0 45 CCCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147452669 BE For-Sale Anodyne S1PR2 20 48 CCCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147452669 BE For-Sale Anodyne NOS3 15 43 CCCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147452669 BE For-Sale Anodyne DNPEP 0 44 CCCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147452669 BE For-Sale Anodyne DPP7 19 49 CCCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147452669 BE For-Sale Anodyne DPP8 0 47 CCCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147452669 BE For-Sale Anodyne DPP9 0 47 CCCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147452669 BE For-Sale Anodyne SIRT1 24 42 CCCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147452669 BE For-Sale Anodyne METAP2 0 43 CCCC[C@@H](N)C(=O)NCCCCC(C)C ZINC000147452669 BE For-Sale Anodyne NOD1 87 52 Cn1cc(Cl)cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147452680 GF On-Demand Anodyne DRD2 16 40 Cn1cc(Cl)cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147452680 GF On-Demand Anodyne HTR4 61 36 Cn1cc(Cl)cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147452680 GF On-Demand Anodyne APP 47 39 Cn1cc(Cl)cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147452680 GF On-Demand Anodyne SLC6A9 51 39 Cn1cc(Cl)cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147452680 GF On-Demand Anodyne EPHX2 31 41 Cn1cc(Cl)cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147452680 GF On-Demand Anodyne TGM2 61 42 Cn1cc(Cl)cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147452680 GF On-Demand Anodyne CACNA1I 78 42 Cn1cc(Cl)cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147452680 GF On-Demand Anodyne F13A1 57 42 Cn1cc(Cl)cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147452680 GF On-Demand Anodyne AKR1C3 44 35 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C)cc1OCC(F)(F)F)C2 ZINC000147452797 GI On-Demand Anodyne ROCK2 43 51 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)ccc1F ZINC000147452809 DH On-Demand Anodyne RARA 29 43 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)ccc1F ZINC000147452809 DH On-Demand Anodyne CPT1A 80 44 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)ccc1F ZINC000147452809 DH On-Demand Anodyne CPT2 48 38 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)ccc1F ZINC000147452809 DH On-Demand Anodyne PRNP 21 42 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)ccc1F ZINC000147452809 DH On-Demand Anodyne NR1H4 19 42 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)ccc1F ZINC000147452809 DH On-Demand Anodyne FABH 0 40 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)ccc1F ZINC000147452809 DH On-Demand Anodyne TAAR1 34 43 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)ccc1F ZINC000147452809 DH On-Demand Anodyne KCNK3 77 45 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)ccc1F ZINC000147452809 DH On-Demand Anodyne KCNK9 39 43 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)ccc1F ZINC000147452809 DH On-Demand Anodyne TMPRSS4 0 44 COc1ccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452862 EI On-Demand Anodyne SDH1 0 43 COc1ccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452862 EI On-Demand Anodyne MMP13 15 40 COc1ccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452862 EI On-Demand Anodyne ACACB 26 42 COc1ccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452862 EI On-Demand Anodyne MMP9 23 40 COc1ccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452862 EI On-Demand Anodyne MMP1 21 40 COc1ccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147452862 EI On-Demand Anodyne DXR 23 42 Cc1ccc(C(=O)Nc2ccncc2Br)cc1N ZINC000147452871 DF For-Sale Anodyne KIT 15 43 Cc1ccc(C(=O)Nc2ccncc2Br)cc1N ZINC000147452871 DF For-Sale Anodyne HDAC1 29 42 Cc1ccc(C(=O)Nc2ccncc2Br)cc1N ZINC000147452871 DF For-Sale Anodyne SIRT2 22 45 CC(C)CCO[C@@H](C)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147452874 EH On-Demand Anodyne GRIN2B 21 42 CC(C)CCO[C@@H](C)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147452874 EH On-Demand Anodyne TRPV1 15 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccnc(Cl)c1 ZINC000147452981 GF On-Demand Anodyne HTR4 43 36 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccnc(Cl)c1 ZINC000147452981 GF On-Demand Anodyne F10 17 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccnc(Cl)c1 ZINC000147452981 GF On-Demand Anodyne EPHX2 24 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccnc(Cl)c1 ZINC000147452981 GF On-Demand Anodyne TGM2 63 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccnc(Cl)c1 ZINC000147452981 GF On-Demand Anodyne CACNA1I 71 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccnc(Cl)c1 ZINC000147452981 GF On-Demand Anodyne F13A1 55 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccnc(Cl)c1 ZINC000147452981 GF On-Demand Anodyne AKR1C3 47 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccnc(Cl)c1 ZINC000147452981 GF On-Demand Anodyne NAMPT 59 42 CCOC(=O)c1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)cc1 ZINC000147452992 GE On-Demand Anodyne CHRM3 18 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc([N+](=O)[O-])s2)c1 ZINC000147453028 EG On-Demand Bother USP47 42 35 CC(C)CCO[C@H](C)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147453072 EH On-Demand Anodyne GRIN2B 21 42 CC(C)CCO[C@H](C)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147453072 EH On-Demand Anodyne TRPV1 15 43 COc1cccc([C@H](C)NC(=O)c2cc(C)ccc2Br)c1 ZINC000147453091 EI On-Demand Anodyne MTNR1A 22 41 COc1cccc([C@H](C)NC(=O)c2cc(C)ccc2Br)c1 ZINC000147453091 EI On-Demand Anodyne MTNR1B 26 41 COc1cccc([C@H](C)NC(=O)c2cc(C)ccc2Br)c1 ZINC000147453091 EI On-Demand Anodyne KCNK3 26 40 C=CCOc1ccc(Cl)cc1O ZINC000147453145 AF For-Sale Mild FABI 16 50 C=CCOc1ccc(Cl)cc1O ZINC000147453145 AF For-Sale Mild S1PR4 0 40 C=CCOc1ccc(Cl)cc1O ZINC000147453145 AF For-Sale Mild CBR1 16 50 CS(=O)(=O)c1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147453195 FF For-Sale Reactive PREP 32 40 CCOC(=O)c1ccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)cc1 ZINC000147453204 GE On-Demand Anodyne CHRM3 18 41 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne F2 23 40 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne FKBP1A 37 43 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne DRD4 42 34 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne ACHE 20 41 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne GRIN2B 41 38 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne SIGMAR1 21 47 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne MMP13 69 42 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne CCR3 29 40 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne ADAM17 28 42 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne MTNR1A 69 43 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne MTNR1B 70 43 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne MMP2 32 42 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne MMP3 61 42 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne MMP8 30 42 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne CAPN1 17 40 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne MMP9 45 42 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne EPHX2 19 40 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne TGM2 71 44 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne ST14 44 35 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne MMP7 53 42 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne MMP1 54 42 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne F13A1 74 44 COc1cccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147453244 HF On-Demand Anodyne AKR1C3 31 47 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)ccc2F)c1 ZINC000147453250 DH On-Demand Anodyne ATF1 57 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)ccc2F)c1 ZINC000147453250 DH On-Demand Anodyne NFKB1 53 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)ccc2F)c1 ZINC000147453250 DH On-Demand Anodyne KCNK3 45 38 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)ccc2F)c1 ZINC000147453250 DH On-Demand Anodyne TMPRSS4 0 45 O=C(NC[C@@H]1CCCCO1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147453298 DF On-Demand Anodyne CACNA1I 55 37 COc1cccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)c1 ZINC000147453325 EI On-Demand Anodyne MTNR1A 22 41 COc1cccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)c1 ZINC000147453325 EI On-Demand Anodyne MTNR1B 26 41 COc1cccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)c1 ZINC000147453325 EI On-Demand Anodyne KCNK3 26 40 Cc1cc(NC(=O)C2(N)CCC2)c2ccccc2n1 ZINC000147453331 CE For-Sale Anodyne ADAM17 86 41 CS(=O)(=O)c1cccc(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147453374 FF For-Sale Reactive PREP 32 40 Nc1cc(C(=O)Nc2ccncc2Br)ccc1F ZINC000147453385 DF For-Sale Anodyne ROCK2 39 42 Nc1cc(C(=O)Nc2ccncc2Br)ccc1F ZINC000147453385 DF For-Sale Anodyne HDAC1 35 43 Cc1c(O)cccc1C(=O)N1CC[C@H](C(=O)O)C1 ZINC000147453428 BD For-Sale Anodyne SLC6A1 95 38 Cc1c(O)cccc1C(=O)N1CC[C@H](C(=O)O)C1 ZINC000147453428 BD For-Sale Anodyne L3MBTL1 0 41 Cc1c(O)cccc1C(=O)N1CC[C@H](C(=O)O)C1 ZINC000147453428 BD For-Sale Anodyne L3MBTL3 49 36 Cc1c(O)cccc1C(=O)N1CC[C@H](C(=O)O)C1 ZINC000147453428 BD For-Sale Anodyne TP53BP1 0 41 COC(=O)c1ccc(N2CCN(CC(N)=S)CC2)nc1C ZINC000147453440 DC For-Sale Anodyne SLC27A1 58 35 O=C(Cc1cccc(Cl)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147453478 DH On-Demand Anodyne PPIA 20 48 O=C(Cc1cccc(Cl)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147453478 DH On-Demand Anodyne PTGER1 32 47 O=C(Cc1cccc(Cl)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147453478 DH On-Demand Anodyne KCNQ2 23 49 O=C(Cc1cccc(Cl)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147453478 DH On-Demand Anodyne CSNK1D 20 46 O=C(Cc1cccc(Cl)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147453478 DH On-Demand Anodyne UL80 17 42 O=C(Cc1cccc(Cl)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147453478 DH On-Demand Anodyne AKR1C3 35 52 O=C(Cc1cccc(Cl)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147453478 DH On-Demand Anodyne PFK 0 46 O=C(NC[C@H]1CCCCO1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147453516 DF On-Demand Anodyne CACNA1I 55 37 Cc1cc(NC(=O)CC2(CN)CCC2)c2ccccc2n1 ZINC000147453554 CG For-Sale Anodyne ADAM17 77 48 COc1cc(C(=O)NCc2ccccc2Br)ccc1F ZINC000147453597 EH On-Demand Anodyne DRD3 17 44 COc1cc(C(=O)NCc2ccccc2Br)ccc1F ZINC000147453597 EH On-Demand Anodyne PPARA 19 44 COc1cc(C(=O)NCc2ccccc2Br)ccc1F ZINC000147453597 EH On-Demand Anodyne CPT1A 43 30 COc1cc(C(=O)NCc2ccccc2Br)ccc1F ZINC000147453597 EH On-Demand Anodyne PPARD 24 44 COc1cc(C(=O)NCc2ccccc2Br)ccc1F ZINC000147453597 EH On-Demand Anodyne MT-ND1 15 41 COc1cc(C(=O)NCc2ccccc2Br)ccc1F ZINC000147453597 EH On-Demand Anodyne TAAR1 17 44 COc1cc(C(=O)NCc2ccccc2Br)ccc1F ZINC000147453597 EH On-Demand Anodyne GLMU 0 43 Nc1cc(Cl)ccc1C(=O)Nc1ccncc1Br ZINC000147453600 EG For-Sale Anodyne F10 31 40 Nc1cc(Cl)ccc1C(=O)Nc1ccncc1Br ZINC000147453600 EG For-Sale Anodyne KCNMA1 23 40 Cc1c(O)cccc1C(=O)N1CC[C@@H](C(=O)O)C1 ZINC000147453645 BD For-Sale Anodyne SLC6A1 95 38 Cc1c(O)cccc1C(=O)N1CC[C@@H](C(=O)O)C1 ZINC000147453645 BD For-Sale Anodyne L3MBTL1 0 41 Cc1c(O)cccc1C(=O)N1CC[C@@H](C(=O)O)C1 ZINC000147453645 BD For-Sale Anodyne L3MBTL3 49 36 Cc1c(O)cccc1C(=O)N1CC[C@@H](C(=O)O)C1 ZINC000147453645 BD For-Sale Anodyne TP53BP1 0 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2Cl)c1 ZINC000147453647 EI On-Demand Anodyne PPIA 17 47 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2Cl)c1 ZINC000147453647 EI On-Demand Anodyne ATF1 60 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2Cl)c1 ZINC000147453647 EI On-Demand Anodyne NR1H4 16 44 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2Cl)c1 ZINC000147453647 EI On-Demand Anodyne NFKB1 55 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2Cl)c1 ZINC000147453647 EI On-Demand Anodyne ACPS 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2Cl)c1 ZINC000147453647 EI On-Demand Anodyne AKR1C3 37 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2Cl)c1 ZINC000147453647 EI On-Demand Anodyne SMO 23 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2Cl)c1 ZINC000147453647 EI On-Demand Anodyne KCNK3 97 44 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2Cl)c1 ZINC000147453647 EI On-Demand Anodyne KCNK9 72 37 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2Cl)c1 ZINC000147453647 EI On-Demand Anodyne TMPRSS4 0 43 COc1ccc(NC(=O)Nc2nccs2)c(C)c1 ZINC000147453665 CG On-Demand Anodyne MAP 0 57 COc1ccc(NC(=O)Nc2nccs2)c(C)c1 ZINC000147453665 CG On-Demand Anodyne MAP1 127 43 COc1ccc(NC(=O)Nc2nccs2)c(C)c1 ZINC000147453665 CG On-Demand Anodyne KDR 22 43 COc1ccc(NC(=O)Nc2nccs2)c(C)c1 ZINC000147453665 CG On-Demand Anodyne PDGFRA 43 38 CC(C)(C)OC(=O)N1CC[C@H](Nc2ncc(Cl)cc2[N+](=O)[O-])C1 ZINC000147453708 EG On-Demand Bother GPR119 37 43 COc1ccc(NC(=O)C(=O)N2CC=C(c3c(C)[nH]c4ccccc34)CC2)cc1OC ZINC000147453713 HH On-Demand Anodyne ENPP1 69 35 O=C(O)[C@]1(O)C[C@H](O)[C@@H](CO)O1 ZINC000147453737 AA For-Sale Anodyne AROB 48 31 COc1cccc(/C=C\C(=O)N2CCC[C@@H]2CN2CCCC2)c1 ZINC000147453746 DF On-Demand Anodyne UTS2R 46 33 CC(C)CCCCNC(=O)CCCCCN ZINC000147453780 BE For-Sale Anodyne NMT1 39 54 CC(C)CCCCNC(=O)CCCCCN ZINC000147453780 BE For-Sale Anodyne GRIA1 55 38 CC(C)CCCCNC(=O)CCCCCN ZINC000147453780 BE For-Sale Anodyne EPHX2 0 42 CC(C)CCCCNC(=O)CCCCCN ZINC000147453780 BE For-Sale Anodyne DHPS 23 40 CC(C)CCCCNC(=O)CCCCCN ZINC000147453780 BE For-Sale Anodyne POLG_WNV 56 32 CC(C)CCCCNC(=O)CCCCCN ZINC000147453780 BE For-Sale Anodyne DHS 0 40 CC(C)CCCCNC(=O)CCCCCN ZINC000147453780 BE For-Sale Anodyne NOD1 64 48 CC(C)CCCCNC(=O)CCCCCN ZINC000147453780 BE For-Sale Anodyne APHA 0 45 N#Cc1ccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147453796 HF On-Demand Mild ADAM17 16 40 N#Cc1ccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147453796 HF On-Demand Mild ITGA4 18 43 N#Cc1ccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147453796 HF On-Demand Mild TGM2 67 44 N#Cc1ccc(CCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147453796 HF On-Demand Mild F13A1 65 44 Nc1ccc(F)c(C(=O)Nc2ccncc2Br)c1 ZINC000147453836 DF For-Sale Anodyne ROCK2 27 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2Cl)c1 ZINC000147453889 GJ On-Demand Anodyne AVPR2 15 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2Cl)c1 ZINC000147453889 GJ On-Demand Anodyne PPIA 15 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2Cl)c1 ZINC000147453889 GJ On-Demand Anodyne ATF1 40 38 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2Cl)c1 ZINC000147453889 GJ On-Demand Anodyne PYGL 19 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2Cl)c1 ZINC000147453889 GJ On-Demand Anodyne SMO 23 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2Cl)c1 ZINC000147453889 GJ On-Demand Anodyne GPR35 39 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2Cl)c1 ZINC000147453889 GJ On-Demand Anodyne KCNK3 19 42 Cc1ccc(Br)c(C(=O)NCc2ccc(F)cc2F)c1 ZINC000147453904 EH On-Demand Anodyne P2RX7 60 48 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000147453913 HG On-Demand Anodyne P2RY1 58 41 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000147453913 HG On-Demand Anodyne CTSS 26 42 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000147453913 HG On-Demand Anodyne EPHX2 65 46 CC(C)(C)OC(=O)N1CC[C@@H](Nc2ncc(Cl)cc2[N+](=O)[O-])C1 ZINC000147453924 EG On-Demand Bother GPR119 37 43 CCOC(=O)c1ccc([N+](=O)[O-])cc1C#N ZINC000147453940 BD In-Stock Mild CACNA1C 62 47 CCOC(=O)c1ccc([N+](=O)[O-])cc1C#N ZINC000147453940 BD In-Stock Mild CACNA1D 93 47 CCOC(=O)c1ccc([N+](=O)[O-])cc1C#N ZINC000147453940 BD In-Stock Mild CCR3 0 41 CCOC(=O)c1ccc([N+](=O)[O-])cc1C#N ZINC000147453940 BD In-Stock Mild CTRB1 31 47 CCOC(=O)c1ccc([N+](=O)[O-])cc1C#N ZINC000147453940 BD In-Stock Mild SLC27A4 45 33 COc1cccc(/C=C\C(=O)N2CCC[C@H]2CN2CCCC2)c1 ZINC000147453977 DF On-Demand Anodyne UTS2R 46 33 CC[C@H](NC(=O)NCc1sccc1Br)C(=O)O ZINC000147453989 DE On-Demand Anodyne ANPEP 26 41 COc1cc(CNCCCCC(C)C)cc([N+](=O)[O-])c1 ZINC000147454018 CH For-Sale Bother LEF 41 39 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1C ZINC000147454091 GE On-Demand Anodyne HTR4 60 37 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1C ZINC000147454091 GE On-Demand Anodyne EPHX2 26 40 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1C ZINC000147454091 GE On-Demand Anodyne TGM2 69 46 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1C ZINC000147454091 GE On-Demand Anodyne CACNA1I 64 36 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)n1C ZINC000147454091 GE On-Demand Anodyne F13A1 70 46 COc1ccc(OC)c(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147454096 FG For-Sale Reactive FKBP1A 19 40 COc1ccc(OC)c(C(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147454096 FG For-Sale Reactive ACKR3 63 34 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000147454105 HG On-Demand Anodyne P2RY1 58 41 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000147454105 HG On-Demand Anodyne CTSS 26 42 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(OC(F)(F)F)cc2)C1 ZINC000147454105 HG On-Demand Anodyne EPHX2 65 46 O=C(O)c1cc(Cl)cc(NC(=O)C2CC2)c1 ZINC000147454109 BE On-Demand Anodyne CACNA1I 54 37 O=C(O)c1cc(Cl)cc(NC(=O)C2CC2)c1 ZINC000147454109 BE On-Demand Anodyne HCAR1 0 44 Cc1[nH]c2ccccc2c1C1=CCN(C(=O)C(=O)Nc2cccc3cnccc23)CC1 ZINC000147454140 HI On-Demand Anodyne TRPV1 45 39 COC(=O)c1ccc(N2CCC[C@H](C(C)=O)C2)nc1C ZINC000147454149 CD On-Demand Anodyne GPBAR1 25 40 CCCCCCCOc1c(F)cc(/C=C/C(=O)O)cc1F ZINC000147454177 CI For-Sale Mild LTB4R 24 42 CCCCCCCOc1c(F)cc(/C=C/C(=O)O)cc1F ZINC000147454177 CI For-Sale Mild PLA2G4B 84 35 CCCCCCCOc1c(F)cc(/C=C/C(=O)O)cc1F ZINC000147454177 CI For-Sale Mild AKR1C3 25 41 CCCCCCCOc1c(F)cc(/C=C/C(=O)O)cc1F ZINC000147454177 CI For-Sale Mild NFE2L2 0 41 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147454208 HG On-Demand Anodyne PLG 17 43 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147454208 HG On-Demand Anodyne CNR2 17 43 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147454208 HG On-Demand Anodyne MAPK14 45 40 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147454208 HG On-Demand Anodyne MAPK13 46 34 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147454208 HG On-Demand Anodyne PLAU 30 48 Cc1cc(C(=O)NC2CCCCC2)ccc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147454208 HG On-Demand Anodyne ST14 24 48 C[C@H](CNc1nccn(C2CC2)c1=O)CC(=O)O ZINC000147454215 CD On-Demand Anodyne CASP3 76 38 C[C@H](CNc1nccn(C2CC2)c1=O)CC(=O)O ZINC000147454215 CD On-Demand Anodyne CASP8 57 38 C[C@H](CNc1nccn(C2CC2)c1=O)CC(=O)O ZINC000147454215 CD On-Demand Anodyne CASP1 49 32 C[C@H](CNc1nccn(C2CC2)c1=O)CC(=O)O ZINC000147454215 CD On-Demand Anodyne CASP7 59 38 Nc1ccc2[nH]c(C(=O)Nc3ccncc3Br)cc2c1 ZINC000147454270 EG For-Sale Anodyne PYGL 47 37 CN1N=C(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCC1=O ZINC000147454284 GC On-Demand Anodyne HTR4 57 39 CN1N=C(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCC1=O ZINC000147454284 GC On-Demand Anodyne EPHX2 18 40 CN1N=C(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCC1=O ZINC000147454284 GC On-Demand Anodyne TGM2 55 42 CN1N=C(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCC1=O ZINC000147454284 GC On-Demand Anodyne CACNA1I 60 38 CN1N=C(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCC1=O ZINC000147454284 GC On-Demand Anodyne F13A1 43 42 COCCn1cc(C(=O)[C@H](C#N)c2nc(C)cs2)c2ccccc21 ZINC000147454305 EH On-Demand Mild CNR1 25 48 COCCn1cc(C(=O)[C@H](C#N)c2nc(C)cs2)c2ccccc21 ZINC000147454305 EH On-Demand Mild CNR2 20 48 COC(=O)c1cccc(OCC(F)(F)F)c1[N+](=O)[O-] ZINC000147454310 CE Annotated Bother CACNA1C 21 42 COC(=O)c1cccc(OCC(F)(F)F)c1[N+](=O)[O-] ZINC000147454310 CE Annotated Bother CACNA1D 37 42 COc1ccc(OC)c(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147454319 FG For-Sale Reactive FKBP1A 19 40 COc1ccc(OC)c(C(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147454319 FG For-Sale Reactive ACKR3 63 34 O=C(CCCc1cccs1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147454337 DI On-Demand Anodyne PTPRF 22 50 C[C@H](NC(=O)c1ccc(Br)c(Cl)c1)c1ccc(C#N)cc1 ZINC000147454348 FI On-Demand Mild PTGER4 22 43 C[C@H](NC(=O)c1ccc(Br)c(Cl)c1)c1ccc(C#N)cc1 ZINC000147454348 FI On-Demand Mild CTSG 17 41 C[C@H](NC(=O)c1ccc(Br)c(Cl)c1)c1ccc(C#N)cc1 ZINC000147454348 FI On-Demand Mild CTRB_BOVIN 46 34 COC(=O)c1ccc(N2CCC[C@@H](C(C)=O)C2)nc1C ZINC000147454382 CD On-Demand Anodyne GPBAR1 25 40 CC[C@@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454422 CF On-Demand Anodyne KCNH2 0 45 CC[C@@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454422 CF On-Demand Anodyne LTA4H 54 51 CC[C@@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454422 CF On-Demand Anodyne HRH3 78 42 CC[C@@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454422 CF On-Demand Anodyne SIGMAR1 33 46 CC[C@@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454422 CF On-Demand Anodyne NPY1R 41 35 CC[C@@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454422 CF On-Demand Anodyne HTR5A 24 42 CC[C@@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454422 CF On-Demand Anodyne CHRNA10 41 40 CC[C@@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454422 CF On-Demand Anodyne GRIN3A 0 42 CC[C@@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454422 CF On-Demand Anodyne PSMB2 49 41 CC[C@@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454422 CF On-Demand Anodyne PSMB1 42 41 CC[C@@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454422 CF On-Demand Anodyne MEN1 53 42 C[C@@H](CNc1nccn(C2CC2)c1=O)CC(=O)O ZINC000147454443 CD On-Demand Anodyne CASP3 76 38 C[C@@H](CNc1nccn(C2CC2)c1=O)CC(=O)O ZINC000147454443 CD On-Demand Anodyne CASP8 57 38 C[C@@H](CNc1nccn(C2CC2)c1=O)CC(=O)O ZINC000147454443 CD On-Demand Anodyne CASP1 49 32 C[C@@H](CNc1nccn(C2CC2)c1=O)CC(=O)O ZINC000147454443 CD On-Demand Anodyne CASP7 59 38 NC1(C(=O)Nc2ccccc2SC(F)F)CCC1 ZINC000147454456 CF For-Sale Anodyne CETP 25 50 COc1csc2ccc([N+](=O)[O-])cc12 ZINC000147454487 BF For-Sale Bother SNCA 39 40 COCCn1cc(C(=O)[C@@H](C#N)c2nc(C)cs2)c2ccccc21 ZINC000147454524 EH On-Demand Mild CNR1 25 48 COCCn1cc(C(=O)[C@@H](C#N)c2nc(C)cs2)c2ccccc21 ZINC000147454524 EH On-Demand Mild CNR2 20 48 C[C@@H](NC(=O)c1ccc(Br)c(Cl)c1)c1ccc(C#N)cc1 ZINC000147454530 FI On-Demand Mild PTGER4 19 43 C[C@@H](NC(=O)c1ccc(Br)c(Cl)c1)c1ccc(C#N)cc1 ZINC000147454530 FI On-Demand Mild CTRB_BOVIN 46 34 Cc1[nH]c2ccccc2c1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147454531 HG On-Demand Anodyne HTR4 73 44 Cc1[nH]c2ccccc2c1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147454531 HG On-Demand Anodyne EPHX2 17 40 Cc1[nH]c2ccccc2c1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147454531 HG On-Demand Anodyne TGM2 54 42 Cc1[nH]c2ccccc2c1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147454531 HG On-Demand Anodyne CACNA1I 52 33 Cc1[nH]c2ccccc2c1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147454531 HG On-Demand Anodyne F13A1 47 42 Cc1nc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)s1 ZINC000147454555 DG On-Demand Anodyne JUN 15 43 C=CC(=O)OCCCOc1ccc(O)cc1 ZINC000147454570 BD For-Sale Anodyne ALDH2 47 35 C=CC(=O)OCCCOc1ccc(O)cc1 ZINC000147454570 BD For-Sale Anodyne PLA2G4B 43 31 C=CC(=O)OCCCOc1ccc(O)cc1 ZINC000147454570 BD For-Sale Anodyne ESRRG 42 30 C=CC(=O)OCCCOc1ccc(O)cc1 ZINC000147454570 BD For-Sale Anodyne AKR1B10 34 40 CC[C@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454652 CF On-Demand Anodyne KCNH2 0 45 CC[C@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454652 CF On-Demand Anodyne LTA4H 54 51 CC[C@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454652 CF On-Demand Anodyne HRH3 78 42 CC[C@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454652 CF On-Demand Anodyne SIGMAR1 33 46 CC[C@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454652 CF On-Demand Anodyne NPY1R 41 35 CC[C@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454652 CF On-Demand Anodyne HTR5A 24 42 CC[C@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454652 CF On-Demand Anodyne CHRNA10 41 40 CC[C@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454652 CF On-Demand Anodyne GRIN3A 0 42 CC[C@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454652 CF On-Demand Anodyne PSMB2 49 41 CC[C@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454652 CF On-Demand Anodyne PSMB1 42 41 CC[C@H]1CN(CCCOc2ccccc2)CC[C@@H]1N ZINC000147454652 CF On-Demand Anodyne MEN1 53 42 CC(C)Cn1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147454685 CD For-Sale Anodyne CASP3 74 35 CC(C)Cn1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147454685 CD For-Sale Anodyne CASP8 52 35 CC(C)Cn1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147454685 CD For-Sale Anodyne CASP1 42 35 CC(C)Cn1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147454685 CD For-Sale Anodyne CASP7 46 35 NCC1(CC(=O)Nc2ccccc2SC(F)F)CCC1 ZINC000147454695 DG For-Sale Anodyne CETP 0 40 Cc1ccc(Br)c(C(=O)N[C@@H](C)c2ccc(C#N)cc2)c1 ZINC000147454717 EI On-Demand Mild SDH1 0 43 CCCCCCCCOc1ccc(CNC(C)(C)C)nc1 ZINC000147454720 CJ For-Sale Mild KCNQ1 0 41 CCCCCCCCOc1ccc(CNC(C)(C)C)nc1 ZINC000147454720 CJ For-Sale Mild PLA2G4B 73 40 NS(=O)(=O)c1cc(Br)c(OCc2ccncc2Cl)cc1F ZINC000147454742 GF For-Sale Anodyne CA14 21 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(Cl)c[nH]1 ZINC000147454746 GE On-Demand Anodyne HTR4 48 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(Cl)c[nH]1 ZINC000147454746 GE On-Demand Anodyne TGM2 56 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(Cl)c[nH]1 ZINC000147454746 GE On-Demand Anodyne CACNA1I 54 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(Cl)c[nH]1 ZINC000147454746 GE On-Demand Anodyne F13A1 51 43 CC(C)CCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147454777 CG On-Demand Anodyne CCKBR 65 42 CC(C)CCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147454777 CG On-Demand Anodyne CACNA1I 41 32 CC(C)CCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147454777 CG On-Demand Anodyne HCAR1 0 41 COc1cc(NCC(=O)Nc2cccc(C)c2)ccc1Br ZINC000147454783 EH On-Demand Anodyne KIT 20 43 COc1cc(NCC(=O)Nc2cccc(C)c2)ccc1Br ZINC000147454783 EH On-Demand Anodyne CCKAR 0 40 COc1cc(NCC(=O)Nc2cccc(C)c2)ccc1Br ZINC000147454783 EH On-Demand Anodyne KDR 23 43 COc1cc(NCC(=O)Nc2cccc(C)c2)ccc1Br ZINC000147454783 EH On-Demand Anodyne FLT3 16 42 COc1cc(NCC(=O)Nc2cccc(C)c2)ccc1Br ZINC000147454783 EH On-Demand Anodyne IMPDH2 0 54 COc1cc(NCC(=O)Nc2cccc(C)c2)ccc1Br ZINC000147454783 EH On-Demand Anodyne ENPP1 78 38 COc1cc(NCC(=O)Nc2cccc(C)c2)ccc1Br ZINC000147454783 EH On-Demand Anodyne PSBA 0 43 COc1cc(NCC(=O)Nc2cccc(C)c2)ccc1Br ZINC000147454783 EH On-Demand Anodyne KCNK3 81 44 COc1cc(NCC(=O)Nc2cccc(C)c2)ccc1Br ZINC000147454783 EH On-Demand Anodyne KCNK9 72 44 CCNCCC(=O)NCCCCC(C)C ZINC000147454811 BD For-Sale Anodyne NOD1 24 40 Cc1nc(N2CC(C(=O)O)C2)c(C#N)cc1C(=O)OC(C)C ZINC000147454872 DD For-Sale Anodyne NR3C2 42 32 Cc1nc(N2CC(C(=O)O)C2)c(C#N)cc1C(=O)OC(C)C ZINC000147454872 DD For-Sale Anodyne P2RY12 41 55 CC(C)Cn1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147454886 CD For-Sale Anodyne CASP3 74 35 CC(C)Cn1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147454886 CD For-Sale Anodyne CASP8 52 35 CC(C)Cn1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147454886 CD For-Sale Anodyne CASP1 42 35 CC(C)Cn1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147454886 CD For-Sale Anodyne CASP7 46 35 C=CCCOCC(=O)Nc1ccc(C(=O)NC2CCCCC2)cc1C ZINC000147454896 EH On-Demand Mild PLAU 16 40 Cc1cncn1CCCN/C(=C\[N+](=O)[O-])Nc1ccc2c(c1)OCO2 ZINC000147454911 EE Annotated Anodyne QPCT 109 90 Cc1cncn1CCCN/C(=C\[N+](=O)[O-])Nc1ccc2c(c1)OCO2 ZINC000147454911 EE Annotated Anodyne DYRK2 46 35 Cc1ccc(Br)c(C(=O)N[C@H](C)c2ccc(C#N)cc2)c1 ZINC000147454928 EI On-Demand Mild SDH1 0 43 NC1(C(=O)NCc2cccc(C(F)(F)F)c2)CCC1 ZINC000147454938 CE On-Demand Anodyne TACR1 26 47 NC1(C(=O)NCc2cccc(C(F)(F)F)c2)CCC1 ZINC000147454938 CE On-Demand Anodyne PHES 0 40 NC1(C(=O)NCc2cccc(C(F)(F)F)c2)CCC1 ZINC000147454938 CE On-Demand Anodyne CCL2 0 44 NC1(C(=O)NCc2cccc(C(F)(F)F)c2)CCC1 ZINC000147454938 CE On-Demand Anodyne PDS 45 45 CC(C)(C)c1cc(NC(=O)[C@@H]2C[C@H](O)CN2CC2CCOCC2)on1 ZINC000147454961 FD Annotated Anodyne CNR2 16 51 C=C(CCl)c1ccc(O)cc1 ZINC000147454962 AF For-Sale Reactive ESR1 16 41 COc1cc(NCC(=O)Nc2cccc(Cl)c2)ccc1Br ZINC000147454968 FI On-Demand Anodyne HTR2A 22 50 COc1cc(NCC(=O)Nc2cccc(Cl)c2)ccc1Br ZINC000147454968 FI On-Demand Anodyne CPT1A 45 31 COc1cc(NCC(=O)Nc2cccc(Cl)c2)ccc1Br ZINC000147454968 FI On-Demand Anodyne KDR 15 41 COc1cc(NCC(=O)Nc2cccc(Cl)c2)ccc1Br ZINC000147454968 FI On-Demand Anodyne IMPDH2 0 44 COc1cc(NCC(=O)Nc2cccc(Cl)c2)ccc1Br ZINC000147454968 FI On-Demand Anodyne ENPP1 76 39 COc1cc(NCC(=O)Nc2cccc(Cl)c2)ccc1Br ZINC000147454968 FI On-Demand Anodyne PSBA 0 42 COc1cc(NCC(=O)Nc2cccc(Cl)c2)ccc1Br ZINC000147454968 FI On-Demand Anodyne KCNK3 46 38 COc1cc(NCC(=O)Nc2cccc(Cl)c2)ccc1Br ZINC000147454968 FI On-Demand Anodyne KCNK9 43 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnc2ccccc2n1 ZINC000147454995 HE On-Demand Anodyne HTR4 46 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnc2ccccc2n1 ZINC000147454995 HE On-Demand Anodyne GRIN2B 29 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnc2ccccc2n1 ZINC000147454995 HE On-Demand Anodyne CCR1 41 39 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnc2ccccc2n1 ZINC000147454995 HE On-Demand Anodyne GRM1 15 49 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnc2ccccc2n1 ZINC000147454995 HE On-Demand Anodyne EPHX2 15 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnc2ccccc2n1 ZINC000147454995 HE On-Demand Anodyne TGM2 63 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnc2ccccc2n1 ZINC000147454995 HE On-Demand Anodyne CACNA1I 52 33 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnc2ccccc2n1 ZINC000147454995 HE On-Demand Anodyne F13A1 57 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnc2ccccc2n1 ZINC000147454995 HE On-Demand Anodyne NAMPT 52 41 O=C1c2ccc(Cl)cc2C(=O)c2cc3ccccc3cc21 ZINC000147455069 CI For-Sale Clean ALDH1A1 17 40 O=C1c2ccc(Cl)cc2C(=O)c2cc3ccccc3cc21 ZINC000147455069 CI For-Sale Clean USP7 24 45 NC[C@@]1(NCC(F)F)CCCN(Cc2ccccc2)C1 ZINC000147455080 CD For-Sale Anodyne NPFFR1 48 48 C[C@H](CNc1cc(C#N)c2ccccc2n1)CC(=O)O ZINC000147455104 CF For-Sale Mild METG 81 42 NCC1(CC(=O)NCc2cccc(C(F)(F)F)c2)CCC1 ZINC000147455131 DF For-Sale Anodyne TACR1 26 42 NCC1(CC(=O)NCc2cccc(C(F)(F)F)c2)CCC1 ZINC000147455131 DF For-Sale Anodyne CCR2 82 38 NCC1(CC(=O)NCc2cccc(C(F)(F)F)c2)CCC1 ZINC000147455131 DF For-Sale Anodyne PDS 38 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C12CC3CC(CC(C3)C1)C2 ZINC000147455195 HG On-Demand Anodyne HSD11B1 29 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C12CC3CC(CC(C3)C1)C2 ZINC000147455195 HG On-Demand Anodyne EPHX2 42 47 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C12CC3CC(CC(C3)C1)C2 ZINC000147455195 HG On-Demand Anodyne TGM2 82 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C12CC3CC(CC(C3)C1)C2 ZINC000147455195 HG On-Demand Anodyne F13A1 86 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C12CC3CC(CC(C3)C1)C2 ZINC000147455195 HG On-Demand Anodyne NAMPT 39 40 Cc1cc(OC(C)C)nn1-c1ccccn1 ZINC000147455274 BE For-Sale Anodyne SLC11A2 46 33 C[C@@H](CNc1cc(C#N)c2ccccc2n1)CC(=O)O ZINC000147455309 CF For-Sale Mild METG 81 42 NC[C@]1(NCC(F)F)CCCN(Cc2ccccc2)C1 ZINC000147455319 CD For-Sale Anodyne NPFFR1 48 48 NC1(C(=O)Nc2cccc3ncccc23)CCC1 ZINC000147455337 BE For-Sale Anodyne P2RX7 0 52 NC1(C(=O)Nc2cccc3ncccc23)CCC1 ZINC000147455337 BE For-Sale Anodyne G2YM83_BOTF4 51 32 COC(=O)CC(=O)c1cc(Br)ccc1F ZINC000147455353 CE For-Sale Anodyne FAS 22 40 Nc1ccc(-c2nc3ccccc3[nH]2)c(F)c1 ZINC000147455417 BF For-Sale Anodyne PLG 0 40 Nc1ccc(-c2nc3ccccc3[nH]2)c(F)c1 ZINC000147455417 BF For-Sale Anodyne PDGFRB 0 49 Nc1ccc(-c2nc3ccccc3[nH]2)c(F)c1 ZINC000147455417 BF For-Sale Anodyne MAP 0 48 Nc1ccc(-c2nc3ccccc3[nH]2)c(F)c1 ZINC000147455417 BF For-Sale Anodyne PLAUR 44 45 Nc1ccc(-c2nc3ccccc3[nH]2)c(F)c1 ZINC000147455417 BF For-Sale Anodyne FGFR1 0 43 Nc1ccc(-c2nc3ccccc3[nH]2)c(F)c1 ZINC000147455417 BF For-Sale Anodyne FLT1 26 43 Nc1ccc(-c2nc3ccccc3[nH]2)c(F)c1 ZINC000147455417 BF For-Sale Anodyne SHH 19 41 Nc1ccc(-c2nc3ccccc3[nH]2)c(F)c1 ZINC000147455417 BF For-Sale Anodyne SCD1 0 42 Nc1ccc(-c2nc3ccccc3[nH]2)c(F)c1 ZINC000147455417 BF For-Sale Anodyne METAP2 0 48 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne PPIA 18 48 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne JUN 23 45 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne PLA2G7 25 40 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne ATF1 58 40 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne GRM4 55 45 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne NR1H4 16 42 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne GRM5 29 55 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne SORT1 27 49 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne NFKB1 54 40 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne SCN10A 45 39 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne TAAR1 15 42 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne AKR1C3 37 44 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne SHH 47 40 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne KCNK3 109 43 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455441 CF On-Demand Anodyne KCNK9 69 43 COc1cc(NCC(=O)Nc2ccccc2Br)ccc1Br ZINC000147455482 HI On-Demand Anodyne ENPP1 69 34 CC[C@@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455499 CE On-Demand Anodyne TIMP3 62 33 CC[C@@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455499 CE On-Demand Anodyne SLC6A11 0 40 CC[C@@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455499 CE On-Demand Anodyne SLC6A12 0 40 CC[C@@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455499 CE On-Demand Anodyne EPHX2 15 42 CC[C@@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455499 CE On-Demand Anodyne BIRC2 43 34 CC[C@@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455499 CE On-Demand Anodyne METAP2 0 42 O=C(c1cccc(C(F)(F)F)c1)c1cncs1 ZINC000147455521 CG For-Sale Anodyne CCR2 29 42 CCOc1cc(N)cc(C(=O)Nc2ccncc2Br)c1 ZINC000147455557 EG For-Sale Anodyne SIRT2 18 40 NCC1(CC(=O)Nc2cccc3ncccc23)CCC1 ZINC000147455588 CF For-Sale Anodyne P2RX7 19 41 CCNc1nc(Cl)nc(Oc2cc(C)cc(C)c2C)n1 ZINC000147455627 CH For-Sale Anodyne PPX1 0 46 Cc1noc(CCC(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1 ZINC000147455660 DE On-Demand Anodyne HCAR2 38 41 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147455673 GD On-Demand Anodyne HTR4 53 36 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147455673 GD On-Demand Anodyne GRIN2B 30 41 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147455673 GD On-Demand Anodyne EPHX2 21 43 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147455673 GD On-Demand Anodyne TGM2 63 46 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147455673 GD On-Demand Anodyne CACNA1I 64 42 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147455673 GD On-Demand Anodyne F13A1 49 42 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147455673 GD On-Demand Anodyne HPGDS 31 41 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cn1 ZINC000147455673 GD On-Demand Anodyne NAMPT 60 46 O=C(O)CCCCOCc1ccccc1Br ZINC000147455725 CG For-Sale Anodyne FFAR1 28 53 O=C(O)CCCCOCc1ccccc1Br ZINC000147455725 CG For-Sale Anodyne FFAR4 55 38 CC[C@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455734 CE For-Sale Anodyne TIMP3 62 33 CC[C@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455734 CE For-Sale Anodyne SLC6A11 0 40 CC[C@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455734 CE For-Sale Anodyne SLC6A12 0 40 CC[C@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455734 CE For-Sale Anodyne EPHX2 15 42 CC[C@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455734 CE For-Sale Anodyne BIRC2 43 34 CC[C@H]1CN([C@@H](C)C(=O)Nc2ccccc2)CC[C@@H]1N ZINC000147455734 CE For-Sale Anodyne METAP2 0 42 Nc1cccc(CC(=O)Nc2ccncc2Br)c1 ZINC000147455779 DF For-Sale Anodyne CA5B 47 44 Nc1cccc(CC(=O)Nc2ccncc2Br)c1 ZINC000147455779 DF For-Sale Anodyne CA5A 53 44 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne F2 79 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne PLG 31 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne ACE 37 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne OPRM1 22 44 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne OPRD1 17 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne CELA1 46 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne ELANE 48 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne TRHR 67 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne HLA-DRB3 66 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne CTRA_BOVIN 40 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne TRY1_BOVIN 97 38 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne NTSR1 125 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne NTSR2 80 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne HLA-A 42 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne LGMN 80 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne CCKBR 42 39 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne C5AR1 25 44 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne TPP2 45 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne XIAP 50 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne BRCA1 59 31 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455780 HG On-Demand Anodyne TMPRSS11D 60 36 CC(C)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147455830 BF For-Sale Anodyne CETP 0 43 CC(C)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147455830 BF For-Sale Anodyne SOAT1 23 40 CC(C)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147455830 BF For-Sale Anodyne ACAT 0 50 COc1cc(C(=O)NCc2ccc(C#N)cc2)ccc1F ZINC000147455855 CF On-Demand Mild U38 0 45 COC(=O)Cc1csc(-c2ccc(OC)c(Cl)c2)n1 ZINC000147455860 CG For-Sale Anodyne DCK 43 40 COC(=O)Cc1csc(-c2ccc(OC)c(Cl)c2)n1 ZINC000147455860 CG For-Sale Anodyne PDE4D 0 44 COC(=O)Cc1csc(-c2ccc(OC)c(Cl)c2)n1 ZINC000147455860 CG For-Sale Anodyne PPARD 18 40 COC(=O)Cc1csc(-c2ccc(OC)c(Cl)c2)n1 ZINC000147455860 CG For-Sale Anodyne KMO 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc[nH]2)c1 ZINC000147455875 CF On-Demand Anodyne PPIA 15 50 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc[nH]2)c1 ZINC000147455875 CF On-Demand Anodyne PRNP 16 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc[nH]2)c1 ZINC000147455875 CF On-Demand Anodyne AKR1C3 26 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc[nH]2)c1 ZINC000147455875 CF On-Demand Anodyne HCAR1 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc[nH]2)c1 ZINC000147455875 CF On-Demand Anodyne KCNK3 58 44 CC(C)[C@H](OCc1ccccc1Br)C(=O)O ZINC000147455928 CG For-Sale Anodyne SLC1A6 0 43 CC(C)[C@H](OCc1ccccc1Br)C(=O)O ZINC000147455928 CG For-Sale Anodyne SLC1A7 0 43 CC1(C)[C@@H]2CC[C@](CN)(CC(=O)O)[C@H]21 ZINC000147455966 AD For-Sale Anodyne CACNA2D1 77 54 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne F2 79 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne PLG 31 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne ACE 37 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne OPRM1 22 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne CELA1 46 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne ELANE 48 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne TRHR 67 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne HLA-DRB3 66 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne CTRA_BOVIN 40 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne TRY1_BOVIN 97 38 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne NTSR1 125 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne NTSR2 80 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne HLA-A 42 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne LGMN 80 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne C5AR1 15 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne TPP2 45 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne XIAP 50 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne BRCA1 59 31 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147455996 HG On-Demand Anodyne TMPRSS11D 60 36 COc1cc(NCc2ccc(OCC#N)cc2)ccc1Br ZINC000147455998 EH For-Sale Mild DRTS_TRYCR 48 36 Oc1ccc(CNCc2nc3ccccc3[nH]2)nc1 ZINC000147455999 CD For-Sale Anodyne CXCR4 27 40 Oc1ccc(CNCc2nc3ccccc3[nH]2)nc1 ZINC000147455999 CD For-Sale Anodyne FABK 0 42 CC(C)c1ccccc1NC(=O)CC1(CN)CCC1 ZINC000147456055 CG For-Sale Anodyne KCNQ2 46 32 CC(C)c1ccccc1NC(=O)CC1(CN)CCC1 ZINC000147456055 CG For-Sale Anodyne ACAT 0 48 COC(=O)Cc1csc(-c2ccc(C3CC3)cc2)n1 ZINC000147456062 CG For-Sale Anodyne AVPR1B 22 41 COC(=O)Cc1csc(-c2ccc(C3CC3)cc2)n1 ZINC000147456062 CG For-Sale Anodyne DGAT1 18 42 Cc1cc(Cl)cc(C(=O)NCc2ccc(C#N)cc2)c1 ZINC000147456083 CG On-Demand Mild CTSV 26 42 Cc1cc(Cl)cc(C(=O)NCc2ccc(C#N)cc2)c1 ZINC000147456083 CG On-Demand Mild CACNA1I 38 41 Cc1c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cnn1C ZINC000147456126 CE On-Demand Anodyne JUN 23 45 Cc1c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cnn1C ZINC000147456126 CE On-Demand Anodyne ATF1 59 41 Cc1c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cnn1C ZINC000147456126 CE On-Demand Anodyne NFKB1 54 41 CC(C)[C@@H](OCc1ccccc1Br)C(=O)O ZINC000147456150 CG For-Sale Anodyne SLC1A6 0 43 CC(C)[C@@H](OCc1ccccc1Br)C(=O)O ZINC000147456150 CG For-Sale Anodyne SLC1A7 0 43 Cc1ncc([N+](=O)[O-])cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147456162 HE On-Demand Bother EPHX2 21 43 Cc1ncc([N+](=O)[O-])cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147456162 HE On-Demand Bother TGM2 58 40 Cc1ncc([N+](=O)[O-])cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147456162 HE On-Demand Bother CACNA1I 51 33 Cc1ncc([N+](=O)[O-])cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147456162 HE On-Demand Bother F13A1 47 40 Cc1ncc([N+](=O)[O-])cc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147456162 HE On-Demand Bother NAMPT 42 39 CC[C@H](NC(=O)N1CC[C@]2(O)CCCC[C@@H]2C1)C(=O)O ZINC000147456168 CD For-Sale Anodyne CCKBR 40 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne F2 79 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne PLG 31 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne ACE 37 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne OPRM1 22 44 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne OPRD1 17 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne CELA1 46 34 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne ELANE 48 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne TRHR 67 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne HLA-DRB3 66 40 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne CTRA_BOVIN 40 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne TRY1_BOVIN 97 38 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne NTSR1 125 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne NTSR2 80 37 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne HLA-A 42 33 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne LGMN 80 35 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne CCKBR 42 39 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne C5AR1 25 44 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne TPP2 45 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne XIAP 50 41 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne BRCA1 59 31 CCCC[C@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456174 HG On-Demand Anodyne TMPRSS11D 60 36 C[C@H](OC[C@@H]1CCCO1)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147456219 EF On-Demand Anodyne GRIN2B 0 40 C[C@H](OC[C@@H]1CCCO1)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147456219 EF On-Demand Anodyne SCN9A 0 51 COCCCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147456226 DF On-Demand Anodyne CACNA1I 44 34 COc1cc(NCC(=O)NC2CCCCC2)ccc1Br ZINC000147456260 EG On-Demand Anodyne EPHX2 25 44 COc1cc(NCC(=O)NC2CCCCC2)ccc1Br ZINC000147456260 EG On-Demand Anodyne ENPP1 49 30 COc1ccc(CCNC(=O)CC2(CN)CCC2)cc1 ZINC000147456276 CD For-Sale Anodyne MTNR1A 112 40 COc1ccc(CCNC(=O)CC2(CN)CCC2)cc1 ZINC000147456276 CD For-Sale Anodyne MTNR1B 90 40 COc1ccc(CCNC(=O)CC2(CN)CCC2)cc1 ZINC000147456276 CD For-Sale Anodyne CA9 23 52 COc1ccc(CCNC(=O)CC2(CN)CCC2)cc1 ZINC000147456276 CD For-Sale Anodyne PROKR1 41 32 COC(=O)c1ccc(Sc2ccccc2C(=O)O)nc1C ZINC000147456324 DG For-Sale Anodyne ALS 57 39 C[C@H](OCc1ccccc1Br)C(=O)O ZINC000147456368 CE For-Sale Anodyne ANPEP 16 40 C[C@H](OCc1ccccc1Br)C(=O)O ZINC000147456368 CE For-Sale Anodyne THRB 15 41 C[C@H](OCc1ccccc1Br)C(=O)O ZINC000147456368 CE For-Sale Anodyne ACE2 44 34 N#CC1(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCCC1 ZINC000147456387 GE On-Demand Mild CTSK 15 43 N#CC1(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCCC1 ZINC000147456387 GE On-Demand Mild EPHX2 16 45 N#CC1(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCCC1 ZINC000147456387 GE On-Demand Mild TGM2 62 46 N#CC1(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCCC1 ZINC000147456387 GE On-Demand Mild F13A1 61 46 N#CC1(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CCCC1 ZINC000147456387 GE On-Demand Mild NAMPT 39 43 CC[C@H](NC(=O)N1CC[C@@]2(O)CCCC[C@@H]2C1)C(=O)O ZINC000147456394 CD For-Sale Anodyne CCKBR 40 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne F2 79 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne PLG 31 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne ACE 37 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne OPRM1 22 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne CELA1 46 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne ELANE 48 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne TRHR 67 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne HLA-DRB3 66 40 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne CTRA_BOVIN 40 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne TRY1_BOVIN 97 38 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne NTSR1 125 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne NTSR2 80 37 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne HLA-A 42 33 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne LGMN 80 35 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne C5AR1 15 44 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne TPP2 45 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne XIAP 50 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne BRCA1 59 31 CCCC[C@@H](NC(N)=O)C(=O)N1CCC[C@H]1C(=O)Nc1cc(Cl)cc(Cl)c1 ZINC000147456397 HG On-Demand Anodyne TMPRSS11D 60 36 O=S(=O)(c1c(F)cc(F)cc1F)N1CCN(CCBr)CC1 ZINC000147456410 GD For-Sale Reactive PKM 33 49 C[C@@H](CCP(=O)(O)O)CC(C)(C)C ZINC000147456419 BF For-Sale Anodyne GRM6 20 42 C[C@@H](OC[C@@H]1CCCO1)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147456424 EF On-Demand Anodyne GRIN2B 0 40 C[C@@H](OC[C@@H]1CCCO1)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147456424 EF On-Demand Anodyne SCN9A 0 51 CCN(CC)[C@@H](C)CNC(=O)CNC(=O)c1ccccc1 ZINC000147456459 CD On-Demand Anodyne CA2 24 42 CCN(CC)[C@@H](C)CNC(=O)CNC(=O)c1ccccc1 ZINC000147456459 CD On-Demand Anodyne KCNK3 41 34 COc1cc(NCc2cccc([N+](=O)[O-])c2C)ccc1Br ZINC000147456497 FI On-Demand Bother COLA 45 34 NC1(C(=O)Nc2ccc3c(c2)Cc2ccccc2-3)CCC1 ZINC000147456505 CG On-Demand Anodyne SLC1A1 28 53 NC1(C(=O)Nc2ccc3c(c2)Cc2ccccc2-3)CCC1 ZINC000147456505 CG On-Demand Anodyne SLC1A3 33 53 COC(=O)c1ccc(Sc2cc(C(=O)O)ccn2)nc1C ZINC000147456527 DE For-Sale Anodyne KDM4C 0 53 COC(=O)c1ccc(Sc2cc(C(=O)O)ccn2)nc1C ZINC000147456527 DE For-Sale Anodyne KDM3A 0 53 COC(=O)c1ccc(Sc2cc(C(=O)O)ccn2)nc1C ZINC000147456527 DE For-Sale Anodyne KDM5C 0 53 COC(=O)c1ccc(Sc2cc(C(=O)O)ccn2)nc1C ZINC000147456527 DE For-Sale Anodyne FTO 0 40 O=C(O)c1cc(Cl)cc(NC(=O)[C@H]2CC=CCC2)c1 ZINC000147456559 CG On-Demand Anodyne INHA 15 43 CC[C@H](NC(=O)N1CC[C@]2(O)CCCC[C@H]2C1)C(=O)O ZINC000147456597 CD For-Sale Anodyne CCKBR 40 37 C[C@H](CCP(=O)(O)O)CC(C)(C)C ZINC000147456605 BF For-Sale Anodyne GRM6 20 42 CC(C)C(C)(C)C(=O)NCC#N ZINC000147456623 AD On-Demand Mild PAPA1_CARPA 55 40 CC(C)C(C)(C)C(=O)NCC#N ZINC000147456623 AD On-Demand Mild CTSS 23 44 C[C@H](OC[C@H]1CCCO1)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147456629 EF On-Demand Anodyne GRIN2B 0 40 C[C@H](OC[C@H]1CCCO1)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147456629 EF On-Demand Anodyne SCN9A 0 51 CCN(CC)[C@H](C)CNC(=O)CNC(=O)c1ccccc1 ZINC000147456634 CD On-Demand Anodyne CA2 24 42 CCN(CC)[C@H](C)CNC(=O)CNC(=O)c1ccccc1 ZINC000147456634 CD On-Demand Anodyne KCNK3 41 34 Cc1ccc(Br)c(C(=O)N[C@@H](C)c2cc(F)ccc2F)c1 ZINC000147456685 FJ On-Demand Anodyne SDH1 0 45 O=C(O)c1cc(Cl)cc(NC(=O)[C@@H]2CC=CCC2)c1 ZINC000147456758 CG On-Demand Anodyne INHA 15 43 CCNc1ccc(C(=O)NCCNC(=O)N(C)C)cc1 ZINC000147456759 CD For-Sale Anodyne KCNQ1 0 45 CC[C@H](NC(=O)N1CC[C@@]2(O)CCCC[C@H]2C1)C(=O)O ZINC000147456797 CD For-Sale Anodyne CCKBR 40 37 C[C@@H](OC[C@H]1CCCO1)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147456837 EF On-Demand Anodyne GRIN2B 0 40 C[C@@H](OC[C@H]1CCCO1)C(=O)NCc1ccc(OC(F)(F)F)cc1 ZINC000147456837 EF On-Demand Anodyne SCN9A 0 51 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne DRD4 40 32 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne HTR4 48 36 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne F10 15 44 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne CHRM5 19 40 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne GRIN2B 25 46 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne CNR2 15 43 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne MAPK14 25 45 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne PLD1 45 36 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne EPHX2 37 42 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne PLD2 41 36 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne TGM2 71 45 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne CACNA1I 71 43 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne F13A1 64 42 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne AKR1C3 47 36 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147456877 GF On-Demand Anodyne SFRP1 38 41 Cc1ccc(Br)c(C(=O)N[C@H](C)c2cc(F)ccc2F)c1 ZINC000147456879 FJ On-Demand Anodyne SDH1 0 45 O=C(C[C@H]1C=CCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147456947 CG For-Sale Anodyne CACNA1I 45 34 O=C(c1cccnc1SC(F)(F)F)N1CCC(N2CCNC2=O)CC1 ZINC000147456960 FE On-Demand Anodyne CALCRL 21 41 O=C(c1cccnc1SC(F)(F)F)N1CCC(N2CCNC2=O)CC1 ZINC000147456960 FE On-Demand Anodyne L3MBTL3 43 38 C[C@H](CNc1c(C(N)=O)cnc2ccccc12)CC(=O)O ZINC000147456973 CD For-Sale Anodyne PDE4B 17 42 C[C@H](CNc1c(C(N)=O)cnc2ccccc12)CC(=O)O ZINC000147456973 CD For-Sale Anodyne CSF1R 66 47 CCNC(=O)CNc1ccc(Br)c(OC)c1 ZINC000147456993 CE For-Sale Anodyne ENPP1 69 36 Cc1ccc(S(=O)(=O)N2CCN(CCBr)CC2)cc1C ZINC000147457118 FE For-Sale Reactive PKM 45 40 O=C(C[C@@H]1C=CCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147457138 CG For-Sale Anodyne CACNA1I 45 34 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne F2 21 42 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne FKBP1A 19 40 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne SLC6A1 66 32 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne CHRM5 24 40 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne LPL 47 38 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne CCR5 15 41 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne MMP3 27 41 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne MMP9 20 41 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne EPHX2 45 52 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne TGM2 71 43 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne MMP1 31 41 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne PDE8B 16 42 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne F13A1 77 43 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne AKR1C3 19 40 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne SFRP1 78 38 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne WNT3 59 33 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne AKR1C1 21 42 CC(=O)N1CCC[C@@H](C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1 ZINC000147457139 HD On-Demand Anodyne NAMPT 36 44 Nc1ccc(CCC(=O)Nc2ccncc2Br)cc1 ZINC000147457147 DF For-Sale Clean HCAR2 17 41 COc1cc(C(=O)N(C)Cc2cccc(Br)c2)ccc1F ZINC000147457151 FH On-Demand Anodyne GYS1 28 43 COc1cc(C(=O)N(C)Cc2cccc(Br)c2)ccc1F ZINC000147457151 FH On-Demand Anodyne HSD17B2 30 49 COc1cc(C(=O)N(C)Cc2cccc(Br)c2)ccc1F ZINC000147457151 FH On-Demand Anodyne LIMK2 36 41 C[C@@H](CNc1c(C(N)=O)cnc2ccccc12)CC(=O)O ZINC000147457189 CD For-Sale Anodyne PDE4B 17 42 C[C@@H](CNc1c(C(N)=O)cnc2ccccc12)CC(=O)O ZINC000147457189 CD For-Sale Anodyne CSF1R 66 47 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(OCCCC#N)c1 ZINC000147457222 HH On-Demand Mild KCNK3 59 41 CCCS(=O)(=O)Nc1ccccc1C(=O)Nc1cccc(OCCCC#N)c1 ZINC000147457222 HH On-Demand Mild KCNK9 56 41 COC(=O)c1ccc(Sc2cccc(C(=O)O)c2)nc1C ZINC000147457248 DG For-Sale Anodyne ALS 66 33 CCCNC(=O)CNc1ccc(Br)c(OC)c1 ZINC000147457249 DE On-Demand Anodyne ENPP1 50 32 CCCC[C@H](NC(N)=O)C(=O)N(C)Cc1ccccc1[N+](=O)[O-] ZINC000147457256 DD On-Demand Bother COLA 110 44 C[C@H]1CCC[C@@H](C)N1NC(=O)/C=C/c1cccc(N)c1 ZINC000147457270 CF For-Sale Anodyne HDAC8 62 39 Cc1oc(CN)cc1COc1ccc(Cl)c(F)c1 ZINC000147457339 CG For-Sale Anodyne PTGER4 0 43 CN1CC(=O)N(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1=O ZINC000147457356 HC On-Demand Anodyne EPHX2 15 41 CN1CC(=O)N(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1=O ZINC000147457356 HC On-Demand Anodyne TGM2 59 42 CN1CC(=O)N(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1=O ZINC000147457356 HC On-Demand Anodyne CACNA1I 41 35 CN1CC(=O)N(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)C1=O ZINC000147457356 HC On-Demand Anodyne F13A1 60 42 CCN(CC)[C@@H](C)CNC(=O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000147457364 FD On-Demand Anodyne SLC5A7 30 40 CCN(CC)[C@@H](C)CNC(=O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000147457364 FD On-Demand Anodyne MT-ND1 25 41 CCN(CC)[C@@H](C)CNC(=O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000147457364 FD On-Demand Anodyne HCRTR2 15 43 Cc1cc(F)ccc1S(=O)(=O)N1CCN(CCBr)CC1 ZINC000147457386 FD For-Sale Reactive EPHX2 17 50 CN1C[C@H](C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1=O ZINC000147457392 CD On-Demand Anodyne INHA 30 53 COc1ccc([N+](=O)[O-])c(C(=O)N2CCC(N3CCNC3=O)CC2)c1 ZINC000147457393 ED On-Demand Bother OXTR 26 41 Nc1cc(Cl)cc(C(=O)Nc2ccncc2Br)c1 ZINC000147457398 EG For-Sale Anodyne IKBKG 0 40 NC1(C(=O)N2CCN(Cc3ccccc3)CC2)CCC1 ZINC000147457437 CD On-Demand Anodyne DRD2 0 45 NC1(C(=O)N2CCN(Cc3ccccc3)CC2)CCC1 ZINC000147457437 CD On-Demand Anodyne DRD3 0 41 NC1(C(=O)N2CCN(Cc3ccccc3)CC2)CCC1 ZINC000147457437 CD On-Demand Anodyne FAAH 0 49 NC1(C(=O)N2CCN(Cc3ccccc3)CC2)CCC1 ZINC000147457437 CD On-Demand Anodyne MGLL 0 50 NC1(C(=O)N2CCN(Cc3ccccc3)CC2)CCC1 ZINC000147457437 CD On-Demand Anodyne ABHD6 0 46 CC[C@H](OCc1ccccc1Br)C(=O)O ZINC000147457444 CF For-Sale Anodyne ACE2 42 33 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CCN3CCCC3)cc1)C2 ZINC000147457447 GH On-Demand Anodyne HRH3 17 50 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CCN3CCCC3)cc1)C2 ZINC000147457447 GH On-Demand Anodyne SIGMAR1 23 44 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CCN3CCCC3)cc1)C2 ZINC000147457447 GH On-Demand Anodyne HDAC8 18 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CCN3CCCC3)cc1)C2 ZINC000147457447 GH On-Demand Anodyne MTNR1A 32 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CCN3CCCC3)cc1)C2 ZINC000147457447 GH On-Demand Anodyne MTNR1B 33 40 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CCN3CCCC3)cc1)C2 ZINC000147457447 GH On-Demand Anodyne ROCK2 37 51 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CCN3CCCC3)cc1)C2 ZINC000147457447 GH On-Demand Anodyne ABCB1 23 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CCN3CCCC3)cc1)C2 ZINC000147457447 GH On-Demand Anodyne CFTR 40 33 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CCN3CCCC3)cc1)C2 ZINC000147457447 GH On-Demand Anodyne MCHR1 25 40 N#CCCCOc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147457455 FE On-Demand Mild ADORA2B 32 40 N#CCCCOc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147457455 FE On-Demand Mild PLA2G4B 51 40 N#CCCCOc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147457455 FE On-Demand Mild ACR 47 39 N#CCCCOc1cccc(NC(=O)COc2ccc(C(N)=O)cc2)c1 ZINC000147457455 FE On-Demand Mild HIF1A 22 41 CCCC[C@@H](NC(N)=O)C(=O)N(C)Cc1ccccc1[N+](=O)[O-] ZINC000147457471 DD On-Demand Bother COLA 110 44 CC(C)CCCCNC[C@H](O)COCc1ccc(Cl)cc1 ZINC000147457481 DH For-Sale Anodyne ADRB2 24 43 CC(C)CCCCNC[C@H](O)COCc1ccc(Cl)cc1 ZINC000147457481 DH For-Sale Anodyne ADRB1 33 40 CC(C)CCCCNC[C@H](O)COCc1ccc(Cl)cc1 ZINC000147457481 DH For-Sale Anodyne ADRB3 27 40 COc1cc(NCC(=O)Nc2cccc(Br)c2)ccc1Br ZINC000147457486 HI For-Sale Anodyne EGFR 34 42 COc1cc(NCC(=O)Nc2cccc(Br)c2)ccc1Br ZINC000147457486 HI For-Sale Anodyne IMPDH2 0 48 COc1cc(NCC(=O)Nc2cccc(Br)c2)ccc1Br ZINC000147457486 HI For-Sale Anodyne ENPP1 77 39 COc1cc(NCC(=O)Nc2cccc(Br)c2)ccc1Br ZINC000147457486 HI For-Sale Anodyne KCNK3 41 39 C[C@H]1CCC[C@H](C)N1NC(=O)/C=C/c1cccc(N)c1 ZINC000147457495 CF For-Sale Anodyne HDAC8 62 39 CCCCCCCCCCC(=O)c1cncs1 ZINC000147457532 CJ For-Sale Mild THRA 47 35 CCCCCCCCCCC(=O)c1cncs1 ZINC000147457532 CJ For-Sale Mild CDC25B 65 38 CCCCCCCCCCC(=O)c1cncs1 ZINC000147457532 CJ For-Sale Mild FAAH 25 40 CCCCCCCCCCC(=O)c1cncs1 ZINC000147457532 CJ For-Sale Mild FFAR1 0 43 CCCCCCCCCCC(=O)c1cncs1 ZINC000147457532 CJ For-Sale Mild CQSS 56 34 CCN(CC)[C@H](C)CNC(=O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000147457571 FD On-Demand Anodyne SLC5A7 30 40 CCN(CC)[C@H](C)CNC(=O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000147457571 FD On-Demand Anodyne MT-ND1 25 41 CCN(CC)[C@H](C)CNC(=O)CNC(=O)c1ccc(OC)c(OC)c1 ZINC000147457571 FD On-Demand Anodyne HCRTR2 15 43 O=C(CN1CCCC1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457579 GC On-Demand Anodyne EPHX2 24 45 O=C(CN1CCCC1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457579 GC On-Demand Anodyne TGM2 76 46 O=C(CN1CCCC1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457579 GC On-Demand Anodyne CACNA1I 42 34 O=C(CN1CCCC1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457579 GC On-Demand Anodyne F13A1 86 46 O=C(CN1CCCC1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457579 GC On-Demand Anodyne AKR1C3 55 37 O=C(CN1CCCC1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457579 GC On-Demand Anodyne NAMPT 25 40 CN1C[C@@H](C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1=O ZINC000147457619 CD On-Demand Anodyne INHA 30 53 CC[C@@H](OCc1ccccc1Br)C(=O)O ZINC000147457646 CF For-Sale Anodyne ACE2 42 33 NC(=O)[C@@H]1NC[C@H](O)[C@@H](O)[C@@H]1O ZINC000147457650 AA For-Sale Anodyne GANAB 0 40 NC(=O)[C@@H]1NC[C@H](O)[C@@H](O)[C@@H]1O ZINC000147457650 AA For-Sale Anodyne GANC 0 40 NC(=O)[C@@H]1NC[C@H](O)[C@@H](O)[C@@H]1O ZINC000147457650 AA For-Sale Anodyne AGLC 0 40 NC(=O)[C@@H]1NC[C@H](O)[C@@H](O)[C@@H]1O ZINC000147457650 AA For-Sale Anodyne Q43014_PRUAV 0 40 NC(=O)[C@@H]1NC[C@H](O)[C@@H](O)[C@@H]1O ZINC000147457650 AA For-Sale Anodyne LACA 0 40 NC(=O)[C@@H]1NC[C@H](O)[C@@H](O)[C@@H]1O ZINC000147457650 AA For-Sale Anodyne AGL 0 40 NC(=O)[C@@H]1NC[C@H](O)[C@@H](O)[C@@H]1O ZINC000147457650 AA For-Sale Anodyne SGA1 0 42 CC(C)CCCCNC[C@@H](O)COCc1ccc(Cl)cc1 ZINC000147457657 DH For-Sale Anodyne ADRB2 24 43 CC(C)CCCCNC[C@@H](O)COCc1ccc(Cl)cc1 ZINC000147457657 DH For-Sale Anodyne ADRB1 33 40 CC(C)CCCCNC[C@@H](O)COCc1ccc(Cl)cc1 ZINC000147457657 DH For-Sale Anodyne ADRB3 27 40 COc1ccc2c(c1)OC[C@H](C(=O)N[C@@H](C)COc1ccc(F)cc1F)C2 ZINC000147457687 GG On-Demand Anodyne ROCK2 25 40 C[C@@H]1CCC[C@@H](C)N1NC(=O)/C=C/c1cccc(N)c1 ZINC000147457701 CF For-Sale Anodyne HDAC8 62 39 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(Cl)c(Cl)c2)C1 ZINC000147457709 GH On-Demand Anodyne NPY2R 45 36 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(Cl)c(Cl)c2)C1 ZINC000147457709 GH On-Demand Anodyne ENV 43 33 COc1cc(NCC(=O)Nc2ccccc2)ccc1Br ZINC000147457728 EH On-Demand Anodyne TSHR 40 30 COc1cc(NCC(=O)Nc2ccccc2)ccc1Br ZINC000147457728 EH On-Demand Anodyne CETP 0 40 COc1cc(NCC(=O)Nc2ccccc2)ccc1Br ZINC000147457728 EH On-Demand Anodyne CPT1A 45 32 COc1cc(NCC(=O)Nc2ccccc2)ccc1Br ZINC000147457728 EH On-Demand Anodyne MTNR1B 18 42 COc1cc(NCC(=O)Nc2ccccc2)ccc1Br ZINC000147457728 EH On-Demand Anodyne IMPDH2 0 48 COc1cc(NCC(=O)Nc2ccccc2)ccc1Br ZINC000147457728 EH On-Demand Anodyne ENPP1 75 37 COc1cc(NCC(=O)Nc2ccccc2)ccc1Br ZINC000147457728 EH On-Demand Anodyne DRTS_TRYCR 43 30 COc1cccc(N)c1C(=O)Nc1ccncc1Br ZINC000147457811 DF For-Sale Anodyne HDAC1 20 40 CCN(CC)[C@@H](C)CNC(=O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000147457813 ED On-Demand Bother CACNA1D 47 33 CCN(CC)[C@@H](C)CNC(=O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000147457813 ED On-Demand Bother CCR2 31 44 CC(C)(C)C(=O)NCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457835 GD On-Demand Anodyne EPHX2 31 45 CC(C)(C)C(=O)NCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457835 GD On-Demand Anodyne TGM2 76 45 CC(C)(C)C(=O)NCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457835 GD On-Demand Anodyne CACNA1I 61 40 CC(C)(C)C(=O)NCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457835 GD On-Demand Anodyne F13A1 78 45 CC(C)(C)C(=O)NCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457835 GD On-Demand Anodyne AKR1C3 43 36 CC(C)(C)C(=O)NCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147457835 GD On-Demand Anodyne SFRP1 61 41 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1OCC(F)(F)F ZINC000147457843 FD On-Demand Anodyne PCSK5 50 31 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1OCC(F)(F)F ZINC000147457843 FD On-Demand Anodyne FURIN 45 32 C[C@H](CNc1ccc(C(N)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147457853 CD For-Sale Bother TAAR1 15 41 COc1ccc2c(c1)OC[C@H](C(=O)N[C@H](C)COc1ccc(F)cc1F)C2 ZINC000147457887 GG On-Demand Anodyne ROCK2 25 40 Cc1cc(Cl)cc(C(=O)N(C)Cc2cccc(C#N)c2)c1 ZINC000147457896 CH On-Demand Mild HSD17B2 25 44 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(Cl)c(Cl)c2)C1 ZINC000147457912 GH On-Demand Anodyne NPY2R 45 36 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(Cl)c(Cl)c2)C1 ZINC000147457912 GH On-Demand Anodyne ENV 43 33 NS(=O)(=O)c1cc(Br)c(OCCCN2CCCC2)cc1F ZINC000147457945 GE For-Sale Anodyne HRH3 45 49 COc1cc(NCC(=O)NC2CC2)ccc1Br ZINC000147457952 CE On-Demand Anodyne ENPP1 50 31 COCCOCCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147457962 DD On-Demand Anodyne CACNA1I 43 34 NC(=O)C1(c2cccc([N+](=O)[O-])c2)CC1 ZINC000147457997 BD In-Stock Bother CACNA1C 52 35 NC(=O)C1(c2cccc([N+](=O)[O-])c2)CC1 ZINC000147457997 BD In-Stock Bother CACNA1D 84 35 NC(=O)C1(c2cccc([N+](=O)[O-])c2)CC1 ZINC000147457997 BD In-Stock Bother UREA_CANEN 16 40 COC(=O)Oc1ccc(C)c(F)c1 ZINC000147458004 AE For-Sale Anodyne LEF 51 37 CCN(CC)[C@H](C)CNC(=O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000147458018 ED On-Demand Bother CACNA1D 47 33 CCN(CC)[C@H](C)CNC(=O)CNC(=O)c1cccc([N+](=O)[O-])c1 ZINC000147458018 ED On-Demand Bother CCR2 31 44 COC(=O)[C@@H](C)C[C@@H](c1cccc(Cl)c1)[C@H](O)c1ccc(Cl)cc1 ZINC000147458039 FK For-Sale Anodyne CNR1 17 40 Nc1ccc(Cl)cc1C(=O)Nc1ccncc1Br ZINC000147458043 EG For-Sale Anodyne F10 32 41 Nc1ccc(Cl)cc1C(=O)Nc1ccncc1Br ZINC000147458043 EG For-Sale Anodyne HDAC1 0 40 Nc1ccc(Cl)cc1C(=O)Nc1ccncc1Br ZINC000147458043 EG For-Sale Anodyne KCNMA1 26 43 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne DRD2 18 43 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne CNR1 21 43 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne DRD3 16 43 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne HTR4 91 50 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne CNR2 27 40 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne HTR6 30 42 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne EPHX2 19 42 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne TGM2 61 43 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne CACNA1I 59 35 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne F13A1 56 43 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne AKR1C3 20 40 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne AKR1C1 21 40 Cn1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c2ccccc21 ZINC000147458050 HG On-Demand Anodyne NAMPT 42 38 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1OCC(F)(F)F ZINC000147458059 FD On-Demand Anodyne PCSK5 50 31 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1OCC(F)(F)F ZINC000147458059 FD On-Demand Anodyne FURIN 45 32 O=C(Cc1cccc(C(F)(F)F)c1)c1cncs1 ZINC000147458061 CH For-Sale Anodyne CSNK1D 24 45 C[C@@H](CNc1ccc(C(N)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147458072 CD For-Sale Bother TAAR1 15 41 COc1ccc2c(c1)OC[C@@H](C(=O)N[C@@H](C)COc1ccc(F)cc1F)C2 ZINC000147458086 GG On-Demand Anodyne ROCK2 25 40 NCC1(CC(=O)NCc2ccccc2Cl)CCC1 ZINC000147458160 CE For-Sale Anodyne P2RX7 38 43 COc1cc(NCC(=O)Nc2ccc(Cl)cc2)ccc1Br ZINC000147458167 FI On-Demand Anodyne HTR2A 35 46 COc1cc(NCC(=O)Nc2ccc(Cl)cc2)ccc1Br ZINC000147458167 FI On-Demand Anodyne COLA 50 35 COc1cc(NCC(=O)Nc2ccc(Cl)cc2)ccc1Br ZINC000147458167 FI On-Demand Anodyne CPT1A 48 35 COc1cc(NCC(=O)Nc2ccc(Cl)cc2)ccc1Br ZINC000147458167 FI On-Demand Anodyne CPT1B 40 34 COc1cc(NCC(=O)Nc2ccc(Cl)cc2)ccc1Br ZINC000147458167 FI On-Demand Anodyne ENPP1 75 39 COc1cc(NCC(=O)Nc2ccc(Cl)cc2)ccc1Br ZINC000147458167 FI On-Demand Anodyne DRTS_TRYCR 43 29 COc1cc(NCC(=O)Nc2ccc(Cl)cc2)ccc1Br ZINC000147458167 FI On-Demand Anodyne PSBA 0 42 CC(=O)Nc1cccc(/C=C\c2ccsc2C(=O)O)c1 ZINC000147458179 CH For-Sale Anodyne AKR1C3 29 41 CC(=O)Nc1cccc(/C=C\c2ccsc2C(=O)O)c1 ZINC000147458179 CH For-Sale Anodyne KCNK3 71 37 COC(=O)[C@H](C)C[C@@H](c1cccc(Cl)c1)[C@H](O)c1ccc(Cl)cc1 ZINC000147458245 FK For-Sale Anodyne CNR1 17 40 CC1(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CCCC1 ZINC000147458250 CH On-Demand Anodyne RARA 43 37 CC1(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CCCC1 ZINC000147458250 CH On-Demand Anodyne HCAR1 0 40 CCc1cc(Br)ccc1NCc1ccc(C(N)=O)cc1 ZINC000147458255 EH On-Demand Anodyne MVFR 0 40 COc1ccc(C(=O)Nc2ccncc2Br)cc1N ZINC000147458273 DF For-Sale Anodyne HDAC1 25 40 COc1ccc(C(=O)Nc2ccncc2Br)cc1N ZINC000147458273 DF For-Sale Anodyne HDAC2 20 40 COc1ccc(C(=O)Nc2ccncc2Br)cc1N ZINC000147458273 DF For-Sale Anodyne TAAR1 22 40 COc1ccc(C(=O)Nc2ccncc2Br)cc1N ZINC000147458273 DF For-Sale Anodyne SIRT2 17 42 C[C@H](CNc1ccc(S(C)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147458285 DD On-Demand Bother BDKRB1 0 47 C[C@H](CNc1ccc(S(C)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147458285 DD On-Demand Bother COLA 67 34 O=C(Nc1nc2ccc(Cl)cc2s1)[C@@H]1CCCN1C1CCOCC1 ZINC000147458294 FH Annotated Anodyne CASR 18 47 O=C(Nc1nc2ccc(Cl)cc2s1)[C@@H]1CCCN1C1CCOCC1 ZINC000147458294 FH Annotated Anodyne LCK 25 40 O=C(Nc1nc2ccc(Cl)cc2s1)[C@@H]1CCCN1C1CCOCC1 ZINC000147458294 FH Annotated Anodyne CSNK1D 34 41 O=C(Nc1nc2ccc(Cl)cc2s1)[C@@H]1CCCN1C1CCOCC1 ZINC000147458294 FH Annotated Anodyne HSD17B1 33 40 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne DRD2 43 47 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne DRD4 41 32 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne ACHE 17 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne DRD3 39 42 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne HTR4 45 37 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne F10 17 46 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne GRIN2B 17 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne CPT1A 78 37 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne CPT2 49 36 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne EPHX2 22 41 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne TGM2 62 49 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne CPT1B 53 35 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne CACNA1I 76 42 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne F13A1 48 41 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne AKR1C3 40 38 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne SFRP1 29 40 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1F ZINC000147458311 HF On-Demand Anodyne ACKR3 72 37 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N(C)C ZINC000147458317 DD On-Demand Anodyne KLK3 58 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N(C)C ZINC000147458317 DD On-Demand Anodyne CXCR2 59 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N(C)C ZINC000147458317 DD On-Demand Anodyne CXCR1 70 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N(C)C ZINC000147458317 DD On-Demand Anodyne POLG_WNV 74 33 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N(C)C ZINC000147458317 DD On-Demand Anodyne NPFFR1 42 33 CCN(CC)[C@@H](C)CNC(=O)CNC(=O)c1cc(C)cc(C)c1 ZINC000147458320 DD On-Demand Anodyne ECR 35 41 COc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cn1 ZINC000147458360 HD On-Demand Anodyne ADRB2 22 47 COc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cn1 ZINC000147458360 HD On-Demand Anodyne ADRB1 62 40 COc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cn1 ZINC000147458360 HD On-Demand Anodyne ADRB3 18 47 COc1ccc(NC(=O)C2(N)CCC2)cc1OC ZINC000147458373 CD On-Demand Anodyne QRFPR 41 34 COc1ccc(NC(=O)C2(N)CCC2)cc1OC ZINC000147458373 CD On-Demand Anodyne ENPP1 66 39 COc1ccc(NC(=O)C2(N)CCC2)cc1OC ZINC000147458373 CD On-Demand Anodyne DRTS_TRYCR 46 33 COC(=O)[C@@H]1[C@H](O)C[C@@H]2CC(=O)C[C@@H]12 ZINC000147458381 AC For-Sale Anodyne SLC6A1 45 32 COc1cc(NCC(=O)Nc2ccc(F)cc2)ccc1Br ZINC000147458392 FH On-Demand Anodyne HTR2A 20 46 COc1cc(NCC(=O)Nc2ccc(F)cc2)ccc1Br ZINC000147458392 FH On-Demand Anodyne ENPP1 65 38 COc1cc(NCC(=O)Nc2ccc(F)cc2)ccc1Br ZINC000147458392 FH On-Demand Anodyne DRTS_TRYCR 43 29 CC(C)NCc1coc(COc2ccc(Cl)c(F)c2)c1 ZINC000147458422 CI For-Sale Anodyne DAO 15 42 COC(=O)[C@@H](C)C[C@H](c1cccc(Cl)c1)[C@@H](O)c1ccc(Cl)cc1 ZINC000147458460 FK For-Sale Anodyne CNR1 17 40 C[C@@H](CNc1ccc(S(C)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147458490 DD On-Demand Bother BDKRB1 0 47 C[C@@H](CNc1ccc(S(C)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147458490 DD On-Demand Bother COLA 67 34 O=C(CCc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147458519 HF On-Demand Anodyne FKBP1A 19 48 O=C(CCc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147458519 HF On-Demand Anodyne GRIN2B 41 40 O=C(CCc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147458519 HF On-Demand Anodyne SIGMAR1 22 41 O=C(CCc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147458519 HF On-Demand Anodyne CCR3 51 46 O=C(CCc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147458519 HF On-Demand Anodyne EPHX2 19 42 O=C(CCc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147458519 HF On-Demand Anodyne TGM2 80 46 O=C(CCc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147458519 HF On-Demand Anodyne F13A1 88 46 O=C(CCc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147458519 HF On-Demand Anodyne NAMPT 45 38 CCN(CC)[C@H](C)CNC(=O)CNC(=O)c1cc(C)cc(C)c1 ZINC000147458527 DD On-Demand Anodyne ECR 35 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N(C)C ZINC000147458530 DD On-Demand Anodyne KLK3 58 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N(C)C ZINC000147458530 DD On-Demand Anodyne CXCR2 59 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N(C)C ZINC000147458530 DD On-Demand Anodyne CXCR1 70 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N(C)C ZINC000147458530 DD On-Demand Anodyne POLG_WNV 74 33 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1C(=O)N(C)C ZINC000147458530 DD On-Demand Anodyne NPFFR1 42 33 COc1ccc(CCC(=O)NNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147458555 GE On-Demand Reactive MTNR1A 56 42 COc1ccc(CCC(=O)NNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147458555 GE On-Demand Reactive MTNR1B 50 36 COc1ccc(CCC(=O)NNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147458555 GE On-Demand Reactive ROCK2 27 43 COc1ccc(CCC(=O)NNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147458555 GE On-Demand Reactive HCAR2 18 43 N[C@@H](COCc1ccccc1Br)C(=O)O ZINC000147458581 CD For-Sale Anodyne CACNA2D1 24 57 N[C@@H](COCc1ccccc1Br)C(=O)O ZINC000147458581 CD For-Sale Anodyne GRIK3 21 40 N[C@@H](COCc1ccccc1Br)C(=O)O ZINC000147458581 CD For-Sale Anodyne SLC1A1 32 49 N[C@@H](COCc1ccccc1Br)C(=O)O ZINC000147458581 CD For-Sale Anodyne KYNU 0 40 N[C@@H](COCc1ccccc1Br)C(=O)O ZINC000147458581 CD For-Sale Anodyne KIF11 28 46 COc1cc(NCC(=O)NCCC(C)C)ccc1Br ZINC000147458587 EG For-Sale Anodyne ENPP1 67 33 Fc1cccc(NC(=S)S)c1 ZINC000147458600 AE For-Sale Anodyne KCNK3 20 45 COc1ccc(NC(=O)CC2(CN)CCC2)cc1OC ZINC000147458601 CE For-Sale Anodyne QRFPR 41 34 COc1ccc(NC(=O)CC2(CN)CCC2)cc1OC ZINC000147458601 CE For-Sale Anodyne ENPP1 89 44 COc1ccc(NC(=O)CC2(CN)CCC2)cc1OC ZINC000147458601 CE For-Sale Anodyne DRTS_TRYCR 47 33 Cc1cccc(-c2cnc(N)c(-c3nnc(-c4ccccc4)o3)n2)c1 ZINC000147458670 EH For-Sale Anodyne ATM 30 42 Cc1cccc(-c2cnc(N)c(-c3nnc(-c4ccccc4)o3)n2)c1 ZINC000147458670 EH For-Sale Anodyne ATR 40 51 COC(=O)[C@H](C)C[C@H](c1cccc(Cl)c1)[C@@H](O)c1ccc(Cl)cc1 ZINC000147458681 FK For-Sale Anodyne CNR1 17 40 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)s1 ZINC000147458688 DH On-Demand Anodyne JUN 23 46 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)s1 ZINC000147458688 DH On-Demand Anodyne ATF1 59 41 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)s1 ZINC000147458688 DH On-Demand Anodyne NFKB1 54 41 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)s1 ZINC000147458688 DH On-Demand Anodyne TMPRSS4 0 40 CC(C)CCCCNC[C@H](O)c1ccc2ccccc2c1 ZINC000147458748 CI For-Sale Anodyne ADRB2 60 46 CC(C)CCCCNC[C@H](O)c1ccc2ccccc2c1 ZINC000147458748 CI For-Sale Anodyne ADRB1 49 42 CC(C)CCCCNC[C@H](O)c1ccc2ccccc2c1 ZINC000147458748 CI For-Sale Anodyne ADRB3 55 42 N[C@H](COCc1ccccc1Br)C(=O)O ZINC000147458765 CD For-Sale Anodyne CACNA2D1 24 57 N[C@H](COCc1ccccc1Br)C(=O)O ZINC000147458765 CD For-Sale Anodyne GRIK3 21 40 N[C@H](COCc1ccccc1Br)C(=O)O ZINC000147458765 CD For-Sale Anodyne SLC1A1 32 49 N[C@H](COCc1ccccc1Br)C(=O)O ZINC000147458765 CD For-Sale Anodyne KYNU 0 40 N[C@H](COCc1ccccc1Br)C(=O)O ZINC000147458765 CD For-Sale Anodyne KIF11 28 46 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)oc2ccccc12 ZINC000147458780 HH On-Demand Anodyne HTR4 65 41 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)oc2ccccc12 ZINC000147458780 HH On-Demand Anodyne MMP13 19 44 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)oc2ccccc12 ZINC000147458780 HH On-Demand Anodyne EPHX2 22 42 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)oc2ccccc12 ZINC000147458780 HH On-Demand Anodyne TGM2 60 43 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)oc2ccccc12 ZINC000147458780 HH On-Demand Anodyne CACNA1I 57 36 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)oc2ccccc12 ZINC000147458780 HH On-Demand Anodyne F13A1 56 43 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)oc2ccccc12 ZINC000147458780 HH On-Demand Anodyne CCR8 49 33 Cc1c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)oc2ccccc12 ZINC000147458780 HH On-Demand Anodyne NAMPT 40 38 COc1ccc(CNC(=O)C2(N)CCC2)cc1 ZINC000147458795 BD On-Demand Anodyne ANPEP 20 49 COc1ccc(CNC(=O)C2(N)CCC2)cc1 ZINC000147458795 BD On-Demand Anodyne TRPV1 29 43 COc1ccc(CNC(=O)C2(N)CCC2)cc1 ZINC000147458795 BD On-Demand Anodyne MTNR1A 42 37 COc1ccc(CNC(=O)C2(N)CCC2)cc1 ZINC000147458795 BD On-Demand Anodyne MMP8 15 40 COc1ccc(CNC(=O)C2(N)CCC2)cc1 ZINC000147458795 BD On-Demand Anodyne CA12 15 51 COc1ccc(CNC(=O)C2(N)CCC2)cc1 ZINC000147458795 BD On-Demand Anodyne DPP7 15 47 COc1ccc(CNC(=O)C2(N)CCC2)cc1 ZINC000147458795 BD On-Demand Anodyne CA9 26 51 COc1ccc(CNC(=O)C2(N)CCC2)cc1 ZINC000147458795 BD On-Demand Anodyne MMP1 38 41 COc1ccc(CNC(=O)C2(N)CCC2)cc1 ZINC000147458795 BD On-Demand Anodyne U38 0 45 COc1ccc(CNC(=O)C2(N)CCC2)cc1 ZINC000147458795 BD On-Demand Anodyne PROKR1 56 35 COc1ccc(CNC(=O)C2(N)CCC2)cc1 ZINC000147458795 BD On-Demand Anodyne KCNJ2 0 43 O=C(O)c1cc(Cl)cc(NC(=O)c2csc(Br)c2)c1 ZINC000147458898 FI On-Demand Anodyne PPIA 16 46 O=C(O)c1cc(Cl)cc(NC(=O)c2csc(Br)c2)c1 ZINC000147458898 FI On-Demand Anodyne KCNK3 43 40 CC(C)CCCCNC[C@@H](O)c1ccc2ccccc2c1 ZINC000147458949 CI For-Sale Anodyne ADRB2 60 46 CC(C)CCCCNC[C@@H](O)c1ccc2ccccc2c1 ZINC000147458949 CI For-Sale Anodyne ADRB1 49 42 CC(C)CCCCNC[C@@H](O)c1ccc2ccccc2c1 ZINC000147458949 CI For-Sale Anodyne ADRB3 55 42 COc1ccc(N)c(C(=O)Nc2ccncc2Br)c1 ZINC000147458960 DF For-Sale Anodyne AKR1C2 50 36 COc1ncccc1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147458973 HD On-Demand Anodyne ADRB2 20 46 CCCC[C@H](NC(N)=O)C(=O)N1CCN(c2ccc([N+](=O)[O-])nc2)CC1 ZINC000147458987 FC On-Demand Bother P2RY12 184 40 CC[C@@H]1CN(CCOc2ccccc2OC)CC[C@@H]1N ZINC000147458993 CE On-Demand Anodyne HTR1A 24 41 CC[C@@H]1CN(CCOc2ccccc2OC)CC[C@@H]1N ZINC000147458993 CE On-Demand Anodyne DRD2 23 44 COc1ccc(CNC(=O)CC2(CN)CCC2)cc1 ZINC000147459009 CD For-Sale Anodyne MTNR1A 65 39 COc1ccc(CNC(=O)CC2(CN)CCC2)cc1 ZINC000147459009 CD For-Sale Anodyne MTNR1B 55 39 COc1ccc(CNC(=O)CC2(CN)CCC2)cc1 ZINC000147459009 CD For-Sale Anodyne TPSAB1 18 41 COc1ccc(CNC(=O)CC2(CN)CCC2)cc1 ZINC000147459009 CD For-Sale Anodyne CA9 23 51 COc1ccc(CNC(=O)CC2(CN)CCC2)cc1 ZINC000147459009 CD For-Sale Anodyne PROKR1 58 32 COc1ccc(CNC(=O)CC2(CN)CCC2)cc1 ZINC000147459009 CD For-Sale Anodyne KCNJ2 0 41 CC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147459033 HF On-Demand Anodyne HTR4 51 36 CC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147459033 HF On-Demand Anodyne MMP13 16 41 CC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147459033 HF On-Demand Anodyne ITGA4 22 41 CC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147459033 HF On-Demand Anodyne EPHX2 20 43 CC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147459033 HF On-Demand Anodyne TGM2 69 44 CC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147459033 HF On-Demand Anodyne CACNA1I 58 34 CC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147459033 HF On-Demand Anodyne F13A1 66 44 CC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147459033 HF On-Demand Anodyne SIRT3 42 34 CC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147459033 HF On-Demand Anodyne SIRT2 40 35 CC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147459033 HF On-Demand Anodyne SIRT1 42 34 CC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)s1 ZINC000147459033 HF On-Demand Anodyne SFRP1 52 39 COc1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1Br ZINC000147459099 HI For-Sale Reactive ACKR3 67 36 COc1ccc(S(=O)(=O)CC[C@H](O)c2ccccc2)cc1 ZINC000147459141 DF On-Demand Anodyne BMP1 73 39 COc1ccc(S(=O)(=O)CC[C@H](O)c2ccccc2)cc1 ZINC000147459141 DF On-Demand Anodyne MMP13 45 59 COc1ccc(S(=O)(=O)CC[C@H](O)c2ccccc2)cc1 ZINC000147459141 DF On-Demand Anodyne MMP2 37 47 COc1ccc(S(=O)(=O)CC[C@H](O)c2ccccc2)cc1 ZINC000147459141 DF On-Demand Anodyne MMP3 43 40 COc1ccc(S(=O)(=O)CC[C@H](O)c2ccccc2)cc1 ZINC000147459141 DF On-Demand Anodyne MMP8 25 42 COc1ccc(S(=O)(=O)CC[C@H](O)c2ccccc2)cc1 ZINC000147459141 DF On-Demand Anodyne MMP14 20 47 COc1ccc(S(=O)(=O)CC[C@H](O)c2ccccc2)cc1 ZINC000147459141 DF On-Demand Anodyne MMP9 38 42 COc1ccc(S(=O)(=O)CC[C@H](O)c2ccccc2)cc1 ZINC000147459141 DF On-Demand Anodyne MMP1 47 42 Cc1cccc(N)c1C(=O)Nc1ccncc1Br ZINC000147459183 DF For-Sale Anodyne HDAC1 21 42 Nc1cc(Cl)c(S(=O)(=O)CCO)cc1S(=O)(=O)CCO ZINC000147459184 EB For-Sale Anodyne CAH_METTE 19 52 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(c2ccc([N+](=O)[O-])nc2)CC1 ZINC000147459195 FC On-Demand Bother P2RY12 184 40 CC[C@H]1CN(CCOc2ccccc2OC)CC[C@@H]1N ZINC000147459202 CE On-Demand Anodyne HTR1A 24 41 CC[C@H]1CN(CCOc2ccccc2OC)CC[C@@H]1N ZINC000147459202 CE On-Demand Anodyne DRD2 23 44 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c(C)c1 ZINC000147459226 HG On-Demand Anodyne ADRB2 21 43 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c(C)c1 ZINC000147459226 HG On-Demand Anodyne ADRB1 48 35 O=C(c1cncs1)[C@@H]1CCCc2cccnc21 ZINC000147459233 BF For-Sale Anodyne CXCR4 51 34 CC(C)C[C@H](N)C(=O)NN1[C@@H](C)CCC[C@H]1C ZINC000147459253 BD For-Sale Anodyne AMPX_VIBPR 0 47 CC(C)CCO[C@H](C)C(=O)N1CCc2sccc2[C@H]1C ZINC000147459263 CH On-Demand Anodyne TRPM8 16 40 O=C(Nc1cc(C(F)(F)F)ccn1)[C@@H]1CCCN1C1CCOCC1 ZINC000147459264 EF On-Demand Anodyne MAPK10 16 44 O=C(Nc1cc(C(F)(F)F)ccn1)[C@@H]1CCCN1C1CCOCC1 ZINC000147459264 EF On-Demand Anodyne MAP3K12 33 43 COC(=O)c1cc(CNc2ccc(Br)c(OC)c2)oc1C ZINC000147459267 FH On-Demand Anodyne DRTS_TRYCR 45 32 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCCC2 ZINC000147459268 HG On-Demand Anodyne NPY2R 53 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCCC2 ZINC000147459268 HG On-Demand Anodyne NPY5R 17 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCCC2 ZINC000147459268 HG On-Demand Anodyne EPHX2 17 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCCC2 ZINC000147459268 HG On-Demand Anodyne TGM2 60 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCCC2 ZINC000147459268 HG On-Demand Anodyne CACNA1I 59 33 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCCC2 ZINC000147459268 HG On-Demand Anodyne F13A1 42 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCCC2 ZINC000147459268 HG On-Demand Anodyne AKR1C3 58 36 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCCC2 ZINC000147459268 HG On-Demand Anodyne NAMPT 38 44 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccccc2N2CCCCCC2)C1 ZINC000147459288 HH On-Demand Anodyne KCNQ2 88 43 COc1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1Br ZINC000147459322 HI For-Sale Reactive ACKR3 67 36 CCCCc1ccc(Oc2cc(C(N)=O)ccc2N)cc1 ZINC000147459380 CH For-Sale Anodyne INHA 100 43 CCCCc1ccc(Oc2cc(C(N)=O)ccc2N)cc1 ZINC000147459380 CH For-Sale Anodyne PLA2G4A 34 47 CCCCc1ccc(Oc2cc(C(N)=O)ccc2N)cc1 ZINC000147459380 CH For-Sale Anodyne SELE 41 39 CCCCc1ccc(Oc2cc(C(N)=O)ccc2N)cc1 ZINC000147459380 CH For-Sale Anodyne ICAM1 37 49 CCCCc1ccc(Oc2cc(C(N)=O)ccc2N)cc1 ZINC000147459380 CH For-Sale Anodyne PLA2G4B 66 33 CCCCc1ccc(Oc2cc(C(N)=O)ccc2N)cc1 ZINC000147459380 CH For-Sale Anodyne S1PR1 15 42 CCCCc1ccc(Oc2cc(C(N)=O)ccc2N)cc1 ZINC000147459380 CH For-Sale Anodyne ENR 0 49 O=C(O)c1cc(Cl)cnc1NC1CC1 ZINC000147459411 BE For-Sale Anodyne TYRO3 42 38 Cc1cccc(C)c1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147459441 HG On-Demand Anodyne ADRB2 31 43 Cc1cccc(C)c1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147459441 HG On-Demand Anodyne ADRB1 56 36 Cc1cccc(C)c1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147459441 HG On-Demand Anodyne ABCB1 47 37 CCOC(=O)Cc1csc(-c2cc(Cl)ccc2F)n1 ZINC000147459447 CH For-Sale Anodyne PTGER1 24 48 CCOC(=O)Cc1csc(-c2cc(Cl)ccc2F)n1 ZINC000147459447 CH For-Sale Anodyne DPP8 41 34 CCOC(=O)Cc1csc(-c2cc(Cl)ccc2F)n1 ZINC000147459447 CH For-Sale Anodyne DPP9 40 34 CCc1cc(Br)ccc1NCc1cccc(C(N)=O)c1 ZINC000147459450 EH On-Demand Anodyne MVFR 0 51 O=C(c1cncs1)[C@H]1CCCc2cccnc21 ZINC000147459464 BF For-Sale Anodyne CXCR4 51 34 COc1cc(NC(=O)CC2(CN)CCC2)cc(OC)c1 ZINC000147459481 CE For-Sale Anodyne MTNR1B 27 41 CC(C)CCO[C@H](C)C(=O)N1CCc2sccc2[C@@H]1C ZINC000147459483 CH On-Demand Anodyne TRPM8 16 40 CC[C@@H](C)NC(=O)CNc1ccc(Br)c(OC)c1 ZINC000147459491 DF On-Demand Anodyne ENPP1 50 31 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccccc2N2CCCCCC2)C1 ZINC000147459495 HH On-Demand Anodyne KCNQ2 88 43 CC(C)C[C@H](N)C(=O)NN1[C@@H](C)CCC[C@@H]1C ZINC000147459497 BD For-Sale Anodyne AMPX_VIBPR 0 47 CCc1cc(Br)ccc1NC(=O)N[C@@H](CC)C(=O)O ZINC000147459518 EF For-Sale Anodyne FOLH1 25 40 CCc1cc(Br)ccc1NC(=O)N[C@@H](CC)C(=O)O ZINC000147459518 EF For-Sale Anodyne ANPEP 29 42 CCc1cc(Br)ccc1NC(=O)N[C@@H](CC)C(=O)O ZINC000147459518 EF For-Sale Anodyne ACE2 54 33 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(Cl)cc1F ZINC000147459519 HG On-Demand Anodyne DRD2 20 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(Cl)cc1F ZINC000147459519 HG On-Demand Anodyne DRD4 15 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(Cl)cc1F ZINC000147459519 HG On-Demand Anodyne HTR4 53 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(Cl)cc1F ZINC000147459519 HG On-Demand Anodyne CHRM5 15 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(Cl)cc1F ZINC000147459519 HG On-Demand Anodyne CNR2 17 47 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(Cl)cc1F ZINC000147459519 HG On-Demand Anodyne APP 46 36 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(Cl)cc1F ZINC000147459519 HG On-Demand Anodyne SLC6A9 70 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(Cl)cc1F ZINC000147459519 HG On-Demand Anodyne EPHX2 33 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(Cl)cc1F ZINC000147459519 HG On-Demand Anodyne TGM2 65 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(Cl)cc1F ZINC000147459519 HG On-Demand Anodyne CACNA1I 74 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(Cl)cc1F ZINC000147459519 HG On-Demand Anodyne F13A1 61 43 C[C@H](CNc1cccc(Cl)c1C(N)=O)CC(=O)O ZINC000147459543 CD For-Sale Anodyne CXCL8 50 38 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@@H]1CCCBr ZINC000147459570 FI For-Sale Reactive CACNA1B 53 35 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@@H]1CCCBr ZINC000147459570 FI For-Sale Reactive PREP 31 41 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@@H]1CCCBr ZINC000147459570 FI For-Sale Reactive CCR2 62 43 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@@H]1CCCBr ZINC000147459570 FI For-Sale Reactive SFRP1 51 34 CCN(CC)[C@@H](C)CNC(=O)CNC(=O)c1cccc(Br)c1 ZINC000147459589 FE On-Demand Anodyne CCR2 38 42 NC(=O)[C@@H](N)COCc1ccccc1Br ZINC000147459603 CC For-Sale Anodyne CACNA2D1 0 47 Nc1ccc(C(=O)Nc2ccncc2Br)cc1F ZINC000147459620 DF For-Sale Anodyne ROCK1 25 41 Nc1ccc(C(=O)Nc2ccncc2Br)cc1F ZINC000147459620 DF For-Sale Anodyne ROCK2 45 44 Nc1ccc(C(=O)Nc2ccncc2Br)cc1F ZINC000147459620 DF For-Sale Anodyne HDAC1 41 45 Nc1ccc(C(=O)Nc2ccncc2Br)cc1F ZINC000147459620 DF For-Sale Anodyne HDAC2 20 42 CCc1ccccc1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147459668 HG On-Demand Anodyne ADRB2 23 44 CCc1ccccc1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147459668 HG On-Demand Anodyne ADRB1 56 38 CCc1ccccc1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147459668 HG On-Demand Anodyne CXCL8 53 34 CCc1ccccc1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147459668 HG On-Demand Anodyne PDS 15 46 CCOC(=O)Cc1csc(Cc2cccnc2)n1 ZINC000147459686 CE For-Sale Anodyne TBXAS1 18 40 CC(C)C[C@H](N)C(=O)NN1[C@H](C)CCC[C@H]1C ZINC000147459693 BD For-Sale Anodyne AMPX_VIBPR 0 47 NC1(C(=O)Nc2ccc(C(F)(F)F)cc2)CCC1 ZINC000147459694 CF On-Demand Anodyne DHODH 35 42 NC1(C(=O)Nc2ccc(C(F)(F)F)cc2)CCC1 ZINC000147459694 CF On-Demand Anodyne KIF11 0 51 CC(C)CCO[C@@H](C)C(=O)N1CCc2sccc2[C@H]1C ZINC000147459699 CH On-Demand Anodyne TRPM8 16 40 Cc1noc(C(C)C)c1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147459729 HF On-Demand Anodyne HTR4 62 39 Cc1noc(C(C)C)c1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147459729 HF On-Demand Anodyne TGM2 54 42 Cc1noc(C(C)C)c1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147459729 HF On-Demand Anodyne CACNA1I 49 33 Cc1noc(C(C)C)c1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147459729 HF On-Demand Anodyne F13A1 46 42 CC[C@H](NC(=O)NCc1cccc2cccnc12)C(=O)O ZINC000147459731 CD On-Demand Anodyne ANPEP 18 45 CC[C@H](NC(=O)NCc1cccc2cccnc12)C(=O)O ZINC000147459731 CD On-Demand Anodyne ACE2 49 39 CC[C@H](C)NC(=O)CNc1ccc(Br)c(OC)c1 ZINC000147459743 DF On-Demand Anodyne ENPP1 50 31 C[C@@H](CNc1cccc(Cl)c1C(N)=O)CC(=O)O ZINC000147459749 CD For-Sale Anodyne CXCL8 50 38 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne RARA 16 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne PPIA 18 49 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne CPT1A 37 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne PRNP 28 49 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne NR1H4 15 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne TAAR1 23 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne AKR1C3 28 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne PTPA 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne HCAR1 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne GPR35 47 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne SENP1 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2)c1 ZINC000147459761 FI On-Demand Anodyne KCNK3 63 47 CCCCc1ccc(Oc2cc(Cl)c(Cl)cc2N)cc1 ZINC000147459783 DK For-Sale Anodyne INHA 95 42 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@H]1CCCBr ZINC000147459796 FI For-Sale Reactive CACNA1B 53 35 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@H]1CCCBr ZINC000147459796 FI For-Sale Reactive PREP 31 41 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@H]1CCCBr ZINC000147459796 FI For-Sale Reactive CCR2 62 43 O=C(c1cccc(C(F)(F)F)c1)N1CCC[C@H]1CCCBr ZINC000147459796 FI For-Sale Reactive SFRP1 51 34 CCN(CC)[C@H](C)CNC(=O)CNC(=O)c1cccc(Br)c1 ZINC000147459818 FE On-Demand Anodyne CCR2 41 42 NC(=O)[C@H](N)COCc1ccccc1Br ZINC000147459837 CC For-Sale Anodyne CACNA2D1 0 47 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c(F)c1 ZINC000147459872 HF On-Demand Anodyne ADRB2 17 41 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c(F)c1 ZINC000147459872 HF On-Demand Anodyne ADRB1 47 37 NCC1(CC(=O)Nc2ccc(C(F)(F)F)cc2)CCC1 ZINC000147459892 CG For-Sale Anodyne DHODH 32 40 NCC1(CC(=O)Nc2ccc(C(F)(F)F)cc2)CCC1 ZINC000147459892 CG For-Sale Anodyne TRPV1 15 42 NCC1(CC(=O)Nc2ccc(C(F)(F)F)cc2)CCC1 ZINC000147459892 CG For-Sale Anodyne EPHX2 29 40 NCC1(CC(=O)Nc2ccc(C(F)(F)F)cc2)CCC1 ZINC000147459892 CG For-Sale Anodyne SLC1A2 39 40 CC(C)CCO[C@@H](C)C(=O)N1CCc2sccc2[C@@H]1C ZINC000147459909 CH On-Demand Anodyne TRPM8 16 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCC2 ZINC000147459928 HG On-Demand Anodyne NPY2R 57 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCC2 ZINC000147459928 HG On-Demand Anodyne NPY5R 20 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCC2 ZINC000147459928 HG On-Demand Anodyne EPHX2 17 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCC2 ZINC000147459928 HG On-Demand Anodyne TGM2 59 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCC2 ZINC000147459928 HG On-Demand Anodyne CACNA1I 55 33 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCC2 ZINC000147459928 HG On-Demand Anodyne F13A1 42 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCC2 ZINC000147459928 HG On-Demand Anodyne AKR1C3 58 36 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2c(s1)CCC2 ZINC000147459928 HG On-Demand Anodyne NAMPT 31 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NCc3ccccc3)cc1)C2 ZINC000147459971 HH On-Demand Anodyne TSHR 40 30 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NCc3ccccc3)cc1)C2 ZINC000147459971 HH On-Demand Anodyne MMP13 27 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NCc3ccccc3)cc1)C2 ZINC000147459971 HH On-Demand Anodyne HDAC8 21 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NCc3ccccc3)cc1)C2 ZINC000147459971 HH On-Demand Anodyne MTNR1A 36 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NCc3ccccc3)cc1)C2 ZINC000147459971 HH On-Demand Anodyne MTNR1B 37 41 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NCc3ccccc3)cc1)C2 ZINC000147459971 HH On-Demand Anodyne ROCK2 55 49 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C(=O)NCc3ccccc3)cc1)C2 ZINC000147459971 HH On-Demand Anodyne NOD2 39 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne PPIA 18 48 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne TBXAS1 51 37 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne PRNP 17 45 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne GRM5 15 53 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne SCN10A 48 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne CSF1R 24 54 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne IKBKG 0 49 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne TAAR1 17 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne AKR1C3 30 44 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne SHH 25 52 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne NAMPT 26 52 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne KCNK3 77 46 O=C(O)c1cc(Cl)cc(NC(=O)c2cccnc2)c1 ZINC000147459985 CF On-Demand Anodyne KCNK9 28 40 O=C(NC[C@@H]1CCCOC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147459987 DF On-Demand Anodyne CACNA1I 70 40 COc1cc(NCC(=O)NC2CCCCCC2)ccc1Br ZINC000147459996 FH On-Demand Anodyne EPHX2 25 44 COc1cc(NCC(=O)NC2CCCCCC2)ccc1Br ZINC000147459996 FH On-Demand Anodyne ENPP1 49 30 CC(C)CCCCNC[C@H](O)COCc1ccccc1Cl ZINC000147460096 DH For-Sale Anodyne GRIN1 16 43 N#Cc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147460110 HE On-Demand Mild ADRB2 19 42 N#Cc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147460110 HE On-Demand Mild ADRB1 63 42 NCC1(CC(=O)NC2CCCCCCC2)CCC1 ZINC000147460120 CF For-Sale Anodyne CACNA2D1 61 49 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1CCS(=O)(=O)C1 ZINC000147460121 HC On-Demand Anodyne EPHX2 31 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1CCS(=O)(=O)C1 ZINC000147460121 HC On-Demand Anodyne TGM2 75 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1CCS(=O)(=O)C1 ZINC000147460121 HC On-Demand Anodyne F13A1 80 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1CCS(=O)(=O)C1 ZINC000147460121 HC On-Demand Anodyne NAMPT 36 41 CC(C)(C)c1ccc(C(=O)c2cncs2)cc1 ZINC000147460138 BH For-Sale Anodyne MAP3K5 43 33 CN1CCN(c2ncnc3cc(Br)ccc23)CC1 ZINC000147460146 DE On-Demand Anodyne PDE3A 44 33 CN1CCN(c2ncnc3cc(Br)ccc23)CC1 ZINC000147460146 DE On-Demand Anodyne PDGFRB 64 46 CN1CCN(c2ncnc3cc(Br)ccc23)CC1 ZINC000147460146 DE On-Demand Anodyne HRH4 35 63 CN1CCN(c2ncnc3cc(Br)ccc23)CC1 ZINC000147460146 DE On-Demand Anodyne AKT2 16 41 CN1CCN(c2ncnc3cc(Br)ccc23)CC1 ZINC000147460146 DE On-Demand Anodyne AKT3 18 41 CN1CCN(c2ncnc3cc(Br)ccc23)CC1 ZINC000147460146 DE On-Demand Anodyne PDE3B 66 34 CC(C)NC(=O)N1CC(NC(=O)[C@@H]2N[C@H](CC(C)(C)C)[C@]3(C(=O)Nc4cc(Cl)ccc43)[C@H]2c2cccc(Cl)c2F)C1 ZINC000147460184 KJ Annotated Anodyne MDM2 101 68 O=C(NC[C@H]1CCCOC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147460187 DF On-Demand Anodyne CACNA1I 70 40 CCN(C)C(=O)CNc1ccc(Br)c(OC)c1 ZINC000147460206 DE On-Demand Anodyne DRTS_TRYCR 44 32 O=C([C@H]1CCCc2ccccc21)N1CCC[C@@H]1CCCBr ZINC000147460208 FI For-Sale Reactive PREP 48 35 O=C([C@H]1CCCc2ccccc21)N1CCC[C@@H]1CCCBr ZINC000147460208 FI For-Sale Reactive HTR3B 0 40 CCOCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147460212 CE On-Demand Anodyne HCAR1 0 44 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(-c2ccnc(C)n2)c1 ZINC000147460216 EF On-Demand Anodyne ABL1 15 42 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(-c2ccnc(C)n2)c1 ZINC000147460216 EF On-Demand Anodyne HDAC10 49 35 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(-c2ccnc(C)n2)c1 ZINC000147460216 EF On-Demand Anodyne MTNN 18 40 CC[C@@]12CCCC[C@@H](Cc3ccc(O)cc31)[C@H]2N ZINC000147460237 BG For-Sale Anodyne OPRM1 24 65 CC[C@@]12CCCC[C@@H](Cc3ccc(O)cc31)[C@H]2N ZINC000147460237 BG For-Sale Anodyne OPRK1 23 47 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(C(=O)N3CCCC3)cc2)C1 ZINC000147460239 HE On-Demand Anodyne EPHX2 19 46 C[C@@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(C(=O)N3CCCC3)cc2)C1 ZINC000147460239 HE On-Demand Anodyne L3MBTL3 68 39 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CASP3 17 45 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne KLK3 76 38 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CTSB 64 46 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne PAPA1_CARPA 64 40 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CYSP_TRYCR 61 44 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CTSK 42 43 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CTSL 47 43 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne PGA 23 45 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CAPNS1 67 38 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne MMP11 54 31 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CTSS 18 40 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CAPN1 77 44 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CASP1 22 44 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CAPN2 119 46 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CASP6 23 41 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne CASP9 29 41 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne NPR 68 35 O=C(N[C@@H](CSc1ccccc1)[C@@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460240 IK For-Sale Anodyne PSMB5 33 44 COCCOc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1F ZINC000147460241 FI On-Demand Anodyne KDR 15 41 COCCOc1ccc(NC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)cc1F ZINC000147460241 FI On-Demand Anodyne MET 60 39 CC(C)CCCCNC[C@@H](O)COCc1ccccc1Cl ZINC000147460308 DH For-Sale Anodyne GRIN1 16 43 CC(C)CCCCNC[C@@H](O)COCc1ccccc1Cl ZINC000147460308 DH For-Sale Anodyne ADRB3 20 40 C[C@H](CCI)NC(=O)OC(C)(C)C ZINC000147460334 CF For-Sale Reactive PAPA1_CARPA 46 42 C[C@H](CCI)NC(=O)OC(C)(C)C ZINC000147460334 CF For-Sale Reactive CTSK 25 49 C[C@H](CCI)NC(=O)OC(C)(C)C ZINC000147460334 CF For-Sale Reactive PGA5 45 40 CCc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147460340 HG On-Demand Anodyne ADRB2 27 45 CCc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147460340 HG On-Demand Anodyne ADRB1 61 35 CCc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147460340 HG On-Demand Anodyne ADRB3 24 45 CCc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147460340 HG On-Demand Anodyne PDS 26 47 NS(=O)(=O)c1cc(Br)c(OCCn2ccnc2)cc1F ZINC000147460352 FD For-Sale Anodyne TBXAS1 29 42 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA2 167 59 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA6 33 44 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA1 143 59 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA7 96 56 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA13 42 44 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA5B 61 55 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA4 112 59 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA5A 65 55 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA14 73 56 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA12 106 53 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA9 117 55 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CAH_METTE 36 44 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CYNT 47 51 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne NCE103 39 44 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne CA15 27 44 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne MTCA1 51 52 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne P96878_MYCTU 65 52 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne NAMPT 69 38 NC1(C(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460377 CB On-Demand Anodyne A6YCJ1_9METZ 34 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne DRD3 15 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne HTR4 52 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne GRIN2B 50 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne CYP51A1 24 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne PYGL 72 39 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne PLD1 37 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne EPHX2 15 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne PLD2 35 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne TGM2 59 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne CACNA1I 57 33 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne F13A1 55 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne AKR1C3 32 49 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc2ccccc2[nH]1 ZINC000147460401 GF On-Demand Anodyne NAMPT 43 48 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)o2)c1 ZINC000147460414 EH On-Demand Anodyne PPIA 15 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)o2)c1 ZINC000147460414 EH On-Demand Anodyne SCN10A 21 41 O=C([C@@H]1CCCc2ccccc21)N1CCC[C@@H]1CCCBr ZINC000147460421 FI For-Sale Reactive PREP 48 35 O=C([C@@H]1CCCc2ccccc21)N1CCC[C@@H]1CCCBr ZINC000147460421 FI For-Sale Reactive HTR3B 0 40 O=C(c1cncs1)c1cccc2ccccc12 ZINC000147460426 BH For-Sale Anodyne CNR1 0 40 COCCOc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1F ZINC000147460438 FI On-Demand Anodyne KDR 15 41 COCCOc1ccc(NC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)cc1F ZINC000147460438 FI On-Demand Anodyne MET 60 39 CC[C@@H]1CN(CCc2ccc(OC)cc2)CC[C@@H]1N ZINC000147460449 CE On-Demand Anodyne SIGMAR1 28 57 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CASP3 17 45 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne KLK3 76 38 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CTSB 64 46 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne PAPA1_CARPA 64 40 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CYSP_TRYCR 61 44 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CTSK 42 43 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CTSL 47 43 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne PGA 23 45 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CAPNS1 67 38 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne MMP11 54 31 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CTSS 18 40 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CAPN1 77 44 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CASP1 22 44 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CAPN2 119 46 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CASP6 23 41 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne CASP9 29 41 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne NPR 68 35 O=C(N[C@@H](CSc1ccccc1)[C@H](O)CSc1ccccc1)OCc1ccccc1 ZINC000147460454 IK For-Sale Anodyne PSMB5 33 44 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(C(=O)N3CCCC3)cc2)C1 ZINC000147460467 HE On-Demand Anodyne EPHX2 19 46 C[C@H]1CCCN(C(C)(C)CNC(=O)C(=O)Nc2ccc(C(=O)N3CCCC3)cc2)C1 ZINC000147460467 HE On-Demand Anodyne L3MBTL3 68 39 COc1cc(NCC(=O)Nc2ccc(Br)cc2)ccc1Br ZINC000147460509 HI On-Demand Anodyne HTR2A 17 44 COc1cc(NCC(=O)Nc2ccc(Br)cc2)ccc1Br ZINC000147460509 HI On-Demand Anodyne FPR2 21 42 COc1cc(NCC(=O)Nc2ccc(Br)cc2)ccc1Br ZINC000147460509 HI On-Demand Anodyne ENPP1 77 40 Cc1ccc(F)c(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147460568 HF On-Demand Anodyne ADRB2 18 41 Cc1ccc(F)c(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147460568 HF On-Demand Anodyne ADRB1 47 37 CCOC[C@H](C)NC(=O)Nc1cc(NC(=O)Nc2ccccc2)ccc1C ZINC000147460581 FI On-Demand Anodyne LPL 47 37 CCOC[C@H](C)NC(=O)Nc1cc(NC(=O)Nc2ccccc2)ccc1C ZINC000147460581 FI On-Demand Anodyne CA1 47 38 CCOC[C@H](C)NC(=O)Nc1cc(NC(=O)Nc2ccccc2)ccc1C ZINC000147460581 FI On-Demand Anodyne PYGL 22 43 CN[C@H](C)C(=O)NN1[C@@H](C)CCC[C@H]1C ZINC000147460585 BC For-Sale Anodyne BIRC2 45 33 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA2 132 63 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA6 24 40 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA1 110 56 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA7 67 56 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA13 26 41 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA5B 58 56 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA4 97 63 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA5A 61 56 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA14 58 50 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA12 80 54 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne TPSAB1 15 41 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA9 84 56 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CAH_METTE 25 41 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CYNT 34 46 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne NCE103 35 41 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA15 16 41 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne MTCA1 40 47 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne P96878_MYCTU 50 47 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne CA 0 41 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne NAMPT 43 34 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne A6YCJ1_9METZ 24 41 NCC1(CC(=O)NCc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147460610 DC For-Sale Anodyne Q5TU56_ANOGA 0 40 O=C([C@H]1CCCc2ccccc21)N1CCC[C@H]1CCCBr ZINC000147460620 FI For-Sale Reactive PREP 48 35 O=C([C@H]1CCCc2ccccc21)N1CCC[C@H]1CCCBr ZINC000147460620 FI For-Sale Reactive HTR3B 0 40 CC[C@H](NC(=O)Nc1c(C)cc(C)cc1Br)C(=O)O ZINC000147460644 EG For-Sale Anodyne PYGL 42 43 CC[C@H]1CN(CCc2ccc(OC)cc2)CC[C@@H]1N ZINC000147460646 CE On-Demand Anodyne SIGMAR1 28 57 COCCOc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1F ZINC000147460660 FI On-Demand Anodyne KDR 15 41 COCCOc1ccc(NC(=O)[C@H]2C[C@H]2c2cccc(Cl)c2)cc1F ZINC000147460660 FI On-Demand Anodyne MET 60 39 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne FKBP1A 24 43 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne GRIN2B 37 47 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne TBXAS1 49 42 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne PTAFR 27 40 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne KCNA5 15 42 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne MMP13 16 41 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne CHRNA7 51 44 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne C3AR1 49 43 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne MMP9 15 41 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne TGM2 90 48 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne MMP7 17 41 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne CYP2C9 16 48 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne MMP1 15 41 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne F13A1 96 48 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne ACHP_LYMST 25 44 O=C(CCc1cccnc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460664 GE On-Demand Anodyne NAMPT 113 53 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)nc2)c1 ZINC000147460666 DG On-Demand Anodyne JUN 23 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)nc2)c1 ZINC000147460666 DG On-Demand Anodyne ATF1 57 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)nc2)c1 ZINC000147460666 DG On-Demand Anodyne CPT1A 34 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)nc2)c1 ZINC000147460666 DG On-Demand Anodyne NFKB1 53 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)nc2)c1 ZINC000147460666 DG On-Demand Anodyne P4HTM 0 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)nc2)c1 ZINC000147460666 DG On-Demand Anodyne KCNK3 44 40 Cc1cc(N2CCOCC2)ccc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@H](C)C1 ZINC000147460692 HE On-Demand Anodyne HRH3 27 46 Nc1ccc(CC(=O)Nc2ccncc2Br)cc1 ZINC000147460699 DF For-Sale Clean CA2 15 43 Nc1ccc(CC(=O)Nc2ccncc2Br)cc1 ZINC000147460699 DF For-Sale Clean CA7 16 42 Nc1ccc(CC(=O)Nc2ccncc2Br)cc1 ZINC000147460699 DF For-Sale Clean CA5B 47 42 Nc1ccc(CC(=O)Nc2ccncc2Br)cc1 ZINC000147460699 DF For-Sale Clean CA5A 53 42 Nc1ccc(CC(=O)Nc2ccncc2Br)cc1 ZINC000147460699 DF For-Sale Clean CA9 28 41 COc1cc(OCC(=O)NCc2ccc(OC(F)(F)F)cc2)ccc1[N+](=O)[O-] ZINC000147460739 HG On-Demand Bother CSNK1D 17 41 COCc1nc(C(=O)Nc2ccc(OC)c(Cc3ccccc3)c2)cs1 ZINC000147460741 FI On-Demand Anodyne TSHR 71 37 COCc1nc(C(=O)Nc2ccc(OC)c(Cc3ccccc3)c2)cs1 ZINC000147460741 FI On-Demand Anodyne PTGER1 37 47 COCc1nc(C(=O)Nc2ccc(OC)c(Cc3ccccc3)c2)cs1 ZINC000147460741 FI On-Demand Anodyne CPT1A 43 30 COCc1nc(C(=O)Nc2ccc(OC)c(Cc3ccccc3)c2)cs1 ZINC000147460741 FI On-Demand Anodyne GRM4 30 44 COCc1nc(C(=O)Nc2ccc(OC)c(Cc3ccccc3)c2)cs1 ZINC000147460741 FI On-Demand Anodyne QRFPR 40 34 COCc1nc(C(=O)Nc2ccc(OC)c(Cc3ccccc3)c2)cs1 ZINC000147460741 FI On-Demand Anodyne ENPP1 69 33 COc1ccc(OCCNc2ccc(Br)c(OC)c2)cc1 ZINC000147460750 FH On-Demand Anodyne UTS2R 0 41 COc1ccc(OCCNc2ccc(Br)c(OC)c2)cc1 ZINC000147460750 FH On-Demand Anodyne DRTS_TRYCR 45 33 CCCOc1ccc(C(=O)c2cncs2)cc1 ZINC000147460762 BG For-Sale Anodyne PLA2G4B 78 38 NS(=O)(=O)c1cc(Br)c(OCCCn2ccnc2)cc1F ZINC000147460775 GD For-Sale Anodyne TBXAS1 38 40 NS(=O)(=O)c1cc(Br)c(OCCCn2ccnc2)cc1F ZINC000147460775 GD For-Sale Anodyne HMOX2 41 42 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147460792 HK On-Demand Anodyne LPL 61 38 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147460792 HK On-Demand Anodyne CCKBR 45 39 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147460792 HK On-Demand Anodyne EPHX2 42 58 CN[C@H](C)C(=O)NN1[C@@H](C)CCC[C@@H]1C ZINC000147460793 BC For-Sale Anodyne BIRC2 45 33 Cc1cc(C)cc(NC(=O)C(=O)NC[C@@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147460823 HG On-Demand Anodyne ADRB2 27 47 Cc1cc(C)cc(NC(=O)C(=O)NC[C@@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147460823 HG On-Demand Anodyne ADRB1 60 35 O=C([C@@H]1CCCc2ccccc21)N1CCC[C@H]1CCCBr ZINC000147460826 FI For-Sale Reactive PREP 48 35 O=C([C@@H]1CCCc2ccccc21)N1CCC[C@H]1CCCBr ZINC000147460826 FI For-Sale Reactive HTR3B 0 40 CC[C@H](NC(=O)NC[C@@H](C)N1CCCC1)C(=O)O ZINC000147460830 CC For-Sale Anodyne RIR1_HHV11 52 37 COc1ccc(OC)c(NC(=O)C2(N)CCC2)c1 ZINC000147460848 CD For-Sale Anodyne CYP1B1 37 42 COc1ccc(OC)c(NC(=O)C2(N)CCC2)c1 ZINC000147460848 CD For-Sale Anodyne AKR1C2 51 37 COCCOc1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1F ZINC000147460871 GG On-Demand Anodyne ROCK2 34 49 COCCOc1ccc(NC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1F ZINC000147460871 GG On-Demand Anodyne MET 40 35 O=C(Cc1ccc(Br)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147460881 FH On-Demand Anodyne PFK 0 41 COc1ccc(C)cc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460882 HF On-Demand Anodyne TSHR 47 31 COc1ccc(C)cc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460882 HF On-Demand Anodyne DRD4 22 44 COc1ccc(C)cc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460882 HF On-Demand Anodyne DRD3 23 41 COc1ccc(C)cc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460882 HF On-Demand Anodyne HTR4 37 40 COc1ccc(C)cc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460882 HF On-Demand Anodyne EPHX2 35 42 COc1ccc(C)cc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460882 HF On-Demand Anodyne TGM2 64 47 COc1ccc(C)cc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460882 HF On-Demand Anodyne CACNA1I 57 37 COc1ccc(C)cc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460882 HF On-Demand Anodyne F13A1 64 41 COc1ccc(C)cc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147460882 HF On-Demand Anodyne ACKR3 63 35 Cc1cc(N2CCOCC2)ccc1NC(=O)C(=O)NCC(C)(C)N1CCC[C@@H](C)C1 ZINC000147460917 HE On-Demand Anodyne HRH3 27 46 CN[C@H](C)C(=O)NN1[C@H](C)CCC[C@H]1C ZINC000147460987 BC For-Sale Anodyne BIRC2 45 33 CCC[C@@H](C)NC(=O)CNc1ccc(Br)c(OC)c1 ZINC000147460993 EG For-Sale Anodyne ENPP1 60 32 CC(=O)Nc1cccc(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147460997 CF For-Sale Anodyne CSNK2A1 32 46 CC(=O)Nc1cccc(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147460997 CF For-Sale Anodyne SORT1 27 41 CC(=O)Nc1cccc(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147460997 CF For-Sale Anodyne MAPK8 16 43 CC(=O)Nc1cccc(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147460997 CF For-Sale Anodyne AKR1C3 58 44 CC(=O)Nc1cccc(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147460997 CF For-Sale Anodyne AKR1C2 75 43 CC(=O)Nc1cccc(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147460997 CF For-Sale Anodyne RHOA 0 42 CC(=O)Nc1cccc(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147460997 CF For-Sale Anodyne KCNK3 109 39 CC(=O)Nc1cccc(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147460997 CF For-Sale Anodyne KCNK9 73 38 CC(C)(C)C[C@H]1N[C@@H](C(=O)N[C@H]2CC[C@@H](O)C2)[C@H](c2cccc(Cl)c2F)[C@@]12C(=O)Nc1cc(Cl)ccc12 ZINC000147461002 KJ Annotated Anodyne MDM2 66 60 Cc1nn(C(F)F)c(C)c1CC(=O)NCc1ccc(N(C)C)nc1 ZINC000147461003 EE On-Demand Anodyne P2RX7 59 48 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147461029 HK On-Demand Anodyne LPL 61 38 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147461029 HK On-Demand Anodyne CCKBR 45 39 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147461029 HK On-Demand Anodyne EPHX2 42 58 CC[C@H](NC(=O)NC[C@H](C)N1CCCC1)C(=O)O ZINC000147461033 CC For-Sale Anodyne RIR1_HHV11 52 37 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1cc(F)cc(F)c1 ZINC000147461043 HF On-Demand Anodyne ADRB2 20 42 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1cc(F)cc(F)c1 ZINC000147461043 HF On-Demand Anodyne ADRB1 63 39 COc1ccc(OC)c(NC(=O)CC2(CN)CCC2)c1 ZINC000147461060 CE For-Sale Anodyne MTNR1A 66 41 COc1ccc(OC)c(NC(=O)CC2(CN)CCC2)c1 ZINC000147461060 CE For-Sale Anodyne MTNR1B 59 41 COc1ccc(OC)c(NC(=O)CC2(CN)CCC2)c1 ZINC000147461060 CE For-Sale Anodyne AKR1C2 40 33 COCCOc1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1F ZINC000147461098 GG On-Demand Anodyne ROCK2 34 49 COCCOc1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1F ZINC000147461098 GG On-Demand Anodyne MET 40 35 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne PPIA 18 52 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne KCNJ11 31 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne ECR 16 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne CPT1A 41 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne PPARD 0 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne GRM5 22 66 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne FABH 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne LUCI_LUCLA 24 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne TAAR1 36 46 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne AKR1C3 40 49 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne SENP1 0 51 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne KCNK3 110 61 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2)c1 ZINC000147461107 CG On-Demand Anodyne KCNK9 54 53 N#Cc1ccc(NC(=O)c2csc(I)c2)c(N)c1 ZINC000147461142 FG For-Sale Mild HDAC1 25 43 CNCc1cc(COc2ccc(Cl)c(F)c2)c(C)o1 ZINC000147461166 CH For-Sale Anodyne PTGER4 0 41 CCC[C@H](C)NC(=O)CNc1ccc(Br)c(OC)c1 ZINC000147461187 EG For-Sale Anodyne ENPP1 60 32 CC(C)n1c2ccccc2c2ccc(C(=O)O)cc21 ZINC000147461188 CI For-Sale Anodyne NPY2R 16 52 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147461236 HK On-Demand Anodyne LPL 61 38 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147461236 HK On-Demand Anodyne CCKBR 45 39 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147461236 HK On-Demand Anodyne EPHX2 42 58 Cc1cc(F)ccc1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147461241 HF On-Demand Anodyne ADRB2 18 42 Cc1cc(F)ccc1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147461241 HF On-Demand Anodyne ADRB1 55 35 O=C(O)c1ccc(COCc2ccccc2Br)cc1 ZINC000147461259 DH For-Sale Anodyne SRD5A2 31 44 O=C(O)c1ccc(COCc2ccccc2Br)cc1 ZINC000147461259 DH For-Sale Anodyne FOLH1 16 43 O=C(O)c1ccc(COCc2ccccc2Br)cc1 ZINC000147461259 DH For-Sale Anodyne PTGER1 20 48 CC[C@H](NC(=O)Nc1ccc(C)nc1)C(=O)O ZINC000147461267 BD On-Demand Anodyne ACE2 43 31 C[C@@H](N)C(=O)NCCc1ccc(O)c(O)c1 ZINC000147461311 BC For-Sale Clean NCE103 37 40 C[C@@H](N)C(=O)NCCc1ccc(O)c(O)c1 ZINC000147461311 BC For-Sale Clean P96878_MYCTU 18 40 Cc1cnc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147461322 CE On-Demand Anodyne JUN 23 45 Cc1cnc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147461322 CE On-Demand Anodyne ATF1 58 40 Cc1cnc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147461322 CE On-Demand Anodyne NFKB1 53 40 Cc1cnc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147461322 CE On-Demand Anodyne P4HTM 0 40 Cc1occc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147461329 FE On-Demand Anodyne HTR4 63 38 Cc1occc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147461329 FE On-Demand Anodyne LPL 45 35 Cc1occc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147461329 FE On-Demand Anodyne EPHX2 23 42 Cc1occc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147461329 FE On-Demand Anodyne TGM2 67 46 Cc1occc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147461329 FE On-Demand Anodyne CACNA1I 58 35 Cc1occc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147461329 FE On-Demand Anodyne F13A1 68 46 Nc1cc(C(=O)Nc2ccncc2Br)ccc1Br ZINC000147461374 FG For-Sale Anodyne HDAC1 31 44 Nc1cc(C(=O)Nc2ccncc2Br)ccc1Br ZINC000147461374 FG For-Sale Anodyne HDAC2 17 42 Nc1cc(C(=O)Nc2ccncc2Br)ccc1Br ZINC000147461374 FG For-Sale Anodyne HDAC3 0 45 COc1cc(-c2nc(-c3ccc(O)cc3)no2)ccc1F ZINC000147461378 CG On-Demand Anodyne LUCI_PHOPE 42 48 NC(=O)NCCNC(=O)c1cc(N)nc2ccccc12 ZINC000147461389 CC For-Sale Anodyne BCHE 47 38 NC(=O)NCCNC(=O)c1cc(N)nc2ccccc12 ZINC000147461389 CC For-Sale Anodyne ACACB 26 43 NC(=O)NCCNC(=O)c1cc(N)nc2ccccc12 ZINC000147461389 CC For-Sale Anodyne TACR3 36 49 NC(=O)NCCNC(=O)c1cc(N)nc2ccccc12 ZINC000147461389 CC For-Sale Anodyne POLR1A 53 33 CCNCc1cc(COc2ccc(Cl)c(F)c2)c(C)o1 ZINC000147461393 CI For-Sale Anodyne PTGER4 0 42 COc1cc(NCC(=O)Nc2ccccc2Cl)ccc1Br ZINC000147461409 FI On-Demand Anodyne GRM4 30 40 COc1cc(NCC(=O)Nc2ccccc2Cl)ccc1Br ZINC000147461409 FI On-Demand Anodyne EPHB3 36 40 COc1cc(NCC(=O)Nc2ccccc2Cl)ccc1Br ZINC000147461409 FI On-Demand Anodyne ENPP1 62 33 O=C(c1ccccc1[N+](=O)[O-])N1CCC[C@@H]1CCCBr ZINC000147461410 EG For-Sale Reactive HCRTR1 16 44 O=C(c1ccccc1[N+](=O)[O-])N1CCC[C@@H]1CCCBr ZINC000147461410 EG For-Sale Reactive PREP 41 36 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147461444 HK On-Demand Anodyne LPL 61 38 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147461444 HK On-Demand Anodyne CCKBR 45 39 Cc1ccc(NC(=O)Nc2ccccc2)cc1NC(=O)N[C@H]1C[C@H]1c1ccccc1 ZINC000147461444 HK On-Demand Anodyne EPHX2 42 58 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461454 ED On-Demand Anodyne F10 19 40 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461454 ED On-Demand Anodyne KLK3 48 37 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461454 ED On-Demand Anodyne CTSK 17 44 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461454 ED On-Demand Anodyne NPFFR2 41 37 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461454 ED On-Demand Anodyne GRIA1 55 33 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461454 ED On-Demand Anodyne PCSK5 61 40 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461454 ED On-Demand Anodyne FURIN 70 42 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461454 ED On-Demand Anodyne CTSS 15 44 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461454 ED On-Demand Anodyne POLG_WNV 78 36 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461454 ED On-Demand Anodyne QRFPR 45 39 CCCC[C@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461454 ED On-Demand Anodyne NPFFR1 55 37 N#Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1 ZINC000147461494 HE On-Demand Mild ADRB2 22 43 N#Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1 ZINC000147461494 HE On-Demand Mild ADRB1 70 43 N#Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1 ZINC000147461494 HE On-Demand Mild ADRB3 19 41 CN(C)C(=O)CCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147461510 DD On-Demand Anodyne CACNA1H 24 41 O=C(O)c1ccccc1OCCOCc1ccccc1Br ZINC000147461520 FH For-Sale Anodyne FOLH1 15 40 Oc1ccc(CNn2cnnc2)cc1 ZINC000147461535 AC For-Sale Anodyne H9TVJ1_CHISP 43 34 Cc1noc(C)c1CCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147461548 HE On-Demand Anodyne TGM2 63 40 Cc1noc(C)c1CCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147461548 HE On-Demand Anodyne ADAMTS4 41 40 Cc1noc(C)c1CCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147461548 HE On-Demand Anodyne ADAMTS5 15 40 Cc1noc(C)c1CCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147461548 HE On-Demand Anodyne F13A1 62 40 CC(C)=CC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147461549 CF On-Demand Anodyne HCAR1 0 43 CC(C)=CC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147461549 CF On-Demand Anodyne PARP15 0 40 O=C(c1ccccc1[N+](=O)[O-])N1CCC[C@H]1CCCBr ZINC000147461611 EG For-Sale Reactive HCRTR1 16 44 O=C(c1ccccc1[N+](=O)[O-])N1CCC[C@H]1CCCBr ZINC000147461611 EG For-Sale Reactive PREP 41 36 COc1cc(NCC(=O)Nc2ccccc2F)ccc1Br ZINC000147461645 FH On-Demand Anodyne HTR2A 16 48 COc1cc(NCC(=O)Nc2ccccc2F)ccc1Br ZINC000147461645 FH On-Demand Anodyne GRM4 16 40 COc1cc(NCC(=O)Nc2ccccc2F)ccc1Br ZINC000147461645 FH On-Demand Anodyne PDGFRA 15 40 COc1cc(NCC(=O)Nc2ccccc2F)ccc1Br ZINC000147461645 FH On-Demand Anodyne ENPP1 55 32 COc1cc(NCC(=O)Nc2ccccc2F)ccc1Br ZINC000147461645 FH On-Demand Anodyne GLMU 0 42 CCOC(=O)[C@@H](Br)c1cccnc1 ZINC000147461652 BE For-Sale Reactive TBXAS1 24 41 CCOC(=O)[C@@H](Br)c1cccnc1 ZINC000147461652 BE For-Sale Reactive KCNA5 26 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461655 ED On-Demand Anodyne F10 19 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461655 ED On-Demand Anodyne KLK3 48 37 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461655 ED On-Demand Anodyne CTSK 17 44 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461655 ED On-Demand Anodyne NPFFR2 41 37 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461655 ED On-Demand Anodyne GRIA1 55 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461655 ED On-Demand Anodyne PCSK5 61 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461655 ED On-Demand Anodyne FURIN 70 42 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461655 ED On-Demand Anodyne CTSS 15 44 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461655 ED On-Demand Anodyne POLG_WNV 78 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461655 ED On-Demand Anodyne QRFPR 45 39 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccc(C(=O)N(C)C)c1 ZINC000147461655 ED On-Demand Anodyne NPFFR1 55 37 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccc(F)cc1F ZINC000147461721 HF On-Demand Anodyne ADRB2 15 41 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccc(F)cc1F ZINC000147461721 HF On-Demand Anodyne ADRB1 56 39 COc1cc(OC)c(NC(=O)C2(N)CCC2)cc1Cl ZINC000147461722 CE For-Sale Anodyne HTR4 39 43 COc1cc(OCC(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)ccc1[N+](=O)[O-] ZINC000147461751 HI On-Demand Bother GYRB 43 35 COc1cc(OCC(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)ccc1[N+](=O)[O-] ZINC000147461751 HI On-Demand Bother CETP 83 59 COc1cc(OCC(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)ccc1[N+](=O)[O-] ZINC000147461751 HI On-Demand Bother FASN 20 40 COc1cc(OCC(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)ccc1[N+](=O)[O-] ZINC000147461751 HI On-Demand Bother AGPAT2 23 40 COc1cc(OCC(=O)Nc2ccc(-c3nc4ccccc4o3)cc2)ccc1[N+](=O)[O-] ZINC000147461751 HI On-Demand Bother IMDH_CRYPV 48 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne AVPR2 20 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne PPIA 17 49 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne ECR 44 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne ATF1 48 38 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne NR1H4 15 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne NFKB1 44 38 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne TAAR1 19 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne AKR1C3 38 45 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne NR2E3 61 36 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne AKR1C2 25 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne SMO 28 49 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne KCNK3 96 52 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Cl)c2Cl)c1 ZINC000147461775 EJ On-Demand Anodyne KCNK9 69 38 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne F2 21 42 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne FKBP1A 17 41 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne HTR4 58 37 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne GRIN2B 42 42 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne SIGMAR1 22 52 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne MMP13 37 42 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne CAPNS1 28 43 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne MMP2 27 42 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne CAPN1 16 42 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne EPHX2 36 44 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne TGM2 80 48 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne MMP1 31 41 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne CACNA1I 66 47 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne F13A1 85 48 Cc1ccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147461801 GF On-Demand Anodyne NAMPT 57 40 Oc1ccc(-c2noc(-c3cccc(Cl)c3F)n2)cc1 ZINC000147461815 CH On-Demand Anodyne LUCI_PHOPE 39 46 CCOC(=O)Cc1csc(-c2cc(C)ccn2)n1 ZINC000147461817 CF For-Sale Anodyne SREBF2 0 41 NS(=O)(=O)c1cc(Br)c(OCCN2CCCC2)cc1F ZINC000147461843 FD For-Sale Anodyne LTA4H 27 43 CCNc1ccc(C(=O)NCCNC(N)=O)cc1[N+](=O)[O-] ZINC000147461871 CC For-Sale Bother DRTS_TOXGO 15 41 CCNc1ccc(C(=O)NCCNC(N)=O)cc1[N+](=O)[O-] ZINC000147461871 CC For-Sale Bother TAAR1 20 54 CCOC(=O)[C@H](Br)c1cccnc1 ZINC000147461883 BE For-Sale Reactive TBXAS1 24 41 CCOC(=O)[C@H](Br)c1cccnc1 ZINC000147461883 BE For-Sale Reactive KCNA5 26 43 Cc1[nH]c(SCC(=O)Nc2ccc(NC(=O)C3CC3)cc2)nc1Cc1ccccc1 ZINC000147461891 HI On-Demand Anodyne ENPP1 79 38 COc1cc(OC)c(NC(=O)CC2(CN)CCC2)cc1Cl ZINC000147461922 DF For-Sale Anodyne HTR4 39 42 CNC(=O)CCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147461947 CD On-Demand Anodyne CACNA1H 24 42 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1cc(F)ccc1F ZINC000147461976 HF On-Demand Anodyne ADRB2 16 41 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1cc(F)ccc1F ZINC000147461976 HF On-Demand Anodyne ADRB1 53 39 O=C(O)c1cc(Cl)cc(NC(=O)C2CCCCC2)c1 ZINC000147461979 CH On-Demand Anodyne INHA 25 51 O=C(O)c1cc(Cl)cc(NC(=O)C2CCCCC2)c1 ZINC000147461979 CH On-Demand Anodyne EPHX2 17 44 O=C(O)c1cc(Cl)cc(NC(=O)C2CCCCC2)c1 ZINC000147461979 CH On-Demand Anodyne CACNA1I 41 35 O=C(O)c1cc(Cl)cc(NC(=O)C2CCCCC2)c1 ZINC000147461979 CH On-Demand Anodyne RHOA 0 44 O=C(O)c1cc(Cl)cc(NC(=O)C2CCCCC2)c1 ZINC000147461979 CH On-Demand Anodyne HCAR1 0 41 O=C(Nc1cccc(Br)c1)Nc1cc(NC(=O)Nc2cccc(Br)c2)cc(C(=O)O)c1 ZINC000147461987 KK For-Sale Anodyne EGFR 39 43 O=C(Nc1cccc(Br)c1)Nc1cc(NC(=O)Nc2cccc(Br)c2)cc(C(=O)O)c1 ZINC000147461987 KK For-Sale Anodyne PPIA 41 49 O=C(Nc1cccc(Br)c1)Nc1cc(NC(=O)Nc2cccc(Br)c2)cc(C(=O)O)c1 ZINC000147461987 KK For-Sale Anodyne KIT 16 43 O=C(Nc1cccc(Br)c1)Nc1cc(NC(=O)Nc2cccc(Br)c2)cc(C(=O)O)c1 ZINC000147461987 KK For-Sale Anodyne KDR 16 43 O=C(Nc1cccc(Br)c1)Nc1cc(NC(=O)Nc2cccc(Br)c2)cc(C(=O)O)c1 ZINC000147461987 KK For-Sale Anodyne EPHX2 26 48 O=C(Nc1cccc(Br)c1)Nc1cc(NC(=O)Nc2cccc(Br)c2)cc(C(=O)O)c1 ZINC000147461987 KK For-Sale Anodyne TAAR1 17 44 O=C(Nc1cccc(Br)c1)Nc1cc(NC(=O)Nc2cccc(Br)c2)cc(C(=O)O)c1 ZINC000147461987 KK For-Sale Anodyne AKR1C3 41 51 O=C(Nc1cccc(Br)c1)Nc1cc(NC(=O)Nc2cccc(Br)c2)cc(C(=O)O)c1 ZINC000147461987 KK For-Sale Anodyne KCNK3 119 41 O=C(Nc1cccc(Br)c1)Nc1cc(NC(=O)Nc2cccc(Br)c2)cc(C(=O)O)c1 ZINC000147461987 KK For-Sale Anodyne KCNK9 79 40 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne PRSS1 15 41 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne DRD2 26 44 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne DRD4 44 35 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne ACHE 22 45 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne DRD3 23 43 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne HTR4 54 40 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne F10 28 41 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne GRIN2B 51 40 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne SIGMAR1 16 50 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne TRY2_BOVIN 77 39 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne CCR3 31 40 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne CCR2 31 40 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne EPHX2 22 42 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne TGM2 74 49 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne ST14 89 36 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne CACNA1I 68 45 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne F13A1 73 49 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne AKR1C3 62 41 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne NAMPT 46 42 COCc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147462007 HF On-Demand Anodyne TMPRSS6 59 34 Cc1cc(C)c(C)c(Oc2nc(N)ncc2Cl)c1 ZINC000147462074 CG For-Sale Anodyne P2RX2 40 36 COC(=O)[C@H](C)OCc1ccccc1Br ZINC000147462077 CF For-Sale Anodyne ANPEP 21 42 CC1(NC(=O)Nc2cc(Br)cc(C(=O)O)c2)CCCCC1 ZINC000147462134 FH For-Sale Anodyne RARA 41 35 CSCC[C@H](N)C(=O)NCCc1ccc(O)c(O)c1 ZINC000147462166 CC For-Sale Clean OPRM1 18 43 CSCC[C@H](N)C(=O)NCCc1ccc(O)c(O)c1 ZINC000147462166 CC For-Sale Clean OPRD1 18 43 CSCC[C@H](N)C(=O)NCCc1ccc(O)c(O)c1 ZINC000147462166 CC For-Sale Clean ALOX15 26 49 O=C(NC[C@@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1c(F)cccc1F ZINC000147462190 HF On-Demand Anodyne ADRB2 17 44 O=C(NC[C@@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1c(F)cccc1F ZINC000147462190 HF On-Demand Anodyne ADRB1 55 39 O=C(COc1ccc([N+](=O)[O-])cc1)Nc1ccccc1Nc1ccccc1 ZINC000147462256 FI On-Demand Bother AKR1C3 24 52 O=C(COc1ccc([N+](=O)[O-])cc1)Nc1ccccc1Nc1ccccc1 ZINC000147462256 FI On-Demand Bother AKR1C2 49 52 Cc1cc(C)c(Nc2ccc(C(=O)O)c(C)n2)c(C)c1 ZINC000147462260 CH For-Sale Anodyne SORT1 25 41 COC(=O)[C@@H](C)OCc1ccccc1Br ZINC000147462288 CF For-Sale Anodyne ANPEP 21 42 COc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1OC ZINC000147462310 FG For-Sale Reactive DRD2 40 40 COc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1OC ZINC000147462310 FG For-Sale Reactive HCRTR1 24 49 COc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1OC ZINC000147462310 FG For-Sale Reactive HCRTR2 0 49 COc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1OC ZINC000147462310 FG For-Sale Reactive ACKR3 66 35 CC1(NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)CCCCC1 ZINC000147462334 DH On-Demand Anodyne RARA 41 35 CC1(NC(=O)Nc2cc(Cl)cc(C(=O)O)c2)CCCCC1 ZINC000147462334 DH On-Demand Anodyne CACNA1I 40 33 CCOc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147462375 CF On-Demand Anodyne PIK3CA 22 42 CCOc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147462375 CF On-Demand Anodyne PTPN7 0 47 CCOc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147462375 CF On-Demand Anodyne Q50565_METTH 0 49 CCOc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147462375 CF On-Demand Anodyne FABK 0 42 CCOc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147462375 CF On-Demand Anodyne ISPD 0 45 CC(C)N(C)CCCNC(=O)CCNS(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000147462389 GD On-Demand Bother TBXA2R 17 42 CC(C)N(C)CCCNC(=O)CCNS(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000147462389 GD On-Demand Bother CACNA1D 48 32 CC(C)N(C)CCCNC(=O)CCNS(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000147462389 GD On-Demand Bother COLA 31 41 CC(C)N(C)CCCNC(=O)CCNS(=O)(=O)c1cccc([N+](=O)[O-])c1 ZINC000147462389 GD On-Demand Bother CA5A 18 40 O=S(=O)(NC[C@@H]1CCCO[C@@H]1c1ccccc1)N1CCOCC1 ZINC000147462393 ED On-Demand Anodyne PGA5 45 32 CNc1cc(C(=O)NCCNC(N)=O)nc2ccccc12 ZINC000147462405 CC For-Sale Anodyne HTR3A 17 43 CNc1cc(C(=O)NCCNC(N)=O)nc2ccccc12 ZINC000147462405 CC For-Sale Anodyne BCHE 42 36 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccc(F)c(F)c1 ZINC000147462442 HF On-Demand Anodyne ADRB2 19 41 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccc(F)c(F)c1 ZINC000147462442 HF On-Demand Anodyne ADRB1 62 41 CC(Nc1ccc(Cl)cc1)=C(C#N)C#N ZINC000147462496 BG For-Sale Reactive DHODH 18 44 COc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1OC ZINC000147462509 FG For-Sale Reactive DRD2 40 40 COc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1OC ZINC000147462509 FG For-Sale Reactive HCRTR1 24 49 COc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1OC ZINC000147462509 FG For-Sale Reactive HCRTR2 0 49 COc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1OC ZINC000147462509 FG For-Sale Reactive ACKR3 66 35 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne F2 28 43 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne ACE 99 46 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne OPRM1 105 43 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne OPRD1 97 43 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne MME 133 50 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne ANPEP 96 36 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne TACR1 26 47 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne CTSB 42 38 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne TRY2_BOVIN 42 33 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne PAPA1_CARPA 47 35 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne CYSP_TRYCR 54 39 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne CTSL 46 38 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne CPA1 41 37 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne SLC15A1 0 50 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne NPFFR2 53 36 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne TIMP3 48 33 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne TPH1 59 31 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne DPP4 20 48 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne CTRB1 31 40 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne AMY2 42 29 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne CAPNS1 80 35 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne F11 44 35 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne YARS 89 42 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne DNPEP 0 40 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne CAPN1 70 39 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne CAPN2 45 35 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne ACE2 66 37 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne DPP7 51 39 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne LAP3 70 38 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne CTSC 40 34 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne POL 0 41 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne AMP1_PLAFQ 54 38 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne XIAP 61 39 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne DPP8 23 44 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne NAAA 56 40 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne SLC15A2 0 49 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462527 CD For-Sale Anodyne VM1B1_BOTAS 0 43 COc1cc(C(=O)NCc2cc(Br)ccc2F)ccc1F ZINC000147462567 FH On-Demand Anodyne PPARA 16 43 COc1cc(C(=O)NCc2cc(Br)ccc2F)ccc1F ZINC000147462567 FH On-Demand Anodyne PPARD 24 43 COc1cc(C(=O)NCc2cc(Br)ccc2F)ccc1F ZINC000147462567 FH On-Demand Anodyne MT-ND1 17 42 O=S(=O)(NC[C@@H]1CCCO[C@H]1c1ccccc1)N1CCOCC1 ZINC000147462613 ED On-Demand Anodyne PGA5 45 32 Cc1ccc(F)cc1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147462642 HF On-Demand Anodyne ADRB2 22 45 Cc1ccc(F)cc1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147462642 HF On-Demand Anodyne ADRB1 60 37 N#Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147462661 DG On-Demand Mild ABCC9 23 40 N#Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147462661 DG On-Demand Mild PPIA 15 49 N#Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147462661 DG On-Demand Mild KCNJ11 26 45 N#Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147462661 DG On-Demand Mild CPT1A 23 40 N#Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147462661 DG On-Demand Mild ITGA4 45 31 N#Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147462661 DG On-Demand Mild GRM5 19 53 N#Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147462661 DG On-Demand Mild MCHR1 27 41 N#Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147462661 DG On-Demand Mild TAAR1 24 43 N#Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147462661 DG On-Demand Mild AKR1C3 33 46 N#Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147462661 DG On-Demand Mild KCNK3 100 50 N#Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147462661 DG On-Demand Mild KCNK9 48 44 CCn1c(CC(=O)c2cncs2)nc2ccccc21 ZINC000147462732 CF For-Sale Anodyne IMDH_CRYPV 21 41 CCNc1cc(C(=O)NCCNC(N)=O)ccc1[N+](=O)[O-] ZINC000147462738 CC For-Sale Bother TAAR1 15 44 Cc1nc(Nc2cccc3ccccc23)ccc1C(=O)O ZINC000147462749 CH For-Sale Anodyne PTGER4 0 40 Cc1nc(Nc2cccc3ccccc23)ccc1C(=O)O ZINC000147462749 CH For-Sale Anodyne MAPK8 16 45 Cc1nc(Nc2cccc3ccccc23)ccc1C(=O)O ZINC000147462749 CH For-Sale Anodyne MCL1 22 41 Cc1nc(Nc2cccc3ccccc23)ccc1C(=O)O ZINC000147462749 CH For-Sale Anodyne AKR1C3 26 42 Cc1nc(Nc2cccc3ccccc23)ccc1C(=O)O ZINC000147462749 CH For-Sale Anodyne AKR1C2 61 42 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne F2 28 43 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne ACE 99 46 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne OPRM1 105 43 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne OPRD1 97 43 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne MME 133 50 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne ANPEP 96 36 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne TACR1 26 47 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne CTSB 42 38 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne TRY2_BOVIN 42 33 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne PAPA1_CARPA 47 35 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne CYSP_TRYCR 54 39 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne CTSL 46 38 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne CPA1 41 37 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne SLC15A1 0 50 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne NPFFR2 53 36 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne TIMP3 48 33 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne TPH1 59 31 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne DPP4 20 48 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne CTRB1 31 40 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne AMY2 42 29 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne CAPNS1 80 35 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne F11 44 35 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne YARS 89 42 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne DNPEP 0 40 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne CAPN1 70 39 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne CAPN2 45 35 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne ACE2 66 37 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne DPP7 51 39 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne LAP3 70 38 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne CTSC 40 34 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne POL 0 41 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne AMP1_PLAFQ 54 38 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne XIAP 61 39 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne DPP8 23 44 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne NAAA 56 40 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne SLC15A2 0 49 C[C@H]1CCC[C@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462761 CD For-Sale Anodyne VM1B1_BOTAS 0 43 CC(C)CCCCNC(=O)CNC(=O)c1ccc(N)cc1 ZINC000147462787 CD For-Sale Anodyne CA2 26 43 CC(C)CCCCNC(=O)CNC(=O)c1ccc(N)cc1 ZINC000147462787 CD For-Sale Anodyne FOLH1 32 40 NCC1(CC(=O)Nc2ccc(C(N)=O)cc2)CCC1 ZINC000147462790 CD For-Sale Anodyne ACR 47 32 CCCCc1ccc(O[C@@H](CN)c2ccccc2)cc1 ZINC000147462794 CI For-Sale Anodyne SCN2A 18 42 CCCCc1ccc(O[C@@H](CN)c2ccccc2)cc1 ZINC000147462794 CI For-Sale Anodyne TAAR1 28 43 Cc1ccc(Br)c(C(=O)NCc2cc(Br)ccc2F)c1 ZINC000147462799 HJ On-Demand Anodyne P2RX7 19 40 CN(CC(C)(C)C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147462803 CH On-Demand Anodyne CACNA1I 41 31 O=S(=O)(NC[C@H]1CCCO[C@@H]1c1ccccc1)N1CCOCC1 ZINC000147462819 ED On-Demand Anodyne PGA5 45 32 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1F ZINC000147462849 HF On-Demand Anodyne ADRB2 25 43 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1F ZINC000147462849 HF On-Demand Anodyne ADRB1 66 41 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1F ZINC000147462849 HF On-Demand Anodyne ADRB3 18 43 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1F ZINC000147462849 HF On-Demand Anodyne ENV 43 34 CN(Cc1cscn1)C(=O)NCCNC(=O)c1ccco1 ZINC000147462852 DD On-Demand Anodyne CYP3A4 15 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2F)c1 ZINC000147462862 EI On-Demand Anodyne RARA 32 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2F)c1 ZINC000147462862 EI On-Demand Anodyne PPIA 15 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2F)c1 ZINC000147462862 EI On-Demand Anodyne ATF1 58 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2F)c1 ZINC000147462862 EI On-Demand Anodyne CPT1A 48 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2F)c1 ZINC000147462862 EI On-Demand Anodyne CPT2 40 35 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2F)c1 ZINC000147462862 EI On-Demand Anodyne PYGL 25 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2F)c1 ZINC000147462862 EI On-Demand Anodyne NFKB1 54 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2F)c1 ZINC000147462862 EI On-Demand Anodyne AKR1C3 21 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2F)c1 ZINC000147462862 EI On-Demand Anodyne HCAR1 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2F)c1 ZINC000147462862 EI On-Demand Anodyne KCNK3 38 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2F)c1 ZINC000147462862 EI On-Demand Anodyne TMPRSS4 0 49 CCOC(=O)c1ccc2c(C3CCCC3)c(-c3ccccn3)sc2c1 ZINC000147462876 FK For-Sale Anodyne NS5B 0 43 COc1cccc(Sc2ccccc2C2(O)CCNCC2)c1 ZINC000147462879 DG For-Sale Anodyne HTR3A 18 57 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147462902 EE On-Demand Anodyne MAPK14 24 42 CC[C@H](NC(=O)N1CC[C@H]2NC(=O)CC[C@@H]2C1)C(=O)O ZINC000147462905 CC For-Sale Anodyne TRHR 49 34 Cc1cnn(CC(=O)Nc2cnn(CC(=O)NC3CC3)c2)c1 ZINC000147462947 DC On-Demand Anodyne PANC 51 33 CCCCc1ccc(O[C@H](CN)c2ccccc2)cc1 ZINC000147462972 CI For-Sale Anodyne SCN2A 18 42 CCCCc1ccc(O[C@H](CN)c2ccccc2)cc1 ZINC000147462972 CI For-Sale Anodyne TAAR1 28 43 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne F2 28 43 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne ACE 99 46 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne OPRM1 105 43 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne OPRD1 97 43 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne MME 133 50 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne ANPEP 96 36 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne TACR1 26 47 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne CTSB 42 38 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne TRY2_BOVIN 42 33 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne PAPA1_CARPA 47 35 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne CYSP_TRYCR 54 39 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne CTSL 46 38 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne CPA1 41 37 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne SLC15A1 0 50 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne NPFFR2 53 36 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne TIMP3 48 33 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne TPH1 59 31 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne DPP4 20 48 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne CTRB1 31 40 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne AMY2 42 29 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne CAPNS1 80 35 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne F11 44 35 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne YARS 89 42 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne DNPEP 0 40 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne CAPN1 70 39 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne CAPN2 45 35 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne ACE2 66 37 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne DPP7 51 39 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne LAP3 70 38 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne CTSC 40 34 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne POL 0 41 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne AMP1_PLAFQ 54 38 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne XIAP 61 39 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne DPP8 23 44 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne NAAA 56 40 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne SLC15A2 0 49 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@H](N)Cc1ccccc1 ZINC000147462980 CD For-Sale Anodyne VM1B1_BOTAS 0 43 Nc1c(Cl)cccc1C(=O)Nc1ccncc1Br ZINC000147462985 EG For-Sale Anodyne JAK1 0 41 Nc1c(Cl)cccc1C(=O)Nc1ccncc1Br ZINC000147462985 EG For-Sale Anodyne GRM4 36 40 Nc1c(Cl)cccc1C(=O)Nc1ccncc1Br ZINC000147462985 EG For-Sale Anodyne TYK2 31 40 Nc1c(Cl)cccc1C(=O)Nc1ccncc1Br ZINC000147462985 EG For-Sale Anodyne EPHB3 50 38 Nc1c(Cl)cccc1C(=O)Nc1ccncc1Br ZINC000147462985 EG For-Sale Anodyne G2YM83_BOTF4 65 33 O=S(=O)(NC[C@H]1CCCO[C@H]1c1ccccc1)N1CCOCC1 ZINC000147463022 ED On-Demand Anodyne PGA5 45 32 O=C(O)CCCOCc1ccccc1Br ZINC000147463031 CF For-Sale Anodyne FFAR1 30 55 O=C(O)CCCOCc1ccccc1Br ZINC000147463031 CF For-Sale Anodyne FFAR4 56 38 Cc1ccc(S(=O)(=O)N(CC(=O)Nc2cccc(C)c2C)Cc2cccc(Cl)c2)cc1 ZINC000147463074 JK In-Stock Anodyne MMP2 16 45 Cc1ccc(S(=O)(=O)N(CC(=O)Nc2cccc(C)c2C)Cc2cccc(Cl)c2)cc1 ZINC000147463074 JK In-Stock Anodyne MMP8 34 45 Cc1ccc(S(=O)(=O)N(CC(=O)Nc2cccc(C)c2C)Cc2cccc(Cl)c2)cc1 ZINC000147463074 JK In-Stock Anodyne MMP9 19 45 Cc1ccc(S(=O)(=O)N(CC(=O)Nc2cccc(C)c2C)Cc2cccc(Cl)c2)cc1 ZINC000147463074 JK In-Stock Anodyne MMP1 25 45 Cc1ccc(S(=O)(=O)N(CC(=O)Nc2cccc(C)c2C)Cc2cccc(Cl)c2)cc1 ZINC000147463074 JK In-Stock Anodyne DAGLA 28 44 Cc1ccc(S(=O)(=O)N(CC(=O)Nc2cccc(C)c2C)Cc2cccc(Cl)c2)cc1 ZINC000147463074 JK In-Stock Anodyne RORC 22 44 CCS(=O)(=O)N1CCC(NC(=O)NNC(=O)c2ccc(C)s2)CC1 ZINC000147463080 FC On-Demand Reactive EPHX2 34 48 CC(C)(C)SCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147463083 DH On-Demand Anodyne CACNA1H 22 41 CC(C)(C)SCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147463083 DH On-Demand Anodyne CACNA1I 44 35 CC(C)(C)SCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147463083 DH On-Demand Anodyne HCAR1 0 44 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccc(Cl)cc1 ZINC000147463106 HG On-Demand Anodyne ADRB2 26 44 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccc(Cl)cc1 ZINC000147463106 HG On-Demand Anodyne ADRB1 64 39 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccc(Cl)cc1 ZINC000147463106 HG On-Demand Anodyne ADRB3 32 44 CC[C@H](NC(=O)N1CC[C@@H]2NC(=O)CC[C@@H]2C1)C(=O)O ZINC000147463121 CC For-Sale Anodyne TRHR 49 34 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne PLG 18 47 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne CA2 20 51 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne HTR4 56 36 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne F10 22 42 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne GRIN2B 35 45 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne CCR3 19 42 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne EPHX2 21 45 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne TGM2 81 51 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne ST14 64 35 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne CACNA1I 66 40 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne F13A1 78 48 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne AKR1C3 45 36 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne SFRP1 17 41 NC(=O)c1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147463145 HD On-Demand Anodyne NAMPT 43 42 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147463172 EE On-Demand Anodyne MAPK14 24 42 CCOc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147463200 CG For-Sale Anodyne CACNA2D1 35 40 CCOc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147463200 CG For-Sale Anodyne AKR1C3 31 45 CCOc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147463200 CG For-Sale Anodyne AKR1C2 77 45 Nc1ccccc1CC(=O)Nc1ccncc1Br ZINC000147463203 DF For-Sale Anodyne CA5B 37 40 Nc1ccccc1CC(=O)Nc1ccncc1Br ZINC000147463203 DF For-Sale Anodyne CA5A 42 40 Nc1ccccc1CC(=O)Nc1ccncc1Br ZINC000147463203 DF For-Sale Anodyne CA9 20 45 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(C)cc1OCC(=O)N(C)C)C2 ZINC000147463221 GF On-Demand Anodyne ROCK2 47 53 CNS(=O)(=O)c1cccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@@H](C)C2)c1 ZINC000147463225 HD On-Demand Anodyne ST14 40 36 CCc1ncc(C(=O)NCc2c(C)nn(Cc3ccccc3)c2C)s1 ZINC000147463231 FG On-Demand Anodyne P2RX7 32 47 CCOC(=O)C/C(=N/OC)c1ccc(OC)cc1 ZINC000147463263 CD For-Sale Mild PTGS2 29 43 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463305 DF On-Demand Anodyne ACE 52 44 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463305 DF On-Demand Anodyne OPRM1 50 47 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463305 DF On-Demand Anodyne OPRD1 77 44 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463305 DF On-Demand Anodyne OPRK1 22 44 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463305 DF On-Demand Anodyne MME 55 44 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463305 DF On-Demand Anodyne ANPEP 55 33 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463305 DF On-Demand Anodyne SLC15A1 0 46 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463305 DF On-Demand Anodyne YARS 53 40 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463305 DF On-Demand Anodyne LAP3 45 36 N[C@@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463305 DF On-Demand Anodyne SLC15A2 0 46 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)no1 ZINC000147463316 CF In-Stock Anodyne PPIA 20 40 CC[C@H](NC(=O)N1CC[C@H]2NC(=O)CC[C@H]2C1)C(=O)O ZINC000147463318 CC For-Sale Anodyne TRHR 49 34 NC(=O)NCCNC(=O)c1cccc(C(F)(F)F)c1N ZINC000147463342 CC For-Sale Anodyne P2RX7 43 35 COc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147463370 HE On-Demand Anodyne ADRB2 34 52 COc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147463370 HE On-Demand Anodyne ADRB1 63 40 COc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147463370 HE On-Demand Anodyne ADRB3 29 52 COc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147463370 HE On-Demand Anodyne MTNR1A 28 43 COc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147463370 HE On-Demand Anodyne MTNR1B 35 43 COc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147463370 HE On-Demand Anodyne TAAR1 33 44 COc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147463370 HE On-Demand Anodyne KCNK3 46 34 COc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147463370 HE On-Demand Anodyne PDS 26 41 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147463372 EE On-Demand Anodyne MAPK14 24 42 O=C(Cn1ccccc1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147463389 GD On-Demand Anodyne EPHX2 22 43 O=C(Cn1ccccc1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147463389 GD On-Demand Anodyne TGM2 66 44 O=C(Cn1ccccc1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147463389 GD On-Demand Anodyne CACNA1I 42 34 O=C(Cn1ccccc1=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147463389 GD On-Demand Anodyne F13A1 66 44 CNS(=O)(=O)c1cccc(NC(=O)C(=O)NCC(C)(C)N2CCC[C@H](C)C2)c1 ZINC000147463404 HD On-Demand Anodyne ST14 40 36 COc1cccc(C(=O)Nc2ccncc2Br)c1N ZINC000147463444 DF For-Sale Anodyne GRM4 18 40 COc1cccc(C(=O)Nc2ccncc2Br)c1N ZINC000147463444 DF For-Sale Anodyne KCNK3 54 44 COc1cccc(C(=O)Nc2ccncc2Br)c1N ZINC000147463444 DF For-Sale Anodyne KCNK9 49 44 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463469 DF On-Demand Anodyne ACE 52 44 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463469 DF On-Demand Anodyne OPRM1 50 44 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463469 DF On-Demand Anodyne OPRD1 45 44 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463469 DF On-Demand Anodyne MME 55 44 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463469 DF On-Demand Anodyne ANPEP 55 33 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463469 DF On-Demand Anodyne YARS 53 40 N[C@H](Cc1ccccc1)C(=O)N[C@@H]1CCSc2ccccc21 ZINC000147463469 DF On-Demand Anodyne LAP3 45 36 COc1ccccc1CNc1ccc(C(=O)O)c(C)n1 ZINC000147463486 CF For-Sale Anodyne ALS 43 36 CCc1ncc(C(=O)Nc2nc(-c3cccc(F)c3)cs2)s1 ZINC000147463495 EI On-Demand Anodyne MPL 77 40 CCc1ncc(C(=O)Nc2nc(-c3cccc(F)c3)cs2)s1 ZINC000147463495 EI On-Demand Anodyne ROCK1 22 45 CCc1ncc(C(=O)Nc2nc(-c3cccc(F)c3)cs2)s1 ZINC000147463495 EI On-Demand Anodyne ROCK2 17 46 CCc1ncc(C(=O)Nc2nc(-c3cccc(F)c3)cs2)s1 ZINC000147463495 EI On-Demand Anodyne HDAC9 16 53 CCc1ncc(C(=O)Nc2nc(-c3cccc(F)c3)cs2)s1 ZINC000147463495 EI On-Demand Anodyne TRPA1 20 49 CNCCC(=O)NCCCCC(C)C ZINC000147463512 BD For-Sale Anodyne NOD1 19 40 CC[C@H](NC(=O)N1CC[C@@H]2NC(=O)CC[C@H]2C1)C(=O)O ZINC000147463524 CC For-Sale Anodyne TRHR 49 34 CC(C)(C)C(=O)NCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147463537 DE On-Demand Anodyne CACNA1H 22 40 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147463596 EE On-Demand Anodyne MAPK14 24 42 O=C(Cn1cc(NC(=O)C(=O)c2ccc3c(c2)CCC3)cn1)NC1CC1 ZINC000147463604 FD On-Demand Anodyne PANC 49 32 Cc1cc(C)c(C)c(Oc2nc(N)cn3ccnc23)c1 ZINC000147463616 CG For-Sale Anodyne HIVRT 0 47 COc1ccccc1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147463631 HE On-Demand Anodyne ADRB2 29 49 COc1ccccc1NC(=O)C(=O)NC[C@H](O)COc1cccc(Cl)c1Cl ZINC000147463631 HE On-Demand Anodyne ADRB1 58 37 Cc1cc(Cl)cc(-c2nc(-c3cccc(O)c3)no2)c1 ZINC000147463657 CI For-Sale Anodyne GRM5 26 45 Cc1cc(Cl)cc(-c2nc(-c3cccc(O)c3)no2)c1 ZINC000147463657 CI For-Sale Anodyne HSD17B1 37 41 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463658 DF On-Demand Anodyne ACE 52 44 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463658 DF On-Demand Anodyne OPRM1 50 47 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463658 DF On-Demand Anodyne OPRD1 77 44 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463658 DF On-Demand Anodyne OPRK1 22 44 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463658 DF On-Demand Anodyne MME 55 44 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463658 DF On-Demand Anodyne ANPEP 55 33 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463658 DF On-Demand Anodyne SLC15A1 0 46 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463658 DF On-Demand Anodyne YARS 53 40 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463658 DF On-Demand Anodyne LAP3 45 36 N[C@@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463658 DF On-Demand Anodyne SLC15A2 0 46 Nc1ccc(C(=O)Nc2ccncc2Br)c(Cl)c1 ZINC000147463714 EG For-Sale Anodyne GRM4 21 41 COc1cc(NC(=O)c2ccc(C(N)=S)cc2)ccc1Br ZINC000147463720 FG On-Demand Anodyne COLA 44 35 COc1cc(NC(=O)c2ccc(C(N)=S)cc2)ccc1Br ZINC000147463720 FG On-Demand Anodyne CPT1A 44 33 COc1cc(NC(=O)c2ccc(C(N)=S)cc2)ccc1Br ZINC000147463720 FG On-Demand Anodyne CPT2 42 31 COc1cc(NC(=O)c2ccc(C(N)=S)cc2)ccc1Br ZINC000147463720 FG On-Demand Anodyne PLAU 20 40 COc1cc(NC(=O)c2ccc(C(N)=S)cc2)ccc1Br ZINC000147463720 FG On-Demand Anodyne TAAR1 32 43 COc1cc(NC(=O)c2ccc(C(N)=S)cc2)ccc1Br ZINC000147463720 FG On-Demand Anodyne PPO2 16 41 COc1cc(NC(=O)c2ccc(C(N)=S)cc2)ccc1Br ZINC000147463720 FG On-Demand Anodyne ENPP1 76 37 COc1cc(NC(=O)c2ccc(C(N)=S)cc2)ccc1Br ZINC000147463720 FG On-Demand Anodyne SMO 23 44 COc1cc(NC(=O)c2ccc(C(N)=S)cc2)ccc1Br ZINC000147463720 FG On-Demand Anodyne KCNK3 91 43 COc1cc(NC(=O)c2ccc(C(N)=S)cc2)ccc1Br ZINC000147463720 FG On-Demand Anodyne KCNK9 60 39 NC1(C(=O)Nc2ccc(OC(F)(F)F)cc2)CCC1 ZINC000147463729 CE On-Demand Anodyne MMP2 27 40 NC1(C(=O)Nc2ccc(OC(F)(F)F)cc2)CCC1 ZINC000147463729 CE On-Demand Anodyne EPHX2 66 52 CC[C@H](NC(=O)Nc1ccc(C#N)cc1F)C(=O)O ZINC000147463734 CD For-Sale Mild ACE2 45 34 C[C@H](CNc1ccccc1S(N)(=O)=O)CC(=O)O ZINC000147463758 CC For-Sale Anodyne CA2 60 50 C[C@H](CNc1ccccc1S(N)(=O)=O)CC(=O)O ZINC000147463758 CC For-Sale Anodyne CA7 19 46 C[C@H](CNc1ccccc1S(N)(=O)=O)CC(=O)O ZINC000147463758 CC For-Sale Anodyne CA4 54 49 C[C@H](CNc1ccccc1S(N)(=O)=O)CC(=O)O ZINC000147463758 CC For-Sale Anodyne CA12 17 46 C[C@H](CNc1ccccc1S(N)(=O)=O)CC(=O)O ZINC000147463758 CC For-Sale Anodyne CA9 17 49 Cc1cccc(COc2c(Cl)cc(/C=c3\sc4nc5ccccc5n4c3=O)cc2Cl)c1 ZINC000147463791 JK In-Stock Anodyne MAPT 53 33 CCCOc1ccc(Oc2nc(N)nc(OC)n2)cc1 ZINC000147463803 CE For-Sale Anodyne DRTS_PLAFK 23 45 CCCOc1ccc(Oc2nc(N)nc(OC)n2)cc1 ZINC000147463803 CE For-Sale Anodyne ACACA 32 40 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1C(C)C ZINC000147463808 HH On-Demand Anodyne HTR4 67 41 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1C(C)C ZINC000147463808 HH On-Demand Anodyne EPHX2 24 40 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1C(C)C ZINC000147463808 HH On-Demand Anodyne TGM2 64 43 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1C(C)C ZINC000147463808 HH On-Demand Anodyne CACNA1I 59 35 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)n1C(C)C ZINC000147463808 HH On-Demand Anodyne F13A1 64 43 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463863 DF On-Demand Anodyne OPRM1 50 47 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463863 DF On-Demand Anodyne OPRD1 77 44 N[C@H](Cc1ccccc1)C(=O)N[C@H]1CCSc2ccccc21 ZINC000147463863 DF On-Demand Anodyne OPRK1 22 44 Cc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1C ZINC000147463877 HG On-Demand Anodyne ADRB2 24 41 Cc1cccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1C ZINC000147463877 HG On-Demand Anodyne ADRB1 51 34 Cc1ccc(N)cc1C(=O)Nc1ccncc1Br ZINC000147463903 DF For-Sale Anodyne BTK 30 40 COc1cc(-c2nc(-c3cccc(O)c3)no2)ccc1F ZINC000147463908 CG For-Sale Anodyne HSD17B1 35 41 COc1cc(-c2nc(-c3cccc(O)c3)no2)ccc1F ZINC000147463908 CG For-Sale Anodyne HSD17B2 21 41 COc1cc(-c2nc(-c3cccc(O)c3)no2)ccc1F ZINC000147463908 CG For-Sale Anodyne LUCI_PHOPE 41 47 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne MAOB 21 51 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne COLA 41 38 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne CPT1A 43 34 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne HPSE 15 48 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne PLAU 15 40 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne IMPDH2 0 47 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne TAAR1 36 43 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne SHH 24 41 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne ENPP1 75 38 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne GLMU 0 42 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne KCNK3 82 38 COc1cc(NC(=O)c2ccc3cn[nH]c3c2)ccc1Br ZINC000147463946 EH For-Sale Anodyne KCNK9 59 38 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1SC1CCCC1 ZINC000147463947 EH On-Demand Anodyne CTSK 42 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1SC1CCCC1 ZINC000147463947 EH On-Demand Anodyne NPFFR2 45 31 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1SC1CCCC1 ZINC000147463947 EH On-Demand Anodyne HDAC10 43 36 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1SC1CCCC1 ZINC000147463947 EH On-Demand Anodyne HDAC11 57 36 NCC1(CC(=O)Nc2ccc(OC(F)(F)F)cc2)CCC1 ZINC000147463948 DG For-Sale Anodyne P2RY1 62 44 NCC1(CC(=O)Nc2ccc(OC(F)(F)F)cc2)CCC1 ZINC000147463948 DG For-Sale Anodyne EPHX2 60 47 NCC1(CC(=O)Nc2ccc(OC(F)(F)F)cc2)CCC1 ZINC000147463948 DG For-Sale Anodyne ACR 41 36 C[C@@H](CNc1ccccc1S(N)(=O)=O)CC(=O)O ZINC000147463970 CC For-Sale Anodyne CA2 60 50 C[C@@H](CNc1ccccc1S(N)(=O)=O)CC(=O)O ZINC000147463970 CC For-Sale Anodyne CA7 19 46 C[C@@H](CNc1ccccc1S(N)(=O)=O)CC(=O)O ZINC000147463970 CC For-Sale Anodyne CA4 54 49 C[C@@H](CNc1ccccc1S(N)(=O)=O)CC(=O)O ZINC000147463970 CC For-Sale Anodyne CA12 17 46 C[C@@H](CNc1ccccc1S(N)(=O)=O)CC(=O)O ZINC000147463970 CC For-Sale Anodyne CA9 17 49 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne F2 21 40 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne FKBP1A 16 40 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne CHRM5 22 42 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne GRIN2B 48 35 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne NPY2R 17 41 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne MMP2 15 40 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne MMP3 29 40 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne CAPN1 15 41 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne MMP9 22 40 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne EPHX2 60 56 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne TGM2 85 45 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne MMP1 31 40 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne F13A1 94 45 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne SFRP1 93 38 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne WNT3 62 33 CC(=O)N1CCC(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)CC1 ZINC000147464031 HD On-Demand Anodyne NAMPT 42 40 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147464041 HJ On-Demand Anodyne MAPK11 30 41 Cc1nc(-c2ccc(Cl)s2)sc1C(=O)Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147464041 HJ On-Demand Anodyne MAPK14 25 45 Cc1nc(NC23CC4CC(CC(C4)C2)C3)ccc1C(=O)O ZINC000147464089 CG For-Sale Anodyne EPHX2 52 43 Nc1cc(C(=O)Nc2ccncc2Br)cc(Cl)c1Cl ZINC000147464090 FH For-Sale Anodyne HDAC1 0 41 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1C ZINC000147464095 HG On-Demand Anodyne ADRB2 28 45 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1C ZINC000147464095 HG On-Demand Anodyne ADRB1 62 36 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1C ZINC000147464095 HG On-Demand Anodyne GRIN1 21 40 Cc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1C ZINC000147464095 HG On-Demand Anodyne ADRB3 23 45 Cc1ccc(Br)c(-c2nc(-c3cccc(O)c3)no2)c1 ZINC000147464114 EI For-Sale Anodyne HSD17B1 33 40 COc1ccc(CNc2nc(Cl)cs2)c(OC)c1 ZINC000147464125 CG On-Demand Anodyne DRTS_TOXGO 19 46 COc1cc(NC(=O)CCC(C)=O)ccc1Br ZINC000147464155 DF On-Demand Anodyne CASP2 21 45 COc1cc(NC(=O)CCC(C)=O)ccc1Br ZINC000147464155 DF On-Demand Anodyne CASP6 20 45 COc1cc(NC(=O)CCC(C)=O)ccc1Br ZINC000147464155 DF On-Demand Anodyne CASP7 0 45 COc1cc(NC(=O)CCC(C)=O)ccc1Br ZINC000147464155 DF On-Demand Anodyne IMPDH2 0 46 COc1cc(NC(=O)CCC(C)=O)ccc1Br ZINC000147464155 DF On-Demand Anodyne ENPP1 64 39 COc1cc(NC(=O)CCC(C)=O)ccc1Br ZINC000147464155 DF On-Demand Anodyne PARP10 0 49 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1SC1CCCC1 ZINC000147464165 EH On-Demand Anodyne CTSK 42 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1SC1CCCC1 ZINC000147464165 EH On-Demand Anodyne NPFFR2 45 31 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1SC1CCCC1 ZINC000147464165 EH On-Demand Anodyne HDAC10 43 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1SC1CCCC1 ZINC000147464165 EH On-Demand Anodyne HDAC11 57 36 Cc1occc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147464195 CG On-Demand Anodyne JUN 19 41 Cc1occc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147464195 CG On-Demand Anodyne ATF1 54 37 Cc1occc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147464195 CG On-Demand Anodyne NFKB1 49 37 Cc1occc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147464195 CG On-Demand Anodyne HCAR1 0 40 Cc1occc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147464195 CG On-Demand Anodyne KCNK3 48 37 Cc1occc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147464195 CG On-Demand Anodyne TMPRSS4 0 41 CCCOc1ccc(Oc2cc(NCC)nc(N)n2)cc1 ZINC000147464231 CG For-Sale Anodyne ACACA 34 40 CC[C@@H]1CN(C[C@@H]2CCCc3ccccc32)CC[C@@H]1N ZINC000147464276 CG For-Sale Anodyne SIGMAR1 15 46 CC[C@@H]1CN(C[C@@H]2CCCc3ccccc32)CC[C@@H]1N ZINC000147464276 CG For-Sale Anodyne EBP 24 42 CC(=O)N[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464289 GD On-Demand Anodyne CHRM5 18 41 CC(=O)N[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464289 GD On-Demand Anodyne CASP2 54 34 CC(=O)N[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464289 GD On-Demand Anodyne PCSK5 23 42 CC(=O)N[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464289 GD On-Demand Anodyne FURIN 24 42 CC(=O)N[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464289 GD On-Demand Anodyne EPHX2 17 42 CC(=O)N[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464289 GD On-Demand Anodyne TGM2 65 43 CC(=O)N[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464289 GD On-Demand Anodyne F13A1 69 43 CC(=O)N[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464289 GD On-Demand Anodyne BRCA1 53 36 Cc1cc(C(=O)Nc2ccncc2Br)ccc1N ZINC000147464321 DF For-Sale Anodyne KIT 15 43 Cc1cc(C(=O)Nc2ccncc2Br)ccc1N ZINC000147464321 DF For-Sale Anodyne HDAC1 42 46 Cc1cc(C(=O)Nc2ccncc2Br)ccc1N ZINC000147464321 DF For-Sale Anodyne HDAC2 22 43 Cc1cc(C(=O)Nc2ccncc2Br)ccc1N ZINC000147464321 DF For-Sale Anodyne SIRT2 26 46 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)c(OC)c1 ZINC000147464325 CF For-Sale Anodyne CYP1B1 17 45 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)c(OC)c1 ZINC000147464325 CF For-Sale Anodyne LUCI_LUCLA 18 45 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)c(OC)c1 ZINC000147464325 CF For-Sale Anodyne AKR1C3 37 52 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)c(OC)c1 ZINC000147464325 CF For-Sale Anodyne AKR1C2 79 52 Oc1cccc(-c2noc(-c3cccc(Cl)c3F)n2)c1 ZINC000147464333 CH For-Sale Anodyne GRM5 20 40 Oc1cccc(-c2noc(-c3cccc(Cl)c3F)n2)c1 ZINC000147464333 CH For-Sale Anodyne HSD17B1 32 41 CN1CCC(n2cc(-c3ccn4c(-c5cccc(NC(=O)NCC(F)(F)F)c5)cnc4c3)cn2)CC1 ZINC000147464336 JJ Annotated Anodyne MAP3K7 49 35 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccc(F)cc1 ZINC000147464350 HF On-Demand Anodyne ADRB2 25 44 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccc(F)cc1 ZINC000147464350 HF On-Demand Anodyne ADRB1 67 46 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccc(F)cc1 ZINC000147464350 HF On-Demand Anodyne ADRB3 23 44 CCC[C@H](NC(N)=O)C(=O)Nc1cnn(CC(=O)NC2CC2)c1 ZINC000147464357 DB On-Demand Anodyne PANC 45 32 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne THRA 56 42 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne SRD5A2 29 41 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne INHA 109 47 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne MPL 20 40 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne RXRG 29 46 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne RARB 38 56 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne RXRA 26 46 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne RXRB 21 46 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne PLA2G4A 45 46 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne S1PR4 22 41 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne PPARD 46 39 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne GRM2 20 45 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne PLA2G4B 104 46 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne S1PR1 23 44 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne TTR 0 43 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne PLM2_PLAFA 47 34 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne FFAR1 27 41 CCCCc1ccc(Oc2ccc(C(=O)O)cc2C)cc1 ZINC000147464381 CJ For-Sale Anodyne YOPH 0 42 CCNC(=O)c1ccc(NC(=O)NCc2cccc(NC(=O)[C@@H]3CCCO3)c2)cc1 ZINC000147464393 HF On-Demand Anodyne ROCK2 23 43 CCc1noc(C)c1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147464454 DG On-Demand Anodyne GHSR 0 44 CC(=O)N[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464476 GD On-Demand Anodyne CHRM5 18 41 CC(=O)N[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464476 GD On-Demand Anodyne CASP2 54 34 CC(=O)N[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464476 GD On-Demand Anodyne PCSK5 23 42 CC(=O)N[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464476 GD On-Demand Anodyne FURIN 24 42 CC(=O)N[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464476 GD On-Demand Anodyne EPHX2 17 42 CC(=O)N[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464476 GD On-Demand Anodyne TGM2 65 43 CC(=O)N[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464476 GD On-Demand Anodyne F13A1 69 43 CC(=O)N[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C(C)C ZINC000147464476 GD On-Demand Anodyne BRCA1 53 36 O=C1C[C@H](OC(=S)c2ccccc2)N1 ZINC000147464478 BD For-Sale Anodyne Q8WSF8_APLCA 43 35 CC[C@H]1CN(C[C@@H]2CCCc3ccccc32)CC[C@@H]1N ZINC000147464481 CG For-Sale Anodyne SIGMAR1 15 46 CC[C@H]1CN(C[C@@H]2CCCc3ccccc32)CC[C@@H]1N ZINC000147464481 CG For-Sale Anodyne EBP 24 42 Cc1ccc(Cl)c(Nc2ccc(C(=O)O)c(C)n2)c1Cl ZINC000147464526 DI For-Sale Anodyne CXCL8 16 48 Cc1ccc(Cl)c(Nc2ccc(C(=O)O)c(C)n2)c1Cl ZINC000147464526 DI For-Sale Anodyne FABP2 0 59 Cc1ccc(Cl)c(Nc2ccc(C(=O)O)c(C)n2)c1Cl ZINC000147464526 DI For-Sale Anodyne FABP1 20 59 CCC[C@@H](NC(N)=O)C(=O)Nc1cnn(CC(=O)NC2CC2)c1 ZINC000147464539 DB On-Demand Anodyne PANC 45 32 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccccc1Cl ZINC000147464547 HG On-Demand Anodyne ADRB2 29 40 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccccc1Cl ZINC000147464547 HG On-Demand Anodyne ADRB1 59 38 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccccc1Cl ZINC000147464547 HG On-Demand Anodyne ADRB3 15 45 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccccc1Cl ZINC000147464547 HG On-Demand Anodyne CXCL8 41 33 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccccc1Cl ZINC000147464547 HG On-Demand Anodyne ABCB1 41 35 CCNC(=O)c1cccc(N[C@@H]2CCO[C@@H]2C)c1 ZINC000147464576 BE On-Demand Anodyne KCNK3 47 33 COc1ccc(C(=O)[C@@H](O)c2ccc(Br)cc2)cc1 ZINC000147464587 DG For-Sale Anodyne CES2 28 46 COc1ccc(C(=O)[C@@H](O)c2ccc(Br)cc2)cc1 ZINC000147464587 DG For-Sale Anodyne DXR 20 40 CCNC(=O)c1ccc(NC(=O)NCc2cccc(NC(=O)[C@H]3CCCO3)c2)cc1 ZINC000147464605 HF On-Demand Anodyne ROCK2 23 43 CCCOc1ccc(Oc2cc(NC)nc(C)n2)cc1 ZINC000147464641 CG For-Sale Anodyne ACACA 39 41 O=C1C[C@@H](OC(=S)c2ccccc2)N1 ZINC000147464690 BD For-Sale Anodyne Q8WSF8_APLCA 43 35 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1Cl ZINC000147464722 CG For-Sale Anodyne GRM4 15 45 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1Cl ZINC000147464722 CG For-Sale Anodyne AGPAT2 40 39 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1Cl ZINC000147464722 CG For-Sale Anodyne CSF1R 22 40 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1Cl ZINC000147464722 CG For-Sale Anodyne AKR1C3 43 42 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1Cl ZINC000147464722 CG For-Sale Anodyne AKR1C2 82 42 CNC(=O)Cn1cc(NC(=O)c2ccccc2S(=O)(=O)N2CCCCC2)cn1 ZINC000147464758 HD On-Demand Anodyne CCR8 41 31 CNC(=O)Cn1cc(NC(=O)c2ccccc2S(=O)(=O)N2CCCCC2)cn1 ZINC000147464758 HD On-Demand Anodyne PANC 50 33 CCNC(=O)c1cccc(N[C@H]2CCO[C@@H]2C)c1 ZINC000147464769 BE On-Demand Anodyne KCNK3 47 33 CN[C@H](C)C(=O)NCCCCC(C)C ZINC000147464795 BD For-Sale Anodyne SIRT1 25 41 CCOC(=O)[C@@H]1CCCN(S(=O)(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)C1 ZINC000147464805 HE On-Demand Anodyne SLC6A1 74 33 COCc1nc(C(=O)N2CCc3sccc3[C@@H]2c2ccccc2)cs1 ZINC000147464807 FI On-Demand Anodyne TRPM8 20 46 COc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1 ZINC000147464813 HE On-Demand Anodyne ADRB2 44 58 COc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1 ZINC000147464813 HE On-Demand Anodyne ADRB1 69 49 COc1ccc(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)cc1 ZINC000147464813 HE On-Demand Anodyne ADRB3 44 58 COc1ccc(C(=O)[C@H](O)c2ccc(Br)cc2)cc1 ZINC000147464815 DG For-Sale Anodyne CES2 28 46 COc1ccc(C(=O)[C@H](O)c2ccc(Br)cc2)cc1 ZINC000147464815 DG For-Sale Anodyne DXR 20 40 CCNC(=O)c1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147464837 HF On-Demand Anodyne CHRM3 23 43 CCNC(=O)c1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147464837 HF On-Demand Anodyne CCR3 21 43 CCNC(=O)c1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147464837 HF On-Demand Anodyne MTOR 54 37 CCNC(=O)c1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147464837 HF On-Demand Anodyne EPHX2 18 44 CCNC(=O)c1ccc(NC(=O)NCc2cccc(CN3CCO[C@H](C)C3)c2)cc1 ZINC000147464837 HF On-Demand Anodyne NOD2 40 34 O=C(Nc1ccccc1OC[C@@H]1CCCCO1)c1cnn(-c2ccccc2Cl)c1 ZINC000147464843 HJ On-Demand Anodyne EPHB3 42 35 CNc1nc(C(=O)NCCNC(N)=O)cc2ccccc12 ZINC000147464871 CC For-Sale Anodyne PLA2G7 18 40 CCCCO[C@@H](C)C(=O)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147464883 GG On-Demand Anodyne P2RX7 32 41 CCCCO[C@@H](C)C(=O)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147464883 GG On-Demand Anodyne RBP4 52 37 CCCCO[C@@H](C)C(=O)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147464883 GG On-Demand Anodyne SCD1 24 51 CCCCO[C@@H](C)C(=O)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147464883 GG On-Demand Anodyne SCD 25 49 CCC(C)(C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147464912 CG On-Demand Anodyne NPY2R 15 46 CCC(C)(C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147464912 CG On-Demand Anodyne CACNA1I 42 32 CCC(C)(C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147464912 CG On-Demand Anodyne HCAR1 0 43 Cc1nc(Nc2cccc3cccnc23)ccc1C(=O)O ZINC000147464922 CG For-Sale Anodyne AKR1C2 42 37 Cc1nc(Nc2cccc3cccnc23)ccc1C(=O)O ZINC000147464922 CG For-Sale Anodyne EGLN1 0 40 Cc1nc(Nc2cccc3cccnc23)ccc1C(=O)O ZINC000147464922 CG For-Sale Anodyne FTO 0 40 CC(C)(NC(=O)Nc1cc(Cl)cc(C(=O)O)c1)C(N)=O ZINC000147464961 CD For-Sale Anodyne IMDH_CRYPV 40 36 CC(C)(NC(=O)Nc1cc(Cl)cc(C(=O)O)c1)C(N)=O ZINC000147464961 CD For-Sale Anodyne HCAR1 0 40 CCNC(=O)c1cccc(N[C@@H]2CCO[C@H]2C)c1 ZINC000147464981 BE On-Demand Anodyne KCNK3 47 33 O=C(COc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147464985 HE On-Demand Anodyne CHRM5 19 41 O=C(COc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147464985 HE On-Demand Anodyne SIGMAR1 15 41 O=C(COc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147464985 HE On-Demand Anodyne MMP13 45 42 O=C(COc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147464985 HE On-Demand Anodyne ADAM17 43 41 O=C(COc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147464985 HE On-Demand Anodyne MMP3 29 40 O=C(COc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147464985 HE On-Demand Anodyne EPHX2 22 45 O=C(COc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147464985 HE On-Demand Anodyne TGM2 67 43 O=C(COc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147464985 HE On-Demand Anodyne F13A1 67 43 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1cccc(Cl)c1 ZINC000147465000 HG On-Demand Anodyne ADRB2 23 43 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1cccc(Cl)c1 ZINC000147465000 HG On-Demand Anodyne ADRB1 60 37 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1cccc(Cl)c1 ZINC000147465000 HG On-Demand Anodyne ADRB3 20 43 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1cccc(Cl)c1 ZINC000147465000 HG On-Demand Anodyne PDS 18 43 CN[C@@H](C)C(=O)NCCCCC(C)C ZINC000147465022 BD For-Sale Anodyne SIRT1 25 41 COCc1nc(C(=O)N2CCc3sccc3[C@H]2c2ccccc2)cs1 ZINC000147465028 FI On-Demand Anodyne TRPM8 20 46 CCNC(=O)c1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147465056 HF On-Demand Anodyne CHRM3 23 43 CCNC(=O)c1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147465056 HF On-Demand Anodyne CCR3 21 43 CCNC(=O)c1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147465056 HF On-Demand Anodyne MTOR 54 37 CCNC(=O)c1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147465056 HF On-Demand Anodyne EPHX2 18 44 CCNC(=O)c1ccc(NC(=O)NCc2cccc(CN3CCO[C@@H](C)C3)c2)cc1 ZINC000147465056 HF On-Demand Anodyne NOD2 40 34 Cc1cc(Cl)cc(-c2nc(-c3ccccc3N)no2)c1 ZINC000147465059 CH For-Sale Anodyne LUCI_PHOPE 35 41 Cc1ccc(NC[C@@H](C)CC(=O)O)cc1[N+](=O)[O-] ZINC000147465077 CE For-Sale Bother COLA 46 33 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccccc1OC[C@@H]1CCCCO1)C2 ZINC000147465084 GH On-Demand Anodyne ROCK2 32 45 CCCCO[C@H](C)C(=O)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147465086 GG On-Demand Anodyne P2RX7 32 41 CCCCO[C@H](C)C(=O)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147465086 GG On-Demand Anodyne RBP4 52 37 CCCCO[C@H](C)C(=O)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147465086 GG On-Demand Anodyne SCD1 24 51 CCCCO[C@H](C)C(=O)N1CCN(C(=O)c2ccccc2C(F)(F)F)CC1 ZINC000147465086 GG On-Demand Anodyne SCD 25 49 CCOc1ccccc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147465125 CG For-Sale Anodyne PPIA 15 41 CCOc1ccccc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147465125 CG For-Sale Anodyne MAPK8 18 46 CCOc1ccccc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147465125 CG For-Sale Anodyne AKR1C2 50 37 CCOc1ccccc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147465125 CG For-Sale Anodyne HCN1 49 33 CCOc1ccccc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147465125 CG For-Sale Anodyne HCN4 41 32 COCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147465152 CE On-Demand Anodyne CACNA1I 51 35 COCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147465152 CE On-Demand Anodyne HCAR1 0 40 N[C@H](Cc1ccc(O)cc1)[C@@H]1COc2ccccc21 ZINC000147465207 CE For-Sale Anodyne YARS 51 33 Nc1cc(C(=O)Nc2ccncc2Br)ccc1Cl ZINC000147465216 EG For-Sale Anodyne HDAC1 32 42 Nc1cc(C(=O)Nc2ccncc2Br)ccc1Cl ZINC000147465216 EG For-Sale Anodyne HDAC3 0 42 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1cccc(F)c1 ZINC000147465217 HF On-Demand Anodyne ADRB2 19 42 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1cccc(F)c1 ZINC000147465217 HF On-Demand Anodyne ADRB1 64 38 C[C@@H](CCC(=O)O)OCc1ccccc1Br ZINC000147465244 CG For-Sale Anodyne THRA 15 40 C[C@@H](CCC(=O)O)OCc1ccccc1Br ZINC000147465244 CG For-Sale Anodyne FFAR1 25 51 C[C@@H](CCC(=O)O)OCc1ccccc1Br ZINC000147465244 CG For-Sale Anodyne FFAR4 46 39 CCNC(=O)c1cccc(N[C@H]2CCO[C@H]2C)c1 ZINC000147465245 BE On-Demand Anodyne KCNK3 47 33 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccccc1OC[C@H]1CCCCO1)C2 ZINC000147465251 GH On-Demand Anodyne ROCK2 32 45 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)no1 ZINC000147465254 FD On-Demand Anodyne HTR4 56 38 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)no1 ZINC000147465254 FD On-Demand Anodyne LPL 45 35 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)no1 ZINC000147465254 FD On-Demand Anodyne EPHX2 31 41 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)no1 ZINC000147465254 FD On-Demand Anodyne TGM2 61 43 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)no1 ZINC000147465254 FD On-Demand Anodyne CACNA1I 51 38 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)no1 ZINC000147465254 FD On-Demand Anodyne F13A1 63 43 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)no1 ZINC000147465254 FD On-Demand Anodyne NAMPT 43 38 Cc1cccc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147465294 CG For-Sale Anodyne ADRB2 63 62 Cc1cccc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147465294 CG For-Sale Anodyne ADRB1 76 63 Cc1cccc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147465294 CG For-Sale Anodyne GRIN1 26 41 Cc1cccc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147465294 CG For-Sale Anodyne ADRB3 46 43 Cc1cccc(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147465294 CG For-Sale Anodyne ABCB1 0 43 Cc1ccc(NC[C@H](C)CC(=O)O)cc1[N+](=O)[O-] ZINC000147465301 CE For-Sale Bother COLA 46 33 Cc1nc(NCCc2ccc(F)cc2)ccc1C(=O)O ZINC000147465314 CF For-Sale Anodyne PTGDR 29 48 Cc1nc(NCCc2ccc(F)cc2)ccc1C(=O)O ZINC000147465314 CF For-Sale Anodyne HAO2 42 43 O=C(CCOCC(F)(F)F)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147465377 EF On-Demand Anodyne ATF1 44 34 O=C(CCOCC(F)(F)F)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147465377 EF On-Demand Anodyne NFKB1 41 34 N[C@H](Cc1ccc(O)cc1)[C@H]1COc2ccccc21 ZINC000147465393 CE For-Sale Anodyne YARS 51 33 CCCCc1ccc(OC[C@H](NC)C(C)C)cc1 ZINC000147465395 BH For-Sale Anodyne ADRB1 16 46 CCCCc1ccc(OC[C@H](NC)C(C)C)cc1 ZINC000147465395 BH For-Sale Anodyne SCN2A 16 42 CCCCc1ccc(OC[C@H](NC)C(C)C)cc1 ZINC000147465395 BH For-Sale Anodyne S1PR4 23 45 CCCCc1ccc(OC[C@H](NC)C(C)C)cc1 ZINC000147465395 BH For-Sale Anodyne S1PR2 32 45 CCCCc1ccc(OC[C@H](NC)C(C)C)cc1 ZINC000147465395 BH For-Sale Anodyne S1PR5 16 45 C[C@H](CCC(=O)O)OCc1ccccc1Br ZINC000147465446 CG For-Sale Anodyne THRA 15 40 C[C@H](CCC(=O)O)OCc1ccccc1Br ZINC000147465446 CG For-Sale Anodyne FFAR1 25 51 C[C@H](CCC(=O)O)OCc1ccccc1Br ZINC000147465446 CG For-Sale Anodyne FFAR4 46 39 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccccc1F ZINC000147465447 HF On-Demand Anodyne ADRB2 19 42 O=C(NC[C@H](O)COc1cccc(Cl)c1Cl)C(=O)Nc1ccccc1F ZINC000147465447 HF On-Demand Anodyne ADRB1 57 48 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccccc1OC[C@H]1CCCCO1)C2 ZINC000147465467 GH On-Demand Anodyne ROCK2 32 45 Cc1cccc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147465512 CG For-Sale Anodyne ADRB2 63 62 Cc1cccc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147465512 CG For-Sale Anodyne ADRB1 76 63 Cc1cccc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147465512 CG For-Sale Anodyne GRIN1 26 41 Cc1cccc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147465512 CG For-Sale Anodyne ADRB3 46 43 Cc1cccc(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147465512 CG For-Sale Anodyne ABCB1 0 43 COc1cc(-c2nc(-c3ccccc3N)no2)ccc1F ZINC000147465521 CG For-Sale Anodyne LUCI_PHOPE 54 57 COC(=O)[C@H](NC(=O)c1cc2cc(Cl)ccc2o1)c1ccccc1 ZINC000147465529 EH On-Demand Anodyne TACR3 15 49 CCCCCCCCCCCCC(=O)c1cncs1 ZINC000147465537 CK For-Sale Mild CDC25B 65 38 CCCCCCCCCCCCC(=O)c1cncs1 ZINC000147465537 CK For-Sale Mild FAAH 27 47 CCCCCCCCCCCCC(=O)c1cncs1 ZINC000147465537 CK For-Sale Mild FFAR1 0 43 CCCCCCCCCCCCC(=O)c1cncs1 ZINC000147465537 CK For-Sale Mild CQSS 56 34 CN(CCCNC(=O)C1(N)CCC1)Cc1ccccc1 ZINC000147465546 CD On-Demand Anodyne ACHE 28 45 Cc1ccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465557 HF On-Demand Anodyne MMP13 55 45 Cc1ccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465557 HF On-Demand Anodyne MMP2 41 38 Cc1ccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465557 HF On-Demand Anodyne MMP3 41 38 Cc1ccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465557 HF On-Demand Anodyne EPHX2 32 43 Cc1ccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465557 HF On-Demand Anodyne TGM2 60 43 Cc1ccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465557 HF On-Demand Anodyne MMP1 36 44 Cc1ccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465557 HF On-Demand Anodyne F13A1 60 43 CCS(=O)(=O)N1CCC(NC(=O)N(C)Cc2cscn2)CC1 ZINC000147465589 ED On-Demand Anodyne NPY2R 15 46 CC1(C)C[C@@H]1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147465593 CF For-Sale Anodyne CACNA1I 40 31 N[C@@H](Cc1ccc(O)cc1)[C@@H]1COc2ccccc21 ZINC000147465611 CE For-Sale Anodyne YARS 51 33 CCCCc1ccc(OC[C@@H](NC)C(C)C)cc1 ZINC000147465614 BH For-Sale Anodyne ADRB1 16 46 CCCCc1ccc(OC[C@@H](NC)C(C)C)cc1 ZINC000147465614 BH For-Sale Anodyne SCN2A 16 42 CCCCc1ccc(OC[C@@H](NC)C(C)C)cc1 ZINC000147465614 BH For-Sale Anodyne S1PR4 23 45 CCCCc1ccc(OC[C@@H](NC)C(C)C)cc1 ZINC000147465614 BH For-Sale Anodyne S1PR2 32 45 CCCCc1ccc(OC[C@@H](NC)C(C)C)cc1 ZINC000147465614 BH For-Sale Anodyne S1PR5 16 45 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive CACNA2D1 41 42 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive GRIA3 24 44 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive GRM8 28 44 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive GRIA1 20 44 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive GRIA2 20 44 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive GRIK3 47 44 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive GCLC 65 31 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive GRIA4 16 44 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive GRIK5 28 44 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive GRIK2 28 44 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive KYNU 57 31 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive GRIK1 57 44 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive SLC17A8 0 41 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive KIF11 34 41 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive GLNA 59 37 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive LUXS 57 35 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive BHMT 61 39 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive ASD 0 50 N[C@@H](CSCl)C(=O)O ZINC000147465669 AC For-Sale Reactive BHMT2 58 38 CCc1ncc(C(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)s1 ZINC000147465684 FG On-Demand Anodyne PTR1 50 36 CCc1ncc(C(=O)NCc2ccc(C(=O)N3CCCCC3)cc2)s1 ZINC000147465684 FG On-Demand Anodyne L3MBTL3 60 36 Cc1ccc(C)c(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147465693 HG On-Demand Anodyne ADRB2 24 45 Cc1ccc(C)c(NC(=O)C(=O)NC[C@H](O)COc2cccc(Cl)c2Cl)c1 ZINC000147465693 HG On-Demand Anodyne ADRB1 56 36 COc1ccc(CCC(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147465701 FH For-Sale Reactive FKBP1A 29 42 COc1ccc(CCC(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147465701 FH For-Sale Reactive SLC18A2 35 43 COc1ccc(CCC(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147465701 FH For-Sale Reactive FKBP12.6 0 42 COc1ccc(CCC(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147465701 FH For-Sale Reactive FAP 0 44 COC(=O)COCc1cccc(Br)c1 ZINC000147465707 CE For-Sale Anodyne HCAR2 16 48 Cc1ccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465774 HF On-Demand Anodyne MMP13 55 45 Cc1ccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465774 HF On-Demand Anodyne MMP2 41 38 Cc1ccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465774 HF On-Demand Anodyne MMP3 41 38 Cc1ccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465774 HF On-Demand Anodyne EPHX2 32 43 Cc1ccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465774 HF On-Demand Anodyne TGM2 60 43 Cc1ccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465774 HF On-Demand Anodyne MMP1 36 44 Cc1ccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147465774 HF On-Demand Anodyne F13A1 60 43 NC1(C(=O)Nc2ccc3c(c2)OC(F)(F)O3)CCC1 ZINC000147465784 CD On-Demand Anodyne BRAF 30 40 COc1cc(Cl)c(C)cc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147465788 DH For-Sale Anodyne AKR1C2 70 38 CC1(C)C[C@H]1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147465794 CF For-Sale Anodyne CACNA1I 40 31 N[C@@H](Cc1ccc(O)cc1)[C@H]1COc2ccccc21 ZINC000147465807 CE For-Sale Anodyne YARS 51 33 CCCCc1ccc(OC[C@H](N)C(C)C)cc1 ZINC000147465843 BG For-Sale Anodyne SCN2A 18 41 CCCCc1ccc(OC[C@H](N)C(C)C)cc1 ZINC000147465843 BG For-Sale Anodyne S1PR4 30 50 CCCCc1ccc(OC[C@H](N)C(C)C)cc1 ZINC000147465843 BG For-Sale Anodyne S1PR3 20 50 CCCCc1ccc(OC[C@H](N)C(C)C)cc1 ZINC000147465843 BG For-Sale Anodyne S1PR2 29 50 CCCCc1ccc(OC[C@H](N)C(C)C)cc1 ZINC000147465843 BG For-Sale Anodyne S1PR5 27 50 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive CACNA2D1 31 41 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive GRIA3 25 44 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive GRM8 28 44 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive GRIA1 20 44 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive GRIA2 20 44 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive GRIK3 47 44 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive GCLC 65 31 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive GRIA4 16 44 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive GRIK5 28 44 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive GRIK2 48 44 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive KYNU 57 31 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive GRIK1 57 44 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive SLC17A8 0 41 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive KIF11 26 41 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive GLNA 59 37 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive LUXS 57 35 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive BHMT 61 39 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive ASD 0 50 N[C@H](CSCl)C(=O)O ZINC000147465846 AC For-Sale Reactive BHMT2 58 38 COc1ccsc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147465856 DG On-Demand Anodyne F10 50 33 COc1ccsc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147465856 DG On-Demand Anodyne COLA 74 38 COc1ccsc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147465856 DG On-Demand Anodyne CPT1A 72 38 COc1ccsc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147465856 DG On-Demand Anodyne CPT2 47 37 COc1ccsc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147465856 DG On-Demand Anodyne CPT1B 53 37 COc1ccc(OC)c(CNC(=O)NNC(=O)c2ccc(C)s2)c1 ZINC000147465860 EE On-Demand Reactive MTNR1B 24 44 COc1ccc(OC)c(CNC(=O)NNC(=O)c2ccc(C)s2)c1 ZINC000147465860 EE On-Demand Reactive MT-ND1 18 49 O=C(N[C@@H]1CCc2cc(Cl)ccc21)c1ccc2c(c1)COC2 ZINC000147465870 DH On-Demand Anodyne BDKRB1 18 40 COc1ccc(CCC(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147465899 FH For-Sale Reactive FKBP1A 29 42 COc1ccc(CCC(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147465899 FH For-Sale Reactive SLC18A2 35 43 COc1ccc(CCC(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147465899 FH For-Sale Reactive FKBP12.6 0 42 COc1ccc(CCC(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147465899 FH For-Sale Reactive FAP 0 44 CCc1ncc(C(=O)NCCOc2ccc3ccccc3c2)s1 ZINC000147465904 EH On-Demand Anodyne MTNR1A 42 41 CCc1ncc(C(=O)NCCOc2ccc3ccccc3c2)s1 ZINC000147465904 EH On-Demand Anodyne MTNR1B 26 41 C[C@H](CNc1cc(F)ccc1[N+](=O)[O-])CC(=O)O ZINC000147465914 CE For-Sale Bother COLA 41 37 Nc1ccccc1-c1noc(-c2cccc(Cl)c2F)n1 ZINC000147465941 CH For-Sale Anodyne LUCI_PHOPE 31 40 O=C(O)CCCCOCc1cccc(Br)c1 ZINC000147465953 CG For-Sale Anodyne TBXAS1 15 40 O=C(O)CCCCOCc1cccc(Br)c1 ZINC000147465953 CG For-Sale Anodyne FFAR1 42 56 O=C(O)CCCCOCc1cccc(Br)c1 ZINC000147465953 CG For-Sale Anodyne FFAR4 23 56 NCC1(CC(=O)Nc2ccc3c(c2)OC(F)(F)O3)CCC1 ZINC000147465992 CE For-Sale Anodyne KIT 23 40 NCC1(CC(=O)Nc2ccc3c(c2)OC(F)(F)O3)CCC1 ZINC000147465992 CE For-Sale Anodyne BRAF 30 40 CCCNc1cncc(Oc2ccc(OCCC)cc2)n1 ZINC000147465994 CH For-Sale Anodyne ACACA 34 41 CCCNc1cncc(Oc2ccc(OCCC)cc2)n1 ZINC000147465994 CH For-Sale Anodyne ACACB 18 41 O=C(CCCc1cccs1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147466014 HG On-Demand Anodyne ADAM17 17 42 O=C(CCCc1cccs1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147466014 HG On-Demand Anodyne EPHX2 17 41 O=C(CCCc1cccs1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147466014 HG On-Demand Anodyne PTPRF 18 40 O=C(CCCc1cccs1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147466014 HG On-Demand Anodyne TGM2 77 44 O=C(CCCc1cccs1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147466014 HG On-Demand Anodyne F13A1 83 44 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne OPRD1 15 42 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne ANPEP 21 40 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne NPY1R 36 45 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne KLK3 59 38 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne NPFFR2 34 44 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne GRIA1 76 38 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne PCSK5 62 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne FURIN 69 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne CAPN2 58 39 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne F7 20 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne TPSAB1 17 43 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne PROC 49 39 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne POLG_WNV 65 34 CCCC[C@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466026 DD On-Demand Anodyne NPFFR1 53 44 CCCCc1ccc(OC[C@@H](N)C(C)C)cc1 ZINC000147466032 BG For-Sale Anodyne SCN2A 18 41 CCCCc1ccc(OC[C@@H](N)C(C)C)cc1 ZINC000147466032 BG For-Sale Anodyne S1PR4 30 50 CCCCc1ccc(OC[C@@H](N)C(C)C)cc1 ZINC000147466032 BG For-Sale Anodyne S1PR3 20 50 CCCCc1ccc(OC[C@@H](N)C(C)C)cc1 ZINC000147466032 BG For-Sale Anodyne S1PR2 29 50 CCCCc1ccc(OC[C@@H](N)C(C)C)cc1 ZINC000147466032 BG For-Sale Anodyne S1PR5 27 50 Cn1cc(CNC(=O)Nc2cc(Br)cc(C(=O)O)c2)cn1 ZINC000147466039 FE For-Sale Anodyne NAMPT 33 42 Cc1nc(Nc2ccccc2C(F)(F)F)ccc1C(=O)O ZINC000147466057 CH For-Sale Anodyne SORT1 29 43 Cc1nc(Nc2ccccc2C(F)(F)F)ccc1C(=O)O ZINC000147466057 CH For-Sale Anodyne MAPK8 20 41 Cc1nc(Nc2ccccc2C(F)(F)F)ccc1C(=O)O ZINC000147466057 CH For-Sale Anodyne RBP4 82 41 Cc1nc(Nc2ccccc2C(F)(F)F)ccc1C(=O)O ZINC000147466057 CH For-Sale Anodyne AKR1C3 29 49 Cc1nc(Nc2ccccc2C(F)(F)F)ccc1C(=O)O ZINC000147466057 CH For-Sale Anodyne AKR1C2 59 39 CCN(CC)[C@H](C)CNC(=O)CCNS(=O)(=O)c1ccc(C)c(C)c1 ZINC000147466075 FD On-Demand Anodyne LEF 44 35 C[C@@H](CSCl)C(=O)O ZINC000147466078 AD For-Sale Reactive BHMT2 44 29 CCCN(C(=O)c1ccc2c(c1)COC2)[C@@H]1CCc2ccccc2C1 ZINC000147466093 EI On-Demand Anodyne HTR1A 20 49 CCCN(C(=O)c1ccc2c(c1)COC2)[C@@H]1CCc2ccccc2C1 ZINC000147466093 EI On-Demand Anodyne DRD2 23 42 CCCN(C(=O)c1ccc2c(c1)COC2)[C@@H]1CCc2ccccc2C1 ZINC000147466093 EI On-Demand Anodyne HTR1D 18 40 CCCN(C(=O)c1ccc2c(c1)COC2)[C@@H]1CCc2ccccc2C1 ZINC000147466093 EI On-Demand Anodyne HTR1B 17 40 CCCN(C(=O)c1ccc2c(c1)COC2)[C@@H]1CCc2ccccc2C1 ZINC000147466093 EI On-Demand Anodyne DRD3 36 42 C=Cc1ccc2cc(OC)ccc2c1Cl ZINC000147466111 BI For-Sale Anodyne CYP1B1 45 43 C=Cc1ccc2cc(OC)ccc2c1Cl ZINC000147466111 BI For-Sale Anodyne AHR 23 40 C=Cc1ccc2cc(OC)ccc2c1Cl ZINC000147466111 BI For-Sale Anodyne CYP1A1 40 43 C=Cc1ccc2cc(OC)ccc2c1Cl ZINC000147466111 BI For-Sale Anodyne CYP1A2 20 43 C[C@@H](CNc1cc(F)ccc1[N+](=O)[O-])CC(=O)O ZINC000147466121 CE For-Sale Bother COLA 41 37 CC(C)[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466172 CG For-Sale Anodyne SLC1A6 0 48 CC(C)[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466172 CG For-Sale Anodyne SLC1A7 0 48 CC(C)[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466172 CG For-Sale Anodyne FFAR1 19 46 CC(C)CCCCNC(=O)CC[C@@H](C)N ZINC000147466173 BE For-Sale Anodyne NOD1 46 45 NC1(C(=O)Nc2ccccc2OC(F)(F)F)CCC1 ZINC000147466203 CE For-Sale Anodyne P2RY1 55 40 CCCOc1ccc(Oc2cncc(NCC)n2)cc1 ZINC000147466216 CG For-Sale Anodyne ACACA 34 41 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne ANPEP 21 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne NPY1R 28 45 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne KLK3 59 38 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne NPFFR2 34 44 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne GRIA1 76 38 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne PCSK5 62 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne FURIN 69 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne CAPN2 58 39 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne F7 20 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne TPSAB1 17 43 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne PROC 49 39 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne POLG_WNV 65 34 CCCC[C@@H](NC(N)=O)C(=O)NCc1ccc(COC)cc1 ZINC000147466231 DD On-Demand Anodyne NPFFR1 53 44 CCNC(=O)c1ccc(NC(=O)N2CCC(NC(=O)c3ccoc3)CC2)cc1 ZINC000147466262 GE On-Demand Anodyne EPHX2 36 42 Cn1cc(CNC(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147466263 DE On-Demand Anodyne CACNA1I 56 38 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne KIT 15 43 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne LCK 29 40 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne KDR 17 40 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne NPY5R 18 46 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne SORT1 34 52 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne TEK 25 40 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne BTK 24 40 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne AKR1C3 50 57 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne SHH 23 41 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne AKR1C4 0 40 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne AKR1C2 58 59 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne UL23 0 40 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne TRPM4 0 59 Cc1nc(Nc2cccc(C(F)(F)F)c2)ccc1C(=O)O ZINC000147466268 CH For-Sale Anodyne KCNK3 21 42 C[C@H](CSCl)C(=O)O ZINC000147466280 AD For-Sale Reactive BHMT2 44 29 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1[N+](=O)[O-] ZINC000147466321 HF On-Demand Bother TGM2 65 44 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1[N+](=O)[O-] ZINC000147466321 HF On-Demand Bother CACNA1I 63 41 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1[N+](=O)[O-] ZINC000147466321 HF On-Demand Bother F13A1 59 42 CCOC(=O)Cc1csc(-c2ccc(F)cc2Cl)n1 ZINC000147466334 CH For-Sale Anodyne P2RX7 41 37 Nc1ccc(Cl)c(C(=O)Nc2ccncc2Br)c1 ZINC000147466339 EG For-Sale Anodyne TYK2 16 51 Nc1ccc(Cl)c(C(=O)Nc2ccncc2Br)c1 ZINC000147466339 EG For-Sale Anodyne CSF1R 15 43 C[C@H](CNc1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147466351 CD On-Demand Anodyne PTGS2 19 46 C[C@H](CNc1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147466351 CD On-Demand Anodyne O49150_SOLTU 41 34 CC(C)CCCCNC(=O)CC[C@H](C)N ZINC000147466357 BE For-Sale Anodyne NOD1 46 45 CC(C)[C@@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466375 CG For-Sale Anodyne SLC1A6 0 48 CC(C)[C@@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466375 CG For-Sale Anodyne SLC1A7 0 48 CC(C)[C@@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466375 CG For-Sale Anodyne FFAR1 19 46 CCCCCCCCCCN1CC[C@H](N)[C@H](CC)C1 ZINC000147466402 CI For-Sale Mild GNAI1 0 46 CCCCCCCCCCN1CC[C@H](N)[C@H](CC)C1 ZINC000147466402 CI For-Sale Mild GNAI3 0 46 CCCCCCCCCCN1CC[C@H](N)[C@H](CC)C1 ZINC000147466402 CI For-Sale Mild GNAO1 0 46 CCCCCCCCCCN1CC[C@H](N)[C@H](CC)C1 ZINC000147466402 CI For-Sale Mild ZM.86993 0 43 O=C(Nc1cc(Cl)ccc1Br)c1ccncc1F ZINC000147466412 EH On-Demand Anodyne GRM4 21 41 O=C(Nc1cc(Cl)ccc1Br)c1ccncc1F ZINC000147466412 EH On-Demand Anodyne KCNMA1 25 43 N#C[C@@]12C[C@@H]1CN(Cc1ccccc1)C2 ZINC000147466424 AE For-Sale Mild SIGMAR1 43 43 O=C(CCc1cccs1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147466482 DH On-Demand Anodyne PTPRF 19 42 COC(=O)[C@@H](NC(=O)c1cc2cc(Cl)ccc2o1)c1ccccc1 ZINC000147466487 EH On-Demand Anodyne TACR3 15 49 C[C@@H](CNc1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147466538 CD On-Demand Anodyne PTGS2 19 46 C[C@@H](CNc1ccc(S(C)(=O)=O)cc1)CC(=O)O ZINC000147466538 CD On-Demand Anodyne O49150_SOLTU 41 34 Cc1cccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466570 HF On-Demand Anodyne CHRM5 19 41 Cc1cccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466570 HF On-Demand Anodyne MMP13 26 40 Cc1cccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466570 HF On-Demand Anodyne EPHX2 36 43 Cc1cccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466570 HF On-Demand Anodyne TGM2 59 42 Cc1cccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466570 HF On-Demand Anodyne CACNA1I 41 33 Cc1cccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466570 HF On-Demand Anodyne F13A1 54 42 Cc1cccc(O[C@@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466570 HF On-Demand Anodyne AKR1C3 43 36 Cc1c(N)cccc1C(=O)Nc1ccncc1Br ZINC000147466581 DF For-Sale Anodyne G2YM83_BOTF4 43 31 C[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466585 CE For-Sale Anodyne MAOB 21 50 C[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466585 CE For-Sale Anodyne SLC1A6 0 40 C[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466585 CE For-Sale Anodyne SLC1A7 0 40 C[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466585 CE For-Sale Anodyne ADAMTS4 24 50 C[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466585 CE For-Sale Anodyne FFAR1 38 51 C[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147466585 CE For-Sale Anodyne PDS 51 42 C[C@@H](NC(=O)c1ccc2c(c1)COC2)c1ccc(F)c(Cl)c1 ZINC000147466608 DI On-Demand Anodyne UTS2 41 32 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne DRD4 23 49 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne LTA4H 15 45 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne SCN2A 21 45 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne S1PR4 41 47 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne LPAR2 45 50 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne S1PR3 56 50 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne SLC2A1 26 41 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne PLA2G4B 79 38 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne FAAH 16 40 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne S1PR2 81 50 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne S1PR1 28 50 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne S1PR5 28 48 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne CYP1A2 15 41 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne CYP2C19 19 41 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne TAAR1 21 43 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne HT1 0 41 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne PPO2 22 44 CCCCc1ccc(OCCCNCCC)cc1 ZINC000147466620 BH For-Sale Anodyne LMGT2 0 41 CCCCCCCCCCN1CC[C@@H](N)[C@H](CC)C1 ZINC000147466626 CI For-Sale Mild GNAI1 0 46 CCCCCCCCCCN1CC[C@@H](N)[C@H](CC)C1 ZINC000147466626 CI For-Sale Mild GNAI3 0 46 CCCCCCCCCCN1CC[C@@H](N)[C@H](CC)C1 ZINC000147466626 CI For-Sale Mild GNAO1 0 46 CCCCCCCCCCN1CC[C@@H](N)[C@H](CC)C1 ZINC000147466626 CI For-Sale Mild ZM.86993 0 43 Cc1nc(Nc2ccc(C(C)(C)C)cc2)ccc1C(=O)O ZINC000147466699 CI For-Sale Anodyne SORT1 30 43 Cc1nc(Nc2ccc(C(C)(C)C)cc2)ccc1C(=O)O ZINC000147466699 CI For-Sale Anodyne AKR1C3 40 54 Cc1nc(Nc2ccc(C(C)(C)C)cc2)ccc1C(=O)O ZINC000147466699 CI For-Sale Anodyne AKR1C2 76 50 CSCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147466702 CE On-Demand Anodyne CACNA1H 15 40 CSCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147466702 CE On-Demand Anodyne CACNA1I 50 34 CSCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147466702 CE On-Demand Anodyne HCAR1 0 42 C[C@H](CNc1ccc(S(=O)(=O)C(F)(F)F)cc1)CC(=O)O ZINC000147466766 EF For-Sale Anodyne CA2 18 45 CCNC(=O)c1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147466772 HI On-Demand Anodyne RAF1 32 40 CCNC(=O)c1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147466772 HI On-Demand Anodyne ROCK2 41 49 CCNC(=O)c1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147466772 HI On-Demand Anodyne MET 50 45 CCNC(=O)c1ccc(NC(=O)NCc2ccc(Oc3cccnc3)c(F)c2)cc1 ZINC000147466772 HI On-Demand Anodyne NAMPT 86 49 Cc1cccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466778 HF On-Demand Anodyne CHRM5 19 41 Cc1cccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466778 HF On-Demand Anodyne MMP13 26 40 Cc1cccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466778 HF On-Demand Anodyne EPHX2 36 43 Cc1cccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466778 HF On-Demand Anodyne TGM2 59 42 Cc1cccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466778 HF On-Demand Anodyne CACNA1I 41 33 Cc1cccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466778 HF On-Demand Anodyne F13A1 54 42 Cc1cccc(O[C@H](C)C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147466778 HF On-Demand Anodyne AKR1C3 43 36 O=C(O)[C@@H](OCc1cccc(Br)c1)C1CC1 ZINC000147466834 CF For-Sale Anodyne HCAR2 16 47 O=C(O)[C@@H](OCc1cccc(Br)c1)C1CC1 ZINC000147466834 CF For-Sale Anodyne FFAR1 19 47 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne DRTS_PLAFK 18 44 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne DRD4 19 40 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne INHA 44 33 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne LTA4H 28 41 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne SCN2A 23 47 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne S1PR4 34 49 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne LPAR2 41 49 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne S1PR3 47 49 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne SLC2A1 22 43 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne PLA2G4B 82 40 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne FAAH 17 41 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne S1PR2 68 49 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne S1PR1 25 49 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne S1PR5 28 49 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne CYP1A2 15 43 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne CYP2C9 16 43 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne CYP2C19 20 43 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne TAAR1 29 54 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne HT1 0 43 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne PPO2 24 46 CCCCc1ccc(OCCCNC)cc1 ZINC000147466841 BG For-Sale Anodyne LMGT2 0 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne AVPR2 49 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne AVPR1A 26 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne DHODH 18 51 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne PPIA 17 49 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne JUN 22 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne ECR 62 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne ATF1 57 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne PYGL 22 50 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne PRNP 26 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne GRM4 54 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne NR1H4 17 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne F12 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne NFKB1 53 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne TYK2 25 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne ACPS 0 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne EPHB3 41 36 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne TAAR1 15 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne AKR1C3 46 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne NR2E3 72 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne SHH 49 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne CYA 0 48 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne AKR1C2 36 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne SMO 35 61 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne GALE 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne HCAR1 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne Q25615_ONCVO 49 33 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne KCNK3 100 60 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Cl)c1 ZINC000147466916 DH On-Demand Anodyne KCNK9 72 38 NCC1(CC(=O)Nc2ccc(Cl)c(Cl)c2)CCC1 ZINC000147466921 CG For-Sale Anodyne SLC1A1 35 40 NCC1(CC(=O)Nc2ccc(Cl)c(Cl)c2)CCC1 ZINC000147466921 CG For-Sale Anodyne SLC1A3 40 40 NCC1(CC(=O)Nc2ccc(Cl)c(Cl)c2)CCC1 ZINC000147466921 CG For-Sale Anodyne SLC1A2 34 40 NCC1(CC(=O)Nc2ccc(Cl)c(Cl)c2)CCC1 ZINC000147466921 CG For-Sale Anodyne ENV 42 34 NCC1(CC(=O)Nc2ccc(Cl)c(Cl)c2)CCC1 ZINC000147466921 CG For-Sale Anodyne IMDH_CRYPV 31 41 NCC1(CC(=O)Nc2ccc(Cl)c(Cl)c2)CCC1 ZINC000147466921 CG For-Sale Anodyne P95276_MYCTO 0 44 NCC1(CC(=O)Nc2ccc(Cl)c(Cl)c2)CCC1 ZINC000147466921 CG For-Sale Anodyne PPX1 0 43 O=C(NC[C@H]1CC=CCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147466927 DH On-Demand Anodyne CACNA1I 73 42 CCCOc1ccc(Oc2cc(NCC)ncn2)cc1 ZINC000147466946 CG For-Sale Anodyne ACACA 35 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne DRD2 21 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne DRD4 21 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne ACHE 15 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne DRD3 15 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne HTR4 66 39 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne GRIN2B 28 47 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne SIGMAR1 19 49 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne CCR3 48 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne EPHX2 30 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne TGM2 74 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne CACNA1I 90 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne F13A1 71 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne AKR1C3 57 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne SFRP1 57 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cc(F)cc(F)c1 ZINC000147466991 GF On-Demand Anodyne NAMPT 45 41 C[C@@H](CNc1ccc(S(=O)(=O)C(F)(F)F)cc1)CC(=O)O ZINC000147466994 EF For-Sale Anodyne CA2 18 45 CC(C)CCCCNC(=O)[C@H](N)CC(=O)O ZINC000147467003 BC For-Sale Anodyne NOS3 15 43 CC(C)CCCCNC(=O)[C@H](N)CC(=O)O ZINC000147467003 BC For-Sale Anodyne DNPEP 0 40 CC(C)CCCCNC(=O)[C@H](N)CC(=O)O ZINC000147467003 BC For-Sale Anodyne ENPEP 44 30 CC(C)CCCCNC(=O)[C@H](N)CC(=O)O ZINC000147467003 BC For-Sale Anodyne SIRT1 46 43 CC(C)CCCCNC(=O)[C@H](N)CC(=O)O ZINC000147467003 BC For-Sale Anodyne SLC15A2 0 48 CC(C)CCCCNC(=O)[C@H](N)CC(=O)O ZINC000147467003 BC For-Sale Anodyne NOD1 34 43 CCNC(=O)c1ccc(NC(=O)NC[C@@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147467023 GH On-Demand Anodyne MTOR 52 41 O=C(O)[C@H](OCc1cccc(Br)c1)C1CC1 ZINC000147467038 CF For-Sale Anodyne HCAR2 16 47 O=C(O)[C@H](OCc1cccc(Br)c1)C1CC1 ZINC000147467038 CF For-Sale Anodyne FFAR1 19 47 CCc1ncc(C(=O)N(C)CCOc2cccc(C)c2)s1 ZINC000147467044 DG On-Demand Anodyne HSD17B2 29 44 O=C(NC[C@@H]1CC=CCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147467106 DH On-Demand Anodyne CACNA1I 73 42 CCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147467108 CG On-Demand Anodyne ACAT 0 46 CCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147467108 CG On-Demand Anodyne HCAR1 0 41 CCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147467108 CG On-Demand Anodyne PARP10 0 40 CCOC(=O)c1ncc(OCC)cc1OCC ZINC000147467117 BE For-Sale Anodyne GABRA5 40 31 O=C(O)[C@@H]1Cc2cc(S(=O)(=O)N3CCCC3)ccc2O1 ZINC000147467163 CC On-Demand Anodyne EPHX2 17 47 O=C(O)[C@@H]1Cc2cc(S(=O)(=O)N3CCCC3)ccc2O1 ZINC000147467163 CC On-Demand Anodyne PKM 34 43 O=C(O)[C@@H]1Cc2cc(S(=O)(=O)N3CCCC3)ccc2O1 ZINC000147467163 CC On-Demand Anodyne AKR1C3 55 44 O=C(O)[C@@H]1Cc2cc(S(=O)(=O)N3CCCC3)ccc2O1 ZINC000147467163 CC On-Demand Anodyne AKR1C1 22 40 CC(C)CCCCNC(=O)[C@@H](N)CC(=O)O ZINC000147467184 BC For-Sale Anodyne NOS3 15 43 CC(C)CCCCNC(=O)[C@@H](N)CC(=O)O ZINC000147467184 BC For-Sale Anodyne DNPEP 0 40 CC(C)CCCCNC(=O)[C@@H](N)CC(=O)O ZINC000147467184 BC For-Sale Anodyne ENPEP 44 30 CC(C)CCCCNC(=O)[C@@H](N)CC(=O)O ZINC000147467184 BC For-Sale Anodyne SIRT1 46 43 CC(C)CCCCNC(=O)[C@@H](N)CC(=O)O ZINC000147467184 BC For-Sale Anodyne SLC15A2 0 48 CC(C)CCCCNC(=O)[C@@H](N)CC(=O)O ZINC000147467184 BC For-Sale Anodyne NOD1 34 43 COc1cc(-c2nc(-c3ccc(N)cc3)no2)ccc1F ZINC000147467190 CG For-Sale Anodyne LUCI_PHOPE 42 48 CCCCc1ccc(OC[C@H](NCCC)C(C)C)cc1 ZINC000147467194 CI For-Sale Anodyne ADRB1 17 47 CCCCc1ccc(OC[C@H](NCCC)C(C)C)cc1 ZINC000147467194 CI For-Sale Anodyne SCN2A 18 40 CCCCc1ccc(OC[C@H](NCCC)C(C)C)cc1 ZINC000147467194 CI For-Sale Anodyne S1PR4 25 43 CCCCc1ccc(OC[C@H](NCCC)C(C)C)cc1 ZINC000147467194 CI For-Sale Anodyne S1PR3 21 43 CCCCc1ccc(OC[C@H](NCCC)C(C)C)cc1 ZINC000147467194 CI For-Sale Anodyne S1PR2 41 43 CCCCc1ccc(OC[C@H](NCCC)C(C)C)cc1 ZINC000147467194 CI For-Sale Anodyne S1PR5 16 43 Cc1nc(Nc2cccc3c2CCCC3)ccc1C(=O)O ZINC000147467199 CH For-Sale Anodyne NISCH 18 48 Cc1nc(Nc2cccc3c2CCCC3)ccc1C(=O)O ZINC000147467199 CH For-Sale Anodyne AKR1C2 42 39 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne HTR1A 26 41 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne DRD2 43 46 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne DRD4 27 44 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne ACHE 18 44 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne ADRA1D 27 41 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne ADRA1A 22 41 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne ADRA1B 22 41 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne DRD3 40 41 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne HTR4 46 37 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne CHRM5 27 42 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne TACR1 25 42 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne HTR7 24 40 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne SIGMAR1 15 50 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne MMP13 30 40 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne CCR3 25 42 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne KCNA3 42 37 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne ADAM17 18 42 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne MMP2 18 41 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne MMP3 33 40 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne MMP8 18 40 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne MMP9 24 40 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne EPHX2 27 43 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne TGM2 70 55 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne MMP7 31 40 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne MMP1 30 40 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne CACNA1I 57 39 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne F13A1 74 44 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne MBTPS1 54 36 COc1ccccc1CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467204 HE On-Demand Anodyne ACKR3 48 35 CCCCNC(=O)COc1cc(F)c(S(N)(=O)=O)cc1Br ZINC000147467229 GD For-Sale Anodyne ASAH1 41 32 CCNC(=O)c1ccc(NC(=O)NC[C@H]2CCCO[C@@H]2c2ccccc2)cc1 ZINC000147467232 GH On-Demand Anodyne MTOR 52 41 COC(=O)CCOCc1cccc(Br)c1 ZINC000147467250 CF In-Stock Anodyne HCAR2 15 46 CCOC(=O)Cc1csc(-c2cc(F)cc(Br)c2)n1 ZINC000147467268 EH For-Sale Anodyne DCK 40 34 O=C(c1nccc2ccccc12)N1CCC[C@@H]1CCCBr ZINC000147467285 EI For-Sale Reactive HCRTR1 32 48 O=C(c1nccc2ccccc12)N1CCC[C@@H]1CCCBr ZINC000147467285 EI For-Sale Reactive HCRTR2 25 48 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2F)c1 ZINC000147467330 DH On-Demand Anodyne ATF1 56 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2F)c1 ZINC000147467330 DH On-Demand Anodyne CPT1A 27 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2F)c1 ZINC000147467330 DH On-Demand Anodyne PYGL 16 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2F)c1 ZINC000147467330 DH On-Demand Anodyne NFKB1 52 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2F)c1 ZINC000147467330 DH On-Demand Anodyne KCNK3 42 38 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2F)c1 ZINC000147467330 DH On-Demand Anodyne TMPRSS4 0 44 O=C(O)[C@H]1Cc2cc(S(=O)(=O)N3CCCC3)ccc2O1 ZINC000147467359 CC On-Demand Anodyne EPHX2 17 47 O=C(O)[C@H]1Cc2cc(S(=O)(=O)N3CCCC3)ccc2O1 ZINC000147467359 CC On-Demand Anodyne PKM 34 43 O=C(O)[C@H]1Cc2cc(S(=O)(=O)N3CCCC3)ccc2O1 ZINC000147467359 CC On-Demand Anodyne AKR1C3 55 44 O=C(O)[C@H]1Cc2cc(S(=O)(=O)N3CCCC3)ccc2O1 ZINC000147467359 CC On-Demand Anodyne AKR1C1 22 40 CCCCc1ccc(OC[C@@H](NCCC)C(C)C)cc1 ZINC000147467403 CI For-Sale Anodyne ADRB1 17 47 CCCCc1ccc(OC[C@@H](NCCC)C(C)C)cc1 ZINC000147467403 CI For-Sale Anodyne SCN2A 18 40 CCCCc1ccc(OC[C@@H](NCCC)C(C)C)cc1 ZINC000147467403 CI For-Sale Anodyne S1PR4 25 43 CCCCc1ccc(OC[C@@H](NCCC)C(C)C)cc1 ZINC000147467403 CI For-Sale Anodyne S1PR3 21 43 CCCCc1ccc(OC[C@@H](NCCC)C(C)C)cc1 ZINC000147467403 CI For-Sale Anodyne S1PR2 41 43 CCCCc1ccc(OC[C@@H](NCCC)C(C)C)cc1 ZINC000147467403 CI For-Sale Anodyne S1PR5 16 43 C[C@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467404 CE On-Demand Anodyne PPARA 0 45 C[C@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467404 CE On-Demand Anodyne P2RY1 51 32 C[C@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467404 CE On-Demand Anodyne NPY5R 34 41 C[C@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467404 CE On-Demand Anodyne EPHX2 59 44 C[C@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467404 CE On-Demand Anodyne GIPR 23 41 C[C@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467404 CE On-Demand Anodyne PSBA 0 43 Cc1nc(Nc2cc(Cl)c(Cl)cc2Cl)ccc1C(=O)O ZINC000147467433 EJ For-Sale Anodyne SORT1 25 43 Cc1nc(Nc2cc(Cl)c(Cl)cc2Cl)ccc1C(=O)O ZINC000147467433 EJ For-Sale Anodyne AKR1C2 71 37 Cc1nc(Nc2cc(Cl)c(Cl)cc2Cl)ccc1C(=O)O ZINC000147467433 EJ For-Sale Anodyne AKR1C1 44 37 COc1ccc(N)cc1C(=O)Nc1ccncc1Br ZINC000147467444 DF For-Sale Anodyne KCNMA1 23 40 CSc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467456 HG On-Demand Anodyne HTR4 66 42 CSc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467456 HG On-Demand Anodyne EPHX2 18 43 CSc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467456 HG On-Demand Anodyne TGM2 67 44 CSc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467456 HG On-Demand Anodyne CACNA1I 62 34 CSc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467456 HG On-Demand Anodyne F13A1 68 44 CSc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467456 HG On-Demand Anodyne HCN1 54 30 CCNC(=O)c1ccc(NC(=O)NC[C@@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147467464 GH On-Demand Anodyne MTOR 52 41 CC[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147467477 CF For-Sale Anodyne PPARG 15 43 CC[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147467477 CF For-Sale Anodyne FFAR1 18 46 CC[C@H](OCc1cccc(Br)c1)C(=O)O ZINC000147467477 CF For-Sale Anodyne PDS 60 43 O=C(c1nccc2ccccc12)N1CCC[C@H]1CCCBr ZINC000147467531 EI For-Sale Reactive HCRTR1 32 48 O=C(c1nccc2ccccc12)N1CCC[C@H]1CCCBr ZINC000147467531 EI For-Sale Reactive HCRTR2 25 48 Cc1ccsc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147467595 CH On-Demand Anodyne PPIA 16 41 Cc1ccccc1C1(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CCOCC1 ZINC000147467604 GJ On-Demand Anodyne MDM2 46 32 C[C@H](CNc1ccc(S(=O)(=O)NC2CC2)cc1)CC(=O)O ZINC000147467618 DD For-Sale Anodyne TBXA2R 15 40 C[C@H](CNc1ccc(S(=O)(=O)NC2CC2)cc1)CC(=O)O ZINC000147467618 DD For-Sale Anodyne SFRP1 87 35 C[C@H](CNc1ccc(S(=O)(=O)NC2CC2)cc1)CC(=O)O ZINC000147467618 DD For-Sale Anodyne WNT3 56 35 C[C@@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467622 CE On-Demand Anodyne PPARA 0 45 C[C@@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467622 CE On-Demand Anodyne P2RY1 51 32 C[C@@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467622 CE On-Demand Anodyne NPY5R 34 41 C[C@@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467622 CE On-Demand Anodyne EPHX2 59 44 C[C@@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467622 CE On-Demand Anodyne GIPR 23 41 C[C@@H](O)CN(C)C(=O)Nc1ccc(OC(F)(F)F)cc1 ZINC000147467622 CE On-Demand Anodyne PSBA 0 43 Nc1ccc(-c2noc(-c3cccc(Cl)c3F)n2)cc1 ZINC000147467629 CH For-Sale Anodyne LUCI_PHOPE 39 46 CCNC(=O)c1ccc(NC(=O)NC[C@H]2CCCO[C@H]2c2ccccc2)cc1 ZINC000147467660 GH On-Demand Anodyne MTOR 52 41 CC[C@@H](OCc1cccc(Br)c1)C(=O)O ZINC000147467673 CF For-Sale Anodyne PPARG 15 43 CC[C@@H](OCc1cccc(Br)c1)C(=O)O ZINC000147467673 CF For-Sale Anodyne FFAR1 18 46 CC[C@@H](OCc1cccc(Br)c1)C(=O)O ZINC000147467673 CF For-Sale Anodyne PDS 60 43 O=C(CC1CCCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467682 GG On-Demand Anodyne F2 15 40 O=C(CC1CCCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467682 GG On-Demand Anodyne CHRM5 19 42 O=C(CC1CCCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467682 GG On-Demand Anodyne CAPN1 17 40 O=C(CC1CCCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467682 GG On-Demand Anodyne EPHX2 32 55 O=C(CC1CCCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467682 GG On-Demand Anodyne TGM2 83 49 O=C(CC1CCCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467682 GG On-Demand Anodyne F13A1 87 49 O=C(CC1CCCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467682 GG On-Demand Anodyne AKR1C3 54 37 O=C(CC1CCCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147467682 GG On-Demand Anodyne NAMPT 34 44 CS(=O)(=O)c1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147467757 FF For-Sale Reactive LOX1.1 41 33 CS(=O)(=O)c1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147467757 FF For-Sale Reactive O49150_SOLTU 49 33 C[C@@H](CNc1ccc(S(=O)(=O)NC2CC2)cc1)CC(=O)O ZINC000147467791 DD For-Sale Anodyne TBXA2R 15 40 C[C@@H](CNc1ccc(S(=O)(=O)NC2CC2)cc1)CC(=O)O ZINC000147467791 DD For-Sale Anodyne SFRP1 87 35 C[C@@H](CNc1ccc(S(=O)(=O)NC2CC2)cc1)CC(=O)O ZINC000147467791 DD For-Sale Anodyne WNT3 56 35 Cc1ccccc1C1(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CCOCC1 ZINC000147467794 GJ On-Demand Anodyne MDM2 46 32 COc1ccc(Cl)cc1NC(=O)C1(N)CCC1 ZINC000147467807 CE For-Sale Anodyne COLA 54 34 COc1ccc(Cl)cc1NC(=O)C1(N)CCC1 ZINC000147467807 CE For-Sale Anodyne CPT1A 51 34 COc1ccc(Cl)cc1NC(=O)C1(N)CCC1 ZINC000147467807 CE For-Sale Anodyne KCNMA1 36 43 COc1ccc(Cl)cc1NC(=O)C1(N)CCC1 ZINC000147467807 CE For-Sale Anodyne CPT1B 42 32 COc1ccc(Cl)cc1NC(=O)C1(N)CCC1 ZINC000147467807 CE For-Sale Anodyne RBP4 26 46 O=C(NCC1(CO)CC1)NC12CC3CC(CC(C3)C1)C2 ZINC000147467833 CE For-Sale Anodyne EPHX2 127 63 O=C(NCC1(CO)CC1)NC12CC3CC(CC(C3)C1)C2 ZINC000147467833 CE For-Sale Anodyne P95276_MYCTO 0 45 COC(=O)C[C@@H](C)C(=O)N1CCc2sccc2[C@@H]1c1ccccc1 ZINC000147467878 EG On-Demand Anodyne TRPM8 24 52 CCOC(=O)CCOCc1cccc(Br)c1 ZINC000147467895 CF For-Sale Anodyne HCAR2 16 47 CCOC(=O)CCOCc1cccc(Br)c1 ZINC000147467895 CF For-Sale Anodyne FFAR1 25 44 Cc1ccc(Cn2cnnc2)cc1 ZINC000147467903 AD For-Sale Anodyne CYP11B1 16 60 CS(=O)(=O)c1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147467939 FF For-Sale Reactive LOX1.1 41 33 CS(=O)(=O)c1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147467939 FF For-Sale Reactive O49150_SOLTU 49 33 Cn1nc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccc1=O ZINC000147467950 GC On-Demand Anodyne HTR4 64 40 Cn1nc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccc1=O ZINC000147467950 GC On-Demand Anodyne GRIN2B 23 41 Cn1nc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccc1=O ZINC000147467950 GC On-Demand Anodyne EPHX2 19 42 Cn1nc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccc1=O ZINC000147467950 GC On-Demand Anodyne TGM2 60 43 Cn1nc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccc1=O ZINC000147467950 GC On-Demand Anodyne CACNA1I 59 37 Cn1nc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)ccc1=O ZINC000147467950 GC On-Demand Anodyne F13A1 55 43 CCOc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCc2cc(OC)cc(OC)c2)cc(N2CCCC2=O)c1 ZINC000147467952 KH Annotated Anodyne CTSD 68 60 CCOc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCc2cc(OC)cc(OC)c2)cc(N2CCCC2=O)c1 ZINC000147467952 KH Annotated Anodyne BACE2 72 60 CCOc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCc2cc(OC)cc(OC)c2)cc(N2CCCC2=O)c1 ZINC000147467952 KH Annotated Anodyne BACE1 96 82 CCOc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCc2cc(OC)cc(OC)c2)cc(N2CCCC2=O)c1 ZINC000147467952 KH Annotated Anodyne PLM1_PLAFA 61 46 CCOc1cc(C(=O)N[C@@H](Cc2ccccc2)[C@@H](O)CNCc2cc(OC)cc(OC)c2)cc(N2CCCC2=O)c1 ZINC000147467952 KH Annotated Anodyne PLM2_PLAFA 41 55 Cc1nc(Nc2cccc3ncccc23)ccc1C(=O)O ZINC000147467960 CG For-Sale Anodyne P2RX7 0 45 Cc1nc(Nc2cccc3ncccc23)ccc1C(=O)O ZINC000147467960 CG For-Sale Anodyne MAPK8 16 44 Cc1ccccc1C1(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CCOCC1 ZINC000147467982 GJ On-Demand Anodyne MDM2 46 32 COc1ccc(Cl)cc1NC(=O)CC1(CN)CCC1 ZINC000147468026 CF For-Sale Anodyne CPT1A 43 30 COc1ccc(Cl)cc1NC(=O)CC1(CN)CCC1 ZINC000147468026 CF For-Sale Anodyne RBP4 25 43 CC(C)CCCCNC(=O)CCCCN ZINC000147468064 BE For-Sale Anodyne NMT1 32 52 CC(C)CCCCNC(=O)CCCCN ZINC000147468064 BE For-Sale Anodyne GRIA1 48 39 CC(C)CCCCNC(=O)CCCCN ZINC000147468064 BE For-Sale Anodyne EPHX2 0 40 CC(C)CCCCNC(=O)CCCCN ZINC000147468064 BE For-Sale Anodyne POLG_WNV 62 33 CC(C)CCCCNC(=O)CCCCN ZINC000147468064 BE For-Sale Anodyne PAO 46 37 CC(C)CCCCNC(=O)CCCCN ZINC000147468064 BE For-Sale Anodyne NOD1 45 46 CC(C)CCCCNC(=O)CCCCN ZINC000147468064 BE For-Sale Anodyne APHA 0 42 COC(=O)C[C@@H](C)C(=O)N1CCc2sccc2[C@H]1c1ccccc1 ZINC000147468066 EG On-Demand Anodyne TRPM8 24 52 COc1ccc(C(=O)O)c(NS(=O)(=O)N(C)C(C)C)c1 ZINC000147468143 DD On-Demand Anodyne AKR1C3 29 53 COc1ccc(C(=O)O)c(NS(=O)(=O)N(C)C(C)C)c1 ZINC000147468143 DD On-Demand Anodyne AKR1C2 72 53 CC[C@@H]1CN(CC(=O)Nc2ccccc2F)CC[C@@H]1N ZINC000147468172 CD On-Demand Anodyne DRD4 0 53 O=C(O)/C=C/COCc1cccc(Br)c1 ZINC000147468215 CF For-Sale Anodyne HCAR2 30 63 CCOC(=O)Cc1csc(Cc2cccc(Cl)c2)n1 ZINC000147468216 CG On-Demand Anodyne PTGER1 23 49 CN(C)S(=O)(=O)c1cccc(Nc2ncc(-c3ccc(F)cc3)o2)c1 ZINC000147468230 FG For-Sale Anodyne IMPDH2 0 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)cc(F)c2)c1 ZINC000147468235 DH On-Demand Anodyne PPIA 15 50 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)cc(F)c2)c1 ZINC000147468235 DH On-Demand Anodyne CPT1A 17 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)cc(F)c2)c1 ZINC000147468235 DH On-Demand Anodyne CACNA1I 47 37 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)cc(F)c2)c1 ZINC000147468235 DH On-Demand Anodyne HCAR1 0 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)cc(F)c2)c1 ZINC000147468235 DH On-Demand Anodyne KCNK3 36 41 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)NC3CCCCC3)cc2)C1 ZINC000147468236 HF On-Demand Anodyne HTR4 43 36 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)NC3CCCCC3)cc2)C1 ZINC000147468236 HF On-Demand Anodyne CNR2 17 41 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)NC3CCCCC3)cc2)C1 ZINC000147468236 HF On-Demand Anodyne EPHX2 28 41 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)NC3CCCCC3)cc2)C1 ZINC000147468236 HF On-Demand Anodyne CACNA1I 61 35 Cc1nc(Nc2ccccc2C(C)C)ccc1C(=O)O ZINC000147468247 CH For-Sale Anodyne MAPK8 15 41 Cc1nc(Nc2ccccc2C(C)C)ccc1C(=O)O ZINC000147468247 CH For-Sale Anodyne AKR1C2 48 38 Fc1ccc(CN2CCCC2)cc1Cl ZINC000147468309 BG On-Demand Anodyne DRD2 0 46 Fc1ccc(CN2CCCC2)cc1Cl ZINC000147468309 BG On-Demand Anodyne OPRK1 25 41 Fc1ccc(CN2CCCC2)cc1Cl ZINC000147468309 BG On-Demand Anodyne HRH3 24 53 Fc1ccc(CN2CCCC2)cc1Cl ZINC000147468309 BG On-Demand Anodyne SIGMAR1 46 50 Fc1ccc(CN2CCCC2)cc1Cl ZINC000147468309 BG On-Demand Anodyne CXCR4 20 42 Fc1ccc(CN2CCCC2)cc1Cl ZINC000147468309 BG On-Demand Anodyne LSS 17 42 Fc1ccc(CN2CCCC2)cc1Cl ZINC000147468309 BG On-Demand Anodyne CACNA1G 20 44 Cc1c(N)cc(C(=O)Nc2ccncc2Br)cc1F ZINC000147468335 DG For-Sale Anodyne HDAC1 28 42 CC[C@H]1CN(CC(=O)Nc2ccccc2F)CC[C@@H]1N ZINC000147468367 CD On-Demand Anodyne DRD4 0 53 CCC[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468374 HH On-Demand Anodyne CHRM5 32 48 CCC[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468374 HH On-Demand Anodyne KCNQ2 39 46 CCC[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468374 HH On-Demand Anodyne MMP13 19 41 CCC[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468374 HH On-Demand Anodyne CCR5 41 39 CCC[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468374 HH On-Demand Anodyne EPHX2 24 45 CCC[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468374 HH On-Demand Anodyne TGM2 64 44 CCC[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468374 HH On-Demand Anodyne MMP1 17 40 CCC[C@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468374 HH On-Demand Anodyne F13A1 65 44 Cc1cc(Cl)cc(-c2nc(-c3cccc(N)c3)no2)c1 ZINC000147468422 CH On-Demand Anodyne GRM5 23 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)s2)c1 ZINC000147468437 FI On-Demand Anodyne PPIA 15 42 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)NC3CCCCC3)cc2)C1 ZINC000147468446 HF On-Demand Anodyne HTR4 43 36 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)NC3CCCCC3)cc2)C1 ZINC000147468446 HF On-Demand Anodyne CNR2 17 41 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)NC3CCCCC3)cc2)C1 ZINC000147468446 HF On-Demand Anodyne EPHX2 28 41 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)NC3CCCCC3)cc2)C1 ZINC000147468446 HF On-Demand Anodyne CACNA1I 61 35 CCCOc1ccc(Oc2cc(C)nc(NC)n2)cc1 ZINC000147468480 CG For-Sale Anodyne ACACA 41 40 CCCOc1ccc(Oc2cc(C)nc(NC)n2)cc1 ZINC000147468480 CG For-Sale Anodyne ACACB 15 40 COc1ccc(CCNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147468483 CF For-Sale Anodyne P2RX1 25 48 COc1ccc(CCNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147468483 CF For-Sale Anodyne PTGDR 38 58 COc1ccc(CCNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147468483 CF For-Sale Anodyne CA9 20 41 COc1ccc(CCNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147468483 CF For-Sale Anodyne AKR1C3 23 41 COc1ccc(CCNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147468483 CF For-Sale Anodyne PROKR1 62 35 COc1ccc(CCNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147468483 CF For-Sale Anodyne AKR1C2 55 41 N[C@@H](COCc1cccc(Br)c1)C(=O)O ZINC000147468499 CD For-Sale Anodyne CACNA2D1 33 56 N[C@@H](COCc1cccc(Br)c1)C(=O)O ZINC000147468499 CD For-Sale Anodyne SLC1A1 33 53 N[C@@H](COCc1cccc(Br)c1)C(=O)O ZINC000147468499 CD For-Sale Anodyne KIF11 24 41 CCC[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468566 HH On-Demand Anodyne CHRM5 32 48 CCC[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468566 HH On-Demand Anodyne KCNQ2 39 46 CCC[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468566 HH On-Demand Anodyne MMP13 19 41 CCC[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468566 HH On-Demand Anodyne CCR5 41 39 CCC[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468566 HH On-Demand Anodyne EPHX2 24 45 CCC[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468566 HH On-Demand Anodyne TGM2 64 44 CCC[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468566 HH On-Demand Anodyne MMP1 17 40 CCC[C@@H](C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147468566 HH On-Demand Anodyne F13A1 65 44 CCCCc1ccc(OC[C@H](NCC)C(C)C)cc1 ZINC000147468626 CI For-Sale Anodyne ADRB1 15 51 CCCCc1ccc(OC[C@H](NCC)C(C)C)cc1 ZINC000147468626 CI For-Sale Anodyne SCN2A 15 41 CCCCc1ccc(OC[C@H](NCC)C(C)C)cc1 ZINC000147468626 CI For-Sale Anodyne S1PR4 18 42 CCCCc1ccc(OC[C@H](NCC)C(C)C)cc1 ZINC000147468626 CI For-Sale Anodyne S1PR2 23 42 N[C@H](COCc1cccc(Br)c1)C(=O)O ZINC000147468675 CD For-Sale Anodyne CACNA2D1 33 56 N[C@H](COCc1cccc(Br)c1)C(=O)O ZINC000147468675 CD For-Sale Anodyne SLC1A1 33 53 N[C@H](COCc1cccc(Br)c1)C(=O)O ZINC000147468675 CD For-Sale Anodyne KIF11 24 41 Cc1nc(Nc2ccc(F)c(F)c2F)ccc1C(=O)O ZINC000147468695 CG For-Sale Anodyne AKR1C2 51 35 COc1cc(NS(=O)(=O)c2ccc(Br)cc2)ccc1Br ZINC000147468698 HI On-Demand Anodyne CA2 15 42 COc1cc(NS(=O)(=O)c2ccc(Br)cc2)ccc1Br ZINC000147468698 HI On-Demand Anodyne CA1 17 40 COc1cc(NS(=O)(=O)c2ccc(Br)cc2)ccc1Br ZINC000147468698 HI On-Demand Anodyne HTR6 30 59 COc1cc(NS(=O)(=O)c2ccc(Br)cc2)ccc1Br ZINC000147468698 HI On-Demand Anodyne CA4 20 41 COc1cc(NS(=O)(=O)c2ccc(Br)cc2)ccc1Br ZINC000147468698 HI On-Demand Anodyne GHSR 23 47 COc1cc(NS(=O)(=O)c2ccc(Br)cc2)ccc1Br ZINC000147468698 HI On-Demand Anodyne ALPL 25 40 COc1cc(NS(=O)(=O)c2ccc(Br)cc2)ccc1Br ZINC000147468698 HI On-Demand Anodyne IDO1 32 50 COc1cc(NS(=O)(=O)c2ccc(Br)cc2)ccc1Br ZINC000147468698 HI On-Demand Anodyne FFAR4 29 40 CCCOc1ccc(Oc2cc(N)cc([N+](=O)[O-])c2)cc1 ZINC000147468708 CH For-Sale Bother ACR 20 40 CCCOc1ccc(Oc2cc(N)cc([N+](=O)[O-])c2)cc1 ZINC000147468708 CH For-Sale Bother ENR 0 40 CC(C)CCCCNC(=O)c1cc2ccccc2cc1N ZINC000147468761 CH For-Sale Anodyne POLR1A 62 37 CCCCc1ccc(OC[C@@H](NCC)C(C)C)cc1 ZINC000147468814 CI For-Sale Anodyne ADRB1 15 51 CCCCc1ccc(OC[C@@H](NCC)C(C)C)cc1 ZINC000147468814 CI For-Sale Anodyne SCN2A 15 41 CCCCc1ccc(OC[C@@H](NCC)C(C)C)cc1 ZINC000147468814 CI For-Sale Anodyne S1PR4 18 42 CCCCc1ccc(OC[C@@H](NCC)C(C)C)cc1 ZINC000147468814 CI For-Sale Anodyne S1PR2 23 42 CC(C)Oc1cccc(C(=O)c2cncs2)c1 ZINC000147468884 BG For-Sale Anodyne HSD17B2 17 50 COc1cc(-c2nc(-c3cccc(N)c3)no2)ccc1F ZINC000147468895 CG On-Demand Anodyne LUCI_PHOPE 41 47 Cc1noc(C)c1CC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147468896 DF In-Stock Anodyne P2RX7 15 51 CCCOc1ccc(Oc2ccnc(N)n2)cc1 ZINC000147468924 BF For-Sale Anodyne DRTS_PLAFK 20 49 O=C(O)CCCCCOCc1cccc(Br)c1 ZINC000147468997 DH For-Sale Anodyne PLA2G4B 47 39 O=C(O)CCCCCOCc1cccc(Br)c1 ZINC000147468997 DH For-Sale Anodyne HCAR2 0 48 O=C(O)CCCCCOCc1cccc(Br)c1 ZINC000147468997 DH For-Sale Anodyne FFAR1 39 54 O=C(O)CCCCCOCc1cccc(Br)c1 ZINC000147468997 DH For-Sale Anodyne FFAR4 22 54 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccccc2OC)CC1 ZINC000147469010 GD On-Demand Anodyne F2 20 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccccc2OC)CC1 ZINC000147469010 GD On-Demand Anodyne GHRHR 43 34 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccccc2OC)CC1 ZINC000147469010 GD On-Demand Anodyne P2RY12 207 41 CCCC[C@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccccc2OC)CC1 ZINC000147469010 GD On-Demand Anodyne TRY2_BOVIN 61 34 CC(=O)Cc1ccc(N)c(O)c1 ZINC000147469024 AD For-Sale Anodyne NCE103 25 41 CCCc1nc(C(F)(F)F)ccc1/C=C/C(=O)N[C@@H](C)c1cc(F)c(NS(C)(=O)=O)c(F)c1 ZINC000147469074 JJ In-Stock Anodyne KCNQ2 51 36 CCCc1nc(C(F)(F)F)ccc1/C=C/C(=O)N[C@@H](C)c1cc(F)c(NS(C)(=O)=O)c(F)c1 ZINC000147469074 JJ In-Stock Anodyne TRPV1 118 46 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1OC ZINC000147469084 CF For-Sale Anodyne SYK 41 42 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1OC ZINC000147469084 CF For-Sale Anodyne AKR1C3 45 45 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1OC ZINC000147469084 CF For-Sale Anodyne ABCG2 21 41 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1OC ZINC000147469084 CF For-Sale Anodyne AKR1C2 91 45 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1OC ZINC000147469084 CF For-Sale Anodyne ENPP1 76 36 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1OC ZINC000147469084 CF For-Sale Anodyne DRTS_TRYCR 47 34 CCOC(=O)Cc1csc(-c2cc(F)cc(F)c2)n1 ZINC000147469107 CG For-Sale Anodyne DCK 48 37 C=CCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147469111 CF On-Demand Mild HCAR1 0 40 COc1cc(NS(=O)(=O)c2ccccc2C)ccc1Br ZINC000147469132 FH On-Demand Anodyne EDNRA 15 44 COc1cc(NS(=O)(=O)c2ccccc2C)ccc1Br ZINC000147469132 FH On-Demand Anodyne GHSR 0 45 COc1cc(NS(=O)(=O)c2ccccc2C)ccc1Br ZINC000147469132 FH On-Demand Anodyne NR1I2 29 43 COc1cc(NS(=O)(=O)c2ccccc2C)ccc1Br ZINC000147469132 FH On-Demand Anodyne ALPL 34 42 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild DRD4 41 33 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild F10 15 42 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild GRIN2B 22 41 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild CCR3 31 45 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild ITGA4 60 33 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild EPHX2 20 42 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild TGM2 58 42 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild MCHR1 16 41 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild CACNA1I 64 42 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild F13A1 51 42 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild AKR1C3 61 45 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild SFRP1 19 46 N#Cc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147469142 GE On-Demand Mild NAMPT 33 41 CNC(=O)Cn1cc(NC(=O)C(=O)c2ccc3c(c2)CCC3)cn1 ZINC000147469146 EC On-Demand Anodyne PANC 44 31 Nc1cccc(CCC(=O)Nc2ccncc2Br)c1 ZINC000147469185 DF For-Sale Anodyne TRPV1 26 48 Nc1cccc(CCC(=O)Nc2ccncc2Br)c1 ZINC000147469185 DF For-Sale Anodyne HCAR2 19 43 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccccc2OC)CC1 ZINC000147469212 GD On-Demand Anodyne F2 20 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccccc2OC)CC1 ZINC000147469212 GD On-Demand Anodyne GHRHR 43 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccccc2OC)CC1 ZINC000147469212 GD On-Demand Anodyne P2RY12 207 41 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(C(=O)c2ccccc2OC)CC1 ZINC000147469212 GD On-Demand Anodyne TRY2_BOVIN 61 34 CC(C)c1ccc(NC(=O)N2CCN([C@@H](C)c3ccccc3)CC2)cc1 ZINC000147469213 FJ For-Sale Anodyne PDGFRB 42 47 CC(C)c1ccc(NC(=O)N2CCN([C@@H](C)c3ccccc3)CC2)cc1 ZINC000147469213 FJ For-Sale Anodyne TRPV1 15 54 CC(C)c1ccc(NC(=O)N2CCN([C@@H](C)c3ccccc3)CC2)cc1 ZINC000147469213 FJ For-Sale Anodyne NPY2R 58 43 CC(C)c1ccc(NC(=O)N2CCN([C@@H](C)c3ccccc3)CC2)cc1 ZINC000147469213 FJ For-Sale Anodyne NPY5R 18 40 CC(C)c1ccc(NC(=O)N2CCN([C@@H](C)c3ccccc3)CC2)cc1 ZINC000147469213 FJ For-Sale Anodyne EPHX2 22 41 CC(C)c1ccc(NC(=O)N2CCN([C@@H](C)c3ccccc3)CC2)cc1 ZINC000147469213 FJ For-Sale Anodyne TRPM8 22 40 O=C(O)C(F)(F)OCc1cccc(Br)c1 ZINC000147469239 CF For-Sale Anodyne HCAR2 18 51 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3ccccc3C#N)cc2)C1 ZINC000147469256 HG On-Demand Mild HTR4 43 34 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3ccccc3C#N)cc2)C1 ZINC000147469256 HG On-Demand Mild CACNA1I 40 30 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3ccccc3C#N)cc2)C1 ZINC000147469256 HG On-Demand Mild PFKFB3 49 35 COc1ccc2c(c1)OC[C@@H](C(=O)NCC1(c3ccc(Cl)cc3)CCOCC1)C2 ZINC000147469279 HH On-Demand Anodyne MTNR1A 23 40 COc1ccc2c(c1)OC[C@@H](C(=O)NCC1(c3ccc(Cl)cc3)CCOCC1)C2 ZINC000147469279 HH On-Demand Anodyne MTNR1B 18 40 Nc1cccc(-c2noc(-c3cccc(Cl)c3F)n2)c1 ZINC000147469301 CH On-Demand Anodyne GRM5 20 41 COc1ccc(CNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147469309 CF For-Sale Anodyne P2RX1 23 44 COc1ccc(CNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147469309 CF For-Sale Anodyne PTGDR 25 47 COc1ccc(CNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147469309 CF For-Sale Anodyne AKR1C3 23 43 COc1ccc(CNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147469309 CF For-Sale Anodyne SCD 18 40 COc1ccc(CNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147469309 CF For-Sale Anodyne PROKR1 64 35 COc1ccc(CNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147469309 CF For-Sale Anodyne AKR1C2 57 43 COc1ccc(CNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147469309 CF For-Sale Anodyne PRUNE 0 40 COc1ccc(CNc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147469309 CF For-Sale Anodyne PETD 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(C3CC3)on2)c1 ZINC000147469312 DG On-Demand Anodyne S1PR3 0 44 CN(Cc1cscn1)C(=O)NCCc1cccnc1 ZINC000147469322 CD On-Demand Anodyne CYP3A4 18 42 COc1cc(NS(=O)(=O)c2cccc(Br)c2)ccc1Br ZINC000147469363 HI On-Demand Anodyne HTR6 23 52 COc1cc(NS(=O)(=O)c2cccc(Br)c2)ccc1Br ZINC000147469363 HI On-Demand Anodyne GHSR 0 49 COc1cc(NS(=O)(=O)c2cccc(Br)c2)ccc1Br ZINC000147469363 HI On-Demand Anodyne ALPL 25 41 CC(C)c1ccc(NC(=O)N2CCN([C@H](C)c3ccccc3)CC2)cc1 ZINC000147469395 FJ For-Sale Anodyne PDGFRB 42 47 CC(C)c1ccc(NC(=O)N2CCN([C@H](C)c3ccccc3)CC2)cc1 ZINC000147469395 FJ For-Sale Anodyne TRPV1 15 54 CC(C)c1ccc(NC(=O)N2CCN([C@H](C)c3ccccc3)CC2)cc1 ZINC000147469395 FJ For-Sale Anodyne NPY2R 58 43 CC(C)c1ccc(NC(=O)N2CCN([C@H](C)c3ccccc3)CC2)cc1 ZINC000147469395 FJ For-Sale Anodyne NPY5R 18 40 CC(C)c1ccc(NC(=O)N2CCN([C@H](C)c3ccccc3)CC2)cc1 ZINC000147469395 FJ For-Sale Anodyne EPHX2 22 41 CC(C)c1ccc(NC(=O)N2CCN([C@H](C)c3ccccc3)CC2)cc1 ZINC000147469395 FJ For-Sale Anodyne TRPM8 22 40 CCCn1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147469401 CD For-Sale Anodyne CASP3 79 36 CCCn1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147469401 CD For-Sale Anodyne CASP8 56 36 CCCn1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147469401 CD For-Sale Anodyne CASP1 45 33 CCCn1ccnc(NC[C@@H](C)CC(=O)O)c1=O ZINC000147469401 CD For-Sale Anodyne CASP7 56 36 CC(C)(C)OC(=O)N1CCCC[C@@H]1C(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147469410 EE On-Demand Anodyne PREP 63 76 CC(C)(C)OC(=O)N1CCCC[C@@H]1C(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147469410 EE On-Demand Anodyne SFRP1 45 44 CC(C)(C)OC(=O)N1CCCC[C@@H]1C(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147469410 EE On-Demand Anodyne WNT3 56 44 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3ccccc3C#N)cc2)C1 ZINC000147469445 HG On-Demand Mild HTR4 43 34 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3ccccc3C#N)cc2)C1 ZINC000147469445 HG On-Demand Mild CACNA1I 40 30 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3ccccc3C#N)cc2)C1 ZINC000147469445 HG On-Demand Mild PFKFB3 49 35 CC[C@@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469446 CE On-Demand Anodyne LTA4H 54 50 CC[C@@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469446 CE On-Demand Anodyne HRH3 56 40 CC[C@@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469446 CE On-Demand Anodyne SLC6A11 0 41 CC[C@@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469446 CE On-Demand Anodyne EBP 35 47 CC[C@@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469446 CE On-Demand Anodyne SLC6A13 0 41 CC[C@@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469446 CE On-Demand Anodyne PSMB2 51 38 CC[C@@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469446 CE On-Demand Anodyne PSMB1 44 39 COc1ccc(OC)c(C(=O)c2cncs2)c1 ZINC000147469513 BE For-Sale Anodyne LUCI_LUCLA 15 40 CCc1nc(CN(C)C(=O)NCCc2cccnc2)cs1 ZINC000147469531 DE On-Demand Anodyne CYP3A4 19 42 COc1cc(Nc2ccc(C(=O)O)c(C)n2)cc(OC)c1 ZINC000147469554 CF For-Sale Anodyne ZAP70 55 35 COc1cc(Nc2ccc(C(=O)O)c(C)n2)cc(OC)c1 ZINC000147469554 CF For-Sale Anodyne ALS 43 31 COc1cc(Nc2ccc(C(=O)O)c(C)n2)cc(OC)c1 ZINC000147469554 CF For-Sale Anodyne AKR1C3 36 56 COc1cc(Nc2ccc(C(=O)O)c(C)n2)cc(OC)c1 ZINC000147469554 CF For-Sale Anodyne AKR1C2 72 50 COc1cc(NS(=O)(=O)c2ccccc2Br)ccc1Br ZINC000147469557 HI On-Demand Anodyne HTR6 18 43 COc1cc(NS(=O)(=O)c2ccccc2Br)ccc1Br ZINC000147469557 HI On-Demand Anodyne UTS2R 0 43 COc1cc(NS(=O)(=O)c2ccccc2Br)ccc1Br ZINC000147469557 HI On-Demand Anodyne GHSR 0 42 COc1cc(NS(=O)(=O)c2ccccc2Br)ccc1Br ZINC000147469557 HI On-Demand Anodyne NR1I2 26 45 COc1cc(NS(=O)(=O)c2ccccc2Br)ccc1Br ZINC000147469557 HI On-Demand Anodyne ALPL 30 44 Cc1noc(C)c1CNS(=O)(=O)c1cccc2cnccc12 ZINC000147469582 DE On-Demand Anodyne EDNRA 19 46 Cc1noc(C)c1CNS(=O)(=O)c1cccc2cnccc12 ZINC000147469582 DE On-Demand Anodyne P2RX7 22 46 Cc1noc(C)c1CNS(=O)(=O)c1cccc2cnccc12 ZINC000147469582 DE On-Demand Anodyne Q95J97_RABIT 0 58 CCCn1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147469596 CD For-Sale Anodyne CASP3 79 36 CCCn1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147469596 CD For-Sale Anodyne CASP8 56 36 CCCn1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147469596 CD For-Sale Anodyne CASP1 45 33 CCCn1ccnc(NC[C@H](C)CC(=O)O)c1=O ZINC000147469596 CD For-Sale Anodyne CASP7 56 36 C[C@H](NC(=O)c1ccco1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147469597 HD On-Demand Anodyne HTR4 41 38 C[C@H](NC(=O)c1ccco1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147469597 HD On-Demand Anodyne TGM2 65 46 C[C@H](NC(=O)c1ccco1)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147469597 HD On-Demand Anodyne F13A1 62 46 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147469621 EE On-Demand Anodyne PREP 63 76 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147469621 EE On-Demand Anodyne SFRP1 45 44 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)N1CCC[C@H](C(=O)O)C1 ZINC000147469621 EE On-Demand Anodyne WNT3 56 44 CC[C@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469623 CE On-Demand Anodyne LTA4H 54 50 CC[C@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469623 CE On-Demand Anodyne HRH3 56 40 CC[C@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469623 CE On-Demand Anodyne SLC6A11 0 41 CC[C@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469623 CE On-Demand Anodyne EBP 35 47 CC[C@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469623 CE On-Demand Anodyne SLC6A13 0 41 CC[C@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469623 CE On-Demand Anodyne PSMB2 51 38 CC[C@H]1CN(CCOc2ccc(OC)cc2)CC[C@@H]1N ZINC000147469623 CE On-Demand Anodyne PSMB1 44 39 CC(Cl)(Cl)C(=O)Oc1ccccc1 ZINC000147469728 BF On-Demand Anodyne ELANE 25 55 CC(Cl)(Cl)C(=O)Oc1ccccc1 ZINC000147469728 BF On-Demand Anodyne PRTN3 57 37 Cc1nc(Nc2ccc(C(F)(F)F)cc2)ccc1C(=O)O ZINC000147469779 CH For-Sale Anodyne DHODH 15 41 Cc1nc(Nc2ccc(C(F)(F)F)cc2)ccc1C(=O)O ZINC000147469779 CH For-Sale Anodyne TRPV1 21 45 Cc1nc(Nc2ccc(C(F)(F)F)cc2)ccc1C(=O)O ZINC000147469779 CH For-Sale Anodyne SORT1 32 53 Cc1nc(Nc2ccc(C(F)(F)F)cc2)ccc1C(=O)O ZINC000147469779 CH For-Sale Anodyne EPHX2 19 43 Cc1nc(Nc2ccc(C(F)(F)F)cc2)ccc1C(=O)O ZINC000147469779 CH For-Sale Anodyne AKR1C3 38 50 Cc1nc(Nc2ccc(C(F)(F)F)cc2)ccc1C(=O)O ZINC000147469779 CH For-Sale Anodyne AKR1C2 73 39 COc1ccc(C)cc1NC(=O)C1(N)CCC1 ZINC000147469789 BD For-Sale Anodyne KCNMA1 18 44 NC(=O)[C@@H](N)COCc1cccc(Br)c1 ZINC000147469805 CC For-Sale Anodyne CACNA2D1 23 46 CC[C@@H](CCNC(=O)OC(C)(C)C)C(=O)O ZINC000147469808 BE In-Stock Anodyne PAPA1_CARPA 44 42 CC[C@@H](CCNC(=O)OC(C)(C)C)C(=O)O ZINC000147469808 BE In-Stock Anodyne CTSK 27 44 CC[C@@H](CCNC(=O)OC(C)(C)C)C(=O)O ZINC000147469808 BE In-Stock Anodyne SLC22A20 0 48 CC(C)(C)OC(=O)N1CCCC[C@@H]1C(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147469817 EE On-Demand Anodyne PREP 63 76 CC(C)(C)OC(=O)N1CCCC[C@@H]1C(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147469817 EE On-Demand Anodyne SFRP1 45 44 CC(C)(C)OC(=O)N1CCCC[C@@H]1C(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147469817 EE On-Demand Anodyne WNT3 56 44 CC(C)Oc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147469896 HG On-Demand Anodyne HTR4 56 39 CC(C)Oc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147469896 HG On-Demand Anodyne GRIN2B 23 44 CC(C)Oc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147469896 HG On-Demand Anodyne MMP13 51 45 CC(C)Oc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147469896 HG On-Demand Anodyne EPHX2 23 42 CC(C)Oc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147469896 HG On-Demand Anodyne TGM2 65 47 CC(C)Oc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147469896 HG On-Demand Anodyne ST14 15 40 CC(C)Oc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147469896 HG On-Demand Anodyne MMP1 35 44 CC(C)Oc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147469896 HG On-Demand Anodyne CACNA1I 65 39 CC(C)Oc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147469896 HG On-Demand Anodyne F13A1 50 43 COc1ccc(C(=O)c2cncs2)c(OC)c1 ZINC000147469940 BE For-Sale Anodyne LUCI_LUCLA 16 45 CC(C)CCCCNCC(=O)OC(C)(C)C ZINC000147469941 BF For-Sale Anodyne CTSK 0 41 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne DRD4 56 45 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne PPIA 17 49 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne KCNJ11 17 44 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne UL80 19 40 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne ECR 25 47 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne COLA 69 38 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne CPT1A 77 40 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne CPT2 47 37 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne PRNP 21 46 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne PPARD 0 42 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne MTNR1A 25 41 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne MTNR1B 30 42 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne NR1H4 17 49 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne GRM5 19 50 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne CPT1B 44 37 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne SCN10A 25 42 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne CSF1R 21 52 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne FABH 0 44 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne GCK 16 40 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne TAAR1 60 56 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne AKR1C3 67 48 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne AKR1C2 58 45 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne SENP1 0 55 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne PSBA 0 41 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne KCNK3 123 64 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne KCNK9 72 47 COc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147469948 DG On-Demand Anodyne BRPF1 0 52 N[C@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147469959 CD For-Sale Anodyne CACNA1I 62 40 COc1cc(NS(=O)(=O)c2ccc(C(=O)O)s2)ccc1Br ZINC000147469964 GG On-Demand Anodyne GHSR 18 42 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147469981 EE On-Demand Anodyne PREP 63 76 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147469981 EE On-Demand Anodyne SFRP1 45 44 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)N1CCC[C@@H](C(=O)O)C1 ZINC000147469981 EE On-Demand Anodyne WNT3 56 44 NC(=O)[C@H](N)COCc1cccc(Br)c1 ZINC000147469998 CC For-Sale Anodyne CACNA2D1 23 46 COc1ccc(OC)c(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147470036 CF For-Sale Anodyne MAPK8 16 40 COc1ccc(OC)c(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147470036 CF For-Sale Anodyne LUCI_LUCLA 17 43 COc1ccc(OC)c(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147470036 CF For-Sale Anodyne AKR1C3 41 56 COc1ccc(OC)c(Nc2ccc(C(=O)O)c(C)n2)c1 ZINC000147470036 CF For-Sale Anodyne AKR1C2 87 56 CC[C@@H](CCC(=O)O)NC(=O)OC(C)(C)C ZINC000147470040 BE For-Sale Anodyne PAPA1_CARPA 47 44 CC[C@@H](CCC(=O)O)NC(=O)OC(C)(C)C ZINC000147470040 BE For-Sale Anodyne CTSK 33 50 CC[C@@H](CCC(=O)O)NC(=O)OC(C)(C)C ZINC000147470040 BE For-Sale Anodyne ECE1 25 40 CC[C@@H](CCC(=O)O)NC(=O)OC(C)(C)C ZINC000147470040 BE For-Sale Anodyne PGA5 41 37 CC[C@@H](CCC(=O)O)NC(=O)OC(C)(C)C ZINC000147470040 BE For-Sale Anodyne POLG_HCV1 24 47 Cc1cc(S(=O)(=O)Nc2ccncc2Br)cc(N)c1C ZINC000147470054 FF For-Sale Anodyne PTGS1 0 41 CCCOc1ccc(Oc2nc(Cl)nc(NCC)n2)cc1 ZINC000147470112 DH For-Sale Anodyne PETD 0 47 CCCOc1ccc(Oc2nc(Cl)nc(NCC)n2)cc1 ZINC000147470112 DH For-Sale Anodyne Q31945_CHEAL 0 40 CCCOc1ccc(Oc2nc(Cl)nc(NCC)n2)cc1 ZINC000147470112 DH For-Sale Anodyne PPX1 0 47 C[C@@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470122 HG On-Demand Anodyne F2 19 40 C[C@@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470122 HG On-Demand Anodyne GRIN2B 24 41 C[C@@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470122 HG On-Demand Anodyne MMP13 17 41 C[C@@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470122 HG On-Demand Anodyne EPHX2 22 41 C[C@@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470122 HG On-Demand Anodyne TGM2 70 45 C[C@@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470122 HG On-Demand Anodyne CACNA1I 46 35 C[C@@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470122 HG On-Demand Anodyne F13A1 76 45 N[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147470131 CD For-Sale Anodyne CACNA1I 62 40 CCNC(=O)C1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147470148 FG For-Sale Anodyne EPHX2 31 45 CCNC(=O)C1CCN(C(=O)c2ccc(Br)c(Cl)c2)CC1 ZINC000147470148 FG For-Sale Anodyne L3MBTL3 90 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne PPIA 16 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne ECR 26 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne ATF1 47 38 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne PRNP 16 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne NR1H4 17 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne NFKB1 43 38 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne ACPS 0 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne AKR1C3 34 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne NR2E3 43 34 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne CYA 0 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne AKR1C2 25 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne SMO 26 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne Q25615_ONCVO 74 39 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne KCNK3 90 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2I)c1 ZINC000147470158 HH On-Demand Anodyne KCNK9 68 35 CC[C@H](CCC(=O)O)NC(=O)OC(C)(C)C ZINC000147470193 BE For-Sale Anodyne PAPA1_CARPA 35 44 CC[C@H](CCC(=O)O)NC(=O)OC(C)(C)C ZINC000147470193 BE For-Sale Anodyne CTSK 33 50 CC[C@H](CCC(=O)O)NC(=O)OC(C)(C)C ZINC000147470193 BE For-Sale Anodyne ECE1 23 40 CC[C@H](CCC(=O)O)NC(=O)OC(C)(C)C ZINC000147470193 BE For-Sale Anodyne POLG_HCV1 24 47 COc1cc(NS(=O)(=O)c2ccccc2)ccc1Br ZINC000147470206 EG On-Demand Anodyne HTR6 26 42 COc1cc(NS(=O)(=O)c2ccccc2)ccc1Br ZINC000147470206 EG On-Demand Anodyne GHSR 22 45 COc1cc(NS(=O)(=O)c2ccccc2)ccc1Br ZINC000147470206 EG On-Demand Anodyne ALPL 27 43 COc1cc(NS(=O)(=O)c2ccccc2)ccc1Br ZINC000147470206 EG On-Demand Anodyne IDO1 0 42 NC1(C(=O)NC2CCN(Cc3ccccc3)CC2)CCC1 ZINC000147470270 CD On-Demand Anodyne DRD2 24 52 NC1(C(=O)NC2CCN(Cc3ccccc3)CC2)CCC1 ZINC000147470270 CD On-Demand Anodyne ACHE 0 50 NC1(C(=O)NC2CCN(Cc3ccccc3)CC2)CCC1 ZINC000147470270 CD On-Demand Anodyne DRD3 34 58 NC1(C(=O)NC2CCN(Cc3ccccc3)CC2)CCC1 ZINC000147470270 CD On-Demand Anodyne BCHE 27 44 Cc1nc(Nc2ccc(C(N)=O)cc2)ccc1C(=O)O ZINC000147470280 CD For-Sale Anodyne PDE4B 0 40 Cc1nc(Nc2ccc(C(N)=O)cc2)ccc1C(=O)O ZINC000147470280 CD For-Sale Anodyne AKR1C3 49 40 Cc1nc(Nc2ccc(C(N)=O)cc2)ccc1C(=O)O ZINC000147470280 CD For-Sale Anodyne AKR1C2 69 39 Cc1nc(Nc2ccc(C(N)=O)cc2)ccc1C(=O)O ZINC000147470280 CD For-Sale Anodyne RPS27 27 41 O=C(c1cncs1)c1cccc2cnccc12 ZINC000147470286 BF For-Sale Anodyne TRPV1 0 40 CC(C)(COCc1cccc(Br)c1)C(=O)O ZINC000147470307 CG For-Sale Anodyne HCAR2 17 50 CC(C)(COCc1cccc(Br)c1)C(=O)O ZINC000147470307 CG For-Sale Anodyne FFAR1 17 47 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470328 HG On-Demand Anodyne F2 19 40 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470328 HG On-Demand Anodyne GRIN2B 24 41 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470328 HG On-Demand Anodyne MMP13 17 41 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470328 HG On-Demand Anodyne EPHX2 22 41 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470328 HG On-Demand Anodyne TGM2 70 45 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470328 HG On-Demand Anodyne CACNA1I 46 35 C[C@H](CC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccccc1 ZINC000147470328 HG On-Demand Anodyne F13A1 76 45 CCCNc1ccc(Cl)cc1C(=O)NCCNC(N)=O ZINC000147470348 CD For-Sale Anodyne F10 22 40 CCCNc1ccc(Cl)cc1C(=O)NCCNC(N)=O ZINC000147470348 CD For-Sale Anodyne PSBA 0 41 Cn1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147470360 CE On-Demand Anodyne ATF1 46 37 Cn1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147470360 CE On-Demand Anodyne NFKB1 42 37 Cn1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147470360 CE On-Demand Anodyne CACNA1I 50 35 CCNC(=O)C1CCN(C(=O)c2cc(C)ccc2Br)CC1 ZINC000147470381 FF For-Sale Anodyne EPHX2 34 42 CCNC(=O)C1CCN(C(=O)c2cc(C)ccc2Br)CC1 ZINC000147470381 FF For-Sale Anodyne L3MBTL3 61 39 COc1cc(NS(=O)(=O)c2ccccc2C#N)ccc1Br ZINC000147470401 FG On-Demand Mild ALPL 23 42 Cc1nc(Nc2ccc(C(C)C)cc2)ccc1C(=O)O ZINC000147470507 CH For-Sale Anodyne AKR1C2 65 38 CC(C)OC(=O)COCc1cccc(Br)c1 ZINC000147470531 CF For-Sale Anodyne HCAR2 15 45 CO[C@@H](CNC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147470533 DF On-Demand Anodyne BMP1 41 33 CO[C@@H](CNC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147470533 DF On-Demand Anodyne CYP3A4 16 42 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(F)c1 ZINC000147470593 DH On-Demand Anodyne RARA 32 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(F)c1 ZINC000147470593 DH On-Demand Anodyne JUN 23 43 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(F)c1 ZINC000147470593 DH On-Demand Anodyne ATF1 60 42 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(F)c1 ZINC000147470593 DH On-Demand Anodyne CPT1A 37 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(F)c1 ZINC000147470593 DH On-Demand Anodyne NR1H4 16 44 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(F)c1 ZINC000147470593 DH On-Demand Anodyne NFKB1 56 42 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(F)c1 ZINC000147470593 DH On-Demand Anodyne KCNMA1 17 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(F)c1 ZINC000147470593 DH On-Demand Anodyne KCNK3 78 41 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(F)c1 ZINC000147470593 DH On-Demand Anodyne KCNK9 53 41 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(F)c1 ZINC000147470593 DH On-Demand Anodyne TMPRSS4 0 48 COc1cc(NS(=O)(=O)c2cccnc2Cl)ccc1Br ZINC000147470598 GG For-Sale Anodyne CCR4 15 40 COc1cc(NS(=O)(=O)c2cccnc2Cl)ccc1Br ZINC000147470598 GG For-Sale Anodyne GRM4 20 44 COc1cc(NS(=O)(=O)c2cccnc2Cl)ccc1Br ZINC000147470598 GG For-Sale Anodyne ALPL 29 45 Cc1ccc(S(=O)(=O)Nc2ccncc2Br)c(N)c1 ZINC000147470647 EF For-Sale Anodyne NFKBIA 0 48 COc1ccc(CC2CCC2)cc1 ZINC000147470654 AG For-Sale Anodyne SLC18A2 37 66 COc1ccc(CC2CCC2)cc1 ZINC000147470654 AG For-Sale Anodyne SIGMAR1 22 48 COc1ccc(CC2CCC2)cc1 ZINC000147470654 AG For-Sale Anodyne CCR3 18 43 Cc1nc(NCCc2ccccc2F)ccc1C(=O)O ZINC000147470709 CF For-Sale Anodyne PTGDR 19 42 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](C)N1CCc2ccccc21 ZINC000147470714 ED On-Demand Anodyne ACE 17 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](C)N1CCc2ccccc21 ZINC000147470714 ED On-Demand Anodyne PCSK5 53 35 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](C)N1CCc2ccccc21 ZINC000147470714 ED On-Demand Anodyne FURIN 54 31 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](C)N1CCc2ccccc21 ZINC000147470714 ED On-Demand Anodyne POLG_WNV 63 30 CCCC[C@H](NC(N)=O)C(=O)NC[C@@H](C)N1CCc2ccccc21 ZINC000147470714 ED On-Demand Anodyne NPFFR1 48 33 CO[C@H](CNC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147470731 DF On-Demand Anodyne BMP1 41 33 CO[C@H](CNC(=O)N(C)Cc1cscn1)c1ccccc1 ZINC000147470731 DF On-Demand Anodyne CYP3A4 16 42 NC[C@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147470734 CD For-Sale Anodyne CCKBR 44 35 NC[C@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147470734 CD For-Sale Anodyne EPHX2 17 45 NC[C@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147470734 CD For-Sale Anodyne CACNA1I 69 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ncsc2c1 ZINC000147470765 HG On-Demand Anodyne GRIN2B 24 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ncsc2c1 ZINC000147470765 HG On-Demand Anodyne EPHX2 15 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ncsc2c1 ZINC000147470765 HG On-Demand Anodyne TGM2 53 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ncsc2c1 ZINC000147470765 HG On-Demand Anodyne CACNA1I 58 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ncsc2c1 ZINC000147470765 HG On-Demand Anodyne F13A1 27 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ncsc2c1 ZINC000147470765 HG On-Demand Anodyne AKR1C3 50 36 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ncsc2c1 ZINC000147470765 HG On-Demand Anodyne NAMPT 43 40 O=C(O)[C@@H](F)OCc1cccc(Br)c1 ZINC000147470791 CE For-Sale Anodyne CACNA2D1 0 45 O=C(O)[C@@H](F)OCc1cccc(Br)c1 ZINC000147470791 CE For-Sale Anodyne SLC1A6 0 40 O=C(O)[C@@H](F)OCc1cccc(Br)c1 ZINC000147470791 CE For-Sale Anodyne SLC1A7 0 40 O=C(O)[C@@H](F)OCc1cccc(Br)c1 ZINC000147470791 CE For-Sale Anodyne FFAR1 15 48 O=C(CN1CCCC1=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147470809 CD On-Demand Anodyne CACNA1H 19 44 Cc1cccc(N)c1S(=O)(=O)Nc1ccncc1Br ZINC000147470842 EF For-Sale Anodyne PTGS1 0 40 Cc1nc(NCCCN2CCCC[C@@H]2C)ccc1C(=O)O ZINC000147470902 CF For-Sale Anodyne HRH3 61 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](C)N1CCc2ccccc21 ZINC000147470912 ED On-Demand Anodyne PCSK5 53 35 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](C)N1CCc2ccccc21 ZINC000147470912 ED On-Demand Anodyne FURIN 54 31 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](C)N1CCc2ccccc21 ZINC000147470912 ED On-Demand Anodyne POLG_WNV 63 30 CCCC[C@@H](NC(N)=O)C(=O)NC[C@@H](C)N1CCc2ccccc21 ZINC000147470912 ED On-Demand Anodyne NPFFR1 48 33 CCCCCCCC/C=C\CCCCCCCCNC[C@@H](C)N ZINC000147470926 DK For-Sale Mild Q8WS26_TRYCR 34 42 NC[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147470930 CD For-Sale Anodyne CCKBR 44 35 NC[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147470930 CD For-Sale Anodyne EPHX2 17 45 NC[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147470930 CD For-Sale Anodyne CACNA1I 69 43 O=C(O)[C@H](F)OCc1cccc(Br)c1 ZINC000147470984 CE For-Sale Anodyne CACNA2D1 0 45 O=C(O)[C@H](F)OCc1cccc(Br)c1 ZINC000147470984 CE For-Sale Anodyne SLC1A6 0 40 O=C(O)[C@H](F)OCc1cccc(Br)c1 ZINC000147470984 CE For-Sale Anodyne SLC1A7 0 40 O=C(O)[C@H](F)OCc1cccc(Br)c1 ZINC000147470984 CE For-Sale Anodyne FFAR1 15 48 CC(=O)c1c(C)[nH]c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1C ZINC000147470999 HF On-Demand Anodyne HTR4 67 40 CC(=O)c1c(C)[nH]c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1C ZINC000147470999 HF On-Demand Anodyne EPHX2 17 40 CC(=O)c1c(C)[nH]c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1C ZINC000147470999 HF On-Demand Anodyne TGM2 64 43 CC(=O)c1c(C)[nH]c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1C ZINC000147470999 HF On-Demand Anodyne CACNA1I 61 35 CC(=O)c1c(C)[nH]c(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1C ZINC000147470999 HF On-Demand Anodyne F13A1 63 43 COCc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147471010 FJ On-Demand Anodyne PPIA 21 42 COCc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147471010 FJ On-Demand Anodyne UL80 15 40 COCc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147471010 FJ On-Demand Anodyne CPT1A 54 32 COCc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147471010 FJ On-Demand Anodyne ROCK2 17 42 COCc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147471010 FJ On-Demand Anodyne CSF1R 20 40 COCc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147471010 FJ On-Demand Anodyne TAAR1 56 53 COCc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147471010 FJ On-Demand Anodyne ADCYAP1R1 61 34 COCc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147471010 FJ On-Demand Anodyne KCNK3 124 43 COCc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147471010 FJ On-Demand Anodyne KCNK9 84 42 Cc1nn(C)c(C)c1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471025 DF On-Demand Anodyne HPD 44 35 COc1cc(NS(=O)(=O)c2cn[nH]c2C)ccc1Br ZINC000147471033 EE On-Demand Anodyne SGK1 69 39 Cc1csc([C@@H](C#N)C(=O)c2cccc(OCc3cccc(Cl)c3)c2)n1 ZINC000147471057 GK On-Demand Mild MAOB 41 46 Cc1nc(NCCCN2CCCC[C@H]2C)ccc1C(=O)O ZINC000147471099 CF For-Sale Anodyne HRH3 61 40 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](C)N1CCc2ccccc21 ZINC000147471107 ED On-Demand Anodyne PCSK5 53 35 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](C)N1CCc2ccccc21 ZINC000147471107 ED On-Demand Anodyne FURIN 54 31 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](C)N1CCc2ccccc21 ZINC000147471107 ED On-Demand Anodyne POLG_WNV 63 30 CCCC[C@H](NC(N)=O)C(=O)NC[C@H](C)N1CCc2ccccc21 ZINC000147471107 ED On-Demand Anodyne NPFFR1 48 33 CCCCCCCC/C=C\CCCCCCCCNC[C@H](C)N ZINC000147471117 DK For-Sale Mild Q8WS26_TRYCR 34 42 C[C@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471230 FC On-Demand Anodyne CHRM5 21 41 C[C@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471230 FC On-Demand Anodyne MMP13 15 40 C[C@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471230 FC On-Demand Anodyne CAPN1 30 40 C[C@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471230 FC On-Demand Anodyne TGM2 65 46 C[C@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471230 FC On-Demand Anodyne ST14 50 33 C[C@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471230 FC On-Demand Anodyne XIAP 49 34 C[C@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471230 FC On-Demand Anodyne F13A1 76 46 C[C@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471230 FC On-Demand Anodyne TMPRSS6 46 31 CCOC(=O)COCc1cccc(Br)c1 ZINC000147471232 CF For-Sale Anodyne HCAR2 17 49 CCOC(=O)COCc1cccc(Br)c1 ZINC000147471232 CF For-Sale Anodyne FFAR1 21 43 O=C(CC(F)(F)F)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471267 CF On-Demand Anodyne HCAR1 0 43 Cc1csc([C@H](C#N)C(=O)c2cccc(OCc3cccc(Cl)c3)c2)n1 ZINC000147471271 GK On-Demand Mild MAOB 41 46 CCCOc1ccc(Oc2cccc(NC)n2)cc1 ZINC000147471272 CH For-Sale Anodyne ACACA 36 40 CCCOc1ccc(Oc2cccc(NC)n2)cc1 ZINC000147471272 CH For-Sale Anodyne ACACB 18 40 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](C)N1CCc2ccccc21 ZINC000147471330 ED On-Demand Anodyne PCSK5 53 35 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](C)N1CCc2ccccc21 ZINC000147471330 ED On-Demand Anodyne FURIN 54 31 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](C)N1CCc2ccccc21 ZINC000147471330 ED On-Demand Anodyne POLG_WNV 63 30 CCCC[C@@H](NC(N)=O)C(=O)NC[C@H](C)N1CCc2ccccc21 ZINC000147471330 ED On-Demand Anodyne NPFFR1 48 33 Cc1nc(Nc2ccc3c(c2)CCC3)ccc1C(=O)O ZINC000147471332 CG For-Sale Anodyne AKR1C2 48 35 O=C(c1cccc2ccccc12)N1CCC[C@@H]1CCCBr ZINC000147471367 EJ For-Sale Reactive HCRTR1 39 62 O=C(c1cccc2ccccc12)N1CCC[C@@H]1CCCBr ZINC000147471367 EJ For-Sale Reactive PREP 58 45 O=C(c1cccc2ccccc12)N1CCC[C@@H]1CCCBr ZINC000147471367 EJ For-Sale Reactive HCRTR2 21 45 O=C(c1cccc2ccccc12)N1CCC[C@@H]1CCCBr ZINC000147471367 EJ For-Sale Reactive FAP 0 47 O=C(c1cccc2ccccc12)N1CCC[C@@H]1CCCBr ZINC000147471367 EJ For-Sale Reactive NR1D1 42 42 CC(C)N(C)CCCNC(=O)c1ccc(OCc2ccncc2)cc1 ZINC000147471389 EG On-Demand Anodyne SLC6A5 38 41 CCCCCCCOc1ccc(CNCCOC)nc1 ZINC000147471429 CG For-Sale Mild LPAR2 61 46 CCCCCCCOc1ccc(CNCCOC)nc1 ZINC000147471429 CG For-Sale Mild S1PR3 27 46 CCCCCCCOc1ccc(CNCCOC)nc1 ZINC000147471429 CG For-Sale Mild PLA2G4B 72 35 CCCCCCCOc1ccc(CNCCOC)nc1 ZINC000147471429 CG For-Sale Mild S1PR2 66 46 C[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471436 FC On-Demand Anodyne CHRM5 21 41 C[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471436 FC On-Demand Anodyne MMP13 15 40 C[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471436 FC On-Demand Anodyne CAPN1 30 40 C[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471436 FC On-Demand Anodyne TGM2 65 46 C[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471436 FC On-Demand Anodyne ST14 50 33 C[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471436 FC On-Demand Anodyne XIAP 49 34 C[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471436 FC On-Demand Anodyne F13A1 76 46 C[C@@H](NC(N)=O)C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147471436 FC On-Demand Anodyne TMPRSS6 46 31 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne CA2 68 57 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne CA1 59 51 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne CA7 44 34 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne CA5B 59 34 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne CA4 67 56 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne CA5A 63 34 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne CA12 44 57 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne CA9 46 57 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne TTK 23 43 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne CYNT 28 50 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne MTCA1 45 40 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne P96878_MYCTU 58 40 NC1(C(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471443 CC On-Demand Anodyne Q5TU56_ANOGA 0 43 COc1cc(NS(=O)(=O)c2c[nH]c(C(=O)O)c2)ccc1Br ZINC000147471476 GE On-Demand Anodyne HTR6 22 41 O=C(O)c1ccccc1OCCOCc1cccc(Br)c1 ZINC000147471489 FH For-Sale Anodyne PTGER1 27 42 O=C(O)c1ccccc1OCCOCc1cccc(Br)c1 ZINC000147471489 FH For-Sale Anodyne HCAR2 0 44 O=C(O)c1ccccc1OCCOCc1cccc(Br)c1 ZINC000147471489 FH For-Sale Anodyne POBA 0 44 Nc1cc(S(=O)(=O)Nc2ccncc2Br)ccc1Br ZINC000147471498 HF For-Sale Anodyne CA4 15 44 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccccc2OC[C@@H]2CCCCO2)C1 ZINC000147471499 HE On-Demand Anodyne HTR4 63 37 O=C(c1cccc2ccccc12)N1CCC[C@H]1CCCBr ZINC000147471523 EJ For-Sale Reactive HCRTR1 39 62 O=C(c1cccc2ccccc12)N1CCC[C@H]1CCCBr ZINC000147471523 EJ For-Sale Reactive PREP 58 45 O=C(c1cccc2ccccc12)N1CCC[C@H]1CCCBr ZINC000147471523 EJ For-Sale Reactive HCRTR2 21 45 O=C(c1cccc2ccccc12)N1CCC[C@H]1CCCBr ZINC000147471523 EJ For-Sale Reactive FAP 0 47 O=C(c1cccc2ccccc12)N1CCC[C@H]1CCCBr ZINC000147471523 EJ For-Sale Reactive NR1D1 42 42 COc1ccc(Cl)cc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147471578 CG For-Sale Anodyne COLA 50 35 COc1ccc(Cl)cc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147471578 CG For-Sale Anodyne CPT1A 52 35 COc1ccc(Cl)cc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147471578 CG For-Sale Anodyne CPT2 43 35 COc1ccc(Cl)cc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147471578 CG For-Sale Anodyne PYGL 15 41 COc1ccc(Cl)cc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147471578 CG For-Sale Anodyne KCNMA1 28 42 COc1ccc(Cl)cc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147471578 CG For-Sale Anodyne RBP4 29 42 COc1ccc(Cl)cc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147471578 CG For-Sale Anodyne AKR1C3 34 44 COc1ccc(Cl)cc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147471578 CG For-Sale Anodyne AKR1C2 74 44 COc1ccc2c(c1)OC[C@H](C(=O)Nc1c3c(nn1C)CCC3)C2 ZINC000147471591 EE On-Demand Anodyne ROCK2 29 44 NCC1(CC(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471645 CC For-Sale Anodyne CA2 69 65 NCC1(CC(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471645 CC For-Sale Anodyne CA1 61 55 NCC1(CC(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471645 CC For-Sale Anodyne CA7 40 39 NCC1(CC(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471645 CC For-Sale Anodyne CA5B 64 39 NCC1(CC(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471645 CC For-Sale Anodyne CA4 80 65 NCC1(CC(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471645 CC For-Sale Anodyne CA5A 69 39 NCC1(CC(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471645 CC For-Sale Anodyne CA12 37 55 NCC1(CC(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471645 CC For-Sale Anodyne CA9 39 46 NCC1(CC(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471645 CC For-Sale Anodyne TTK 31 41 NCC1(CC(=O)Nc2cccc(S(N)(=O)=O)c2)CCC1 ZINC000147471645 CC For-Sale Anodyne P96878_MYCTU 48 38 Cc1ccc2[nH]c(C(=O)NCCCN(C)C(C)C)cc2c1 ZINC000147471709 CF On-Demand Anodyne CCKAR 19 42 Cc1ccc2[nH]c(C(=O)NCCCN(C)C(C)C)cc2c1 ZINC000147471709 CF On-Demand Anodyne AKR1C3 25 49 CCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471716 BF On-Demand Anodyne CACNA1I 41 32 CCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471716 BF On-Demand Anodyne HCAR1 0 43 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccccc2OC[C@@H]2CCCCO2)C1 ZINC000147471718 HE On-Demand Anodyne HTR4 63 37 Nc1cccc(Cl)c1S(=O)(=O)Nc1ccncc1Br ZINC000147471726 FF For-Sale Anodyne PTGS1 0 40 CCc1nc(CN(C)C(=O)NCCCN2CCN(c3ncccn3)CC2)cs1 ZINC000147471771 HD On-Demand Anodyne HTR1A 37 49 CCc1nc(CN(C)C(=O)NCCCN2CCN(c3ncccn3)CC2)cs1 ZINC000147471771 HD On-Demand Anodyne DRD2 32 41 CCc1nc(CN(C)C(=O)NCCCN2CCN(c3ncccn3)CC2)cs1 ZINC000147471771 HD On-Demand Anodyne HTR2A 32 42 CCc1nc(CN(C)C(=O)NCCCN2CCN(c3ncccn3)CC2)cs1 ZINC000147471771 HD On-Demand Anodyne HTR2C 26 42 CCCCc1ccc(OCCNC2CC2)cc1 ZINC000147471781 BG For-Sale Anodyne KCNQ1 0 40 CCCCc1ccc(OCCNC2CC2)cc1 ZINC000147471781 BG For-Sale Anodyne HRH3 15 49 CCCCc1ccc(OCCNC2CC2)cc1 ZINC000147471781 BG For-Sale Anodyne SCN2A 20 41 CCCCc1ccc(OCCNC2CC2)cc1 ZINC000147471781 BG For-Sale Anodyne S1PR4 21 41 CCCCc1ccc(OCCNC2CC2)cc1 ZINC000147471781 BG For-Sale Anodyne PLA2G4B 58 35 CCCCc1ccc(OCCNC2CC2)cc1 ZINC000147471781 BG For-Sale Anodyne S1PR5 19 41 CCCCc1ccc(OCCNC2CC2)cc1 ZINC000147471781 BG For-Sale Anodyne PPO2 19 40 C/C(=C/C(=O)O)COCc1cccc(Br)c1 ZINC000147471783 CF For-Sale Anodyne RAM2 0 43 O=C(c1ccc2ncccc2c1)N1CCC[C@@H]1CCCBr ZINC000147471796 EI For-Sale Reactive CCR3 0 41 O=C(c1ccc2ncccc2c1)N1CCC[C@@H]1CCCBr ZINC000147471796 EI For-Sale Reactive HCRTR2 0 43 CS(=O)(=O)c1ccc(OCc2cnc(Cl)cn2)cc1 ZINC000147471841 CE On-Demand Anodyne PTGS2 36 49 Cc1cccc(C(C)C)c1NC(=O)C1(N)CCC1 ZINC000147471842 BF For-Sale Anodyne SOAT1 47 43 Cc1cccc(C(C)C)c1NC(=O)C1(N)CCC1 ZINC000147471842 BF For-Sale Anodyne ACAT 0 53 Cc1cccc(OCCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147471878 HF On-Demand Anodyne F2 17 40 Cc1cccc(OCCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147471878 HF On-Demand Anodyne AVPR1B 34 40 Cc1cccc(OCCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147471878 HF On-Demand Anodyne EPHX2 41 44 Cc1cccc(OCCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147471878 HF On-Demand Anodyne TGM2 67 41 Cc1cccc(OCCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147471878 HF On-Demand Anodyne F13A1 68 41 COc1cc(NS(=O)(=O)c2ccc(F)cc2)ccc1Br ZINC000147471907 FG On-Demand Anodyne CA1 16 54 COc1cc(NS(=O)(=O)c2ccc(F)cc2)ccc1Br ZINC000147471907 FG On-Demand Anodyne HTR6 29 43 COc1cc(NS(=O)(=O)c2ccc(F)cc2)ccc1Br ZINC000147471907 FG On-Demand Anodyne CA4 20 54 COc1cc(NS(=O)(=O)c2ccc(F)cc2)ccc1Br ZINC000147471907 FG On-Demand Anodyne GHSR 28 53 COc1cc(NS(=O)(=O)c2ccc(F)cc2)ccc1Br ZINC000147471907 FG On-Demand Anodyne IDO1 24 40 COc1cc(NS(=O)(=O)c2ccc(F)cc2)ccc1Br ZINC000147471907 FG On-Demand Anodyne FFAR4 28 45 COc1cc(NS(=O)(=O)c2ccc(F)cc2)ccc1Br ZINC000147471907 FG On-Demand Anodyne MGAT1 48 37 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne AVPR2 32 42 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne AVPR1A 16 42 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne DHODH 17 45 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne PPIA 23 43 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne JUN 20 40 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne APOB 0 41 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne ECR 51 44 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne KCNA3 44 43 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne ATF1 57 39 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne COLA 74 40 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne CPT1A 72 40 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne CPT2 48 36 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne PYGL 17 47 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne PRNP 27 40 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne KDR 27 42 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne GRM4 32 42 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne NR1H4 17 49 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne ABCB1 0 40 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne MTTP 30 41 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne NFKB1 53 39 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne KCNMA1 35 40 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne CPT1B 47 37 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne ACPS 0 41 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne AKR1C3 44 40 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne SHH 23 46 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne AKR1C2 60 38 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne SMO 33 43 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne GLMU 0 44 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne BRD1 0 42 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne KCNK3 114 61 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne KCNK9 92 60 COc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471924 DG On-Demand Anodyne BRPF1 0 49 CCCOc1ccc(Oc2cc(NC)nc(N)n2)cc1 ZINC000147471928 CF For-Sale Anodyne DRTS_PLAFK 20 44 CCCOc1ccc(Oc2cc(NC)nc(N)n2)cc1 ZINC000147471928 CF For-Sale Anodyne ACACA 35 41 CO[C@@H]1CCC[C@@H]1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147471932 DF For-Sale Anodyne CACNA1I 41 32 C[C@H]1CCC[C@@H](C)N1NC(=O)CC1(CN)CCC1 ZINC000147471966 CD For-Sale Anodyne CACNA2D1 45 41 CC(C)N(C)CCCNC(=O)c1cc2cc(Br)ccc2[nH]1 ZINC000147471975 FG On-Demand Anodyne PYGL 82 50 CC(C)N(C)CCCNC(=O)c1cc2cc(Br)ccc2[nH]1 ZINC000147471975 FG On-Demand Anodyne PYK 69 47 Cc1c(NC(=O)c2ccccc2)cccc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147471979 HJ On-Demand Anodyne GRM5 16 46 Cc1c(NC(=O)c2ccccc2)cccc1NC(=O)c1ccn(-c2cccc(F)c2)n1 ZINC000147471979 HJ On-Demand Anodyne KCNK3 64 43 O=C(c1ccc2ncccc2c1)N1CCC[C@H]1CCCBr ZINC000147472008 EI For-Sale Reactive CCR3 0 41 O=C(c1ccc2ncccc2c1)N1CCC[C@H]1CCCBr ZINC000147472008 EI For-Sale Reactive HCRTR2 0 43 Cc1cccc(C(C)C)c1NC(=O)CC1(CN)CCC1 ZINC000147472064 CH For-Sale Anodyne SOAT1 46 41 Cc1cccc(C(C)C)c1NC(=O)CC1(CN)CCC1 ZINC000147472064 CH For-Sale Anodyne ACAT 0 51 COC(=O)[C@H](C)OCc1cccc(Br)c1 ZINC000147472103 CF For-Sale Anodyne MAOB 16 45 COC(=O)[C@H](C)OCc1cccc(Br)c1 ZINC000147472103 CF For-Sale Anodyne PAPA1_CARPA 22 40 COC(=O)[C@H](C)OCc1cccc(Br)c1 ZINC000147472103 CF For-Sale Anodyne HCAR2 17 49 O=C(CCOc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147472112 HF On-Demand Anodyne GRIN2B 32 43 O=C(CCOc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147472112 HF On-Demand Anodyne MMP13 41 42 O=C(CCOc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147472112 HF On-Demand Anodyne EPHX2 19 47 O=C(CCOc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147472112 HF On-Demand Anodyne TGM2 82 45 O=C(CCOc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147472112 HF On-Demand Anodyne MMP7 46 38 O=C(CCOc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147472112 HF On-Demand Anodyne F13A1 88 45 COc1cc(NS(=O)(=O)c2cccc(C#N)c2)ccc1Br ZINC000147472120 FG On-Demand Mild HTR6 17 43 CO[C@H]1CCC[C@@H]1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147472134 DF For-Sale Anodyne CACNA1I 41 32 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147472143 DG On-Demand Mild CMA1 0 40 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147472143 DG On-Demand Mild CTSG 17 40 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147472143 DG On-Demand Mild CPT1A 28 42 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147472143 DG On-Demand Mild PRNP 27 46 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147472143 DG On-Demand Mild SCN10A 15 43 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147472143 DG On-Demand Mild CTRB_BOVIN 45 34 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147472143 DG On-Demand Mild KCNK3 59 37 O=C(Nc1ccc(Cl)cc1Br)N1CCCCC1 ZINC000147472151 DI For-Sale Anodyne EPHX2 21 42 O=C(Nc1ccc(Cl)cc1Br)N1CCCCC1 ZINC000147472151 DI For-Sale Anodyne RBP4 22 44 Nc1cccc(NCC2CCCC2)c1[N+](=O)[O-] ZINC000147472171 BF For-Sale Bother PRKCQ 44 35 CC(C)CCCCNC(=O)[C@@H](C)CCN ZINC000147472201 BD For-Sale Anodyne SIRT1 36 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)NCC(C)C)c(Cl)c2)c1 ZINC000147472205 HH On-Demand Bother F3 78 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)NCC(C)C)c(Cl)c2)c1 ZINC000147472205 HH On-Demand Bother TAAR1 26 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)NCC(C)C)c(Cl)c2)c1 ZINC000147472205 HH On-Demand Bother AKR1C2 46 38 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)NCC(C)C)c(Cl)c2)c1 ZINC000147472205 HH On-Demand Bother USP7 29 42 COc1ccc([N+](=O)[O-])c(C(=O)Nc2ccc(C(=O)NCC(C)C)c(Cl)c2)c1 ZINC000147472205 HH On-Demand Bother USP47 36 42 C[C@H]1CCC[C@H](C)N1NC(=O)CC1(CN)CCC1 ZINC000147472209 CD For-Sale Anodyne CACNA2D1 45 41 O=C(c1csc2ccccc12)N1CCC[C@@H]1CCCBr ZINC000147472286 FJ For-Sale Reactive HCRTR1 15 45 CO[C@@H]1CCC[C@H]1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147472302 DF For-Sale Anodyne CACNA1I 41 32 COC(=O)[C@@H](C)OCc1cccc(Br)c1 ZINC000147472309 CF For-Sale Anodyne MAOB 16 45 COC(=O)[C@@H](C)OCc1cccc(Br)c1 ZINC000147472309 CF For-Sale Anodyne PAPA1_CARPA 22 40 COC(=O)[C@@H](C)OCc1cccc(Br)c1 ZINC000147472309 CF For-Sale Anodyne HCAR2 17 49 Cc1noc(C)c1CNS(=O)(=O)c1ccc(OCC(C)C)cc1 ZINC000147472347 EF On-Demand Anodyne ADAMTS4 41 33 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Cl)c1 ZINC000147472369 EI For-Sale Anodyne AVPR2 26 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Cl)c1 ZINC000147472369 EI For-Sale Anodyne PPIA 15 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Cl)c1 ZINC000147472369 EI For-Sale Anodyne HTR1F 15 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Cl)c1 ZINC000147472369 EI For-Sale Anodyne ATF1 57 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Cl)c1 ZINC000147472369 EI For-Sale Anodyne CPT1A 0 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Cl)c1 ZINC000147472369 EI For-Sale Anodyne PYGL 25 54 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Cl)c1 ZINC000147472369 EI For-Sale Anodyne NFKB1 53 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Cl)c1 ZINC000147472369 EI For-Sale Anodyne SMO 24 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Cl)c1 ZINC000147472369 EI For-Sale Anodyne GPR35 25 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Cl)c1 ZINC000147472369 EI For-Sale Anodyne KCNK3 42 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Cl)c1 ZINC000147472369 EI For-Sale Anodyne TMPRSS4 0 42 CC(C)CCCCNC(=O)[C@H](C)CCN ZINC000147472411 BD For-Sale Anodyne SIRT1 36 40 C[C@@H]1CCC[C@@H](C)N1NC(=O)CC1(CN)CCC1 ZINC000147472414 CD For-Sale Anodyne CACNA2D1 45 41 CC(C)CNC(=O)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1Cl ZINC000147472452 HI On-Demand Anodyne AVPR2 42 38 CC(C)CNC(=O)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1Cl ZINC000147472452 HI On-Demand Anodyne AVPR1A 18 41 CC(C)CNC(=O)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1Cl ZINC000147472452 HI On-Demand Anodyne GRM4 42 43 CC(C)CNC(=O)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1Cl ZINC000147472452 HI On-Demand Anodyne F3 48 32 O=C(c1csc2ccccc12)N1CCC[C@H]1CCCBr ZINC000147472496 FJ For-Sale Reactive HCRTR1 15 45 CC(C)N(Cc1ccccc1)C(=O)CC1(CN)CCC1 ZINC000147472502 CF For-Sale Anodyne CACNA2D1 46 43 CO[C@H]1CCC[C@H]1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147472517 DF For-Sale Anodyne CACNA1I 41 32 CCOC(=O)[C@@H](C)OCc1cccc(Br)c1 ZINC000147472523 CF For-Sale Anodyne HCAR2 16 48 CCOC(=O)[C@@H](C)OCc1cccc(Br)c1 ZINC000147472523 CF For-Sale Anodyne FFAR1 19 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1COc2ccccc2O1 ZINC000147472553 HE On-Demand Anodyne EPHX2 18 47 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1COc2ccccc2O1 ZINC000147472553 HE On-Demand Anodyne PKM 22 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1COc2ccccc2O1 ZINC000147472553 HE On-Demand Anodyne TGM2 55 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)[C@H]1COc2ccccc2O1 ZINC000147472553 HE On-Demand Anodyne F13A1 50 43 COc1cc(NS(=O)(=O)c2ccc(C)cc2Br)ccc1Br ZINC000147472576 II On-Demand Anodyne UTS2R 0 44 COc1cc(NS(=O)(=O)c2ccc(C)cc2Br)ccc1Br ZINC000147472576 II On-Demand Anodyne ALPL 29 43 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2Cl)c1 ZINC000147472601 EI For-Sale Anodyne PPIA 23 40 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2Cl)c1 ZINC000147472601 EI For-Sale Anodyne JAK1 24 58 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2Cl)c1 ZINC000147472601 EI For-Sale Anodyne TYK2 51 46 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2Cl)c1 ZINC000147472601 EI For-Sale Anodyne TAAR1 27 41 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2Cl)c1 ZINC000147472601 EI For-Sale Anodyne AKR1C3 31 43 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2Cl)c1 ZINC000147472601 EI For-Sale Anodyne KCNK3 60 42 COCc1nc(C(=O)N2CCCN(S(=O)(=O)c3ccc(F)cc3)CC2)cs1 ZINC000147472631 HD On-Demand Anodyne TGM2 45 39 COCc1nc(C(=O)N2CCCN(S(=O)(=O)c3ccc(F)cc3)CC2)cs1 ZINC000147472631 HD On-Demand Anodyne F13A1 51 39 COc1ccc(C)cc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147472634 CG For-Sale Anodyne AKR1C3 36 44 COc1ccc(C)cc1Nc1ccc(C(=O)O)c(C)n1 ZINC000147472634 CG For-Sale Anodyne AKR1C2 73 42 CCCOc1ccc(Oc2cc(NCC)nc(C)n2)cc1 ZINC000147472637 CH For-Sale Anodyne ACACA 38 40 CCCOc1ccc(Oc2cc(NCC)nc(C)n2)cc1 ZINC000147472637 CH For-Sale Anodyne ACACB 19 40 C[C@H]1CCC[C@@H](C)N1NC(=O)c1csc(N)n1 ZINC000147472658 CD For-Sale Anodyne TRPC6 47 39 COc1cc2c(cc1OC)CN(C(=O)C1(N)CCC1)CC2 ZINC000147472692 CD On-Demand Anodyne ABCB1 24 53 Cc1noc(C)c1CNS(=O)(=O)c1ccc2c(c1)CCCC(=O)N2 ZINC000147472714 EE On-Demand Anodyne PKM 41 47 CC(C)(C)OC(=O)N1CCCC[C@@H]1C(=O)N1CCC(C(=O)O)CC1 ZINC000147472730 EE On-Demand Anodyne PREP 62 77 CC(C)(C)OC(=O)N1CCCC[C@@H]1C(=O)N1CCC(C(=O)O)CC1 ZINC000147472730 EE On-Demand Anodyne SFRP1 54 48 CC(C)(C)OC(=O)N1CCCC[C@@H]1C(=O)N1CCC(C(=O)O)CC1 ZINC000147472730 EE On-Demand Anodyne WNT3 62 48 O=C(c1ccc(OC(F)F)cc1)N1CCC[C@@H]1CCCBr ZINC000147472737 FI For-Sale Reactive HCRTR1 18 46 O=C1C[C@@H](C(=O)Nc2ncc(Cc3ccc(F)c(F)c3)s2)c2ccc(F)cc2N1 ZINC000147472740 HI On-Demand Anodyne SCD 30 44 CCOC(=O)[C@H](C)OCc1cccc(Br)c1 ZINC000147472749 CF For-Sale Anodyne HCAR2 16 48 CCOC(=O)[C@H](C)OCc1cccc(Br)c1 ZINC000147472749 CF For-Sale Anodyne FFAR1 19 42 O=C(COc1ccccc1F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147472775 HE On-Demand Anodyne EPHX2 20 40 O=C(COc1ccccc1F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147472775 HE On-Demand Anodyne TGM2 68 43 O=C(COc1ccccc1F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147472775 HE On-Demand Anodyne F13A1 66 43 O=C(COc1ccccc1F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147472775 HE On-Demand Anodyne NAMPT 19 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2Cl)c1 ZINC000147472797 GJ On-Demand Anodyne PPIA 15 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2Cl)c1 ZINC000147472797 GJ On-Demand Anodyne ATF1 47 38 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2Cl)c1 ZINC000147472797 GJ On-Demand Anodyne F12 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2Cl)c1 ZINC000147472797 GJ On-Demand Anodyne NFKB1 44 38 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2Cl)c1 ZINC000147472797 GJ On-Demand Anodyne CSF1R 15 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2Cl)c1 ZINC000147472797 GJ On-Demand Anodyne AKR1C3 18 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2Cl)c1 ZINC000147472797 GJ On-Demand Anodyne KCNK3 21 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2Cl)c1 ZINC000147472797 GJ On-Demand Anodyne TMPRSS4 0 40 Cc1cc(N)cc(C)c1S(=O)(=O)Nc1ccncc1Br ZINC000147472843 FF For-Sale Anodyne PTGS1 0 40 C[C@H]1CCC[C@H](C)N1NC(=O)c1csc(N)n1 ZINC000147472847 CD For-Sale Anodyne TRPC6 47 39 NC1(C(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147472853 CD On-Demand Anodyne ERBB2 0 44 NC1(C(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147472853 CD On-Demand Anodyne MMP2 0 44 NC1(C(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147472853 CD On-Demand Anodyne MMP9 0 43 NC1(C(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147472853 CD On-Demand Anodyne AKR1C3 23 50 CCN(CC)CCC[C@@H](C)Nc1ccc(C(=O)O)c(C)n1 ZINC000147472859 CG For-Sale Anodyne CACNA2D1 26 51 CCN(CC)CCC[C@@H](C)Nc1ccc(C(=O)O)c(C)n1 ZINC000147472859 CG For-Sale Anodyne RBP_CHICK 0 40 O=C1C[C@H](C(=O)Nc2ncc(Cc3ccc(F)c(F)c3)s2)c2ccc(F)cc2N1 ZINC000147472908 HI On-Demand Anodyne SCD 30 44 O=C(c1ccc(OC(F)F)cc1)N1CCC[C@H]1CCCBr ZINC000147472913 FI For-Sale Reactive HCRTR1 18 46 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)N1CCC(C(=O)O)CC1 ZINC000147472924 EE On-Demand Anodyne PREP 62 77 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)N1CCC(C(=O)O)CC1 ZINC000147472924 EE On-Demand Anodyne SFRP1 54 48 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)N1CCC(C(=O)O)CC1 ZINC000147472924 EE On-Demand Anodyne WNT3 62 48 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3ccc(Cl)cc3)nc2)C1 ZINC000147472952 HG On-Demand Anodyne CACNA1I 62 36 CNc1cc(C(=O)NCCNC(N)=O)ccc1[N+](=O)[O-] ZINC000147472960 CC For-Sale Bother GSTM2 47 37 N#Cc1ccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147472974 HE On-Demand Mild MMP13 33 41 N#Cc1ccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147472974 HE On-Demand Mild ADAM17 42 42 N#Cc1ccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147472974 HE On-Demand Mild CPT1A 18 42 N#Cc1ccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147472974 HE On-Demand Mild EPHX2 15 43 N#Cc1ccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147472974 HE On-Demand Mild TRPV4 46 42 N#Cc1ccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147472974 HE On-Demand Mild TGM2 59 42 N#Cc1ccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147472974 HE On-Demand Mild F13A1 56 42 N#Cc1ccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147472974 HE On-Demand Mild MEN1 41 36 COc1cc(C(=O)N2CCN(CCO)CC2)ccc1F ZINC000147472989 CC On-Demand Anodyne DRD4 40 33 COc1cc(C(=O)N2CCN(CCO)CC2)ccc1F ZINC000147472989 CC On-Demand Anodyne SLC29A2 0 42 CCCNCC(=O)NCCCCC(C)C ZINC000147472999 BD For-Sale Anodyne NOD1 32 40 C[C@@H]1CCC[C@@H](C)N1NC(=O)c1csc(N)n1 ZINC000147473015 CD For-Sale Anodyne TRPC6 47 39 O=C(CC1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473034 CH On-Demand Anodyne GRIN1 15 40 O=C(CC1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473034 CH On-Demand Anodyne CACNA1I 61 39 O=C(Nc1cc(Cl)cc(C(=O)O)c1)N[C@@H]1CCCNC1=O ZINC000147473042 DD On-Demand Anodyne GRIN1 19 43 CCN(CC)CCC[C@H](C)Nc1ccc(C(=O)O)c(C)n1 ZINC000147473049 CG For-Sale Anodyne CACNA2D1 26 51 CCN(CC)CCC[C@H](C)Nc1ccc(C(=O)O)c(C)n1 ZINC000147473049 CG For-Sale Anodyne RBP_CHICK 0 40 Nc1cc(S(=O)(=O)Nc2ccncc2Br)ccc1O ZINC000147473093 ED For-Sale Anodyne PTGS1 0 42 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)COCC(=O)O ZINC000147473094 CD For-Sale Bother CACNA1C 51 38 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)COCC(=O)O ZINC000147473094 CD For-Sale Bother CACNA1D 80 37 CCOC(=O)Cc1csc(-c2ccc(Cl)cc2F)n1 ZINC000147473100 CH For-Sale Anodyne PTGER1 22 45 CCOC(=O)Cc1csc(-c2ccc(Cl)cc2F)n1 ZINC000147473100 CH For-Sale Anodyne DPP8 75 37 CCOC(=O)Cc1csc(-c2ccc(Cl)cc2F)n1 ZINC000147473100 CH For-Sale Anodyne DPP9 71 37 NCC1(CC(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147473105 CD For-Sale Anodyne HTR1A 18 42 NCC1(CC(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147473105 CD For-Sale Anodyne CACNA2D1 0 43 NCC1(CC(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147473105 CD For-Sale Anodyne ERBB2 0 45 NCC1(CC(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147473105 CD For-Sale Anodyne MMP2 0 45 NCC1(CC(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147473105 CD For-Sale Anodyne MMP9 0 45 NCC1(CC(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147473105 CD For-Sale Anodyne ADAM10 37 45 NCC1(CC(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147473105 CD For-Sale Anodyne AKR1C3 0 45 NCC1(CC(=O)N2CCN(c3ccccc3)CC2)CCC1 ZINC000147473105 CD For-Sale Anodyne SLC6A7 0 43 COc1cc(NS(=O)(=O)c2ccc(Cl)nc2)ccc1Br ZINC000147473133 GG On-Demand Anodyne HTR6 16 42 CCOC(=O)[C@H](F)OCc1cccc(Br)c1 ZINC000147473140 CF For-Sale Anodyne HCAR2 18 50 CCOC(=O)[C@H](F)OCc1cccc(Br)c1 ZINC000147473140 CF For-Sale Anodyne FFAR1 15 41 COC(=O)c1ccc(-c2ccc(F)cc2)c(OC)c1 ZINC000147473142 CG For-Sale Anodyne GRIN2B 40 42 COC(=O)c1ccc(-c2ccc(F)cc2)c(OC)c1 ZINC000147473142 CG For-Sale Anodyne GYS1 46 34 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3ccc(Cl)cc3)nc2)C1 ZINC000147473163 HG On-Demand Anodyne CACNA1I 62 36 N#Cc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473195 HE On-Demand Mild ADRB1 41 32 N#Cc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473195 HE On-Demand Mild EPHX2 15 43 N#Cc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473195 HE On-Demand Mild TRPV4 41 31 N#Cc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473195 HE On-Demand Mild TGM2 59 42 N#Cc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473195 HE On-Demand Mild F13A1 54 42 O=C(Nc1cc(Cl)cc(C(=O)O)c1)N[C@H]1CCCNC1=O ZINC000147473238 DD On-Demand Anodyne GRIN1 19 43 Cc1cccc(C(C)C)c1Nc1ccc(C(=O)O)c(C)n1 ZINC000147473245 CI For-Sale Anodyne SOAT1 41 34 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)COCC(=O)O ZINC000147473277 CD For-Sale Bother CACNA1C 51 38 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)COCC(=O)O ZINC000147473277 CD For-Sale Bother CACNA1D 80 37 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)c3ccc(C)cc3)c2)c1 ZINC000147473279 HI On-Demand Bother ROCK2 30 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)c3ccc(C)cc3)c2)c1 ZINC000147473279 HI On-Demand Bother TAAR1 43 54 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)c3ccc(C)cc3)c2)c1 ZINC000147473279 HI On-Demand Bother AKR1C3 21 41 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)c3ccc(C)cc3)c2)c1 ZINC000147473279 HI On-Demand Bother KCNK3 104 48 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)c3ccc(C)cc3)c2)c1 ZINC000147473279 HI On-Demand Bother KCNK9 62 39 O=C(O)c1cc(Cl)cc(NC(=O)c2c(Cl)cccc2Cl)c1 ZINC000147473282 EJ On-Demand Anodyne CPT1A 27 42 O=C(O)c1cc(Cl)cc(NC(=O)c2c(Cl)cccc2Cl)c1 ZINC000147473282 EJ On-Demand Anodyne TYK2 73 44 O=C(O)c1cc(Cl)cc(NC(=O)c2c(Cl)cccc2Cl)c1 ZINC000147473282 EJ On-Demand Anodyne TAAR1 31 45 O=C(O)c1cc(Cl)cc(NC(=O)c2c(Cl)cccc2Cl)c1 ZINC000147473282 EJ On-Demand Anodyne AKR1C3 38 49 O=C(O)c1cc(Cl)cc(NC(=O)c2c(Cl)cccc2Cl)c1 ZINC000147473282 EJ On-Demand Anodyne SMO 22 42 O=C(O)c1cc(Cl)cc(NC(=O)c2c(Cl)cccc2Cl)c1 ZINC000147473282 EJ On-Demand Anodyne KCNK3 77 47 O=C(O)c1cc(Cl)cc(NC(=O)c2c(Cl)cccc2Cl)c1 ZINC000147473282 EJ On-Demand Anodyne KCNK9 37 40 O=C(NCc1ccn2ccnc2c1)c1cnc(-c2ccccc2)s1 ZINC000147473297 EG On-Demand Anodyne NAMPT 23 42 C[C@H](Cc1cccc(F)c1)C(=O)NCC1(c2ccccc2)CC1 ZINC000147473313 DH On-Demand Anodyne MME 66 37 C[C@H](Cc1cccc(F)c1)C(=O)NCC1(c2ccccc2)CC1 ZINC000147473313 DH On-Demand Anodyne TACR1 19 46 C[C@H](Cc1cccc(F)c1)C(=O)NCC1(c2ccccc2)CC1 ZINC000147473313 DH On-Demand Anodyne PAPA1_CARPA 24 42 C[C@H](Cc1cccc(F)c1)C(=O)NCC1(c2ccccc2)CC1 ZINC000147473313 DH On-Demand Anodyne CTSL 22 42 C[C@H](Cc1cccc(F)c1)C(=O)NCC1(c2ccccc2)CC1 ZINC000147473313 DH On-Demand Anodyne CPA1 15 42 C[C@H](Cc1cccc(F)c1)C(=O)NCC1(c2ccccc2)CC1 ZINC000147473313 DH On-Demand Anodyne KCNA3 47 37 C[C@H](Cc1cccc(F)c1)C(=O)NCC1(c2ccccc2)CC1 ZINC000147473313 DH On-Demand Anodyne SOAT1 16 45 C[C@H](Cc1cccc(F)c1)C(=O)NCC1(c2ccccc2)CC1 ZINC000147473313 DH On-Demand Anodyne CTSS 18 42 C[C@H](Cc1cccc(F)c1)C(=O)NCC1(c2ccccc2)CC1 ZINC000147473313 DH On-Demand Anodyne ACE2 61 37 C[C@H](Cc1cccc(F)c1)C(=O)NCC1(c2ccccc2)CC1 ZINC000147473313 DH On-Demand Anodyne AMP1_PLAFQ 47 31 CCCOc1ccc(Oc2nc(N)nc(OCC)n2)cc1 ZINC000147473329 CE For-Sale Anodyne DRTS_PLAFK 17 45 CCCOc1ccc(Oc2nc(N)nc(OCC)n2)cc1 ZINC000147473329 CE For-Sale Anodyne ACACA 32 40 CCOC(=O)[C@@H](F)OCc1cccc(Br)c1 ZINC000147473331 CF For-Sale Anodyne HCAR2 18 50 CCOC(=O)[C@@H](F)OCc1cccc(Br)c1 ZINC000147473331 CF For-Sale Anodyne FFAR1 15 41 COc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147473346 CE On-Demand Anodyne CSNK1D 49 64 COc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147473346 CE On-Demand Anodyne PIK3CA 22 48 COc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147473346 CE On-Demand Anodyne ITK 0 58 COc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147473346 CE On-Demand Anodyne LUCI_PHOPE 31 40 COc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147473346 CE On-Demand Anodyne FABK 0 51 COc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147473346 CE On-Demand Anodyne PORCN 0 44 COc1ccc2nc(NC(=O)C3(N)CCC3)sc2c1 ZINC000147473346 CE On-Demand Anodyne ISPD 0 53 COc1cc(NS(=O)(=O)c2ccc(C#N)cc2)ccc1Br ZINC000147473347 FG On-Demand Mild HTR6 20 46 COc1cc(NS(=O)(=O)c2ccc(C#N)cc2)ccc1Br ZINC000147473347 FG On-Demand Mild GHSR 0 44 COc1cc(NS(=O)(=O)c2ccc(C#N)cc2)ccc1Br ZINC000147473347 FG On-Demand Mild IDO1 27 49 Cc1nn(C(F)F)c(C)c1CC(=O)Nc1ccc2oc(C(C)C)nc2c1 ZINC000147473383 FI On-Demand Anodyne IMDH_CRYPV 47 36 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473413 HD On-Demand Anodyne DRD2 19 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473413 HD On-Demand Anodyne DRD4 28 42 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473413 HD On-Demand Anodyne ACHE 37 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473413 HD On-Demand Anodyne CHRM3 15 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473413 HD On-Demand Anodyne CCR3 81 44 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473413 HD On-Demand Anodyne CACNA1I 44 39 Cc1ccc2c(c1)CCN(C(=O)c1cc(S(C)(=O)=O)ccc1OC(C)C)C2 ZINC000147473419 GG On-Demand Anodyne SLC6A9 54 59 CNCc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147473428 CH For-Sale Anodyne MAOB 73 46 CNCc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147473428 CH For-Sale Anodyne F9 0 40 CNCc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147473428 CH For-Sale Anodyne GYS1 42 35 CNCc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147473428 CH For-Sale Anodyne FFAR1 37 41 Cc1noc(C)c1CNS(=O)(=O)c1cccc(Cl)c1F ZINC000147473446 DF On-Demand Anodyne EDNRA 25 44 Cc1cccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147473452 HF On-Demand Anodyne F2 17 41 Cc1cccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147473452 HF On-Demand Anodyne MMP13 18 40 Cc1cccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147473452 HF On-Demand Anodyne EPHX2 39 45 Cc1cccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147473452 HF On-Demand Anodyne TGM2 66 42 Cc1cccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147473452 HF On-Demand Anodyne CACNA1I 41 32 Cc1cccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147473452 HF On-Demand Anodyne F13A1 65 42 Cc1cccc(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147473452 HF On-Demand Anodyne AKR1C3 43 36 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2C)c1 ZINC000147473457 HI On-Demand Bother NR1H4 15 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2C)c1 ZINC000147473457 HI On-Demand Bother PYGM 23 47 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2C)c1 ZINC000147473457 HI On-Demand Bother KCNMA1 31 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2C)c1 ZINC000147473457 HI On-Demand Bother LUCI_LUCLA 23 41 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2C)c1 ZINC000147473457 HI On-Demand Bother TAAR1 32 51 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2C)c1 ZINC000147473457 HI On-Demand Bother AKR1C3 39 52 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2C)c1 ZINC000147473457 HI On-Demand Bother ABCG2 28 44 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2C)c1 ZINC000147473457 HI On-Demand Bother AKR1C2 70 51 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2C)c1 ZINC000147473457 HI On-Demand Bother GPR35 36 40 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2C)c1 ZINC000147473457 HI On-Demand Bother KCNK3 94 46 COc1ccc([N+](=O)[O-])c(C(=O)Nc2cccc(NC(=O)c3ccccc3)c2C)c1 ZINC000147473457 HI On-Demand Bother KCNK9 50 37 CCc1ncc(C(=O)NCCc2ccc(-c3csc(C)n3)cc2)s1 ZINC000147473463 FI On-Demand Anodyne ROCK1 15 44 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)/C=C/C(=O)O ZINC000147473496 CD For-Sale Bother CACNA1C 42 36 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)/C=C/C(=O)O ZINC000147473496 CD For-Sale Bother CACNA1D 65 36 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild CA2 97 49 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild CA1 92 51 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild CA7 40 44 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild CA5B 49 42 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild CA4 72 48 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild CA5A 56 42 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild CA14 33 47 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild CA12 74 51 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild CA9 82 51 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild UREA_CANEN 28 44 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild CYNT 47 49 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild NCE103 31 40 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild MTCA1 60 51 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild P96878_MYCTU 73 51 C=C(C)c1cccc(C(C)(C)NC(=O)Nc2ccc(S(N)(=O)=O)cc2)c1 ZINC000147473528 FG For-Sale Mild IMDH_CRYPV 106 73 COc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147473543 DF For-Sale Anodyne LCK 22 41 COc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147473543 DF For-Sale Anodyne CSNK1D 59 63 COc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147473543 DF For-Sale Anodyne NMT1 36 40 COc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147473543 DF For-Sale Anodyne PIK3CA 20 46 COc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147473543 DF For-Sale Anodyne ITK 0 41 COc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147473543 DF For-Sale Anodyne PIK3CG 18 40 COc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147473543 DF For-Sale Anodyne FABK 0 49 COc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147473543 DF For-Sale Anodyne PORCN 0 49 COc1ccc2nc(NC(=O)CC3(CN)CCC3)sc2c1 ZINC000147473543 DF For-Sale Anodyne ISPD 0 55 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne AVPR2 58 45 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne AVPR1A 33 44 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne PPIA 16 46 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne JUN 22 43 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne ECR 69 43 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne ATF1 55 38 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne PRNP 36 43 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne GRM4 35 47 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne NR1H4 23 46 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne NFKB1 51 38 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne CSF1R 17 41 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne ACPS 0 41 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne CCR8 45 32 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne AKR1C3 45 42 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne NR2E3 47 42 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne SHH 34 40 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne CYA 0 45 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne AKR1C2 37 40 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne SMO 33 45 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne Q25615_ONCVO 42 31 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne E3UJZ5_SPOLI 52 43 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne KCNK3 120 58 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne KCNK9 86 51 Cc1ccccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147473556 CH On-Demand Anodyne TMPRSS4 0 42 CCCOc1ccc(Oc2ncnc(N)c2C(C)C)cc1 ZINC000147473567 CH For-Sale Anodyne ACACA 34 40 CCCOc1ccc(Oc2ncnc(N)c2C(C)C)cc1 ZINC000147473567 CH For-Sale Anodyne ACACB 16 40 COc1cc(NS(=O)(=O)c2ccc(F)cc2Br)ccc1Br ZINC000147473577 II On-Demand Anodyne UTS2R 0 46 O=C([C@@H]1CSc2ccccc21)N1CCC[C@@H]1CCCBr ZINC000147473623 FI For-Sale Reactive PREP 49 33 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473636 HD On-Demand Anodyne DRD2 19 40 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473636 HD On-Demand Anodyne DRD4 28 42 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473636 HD On-Demand Anodyne ACHE 37 40 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473636 HD On-Demand Anodyne CHRM3 15 40 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473636 HD On-Demand Anodyne CCR3 81 44 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(CN3CCN(C)CC3)c2)C1 ZINC000147473636 HD On-Demand Anodyne CACNA1I 44 39 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)/C=C/C(=O)O ZINC000147473686 CD For-Sale Bother CACNA1C 42 36 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)/C=C/C(=O)O ZINC000147473686 CD For-Sale Bother CACNA1D 65 36 COC(=O)[C@H](Br)COCc1cccc(Br)c1 ZINC000147473689 FF For-Sale Reactive HCAR2 16 47 Cc1nc(N2CCN(c3nccs3)CC2)ccc1C(=O)O ZINC000147473691 DD For-Sale Anodyne SORD 88 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(=O)[nH]n1 ZINC000147473722 GC On-Demand Anodyne HTR4 46 36 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(=O)[nH]n1 ZINC000147473722 GC On-Demand Anodyne GRIN2B 27 60 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(=O)[nH]n1 ZINC000147473722 GC On-Demand Anodyne TGM2 57 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(=O)[nH]n1 ZINC000147473722 GC On-Demand Anodyne CACNA1I 51 33 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc(=O)[nH]n1 ZINC000147473722 GC On-Demand Anodyne F13A1 51 43 COc1ccc(N)cc1S(=O)(=O)Nc1ccncc1Br ZINC000147473734 FE For-Sale Anodyne ALPL 27 43 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)c1 ZINC000147473756 DH On-Demand Anodyne AVPR2 29 47 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)c1 ZINC000147473756 DH On-Demand Anodyne JUN 22 45 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)c1 ZINC000147473756 DH On-Demand Anodyne ECR 24 43 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)c1 ZINC000147473756 DH On-Demand Anodyne ATF1 58 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)c1 ZINC000147473756 DH On-Demand Anodyne CPT1A 41 39 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)c1 ZINC000147473756 DH On-Demand Anodyne NR1H4 18 48 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)c1 ZINC000147473756 DH On-Demand Anodyne NFKB1 54 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)c1 ZINC000147473756 DH On-Demand Anodyne KCNK3 83 43 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)c1 ZINC000147473756 DH On-Demand Anodyne KCNK9 58 43 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)c1 ZINC000147473756 DH On-Demand Anodyne TMPRSS4 0 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(C)cc2C)CC1 ZINC000147473794 FF On-Demand Anodyne F2 17 42 CCCC[C@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(C)cc2C)CC1 ZINC000147473794 FF On-Demand Anodyne P2RY12 173 36 O=C([C@H]1CSc2ccccc21)N1CCC[C@@H]1CCCBr ZINC000147473839 FI For-Sale Reactive PREP 49 33 COC(=O)[C@@H](Br)COCc1cccc(Br)c1 ZINC000147473867 FF For-Sale Reactive HCAR2 16 47 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCC(=O)O ZINC000147473930 CD For-Sale Bother CACNA1C 45 38 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCC(=O)O ZINC000147473930 CD For-Sale Bother CACNA1D 70 36 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C)cc2OCC(F)(F)F)C1 ZINC000147473931 HF On-Demand Anodyne CACNA1I 65 36 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother GRIN2B 24 42 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother CCR5 19 43 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother MMP2 27 44 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother MMP8 50 44 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother MMP9 32 44 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother EPHX2 15 44 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother TGM2 78 47 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother MMP1 46 44 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother CACNA1I 36 42 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother F13A1 82 47 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother LUXR 20 42 O=C(Cc1ccc([N+](=O)[O-])cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147473960 HE On-Demand Bother NAMPT 53 40 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CA2 136 51 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CA6 33 40 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CA1 48 33 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CA7 78 47 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CA13 23 40 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CA5B 65 47 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CA4 106 51 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CA5A 70 47 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CA14 58 45 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CA12 99 61 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CA9 111 51 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CAH_METTE 34 44 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne UREA_CANEN 29 44 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne IDO1 0 45 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne CYNT 50 45 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne NCE103 66 42 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne MTCA1 51 51 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne P96878_MYCTU 71 50 NC1(C(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147473990 CC On-Demand Anodyne Q5TU56_ANOGA 0 41 CCc1ncc(C(=O)N2CCN(CCCc3nc(-c4cccs4)no3)CC2)s1 ZINC000147474005 HG On-Demand Anodyne ETHR 42 42 C[C@H](CNc1ccc(Cl)cc1[N+](=O)[O-])CC(=O)O ZINC000147474006 CF For-Sale Bother COLA 48 37 C[C@H](CNc1ccc(Cl)cc1[N+](=O)[O-])CC(=O)O ZINC000147474006 CF For-Sale Bother OXER1 40 34 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(C)cc2C)CC1 ZINC000147474007 FF On-Demand Anodyne F2 17 42 CCCC[C@@H](NC(N)=O)C(=O)N1CCC(C(=O)c2ccc(C)cc2C)CC1 ZINC000147474007 FF On-Demand Anodyne P2RY12 173 36 O=C([C@@H]1CSc2ccccc21)N1CCC[C@H]1CCCBr ZINC000147474067 FI For-Sale Reactive PREP 49 33 C[C@@](O)(COCc1cccc(Br)c1)C(=O)O ZINC000147474091 CD For-Sale Anodyne HCAR2 16 48 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C)cc2OCC(F)(F)F)C1 ZINC000147474118 HF On-Demand Anodyne CACNA1I 65 36 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCC(=O)O ZINC000147474135 CD For-Sale Bother CACNA1C 45 38 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCC(=O)O ZINC000147474135 CD For-Sale Bother CACNA1D 70 36 Nc1cc(C(=O)O)ccc1S(=O)(=O)Nc1ccncc1Br ZINC000147474142 FD For-Sale Anodyne NEU3 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne PPIA 16 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne ECR 30 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne ATF1 57 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne PRNP 21 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne GRM4 35 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne NR1H4 24 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne NFKB1 53 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne KCNMA1 17 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne ACPS 0 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne AKR1C3 39 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne NR2E3 54 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne CYA 0 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne AKR1C2 31 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne SMO 24 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne GALE 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne Q25615_ONCVO 44 33 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne E3UJZ5_SPOLI 24 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne KCNK3 97 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne KCNK9 74 35 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2F)c1 ZINC000147474156 CG On-Demand Anodyne TMPRSS4 0 45 C[C@@H](CNc1ccc(Cl)cc1[N+](=O)[O-])CC(=O)O ZINC000147474184 CF For-Sale Bother COLA 48 37 C[C@@H](CNc1ccc(Cl)cc1[N+](=O)[O-])CC(=O)O ZINC000147474184 CF For-Sale Bother OXER1 40 34 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CA2 151 62 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CA1 132 57 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CA7 72 52 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CA13 23 47 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CA5B 70 52 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CA4 129 62 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CA5A 76 52 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CA14 55 52 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CA12 90 57 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CA9 93 57 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CAH_METTE 28 40 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne CYNT 47 42 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne NCE103 51 41 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne MTCA1 62 47 NCC1(CC(=O)Nc2ccc(S(N)(=O)=O)cc2)CCC1 ZINC000147474189 CC For-Sale Anodyne P96878_MYCTU 77 47 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne HTR1A 21 40 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne DRD2 30 41 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne FKBP1A 28 41 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne DRD4 18 41 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne ADRA1D 26 40 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne ADRA1A 19 40 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne ADRA1B 20 40 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne CHRM5 17 43 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne EPHX2 22 45 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne TGM2 68 48 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne F13A1 72 43 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne MBTPS1 43 32 COc1ccccc1OCC(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474209 HE On-Demand Anodyne ACKR3 62 35 O=C([C@H]1CSc2ccccc21)N1CCC[C@H]1CCCBr ZINC000147474237 FI For-Sale Reactive PREP 49 33 C[C@](O)(COCc1cccc(Br)c1)C(=O)O ZINC000147474255 CD For-Sale Anodyne HCAR2 16 48 Cc1nc(N2c3ccccc3C[C@@H]2C)ccc1C(=O)O ZINC000147474268 CG For-Sale Anodyne DRD4 21 40 Cc1nc(N2c3ccccc3C[C@@H]2C)ccc1C(=O)O ZINC000147474268 CG For-Sale Anodyne TPP2 43 33 COc1cc(NS(=O)(=O)c2ccccc2F)ccc1Br ZINC000147474309 FG On-Demand Anodyne GHSR 0 40 COc1cc(NS(=O)(=O)c2ccccc2F)ccc1Br ZINC000147474309 FG On-Demand Anodyne NR1I2 27 43 COc1cc(NS(=O)(=O)c2ccccc2F)ccc1Br ZINC000147474309 FG On-Demand Anodyne SGK1 27 41 COc1cc(NS(=O)(=O)c2ccccc2F)ccc1Br ZINC000147474309 FG On-Demand Anodyne ALPL 26 41 C[C@@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474310 JI Annotated Anodyne HTR1A 78 43 C[C@@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474310 JI Annotated Anodyne DRD2 55 46 C[C@@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474310 JI Annotated Anodyne DRD4 31 43 C[C@@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474310 JI Annotated Anodyne HTR1D 51 37 C[C@@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474310 JI Annotated Anodyne HTR1B 50 37 C[C@@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474310 JI Annotated Anodyne HTR2A 49 41 C[C@@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474310 JI Annotated Anodyne HTR2C 40 38 C[C@@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474310 JI Annotated Anodyne ADRA1A 30 40 C[C@@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474310 JI Annotated Anodyne DRD3 70 46 C[C@@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474310 JI Annotated Anodyne HTR7 46 40 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CA2 108 54 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CA1 98 54 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CA7 77 54 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CA13 40 42 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CA4 67 48 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CA5A 40 34 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CA14 50 41 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CA12 79 54 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CA9 89 54 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CAH_METTE 42 42 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CYNT 40 44 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne NCE103 35 42 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CA15 25 42 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne MTCA1 39 43 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne P96878_MYCTU 47 43 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne CA 0 44 NS(=O)(=O)c1ccc(OC/C(Cl)=C/Cl)cc1 ZINC000147474352 CE On-Demand Anodyne A6YCJ1_9METZ 28 42 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCC(=O)O ZINC000147474353 CE For-Sale Bother CACNA1D 60 35 Cc1nc(N2c3ccccc3C[C@H]2C)ccc1C(=O)O ZINC000147474379 CG For-Sale Anodyne DRD4 21 40 Cc1nc(N2c3ccccc3C[C@H]2C)ccc1C(=O)O ZINC000147474379 CG For-Sale Anodyne TPP2 43 33 CN1[C@H](C(=O)O)C[C@H]2CCCC[C@H]21 ZINC000147474400 AD For-Sale Anodyne ACE 30 55 O=C(COc1cccc(F)c1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474436 HE On-Demand Anodyne CPT1A 46 35 O=C(COc1cccc(F)c1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474436 HE On-Demand Anodyne EPHX2 21 43 O=C(COc1cccc(F)c1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474436 HE On-Demand Anodyne TGM2 63 42 O=C(COc1cccc(F)c1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474436 HE On-Demand Anodyne F13A1 59 42 O=C(COc1cccc(F)c1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474436 HE On-Demand Anodyne AKR1C3 42 36 O=C(COc1cccc(F)c1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147474436 HE On-Demand Anodyne NAMPT 23 41 C/C(=C/COCc1cccc(Br)c1)C(=O)O ZINC000147474439 CF For-Sale Anodyne HCAR2 18 51 C[C@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474460 JI Annotated Anodyne HTR1A 78 43 C[C@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474460 JI Annotated Anodyne DRD2 55 46 C[C@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474460 JI Annotated Anodyne DRD4 31 43 C[C@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474460 JI Annotated Anodyne HTR1D 51 37 C[C@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474460 JI Annotated Anodyne HTR1B 50 37 C[C@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474460 JI Annotated Anodyne HTR2A 49 41 C[C@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474460 JI Annotated Anodyne HTR2C 40 38 C[C@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474460 JI Annotated Anodyne ADRA1A 30 40 C[C@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474460 JI Annotated Anodyne DRD3 70 46 C[C@H](NC(=O)c1cc2cccc(N3CCN(CCc4ccccn4)CC3)c2o1)c1ccccn1 ZINC000147474460 JI Annotated Anodyne HTR7 46 40 CN(Cc1ccccc1)C(=O)CC1(CN)CCC1 ZINC000147474475 BE For-Sale Anodyne CACNA2D1 33 43 CN(Cc1ccccc1)C(=O)CC1(CN)CCC1 ZINC000147474475 BE For-Sale Anodyne HCRTR1 0 43 CN(Cc1ccccc1)C(=O)CC1(CN)CCC1 ZINC000147474475 BE For-Sale Anodyne TSPO 16 40 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCC(=O)O ZINC000147474519 CE For-Sale Bother CACNA1D 60 35 CC1=C(/C=C/C(C)=C\C=C\C(C)=C/C(=O)OCC(=O)C(C)(C)C)C(C)(C)CCC1 ZINC000147474533 GK For-Sale Anodyne RARA 21 46 CC1=C(/C=C/C(C)=C\C=C\C(C)=C/C(=O)OCC(=O)C(C)(C)C)C(C)(C)CCC1 ZINC000147474533 GK For-Sale Anodyne RARG 22 51 CC1=C(/C=C/C(C)=C\C=C\C(C)=C/C(=O)OCC(=O)C(C)(C)C)C(C)(C)CCC1 ZINC000147474533 GK For-Sale Anodyne RXRG 18 45 CC1=C(/C=C/C(C)=C\C=C\C(C)=C/C(=O)OCC(=O)C(C)(C)C)C(C)(C)CCC1 ZINC000147474533 GK For-Sale Anodyne RARB 22 46 CC1=C(/C=C/C(C)=C\C=C\C(C)=C/C(=O)OCC(=O)C(C)(C)C)C(C)(C)CCC1 ZINC000147474533 GK For-Sale Anodyne RXRA 17 45 CC1=C(/C=C/C(C)=C\C=C\C(C)=C/C(=O)OCC(=O)C(C)(C)C)C(C)(C)CCC1 ZINC000147474533 GK For-Sale Anodyne RBP4 32 61 COc1cc(NS(=O)(=O)c2ccc(Br)s2)ccc1Br ZINC000147474543 II On-Demand Anodyne GHSR 0 48 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(CCC(=O)N3CCCC3)cc2)C1 ZINC000147474583 HE On-Demand Anodyne CCR3 34 40 COC(=O)CC[C@H](NC(=O)c1csc(Br)c1)C(=O)OC ZINC000147474605 FD On-Demand Anodyne CCKBR 41 33 C[C@@H]1CCCN(C(=O)Nc2cc(Br)cc(C(=O)O)c2)[C@@H]1C ZINC000147474651 FH For-Sale Anodyne TRPC6 48 35 Cc1ccc(C)c(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474672 HF On-Demand Anodyne EPHX2 36 45 Cc1ccc(C)c(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474672 HF On-Demand Anodyne TGM2 62 41 Cc1ccc(C)c(OCC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474672 HF On-Demand Anodyne F13A1 59 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2F)c1 ZINC000147474677 DH On-Demand Anodyne PPIA 15 48 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2F)c1 ZINC000147474677 DH On-Demand Anodyne ATF1 57 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2F)c1 ZINC000147474677 DH On-Demand Anodyne NR1H4 16 45 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2F)c1 ZINC000147474677 DH On-Demand Anodyne NFKB1 53 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2F)c1 ZINC000147474677 DH On-Demand Anodyne ACPS 0 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2F)c1 ZINC000147474677 DH On-Demand Anodyne AKR1C3 38 44 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2F)c1 ZINC000147474677 DH On-Demand Anodyne CYA 0 44 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2F)c1 ZINC000147474677 DH On-Demand Anodyne SMO 23 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2F)c1 ZINC000147474677 DH On-Demand Anodyne KCNK3 99 45 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2F)c1 ZINC000147474677 DH On-Demand Anodyne KCNK9 74 37 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(F)c2F)c1 ZINC000147474677 DH On-Demand Anodyne TMPRSS4 0 44 NCc1coc(COc2ccc(Cl)c(F)c2)c1 ZINC000147474706 CG For-Sale Anodyne DAO 17 47 Cc1ncc([N+](=O)[O-])n1CCN1CCC(=O)CC1 ZINC000147474715 CC For-Sale Bother TYMS 37 43 O=C(Nc1cccc(CN2CCOCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147474737 GH On-Demand Anodyne DRD2 16 42 O=C(Nc1cccc(CN2CCOCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147474737 GH On-Demand Anodyne DRD3 17 44 O=C(Nc1cccc(CN2CCOCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147474737 GH On-Demand Anodyne FAAH 22 40 O=C(Nc1cccc(CN2CCOCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147474737 GH On-Demand Anodyne MAPK10 23 42 O=C(Nc1cccc(CN2CCOCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147474737 GH On-Demand Anodyne MCHR1 20 41 O=C(Nc1cccc(CN2CCOCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147474737 GH On-Demand Anodyne AURKA 18 43 O=C(Nc1cccc(CN2CCOCC2)c1)c1cnn(-c2ccccc2Cl)c1 ZINC000147474737 GH On-Demand Anodyne KCNK3 41 37 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(CCC(=O)N3CCCC3)cc2)C1 ZINC000147474794 HE On-Demand Anodyne CCR3 34 40 C[C@H]1CCCN(C(=O)Nc2cc(Br)cc(C(=O)O)c2)[C@@H]1C ZINC000147474799 FH For-Sale Anodyne TRPC6 48 35 C=C(COCc1cccc(Br)c1)C(=O)O ZINC000147474857 CF For-Sale Mild HCAR2 17 50 CCCCO[C@@H](C)C(=O)Nc1ccc2oc(C(C)C)nc2c1 ZINC000147474879 DI On-Demand Anodyne IMDH_CRYPV 47 48 CCCNCc1coc(COc2ccc(Cl)c(F)c2)c1 ZINC000147474882 CI For-Sale Anodyne DAO 15 41 Nc1cc(S(=O)(=O)Nc2ccncc2Br)c(Cl)cc1F ZINC000147474899 GG For-Sale Anodyne SGK1 60 35 O=C(Cc1ccccc1F)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147474902 DG On-Demand Anodyne PTGER1 15 43 O=C(Cc1ccccc1F)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147474902 DG On-Demand Anodyne AKR1C3 25 42 COc1ccc(N(C(=O)Nc2c(C)cccc2C)c2cc(Nc3ccc(N4CCN(C)CC4)cc3)ncn2)c(OC)c1 ZINC000147474927 KK In-Stock Anodyne PDGFRB 43 38 COc1ccc(N(C(=O)Nc2c(C)cccc2C)c2cc(Nc3ccc(N4CCN(C)CC4)cc3)ncn2)c(OC)c1 ZINC000147474927 KK In-Stock Anodyne LCK 45 53 COc1ccc(N(C(=O)Nc2c(C)cccc2C)c2cc(Nc3ccc(N4CCN(C)CC4)cc3)ncn2)c(OC)c1 ZINC000147474927 KK In-Stock Anodyne FGFR1 17 51 COc1ccc(N(C(=O)Nc2c(C)cccc2C)c2cc(Nc3ccc(N4CCN(C)CC4)cc3)ncn2)c(OC)c1 ZINC000147474927 KK In-Stock Anodyne SRC 18 60 COc1ccc(N(C(=O)Nc2c(C)cccc2C)c2cc(Nc3ccc(N4CCN(C)CC4)cc3)ncn2)c(OC)c1 ZINC000147474927 KK In-Stock Anodyne KDR 19 60 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147474953 GF On-Demand Anodyne ACHE 15 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147474953 GF On-Demand Anodyne HRH2 26 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147474953 GF On-Demand Anodyne CASR 33 42 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147474953 GF On-Demand Anodyne ROCK2 37 44 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147474953 GF On-Demand Anodyne FAAH 21 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147474953 GF On-Demand Anodyne EPHX2 17 43 COc1ccc2c(c1)OC[C@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147474953 GF On-Demand Anodyne MCHR1 28 43 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne DRD4 42 33 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne HTR4 48 35 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne LPL 50 36 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne CCR3 61 44 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne EPHX2 43 42 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne TGM2 81 46 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne ST14 63 36 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne MCHR1 29 42 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne CACNA1I 74 45 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne F13A1 87 46 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne AKR1C3 66 41 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne NAMPT 47 39 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne KCNK3 96 37 CC(=O)Nc1cccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147474955 HE On-Demand Anodyne KCNK9 54 37 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147474994 FH For-Sale Anodyne TRPC6 48 35 CCCCO[C@H](C)C(=O)Nc1ccc2oc(C(C)C)nc2c1 ZINC000147475031 DI On-Demand Anodyne IMDH_CRYPV 47 48 CN1CCCC[C@@H]1C(=O)NO ZINC000147475106 AB On-Demand Mild MMP13 16 44 CN1CCCC[C@@H]1C(=O)NO ZINC000147475106 AB On-Demand Mild MMP7 21 44 CN1CCCC[C@@H]1C(=O)NO ZINC000147475106 AB On-Demand Mild MMP1 15 44 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475108 DF On-Demand Anodyne JUN 22 40 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475108 DF On-Demand Anodyne ATF1 55 38 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475108 DF On-Demand Anodyne CPT1A 72 40 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475108 DF On-Demand Anodyne CPT2 47 39 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475108 DF On-Demand Anodyne NFKB1 51 38 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475108 DF On-Demand Anodyne P4HTM 0 43 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475108 DF On-Demand Anodyne TAAR1 31 40 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475108 DF On-Demand Anodyne GPR35 22 46 COc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475108 DF On-Demand Anodyne KCNK3 44 38 C[C@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475109 DC On-Demand Bother CA2 66 39 C[C@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475109 DC On-Demand Bother CA1 56 40 C[C@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475109 DC On-Demand Bother BDKRB1 0 46 C[C@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475109 DC On-Demand Bother COLA 69 34 C[C@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475109 DC On-Demand Bother CA5B 41 39 C[C@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475109 DC On-Demand Bother CA4 73 41 C[C@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475109 DC On-Demand Bother CA5A 46 39 CCNCCC[C@@H](C)Oc1ccc(Cl)c(F)c1 ZINC000147475116 CH For-Sale Anodyne LEF 42 37 C[C@H]1CCCN(C(=O)Nc2cc(Br)cc(C(=O)O)c2)[C@H]1C ZINC000147475123 FH For-Sale Anodyne TRPC6 48 35 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147475148 GF On-Demand Anodyne ACHE 15 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147475148 GF On-Demand Anodyne HRH2 26 43 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147475148 GF On-Demand Anodyne CASR 33 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147475148 GF On-Demand Anodyne ROCK2 37 44 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147475148 GF On-Demand Anodyne FAAH 21 43 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147475148 GF On-Demand Anodyne EPHX2 17 43 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCOCC3)c1)C2 ZINC000147475148 GF On-Demand Anodyne MCHR1 28 43 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)S(=O)(=O)CC(=O)O ZINC000147475190 DD For-Sale Bother CACNA1D 55 35 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)S(=O)(=O)CC(=O)O ZINC000147475190 DD For-Sale Bother COLA 49 38 CCNCCC[C@H](C)Oc1ccc(Cl)c(F)c1 ZINC000147475266 CH For-Sale Anodyne LEF 42 37 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475269 DC On-Demand Bother CA2 66 39 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475269 DC On-Demand Bother CA1 56 40 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475269 DC On-Demand Bother BDKRB1 0 46 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475269 DC On-Demand Bother COLA 69 34 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475269 DC On-Demand Bother CA5B 41 39 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475269 DC On-Demand Bother CA4 73 41 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1[N+](=O)[O-])CC(=O)O ZINC000147475269 DC On-Demand Bother CA5A 46 39 C[C@@H](CCC(=O)O)OCc1cccc(Br)c1 ZINC000147475272 CG For-Sale Anodyne FFAR1 45 53 C[C@@H](CCC(=O)O)OCc1cccc(Br)c1 ZINC000147475272 CG For-Sale Anodyne FFAR4 26 53 Clc1ccc2[nH]cc(C[C@@H]3CCNC3)c2c1 ZINC000147475281 BF For-Sale Anodyne MPO 52 36 Clc1ccc2[nH]cc(C[C@@H]3CCNC3)c2c1 ZINC000147475281 BF For-Sale Anodyne HTR6 21 41 CN1CCCC[C@H]1C(=O)NO ZINC000147475294 AB On-Demand Mild MMP13 16 44 CN1CCCC[C@H]1C(=O)NO ZINC000147475294 AB On-Demand Mild MMP7 21 44 CN1CCCC[C@H]1C(=O)NO ZINC000147475294 AB On-Demand Mild MMP1 15 44 Nc1cc(F)c(F)c(S(=O)(=O)Nc2ccncc2Br)c1 ZINC000147475305 FF For-Sale Anodyne PTGS1 0 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475333 CF On-Demand Anodyne JUN 23 44 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475333 CF On-Demand Anodyne ATF1 57 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475333 CF On-Demand Anodyne CPT1A 41 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475333 CF On-Demand Anodyne PRNP 21 41 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475333 CF On-Demand Anodyne NFKB1 53 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475333 CF On-Demand Anodyne P4HTM 0 48 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475333 CF On-Demand Anodyne SCN10A 33 41 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475333 CF On-Demand Anodyne CSF1R 20 46 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475333 CF On-Demand Anodyne DDR1 40 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cn1 ZINC000147475333 CF On-Demand Anodyne KCNK3 60 39 C[C@@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)[C@@H]1C ZINC000147475335 DH On-Demand Anodyne CACNA1I 42 33 C[C@@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)[C@@H]1C ZINC000147475335 DH On-Demand Anodyne TRPC6 52 38 COc1cc(Cl)ccc1C(=O)N1CCC[C@@H]1CCCBr ZINC000147475336 FI For-Sale Reactive HTR4 48 36 COc1cc(Cl)ccc1C(=O)N1CCC[C@@H]1CCCBr ZINC000147475336 FI For-Sale Reactive ACKR3 61 31 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)S(=O)(=O)CC(=O)O ZINC000147475372 DD For-Sale Bother CACNA1D 55 35 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)S(=O)(=O)CC(=O)O ZINC000147475372 DD For-Sale Bother COLA 49 38 Clc1ccc2[nH]cc(C[C@H]3CCNC3)c2c1 ZINC000147475387 BF For-Sale Anodyne MPO 52 36 Clc1ccc2[nH]cc(C[C@H]3CCNC3)c2c1 ZINC000147475387 BF For-Sale Anodyne HTR6 21 41 CCCNCCCCCOc1ccc(Cl)c(F)c1 ZINC000147475419 CI For-Sale Anodyne DRD4 21 48 CCCNCCCCCOc1ccc(Cl)c(F)c1 ZINC000147475419 CI For-Sale Anodyne PLA2G4B 44 33 C[C@H](CCC(=O)O)OCc1cccc(Br)c1 ZINC000147475453 CG For-Sale Anodyne FFAR1 45 53 C[C@H](CCC(=O)O)OCc1cccc(Br)c1 ZINC000147475453 CG For-Sale Anodyne FFAR4 26 53 COc1cc(Cl)ccc1C(=O)N1CCC[C@H]1CCCBr ZINC000147475459 FI For-Sale Reactive HTR4 48 36 COc1cc(Cl)ccc1C(=O)N1CCC[C@H]1CCCBr ZINC000147475459 FI For-Sale Reactive ACKR3 61 31 C[C@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)[C@@H]1C ZINC000147475464 DH On-Demand Anodyne CACNA1I 42 33 C[C@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)[C@@H]1C ZINC000147475464 DH On-Demand Anodyne TRPC6 52 38 Cc1cc(S(=O)(=O)Nc2ccncc2Br)ccc1N ZINC000147475511 EF For-Sale Anodyne PTGS1 0 40 Cc1cc(S(=O)(=O)Nc2ccncc2Br)ccc1N ZINC000147475511 EF For-Sale Anodyne CA1 15 42 Cc1cc(S(=O)(=O)Nc2ccncc2Br)ccc1N ZINC000147475511 EF For-Sale Anodyne CA4 20 42 Cc1cc(S(=O)(=O)Nc2ccncc2Br)ccc1N ZINC000147475511 EF For-Sale Anodyne CAH_METTE 18 40 Cc1cc(S(=O)(=O)Nc2ccncc2Br)ccc1N ZINC000147475511 EF For-Sale Anodyne CYNT 20 40 CCCN(C)S(=O)(=O)NC(=O)c1ccccc1Cl ZINC000147475516 CD On-Demand Anodyne ECR 48 41 CCCN(C)S(=O)(=O)NC(=O)c1ccccc1Cl ZINC000147475516 CD On-Demand Anodyne E3UJZ5_SPOLI 43 41 Cc1cccc(CC(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147475544 DH On-Demand Anodyne PPIA 19 45 Cc1cccc(CC(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147475544 DH On-Demand Anodyne PTGER1 20 44 Cc1cccc(CC(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147475544 DH On-Demand Anodyne AKR1C3 38 46 Cc1cccc(CC(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147475544 DH On-Demand Anodyne PFK 0 43 Cc1cccc(CC(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147475544 DH On-Demand Anodyne KCNK3 63 44 Cc1cccc(CC(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147475544 DH On-Demand Anodyne KCNK9 44 44 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147475608 DH On-Demand Anodyne CACNA1I 42 33 C[C@H]1[C@H](C)CCCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147475608 DH On-Demand Anodyne TRPC6 52 38 CC(C)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147475666 IK Annotated Anodyne TP53 51 81 CC(C)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147475666 IK Annotated Anodyne MDM2 289 81 CCCNc1cccc(NCC2CCCCC2)n1 ZINC000147475693 BH For-Sale Anodyne GPR39 0 46 COc1cccc([C@@H](CC(C)(C)C)C(=O)O)c1 ZINC000147475708 BG For-Sale Anodyne MTNR1A 37 43 COc1cccc([C@@H](CC(C)(C)C)C(=O)O)c1 ZINC000147475708 BG For-Sale Anodyne MTNR1B 40 43 COc1cccc([C@@H](CC(C)(C)C)C(=O)O)c1 ZINC000147475708 BG For-Sale Anodyne ALS 59 33 COc1cccc([C@@H](CC(C)(C)C)C(=O)O)c1 ZINC000147475708 BG For-Sale Anodyne AKR1C3 21 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1=COCCO1 ZINC000147475709 FD On-Demand Anodyne HTR4 47 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1=COCCO1 ZINC000147475709 FD On-Demand Anodyne PKM 20 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1=COCCO1 ZINC000147475709 FD On-Demand Anodyne TGM2 64 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1=COCCO1 ZINC000147475709 FD On-Demand Anodyne CACNA1I 47 33 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)C1=COCCO1 ZINC000147475709 FD On-Demand Anodyne F13A1 67 43 C[C@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)[C@H]1C ZINC000147475757 DH On-Demand Anodyne CACNA1I 42 33 C[C@H]1CCCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)[C@H]1C ZINC000147475757 DH On-Demand Anodyne TRPC6 52 38 O=C(COc1cccc(Cl)c1)N1CCC[C@@H]1CCCBr ZINC000147475765 FH For-Sale Reactive COLA 135 48 O=C(COc1cccc(Cl)c1)N1CCC[C@@H]1CCCBr ZINC000147475765 FH For-Sale Reactive CPT1A 116 48 O=C(COc1cccc(Cl)c1)N1CCC[C@@H]1CCCBr ZINC000147475765 FH For-Sale Reactive CPT2 51 48 O=C(COc1cccc(Cl)c1)N1CCC[C@@H]1CCCBr ZINC000147475765 FH For-Sale Reactive CHRNA10 48 35 COCCn1cc(C(=O)[C@@H](C#N)c2nc3ccccc3[nH]2)c2ccccc21 ZINC000147475801 FH On-Demand Mild CNR1 24 47 COCCn1cc(C(=O)[C@@H](C#N)c2nc3ccccc3[nH]2)c2ccccc21 ZINC000147475801 FH On-Demand Mild CNR2 19 47 COC(=O)CC[C@@H](NC(=O)c1csc(Br)c1)C(=O)OC ZINC000147475808 FD On-Demand Anodyne CCKBR 41 33 O=C(NCc1ccc(F)cc1F)c1ccccc1Cl ZINC000147475827 CH On-Demand Anodyne P2RX7 106 46 O=C(NCc1ccc(F)cc1F)c1ccccc1Cl ZINC000147475827 CH On-Demand Anodyne ECR 51 44 O=C(NCc1ccc(F)cc1F)c1ccccc1Cl ZINC000147475827 CH On-Demand Anodyne EPHX2 15 44 O=C(NCc1ccc(F)cc1F)c1ccccc1Cl ZINC000147475827 CH On-Demand Anodyne SCN10A 31 41 O=C(NCc1ccc(F)cc1F)c1ccccc1Cl ZINC000147475827 CH On-Demand Anodyne E3UJZ5_SPOLI 38 40 O=C(NCc1ccc(F)cc1F)c1ccccc1Cl ZINC000147475827 CH On-Demand Anodyne KCNK3 15 56 COc1cccc([C@H](CC(C)(C)C)C(=O)O)c1 ZINC000147475868 BG For-Sale Anodyne MTNR1A 37 43 COc1cccc([C@H](CC(C)(C)C)C(=O)O)c1 ZINC000147475868 BG For-Sale Anodyne MTNR1B 40 43 COc1cccc([C@H](CC(C)(C)C)C(=O)O)c1 ZINC000147475868 BG For-Sale Anodyne ALS 59 33 COc1cccc([C@H](CC(C)(C)C)C(=O)O)c1 ZINC000147475868 BG For-Sale Anodyne AKR1C3 21 43 NCC1(CC(=O)N[C@@H]2CCS(=O)(=O)C2)CCC1 ZINC000147475879 CB For-Sale Anodyne CACNA2D1 20 43 O=C(COc1cccc(Cl)c1)N1CCC[C@H]1CCCBr ZINC000147475929 FH For-Sale Reactive COLA 135 48 O=C(COc1cccc(Cl)c1)N1CCC[C@H]1CCCBr ZINC000147475929 FH For-Sale Reactive CPT1A 116 48 O=C(COc1cccc(Cl)c1)N1CCC[C@H]1CCCBr ZINC000147475929 FH For-Sale Reactive CPT2 51 48 O=C(COc1cccc(Cl)c1)N1CCC[C@H]1CCCBr ZINC000147475929 FH For-Sale Reactive CHRNA10 48 35 COC(=O)COc1cc(C(F)(F)F)nn1-c1ccccc1Cl ZINC000147475981 EG For-Sale Anodyne CARM1 69 35 O=C(Cc1ccccc1[N+](=O)[O-])NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476002 HE On-Demand Bother COLA 110 40 O=C(Cc1ccccc1[N+](=O)[O-])NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476002 HE On-Demand Bother EPHX2 18 43 O=C(Cc1ccccc1[N+](=O)[O-])NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476002 HE On-Demand Bother TGM2 74 45 O=C(Cc1ccccc1[N+](=O)[O-])NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476002 HE On-Demand Bother F13A1 80 45 O=C(Cc1ccccc1[N+](=O)[O-])NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476002 HE On-Demand Bother NAMPT 54 40 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCCl ZINC000147476026 CG For-Sale Reactive CACNA1D 58 35 NCC1(CC(=O)N[C@H]2CCS(=O)(=O)C2)CCC1 ZINC000147476045 CB For-Sale Anodyne CACNA2D1 20 43 COCCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147476092 CE On-Demand Anodyne CACNA1I 46 34 O=C(O)CCCCOCc1ccc(Br)cc1 ZINC000147476127 CG For-Sale Anodyne PLA2G4B 26 40 O=C(O)CCCCOCc1ccc(Br)cc1 ZINC000147476127 CG For-Sale Anodyne GBA2 46 35 O=C(O)CCCCOCc1ccc(Br)cc1 ZINC000147476127 CG For-Sale Anodyne FFAR1 15 53 C[C@H]1CCC[C@@H](C)N1NC(=O)CNC(=O)CN ZINC000147476168 BB For-Sale Anodyne UREB 0 43 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCCl ZINC000147476191 CG For-Sale Reactive CACNA1D 58 35 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne F2 30 42 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne DRD2 28 46 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne FKBP1A 36 43 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne DRD4 46 37 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne ACHE 24 45 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne DRD3 26 43 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne HTR4 45 36 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne F10 18 41 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne CHRM5 22 43 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne CHRM3 17 40 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne GRIN2B 47 39 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne SIGMAR1 34 54 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne MMP13 95 44 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne CCR3 42 47 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne HTR6 22 40 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne ADAM17 41 42 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne MTNR1A 65 40 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne MTNR1B 65 40 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne MMP2 43 44 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne MMP3 76 44 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne MMP8 41 44 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne NPY5R 16 41 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne CAPN1 18 42 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne MMP9 59 44 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne EPHX2 25 42 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne PKM 15 42 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne MMP12 26 41 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne TGM2 76 46 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne ST14 43 37 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne MMP7 61 44 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne MMP1 72 44 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne MCHR1 23 40 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne CACNA1I 59 39 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne F13A1 78 46 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne CCR8 24 43 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne AKR1C3 45 42 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne NCE103 16 44 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne NAMPT 48 39 COc1cccc(CC(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147476229 HE On-Demand Anodyne TMPRSS6 47 35 O[C@H](c1cncs1)[C@@H]1CCCc2cccnc21 ZINC000147476262 BF For-Sale Anodyne CXCR4 54 34 CC(C)[C@H](OCc1ccc(Br)cc1)C(=O)O ZINC000147476318 CG For-Sale Anodyne SLC1A6 0 49 CC(C)[C@H](OCc1ccc(Br)cc1)C(=O)O ZINC000147476318 CG For-Sale Anodyne SLC1A7 0 49 O=C(CC[C@@H]1CCCO1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147476327 CF On-Demand Anodyne LDLR 0 40 CN(C)C1(CNC(=O)c2ccccc2NN)CCCC1 ZINC000147476353 CD For-Sale Anodyne KCNA3 42 44 CN(C)C1(CNC(=O)c2ccccc2NN)CCCC1 ZINC000147476353 CD For-Sale Anodyne SLC6A5 16 47 CN(C)C1(CNC(=O)c2ccccc2NN)CCCC1 ZINC000147476353 CD For-Sale Anodyne HCN1 84 41 CN(C)C1(CNC(=O)c2ccccc2NN)CCCC1 ZINC000147476353 CD For-Sale Anodyne HCN4 59 39 C[C@H]1CCC[C@H](C)N1NC(=O)CNC(=O)CN ZINC000147476354 BB For-Sale Anodyne UREB 0 43 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CBr ZINC000147476364 DF For-Sale Reactive CACNA1C 46 39 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CBr ZINC000147476364 DF For-Sale Reactive CACNA1D 75 35 Nc1ccc(F)c(S(=O)(=O)Nc2ccncc2Br)c1 ZINC000147476385 EE For-Sale Anodyne PTGS1 0 45 Nc1ccc(F)c(S(=O)(=O)Nc2ccncc2Br)c1 ZINC000147476385 EE For-Sale Anodyne SGK1 40 39 O[C@H](c1cncs1)[C@H]1CCCc2cccnc21 ZINC000147476406 BF For-Sale Anodyne CXCR4 54 34 COc1ccc(N2CCN(C(=O)C3(N)CCC3)CC2)cc1 ZINC000147476452 CD On-Demand Clean MMP13 15 44 COc1ccc(N2CCN(C(=O)C3(N)CCC3)CC2)cc1 ZINC000147476452 CD On-Demand Clean NPBWR1 52 30 CNC(=O)c1cc(NC[C@@H](C)CC(=O)O)ccn1 ZINC000147476494 CC For-Sale Anodyne RAF1 48 35 CNC(=O)c1cc(NC[C@@H](C)CC(=O)O)ccn1 ZINC000147476494 CC For-Sale Anodyne Q8MMZ8_EIMTE 53 37 O=C(CC[C@H]1CCCO1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147476511 CF On-Demand Anodyne LDLR 0 40 C[C@@H]1CCC[C@@H](C)N1NC(=O)CNC(=O)CN ZINC000147476514 BB For-Sale Anodyne UREB 0 43 CC(C)[C@@H](OCc1ccc(Br)cc1)C(=O)O ZINC000147476534 CG For-Sale Anodyne SLC1A6 0 49 CC(C)[C@@H](OCc1ccc(Br)cc1)C(=O)O ZINC000147476534 CG For-Sale Anodyne SLC1A7 0 49 Cc1ccsc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476543 GF On-Demand Anodyne HTR4 49 37 Cc1ccsc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476543 GF On-Demand Anodyne EPHX2 31 43 Cc1ccsc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476543 GF On-Demand Anodyne TGM2 74 46 Cc1ccsc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476543 GF On-Demand Anodyne CACNA1I 58 35 Cc1ccsc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476543 GF On-Demand Anodyne F13A1 75 46 O[C@@H](c1cncs1)[C@@H]1CCCc2cccnc21 ZINC000147476551 BF For-Sale Anodyne CXCR4 54 34 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CBr ZINC000147476553 DF For-Sale Reactive CACNA1C 46 39 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CBr ZINC000147476553 DF For-Sale Reactive CACNA1D 75 35 Nc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1Br ZINC000147476606 HF For-Sale Anodyne CA2 15 50 Nc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1Br ZINC000147476606 HF For-Sale Anodyne CA4 15 50 Nc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1Br ZINC000147476606 HF For-Sale Anodyne CAH_METTE 20 50 Nc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1Br ZINC000147476606 HF For-Sale Anodyne CYNT 16 50 Nc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1Br ZINC000147476606 HF For-Sale Anodyne CA15 18 50 Nc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1Br ZINC000147476606 HF For-Sale Anodyne CA 0 50 Nc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1Br ZINC000147476606 HF For-Sale Anodyne Q5TU56_ANOGA 0 50 CCCc1c(NCC)ncnc1Oc1ccc(Br)cc1F ZINC000147476616 FJ For-Sale Anodyne HTT 0 40 COC(=O)Cc1csc(-c2ccccc2[N+](=O)[O-])n1 ZINC000147476640 CE For-Sale Bother COLA 75 35 CNC(=O)c1cc(NC[C@H](C)CC(=O)O)ccn1 ZINC000147476657 CC For-Sale Anodyne RAF1 48 35 CNC(=O)c1cc(NC[C@H](C)CC(=O)O)ccn1 ZINC000147476657 CC For-Sale Anodyne Q8MMZ8_EIMTE 53 37 O[C@@H](c1cncs1)[C@H]1CCCc2cccnc21 ZINC000147476713 BF For-Sale Anodyne CXCR4 54 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne CACNA1H 15 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne DRD2 24 48 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne DRD4 45 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne ACHE 15 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne DRD3 30 48 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne HTR4 54 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne F10 28 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne CNR2 15 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne CCR3 33 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne HTR6 16 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne APP 43 35 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne CPT1A 46 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne PPARD 15 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne SLC6A9 48 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne CCR2 37 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne EPHX2 35 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne TGM2 68 49 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne ST14 44 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne CXCR3 23 48 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne MCHR1 18 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne CACNA1I 96 60 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne F13A1 64 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne AKR1C3 63 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne SFRP1 27 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne AKR1C1 23 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(Cl)c1 ZINC000147476756 GG On-Demand Anodyne NAMPT 42 40 C=CC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147476785 BE For-Sale Bother CACNA1C 45 37 C=CC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147476785 BE For-Sale Bother CACNA1D 72 37 C=CC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147476785 BE For-Sale Bother APR 0 40 C[C@H](CNc1cc(Br)ccc1[N+](=O)[O-])CC(=O)O ZINC000147476826 DF For-Sale Bother COLA 67 34 Cc1cc(F)c(S(=O)(=O)Nc2ccncc2Br)cc1N ZINC000147476830 FF For-Sale Anodyne PTGS1 0 43 CC(C)[C@@H](C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147476874 CG On-Demand Anodyne HCAR1 0 44 Cc1noc(C)c1CNS(=O)(=O)c1ccc(I)cc1 ZINC000147476904 GE On-Demand Anodyne EDNRA 23 41 Cc1cc(NN)c(C(=O)NCC2(N(C)C)CCCC2)cn1 ZINC000147476911 CD For-Sale Anodyne SLC6A5 15 43 CCOCCn1c(COc2cccc(CO)c2)nc2ccccc21 ZINC000147476912 EG For-Sale Anodyne HRH1 18 45 CCOCCn1c(COc2cccc(CO)c2)nc2ccccc21 ZINC000147476912 EG For-Sale Anodyne NPY1R 41 34 O=C(CSc1ccncc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476924 HE On-Demand Anodyne GRIN2B 30 41 O=C(CSc1ccncc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476924 HE On-Demand Anodyne EPHX2 15 42 O=C(CSc1ccncc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476924 HE On-Demand Anodyne TGM2 79 46 O=C(CSc1ccncc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476924 HE On-Demand Anodyne F13A1 86 46 O=C(CSc1ccncc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147476924 HE On-Demand Anodyne NAMPT 56 39 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cc(F)ccc2Br)c1 ZINC000147476971 GG On-Demand Bother TAAR1 23 44 C=CC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147476989 BE For-Sale Bother CACNA1C 45 37 C=CC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147476989 BE For-Sale Bother CACNA1D 72 37 C=CC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147476989 BE For-Sale Bother APR 0 40 C[C@@H](CNc1cc(Br)ccc1[N+](=O)[O-])CC(=O)O ZINC000147477008 DF For-Sale Bother COLA 67 34 CCCCCNC(=O)[C@H](C)N1CC[C@H](N)[C@H](CC)C1 ZINC000147477010 CD On-Demand Anodyne TPP2 30 40 CC(C)[C@H](C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147477043 CG On-Demand Anodyne HCAR1 0 44 CNc1cn2ccnc2c(Oc2ccc(Br)cc2F)n1 ZINC000147477068 EG For-Sale Anodyne HIVRT 0 45 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCCC[C@@H]3C)cc2)C1 ZINC000147477080 HE On-Demand Anodyne CACNA1I 40 32 COC(=O)Cc1csc(Cc2ccc(F)cc2Cl)n1 ZINC000147477094 CG For-Sale Anodyne P2RX7 53 39 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne RARA 24 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne PPIA 15 49 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne ATF1 40 38 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne CPT1A 50 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne PYGL 18 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne CXCR2 0 47 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne PRNP 33 49 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne NR1H4 23 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne TAAR1 34 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne AKR1C3 33 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne PTPA 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne SHH 23 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne HCAR1 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2)c1 ZINC000147477210 CG On-Demand Anodyne KCNK3 74 55 C[C@H](CNc1ccc(C(F)(F)F)cc1[N+](=O)[O-])CC(=O)O ZINC000147477214 DG On-Demand Bother AKR1C4 0 50 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](C)Cl ZINC000147477246 CF For-Sale Reactive CACNA1D 51 34 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCCC[C@@H]3C)cc2)C1 ZINC000147477259 HE On-Demand Anodyne CACNA1I 40 32 C[C@H](NC(=O)c1cn(-c2ccccc2)nc1-c1ccc(-c2ccccc2)cc1)C(N)=O ZINC000147477261 HH On-Demand Anodyne CDK2 21 56 NC1(C(=O)N2CCN(c3ccc(F)cc3)CC2)CCC1 ZINC000147477264 CD On-Demand Anodyne AKR1C3 0 52 C[C@@H](Cl)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147477360 CF For-Sale Reactive CACNA1D 51 34 C[C@@H](CNc1ccc(C(F)(F)F)cc1[N+](=O)[O-])CC(=O)O ZINC000147477363 DG On-Demand Bother AKR1C4 0 50 O=C(/C=C/c1ccco1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147477426 FF On-Demand Anodyne TGM2 72 46 O=C(/C=C/c1ccco1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147477426 FF On-Demand Anodyne F13A1 92 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne PPIA 19 47 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne ECR 32 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne ATF1 47 39 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne PRNP 21 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne NR1H4 15 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne F12 0 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne NFKB1 44 39 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne ACPS 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne AKR1C3 38 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne NR2E3 44 34 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne CYA 0 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne AKR1C2 32 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne SMO 27 47 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne HCAR1 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne KCNK3 92 47 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne KCNK9 69 36 O=C(O)c1cc(Cl)cc(NC(=O)c2ccccc2Br)c1 ZINC000147477438 FI On-Demand Anodyne TMPRSS4 0 40 CS(=O)(=O)c1cc(C(=O)Nc2ccccc2CN2CCOCC2)cc([N+](=O)[O-])c1 ZINC000147477440 HE On-Demand Bother BCL2L1 45 34 CS(=O)(=O)c1cc(C(=O)Nc2ccccc2CN2CCOCC2)cc([N+](=O)[O-])c1 ZINC000147477440 HE On-Demand Bother BCL2 40 36 C[C@H](Cl)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147477463 CF For-Sale Reactive CACNA1D 51 34 C[C@@H](NC(=O)c1cn(-c2ccccc2)nc1-c1ccc(-c2ccccc2)cc1)C(N)=O ZINC000147477464 HH On-Demand Anodyne CDK2 21 56 C[C@@H]1Cc2ccccc2N1C(=O)C1(N)CCC1 ZINC000147477531 BD For-Sale Anodyne DRD4 32 51 Cc1noc(C)c1CNS(=O)(=O)c1ccc(S(=O)(=O)N2CCCCC2)cc1 ZINC000147477563 HD On-Demand Anodyne NAMPT 25 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccccc2N2C[C@H](C)O[C@H](C)C2)C1 ZINC000147477567 HE On-Demand Anodyne HTR4 44 36 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccccc2N2C[C@H](C)O[C@H](C)C2)C1 ZINC000147477567 HE On-Demand Anodyne KCNQ2 71 39 Cc1ccc(C(=O)NCC2(N(C)C)CCCC2)c(NN)c1 ZINC000147477572 CD For-Sale Anodyne SLC6A5 15 42 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@](C)(N)c1ccccc1 ZINC000147477584 CE For-Sale Anodyne AMY2 47 32 COc1ccc(S(=O)(=O)Nc2ccncc2Br)c(N)c1 ZINC000147477585 FE For-Sale Anodyne NFKBIA 0 46 CCCNc1cc(Oc2ccc(Br)cc2F)nc(N)n1 ZINC000147477594 EH For-Sale Anodyne AGPAT2 59 44 C[C@H](Cl)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147477627 CF For-Sale Reactive CACNA1D 51 34 O=C(Cc1cccs1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147477631 CG On-Demand Anodyne CA5B 45 50 O=C(Cc1cccs1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147477631 CG On-Demand Anodyne CA5A 47 50 C[C@H]1Cc2ccccc2N1C(=O)C1(N)CCC1 ZINC000147477650 BD For-Sale Anodyne DRD4 32 51 C[C@H](NC(=O)c1cn(-c2ccccc2)nc1-c1ccc(Br)cc1)C(N)=O ZINC000147477671 HF On-Demand Anodyne CDK2 20 52 C[C@@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)[C@H](C)C1 ZINC000147477677 DH For-Sale Anodyne CACNA1I 46 34 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccccc2N2C[C@H](C)O[C@H](C)C2)C1 ZINC000147477705 HE On-Demand Anodyne HTR4 44 36 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccccc2N2C[C@H](C)O[C@H](C)C2)C1 ZINC000147477705 HE On-Demand Anodyne KCNQ2 71 39 CCS(=O)(=O)Nc1ccc(NC(=O)c2cc(F)ccc2NS(C)(=O)=O)cc1 ZINC000147477742 HE On-Demand Anodyne PLA2G7 32 44 CCS(=O)(=O)Nc1ccc(NC(=O)c2cc(F)ccc2NS(C)(=O)=O)cc1 ZINC000147477742 HE On-Demand Anodyne TRPV1 24 40 CCS(=O)(=O)Nc1ccc(NC(=O)c2cc(F)ccc2NS(C)(=O)=O)cc1 ZINC000147477742 HE On-Demand Anodyne Q25615_ONCVO 44 40 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne CA2 17 40 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne CHRM2 33 54 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne DRD2 37 47 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne FKBP1A 18 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne DRD4 44 35 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne ACHE 19 55 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne DRD3 39 41 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne HTR4 57 37 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne F10 33 46 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne CHRM5 22 51 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne GRIN2B 37 46 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne SIGMAR1 22 48 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne MMP13 109 50 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne ADAM17 69 40 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne PLD1 23 42 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne MMP2 59 50 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne MMP3 91 50 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne MMP8 50 50 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne MMP9 81 50 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne EPHX2 29 50 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne MMP12 40 39 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne TGM2 72 55 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne ITGAV 40 36 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne MMP7 68 50 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne MMP1 100 50 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne MCHR1 27 42 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne CACNA1I 67 41 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne F13A1 64 45 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne AKR1C3 48 42 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147477778 GF On-Demand Anodyne NAMPT 47 43 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCl ZINC000147477819 CF For-Sale Reactive CACNA1C 43 38 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCl ZINC000147477819 CF For-Sale Reactive CACNA1D 65 36 O=C(Nc1ccc(C(=O)NO)cc1)OC[C@@H]1CCc2ccccc2C1 ZINC000147477838 EG For-Sale Mild HDAC8 17 42 O=C(Nc1ccc(C(=O)NO)cc1)OC[C@@H]1CCc2ccccc2C1 ZINC000147477838 EG For-Sale Mild CFTR 50 33 O=C(Nc1ccc(C(=O)NO)cc1)OC[C@@H]1CCc2ccccc2C1 ZINC000147477838 EG For-Sale Mild NOD2 44 37 C[C@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)[C@H](C)C1 ZINC000147477846 DH For-Sale Anodyne CACNA1I 46 34 C[C@@H]1Cc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147477848 CE For-Sale Anodyne ACE 16 40 C[C@@H]1Cc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147477848 CE For-Sale Anodyne DRD4 31 50 C[C@@H]1Cc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147477848 CE For-Sale Anodyne TPP2 71 40 O=C(O)c1cc(Cl)cc(NC(=O)C2CCCC2)c1 ZINC000147477891 CG On-Demand Anodyne INHA 23 49 O=C(O)c1cc(Cl)cc(NC(=O)C2CCCC2)c1 ZINC000147477891 CG On-Demand Anodyne CACNA1I 45 36 O=C(O)c1cc(Cl)cc(NC(=O)C2CCCC2)c1 ZINC000147477891 CG On-Demand Anodyne RHOA 0 42 O=C(O)c1cc(Cl)cc(NC(=O)C2CCCC2)c1 ZINC000147477891 CG On-Demand Anodyne HCAR1 0 42 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@](C)(N)c1ccccc1 ZINC000147477907 CE For-Sale Anodyne AMY2 47 32 CCS(=O)(=O)Nc1ccc(NC(=O)c2cc(C)ccc2NS(C)(=O)=O)cc1 ZINC000147477931 HE On-Demand Anodyne PLA2G7 17 43 CCS(=O)(=O)Nc1ccc(NC(=O)c2cc(C)ccc2NS(C)(=O)=O)cc1 ZINC000147477931 HE On-Demand Anodyne Q25615_ONCVO 44 39 CCS(=O)(=O)Nc1ccc(NC(=O)c2cc(C)ccc2NS(C)(=O)=O)cc1 ZINC000147477931 HE On-Demand Anodyne KCNK3 45 32 CCS(=O)(=O)Nc1ccc(NC(=O)c2cc(C)ccc2NS(C)(=O)=O)cc1 ZINC000147477931 HE On-Demand Anodyne KCNK9 43 32 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147477951 HG On-Demand Anodyne HTR1A 16 41 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147477951 HG On-Demand Anodyne HRH2 64 39 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147477951 HG On-Demand Anodyne HTR1D 33 41 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147477951 HG On-Demand Anodyne HTR1B 27 41 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147477951 HG On-Demand Anodyne HTR4 55 39 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147477951 HG On-Demand Anodyne LTA4H 22 44 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147477951 HG On-Demand Anodyne CCR3 99 47 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147477951 HG On-Demand Anodyne EPHX2 23 42 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147477951 HG On-Demand Anodyne CACNA1I 49 33 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147477951 HG On-Demand Anodyne PDS 47 33 CC[C@@H](OCc1ccc(Br)cc1)C(=O)O ZINC000147477963 CF For-Sale Anodyne PPARG 16 44 CC[C@@H](OCc1ccc(Br)cc1)C(=O)O ZINC000147477963 CF For-Sale Anodyne PPARA 20 44 CC[C@@H](OCc1ccc(Br)cc1)C(=O)O ZINC000147477963 CF For-Sale Anodyne CPA1 15 43 Cc1ccccc1OC[C@H](O)CNCCCCC(C)C ZINC000147477966 CG For-Sale Anodyne ADRB2 54 71 Cc1ccccc1OC[C@H](O)CNCCCCC(C)C ZINC000147477966 CG For-Sale Anodyne ADRB1 66 43 Cc1ccccc1OC[C@H](O)CNCCCCC(C)C ZINC000147477966 CG For-Sale Anodyne ADRB3 44 42 Cc1ccccc1OC[C@H](O)CNCCCCC(C)C ZINC000147477966 CG For-Sale Anodyne CYP2D26 0 43 Cc1ccccc1OC[C@H](O)CNCCCCC(C)C ZINC000147477966 CG For-Sale Anodyne CYP2D6 16 44 Cc1ccccc1OC[C@H](O)CNCCCCC(C)C ZINC000147477966 CG For-Sale Anodyne ABCB1 38 46 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCl ZINC000147478029 CF For-Sale Reactive CACNA1C 43 38 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCl ZINC000147478029 CF For-Sale Reactive CACNA1D 65 36 O=C(Nc1ccc(C(=O)NO)cc1)OC[C@H]1CCc2ccccc2C1 ZINC000147478079 EG For-Sale Mild HDAC8 17 42 O=C(Nc1ccc(C(=O)NO)cc1)OC[C@H]1CCc2ccccc2C1 ZINC000147478079 EG For-Sale Mild CFTR 50 33 O=C(Nc1ccc(C(=O)NO)cc1)OC[C@H]1CCc2ccccc2C1 ZINC000147478079 EG For-Sale Mild NOD2 44 37 C[C@H]1Cc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147478082 CE For-Sale Anodyne ACE 16 40 C[C@H]1Cc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147478082 CE For-Sale Anodyne DRD4 31 50 C[C@H]1Cc2ccccc2N1C(=O)CC1(CN)CCC1 ZINC000147478082 CE For-Sale Anodyne TPP2 71 40 C[C@H]1C[C@H](C)CCN1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478083 DH For-Sale Anodyne CACNA1I 46 34 Cc1ccccc1OC[C@@H](O)CNCCCCC(C)C ZINC000147478113 CG For-Sale Anodyne ADRB2 54 71 Cc1ccccc1OC[C@@H](O)CNCCCCC(C)C ZINC000147478113 CG For-Sale Anodyne ADRB1 66 43 Cc1ccccc1OC[C@@H](O)CNCCCCC(C)C ZINC000147478113 CG For-Sale Anodyne ADRB3 44 42 Cc1ccccc1OC[C@@H](O)CNCCCCC(C)C ZINC000147478113 CG For-Sale Anodyne CYP2D26 0 43 Cc1ccccc1OC[C@@H](O)CNCCCCC(C)C ZINC000147478113 CG For-Sale Anodyne CYP2D6 16 44 Cc1ccccc1OC[C@@H](O)CNCCCCC(C)C ZINC000147478113 CG For-Sale Anodyne ABCB1 38 46 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147478126 HG On-Demand Anodyne HTR1A 16 41 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147478126 HG On-Demand Anodyne HRH2 64 39 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147478126 HG On-Demand Anodyne HTR1D 33 41 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147478126 HG On-Demand Anodyne HTR1B 27 41 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147478126 HG On-Demand Anodyne HTR4 55 39 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147478126 HG On-Demand Anodyne LTA4H 22 44 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147478126 HG On-Demand Anodyne CCR3 99 47 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147478126 HG On-Demand Anodyne EPHX2 23 42 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147478126 HG On-Demand Anodyne CACNA1I 49 33 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCCc3ccccc3)c2)C1 ZINC000147478126 HG On-Demand Anodyne PDS 47 33 CCS(=O)(=O)Nc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147478133 GD On-Demand Anodyne CA2 23 46 CCS(=O)(=O)Nc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147478133 GD On-Demand Anodyne PRSS1 15 43 CCS(=O)(=O)Nc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147478133 GD On-Demand Anodyne ADORA2B 45 48 CCS(=O)(=O)Nc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147478133 GD On-Demand Anodyne CA1 46 38 CCS(=O)(=O)Nc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147478133 GD On-Demand Anodyne ACR 70 42 CCS(=O)(=O)Nc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147478133 GD On-Demand Anodyne CA12 27 46 CCS(=O)(=O)Nc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147478133 GD On-Demand Anodyne CA9 28 46 CCS(=O)(=O)Nc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147478133 GD On-Demand Anodyne HIF1A 21 41 CCS(=O)(=O)Nc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147478133 GD On-Demand Anodyne NCE103 34 46 CCS(=O)(=O)Nc1ccc(NC(=O)COc2ccc(C(N)=O)cc2)cc1 ZINC000147478133 GD On-Demand Anodyne P96878_MYCTU 20 41 O=C(Cc1ccc(F)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478178 DG On-Demand Anodyne KCNQ2 17 40 O=C(Cc1ccc(F)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478178 DG On-Demand Anodyne PFK 0 41 O=C(Cc1ccc(F)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478178 DG On-Demand Anodyne RORC 45 38 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478203 DC On-Demand Anodyne TIMP3 40 30 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478203 DC On-Demand Anodyne MMP2 17 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478203 DC On-Demand Anodyne MMP3 32 43 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478203 DC On-Demand Anodyne GRIA1 40 32 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478203 DC On-Demand Anodyne PCSK5 53 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478203 DC On-Demand Anodyne FURIN 58 38 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478203 DC On-Demand Anodyne S1PR5 16 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478203 DC On-Demand Anodyne POLG_WNV 44 33 CN(C)C1(CNC(=O)c2nc(NN)ccc2Cl)CCCC1 ZINC000147478206 DD For-Sale Anodyne P2RX7 21 40 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCCCl ZINC000147478259 CH For-Sale Reactive CACNA1D 50 34 O=C(O)c1ccc(C(F)=C(F)F)cc1 ZINC000147478270 BF For-Sale Anodyne SRD5A2 42 48 O=C(O)c1ccc(C(F)=C(F)F)cc1 ZINC000147478270 BF For-Sale Anodyne SLC7A11 0 41 CC(=O)NC(=O)C(=O)c1ccccc1 ZINC000147478272 AC For-Sale Anodyne EPHX1 0 45 C[C@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)[C@@H](C)C1 ZINC000147478277 DH For-Sale Anodyne CACNA1I 46 34 NC1(C(=O)N2CCN(c3ncccn3)CC2)CCC1 ZINC000147478291 CC On-Demand Anodyne SLC6A7 0 47 COC1=CC=C2[C@H]3Cc4ccc(O)c5c4[C@]2(CCN3C)[C@@H]1O5 ZINC000147478326 CE Annotated Anodyne OPRM1 82 44 COC1=CC=C2[C@H]3Cc4ccc(O)c5c4[C@]2(CCN3C)[C@@H]1O5 ZINC000147478326 CE Annotated Anodyne OPRD1 78 44 COC1=CC=C2[C@H]3Cc4ccc(O)c5c4[C@]2(CCN3C)[C@@H]1O5 ZINC000147478326 CE Annotated Anodyne OPRK1 78 44 NC(=O)NCCCCC(=O)Nc1ccc(Cl)c(C(=O)NC2CC2)c1 ZINC000147478373 FE On-Demand Anodyne PLAU 16 40 NC(=O)NCCCCC(=O)Nc1ccc(Cl)c(C(=O)NC2CC2)c1 ZINC000147478373 FE On-Demand Anodyne ST14 18 40 NC(=O)NCCCCC(=O)Nc1ccc(Cl)c(C(=O)NC2CC2)c1 ZINC000147478373 FE On-Demand Anodyne ENV 40 30 NC(=O)n1nc(-c2ccco2)cc1N ZINC000147478386 AC For-Sale Anodyne ADORA1 33 42 NC(=O)n1nc(-c2ccco2)cc1N ZINC000147478386 AC For-Sale Anodyne ADORA2A 49 40 NC(=O)n1nc(-c2ccco2)cc1N ZINC000147478386 AC For-Sale Anodyne ADORA2B 25 42 NC(=O)n1nc(-c2ccco2)cc1N ZINC000147478386 AC For-Sale Anodyne ADORA3 22 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478403 DC On-Demand Anodyne TIMP3 40 30 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478403 DC On-Demand Anodyne MMP2 17 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478403 DC On-Demand Anodyne MMP3 32 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478403 DC On-Demand Anodyne GRIA1 40 32 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478403 DC On-Demand Anodyne PCSK5 53 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478403 DC On-Demand Anodyne FURIN 58 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478403 DC On-Demand Anodyne S1PR5 16 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(CC(N)=O)cc1 ZINC000147478403 DC On-Demand Anodyne POLG_WNV 44 33 O=C(CCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478406 DH On-Demand Anodyne GRIN1 19 49 O=C(CCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478406 DH On-Demand Anodyne PPIA 23 42 O=C(CCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478406 DH On-Demand Anodyne PTGER1 21 50 O=C(CCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478406 DH On-Demand Anodyne PAM 0 41 O=C(CCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478406 DH On-Demand Anodyne HCAR2 37 43 O=C(CCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478406 DH On-Demand Anodyne VIPR1 23 42 O=C(CCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478406 DH On-Demand Anodyne AKR1C3 31 42 O=C(CCc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478406 DH On-Demand Anodyne PARP10 0 40 Cc1c(N)cccc1S(=O)(=O)Nc1ccncc1Br ZINC000147478419 EF For-Sale Anodyne NFKBIA 0 43 O=C(O)/C=C/COCc1ccc(Br)cc1 ZINC000147478420 CF For-Sale Anodyne HCAR2 22 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc([N+](=O)[O-])o1 ZINC000147478423 GE On-Demand Bother HTR4 45 35 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc([N+](=O)[O-])o1 ZINC000147478423 GE On-Demand Bother EPHX2 15 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc([N+](=O)[O-])o1 ZINC000147478423 GE On-Demand Bother TGM2 68 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc([N+](=O)[O-])o1 ZINC000147478423 GE On-Demand Bother GSR 40 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc([N+](=O)[O-])o1 ZINC000147478423 GE On-Demand Bother CACNA1I 42 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc([N+](=O)[O-])o1 ZINC000147478423 GE On-Demand Bother F13A1 67 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc([N+](=O)[O-])o1 ZINC000147478423 GE On-Demand Bother NAMPT 80 42 Cc1ccc(Br)c(C(=O)NCC(C)(C)c2ccccc2)c1 ZINC000147478446 EI On-Demand Anodyne ECR 46 38 NCC1(CC(=O)N2CCN(c3ncccn3)CC2)CCC1 ZINC000147478478 CC For-Sale Anodyne SLC6A7 0 42 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCCCl ZINC000147478485 CH For-Sale Reactive CACNA1D 50 34 CCc1ccc(OC)cc1F ZINC000147478528 AE For-Sale Anodyne MTR1B_CHICK 62 32 CCc1ccc(OC)cc1F ZINC000147478528 AE For-Sale Anodyne CYP27A1 49 38 NC(=O)n1nc(-c2ccc(F)cc2)cc1N ZINC000147478591 BD For-Sale Anodyne SCN4A 51 47 O=C(Cc1ccccc1Cl)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478606 DH On-Demand Anodyne GRIN1 31 40 O=C(Cc1ccccc1Cl)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478606 DH On-Demand Anodyne PPIA 18 43 O=C(Cc1ccccc1Cl)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478606 DH On-Demand Anodyne CXCL8 34 40 O=C(Cc1ccccc1Cl)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478606 DH On-Demand Anodyne KCNQ2 28 47 O=C(Cc1ccccc1Cl)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478606 DH On-Demand Anodyne AKR1C3 28 42 O=C(Cc1ccccc1Cl)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147478606 DH On-Demand Anodyne PFK 0 41 O[C@@H](Cc1cccc(C(F)(F)F)c1)c1cncs1 ZINC000147478608 CG For-Sale Anodyne PHES 0 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother DRD4 41 33 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother HTR4 42 35 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother CACNA1C 42 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother CACNA1D 55 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother CCR2 20 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother EPHX2 18 52 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother TGM2 71 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother CACNA1I 63 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother F13A1 70 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother AKR1C3 72 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother SFRP1 24 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc([N+](=O)[O-])c1 ZINC000147478629 HE On-Demand Bother NAMPT 40 40 O=C(O)c1cccc(OCCOCc2ccc(Br)cc2)c1 ZINC000147478646 FH For-Sale Anodyne SRD5A2 0 51 O=C(O)c1cccc(OCCOCc2ccc(Br)cc2)c1 ZINC000147478646 FH For-Sale Anodyne CYSLTR1 23 44 O=C(O)c1cccc(OCCOCc2ccc(Br)cc2)c1 ZINC000147478646 FH For-Sale Anodyne PLA2G4B 63 47 O=C(O)c1cccc(OCCOCc2ccc(Br)cc2)c1 ZINC000147478646 FH For-Sale Anodyne ACR 30 43 O=C(O)c1cccc(OCCOCc2ccc(Br)cc2)c1 ZINC000147478646 FH For-Sale Anodyne MDH2 0 40 O=C(O)c1cccc(OCCOCc2ccc(Br)cc2)c1 ZINC000147478646 FH For-Sale Anodyne FFAR1 26 42 O=C(O)c1cccc(OCCOCc2ccc(Br)cc2)c1 ZINC000147478646 FH For-Sale Anodyne AKR1C3 26 45 CN(C)C1(CNC(=O)c2ccnc(NN)c2)CCCC1 ZINC000147478648 CC For-Sale Anodyne SLC6A5 17 48 NC1(C(=O)N2CCN(c3ccccn3)CC2)CCC1 ZINC000147478672 CC On-Demand Anodyne EBP 27 41 NC1(C(=O)N2CCN(c3ccccn3)CC2)CCC1 ZINC000147478672 CC On-Demand Anodyne GRM1 0 47 NC1(C(=O)N2CCN(c3ccccn3)CC2)CCC1 ZINC000147478672 CC On-Demand Anodyne SLC6A7 0 52 COc1c(C)ccc(NC(=O)c2cc(C)ccc2Br)c1C ZINC000147478685 EJ On-Demand Anodyne KCNMA1 22 40 O[C@H](Cc1cccc(C(F)(F)F)c1)c1cncs1 ZINC000147478817 CG For-Sale Anodyne PHES 0 40 Cc1noc(C)c1CNS(=O)(=O)c1cc(S(C)(=O)=O)ccc1Cl ZINC000147478828 GD On-Demand Anodyne EDNRA 22 45 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C)cc2OCc2ccccc2)C1 ZINC000147478830 HG On-Demand Anodyne DRD4 19 43 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C)cc2OCc2ccccc2)C1 ZINC000147478830 HG On-Demand Anodyne HTR4 44 36 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C)cc2OCc2ccccc2)C1 ZINC000147478830 HG On-Demand Anodyne CACNA1I 42 36 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne PPIA 15 44 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne ATF1 59 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne CPT1A 43 38 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne CPT2 40 32 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne NFKB1 55 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne KCNMA1 23 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne ACPS 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne AKR1C3 24 44 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne GALE 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne HCAR1 0 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne KCNK3 43 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2F)c1 ZINC000147478832 EI On-Demand Anodyne TMPRSS4 0 53 N[C@@H](COCc1ccc(Br)cc1)C(=O)O ZINC000147478845 CD For-Sale Anodyne CACNA2D1 31 51 N[C@@H](COCc1ccc(Br)cc1)C(=O)O ZINC000147478845 CD For-Sale Anodyne SLC1A1 24 55 N[C@@H](COCc1ccc(Br)cc1)C(=O)O ZINC000147478845 CD For-Sale Anodyne GRIK1 44 42 N[C@@H](COCc1ccc(Br)cc1)C(=O)O ZINC000147478845 CD For-Sale Anodyne KIF11 17 43 CN(C)C1(CNC(=O)c2ccc(NN)nc2)CCCC1 ZINC000147478857 CC For-Sale Anodyne SLC6A5 17 47 Cc1nc(Nc2ccc3c(c2)OCCO3)ccc1C(=O)O ZINC000147478876 CF For-Sale Anodyne AKR1C2 52 37 NCC1(CC(=O)N2CCN(c3ccccn3)CC2)CCC1 ZINC000147478900 CD For-Sale Anodyne SLC6A7 0 47 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2n1 ZINC000147478951 HG On-Demand Anodyne HTR4 46 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2n1 ZINC000147478951 HG On-Demand Anodyne NPY2R 27 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2n1 ZINC000147478951 HG On-Demand Anodyne TGM2 61 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2n1 ZINC000147478951 HG On-Demand Anodyne CACNA1I 55 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2n1 ZINC000147478951 HG On-Demand Anodyne F13A1 56 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2n1 ZINC000147478951 HG On-Demand Anodyne AKR1C3 20 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2n1 ZINC000147478951 HG On-Demand Anodyne NAMPT 40 39 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CCC(=O)N3CCCC3)cc1)C2 ZINC000147478976 HG On-Demand Anodyne HDAC8 18 45 COc1ccc2c(c1)OC[C@H](C(=O)Nc1ccc(CCC(=O)N3CCCC3)cc1)C2 ZINC000147478976 HG On-Demand Anodyne ROCK2 31 50 CNC(=O)c1ccc(N[C@@H]2CCO[C@@H]2C)cc1 ZINC000147478986 BD For-Sale Anodyne HDAC8 0 42 CC(C)(C)OC(=O)NCC/C=C/C=O ZINC000147478998 AD For-Sale Reactive CTSK 17 44 N[C@H](COCc1ccc(Br)cc1)C(=O)O ZINC000147479027 CD For-Sale Anodyne CACNA2D1 31 51 N[C@H](COCc1ccc(Br)cc1)C(=O)O ZINC000147479027 CD For-Sale Anodyne SLC1A1 24 55 N[C@H](COCc1ccc(Br)cc1)C(=O)O ZINC000147479027 CD For-Sale Anodyne GRIK1 44 42 N[C@H](COCc1ccc(Br)cc1)C(=O)O ZINC000147479027 CD For-Sale Anodyne KIF11 17 43 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C)cc2OCc2ccccc2)C1 ZINC000147479031 HG On-Demand Anodyne DRD4 19 43 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C)cc2OCc2ccccc2)C1 ZINC000147479031 HG On-Demand Anodyne HTR4 44 36 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C)cc2OCc2ccccc2)C1 ZINC000147479031 HG On-Demand Anodyne CACNA1I 42 36 Cn1cc(NC(=O)[C@@H]2CCC(=O)N(Cc3ccccc3)[C@@H]2c2ccccc2)cn1 ZINC000147479138 GH On-Demand Anodyne P2RX7 20 41 Cn1cc(NC(=O)[C@@H]2CCC(=O)N(Cc3ccccc3)[C@@H]2c2ccccc2)cn1 ZINC000147479138 GH On-Demand Anodyne PANC 48 38 CNC(=O)c1ccc(N[C@@H]2CCO[C@H]2C)cc1 ZINC000147479145 BD For-Sale Anodyne HDAC8 0 42 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(CCC(=O)N3CCCC3)cc1)C2 ZINC000147479156 HG On-Demand Anodyne HDAC8 18 45 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(CCC(=O)N3CCCC3)cc1)C2 ZINC000147479156 HG On-Demand Anodyne ROCK2 31 50 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne HTR1A 27 41 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne DRD2 55 52 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne DRD4 31 52 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne ACHE 19 41 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne ADRA1D 26 41 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne ADRA1A 21 41 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne ADRA1B 19 41 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne DRD3 50 48 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne HTR4 86 42 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne CHRM5 15 42 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne HTR7 19 42 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne SIGMAR1 15 48 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne MMP13 27 44 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne CCR3 16 48 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne KCNA3 57 45 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne MMP2 15 44 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne MMP3 28 40 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne SLC6A9 26 48 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne MMP9 26 40 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne EPHX2 26 44 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne TGM2 67 49 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne MMP7 30 40 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne MMP1 30 42 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne CACNA1I 63 36 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne F13A1 67 45 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne AKR1C3 29 40 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne HCN1 81 44 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne HCN4 57 42 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne ACKR3 54 36 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne KCNK3 34 40 COc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479247 GF On-Demand Anodyne KCNK9 26 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccsc2)c1 ZINC000147479285 CG On-Demand Anodyne CPT1A 16 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccsc2)c1 ZINC000147479285 CG On-Demand Anodyne ITGAV 18 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccsc2)c1 ZINC000147479285 CG On-Demand Anodyne HCAR1 0 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccsc2)c1 ZINC000147479285 CG On-Demand Anodyne KCNK3 50 56 NC1(C(=O)N2CCN(c3cccc(Cl)c3)CC2)CCC1 ZINC000147479315 CD On-Demand Anodyne AKR1C3 0 54 CNC(=O)c1ccc(N[C@H]2CCO[C@@H]2C)cc1 ZINC000147479346 BD For-Sale Anodyne HDAC8 0 42 Cc1nc(NCCc2ccc(Cl)cc2Cl)ccc1C(=O)O ZINC000147479353 EI For-Sale Anodyne CNR1 24 42 Cc1nc(NCCc2ccc(Cl)cc2Cl)ccc1C(=O)O ZINC000147479353 EI For-Sale Anodyne PTGDR 31 56 Cc1nc(NCCc2ccc(Cl)cc2Cl)ccc1C(=O)O ZINC000147479353 EI For-Sale Anodyne DPP8 50 32 Cc1nc(NCCc2ccc(Cl)cc2Cl)ccc1C(=O)O ZINC000147479353 EI For-Sale Anodyne DPP9 49 32 Cc1nc(NCCc2ccc(Cl)cc2Cl)ccc1C(=O)O ZINC000147479353 EI For-Sale Anodyne AKR1C2 41 35 Cc1nc(NCCc2ccc(Cl)cc2Cl)ccc1C(=O)O ZINC000147479353 EI For-Sale Anodyne AKR1C1 44 35 Cn1cc(NC(=O)[C@H]2CCC(=O)N(Cc3ccccc3)[C@@H]2c2ccccc2)cn1 ZINC000147479357 GH On-Demand Anodyne P2RX7 20 41 Cn1cc(NC(=O)[C@H]2CCC(=O)N(Cc3ccccc3)[C@@H]2c2ccccc2)cn1 ZINC000147479357 GH On-Demand Anodyne PANC 48 38 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(CN3CCOC3=O)cc2)C1 ZINC000147479359 GD On-Demand Anodyne HTR4 44 39 CC(C)CCCCNCC(=O)O ZINC000147479373 AD For-Sale Anodyne DNPEP 49 31 CN(C)C1(CNC(=O)c2cccc(NN)n2)CCCC1 ZINC000147479380 CC For-Sale Anodyne SLC6A5 15 42 CNC(=O)c1ccc(N[C@H]2CCO[C@H]2C)cc1 ZINC000147479557 BD For-Sale Anodyne HDAC8 0 42 Cn1cc(NC(=O)[C@@H]2CCC(=O)N(Cc3ccccc3)[C@H]2c2ccccc2)cn1 ZINC000147479564 GH On-Demand Anodyne P2RX7 20 41 Cn1cc(NC(=O)[C@@H]2CCC(=O)N(Cc3ccccc3)[C@H]2c2ccccc2)cn1 ZINC000147479564 GH On-Demand Anodyne PANC 48 38 NCC1(CC(=O)N2CCC(C(N)=O)CC2)CCC1 ZINC000147479574 CC For-Sale Anodyne CACNA2D1 36 42 CC[C@H](Br)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147479580 EG For-Sale Reactive CACNA1D 60 34 COc1ccc(-c2nnc(SCC(=O)Nc3ccc(-n4cnnn4)cc3)o2)cc1 ZINC000147479582 HE On-Demand Anodyne ENPP1 72 34 Cc1ccc2c(c1)CCCN2c1ccc(C(=O)O)c(C)n1 ZINC000147479586 CG For-Sale Anodyne SRD5A1 39 42 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(CN3CCOC3=O)cc2)C1 ZINC000147479590 GD On-Demand Anodyne HTR4 44 39 CC(C)CCCCNCc1nc2ccccc2c(=O)[nH]1 ZINC000147479594 CF For-Sale Anodyne METG 51 33 CC(C)CCCCNCc1nc2ccccc2c(=O)[nH]1 ZINC000147479594 CF For-Sale Anodyne PARP3 26 47 CC(C)CCCCNCc1nc2ccccc2c(=O)[nH]1 ZINC000147479594 CF For-Sale Anodyne QTRT1 0 40 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne CA2 15 45 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne HTR4 54 36 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne GRIN2B 28 47 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne LPL 51 35 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne NPY2R 16 40 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne CPT1A 44 36 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne PRNP 47 37 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne EPHX2 41 48 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne TGM2 98 53 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne CACNA1I 66 43 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne F13A1 110 53 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne NOD2 40 34 CC(=O)Nc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147479597 HE On-Demand Anodyne NAMPT 61 46 CC(=O)Nc1cccc(CNC(=O)N(C)Cc2cscn2)c1 ZINC000147479601 DE On-Demand Anodyne GPR142 36 44 COc1ccc(OCCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147479608 FF On-Demand Anodyne SCNN1A 32 43 COc1ccc(OCCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147479608 FF On-Demand Anodyne NQO2 36 40 COc1ccc(OCCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147479608 FF On-Demand Anodyne MTNR1A 92 46 COc1ccc(OCCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147479608 FF On-Demand Anodyne MTNR1B 78 40 COc1ccc(OCCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147479608 FF On-Demand Anodyne ROCK2 33 45 COc1ccc(OCCCNC(=O)[C@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147479608 FF On-Demand Anodyne IKBKE 43 37 Cn1c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc(Cl)c1Cl ZINC000147479722 EH On-Demand Anodyne CACNA1I 50 36 CCOc1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147479748 EH For-Sale Reactive AVPR1A 15 42 CCOc1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147479748 EH For-Sale Reactive HCRTR1 0 49 CCOc1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147479748 EH For-Sale Reactive HRH3 19 41 CCOc1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147479748 EH For-Sale Reactive CHEK2 15 43 CC[C@@H](Br)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147479775 EG For-Sale Reactive CACNA1D 60 34 Cn1cc(NC(=O)[C@H]2CCC(=O)N(Cc3ccccc3)[C@H]2c2ccccc2)cn1 ZINC000147479781 GH On-Demand Anodyne P2RX7 20 41 Cn1cc(NC(=O)[C@H]2CCC(=O)N(Cc3ccccc3)[C@H]2c2ccccc2)cn1 ZINC000147479781 GH On-Demand Anodyne PANC 48 38 Cc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1[N+](=O)[O-] ZINC000147479787 CG For-Sale Bother AKR1C2 54 39 NC1(C(=O)N2CCc3ccccc3C2)CCC1 ZINC000147479794 BD On-Demand Anodyne PREP 23 40 NC1(C(=O)N2CCc3ccccc3C2)CCC1 ZINC000147479794 BD On-Demand Anodyne DPP8 26 43 NC1(C(=O)N2CCc3ccccc3C2)CCC1 ZINC000147479794 BD On-Demand Anodyne SLC7A5 0 44 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne F2 19 46 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne PRSS1 15 46 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne FKBP1A 38 47 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne GRIN2B 57 46 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne SIGMAR1 25 58 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne PREP 43 35 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne MMP2 17 44 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne MMP3 27 40 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne CAPN1 19 40 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne MMP9 19 40 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne EPHX2 22 46 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne TGM2 90 52 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne MMP7 33 40 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne MMP1 22 40 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne CACNA1I 42 37 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne F13A1 98 52 O=C(CCc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147479814 GF On-Demand Anodyne NAMPT 49 44 CN(C)C1(CNC(=O)c2ccc(NN)cc2)CCCC1 ZINC000147479839 CD For-Sale Anodyne SLC6A5 17 48 CCOC(=O)C(F)(F)c1cccc([N+](=O)[O-])c1 ZINC000147479905 BE For-Sale Bother CACNA1C 72 44 CCOC(=O)C(F)(F)c1cccc([N+](=O)[O-])c1 ZINC000147479905 BE For-Sale Bother CACNA1D 98 44 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(-n3nc(C)cc3C)c(F)c2)C1 ZINC000147479910 HE On-Demand Anodyne NPY2R 67 37 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)n1C ZINC000147479949 CF On-Demand Anodyne CACNA1I 41 33 O=C(c1c(F)cccc1F)N1CCN(Cc2ccc([N+](=O)[O-])cc2F)CC1 ZINC000147479965 GF On-Demand Bother FAAH 15 44 COC(=O)Cc1csc(-c2cc(Cl)ccc2F)n1 ZINC000147479966 CG For-Sale Anodyne PTGER1 31 50 COC(=O)Cc1csc(-c2cc(Cl)ccc2F)n1 ZINC000147479966 CG For-Sale Anodyne TSPO 0 41 CC[C@H](Br)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147479969 EG For-Sale Reactive CACNA1D 60 34 Cc1nn(-c2ccc(Cl)c(Cl)c2)c(Cl)c1S(=O)(=O)Cl ZINC000147479982 FI For-Sale Unstable RPA1 42 40 CCOc1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147479995 EH For-Sale Reactive AVPR1A 15 42 CCOc1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147479995 EH For-Sale Reactive HCRTR1 0 49 CCOc1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147479995 EH For-Sale Reactive HRH3 19 41 CCOc1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147479995 EH For-Sale Reactive CHEK2 15 43 Cc1nc(Nc2ccc(S(C)(=O)=O)cc2)ccc1C(=O)O ZINC000147479997 DE For-Sale Anodyne PTGS2 24 44 Cc1nc(Nc2ccc(S(C)(=O)=O)cc2)ccc1C(=O)O ZINC000147479997 DE For-Sale Anodyne AKR1C2 61 38 Cc1nc(Nc2ccc(S(C)(=O)=O)cc2)ccc1C(=O)O ZINC000147479997 DE For-Sale Anodyne MT-CO2 34 42 NCC1(CC(=O)N2CCc3ccccc3C2)CCC1 ZINC000147480003 CE For-Sale Anodyne DPP8 26 44 Cc1cc(F)c(N)cc1S(=O)(=O)Nc1ccncc1Br ZINC000147480004 FF For-Sale Anodyne PTGS1 0 40 COc1cccc(/C=N/CCO)c1 ZINC000147480057 AD For-Sale Mild CYP1B1 27 42 COc1cccc(/C=N/CCO)c1 ZINC000147480057 AD For-Sale Mild G6PC 27 50 COc1cccc(/C=N/CCO)c1 ZINC000147480057 AD For-Sale Mild AHR 24 44 COc1cccc(/C=N/CCO)c1 ZINC000147480057 AD For-Sale Mild CYP1A1 24 42 CN(C)C1(CNC(=O)c2cnc(NN)c(Cl)c2)CCCC1 ZINC000147480092 DD For-Sale Anodyne SLC6A5 16 47 CC(C)CCCCNCc1ccc(I)cc1 ZINC000147480093 EI For-Sale Anodyne FOLH1 22 51 CC(C)CCCCNCc1ccc(I)cc1 ZINC000147480093 EI For-Sale Anodyne FDFT1 0 41 CC(C)CCCCNCc1ccc(I)cc1 ZINC000147480093 EI For-Sale Anodyne S1PR2 29 41 CC(C)CCCCNCc1ccc(I)cc1 ZINC000147480093 EI For-Sale Anodyne LEF 78 39 CC(C)CCCCNCc1ccc(I)cc1 ZINC000147480093 EI For-Sale Anodyne GPM3 0 49 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(-n3nc(C)cc3C)c(F)c2)C1 ZINC000147480121 HE On-Demand Anodyne NPY2R 67 37 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne CHRM5 15 42 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne GRIN2B 35 41 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne MMP13 40 43 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne ADAM17 41 39 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne CPT1A 82 38 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne MMP3 29 41 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne MMP9 23 41 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne EPHX2 25 49 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne TGM2 83 47 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne MMP7 35 41 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne MMP1 34 41 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne F13A1 89 47 O=C(COc1ccccc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147480126 GE On-Demand Anodyne NAMPT 45 39 CN(C)Cc1ccccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147480138 FI On-Demand Anodyne FABH 0 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)ccc2Br)c1 ZINC000147480171 FI On-Demand Anodyne ATF1 55 39 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)ccc2Br)c1 ZINC000147480171 FI On-Demand Anodyne NFKB1 51 39 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(F)ccc2Br)c1 ZINC000147480171 FI On-Demand Anodyne TMPRSS4 0 40 CC[C@@H](Br)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147480173 EG For-Sale Reactive CACNA1D 60 34 COc1cc(S(=O)(=O)Nc2ccncc2Br)ccc1N ZINC000147480216 FE For-Sale Anodyne FFAR4 23 40 CCCc1nn(-c2ccc(Cl)c(Cl)c2)c(Cl)c1S(=O)(=O)Cl ZINC000147480229 GJ For-Sale Unstable RPA1 40 35 CCOc1ccccc1C(=O)N1CCC[C@@H]1CCCBr ZINC000147480235 EH For-Sale Reactive HCRTR1 34 49 CCOc1ccccc1C(=O)N1CCC[C@@H]1CCCBr ZINC000147480235 EH For-Sale Reactive HCRTR2 34 49 CCOc1ccccc1C(=O)N1CCC[C@@H]1CCCBr ZINC000147480235 EH For-Sale Reactive HCN1 58 39 CCOc1ccccc1C(=O)N1CCC[C@@H]1CCCBr ZINC000147480235 EH For-Sale Reactive HCN4 51 39 CC(=O)Nc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147480237 CF For-Sale Anodyne AKR1C3 36 40 CC(=O)Nc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147480237 CF For-Sale Anodyne AKR1C2 65 40 CC(=O)Nc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147480237 CF For-Sale Anodyne MT-CO2 23 40 CCOC(=O)[C@@H](C)c1cccc2ccc(O)cc12 ZINC000147480273 BG For-Sale Anodyne CA7 19 41 CCOC(=O)[C@@H](C)c1cccc2ccc(O)cc12 ZINC000147480273 BG For-Sale Anodyne CA14 17 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne F2 29 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne ADRA2A 15 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne DRD2 15 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne DRD3 18 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne HTR4 54 38 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne F10 25 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne CHRM5 19 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne GRIN2B 36 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne TRY2_BOVIN 70 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne CCR3 25 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne PLD1 32 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne CASP1 34 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne EPHX2 26 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne PLD2 37 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne TGM2 73 53 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne MCHR1 21 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne CACNA1I 69 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne F13A1 65 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne AKR1C3 64 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne SFRP1 27 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2ccccc2c1 ZINC000147480358 HH On-Demand Anodyne NAMPT 49 45 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C(C)(C)CCl ZINC000147480387 CG For-Sale Reactive CACNA1D 48 33 Nc1cc(F)c(S(=O)(=O)Nc2ccncc2Br)c(F)c1 ZINC000147480414 FF For-Sale Anodyne PTGS1 0 42 CCOc1ccccc1C(=O)N1CCC[C@H]1CCCBr ZINC000147480432 EH For-Sale Reactive HCRTR1 34 49 CCOc1ccccc1C(=O)N1CCC[C@H]1CCCBr ZINC000147480432 EH For-Sale Reactive HCRTR2 34 49 CCOc1ccccc1C(=O)N1CCC[C@H]1CCCBr ZINC000147480432 EH For-Sale Reactive HCN1 58 39 CCOc1ccccc1C(=O)N1CCC[C@H]1CCCBr ZINC000147480432 EH For-Sale Reactive HCN4 51 39 CC(C)c1nn(-c2ccc(Cl)c(Cl)c2)c(Cl)c1S(=O)(=O)Cl ZINC000147480456 GJ For-Sale Unstable RPA1 53 35 COC(=O)Cc1csc(CSc2ccc(Br)cc2)n1 ZINC000147480457 FH For-Sale Anodyne FAS 48 42 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCc3cccc(F)c3)c2)C1 ZINC000147480459 HG On-Demand Anodyne F10 15 43 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCc3cccc(F)c3)c2)C1 ZINC000147480459 HG On-Demand Anodyne CCR3 110 44 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCc3cccc(F)c3)c2)C1 ZINC000147480459 HG On-Demand Anodyne CCR5 65 34 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(OCc3cccc(F)c3)c2)C1 ZINC000147480459 HG On-Demand Anodyne CACNA1I 45 33 NCC1(CC(=O)Nc2ccc(F)c(F)c2)CCC1 ZINC000147480474 CE For-Sale Anodyne SLC1A2 45 38 NCC1(CC(=O)Nc2ccc(F)c(F)c2)CCC1 ZINC000147480474 CE For-Sale Anodyne ENV 42 34 CCOC(=O)[C@H](C)c1cccc2ccc(O)cc12 ZINC000147480493 BG For-Sale Anodyne CA7 19 41 CCOC(=O)[C@H](C)c1cccc2ccc(O)cc12 ZINC000147480493 BG For-Sale Anodyne CA14 17 41 CN(C)C1(CNC(=O)c2ccc(NN)nn2)CCCC1 ZINC000147480519 CC For-Sale Anodyne HCN1 40 31 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1ccc(C(=O)N(C)C)c(Cl)c1)C2 ZINC000147480526 GG On-Demand Anodyne ROCK2 31 50 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne CHRM2 28 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne HTR4 49 35 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne F10 16 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne EDNRB 41 35 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne EPHX2 18 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne PKM 35 47 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne TGM2 62 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne MCHR1 16 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne CACNA1I 64 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne F13A1 53 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne AKR1C3 46 35 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1ccc2c(c1)OCO2 ZINC000147480565 HE On-Demand Anodyne SFRP1 31 41 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C(C)(C)CCl ZINC000147480574 CG For-Sale Reactive CACNA1D 48 33 COC(=O)COc1cccc(NC(=O)[C@H]2CC[C@@H](C)O2)c1 ZINC000147480599 CD On-Demand Anodyne F10 15 40 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCc3cccc(F)c3)c2)C1 ZINC000147480633 HG On-Demand Anodyne F10 15 43 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCc3cccc(F)c3)c2)C1 ZINC000147480633 HG On-Demand Anodyne CCR3 110 44 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCc3cccc(F)c3)c2)C1 ZINC000147480633 HG On-Demand Anodyne CCR5 65 34 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(OCc3cccc(F)c3)c2)C1 ZINC000147480633 HG On-Demand Anodyne CACNA1I 45 33 Nc1cc(S(=O)(=O)Nc2ccncc2Br)c(F)cc1F ZINC000147480670 FF For-Sale Anodyne PTGS1 0 42 Cc1nc(Nc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147480671 CF For-Sale Anodyne NOS2 46 30 Cc1nc(Nc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147480671 CF For-Sale Anodyne CLK1 19 41 Cc1nc(Nc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147480671 CF For-Sale Anodyne DYRK2 44 38 Cc1nc(Nc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147480671 CF For-Sale Anodyne AKR1C2 52 37 Cc1nc(Nc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147480671 CF For-Sale Anodyne TRPC6 36 41 Cc1nc(Nc2ccc3c(c2)OCO3)ccc1C(=O)O ZINC000147480671 CF For-Sale Anodyne TRPC3 39 44 COc1ccc(C(=O)N2CCC[C@@H]2CCCBr)c(OC)c1 ZINC000147480676 FG For-Sale Reactive ACKR3 61 31 CNC(=O)c1ccc(NCc2ccon2)c([N+](=O)[O-])c1 ZINC000147480689 CD On-Demand Bother DRTS_TOXGO 15 46 CNC(=O)c1ccc(NCc2ccon2)c([N+](=O)[O-])c1 ZINC000147480689 CD On-Demand Bother TAAR1 15 42 COCc1nn(-c2ccc(Cl)c(Cl)c2)c(Cl)c1S(=O)(=O)Cl ZINC000147480695 GH For-Sale Unstable RPA1 45 36 COc1ccc2ccc(-c3nn(-c4ccccc4)cc3C(=O)N[C@@H](C)C(N)=O)cc2c1 ZINC000147480700 HG On-Demand Anodyne CDK2 19 54 COc1ccc2ccc(-c3nn(-c4ccccc4)cc3C(=O)N[C@@H](C)C(N)=O)cc2c1 ZINC000147480700 HG On-Demand Anodyne CDK4 18 54 O=C(O)[C@@H](F)OCc1ccc(Br)cc1 ZINC000147480709 CE For-Sale Anodyne CPA1 25 49 O=C(O)[C@@H](F)OCc1ccc(Br)cc1 ZINC000147480709 CE For-Sale Anodyne SLC1A6 0 40 O=C(O)[C@@H](F)OCc1ccc(Br)cc1 ZINC000147480709 CE For-Sale Anodyne SLC1A7 0 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnccn1 ZINC000147480762 FD On-Demand Anodyne HTR4 47 36 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnccn1 ZINC000147480762 FD On-Demand Anodyne GRIN2B 26 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnccn1 ZINC000147480762 FD On-Demand Anodyne TGM2 66 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnccn1 ZINC000147480762 FD On-Demand Anodyne CACNA1I 45 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnccn1 ZINC000147480762 FD On-Demand Anodyne F13A1 77 46 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cnccn1 ZINC000147480762 FD On-Demand Anodyne NAMPT 78 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cnsn2)c1 ZINC000147480772 CE On-Demand Anodyne ATF1 47 38 O=C(O)c1cc(Cl)cc(NC(=O)c2cnsn2)c1 ZINC000147480772 CE On-Demand Anodyne NFKB1 43 38 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](C)CCl ZINC000147480797 CF For-Sale Reactive CACNA1C 41 35 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](C)CCl ZINC000147480797 CF For-Sale Reactive CACNA1D 65 34 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](C)CCl ZINC000147480797 CF For-Sale Reactive TRPM8 0 40 CN(C)C1(CNC(=O)c2cc(Cl)nc(NN)c2)CCCC1 ZINC000147480801 DD For-Sale Anodyne SLC6A5 17 50 COC(=O)COc1cccc(NC(=O)[C@H]2CC[C@H](C)O2)c1 ZINC000147480805 CD On-Demand Anodyne F10 15 40 COc1ccc(C(=O)N2CCC[C@H]2CCCBr)c(OC)c1 ZINC000147480851 FG For-Sale Reactive ACKR3 61 31 CCCCC(=O)N(C)N ZINC000147480893 AC For-Sale Reactive CQSS 58 35 COc1ccc2ccc(-c3nn(-c4ccccc4)cc3C(=O)N[C@H](C)C(N)=O)cc2c1 ZINC000147480894 HG On-Demand Anodyne CDK2 19 54 COc1ccc2ccc(-c3nn(-c4ccccc4)cc3C(=O)N[C@H](C)C(N)=O)cc2c1 ZINC000147480894 HG On-Demand Anodyne CDK4 18 54 CCc1nn(-c2ccc(Cl)c(Cl)c2)c(Cl)c1S(=O)(=O)Cl ZINC000147480911 FI For-Sale Unstable RPA1 73 38 CN(C(=O)CC1(CN)CCC1)C1CCCCC1 ZINC000147480925 BE For-Sale Anodyne CACNA2D1 58 47 O=C(O)[C@H](F)OCc1ccc(Br)cc1 ZINC000147480935 CE For-Sale Anodyne CPA1 25 49 O=C(O)[C@H](F)OCc1ccc(Br)cc1 ZINC000147480935 CE For-Sale Anodyne SLC1A6 0 40 O=C(O)[C@H](F)OCc1ccc(Br)cc1 ZINC000147480935 CE For-Sale Anodyne SLC1A7 0 40 COc1ccc2c(c1)OC[C@H](C(=O)N1CCC(CNC(C)=O)CC1)C2 ZINC000147480981 ED On-Demand Anodyne NQO2 31 40 COc1ccc2c(c1)OC[C@H](C(=O)N1CCC(CNC(C)=O)CC1)C2 ZINC000147480981 ED On-Demand Anodyne MTNR1A 64 49 COc1ccc2c(c1)OC[C@H](C(=O)N1CCC(CNC(C)=O)CC1)C2 ZINC000147480981 ED On-Demand Anodyne MTNR1B 54 42 C[C@H](CCl)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147480983 CF For-Sale Reactive CACNA1C 41 35 C[C@H](CCl)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147480983 CF For-Sale Reactive CACNA1D 65 34 C[C@H](CCl)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147480983 CF For-Sale Reactive TRPM8 0 40 CC(C)[C@@H]1C(=O)Nc2ccc(F)cc21 ZINC000147480986 AF For-Sale Anodyne AKR1B1 17 58 Cc1noc(C)c1CNS(=O)(=O)N1CCOCC1 ZINC000147480993 CB On-Demand Anodyne ADAMTS4 35 40 Cc1ccc(OC[C@H](O)CNCCCCC(C)C)c(C)c1 ZINC000147480999 CG For-Sale Anodyne ADRB2 32 51 Cc1ccc(OC[C@H](O)CNCCCCC(C)C)c(C)c1 ZINC000147480999 CG For-Sale Anodyne ADRB1 48 39 Cc1ccc(OC[C@H](O)CNCCCCC(C)C)c(C)c1 ZINC000147480999 CG For-Sale Anodyne ABCB1 0 50 COC(=O)COc1cccc(NC(=O)[C@@H]2CC[C@@H](C)O2)c1 ZINC000147481014 CD On-Demand Anodyne F10 15 40 O=C(O)c1cc(Cl)cc(NC(=O)c2csc(I)c2)c1 ZINC000147481021 HH On-Demand Anodyne PPIA 16 46 O=C(O)c1cc(Cl)cc(NC(=O)c2csc(I)c2)c1 ZINC000147481021 HH On-Demand Anodyne AKR1C3 19 42 O=C(O)c1cc(Cl)cc(NC(=O)c2csc(I)c2)c1 ZINC000147481021 HH On-Demand Anodyne KCNK3 44 40 C=CCCOCC(=O)Nc1ccc(CN2CCN(Cc3ccccc3)CC2)cc1 ZINC000147481031 GH On-Demand Mild ACHE 23 43 C=CCCOCC(=O)Nc1ccc(CN2CCN(Cc3ccccc3)CC2)cc1 ZINC000147481031 GH On-Demand Mild LTA4H 44 50 C=CCCOCC(=O)Nc1ccc(CN2CCN(Cc3ccccc3)CC2)cc1 ZINC000147481031 GH On-Demand Mild SIGMAR1 44 47 C=CCCOCC(=O)Nc1ccc(CN2CCN(Cc3ccccc3)CC2)cc1 ZINC000147481031 GH On-Demand Mild FAAH 23 45 C=CCCOCC(=O)Nc1ccc(CN2CCN(Cc3ccccc3)CC2)cc1 ZINC000147481031 GH On-Demand Mild CACNA1G 19 47 C=CCCOCC(=O)Nc1ccc(CN2CCN(Cc3ccccc3)CC2)cc1 ZINC000147481031 GH On-Demand Mild F13A1 56 37 C=CCCOCC(=O)Nc1ccc(CN2CCN(Cc3ccccc3)CC2)cc1 ZINC000147481031 GH On-Demand Mild NPFFR1 40 35 C=CCCOCC(=O)Nc1ccc(CN2CCN(Cc3ccccc3)CC2)cc1 ZINC000147481031 GH On-Demand Mild NOD2 43 36 N#Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147481050 GE On-Demand Mild HTR4 42 35 N#Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147481050 GE On-Demand Mild GRIN2B 23 48 N#Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147481050 GE On-Demand Mild EPHX2 17 43 N#Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147481050 GE On-Demand Mild TGM2 66 48 N#Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147481050 GE On-Demand Mild CTRB_BOVIN 48 38 N#Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147481050 GE On-Demand Mild CACNA1I 63 38 N#Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147481050 GE On-Demand Mild F13A1 56 44 N#Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147481050 GE On-Demand Mild AKR1C3 40 41 N#Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1 ZINC000147481050 GE On-Demand Mild NAMPT 37 40 O=C(Nc1cc(Br)cc(C(=O)O)c1)NC1CCC1 ZINC000147481061 DF For-Sale Anodyne EPHX2 55 45 COc1cc(CNC(=O)N(C)Cc2cscn2)ccc1O ZINC000147481079 DE On-Demand Anodyne TRPV1 27 47 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(OC3CCCC3)c(Cl)c2)C1 ZINC000147481101 HG On-Demand Anodyne HTR4 51 38 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(OC3CCCC3)c(Cl)c2)C1 ZINC000147481101 HG On-Demand Anodyne CCR3 45 38 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(OC3CCCC3)c(Cl)c2)C1 ZINC000147481101 HG On-Demand Anodyne CACNA1I 70 36 O=[N+]([O-])c1ccncc1OCc1ccccc1 ZINC000147481120 BF For-Sale Bother CYP11B1 15 41 O=[N+]([O-])c1ccncc1OCc1ccccc1 ZINC000147481120 BF For-Sale Bother PPIA 48 43 O=[N+]([O-])c1ccncc1OCc1ccccc1 ZINC000147481120 BF For-Sale Bother CYP11B2 15 50 O=S(=O)(Cl)c1c(C2CC2)nn(-c2ccc(Cl)c(Cl)c2)c1Cl ZINC000147481158 GJ For-Sale Unstable RPA1 41 35 CC(C)[C@H]1C(=O)Nc2ccc(F)cc21 ZINC000147481190 AF For-Sale Anodyne AKR1B1 17 58 NCC1(CC(=O)NCCc2ccccc2)CCC1 ZINC000147481194 BD For-Sale Anodyne CACNA2D1 23 45 NCC1(CC(=O)NCCc2ccccc2)CCC1 ZINC000147481194 BD For-Sale Anodyne CA5B 22 46 NCC1(CC(=O)NCCc2ccccc2)CCC1 ZINC000147481194 BD For-Sale Anodyne SCN5A 0 40 NCC1(CC(=O)NCCc2ccccc2)CCC1 ZINC000147481194 BD For-Sale Anodyne NCE103 25 42 NCC1(CC(=O)NCCc2ccccc2)CCC1 ZINC000147481194 BD For-Sale Anodyne SLC12A5 46 36 NCC1(CC(=O)NCCc2ccccc2)CCC1 ZINC000147481194 BD For-Sale Anodyne CAN2 0 42 Cc1nc(N(C)Cc2cccc(F)c2)ccc1C(=O)O ZINC000147481198 CF For-Sale Anodyne HAO2 62 44 O=C(O)c1ccccc1OCCOCc1ccc(Br)cc1 ZINC000147481199 FH For-Sale Anodyne POBA 0 44 COCc1nc(C(=O)Nc2nc3ccc(OC(F)(F)F)cc3s2)cs1 ZINC000147481200 GI On-Demand Anodyne CSNK1D 55 55 COCc1nc(C(=O)Nc2nc3ccc(OC(F)(F)F)cc3s2)cs1 ZINC000147481200 GI On-Demand Anodyne RAF1 18 41 COCc1nc(C(=O)Nc2nc3ccc(OC(F)(F)F)cc3s2)cs1 ZINC000147481200 GI On-Demand Anodyne HSD17B1 29 41 COCc1nc(C(=O)Nc2nc3ccc(OC(F)(F)F)cc3s2)cs1 ZINC000147481200 GI On-Demand Anodyne SCN10A 29 46 Cc1cccc(OCCC(=O)N2CCC[C@@H]2CCCBr)c1 ZINC000147481207 FH For-Sale Reactive CHRNA10 48 37 C[C@@H](CCl)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147481218 CF For-Sale Reactive CACNA1C 41 35 C[C@@H](CCl)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147481218 CF For-Sale Reactive CACNA1D 65 34 C[C@@H](CCl)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147481218 CF For-Sale Reactive TRPM8 0 40 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC(CNC(C)=O)CC1)C2 ZINC000147481220 ED On-Demand Anodyne NQO2 31 40 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC(CNC(C)=O)CC1)C2 ZINC000147481220 ED On-Demand Anodyne MTNR1A 64 49 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC(CNC(C)=O)CC1)C2 ZINC000147481220 ED On-Demand Anodyne MTNR1B 54 42 Cc1ccc(OC[C@@H](O)CNCCCCC(C)C)c(C)c1 ZINC000147481227 CG For-Sale Anodyne ADRB2 32 51 Cc1ccc(OC[C@@H](O)CNCCCCC(C)C)c(C)c1 ZINC000147481227 CG For-Sale Anodyne ADRB1 48 39 Cc1ccc(OC[C@@H](O)CNCCCCC(C)C)c(C)c1 ZINC000147481227 CG For-Sale Anodyne ABCB1 0 50 COC(=O)COc1cccc(NC(=O)[C@@H]2CC[C@H](C)O2)c1 ZINC000147481242 CD On-Demand Anodyne F10 15 40 CCOC(=O)c1ccc(N(CC)C2CC2)nc1 ZINC000147481285 BE For-Sale Anodyne RXRA 43 39 Cc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147481292 FF On-Demand Anodyne SLC6A1 43 35 Cc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147481292 FF On-Demand Anodyne HTR4 63 42 Cc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147481292 FF On-Demand Anodyne CHRM5 15 46 Cc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147481292 FF On-Demand Anodyne EPHX2 35 43 Cc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147481292 FF On-Demand Anodyne TGM2 67 46 Cc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147481292 FF On-Demand Anodyne CACNA1I 51 36 Cc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147481292 FF On-Demand Anodyne F13A1 73 46 Cc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147481292 FF On-Demand Anodyne CCR8 67 39 Cc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147481292 FF On-Demand Anodyne HCN1 52 31 Cc1ccccc1C(=O)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147481292 FF On-Demand Anodyne HCN4 40 31 O=C(Nc1cc(Cl)cc(C(=O)O)c1)NC1CCC1 ZINC000147481300 CF On-Demand Anodyne EPHX2 54 54 O=C(Nc1cc(Cl)cc(C(=O)O)c1)NC1CCC1 ZINC000147481300 CF On-Demand Anodyne CXCR3 16 49 O=C(Nc1cc(Cl)cc(C(=O)O)c1)NC1CCC1 ZINC000147481300 CF On-Demand Anodyne HCAR1 0 40 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(OC3CCCC3)c(Cl)c2)C1 ZINC000147481331 HG On-Demand Anodyne HTR4 51 38 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(OC3CCCC3)c(Cl)c2)C1 ZINC000147481331 HG On-Demand Anodyne CCR3 45 38 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(OC3CCCC3)c(Cl)c2)C1 ZINC000147481331 HG On-Demand Anodyne CACNA1I 70 36 COC(=O)C(C(=O)OC)[C@H]1CCCC[C@@H]1NS(=O)(=O)c1ccc(C)cc1 ZINC000147481338 GD Annotated Anodyne CASR 27 43 COC(=O)C(C(=O)OC)[C@H]1CCCC[C@@H]1NS(=O)(=O)c1ccc(C)cc1 ZINC000147481338 GD Annotated Anodyne MMP13 20 43 COC(=O)C(C(=O)OC)[C@H]1CCCC[C@@H]1NS(=O)(=O)c1ccc(C)cc1 ZINC000147481338 GD Annotated Anodyne MMP2 25 43 COC(=O)C(C(=O)OC)[C@H]1CCCC[C@@H]1NS(=O)(=O)c1ccc(C)cc1 ZINC000147481338 GD Annotated Anodyne GRIA4 17 41 Cc1nn(-c2cccc(C(F)(F)F)c2)c(Cl)c1S(=O)(=O)Cl ZINC000147481369 FH For-Sale Unstable NPY5R 18 46 CN1CCC(N(C)C(=O)CC2(CN)CCC2)CC1 ZINC000147481405 CD For-Sale Anodyne CACNA2D1 34 41 Cc1cccc(OCCC(=O)N2CCC[C@H]2CCCBr)c1 ZINC000147481409 FH For-Sale Reactive CHRNA10 48 37 C[C@H](CCl)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147481418 CF For-Sale Reactive CACNA1C 41 35 C[C@H](CCl)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147481418 CF For-Sale Reactive CACNA1D 65 34 C[C@H](CCl)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147481418 CF For-Sale Reactive TRPM8 0 40 CC(=O)NCC1CCN(C(=O)c2cnn(-c3ccccc3Cl)c2)CC1 ZINC000147481435 FF On-Demand Anodyne CACNA1I 55 36 CC(=O)NCC1CCN(C(=O)c2cnn(-c3ccccc3Cl)c2)CC1 ZINC000147481435 FF On-Demand Anodyne L3MBTL3 48 33 CN(Cc1cscn1)C(=O)NCCc1ccc(C(C)(C)C)cc1 ZINC000147481479 EH On-Demand Anodyne BMP1 0 40 Cc1cc(C(=O)NCC2(N(C)C)CCCC2)ccc1NN ZINC000147481514 CD For-Sale Anodyne SLC6A5 17 47 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne DRD2 44 55 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne DRD4 41 33 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne ACHE 18 43 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne OXTR 19 40 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne DRD3 44 49 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne AVPR1B 44 31 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne HTR4 90 43 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne SIGMAR1 17 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne MMP13 64 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne CCR3 27 41 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne KCNA3 49 38 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne MTNR1A 46 36 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne MTNR1B 50 37 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne MMP2 34 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne MMP3 59 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne MMP8 33 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne MMP9 50 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne EPHX2 22 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne TGM2 57 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne MMP7 51 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne MMP1 59 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne MCHR1 21 47 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne CACNA1I 58 34 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne F13A1 47 42 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne AKR1C3 37 41 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne AKR1C2 45 33 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(OC)c1 ZINC000147481542 HF On-Demand Anodyne ACKR3 49 35 COc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1O ZINC000147481679 EG For-Sale Reactive HCRTR1 18 46 COc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1O ZINC000147481679 EG For-Sale Reactive ACKR3 61 31 C[C@@H]1CCC[C@H](NC(=O)CC2(CN)CCC2)[C@@H]1C ZINC000147481682 CE For-Sale Anodyne CACNA2D1 41 39 CCC(CC)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147481697 CG On-Demand Anodyne HCAR1 0 42 Nc1nc(Oc2ccc(Br)cc2F)c2ccccc2n1 ZINC000147481703 EH For-Sale Anodyne FOLA 16 40 Nc1nc(Oc2ccc(Br)cc2F)c2ccccc2n1 ZINC000147481703 EH For-Sale Anodyne AGPAT2 27 40 Cc1ccc(NN)c(C(=O)NCC2(N(C)C)CCCC2)c1 ZINC000147481725 CD For-Sale Anodyne SLC6A5 15 43 Cc1ccc(NN)c(C(=O)NCC2(N(C)C)CCCC2)c1 ZINC000147481725 CD For-Sale Anodyne HCN1 44 35 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne CHRM2 15 46 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne DRD2 33 46 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne FKBP1A 25 45 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne DRD4 48 39 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne ACHE 17 44 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne DRD3 32 43 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne HTR4 58 36 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne F10 22 47 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne CHRM5 15 45 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne GRIN2B 30 43 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne SIGMAR1 16 47 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne MMP13 59 47 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne MMP2 33 47 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne MMP3 58 47 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne MMP8 35 47 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne MMP9 44 47 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne EPHX2 30 44 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne PKM 16 43 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne TGM2 68 46 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne ST14 19 41 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne MMP7 49 47 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne MMP1 54 47 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne MCHR1 21 49 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne GCK 26 40 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne CACNA1I 79 42 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne F13A1 63 44 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne AKR1C3 62 44 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne NAMPT 43 42 COc1cc(OC)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147481773 HF On-Demand Anodyne ACKR3 40 35 O=C(NC1CCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CC1)c1cccs1 ZINC000147481797 GH On-Demand Anodyne NPBWR1 50 33 CN(C)Cc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147481813 FI On-Demand Anodyne F2R 0 41 CN(C)Cc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147481813 FI On-Demand Anodyne CSF1R 20 40 CN(C)Cc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147481813 FI On-Demand Anodyne TAAR1 52 49 CN(C)Cc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147481813 FI On-Demand Anodyne KCNK3 110 43 CN(C)Cc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147481813 FI On-Demand Anodyne KCNK9 60 42 CN(C)Cc1cccc(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147481813 FI On-Demand Anodyne LMGT2 0 41 Nc1ccc(S(=O)(=O)Nc2ccncc2Br)c(F)c1 ZINC000147481819 EE For-Sale Anodyne PTGS1 0 40 Cc1nc(Nc2ccc(OC(C)C)cc2)ccc1C(=O)O ZINC000147481828 CH For-Sale Anodyne AKR1C3 34 45 Cc1nc(Nc2ccc(OC(C)C)cc2)ccc1C(=O)O ZINC000147481828 CH For-Sale Anodyne AKR1C2 77 45 C[C@H]1CCC[C@H](NC(=O)CC2(CN)CCC2)[C@@H]1C ZINC000147481866 CE For-Sale Anodyne CACNA2D1 41 39 COc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1O ZINC000147481878 EG For-Sale Reactive HCRTR1 18 46 COc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1O ZINC000147481878 EG For-Sale Reactive ACKR3 61 31 COC(=O)Cc1csc(CSC2CCCCC2)n1 ZINC000147481912 CG For-Sale Anodyne QRFPR 43 36 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne PPIA 15 45 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne JUN 21 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne ATF1 57 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne CPT1A 43 44 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne CPT2 40 31 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne PYGL 23 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne NFKB1 53 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne KCNMA1 24 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne ALPL 41 35 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne CSF1R 16 46 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne AKR1C3 27 45 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne SHH 54 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne SMO 23 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne Q25615_ONCVO 40 35 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccc2Cl)c1 ZINC000147481916 EJ On-Demand Anodyne KCNK3 40 43 CN(Cc1cscn1)C(=O)NCc1ccccc1[N+](=O)[O-] ZINC000147481961 DE On-Demand Bother COLA 87 36 CN(C)C1(CNC(=O)c2cc(NN)ccn2)CCCC1 ZINC000147481963 CC For-Sale Anodyne SLC6A5 15 44 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCN(C)CC3)cc2)C1 ZINC000147481972 HC On-Demand Anodyne MTOR 19 42 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCN(C)CC3)cc2)C1 ZINC000147481972 HC On-Demand Anodyne EPHX2 15 47 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCN(C)CC3)cc2)C1 ZINC000147481972 HC On-Demand Anodyne CACNA1I 53 34 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCN(C)CC3)cc2)C1 ZINC000147481972 HC On-Demand Anodyne L3MBTL3 52 38 O=C(NC1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1)c1cccs1 ZINC000147481983 GH On-Demand Anodyne NPBWR1 50 33 Cc1cc(C)cc(C(=O)c2ccc(C(F)(F)F)cc2)c1 ZINC000147481986 CJ For-Sale Anodyne SRD5A2 39 63 Cc1cc(C)cc(C(=O)c2ccc(C(F)(F)F)cc2)c1 ZINC000147481986 CJ For-Sale Anodyne ECR 26 43 Cc1cc(C)cc(C(=O)c2ccc(C(F)(F)F)cc2)c1 ZINC000147481986 CJ For-Sale Anodyne CES2 15 43 Cc1cc(C)cc(C(=O)c2ccc(C(F)(F)F)cc2)c1 ZINC000147481986 CJ For-Sale Anodyne E3UJZ5_SPOLI 23 43 Cc1cc(C)cc(C(=O)c2ccc(C(F)(F)F)cc2)c1 ZINC000147481986 CJ For-Sale Anodyne KCNK3 21 40 Cc1nc(Nc2cccc(C(C)C)c2)ccc1C(=O)O ZINC000147482030 CH For-Sale Anodyne AKR1C3 44 41 Cc1nc(Nc2cccc(C(C)C)c2)ccc1C(=O)O ZINC000147482030 CH For-Sale Anodyne AKR1C2 59 41 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne DRD2 18 42 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne HTR4 63 39 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne F10 15 40 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne CHRM5 19 40 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne GRIN2B 32 42 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne LPL 46 37 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne MMP13 15 40 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne EPHX2 39 47 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne TGM2 74 45 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne ITGAV 43 35 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne CACNA1I 82 48 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne F13A1 70 45 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne AKR1C3 60 38 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne SFRP1 29 40 Cc1cc(C)cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c1 ZINC000147482041 GG On-Demand Anodyne NAMPT 46 41 O=C(CCc1ncc(-c2ccc(F)cc2F)o1)NCCCCc1ccccc1 ZINC000147482048 GJ On-Demand Anodyne MTNR1A 16 40 O=C(CCc1ncc(-c2ccc(F)cc2F)o1)NCCCCc1ccccc1 ZINC000147482048 GJ On-Demand Anodyne MTNR1B 17 40 O=C(CCc1ncc(-c2ccc(F)cc2F)o1)NCCCCc1ccccc1 ZINC000147482048 GJ On-Demand Anodyne FAAH 86 47 O=C(CCc1ncc(-c2ccc(F)cc2F)o1)NCCCCc1ccccc1 ZINC000147482048 GJ On-Demand Anodyne CES1 62 47 O=C(CCc1ncc(-c2ccc(F)cc2F)o1)NCCCCc1ccccc1 ZINC000147482048 GJ On-Demand Anodyne CES1D 61 37 CC[C@@H](CN)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147482071 CE For-Sale Bother CACNA1C 54 38 CC[C@@H](CN)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147482071 CE For-Sale Bother CACNA1D 86 36 COc1ccc(NC(C)=O)cc1S(=O)(=O)NCc1c(C)noc1C ZINC000147482075 FD On-Demand Anodyne TSHR 40 30 COc1ccc(NC(C)=O)cc1S(=O)(=O)NCc1c(C)noc1C ZINC000147482075 FD On-Demand Anodyne BRD3 18 43 C[C@@H]1CCC[C@@H](NC(=O)CC2(CN)CCC2)[C@@H]1C ZINC000147482084 CE For-Sale Anodyne CACNA2D1 41 39 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne AVPR2 25 41 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne AVPR1A 15 41 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne JUN 22 45 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne ATF1 58 40 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne NR1H4 21 47 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne NFKB1 54 40 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne CSF1R 15 42 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne BTK 25 41 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne AKR1C3 28 41 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne KCNK3 78 46 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne KCNK9 59 46 Cc1ccc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482141 DH On-Demand Anodyne TMPRSS4 0 44 Cc1c(N)ncnc1Oc1ccc(Br)cc1F ZINC000147482166 CG For-Sale Anodyne TRPA1 0 47 CN(C)C1(CNC(=O)c2cccc(F)c2NN)CCCC1 ZINC000147482170 CD For-Sale Anodyne HCN1 69 36 CN(C)C1(CNC(=O)c2cccc(F)c2NN)CCCC1 ZINC000147482170 CD For-Sale Anodyne HCN4 51 34 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCN(C)CC3)cc2)C1 ZINC000147482177 HC On-Demand Anodyne MTOR 19 42 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCN(C)CC3)cc2)C1 ZINC000147482177 HC On-Demand Anodyne EPHX2 15 47 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCN(C)CC3)cc2)C1 ZINC000147482177 HC On-Demand Anodyne CACNA1I 53 34 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCN(C)CC3)cc2)C1 ZINC000147482177 HC On-Demand Anodyne L3MBTL3 52 38 O=C(NC1CCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CC1)c1cccs1 ZINC000147482192 GH On-Demand Anodyne NPBWR1 50 33 CCCOc1cccc(NC(=O)c2cc(C)ccc2Br)c1 ZINC000147482209 EJ On-Demand Anodyne F2R 0 66 CCCOc1cccc(NC(=O)c2cc(C)ccc2Br)c1 ZINC000147482209 EJ On-Demand Anodyne F12 0 41 CCCOc1cccc(NC(=O)c2cc(C)ccc2Br)c1 ZINC000147482209 EJ On-Demand Anodyne SCN10A 25 40 CCCOc1cccc(NC(=O)c2cc(C)ccc2Br)c1 ZINC000147482209 EJ On-Demand Anodyne TAAR1 37 42 CCCOc1cccc(NC(=O)c2cc(C)ccc2Br)c1 ZINC000147482209 EJ On-Demand Anodyne KCNK3 110 47 CCCOc1cccc(NC(=O)c2cc(C)ccc2Br)c1 ZINC000147482209 EJ On-Demand Anodyne KCNK9 89 47 Nc1ccc2c(S(=O)(=O)Nc3ccncc3Br)c[nH]c2c1 ZINC000147482238 FF For-Sale Anodyne SGK1 44 32 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(C(F)(F)F)cc1 ZINC000147482240 EI On-Demand Anodyne CYP3A4 15 44 CC[C@H](CN)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147482249 CE For-Sale Bother CACNA1C 54 38 CC[C@H](CN)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147482249 CE For-Sale Bother CACNA1D 86 36 C[C@H]1CCC[C@@H](NC(=O)CC2(CN)CCC2)[C@@H]1C ZINC000147482257 CE For-Sale Anodyne CACNA2D1 41 39 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne ACHE 15 44 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne HTR4 56 37 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne KCNQ2 15 40 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne SIGMAR1 28 59 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne APP 57 42 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne MMP2 17 42 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne CCR2 16 41 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne EPHX2 32 45 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne TGM2 80 48 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne CXCR3 21 45 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne CA9 15 43 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne PTGDR2 15 45 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne CACNA1I 71 45 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne F13A1 84 48 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne AKR1C3 22 41 O=C(Cc1ccc(Cl)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482275 HG On-Demand Anodyne NAMPT 53 40 NC(=O)[C@@H]1CCCCc2ccccc21 ZINC000147482301 AD For-Sale Anodyne TSPAN17 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne PPARA 0 47 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne PPIA 19 53 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne UL80 16 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne CPT1A 35 45 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne PRNP 22 50 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne CSF1R 17 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne LUCI_LUCLA 16 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne TAAR1 37 47 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne AKR1C3 41 50 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne HCAR1 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne SENP1 0 52 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne KCNK3 107 55 O=C(O)c1cc(Cl)cc(NC(=O)c2cccc(Br)c2)c1 ZINC000147482347 FI On-Demand Anodyne KCNK9 53 48 CN(C)C(=O)NCCNC(=O)c1cc(Cl)ccc1NN ZINC000147482354 CC For-Sale Anodyne F10 31 44 CCN(Cc1ccccc1)c1ccc(C(=O)O)c(C)n1 ZINC000147482426 CG For-Sale Anodyne TSPO 22 42 C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(C(F)(F)F)cc1 ZINC000147482448 EI On-Demand Anodyne CYP3A4 15 44 CC[C@@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147482463 CE For-Sale Bother CACNA1C 54 38 CC[C@@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147482463 CE For-Sale Bother CACNA1D 86 36 O=C(CCC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482491 GG On-Demand Anodyne CHRM5 20 45 O=C(CCC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482491 GG On-Demand Anodyne EPHX2 27 51 O=C(CCC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482491 GG On-Demand Anodyne TGM2 88 48 O=C(CCC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482491 GG On-Demand Anodyne CACNA1I 53 36 O=C(CCC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482491 GG On-Demand Anodyne F13A1 91 48 O=C(CCC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482491 GG On-Demand Anodyne AKR1C3 60 39 O=C(CCC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482491 GG On-Demand Anodyne SFRP1 45 39 O=C(CCC1CCCC1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482491 GG On-Demand Anodyne NAMPT 32 41 CC(C)CCCCNC[C@H](O)COc1ccc(C#N)cc1 ZINC000147482516 CF For-Sale Mild ADRB2 61 46 CC(C)CCCCNC[C@H](O)COc1ccc(C#N)cc1 ZINC000147482516 CF For-Sale Mild ADRB1 76 48 CC(C)CCCCNC[C@H](O)COc1ccc(C#N)cc1 ZINC000147482516 CF For-Sale Mild ADRB3 52 48 CSc1ccc([C@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147482520 FJ On-Demand Anodyne SDH1 0 46 NC(=O)[C@H]1CCCCc2ccccc21 ZINC000147482544 AD For-Sale Anodyne TSPAN17 0 42 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne PPIA 18 52 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne KCNJ11 15 41 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne ECR 33 44 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne CTSL 18 41 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne CPT1A 55 42 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne PRNP 27 49 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne PPARD 23 40 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne NR1H4 0 46 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne GRM5 17 48 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne F12 0 40 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne SCN10A 39 40 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne CSF1R 25 48 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne LUCI_LUCLA 16 40 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne TAAR1 40 46 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne AKR1C3 46 49 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne DDR1 23 44 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne GPR35 23 52 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne KCNK3 139 68 Cc1cccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147482562 CH On-Demand Anodyne KCNK9 78 68 N#CCNC(=O)Cc1nnc(Cc2ccc(-c3ccccc3)cn2)o1 ZINC000147482671 ED Annotated Mild CTSK 27 40 N#CCNC(=O)Cc1nnc(Cc2ccc(-c3ccccc3)cn2)o1 ZINC000147482671 ED Annotated Mild CTSS 32 40 N#CCNC(=O)Cc1nnc(Cc2ccc(-c3ccccc3)cn2)o1 ZINC000147482671 ED Annotated Mild CTSV 46 34 CC[C@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147482675 CE For-Sale Bother CACNA1C 54 38 CC[C@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147482675 CE For-Sale Bother CACNA1D 86 36 CC(C)CCCCNC[C@@H](O)COc1ccc(C#N)cc1 ZINC000147482722 CF For-Sale Mild ADRB2 61 46 CC(C)CCCCNC[C@@H](O)COc1ccc(C#N)cc1 ZINC000147482722 CF For-Sale Mild ADRB1 76 48 CC(C)CCCCNC[C@@H](O)COc1ccc(C#N)cc1 ZINC000147482722 CF For-Sale Mild ADRB3 52 48 CSc1ccc([C@@H](C)NC(=O)c2cc(C)ccc2Br)cc1 ZINC000147482741 FJ On-Demand Anodyne SDH1 0 46 CCN(C(=O)CC1(CN)CCC1)C1CCCCC1 ZINC000147482751 CF For-Sale Anodyne CACNA2D1 53 45 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne DRD2 17 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne DRD4 41 33 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne HTR4 55 37 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne F10 18 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne GRIN2B 28 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne CCR3 45 39 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne CCR2 41 41 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne EPHX2 28 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne TGM2 71 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne CACNA1I 71 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne F13A1 67 44 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne AKR1C3 62 43 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne SFRP1 49 42 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne NAMPT 40 40 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne ACKR3 57 34 O=C(NCC1CCN(S(=O)(=O)c2ccccc2)CC1)c1cccc(F)c1 ZINC000147482758 GF On-Demand Anodyne KCNK3 15 42 CCC[C@@H](C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147482778 CG On-Demand Anodyne CCKBR 46 37 Cc1nc(Nc2ccc(OC(F)F)cc2)ccc1C(=O)O ZINC000147482779 CG For-Sale Anodyne AKR1C3 30 44 Cc1nc(Nc2ccc(OC(F)F)cc2)ccc1C(=O)O ZINC000147482779 CG For-Sale Anodyne AKR1C2 69 44 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(CCN3CCCCC3)cc2)C1 ZINC000147482810 HF On-Demand Anodyne HTR4 45 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(CCN3CCCCC3)cc2)C1 ZINC000147482810 HF On-Demand Anodyne HRH3 21 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(CCN3CCCCC3)cc2)C1 ZINC000147482810 HF On-Demand Anodyne CCR3 67 46 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(CCN3CCCCC3)cc2)C1 ZINC000147482810 HF On-Demand Anodyne CACNA1I 41 38 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(CCN3CCCCC3)cc2)C1 ZINC000147482810 HF On-Demand Anodyne BIRC2 66 37 COc1cc(Br)c(N)cc1S(=O)(=O)Nc1ccncc1Br ZINC000147482883 IF For-Sale Anodyne ALPL 26 42 CC[C@](C)(N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147482902 CE For-Sale Bother CACNA1C 43 38 CC[C@](C)(N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147482902 CE For-Sale Bother CACNA1D 66 34 CCC[C@H](C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147482963 CG On-Demand Anodyne CCKBR 46 37 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne SLC6A3 16 43 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne HTR4 53 35 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne GRIN2B 51 42 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne SIGMAR1 29 47 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne MMP13 20 42 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne CCR3 71 45 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne MMP3 22 40 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne MMP8 18 40 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne EPHX2 25 45 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne TGM2 80 48 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne CACNA1I 56 45 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne F13A1 85 48 O=C(Cc1ccc(F)cc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147482964 GF On-Demand Anodyne NAMPT 58 41 NCC1(CC(=O)Nc2cccc(Cl)c2)CCC1 ZINC000147482986 CF For-Sale Anodyne NADD 0 41 Cc1nc(Nc2ccccc2OC(F)F)ccc1C(=O)O ZINC000147482995 CG For-Sale Anodyne AKR1C2 46 37 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(CCN3CCCCC3)cc2)C1 ZINC000147483033 HF On-Demand Anodyne HTR4 45 40 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(CCN3CCCCC3)cc2)C1 ZINC000147483033 HF On-Demand Anodyne HRH3 21 40 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(CCN3CCCCC3)cc2)C1 ZINC000147483033 HF On-Demand Anodyne CCR3 67 46 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(CCN3CCCCC3)cc2)C1 ZINC000147483033 HF On-Demand Anodyne CACNA1I 41 38 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(CCN3CCCCC3)cc2)C1 ZINC000147483033 HF On-Demand Anodyne BIRC2 66 37 COC(=O)[C@H](Br)COCc1ccc(Br)cc1 ZINC000147483088 FF For-Sale Reactive PLM1_PLAFA 40 42 COC(=O)[C@H](Br)COCc1ccc(Br)cc1 ZINC000147483088 FF For-Sale Reactive PLM2_PLAFA 17 42 CC[C@@](C)(N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147483113 CE For-Sale Bother CACNA1C 43 38 CC[C@@](C)(N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147483113 CE For-Sale Bother CACNA1D 66 34 CC1(C)c2[nH]nc(Nc3nc(Cl)nc(Cl)n3)c2CN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147483128 JH Annotated Anodyne PAK4 24 43 NCC1(CC(=O)Nc2cccc(F)c2)CCC1 ZINC000147483198 BE For-Sale Anodyne FUCA1 16 45 NCC1(CC(=O)Nc2cccc(F)c2)CCC1 ZINC000147483198 BE For-Sale Anodyne KCNK3 15 40 Cc1nc(NCCCN2CCOCC2)ccc1C(=O)O ZINC000147483240 CD For-Sale Anodyne CNR1 22 41 Cc1nc(NCCCN2CCOCC2)ccc1C(=O)O ZINC000147483240 CD For-Sale Anodyne CNR2 0 44 Cc1nc(NCCCN2CCOCC2)ccc1C(=O)O ZINC000147483240 CD For-Sale Anodyne CASR 49 38 Cc1nc(NCCCN2CCOCC2)ccc1C(=O)O ZINC000147483240 CD For-Sale Anodyne FGFR1 15 43 Cc1nc(NCCCN2CCOCC2)ccc1C(=O)O ZINC000147483240 CD For-Sale Anodyne CHRNA7 17 42 Cc1nc(NCCCN2CCOCC2)ccc1C(=O)O ZINC000147483240 CD For-Sale Anodyne PTGDS 42 37 Cc1nc(NCCCN2CCOCC2)ccc1C(=O)O ZINC000147483240 CD For-Sale Anodyne EPHX2 19 40 Cc1nc(NCCCN2CCOCC2)ccc1C(=O)O ZINC000147483240 CD For-Sale Anodyne TLR9 0 40 O=C(Cc1ccsc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147483283 GF On-Demand Anodyne EPHX2 16 43 O=C(Cc1ccsc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147483283 GF On-Demand Anodyne TGM2 74 48 O=C(Cc1ccsc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147483283 GF On-Demand Anodyne F13A1 78 48 O=C(Cc1ccsc1)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147483283 GF On-Demand Anodyne TGM6 0 40 COC(=O)[C@@H](Br)COCc1ccc(Br)cc1 ZINC000147483316 FF For-Sale Reactive PLM1_PLAFA 40 42 COC(=O)[C@@H](Br)COCc1ccc(Br)cc1 ZINC000147483316 FF For-Sale Reactive PLM2_PLAFA 17 42 Nc1cc(S(=O)(=O)Nc2ccncc2Br)ccc1Cl ZINC000147483325 FF For-Sale Anodyne CCR2 0 47 CC(=O)N1CCc2cc(N[C@@H]3CCO[C@@H]3C)ccc21 ZINC000147483333 CE For-Sale Anodyne HSD17B3 46 34 CC[C@](C)(N)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147483340 CE For-Sale Bother CACNA1C 43 38 CC[C@](C)(N)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147483340 CE For-Sale Bother CACNA1D 66 34 CC1(C)c2[nH]nc(Nc3nc(Cl)nc(Cl)n3)c2CN1C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147483347 JH Annotated Anodyne PAK4 24 43 NCC1(CC(=O)Nc2ccc(Cl)cc2)CCC1 ZINC000147483402 CF For-Sale Anodyne CACNA2D1 0 42 Cc1ccc(F)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147483411 DH On-Demand Anodyne JUN 23 44 Cc1ccc(F)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147483411 DH On-Demand Anodyne ATF1 61 42 Cc1ccc(F)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147483411 DH On-Demand Anodyne NR1H4 17 42 Cc1ccc(F)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147483411 DH On-Demand Anodyne NFKB1 56 42 Cc1ccc(F)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147483411 DH On-Demand Anodyne KCNK3 84 42 Cc1ccc(F)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147483411 DH On-Demand Anodyne KCNK9 58 42 Cc1ccc(F)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c1 ZINC000147483411 DH On-Demand Anodyne TMPRSS4 0 49 COC(=O)c1c(Cl)cncc1OCc1ccccc1 ZINC000147483483 CG For-Sale Anodyne PPIA 47 37 COC(=O)c1c(Cl)cncc1OCc1ccccc1 ZINC000147483483 CG For-Sale Anodyne ERBB2 15 43 COC(=O)c1c(Cl)cncc1OCc1ccccc1 ZINC000147483483 CG For-Sale Anodyne PTGER1 57 41 COC(=O)c1c(Cl)cncc1OCc1ccccc1 ZINC000147483483 CG For-Sale Anodyne PDE4D 17 49 O=C(c1ccc2c(c1)CCO2)N1CCC[C@@H]1CCCBr ZINC000147483493 EG For-Sale Reactive GPR183 0 45 CC[C@@](C)(N)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147483518 CE For-Sale Bother CACNA1C 43 38 CC[C@@](C)(N)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147483518 CE For-Sale Bother CACNA1D 66 34 CC(=O)N1CCc2cc(N[C@@H]3CCO[C@H]3C)ccc21 ZINC000147483519 CE For-Sale Anodyne HSD17B3 46 34 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne DRD2 53 47 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne FKBP1A 38 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne DRD4 42 34 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne ACHE 28 53 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne DRD3 48 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne HTR4 67 39 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne CYSLTR1 32 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne F10 25 50 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne GRIN2B 31 42 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne SIGMAR1 16 45 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne PDE4D 15 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne CPT1A 73 36 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne CPT2 48 35 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne SLC9A1 56 31 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne EPHX2 26 50 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne TGM2 67 53 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne CPT1B 49 34 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne MCHR1 23 45 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne CACNA1I 68 44 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne F13A1 61 43 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne AKR1C3 48 40 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne SFRP1 20 40 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne NAMPT 43 43 COc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)cc1OC ZINC000147483546 HF On-Demand Anodyne ACKR3 77 42 CC(C)CCCCNCc1ncccn1 ZINC000147483635 BE For-Sale Anodyne FDFT1 0 42 O=C(c1ccc2c(c1)CCO2)N1CCC[C@H]1CCCBr ZINC000147483663 EG For-Sale Reactive GPR183 0 45 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2F)c1 ZINC000147483664 FI On-Demand Anodyne PPIA 15 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2F)c1 ZINC000147483664 FI On-Demand Anodyne ATF1 55 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2F)c1 ZINC000147483664 FI On-Demand Anodyne NFKB1 51 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2F)c1 ZINC000147483664 FI On-Demand Anodyne AKR1C3 17 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2F)c1 ZINC000147483664 FI On-Demand Anodyne GPR35 53 35 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Br)ccc2F)c1 ZINC000147483664 FI On-Demand Anodyne TMPRSS4 0 43 CC(=O)N1CCc2cc(N[C@H]3CCO[C@@H]3C)ccc21 ZINC000147483689 CE For-Sale Anodyne HSD17B3 46 34 C[C@@H](CCN)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147483721 CE For-Sale Bother CACNA1C 44 37 C[C@@H](CCN)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147483721 CE For-Sale Bother CACNA1D 73 37 CC1(C)c2[nH]nc(Nc3nc(Cl)nc4ccccc34)c2CN1C(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147483739 JK Annotated Anodyne PAK4 19 40 Cc1cc(N)c(C(=O)O)cc1Cl ZINC000147483766 AD For-Sale Anodyne AKR1C2 51 39 Cc1cc(N)c(C(=O)O)cc1Cl ZINC000147483766 AD For-Sale Anodyne AKR1C1 51 39 Cc1cc(N)c(C(=O)O)cc1Cl ZINC000147483766 AD For-Sale Anodyne HAAO 43 35 CC[C@@H]1CN(CC(=O)Nc2ccccc2OC)CC[C@@H]1N ZINC000147483775 CD On-Demand Anodyne DRD4 26 48 N#Cc1ccccc1NC(=O)CC1(CN)CCC1 ZINC000147483778 BE For-Sale Mild CACNA2D1 23 40 O=C(C(=O)N1CCN(c2ncnc3sccc23)CC1)c1ccc2c(c1)CCC2 ZINC000147483781 GF On-Demand Anodyne PDGFRB 44 34 CC(C)Oc1ccc(CNC(=O)N(C)Cc2cscn2)cc1 ZINC000147483786 DG On-Demand Anodyne BMP1 43 36 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne AVPR2 24 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne PPIA 15 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne ATF1 56 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne CPT1A 45 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne CPT2 43 34 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne PYGL 29 54 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne SLC6A9 26 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne NFKB1 52 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne AKR1C3 21 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne SMO 25 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne GPR35 27 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2Cl)c1 ZINC000147483852 EJ On-Demand Anodyne KCNK3 31 44 Cc1noc(C)c1CNS(=O)(=O)c1cccc(F)c1 ZINC000147483877 CD On-Demand Anodyne EDNRA 23 42 CC(C)(C(=O)N1CCC[C@@H]1CCCBr)c1ccccc1 ZINC000147483880 EI For-Sale Reactive CHRM4 15 44 CC(C)(C(=O)N1CCC[C@@H]1CCCBr)c1ccccc1 ZINC000147483880 EI For-Sale Reactive CHRM5 15 44 CC(C)(C(=O)N1CCC[C@@H]1CCCBr)c1ccccc1 ZINC000147483880 EI For-Sale Reactive CHRM3 38 44 CC(C)(C(=O)N1CCC[C@@H]1CCCBr)c1ccccc1 ZINC000147483880 EI For-Sale Reactive PREP 49 34 CC(C)(C(=O)N1CCC[C@@H]1CCCBr)c1ccccc1 ZINC000147483880 EI For-Sale Reactive AMY2 51 35 CC(C)(C(=O)N1CCC[C@@H]1CCCBr)c1ccccc1 ZINC000147483880 EI For-Sale Reactive CYP2J2 47 35 N#Cc1ccccc1N[C@@H](CC(=O)O)C(=O)O ZINC000147483897 BC For-Sale Mild MME 39 40 N#Cc1ccccc1N[C@@H](CC(=O)O)C(=O)O ZINC000147483897 BC For-Sale Mild ACE2 40 34 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)c1 ZINC000147483901 GG On-Demand Anodyne DRD2 20 40 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)c1 ZINC000147483901 GG On-Demand Anodyne HTR4 63 38 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)c1 ZINC000147483901 GG On-Demand Anodyne SLC6A9 46 35 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)c1 ZINC000147483901 GG On-Demand Anodyne EPHX2 39 48 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)c1 ZINC000147483901 GG On-Demand Anodyne TGM2 64 43 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)c1 ZINC000147483901 GG On-Demand Anodyne CACNA1I 62 41 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)c1 ZINC000147483901 GG On-Demand Anodyne F13A1 60 43 Cc1ccc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3)CC2)c(C)c1 ZINC000147483901 GG On-Demand Anodyne CCR8 53 31 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](C)CCN ZINC000147483903 CE For-Sale Bother CACNA1C 44 37 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](C)CCN ZINC000147483903 CE For-Sale Bother CACNA1D 73 37 CC(=O)N1CCc2cc(N[C@H]3CCO[C@H]3C)ccc21 ZINC000147483926 CE For-Sale Anodyne HSD17B3 46 34 Nc1cc(Br)ccc1S(=O)(=O)Nc1ccncc1Br ZINC000147483940 HF For-Sale Anodyne PTGS1 0 40 CC(C)(C)NS(=O)(=O)C[C@H](C1CC1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147483958 KK Annotated Anodyne TP53 42 62 CC(C)(C)NS(=O)(=O)C[C@H](C1CC1)N1C(=O)[C@@](C)(CC(=O)O)C[C@H](c2cccc(Cl)c2)[C@H]1c1ccc(Cl)cc1 ZINC000147483958 KK Annotated Anodyne MDM2 261 87 COc1cccc(-c2cnc(Cl)o2)c1 ZINC000147483970 BG For-Sale Anodyne TUBB2B 24 43 COc1cccc(-c2cnc(Cl)o2)c1 ZINC000147483970 BG For-Sale Anodyne TUBA1A 23 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCC(C)CC3)cc2)C1 ZINC000147483994 HE On-Demand Anodyne EPHX2 16 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCC(C)CC3)cc2)C1 ZINC000147483994 HE On-Demand Anodyne CACNA1I 45 33 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCC(C)CC3)cc2)C1 ZINC000147483994 HE On-Demand Anodyne L3MBTL3 55 36 CC[C@H]1CN(CC(=O)Nc2ccccc2OC)CC[C@@H]1N ZINC000147484005 CD On-Demand Anodyne DRD4 26 48 N#Cc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147484009 BE For-Sale Mild MCHR1 40 42 CCCCCCCCOc1ccc(C=O)nc1 ZINC000147484027 BH For-Sale Mild THRA 65 40 CCCCCCCCOc1ccc(C=O)nc1 ZINC000147484027 BH For-Sale Mild THRB 43 40 CCCCCCCCOc1ccc(C=O)nc1 ZINC000147484027 BH For-Sale Mild LPAR2 25 40 CCCCCCCCOc1ccc(C=O)nc1 ZINC000147484027 BH For-Sale Mild S1PR3 24 40 CCCCCCCCOc1ccc(C=O)nc1 ZINC000147484027 BH For-Sale Mild PLA2G4B 97 42 CCCCCCCCOc1ccc(C=O)nc1 ZINC000147484027 BH For-Sale Mild S1PR2 25 40 CCCCCCCCOc1ccc(C=O)nc1 ZINC000147484027 BH For-Sale Mild CYP2C19 17 40 O=C(CSc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484082 DH On-Demand Anodyne PPIA 15 43 O=C(CSc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484082 DH On-Demand Anodyne AKR1C3 16 41 O=C(CSc1ccccc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484082 DH On-Demand Anodyne FAS 66 44 CC(C)(C(=O)N1CCC[C@H]1CCCBr)c1ccccc1 ZINC000147484089 EI For-Sale Reactive CHRM4 15 44 CC(C)(C(=O)N1CCC[C@H]1CCCBr)c1ccccc1 ZINC000147484089 EI For-Sale Reactive CHRM5 15 44 CC(C)(C(=O)N1CCC[C@H]1CCCBr)c1ccccc1 ZINC000147484089 EI For-Sale Reactive CHRM3 38 44 CC(C)(C(=O)N1CCC[C@H]1CCCBr)c1ccccc1 ZINC000147484089 EI For-Sale Reactive PREP 49 34 CC(C)(C(=O)N1CCC[C@H]1CCCBr)c1ccccc1 ZINC000147484089 EI For-Sale Reactive AMY2 51 35 CC(C)(C(=O)N1CCC[C@H]1CCCBr)c1ccccc1 ZINC000147484089 EI For-Sale Reactive CYP2J2 47 35 C[C@@H](CCN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147484094 CE For-Sale Bother CACNA1C 44 37 C[C@@H](CCN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147484094 CE For-Sale Bother CACNA1D 73 37 COC(=O)N(C)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147484155 FG On-Demand Anodyne MTNR1A 23 48 COC(=O)N(C)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147484155 FG On-Demand Anodyne MTNR1B 15 48 COC(=O)N(C)c1ccc(NC(=O)[C@@H]2COc3cc(OC)ccc3C2)cc1 ZINC000147484155 FG On-Demand Anodyne ROCK2 34 55 OCC[C@@H]1NCc2ccccc21 ZINC000147484175 AD In-Stock Anodyne PRCP 51 40 CSc1nc(N)nc(NC2CC2)n1 ZINC000147484179 AC For-Sale Anodyne ERM 0 66 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCC(C)CC3)cc2)C1 ZINC000147484195 HE On-Demand Anodyne EPHX2 16 40 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCC(C)CC3)cc2)C1 ZINC000147484195 HE On-Demand Anodyne CACNA1I 45 33 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCC(C)CC3)cc2)C1 ZINC000147484195 HE On-Demand Anodyne L3MBTL3 55 36 C[C@H](CCN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147484316 CE For-Sale Bother CACNA1C 44 37 C[C@H](CCN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147484316 CE For-Sale Bother CACNA1D 73 37 C[C@@H](CCC(=O)O)OCc1ccc(Br)cc1 ZINC000147484327 CG For-Sale Anodyne FOLH1 19 40 C[C@@H](CCC(=O)O)OCc1ccc(Br)cc1 ZINC000147484327 CG For-Sale Anodyne FFAR1 24 50 C[C@@H](CCC(=O)O)OCc1ccc(Br)cc1 ZINC000147484327 CG For-Sale Anodyne FFAR4 25 40 CC(C)c1n[nH]c2c(=O)[nH]c(Cc3cccc(OC(F)(F)F)c3)nc12 ZINC000147484337 FG For-Sale Anodyne PDE1C 21 71 CC(C)c1n[nH]c2c(=O)[nH]c(Cc3cccc(OC(F)(F)F)c3)nc12 ZINC000147484337 FG For-Sale Anodyne HAO2 18 47 OCC[C@H]1NCc2ccccc21 ZINC000147484360 AD In-Stock Anodyne PRCP 51 40 COc1ccc(C)cc1C1(CNC(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CCOCC1 ZINC000147484363 HJ On-Demand Anodyne MDM2 62 33 COCc1nc(C(=O)N2CCCCC[C@@H]2c2ccc(OC)cc2)cs1 ZINC000147484435 FI On-Demand Anodyne CPT1A 74 41 COCc1nc(C(=O)N2CCCCC[C@@H]2c2ccc(OC)cc2)cs1 ZINC000147484435 FI On-Demand Anodyne TRPC6 42 40 COCc1nc(C(=O)N2CCCCC[C@@H]2c2ccc(OC)cc2)cs1 ZINC000147484435 FI On-Demand Anodyne TRPC3 34 40 CCCCc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147484478 CI For-Sale Anodyne MPL 16 41 CCCCc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147484478 CI For-Sale Anodyne RARB 15 43 CCCCc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147484478 CI For-Sale Anodyne AGTR1B 54 36 CCCCc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147484478 CI For-Sale Anodyne AKR1C2 48 35 Cc1ccc(F)cc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484496 DH On-Demand Anodyne AVPR2 32 44 Cc1ccc(F)cc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484496 DH On-Demand Anodyne AVPR1A 19 55 Cc1ccc(F)cc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484496 DH On-Demand Anodyne JUN 22 40 Cc1ccc(F)cc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484496 DH On-Demand Anodyne ATF1 56 39 Cc1ccc(F)cc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484496 DH On-Demand Anodyne NR1H4 17 41 Cc1ccc(F)cc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484496 DH On-Demand Anodyne NFKB1 52 39 Cc1ccc(F)cc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484496 DH On-Demand Anodyne BTK 26 41 Cc1ccc(F)cc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484496 DH On-Demand Anodyne AKR1C3 15 40 Cc1ccc(F)cc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484496 DH On-Demand Anodyne KCNK3 69 39 Cc1ccc(F)cc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484496 DH On-Demand Anodyne KCNK9 58 38 Cc1ccc(F)cc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484496 DH On-Demand Anodyne TMPRSS4 0 48 O=C(NCCN1CCCC1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147484522 FE For-Sale Anodyne CACNA1H 26 41 O=C(NCCN1CCCC1)Nc1cc(Br)cc(C(=O)O)c1 ZINC000147484522 FE For-Sale Anodyne CCR3 36 40 CC[C@@H](C)[C@H](N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147484531 CE For-Sale Bother CACNA1C 57 40 CC[C@@H](C)[C@H](N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147484531 CE For-Sale Bother CACNA1D 89 37 NCC1(CC(=O)Nc2ccc(Br)cc2)CCC1 ZINC000147484544 CF For-Sale Anodyne CACNA2D1 0 42 C[C@H](CCC(=O)O)OCc1ccc(Br)cc1 ZINC000147484549 CG For-Sale Anodyne FOLH1 19 40 C[C@H](CCC(=O)O)OCc1ccc(Br)cc1 ZINC000147484549 CG For-Sale Anodyne FFAR1 24 50 C[C@H](CCC(=O)O)OCc1ccc(Br)cc1 ZINC000147484549 CG For-Sale Anodyne FFAR4 25 40 COc1ccc(C)cc1C1(CNC(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CCOCC1 ZINC000147484556 HJ On-Demand Anodyne MDM2 62 33 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(OC(F)F)c3ncccc23)C1 ZINC000147484579 HF On-Demand Anodyne HTR4 45 39 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(OC(F)F)c3ncccc23)C1 ZINC000147484579 HF On-Demand Anodyne CACNA1I 40 31 COCc1nc(C(=O)N2CCCCC[C@H]2c2ccc(OC)cc2)cs1 ZINC000147484653 FI On-Demand Anodyne CPT1A 74 41 COCc1nc(C(=O)N2CCCCC[C@H]2c2ccc(OC)cc2)cs1 ZINC000147484653 FI On-Demand Anodyne TRPC6 42 40 COCc1nc(C(=O)N2CCCCC[C@H]2c2ccc(OC)cc2)cs1 ZINC000147484653 FI On-Demand Anodyne TRPC3 34 40 Cc1cc(N2CCC(C(=O)O)CC2)ccc1C(N)=O ZINC000147484667 CD For-Sale Anodyne SLC6A1 56 37 CCCc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147484678 CH For-Sale Anodyne PDE4B 0 42 CCCc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147484678 CH For-Sale Anodyne PDE4D 0 42 CCCc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1 ZINC000147484678 CH For-Sale Anodyne AKR1C2 59 37 COc1ccc(C)cc1C1(CNC(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CCOCC1 ZINC000147484758 HJ On-Demand Anodyne MDM2 62 33 CCN1CCC[C@H]1C(C)=O ZINC000147484760 AD For-Sale Anodyne HSD11B1 43 35 O=C(NCCN1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484761 DE For-Sale Anodyne CACNA1H 34 54 O=C(NCCN1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484761 DE For-Sale Anodyne DRD4 43 34 O=C(NCCN1CCCC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484761 DE For-Sale Anodyne CACNA1I 54 42 NCC1(CC(=O)Nc2cccc(Br)c2)CCC1 ZINC000147484776 CF For-Sale Anodyne EGFR 64 43 NCC1(CC(=O)Nc2cccc(Br)c2)CCC1 ZINC000147484776 CF For-Sale Anodyne NADD 0 41 NCC1(CC(=O)Nc2cccc(Br)c2)CCC1 ZINC000147484776 CF For-Sale Anodyne PARP10 0 41 CC[C@@H](C)[C@@H](N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147484785 CE For-Sale Bother CACNA1C 57 40 CC[C@@H](C)[C@@H](N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147484785 CE For-Sale Bother CACNA1D 89 37 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(OC(F)F)c3ncccc23)C1 ZINC000147484818 HF On-Demand Anodyne HTR4 45 39 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(OC(F)F)c3ncccc23)C1 ZINC000147484818 HF On-Demand Anodyne CACNA1I 40 31 COC(=O)c1cc(C(F)(F)F)cc(C)c1Cl ZINC000147484855 CG For-Sale Anodyne JUN 22 41 COC(=O)c1cc(C(F)(F)F)cc(C)c1Cl ZINC000147484855 CG For-Sale Anodyne ATF1 56 37 COC(=O)c1cc(C(F)(F)F)cc(C)c1Cl ZINC000147484855 CG For-Sale Anodyne NFKB1 52 37 Nc1cccc(S(=O)(=O)Nc2ccncc2Br)c1 ZINC000147484857 EE For-Sale Anodyne Q5TU56_ANOGA 0 45 Nc1nc(Br)cc(N2CCOCC2)n1 ZINC000147484860 CC For-Sale Anodyne HRH4 43 64 Nc1nc(Br)cc(N2CCOCC2)n1 ZINC000147484860 CC For-Sale Anodyne PIK3CA 15 48 Cc1nn(-c2ccc(Cl)cc2Cl)c(Cl)c1S(=O)(=O)Cl ZINC000147484867 FI For-Sale Unstable CNR1 66 40 O=C(Cc1ccccc1F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147484921 GF On-Demand Anodyne GRIN2B 24 44 O=C(Cc1ccccc1F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147484921 GF On-Demand Anodyne EPHX2 26 45 O=C(Cc1ccccc1F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147484921 GF On-Demand Anodyne TGM2 77 45 O=C(Cc1ccccc1F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147484921 GF On-Demand Anodyne CACNA1I 53 38 O=C(Cc1ccccc1F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147484921 GF On-Demand Anodyne F13A1 79 45 O=C(Cc1ccccc1F)NCC1CCN(S(=O)(=O)c2ccccc2)CC1 ZINC000147484921 GF On-Demand Anodyne NAMPT 42 52 CC(=O)CC(=O)NCCCCC(C)C ZINC000147484924 AD For-Sale Anodyne DNPEP 43 33 C[C@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147484927 BE For-Sale Bother PGR 0 44 C[C@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147484927 BE For-Sale Bother CACNA1C 54 37 C[C@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147484927 BE For-Sale Bother CACNA1D 83 36 C[C@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147484927 BE For-Sale Bother DDX3X 0 44 C[C@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147484927 BE For-Sale Bother TRPM8 0 42 C[C@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147484927 BE For-Sale Bother OSIGBA0132E09-OSIGBA0108L24.11 0 46 O=C(C[C@H]1CCS(=O)(=O)C1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147484933 ED On-Demand Anodyne CACNA1I 56 37 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1F ZINC000147484937 CF For-Sale Anodyne GALR2 23 44 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1F ZINC000147484937 CF For-Sale Anodyne CSF1R 24 40 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1F ZINC000147484937 CF For-Sale Anodyne AKR1C3 40 42 COc1ccc(Nc2ccc(C(=O)O)c(C)n2)cc1F ZINC000147484937 CF For-Sale Anodyne AKR1C2 81 42 NCC1(CC(=O)Nc2ccc(F)cc2)CCC1 ZINC000147485001 BE For-Sale Anodyne CACNA2D1 0 42 NCC1(CC(=O)Nc2ccc(F)cc2)CCC1 ZINC000147485001 BE For-Sale Anodyne FUCA1 22 41 CC[C@H](C)[C@@H](N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147485014 CE For-Sale Bother CACNA1C 57 40 CC[C@H](C)[C@@H](N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147485014 CE For-Sale Bother CACNA1D 89 37 COc1cc2c(cc1OC)CCN(C(=O)c1cnn(-c3ccccc3Cl)c1)CC2 ZINC000147485027 HH On-Demand Anodyne ABCB1B 48 36 CS(=O)(=O)N1CCC[C@H](NC(=O)NCCN2C(=O)c3ccccc3C2=O)C1 ZINC000147485031 GC On-Demand Anodyne BIRC2 44 33 CN1CCC[C@@H]1c1ncc[nH]1 ZINC000147485056 AD For-Sale Anodyne ADRA1A 21 41 CN1CCC[C@@H]1c1ncc[nH]1 ZINC000147485056 AD For-Sale Anodyne CHRNA2 44 45 CN1CCC[C@@H]1c1ncc[nH]1 ZINC000147485056 AD For-Sale Anodyne CHRNA10 50 35 Nc1cc(S(=O)(=O)Nc2ccncc2Br)ccc1F ZINC000147485058 EE For-Sale Anodyne PTGS1 0 42 Nc1cc(S(=O)(=O)Nc2ccncc2Br)ccc1F ZINC000147485058 EE For-Sale Anodyne CA4 16 47 CCCc1nn(-c2ccc(Cl)cc2Cl)c(Cl)c1S(=O)(=O)Cl ZINC000147485099 GJ For-Sale Unstable CNR1 68 43 CCCc1nn(-c2ccc(Cl)cc2Cl)c(Cl)c1S(=O)(=O)Cl ZINC000147485099 GJ For-Sale Unstable CNR2 30 44 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccccc2Oc2c(C)cccc2C)C1 ZINC000147485112 HH On-Demand Anodyne HTR4 60 37 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccccc2Oc2c(C)cccc2C)C1 ZINC000147485112 HH On-Demand Anodyne CACNA1I 45 32 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1F ZINC000147485118 DH On-Demand Anodyne RARA 29 43 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1F ZINC000147485118 DH On-Demand Anodyne CPT1A 76 43 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1F ZINC000147485118 DH On-Demand Anodyne CPT2 46 36 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1F ZINC000147485118 DH On-Demand Anodyne PRNP 21 41 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1F ZINC000147485118 DH On-Demand Anodyne NR1H4 18 41 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1F ZINC000147485118 DH On-Demand Anodyne TAAR1 34 43 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1F ZINC000147485118 DH On-Demand Anodyne DDR1 37 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1F ZINC000147485118 DH On-Demand Anodyne KCNK3 76 44 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1F ZINC000147485118 DH On-Demand Anodyne KCNK9 39 42 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1F ZINC000147485118 DH On-Demand Anodyne TMPRSS4 0 43 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne FKBP1A 32 45 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne GRIN2B 48 55 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne SIGMAR1 22 40 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne CYSP_TRYCR 40 36 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne C3AR1 42 37 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne PREP 38 40 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne AMY2 44 31 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne TGM2 45 49 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne RHODESAIN 0 41 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne F13A1 51 49 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne CCR8 50 48 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne BIRC2 28 48 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne SFRP1 46 36 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne F1PEP1 0 40 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne WNT3 42 34 CC(C)(O)CNC1CCN(C(=O)OCc2ccccc2)CC1 ZINC000147485121 DE On-Demand Anodyne SLC12A5 67 38 C[C@@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147485153 BE For-Sale Bother PGR 0 44 C[C@@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147485153 BE For-Sale Bother CACNA1C 54 37 C[C@@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147485153 BE For-Sale Bother CACNA1D 83 36 C[C@@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147485153 BE For-Sale Bother DDX3X 0 44 C[C@@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147485153 BE For-Sale Bother TRPM8 0 42 C[C@@H](CNc1cccc([N+](=O)[O-])c1)CC(=O)O ZINC000147485153 BE For-Sale Bother OSIGBA0132E09-OSIGBA0108L24.11 0 46 CCc1ncc(C(=O)NCc2ccc(-c3csc(C)n3)cc2)s1 ZINC000147485181 EI On-Demand Anodyne ROCK1 18 43 CCc1ncc(C(=O)NCc2ccc(-c3csc(C)n3)cc2)s1 ZINC000147485181 EI On-Demand Anodyne ROCK2 18 43 CS(=O)(=O)N1CCC[C@H](NC(=O)Nc2ccc(OC[C@@H]3CCCO3)cc2)C1 ZINC000147485208 GD On-Demand Anodyne EPHX2 50 44 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](N)CC(N)=O ZINC000147485223 CC For-Sale Bother CACNA1C 38 40 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](N)CC(N)=O ZINC000147485223 CC For-Sale Bother CACNA1D 59 34 NCC1(CC(=O)Nc2ccccc2Cl)CCC1 ZINC000147485236 CF For-Sale Anodyne KCNQ2 36 41 NCC1(CC(=O)Nc2ccccc2Cl)CCC1 ZINC000147485236 CF For-Sale Anodyne EPHB3 55 34 CS(=O)(=O)N1CCC[C@@H](NC(=O)NCCN2C(=O)c3ccccc3C2=O)C1 ZINC000147485239 GC On-Demand Anodyne BIRC2 44 33 CC(C)CCCCNC[C@H](O)COc1cc(Cl)ccc1Cl ZINC000147485241 EI For-Sale Anodyne ADRB2 31 44 CC(C)CCCCNC[C@H](O)COc1cc(Cl)ccc1Cl ZINC000147485241 EI For-Sale Anodyne ADRB1 46 38 CC(C)CCCCNC[C@H](O)COc1cc(Cl)ccc1Cl ZINC000147485241 EI For-Sale Anodyne GRIN1 26 41 CN1CCC[C@H]1c1ncc[nH]1 ZINC000147485254 AD For-Sale Anodyne ADRA1A 21 41 CN1CCC[C@H]1c1ncc[nH]1 ZINC000147485254 AD For-Sale Anodyne CHRNA2 29 45 CN1CCC[C@H]1c1ncc[nH]1 ZINC000147485254 AD For-Sale Anodyne CHRNA10 50 35 CC[C@@H]1CN(CC(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147485290 CD For-Sale Anodyne DRD4 0 49 CC[C@@H]1CN(CC(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147485290 CD For-Sale Anodyne CCR3 64 38 CC[C@@H]1CN(CC(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147485290 CD For-Sale Anodyne EPHX2 17 42 CC[C@@H]1CN(CC(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147485290 CD For-Sale Anodyne MCHR1 15 40 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccccc2Oc2c(C)cccc2C)C1 ZINC000147485308 HH On-Demand Anodyne HTR4 60 37 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccccc2Oc2c(C)cccc2C)C1 ZINC000147485308 HH On-Demand Anodyne CACNA1I 45 32 CC(C)c1nn(-c2ccc(Cl)cc2Cl)c(Cl)c1S(=O)(=O)Cl ZINC000147485321 GJ For-Sale Unstable CNR1 50 38 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2F)c1 ZINC000147485330 FI For-Sale Anodyne ATF1 48 39 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2F)c1 ZINC000147485330 FI For-Sale Anodyne CPT1A 23 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2F)c1 ZINC000147485330 FI For-Sale Anodyne NFKB1 44 39 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2F)c1 ZINC000147485330 FI For-Sale Anodyne GPR35 50 38 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Br)cc2F)c1 ZINC000147485330 FI For-Sale Anodyne TMPRSS4 0 43 CN(C)CCCCNC(=O)c1cccnc1Oc1ccc(Nc2ccccn2)cc1 ZINC000147485331 HI Annotated Anodyne POLR1A 32 41 CCNc1cccc(NC2CCN(C)CC2)n1 ZINC000147485337 BE For-Sale Anodyne HTR1F 43 34 CC(C)Oc1ccc(C(=O)N2CCC[C@@H]2CCCBr)cc1 ZINC000147485399 FI For-Sale Reactive HCRTR1 15 46 CS(=O)(=O)N1CCC[C@@H](NC(=O)Nc2ccc(OC[C@@H]3CCCO3)cc2)C1 ZINC000147485444 GD On-Demand Anodyne EPHX2 50 44 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](N)CC(N)=O ZINC000147485446 CC For-Sale Bother CACNA1C 38 40 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](N)CC(N)=O ZINC000147485446 CC For-Sale Bother CACNA1D 59 34 CC(C)CCCCNC[C@@H](O)COc1cc(Cl)ccc1Cl ZINC000147485458 EI For-Sale Anodyne ADRB2 31 44 CC(C)CCCCNC[C@@H](O)COc1cc(Cl)ccc1Cl ZINC000147485458 EI For-Sale Anodyne ADRB1 46 38 CC(C)CCCCNC[C@@H](O)COc1cc(Cl)ccc1Cl ZINC000147485458 EI For-Sale Anodyne GRIN1 26 41 CCOC(=O)CCCCCCc1ccc(O)cc1 ZINC000147485494 CG For-Sale Anodyne INHA 69 33 CCOC(=O)CCCCCCc1ccc(O)cc1 ZINC000147485494 CG For-Sale Anodyne GRIA1 46 35 CCOC(=O)CCCCCCc1ccc(O)cc1 ZINC000147485494 CG For-Sale Anodyne FAAH 47 37 CCOC(=O)CCCCCCc1ccc(O)cc1 ZINC000147485494 CG For-Sale Anodyne S1PR2 47 41 CCOC(=O)CCCCCCc1ccc(O)cc1 ZINC000147485494 CG For-Sale Anodyne CES1 53 37 CCOC(=O)CCCCCCc1ccc(O)cc1 ZINC000147485494 CG For-Sale Anodyne S1PR1 18 41 CCOC(=O)CCCCCCc1ccc(O)cc1 ZINC000147485494 CG For-Sale Anodyne PPO2 21 51 CCOC(=O)CCCCCCc1ccc(O)cc1 ZINC000147485494 CG For-Sale Anodyne AKR1B10 24 40 CC[C@H]1CN(CC(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147485495 CD For-Sale Anodyne DRD4 0 49 CC[C@H]1CN(CC(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147485495 CD For-Sale Anodyne CCR3 64 38 CC[C@H]1CN(CC(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147485495 CD For-Sale Anodyne EPHX2 17 42 CC[C@H]1CN(CC(=O)Nc2ccc(F)cc2)CC[C@@H]1N ZINC000147485495 CD For-Sale Anodyne MCHR1 15 40 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@@H](N3CCCC3)CCC[C@H]21 ZINC000147485503 KJ Annotated Anodyne OPRK1 33 75 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@@H](N3CCCC3)CCC[C@H]21 ZINC000147485503 KJ Annotated Anodyne SIGMAR1 17 65 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@@H](N3CCCC3)CCC[C@H]21 ZINC000147485503 KJ Annotated Anodyne CCR3 51 38 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@@H](N3CCCC3)CCC[C@H]21 ZINC000147485503 KJ Annotated Anodyne L3MBTL3 43 37 CCN1C[C@H](C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1=O ZINC000147485541 DD On-Demand Anodyne INHA 30 53 COCc1nn(-c2ccc(Cl)cc2Cl)c(Cl)c1S(=O)(=O)Cl ZINC000147485562 GH For-Sale Unstable CNR1 44 40 CC(C)Oc1ccc(C(=O)N2CCC[C@H]2CCCBr)cc1 ZINC000147485604 FI For-Sale Reactive HCRTR1 15 46 C=CCNCCCCC(C)C ZINC000147485653 AF For-Sale Mild PAOX 27 41 CCCNC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCN(CCC)C2)cc1Cl ZINC000147485654 HE On-Demand Anodyne HTR4 46 41 CCCNC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCN(CCC)C2)cc1Cl ZINC000147485654 HE On-Demand Anodyne SLC6A9 44 35 CCCNC(=O)c1ccc(NC(=O)C(=O)NC[C@@H]2CCN(CCC)C2)cc1Cl ZINC000147485654 HE On-Demand Anodyne CACNA1I 68 38 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](N)CC(N)=O ZINC000147485667 CC For-Sale Bother CACNA1C 38 40 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](N)CC(N)=O ZINC000147485667 CC For-Sale Bother CACNA1D 59 34 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1ccc(OC[C@@H]2CCCO2)cc1 ZINC000147485670 HH On-Demand Anodyne NOS2 98 36 Cc1cccc(CNC(=O)N(C)Cc2cscn2)c1 ZINC000147485672 CF On-Demand Anodyne BMP1 54 39 O=C(NC1CCN(C(=O)[C@H]2C[C@@H]2c2cccc(Cl)c2)CC1)c1ccsc1 ZINC000147485678 GH On-Demand Anodyne NPBWR1 96 38 NCC1(CC(=O)NCc2ccc(F)cc2)CCC1 ZINC000147485694 CD For-Sale Anodyne CACNA2D1 0 40 NCC1(CC(=O)NCc2ccc(F)cc2)CCC1 ZINC000147485694 CD For-Sale Anodyne TPSAB1 18 44 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@@H](N3CCCC3)CCC[C@@H]21 ZINC000147485699 KJ Annotated Anodyne OPRK1 33 75 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@@H](N3CCCC3)CCC[C@@H]21 ZINC000147485699 KJ Annotated Anodyne SIGMAR1 17 65 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@@H](N3CCCC3)CCC[C@@H]21 ZINC000147485699 KJ Annotated Anodyne CCR3 51 38 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@@H](N3CCCC3)CCC[C@@H]21 ZINC000147485699 KJ Annotated Anodyne L3MBTL3 43 37 COC(=O)Cc1csc(-c2c(F)cccc2F)n1 ZINC000147485701 CF For-Sale Anodyne PIM1 17 40 CCN1C[C@@H](C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1=O ZINC000147485749 DD On-Demand Anodyne INHA 30 53 CS(=O)(=O)N1CCC[C@H](NC(=O)NC2CCN(c3ccccc3)CC2)C1 ZINC000147485753 GD On-Demand Anodyne EPHX2 49 53 C[C@H](CNc1ccc(F)cc1C#N)CC(=O)O ZINC000147485758 BE For-Sale Mild SDH1 0 40 C[C@@H](OCc1ccccc1)C(=O)NCCN1CCCS1(=O)=O ZINC000147485761 EC On-Demand Anodyne CAPN1 43 36 C[C@@H](OCc1ccccc1)C(=O)NCCN1CCCS1(=O)=O ZINC000147485761 EC On-Demand Anodyne CAPN2 69 34 C[C@@H](OCc1ccccc1)C(=O)NCCN1CCCS1(=O)=O ZINC000147485761 EC On-Demand Anodyne NPR 46 34 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485770 ED On-Demand Anodyne NPY1R 24 40 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485770 ED On-Demand Anodyne GRIA1 41 32 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485770 ED On-Demand Anodyne PCSK5 56 35 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485770 ED On-Demand Anodyne FURIN 62 36 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485770 ED On-Demand Anodyne MC1R 47 33 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485770 ED On-Demand Anodyne POLG_WNV 66 32 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485770 ED On-Demand Anodyne NPFFR1 46 31 CCCC[C@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485770 ED On-Demand Anodyne HPN 50 34 CCc1nn(-c2ccc(Cl)cc2Cl)c(Cl)c1S(=O)(=O)Cl ZINC000147485780 FI For-Sale Unstable CNR1 60 39 CCc1nn(-c2ccc(Cl)cc2Cl)c(Cl)c1S(=O)(=O)Cl ZINC000147485780 FI For-Sale Unstable CNR2 25 42 O=C(c1cccc(OC(F)F)c1)N1CCC[C@@H]1CCCBr ZINC000147485810 FI For-Sale Reactive PREP 38 40 CCCNC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCN(CCC)C2)cc1Cl ZINC000147485867 HE On-Demand Anodyne HTR4 46 41 CCCNC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCN(CCC)C2)cc1Cl ZINC000147485867 HE On-Demand Anodyne SLC6A9 44 35 CCCNC(=O)c1ccc(NC(=O)C(=O)NC[C@H]2CCN(CCC)C2)cc1Cl ZINC000147485867 HE On-Demand Anodyne CACNA1I 68 38 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](N)CC(N)=O ZINC000147485869 CC For-Sale Bother CACNA1C 38 40 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](N)CC(N)=O ZINC000147485869 CC For-Sale Bother CACNA1D 59 34 O=C(NCc1ccc(-n2ccnc2)c(F)c1)Nc1ccc(OC[C@H]2CCCO2)cc1 ZINC000147485890 HH On-Demand Anodyne NOS2 98 36 O=C(NC1CCN(C(=O)[C@@H]2C[C@H]2c2cccc(Cl)c2)CC1)c1ccsc1 ZINC000147485892 GH On-Demand Anodyne NPBWR1 96 38 Cc1nc(NCCc2cccc(F)c2)ccc1C(=O)O ZINC000147485909 CF For-Sale Anodyne PTGDR 28 43 Cc1nc(NCCc2cccc(F)c2)ccc1C(=O)O ZINC000147485909 CF For-Sale Anodyne NAMPT 23 41 Cc1nc(NCCc2cccc(F)c2)ccc1C(=O)O ZINC000147485909 CF For-Sale Anodyne HAO2 76 46 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@H](N3CCCC3)CCC[C@H]21 ZINC000147485925 KJ Annotated Anodyne OPRK1 33 75 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@H](N3CCCC3)CCC[C@H]21 ZINC000147485925 KJ Annotated Anodyne SIGMAR1 17 65 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@H](N3CCCC3)CCC[C@H]21 ZINC000147485925 KJ Annotated Anodyne CCR3 51 38 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@@H]2[C@H](N3CCCC3)CCC[C@H]21 ZINC000147485925 KJ Annotated Anodyne L3MBTL3 43 37 CCc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)o1 ZINC000147485966 CG For-Sale Anodyne SCN10A 19 41 CCc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)o1 ZINC000147485966 CG For-Sale Anodyne CACNA1I 44 34 CS(=O)(=O)N1CCC[C@@H](NC(=O)NC2CCN(c3ccccc3)CC2)C1 ZINC000147485977 GD On-Demand Anodyne EPHX2 49 53 C[C@@H](CNc1ccc(F)cc1C#N)CC(=O)O ZINC000147485982 BE For-Sale Mild SDH1 0 40 O=S(=O)(Cl)c1c(C2CC2)nn(-c2ccc(Cl)cc2Cl)c1Cl ZINC000147485991 GJ For-Sale Unstable CNR1 51 31 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485996 ED On-Demand Anodyne NPY1R 24 40 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485996 ED On-Demand Anodyne GRIA1 41 32 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485996 ED On-Demand Anodyne PCSK5 56 35 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485996 ED On-Demand Anodyne FURIN 62 36 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485996 ED On-Demand Anodyne MC1R 47 33 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485996 ED On-Demand Anodyne POLG_WNV 66 32 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485996 ED On-Demand Anodyne NPFFR1 46 31 CCCC[C@@H](NC(N)=O)C(=O)NCc1cccnc1-n1cccn1 ZINC000147485996 ED On-Demand Anodyne HPN 50 34 O=C(c1cccc(OC(F)F)c1)N1CCC[C@H]1CCCBr ZINC000147486037 FI For-Sale Reactive PREP 38 40 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CNC1CC1 ZINC000147486061 CD For-Sale Bother CACNA1C 56 41 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CNC1CC1 ZINC000147486061 CD For-Sale Bother CACNA1D 86 35 O=C(NC1CCN(C(=O)[C@@H]2C[C@@H]2c2cccc(Cl)c2)CC1)c1ccsc1 ZINC000147486080 GH On-Demand Anodyne NPBWR1 96 38 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@H]2[C@@H]1CCC[C@H]2N1CCCC1 ZINC000147486140 KJ Annotated Anodyne OPRK1 33 75 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@H]2[C@@H]1CCC[C@H]2N1CCCC1 ZINC000147486140 KJ Annotated Anodyne SIGMAR1 17 65 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@H]2[C@@H]1CCC[C@H]2N1CCCC1 ZINC000147486140 KJ Annotated Anodyne CCR3 51 38 O=C(c1ccccc1)N1CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)[C@H]2[C@@H]1CCC[C@H]2N1CCCC1 ZINC000147486140 KJ Annotated Anodyne L3MBTL3 43 37 Nc1cc(S(=O)(=O)Nc2ccncc2Br)c(Br)cc1F ZINC000147486145 IG For-Sale Anodyne PTGS1 0 40 Cc1nn(C(F)F)c(C)c1CC(=O)NCc1cccnc1-n1cccn1 ZINC000147486197 FE On-Demand Anodyne P2RX7 61 48 C[C@@H]1CCCC[C@@H]1NC(=O)CC1(CN)CCC1 ZINC000147486199 BE For-Sale Anodyne CACNA2D1 41 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)c(Cl)[nH]2)c1 ZINC000147486200 EH On-Demand Anodyne PPIA 15 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)c(Cl)[nH]2)c1 ZINC000147486200 EH On-Demand Anodyne HCAR1 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)c(Cl)[nH]2)c1 ZINC000147486200 EH On-Demand Anodyne KCNK3 25 40 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA2 180 62 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA6 32 42 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA1 152 62 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA7 84 55 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA13 45 42 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA5B 52 44 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA4 145 51 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA5A 56 44 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA14 65 55 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne PTPRB 20 43 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA12 97 62 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA9 110 62 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CAH_METTE 29 42 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CYNT 55 44 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne NCE103 33 43 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne MTCA1 58 45 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne P96878_MYCTU 72 48 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne CA 0 43 C[C@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486228 CC For-Sale Anodyne Q5TU56_ANOGA 0 41 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CNC1CC1 ZINC000147486251 CD For-Sale Bother CACNA1C 56 41 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CNC1CC1 ZINC000147486251 CD For-Sale Bother CACNA1D 86 35 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCC(NC(=O)c3ccsc3)CC1)C2 ZINC000147486297 HF On-Demand Anodyne NPBWR1 81 35 O=C(NC[C@@H]1CCOC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147486305 CE For-Sale Anodyne CACNA1I 73 41 NNc1ccc(C(=O)NCCNC(N)=O)cc1[N+](=O)[O-] ZINC000147486308 CB For-Sale Bother TAAR1 19 40 Cc1nc(Nc2cccc(F)c2C#N)ccc1C(=O)O ZINC000147486340 CF For-Sale Mild AKR1C2 40 35 CCn1cc(NC(=O)NCc2cc(Br)ccc2OC)ccc1=O ZINC000147486360 GF On-Demand Anodyne TSHR 47 31 CCn1cc(NC(=O)NCc2cc(Br)ccc2OC)ccc1=O ZINC000147486360 GF On-Demand Anodyne ENPP1 40 36 O=C(NCCc1ccccc1F)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147486392 HG On-Demand Anodyne MAP1 76 38 Cn1nccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147486405 CE In-Stock Anodyne FLT1 20 40 C[C@H]1CCCC[C@@H]1NC(=O)CC1(CN)CCC1 ZINC000147486419 BE For-Sale Anodyne CACNA2D1 41 41 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA2 180 62 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA6 32 42 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA1 152 62 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA7 84 55 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA13 45 42 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA5B 52 44 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA4 145 51 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA5A 56 44 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA14 65 55 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne PTPRB 20 43 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA12 97 62 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA9 110 62 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CAH_METTE 29 42 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CYNT 55 44 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne NCE103 33 43 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne MTCA1 58 45 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne P96878_MYCTU 72 48 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne CA 0 43 C[C@@H](CNc1ccc(S(N)(=O)=O)cc1)CC(=O)O ZINC000147486448 CC For-Sale Anodyne Q5TU56_ANOGA 0 41 CS(=O)(=O)N1CCC[C@H](NC(=O)NCc2ccc(F)cc2Br)C1 ZINC000147486458 HD On-Demand Anodyne P2RX7 56 48 CS(=O)(=O)N1CCC[C@H](NC(=O)NCc2ccc(F)cc2Br)C1 ZINC000147486458 HD On-Demand Anodyne CCR3 24 46 CS(=O)(=O)N1CCC[C@H](NC(=O)NCc2ccc(F)cc2Br)C1 ZINC000147486458 HD On-Demand Anodyne EPHX2 22 43 CNC(=O)COc1ccc(C(=O)[C@@H](C#N)c2nc3ccccc3[nH]2)cc1OC ZINC000147486464 GE On-Demand Mild HPSE 16 43 CNC(=O)COc1ccc(C(=O)[C@@H](C#N)c2nc3ccccc3[nH]2)cc1OC ZINC000147486464 GE On-Demand Mild ENPP1 68 35 CCCNCC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147486469 CE For-Sale Bother CACNA1C 41 37 CCCNCC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147486469 CE For-Sale Bother CACNA1D 64 34 COc1ccc(C(C)=O)cc1CC(=O)N1CCN(CCOc2ccc(Cl)cc2)CC1 ZINC000147486515 IG On-Demand Anodyne DRD2 21 47 COc1ccc(C(C)=O)cc1CC(=O)N1CCN(CCOc2ccc(Cl)cc2)CC1 ZINC000147486515 IG On-Demand Anodyne HTR2A 25 43 COc1ccc(C(C)=O)cc1CC(=O)N1CCN(CCOc2ccc(Cl)cc2)CC1 ZINC000147486515 IG On-Demand Anodyne HTR4 30 40 COc1ccc(C(C)=O)cc1CC(=O)N1CCN(CCOc2ccc(Cl)cc2)CC1 ZINC000147486515 IG On-Demand Anodyne LTA4H 29 42 COc1ccc(C(C)=O)cc1CC(=O)N1CCN(CCOc2ccc(Cl)cc2)CC1 ZINC000147486515 IG On-Demand Anodyne HRH3 35 43 COc1ccc(C(C)=O)cc1CC(=O)N1CCN(CCOc2ccc(Cl)cc2)CC1 ZINC000147486515 IG On-Demand Anodyne SLC9A1 54 38 COc1ccc(C(C)=O)cc1CC(=O)N1CCN(CCOc2ccc(Cl)cc2)CC1 ZINC000147486515 IG On-Demand Anodyne MCHR1 15 41 COc1ccc(C(C)=O)cc1CC(=O)N1CCN(CCOc2ccc(Cl)cc2)CC1 ZINC000147486515 IG On-Demand Anodyne PSMB1 42 37 O=C(NC[C@H]1CCOC1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147486545 CE For-Sale Anodyne CACNA1I 73 41 Cc1cc(N)c(S(=O)(=O)Nc2ccncc2Br)cc1C ZINC000147486576 FF For-Sale Anodyne PTGS1 0 43 C[C@@H]1CCCC[C@H]1NC(=O)CC1(CN)CCC1 ZINC000147486606 BE For-Sale Anodyne CACNA2D1 41 41 C[C@H](CNc1cccc(F)c1C(N)=O)CC(=O)O ZINC000147486671 CD For-Sale Anodyne DAC 22 40 CCCNCC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147486687 CE For-Sale Bother CACNA1C 41 37 CCCNCC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147486687 CE For-Sale Bother CACNA1D 64 34 CS(=O)(=O)N1CCC[C@@H](NC(=O)NCc2ccc(F)cc2Br)C1 ZINC000147486688 HD On-Demand Anodyne P2RX7 56 48 CS(=O)(=O)N1CCC[C@@H](NC(=O)NCc2ccc(F)cc2Br)C1 ZINC000147486688 HD On-Demand Anodyne CCR3 24 46 CS(=O)(=O)N1CCC[C@@H](NC(=O)NCc2ccc(F)cc2Br)C1 ZINC000147486688 HD On-Demand Anodyne EPHX2 22 43 CCCNc1ncnc(Oc2ccc(Br)cc2F)c1CC ZINC000147486760 FJ For-Sale Anodyne HTT 0 51 CC(C)NCc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147486791 DJ For-Sale Anodyne MAOB 59 46 CC(C)NCc1cccc(COc2ccc(Cl)c(F)c2)c1 ZINC000147486791 DJ For-Sale Anodyne GYS1 44 37 Nc1ccccc1S(=O)(=O)Nc1ccncc1Br ZINC000147486795 EE For-Sale Anodyne CA14 0 40 Nc1ccccc1S(=O)(=O)Nc1ccncc1Br ZINC000147486795 EE For-Sale Anodyne NFKBIA 0 51 C[C@H]1CCCC[C@H]1NC(=O)CC1(CN)CCC1 ZINC000147486805 BE For-Sale Anodyne CACNA2D1 41 41 Cc1nc(Nc2ccc(N(C)C)cc2)ccc1C(=O)O ZINC000147486855 CF For-Sale Anodyne AKR1C2 61 38 C[C@@H](CNc1cccc(F)c1C(N)=O)CC(=O)O ZINC000147486899 CD For-Sale Anodyne DAC 22 40 CCN[C@@H](C)CC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147486903 CF For-Sale Bother CACNA1C 41 37 CCN[C@@H](C)CC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147486903 CF For-Sale Bother CACNA1D 62 34 COC(=O)Cc1csc(Cc2ccc(Cl)cc2Cl)n1 ZINC000147486932 DH For-Sale Anodyne PTGER1 23 49 COc1cc(N)ccc1S(=O)(=O)Nc1ccncc1Br ZINC000147487008 FE For-Sale Anodyne ALPL 25 40 Cc1nc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)o1 ZINC000147487029 CF On-Demand Anodyne JUN 19 45 Cc1nc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)o1 ZINC000147487029 CF On-Demand Anodyne ATF1 47 38 Cc1nc(C)c(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)o1 ZINC000147487029 CF On-Demand Anodyne NFKB1 44 38 NCC1(CC(=O)N[C@@H]2CN3CCC2CC3)CCC1 ZINC000147487043 CC For-Sale Anodyne HTR3A 16 40 CC(C)CCCCNC[C@H](O)COc1cccc(Br)c1 ZINC000147487056 EH For-Sale Anodyne ADRB2 57 47 CC(C)CCCCNC[C@H](O)COc1cccc(Br)c1 ZINC000147487056 EH For-Sale Anodyne ADRB1 68 46 CC(C)CCCCNC[C@H](O)COc1cccc(Br)c1 ZINC000147487056 EH For-Sale Anodyne GRIN1 24 40 CC(C)CCCCNC[C@H](O)COc1cccc(Br)c1 ZINC000147487056 EH For-Sale Anodyne ADRB3 50 42 C[C@H](CNc1ncccc1[N+](=O)[O-])CC(=O)O ZINC000147487097 BD On-Demand Bother COLA 83 34 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(Cl)c2Oc2cccnc2)C1 ZINC000147487132 HG On-Demand Anodyne CACNA1I 45 34 CCN[C@H](C)CC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147487137 CF For-Sale Bother CACNA1C 41 37 CCN[C@H](C)CC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147487137 CF For-Sale Bother CACNA1D 62 34 CN1CCN(CCCCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)CC1 ZINC000147487199 GC On-Demand Bother HTR1A 21 47 CN1CCN(CCCCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)CC1 ZINC000147487199 GC On-Demand Bother DRD4 40 30 CN1CCN(CCCCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)CC1 ZINC000147487199 GC On-Demand Bother DRD3 59 38 CN1CCN(CCCCNC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)CC1 ZINC000147487199 GC On-Demand Bother HRP1_PLAFA 35 45 CNCc1cccc(OCCOc2ccc(Cl)c(F)c2)c1 ZINC000147487213 DH For-Sale Anodyne PDS 45 34 Cc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1N ZINC000147487227 EF For-Sale Anodyne PTGS1 0 41 CC(C)CCCCNC[C@@H](O)COc1cccc(Br)c1 ZINC000147487243 EH For-Sale Anodyne ADRB2 57 47 CC(C)CCCCNC[C@@H](O)COc1cccc(Br)c1 ZINC000147487243 EH For-Sale Anodyne ADRB1 68 46 CC(C)CCCCNC[C@@H](O)COc1cccc(Br)c1 ZINC000147487243 EH For-Sale Anodyne GRIN1 24 40 CC(C)CCCCNC[C@@H](O)COc1cccc(Br)c1 ZINC000147487243 EH For-Sale Anodyne ADRB3 50 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccn2)c1 ZINC000147487244 DG On-Demand Anodyne PPIA 20 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccn2)c1 ZINC000147487244 DG On-Demand Anodyne ATF1 47 39 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccn2)c1 ZINC000147487244 DG On-Demand Anodyne PYGL 24 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccn2)c1 ZINC000147487244 DG On-Demand Anodyne GRM4 64 50 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccn2)c1 ZINC000147487244 DG On-Demand Anodyne PYGM 28 45 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccn2)c1 ZINC000147487244 DG On-Demand Anodyne NFKB1 44 39 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccn2)c1 ZINC000147487244 DG On-Demand Anodyne TYK2 49 32 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccn2)c1 ZINC000147487244 DG On-Demand Anodyne KDM4C 0 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccn2)c1 ZINC000147487244 DG On-Demand Anodyne HCAR1 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccn2)c1 ZINC000147487244 DG On-Demand Anodyne KCNK3 28 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cc(Cl)ccn2)c1 ZINC000147487244 DG On-Demand Anodyne FTO 0 43 NCC1(CC(=O)N[C@H]2CN3CCC2CC3)CCC1 ZINC000147487274 CC For-Sale Anodyne HTR3A 16 40 C[C@@H](CNc1ncccc1[N+](=O)[O-])CC(=O)O ZINC000147487292 BD On-Demand Bother COLA 83 34 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(Cl)c2Oc2cccnc2)C1 ZINC000147487340 HG On-Demand Anodyne CACNA1I 45 34 CCN[C@@H](C)CC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147487345 CF For-Sale Bother CACNA1C 41 37 CCN[C@@H](C)CC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147487345 CF For-Sale Bother CACNA1D 62 34 COCc1nc(C(=O)Nc2ccccc2Oc2ccccc2Cl)cs1 ZINC000147487417 FJ On-Demand Anodyne GRM4 33 40 Nc1ccc(Cl)cc1S(=O)(=O)Nc1ccncc1Br ZINC000147487430 FF For-Sale Anodyne SGK1 41 38 CC(C)CCCCNC[C@H](O)COc1ccc(F)cc1 ZINC000147487441 CF For-Sale Anodyne ADRB2 68 48 CC(C)CCCCNC[C@H](O)COc1ccc(F)cc1 ZINC000147487441 CF For-Sale Anodyne ADRB1 87 50 CC(C)CCCCNC[C@H](O)COc1ccc(F)cc1 ZINC000147487441 CF For-Sale Anodyne GRIN1 22 53 CC(C)CCCCNC[C@H](O)COc1ccc(F)cc1 ZINC000147487441 CF For-Sale Anodyne ADRB3 52 50 CC(C)CCCCNC[C@H](O)COc1ccc(F)cc1 ZINC000147487441 CF For-Sale Anodyne ABCB1 0 45 CC(C)CCCCNC[C@H](O)COc1ccc(F)cc1 ZINC000147487441 CF For-Sale Anodyne LEF 65 37 CC(C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147487451 BF On-Demand Anodyne AKR1C3 21 45 CC(C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147487451 BF On-Demand Anodyne HCAR1 0 46 COc1ccc(CC[C@@]2(C)NC(=O)N(C[C@@H](O)COc3c(C)ccc(C)c3C)C2=O)cc1 ZINC000147487512 IG On-Demand Anodyne CYP2D6 15 42 NCC1(CC(=O)NCCc2cccs2)CCC1 ZINC000147487514 CD For-Sale Anodyne ADAM17 0 43 NCC1(CC(=O)NCCc2cccs2)CCC1 ZINC000147487514 CD For-Sale Anodyne CA5B 30 43 Cc1nc(N2CCC[C@H]3CCCC[C@@H]32)ccc1C(=O)O ZINC000147487516 CG For-Sale Anodyne NR3C2 41 44 CCN[C@H](C)CC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147487560 CF For-Sale Bother CACNA1C 41 37 CCN[C@H](C)CC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147487560 CF For-Sale Bother CACNA1D 62 34 CN(C)CCOc1ccccc1C(=O)Nc1ccc(-n2cncn2)c(F)c1 ZINC000147487607 FF On-Demand Anodyne NPY2R 63 37 CN(C)CCOc1ccccc1C(=O)Nc1ccc(-n2cncn2)c(F)c1 ZINC000147487607 FF On-Demand Anodyne KDR 15 45 CN(C)CCOc1ccccc1C(=O)Nc1ccc(-n2cncn2)c(F)c1 ZINC000147487607 FF On-Demand Anodyne MET 48 43 CN(C)CCOc1ccccc1C(=O)Nc1ccc(-n2cncn2)c(F)c1 ZINC000147487607 FF On-Demand Anodyne KCNK3 54 39 CN(C)CCOc1ccccc1C(=O)Nc1ccc(-n2cncn2)c(F)c1 ZINC000147487607 FF On-Demand Anodyne KCNK9 55 39 CC(C)CCCCNC[C@@H](O)COc1ccc(F)cc1 ZINC000147487645 CF For-Sale Anodyne ADRB2 68 48 CC(C)CCCCNC[C@@H](O)COc1ccc(F)cc1 ZINC000147487645 CF For-Sale Anodyne ADRB1 87 50 CC(C)CCCCNC[C@@H](O)COc1ccc(F)cc1 ZINC000147487645 CF For-Sale Anodyne GRIN1 22 53 CC(C)CCCCNC[C@@H](O)COc1ccc(F)cc1 ZINC000147487645 CF For-Sale Anodyne ADRB3 52 50 CC(C)CCCCNC[C@@H](O)COc1ccc(F)cc1 ZINC000147487645 CF For-Sale Anodyne ABCB1 0 45 CC(C)CCCCNC[C@@H](O)COc1ccc(F)cc1 ZINC000147487645 CF For-Sale Anodyne LEF 65 37 CNc1cc(Oc2ccc(Br)cc2F)nc(N)n1 ZINC000147487658 DF For-Sale Anodyne AGPAT2 44 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne EPHX1 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne RARA 25 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne PPIA 16 53 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne F10 30 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne CPT1A 68 47 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne CPT2 42 35 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne PRNP 34 53 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne NR1H4 20 48 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne SCN10A 24 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne LUCI_LUCLA 24 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne TAAR1 25 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne AKR1C3 38 48 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne PTPA 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne HCAR1 0 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne GPR35 22 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne Q25615_ONCVO 30 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne SENP1 0 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne KCNK3 72 50 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(Cl)cc2)c1 ZINC000147487696 DH On-Demand Anodyne KCNK9 24 40 Cc1nc(N2CCC[C@@H]3CCCC[C@@H]32)ccc1C(=O)O ZINC000147487699 CG For-Sale Anodyne NR3C2 41 44 COc1ccc(CC[C@@]2(C)NC(=O)N(C[C@H](O)COc3c(C)ccc(C)c3C)C2=O)cc1 ZINC000147487720 IG On-Demand Anodyne CYP2D6 15 42 Cc1cc(-c2cnc3c(NCCC(F)(F)F)cc([C@@](C)(O)c4cccc(F)c4O)nn23)ccc1C(=O)NC1CC1 ZINC000147487762 KK Annotated Anodyne TTK 43 73 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C1CNC1 ZINC000147487785 CD For-Sale Bother CACNA1C 49 39 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C1CNC1 ZINC000147487785 CD For-Sale Bother CACNA1D 80 35 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C1CNC1 ZINC000147487785 CD For-Sale Bother TRPM8 0 41 CCNCc1coc(COc2ccc(Cl)c(F)c2)c1 ZINC000147487835 CH For-Sale Anodyne DAO 16 45 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(OC(F)(F)F)cc1 ZINC000147487850 FH On-Demand Anodyne BMP1 47 33 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(OC(F)(F)F)cc1 ZINC000147487850 FH On-Demand Anodyne ACACA 22 40 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(OC(F)(F)F)cc1 ZINC000147487850 FH On-Demand Anodyne ACACB 29 40 C[C@H](NC(=O)N(C)Cc1cscn1)c1ccc(OC(F)(F)F)cc1 ZINC000147487850 FH On-Demand Anodyne CYP3A4 17 42 COC(=O)Cc1csc(-c2ccc(F)cc2Cl)n1 ZINC000147487851 CG For-Sale Anodyne P2RX7 49 37 Cc1cc(N)cc(S(=O)(=O)Nc2ccncc2Br)c1C ZINC000147487882 FF For-Sale Anodyne PTGS1 0 41 COc1ccc(CC[C@]2(C)NC(=O)N(C[C@@H](O)COc3c(C)ccc(C)c3C)C2=O)cc1 ZINC000147487904 IG On-Demand Anodyne CYP2D6 15 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cnccn2)c1 ZINC000147487951 CE On-Demand Anodyne JUN 22 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cnccn2)c1 ZINC000147487951 CE On-Demand Anodyne ATF1 57 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cnccn2)c1 ZINC000147487951 CE On-Demand Anodyne GRM4 51 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cnccn2)c1 ZINC000147487951 CE On-Demand Anodyne NFKB1 52 41 C[C@H](CNc1cc(Cl)ccc1C(N)=O)CC(=O)O ZINC000147487957 CD For-Sale Anodyne OXER1 41 35 CN(CC1CCC1)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147487976 CG For-Sale Anodyne CACNA1I 52 36 Cc1nc(Nc2cccc3cnccc23)ccc1C(=O)O ZINC000147487995 CG For-Sale Anodyne TRPV1 43 46 Cc1nc(Nc2cccc3cnccc23)ccc1C(=O)O ZINC000147487995 CG For-Sale Anodyne MAPK8 17 42 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C1CNC1 ZINC000147488003 CD For-Sale Bother CACNA1C 49 39 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C1CNC1 ZINC000147488003 CD For-Sale Bother CACNA1D 80 35 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C1CNC1 ZINC000147488003 CD For-Sale Bother TRPM8 0 41 C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(OC(F)(F)F)cc1 ZINC000147488058 FH On-Demand Anodyne BMP1 47 33 C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(OC(F)(F)F)cc1 ZINC000147488058 FH On-Demand Anodyne ACACA 22 40 C[C@@H](NC(=O)N(C)Cc1cscn1)c1ccc(OC(F)(F)F)cc1 ZINC000147488058 FH On-Demand Anodyne ACACB 29 40 COc1ccc(C2(CNC(=O)[C@@H]3COc4cc(OC)ccc4C3)CCOCC2)cc1 ZINC000147488095 HG On-Demand Anodyne MTNR1A 31 43 COc1ccc(C2(CNC(=O)[C@@H]3COc4cc(OC)ccc4C3)CCOCC2)cc1 ZINC000147488095 HG On-Demand Anodyne MTNR1B 26 43 COc1ccc(C2(CNC(=O)[C@@H]3COc4cc(OC)ccc4C3)CCOCC2)cc1 ZINC000147488095 HG On-Demand Anodyne ROCK2 21 40 Nc1cccc(NC(=O)C2CC2)c1Cl ZINC000147488116 BE For-Sale Anodyne TYK2 47 40 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2F)c1 ZINC000147488177 DH On-Demand Anodyne PPIA 19 50 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2F)c1 ZINC000147488177 DH On-Demand Anodyne TYK2 31 50 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2F)c1 ZINC000147488177 DH On-Demand Anodyne TAAR1 22 40 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2F)c1 ZINC000147488177 DH On-Demand Anodyne AKR1C3 36 47 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2F)c1 ZINC000147488177 DH On-Demand Anodyne HCAR1 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2F)c1 ZINC000147488177 DH On-Demand Anodyne KCNK3 69 44 O=C(O)c1cc(Cl)cc(NC(=O)c2c(F)cccc2F)c1 ZINC000147488177 DH On-Demand Anodyne TMPRSS4 0 40 C[C@@H](CNc1cc(Cl)ccc1C(N)=O)CC(=O)O ZINC000147488181 CD For-Sale Anodyne OXER1 41 35 NCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147488212 CE In-Stock Anodyne CA2 33 42 NCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147488212 CE In-Stock Anodyne CA1 25 45 NCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147488212 CE In-Stock Anodyne CSNK1D 53 69 NCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147488212 CE In-Stock Anodyne PIK3CA 21 41 NCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147488212 CE In-Stock Anodyne CA4 36 42 NCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147488212 CE In-Stock Anodyne PTPN7 0 40 NCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147488212 CE In-Stock Anodyne PIK3CG 17 41 NCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147488212 CE In-Stock Anodyne FABK 0 41 NCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147488212 CE In-Stock Anodyne PORCN 0 41 NCC(=O)Nc1nc2ccc(OC(F)(F)F)cc2s1 ZINC000147488212 CE In-Stock Anodyne ISPD 0 52 NCC1(CC(=O)N2CCc3ccccc32)CCC1 ZINC000147488227 BE For-Sale Anodyne AVPR2 31 40 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@]1(C)CCNC1 ZINC000147488228 CE For-Sale Bother CACNA1D 54 33 COC(=O)Cc1csc(CSc2ccccc2)n1 ZINC000147488257 CG For-Sale Anodyne FAS 34 40 O=C(CSc1nncs1)Nc1ccc(-n2cncn2)c(F)c1 ZINC000147488263 ED On-Demand Anodyne ENPP1 50 32 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne CA2 29 78 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne OXTR 0 43 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne CA6 16 42 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne CA1 15 42 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne CA4 29 68 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne PRTN3 58 37 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne CA12 17 47 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne CA9 22 68 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne PFMRK 0 42 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne CYNT 50 78 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne MTCA1 21 44 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne P96878_MYCTU 22 44 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne MTCA2 18 42 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne CA 0 47 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne UQCRB 0 56 NS(=O)(=O)c1ccccc1NS(=O)(=O)c1ccc(C(F)(F)F)cc1 ZINC000147488318 GE On-Demand Anodyne Q5TU56_ANOGA 0 42 Cc1[nH]c(=O)c(C#N)cc1-c1ccc(Cl)cc1 ZINC000147488322 BF For-Sale Mild Q9XSW7_PIG 0 69 Cc1nc(NCc2ccc([N+](=O)[O-])cc2)ccc1C(=O)O ZINC000147488353 CF For-Sale Bother U38 0 40 COc1cc(Br)c(S(=O)(=O)NCc2c(C)noc2C)cc1OC ZINC000147488400 HF On-Demand Anodyne EDNRA 15 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cnc(Cl)c(Cl)c2)c1 ZINC000147488421 EH On-Demand Anodyne JUN 23 44 O=C(O)c1cc(Cl)cc(NC(=O)c2cnc(Cl)c(Cl)c2)c1 ZINC000147488421 EH On-Demand Anodyne ATF1 57 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cnc(Cl)c(Cl)c2)c1 ZINC000147488421 EH On-Demand Anodyne NFKB1 53 41 O=C(O)c1cc(Cl)cc(NC(=O)c2cnc(Cl)c(Cl)c2)c1 ZINC000147488421 EH On-Demand Anodyne SCN10A 21 40 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@]1(C)CCNC1 ZINC000147488439 CE For-Sale Bother CACNA1D 54 33 Cc1cc(-c2cnc3c(NCCC(F)(F)F)cc([C@](C)(O)c4cccc(F)c4O)nn23)ccc1C(=O)NC1CC1 ZINC000147488444 KK Annotated Anodyne TTK 43 73 O=C(O)c1sc(-c2cccnc2)nc1Cl ZINC000147488514 BF For-Sale Anodyne CYP11B1 15 40 O=C(O)c1sc(-c2cccnc2)nc1Cl ZINC000147488514 BF For-Sale Anodyne CYP11B2 34 40 O=C(O)c1sc(-c2cccnc2)nc1Cl ZINC000147488514 BF For-Sale Anodyne CYP2E1 47 34 O=C(O)c1sc(-c2cccnc2)nc1Cl ZINC000147488514 BF For-Sale Anodyne CYP2A6 44 38 COc1ccc2c(c1)OC[C@H](C(=O)N1CCc3cc(OC)c(OC)cc3CC1)C2 ZINC000147488516 GF On-Demand Anodyne ADRA2C 45 31 COc1ccc2c(c1)OC[C@H](C(=O)N1CCc3cc(OC)c(OC)cc3CC1)C2 ZINC000147488516 GF On-Demand Anodyne MTNR1A 15 44 COc1ccc2c(c1)OC[C@H](C(=O)N1CCc3cc(OC)c(OC)cc3CC1)C2 ZINC000147488516 GF On-Demand Anodyne MTNR1B 24 45 COc1ccc2c(c1)OC[C@H](C(=O)N1CCc3cc(OC)c(OC)cc3CC1)C2 ZINC000147488516 GF On-Demand Anodyne ROCK2 29 42 COc1ccc2c(c1)OC[C@H](C(=O)N1CCc3cc(OC)c(OC)cc3CC1)C2 ZINC000147488516 GF On-Demand Anodyne SSTR1 42 32 NNc1cc(C(=O)NCCNC(N)=O)nc2ccccc12 ZINC000147488549 CB For-Sale Anodyne HTR3A 15 40 NNc1cc(C(=O)NCCNC(N)=O)nc2ccccc12 ZINC000147488549 CB For-Sale Anodyne BCHE 41 37 O=C(O)c1cc(Cl)cc(NC(=O)N2CC[C@H](O)C2)c1 ZINC000147488618 CD On-Demand Anodyne CACNA1I 46 36 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@]1(C)CCNC1 ZINC000147488650 CE For-Sale Bother CACNA1D 54 33 CCOC(=O)c1cnc(-c2ccc(F)cc2)nc1C ZINC000147488666 CF For-Sale Anodyne JUN 19 47 CCOC(=O)c1cnc(-c2ccc(F)cc2)nc1C ZINC000147488666 CF For-Sale Anodyne ADORA3 0 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne RARA 26 43 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne MAOB 17 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne CPT1A 75 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne CPT2 42 35 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne PRNP 17 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne NR1H4 17 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne KMO 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne TAAR1 36 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne AKR1C3 26 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne HCAR1 0 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne KCNK3 66 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne KCNK9 28 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)c(F)c2)c1 ZINC000147488683 DH On-Demand Anodyne TMPRSS4 0 41 Cc1c(CC(=O)NCCCCN2CCN(C)CC2)nnn1-c1ccccc1 ZINC000147488696 FD On-Demand Anodyne HTR1A 43 47 Cc1c(CC(=O)NCCCCN2CCN(C)CC2)nnn1-c1ccccc1 ZINC000147488696 FD On-Demand Anodyne DRD2 47 41 Cc1c(CC(=O)NCCCCN2CCN(C)CC2)nnn1-c1ccccc1 ZINC000147488696 FD On-Demand Anodyne HTR2A 47 45 Cc1c(CC(=O)NCCCCN2CCN(C)CC2)nnn1-c1ccccc1 ZINC000147488696 FD On-Demand Anodyne HTR2C 39 43 Cc1c(CC(=O)NCCCCN2CCN(C)CC2)nnn1-c1ccccc1 ZINC000147488696 FD On-Demand Anodyne SLC6A4 16 42 Cc1c(CC(=O)NCCCCN2CCN(C)CC2)nnn1-c1ccccc1 ZINC000147488696 FD On-Demand Anodyne DRD3 66 41 Cc1c(CC(=O)NCCCCN2CCN(C)CC2)nnn1-c1ccccc1 ZINC000147488696 FD On-Demand Anodyne HTR7 44 36 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCc3cc(OC)c(OC)cc3CC1)C2 ZINC000147488703 GF On-Demand Anodyne ADRA2C 45 31 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCc3cc(OC)c(OC)cc3CC1)C2 ZINC000147488703 GF On-Demand Anodyne MTNR1A 15 44 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCc3cc(OC)c(OC)cc3CC1)C2 ZINC000147488703 GF On-Demand Anodyne MTNR1B 24 45 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCc3cc(OC)c(OC)cc3CC1)C2 ZINC000147488703 GF On-Demand Anodyne ROCK2 29 42 COc1ccc2c(c1)OC[C@@H](C(=O)N1CCc3cc(OC)c(OC)cc3CC1)C2 ZINC000147488703 GF On-Demand Anodyne SSTR1 42 32 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne ADRB2 34 48 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne ADRB1 48 45 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne ALOX5 20 42 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne PPARG 15 41 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne INHA 56 39 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne ADRB3 37 44 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne LTA4H 23 45 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne SCN2A 20 50 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne S1PR4 30 44 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne PLA2G4B 78 36 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne ABCB1 29 40 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne S1PR2 33 44 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne S1PR1 18 48 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne S1PR5 24 44 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne TAAR1 18 42 CCCCc1ccc(OC[C@H](O)c2ccccc2)cc1 ZINC000147488706 CI For-Sale Anodyne FFAR1 39 44 Cc1cc(C)cc(NC(=O)CC2(CN)CCC2)c1 ZINC000147488710 BF For-Sale Anodyne CACNA2D1 0 42 Nc1cc(Cl)c(Cl)cc1OCc1ccc(Br)cc1 ZINC000147488742 EJ For-Sale Anodyne CCR5 25 45 Nc1cc(Cl)c(Cl)cc1OCc1ccc(Br)cc1 ZINC000147488742 EJ For-Sale Anodyne ACR 22 42 Nc1cc(Cl)c(Cl)cc1OCc1ccc(Br)cc1 ZINC000147488742 EJ For-Sale Anodyne KLK_PIG 25 43 COc1cc(C)c(N)cc1S(=O)(=O)Nc1ccncc1Br ZINC000147488746 FF For-Sale Anodyne ALPL 27 49 CC(C)(C)C(=O)N1CCC[C@H](C(=O)Nc2ccc(-n3cncn3)c(F)c2)C1 ZINC000147488754 FF On-Demand Anodyne NPY2R 28 40 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)c3ccccn3)c2)c1 ZINC000147488779 HG On-Demand Bother ROCK1 25 44 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)c3ccccn3)c2)c1 ZINC000147488779 HG On-Demand Bother GRM4 68 45 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)c3ccccn3)c2)c1 ZINC000147488779 HG On-Demand Bother ROCK2 36 44 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)c3ccccn3)c2)c1 ZINC000147488779 HG On-Demand Bother TAAR1 31 49 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)c3ccccn3)c2)c1 ZINC000147488779 HG On-Demand Bother KCNK3 47 35 CCCNc1ncnc(Oc2ccc(Br)cc2F)c1C ZINC000147488830 EI For-Sale Anodyne HTT 0 51 O=C(O)c1cc(Cl)cc(NC(=O)N2CC[C@@H](O)C2)c1 ZINC000147488832 CD For-Sale Anodyne CACNA1I 46 36 Cc1nc(NCCCc2ccccc2)ccc1C(=O)O ZINC000147488847 CG For-Sale Anodyne SDH1 0 44 Cc1nc(NCCCc2ccccc2)ccc1C(=O)O ZINC000147488847 CG For-Sale Anodyne P2RX1 30 42 Cc1nc(NCCCc2ccccc2)ccc1C(=O)O ZINC000147488847 CG For-Sale Anodyne FAAH 48 37 Cc1nc(NCCCc2ccccc2)ccc1C(=O)O ZINC000147488847 CG For-Sale Anodyne CES1 56 37 Cc1nc(NCCCc2ccccc2)ccc1C(=O)O ZINC000147488847 CG For-Sale Anodyne FOLP 0 41 Cc1nc(NCCCc2ccccc2)ccc1C(=O)O ZINC000147488847 CG For-Sale Anodyne AMP1_PLAFQ 23 40 Cc1nc(NCCCc2ccccc2)ccc1C(=O)O ZINC000147488847 CG For-Sale Anodyne PETD 0 43 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@]1(C)CCNC1 ZINC000147488854 CE For-Sale Bother CACNA1D 54 33 COc1ccc(Br)cc1CNC(=O)Nc1cccc(CN(C)C)c1 ZINC000147488877 GH On-Demand Anodyne TSHR 42 32 COc1ccc(Br)cc1CNC(=O)Nc1cccc(CN(C)C)c1 ZINC000147488877 GH On-Demand Anodyne ROCK2 27 45 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne ADRB2 34 48 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne ADRB1 48 45 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne ALOX5 20 42 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne PPARG 15 41 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne INHA 56 39 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne ADRB3 37 44 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne LTA4H 23 45 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne SCN2A 20 50 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne S1PR4 30 44 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne PLA2G4B 78 36 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne ABCB1 29 40 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne S1PR2 33 44 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne S1PR1 18 48 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne S1PR5 24 44 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne TAAR1 18 42 CCCCc1ccc(OC[C@@H](O)c2ccccc2)cc1 ZINC000147488910 CI For-Sale Anodyne FFAR1 39 44 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne HTR1A 59 53 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne ADRA2A 16 53 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne DRD2 70 53 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne DRD1 29 53 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne DRD4 51 39 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne ACHE 15 41 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne ADRA1D 28 47 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne HTR2A 36 51 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne HTR2C 28 51 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne ADRA1A 36 53 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne ADRA1B 19 47 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne DRD3 110 53 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne HRP1_PLAFA 27 41 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne CHRNA7 15 41 CNC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1OC ZINC000147488939 GC On-Demand Anodyne SLC9A1 60 36 CC(C)(C)C(=O)N1CCC[C@@H](C(=O)Nc2ccc(-n3cncn3)c(F)c2)C1 ZINC000147488952 FF On-Demand Anodyne NPY2R 28 40 CCOc1ncccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147489012 FI On-Demand Anodyne SCN10A 18 40 CCOc1ncccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147489012 FI On-Demand Anodyne FABH 0 40 CCOc1ncccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147489012 FI On-Demand Anodyne G2YM83_BOTF4 68 37 CCc1c(C(=O)O)c(O)nc2ccccc12 ZINC000147489021 BE For-Sale Anodyne DHODH 30 44 CCc1c(C(=O)O)c(O)nc2ccccc12 ZINC000147489021 BE For-Sale Anodyne TACR2 23 43 CCc1c(C(=O)O)c(O)nc2ccccc12 ZINC000147489021 BE For-Sale Anodyne TACR3 63 43 CCc1c(C(=O)O)c(O)nc2ccccc12 ZINC000147489021 BE For-Sale Anodyne CYP73A1 0 45 CC(C)CCCCNS(=O)(=O)c1ccc(S(=O)(=O)Cl)cc1 ZINC000147489025 FF For-Sale Unstable TBXAS1 35 43 COc1ccc(Br)cc1CNC(=O)Nc1nc(C2CC2)cs1 ZINC000147489066 GI On-Demand Anodyne ROCK1 15 40 COc1ccc(Br)cc1CNC(=O)Nc1nc(C2CC2)cs1 ZINC000147489066 GI On-Demand Anodyne ROCK2 21 51 CC1(C)CCN(C(=O)Nc2cc(Br)cc(C(=O)O)c2)CC1 ZINC000147489068 FH For-Sale Anodyne RARA 41 36 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@]1(C)CCCN1 ZINC000147489082 CE For-Sale Bother CACNA1D 54 33 NNc1cc(C(=O)NCCNC(N)=O)c2ccccc2n1 ZINC000147489091 CB For-Sale Anodyne ACACB 25 41 NNc1cc(C(=O)NCCNC(N)=O)c2ccccc2n1 ZINC000147489091 CB For-Sale Anodyne TACR3 27 47 NNc1cc(C(=O)NCCNC(N)=O)c2ccccc2n1 ZINC000147489091 CB For-Sale Anodyne POLR1A 51 31 CC(=O)Nc1ccc(-c2ccc(S(=O)(=O)NCc3c(C)noc3C)cc2)cc1 ZINC000147489122 GG On-Demand Anodyne IDO1 33 45 CNC[C@H](Oc1ccc(Cl)c(F)c1)c1ccccc1 ZINC000147489126 CH For-Sale Anodyne SLC6A2 20 44 CNC[C@H](Oc1ccc(Cl)c(F)c1)c1ccccc1 ZINC000147489126 CH For-Sale Anodyne SLC6A4 17 44 COC(=O)Cc1csc(CSC2CCCC2)n1 ZINC000147489148 CG For-Sale Anodyne QRFPR 44 37 FC(F)(F)COc1ccc2c(c1)CNC2 ZINC000147489165 BE For-Sale Anodyne PNMT 33 45 Cc1cc(C)n([C@@H](C)C(=O)Nc2ccc(-n3cncn3)c(F)c2)n1 ZINC000147489176 EE On-Demand Anodyne NPY2R 59 37 CN1CCN(CCCCNC(=O)c2cc(C(N)=O)cs2)CC1 ZINC000147489178 DC On-Demand Anodyne HTR1A 24 45 CN1CCN(CCCCNC(=O)c2cc(C(N)=O)cs2)CC1 ZINC000147489178 DC On-Demand Anodyne DRD2 37 41 CN1CCN(CCCCNC(=O)c2cc(C(N)=O)cs2)CC1 ZINC000147489178 DC On-Demand Anodyne DRD1 19 40 CN1CCN(CCCCNC(=O)c2cc(C(N)=O)cs2)CC1 ZINC000147489178 DC On-Demand Anodyne DRD4 41 31 CN1CCN(CCCCNC(=O)c2cc(C(N)=O)cs2)CC1 ZINC000147489178 DC On-Demand Anodyne HTR2A 21 41 CN1CCN(CCCCNC(=O)c2cc(C(N)=O)cs2)CC1 ZINC000147489178 DC On-Demand Anodyne DRD3 63 40 CN1CCN(CCCCNC(=O)c2cc(C(N)=O)cs2)CC1 ZINC000147489178 DC On-Demand Anodyne SIRT3 40 32 CN1CCN(CCCCNC(=O)c2cc(C(N)=O)cs2)CC1 ZINC000147489178 DC On-Demand Anodyne SIRT2 47 39 CN1CCN(CCCCNC(=O)c2cc(C(N)=O)cs2)CC1 ZINC000147489178 DC On-Demand Anodyne SIRT1 40 32 CC1(C)CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147489277 DH On-Demand Anodyne CACNA1H 64 42 CC1(C)CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147489277 DH On-Demand Anodyne RARA 41 36 CC1(C)CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147489277 DH On-Demand Anodyne S1PR2 25 42 CC1(C)CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147489277 DH On-Demand Anodyne EPHX2 23 42 CC1(C)CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)CC1 ZINC000147489277 DH On-Demand Anodyne CACNA1I 50 33 NNc1ccc(C(F)(F)F)cc1C(=O)NCCNC(N)=O ZINC000147489297 DC For-Sale Anodyne LIPG 17 41 CNC[C@@H](Oc1ccc(Cl)c(F)c1)c1ccccc1 ZINC000147489298 CH For-Sale Anodyne SLC6A2 20 44 CNC[C@@H](Oc1ccc(Cl)c(F)c1)c1ccccc1 ZINC000147489298 CH For-Sale Anodyne SLC6A4 17 44 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@]1(C)CCCN1 ZINC000147489305 CE For-Sale Bother CACNA1D 54 33 COc1ccc(Br)cc1CNC(=O)Nc1nc(C)c(C)s1 ZINC000147489312 FH On-Demand Anodyne CSNK1D 22 48 COc1ccc(Br)cc1CNC(=O)Nc1nc(C)c(C)s1 ZINC000147489312 FH On-Demand Anodyne ROCK2 16 43 O=C(c1ccc2ccccc2n1)N1CCC[C@@H]1CCCBr ZINC000147489323 EI For-Sale Reactive HCRTR1 24 41 O=C(c1ccc2ccccc2n1)N1CCC[C@@H]1CCCBr ZINC000147489323 EI For-Sale Reactive HCRTR2 0 41 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne PLG 0 40 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne PPARG 24 45 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne MMP13 29 47 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne ROCK1 45 43 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne MTNR1A 40 42 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne MTNR1B 41 42 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne ROCK2 51 41 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne ZAP70 15 41 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne PTGDR 32 45 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne ALS 52 31 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne AKR1C3 29 44 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne STAT6 15 42 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne SCD 26 41 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne AKR1C2 60 42 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne VCP 39 44 COc1cccc(CNc2ccc(C(=O)O)c(C)n2)c1 ZINC000147489331 CF For-Sale Anodyne HAO2 52 39 COC(=O)Cc1csc(-c2ccc(Cl)cn2)n1 ZINC000147489372 CF For-Sale Anodyne F10 49 31 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)o1 ZINC000147489380 CG On-Demand Anodyne SCN10A 31 43 Cc1cc(C)n([C@H](C)C(=O)Nc2ccc(-n3cncn3)c(F)c2)n1 ZINC000147489392 EE On-Demand Anodyne NPY2R 59 37 CN1CCN(CCCCNC(=O)CNC(=O)c2ccsc2)CC1 ZINC000147489434 EC On-Demand Anodyne HTR1A 25 59 CN1CCN(CCCCNC(=O)CNC(=O)c2ccsc2)CC1 ZINC000147489434 EC On-Demand Anodyne DRD2 38 42 CN1CCN(CCCCNC(=O)CNC(=O)c2ccsc2)CC1 ZINC000147489434 EC On-Demand Anodyne DRD1 19 40 CN1CCN(CCCCNC(=O)CNC(=O)c2ccsc2)CC1 ZINC000147489434 EC On-Demand Anodyne DRD4 41 31 CN1CCN(CCCCNC(=O)CNC(=O)c2ccsc2)CC1 ZINC000147489434 EC On-Demand Anodyne DRD3 63 46 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489439 HE On-Demand Bother BMP1 27 41 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489439 HE On-Demand Bother MMP13 20 40 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489439 HE On-Demand Bother COLA 62 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489439 HE On-Demand Bother MMP8 20 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489439 HE On-Demand Bother MMP9 23 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489439 HE On-Demand Bother MMP1 21 40 CCc1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147489474 BF For-Sale Anodyne CACNA2D1 27 40 CC[C@@H](CNC1CC1)Oc1ccc(Cl)c(F)c1 ZINC000147489514 CG For-Sale Anodyne ENV 41 32 Cc1ccc(Br)c(C(=O)Nc2ccc(C(N)=O)cc2C)c1 ZINC000147489520 EG On-Demand Anodyne KCNK3 49 35 CCN(c1cccc(C)c1)c1ccc(C(=O)O)c(C)n1 ZINC000147489536 CH For-Sale Anodyne RXRA 42 36 CCN(c1cccc(C)c1)c1ccc(C(=O)O)c(C)n1 ZINC000147489536 CH For-Sale Anodyne AKR1C2 27 41 CCN(c1cccc(C)c1)c1ccc(C(=O)O)c(C)n1 ZINC000147489536 CH For-Sale Anodyne AKR1C1 29 41 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@]1(C)CCCN1 ZINC000147489546 CE For-Sale Bother CACNA1D 54 33 O=C(c1ccc2ccccc2n1)N1CCC[C@H]1CCCBr ZINC000147489566 EI For-Sale Reactive HCRTR1 24 41 O=C(c1ccc2ccccc2n1)N1CCC[C@H]1CCCBr ZINC000147489566 EI For-Sale Reactive HCRTR2 0 41 COc1cc2c(cc1OC)CCN(C(=O)c1ccc3c(c1)COC3)CC2 ZINC000147489578 FF On-Demand Anodyne ABCB1 19 45 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489643 HE On-Demand Bother BMP1 27 41 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489643 HE On-Demand Bother MMP13 20 40 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489643 HE On-Demand Bother COLA 62 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489643 HE On-Demand Bother MMP8 20 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489643 HE On-Demand Bother MMP9 23 42 COc1ccc([N+](=O)[O-])c(C(=O)N[C@H](C)c2ccc(S(=O)(=O)N(C)C)cc2)c1 ZINC000147489643 HE On-Demand Bother MMP1 21 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489648 DD On-Demand Anodyne HDAC10 43 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489648 DD On-Demand Anodyne PCSK5 42 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489648 DD On-Demand Anodyne FURIN 44 31 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489648 DD On-Demand Anodyne HDAC11 40 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489648 DD On-Demand Anodyne POLG_WNV 51 31 CCCC[C@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489648 DD On-Demand Anodyne NPFFR1 41 32 CCCCc1c(O)c2c(O)cc(O)cc2oc1=O ZINC000147489659 CE For-Sale Anodyne CYP1B1 35 40 CCCCc1c(O)c2c(O)cc(O)cc2oc1=O ZINC000147489659 CE For-Sale Anodyne CCR4 19 47 CCCCc1c(O)c2c(O)cc(O)cc2oc1=O ZINC000147489659 CE For-Sale Anodyne CYP1A1 20 40 CCCCc1c(O)c2c(O)cc(O)cc2oc1=O ZINC000147489659 CE For-Sale Anodyne HSD17B3 23 51 CCCCc1c(O)c2c(O)cc(O)cc2oc1=O ZINC000147489659 CE For-Sale Anodyne NQO1 71 41 CCCCc1ccc(Oc2ccc(N)cc2C(N)=O)cc1 ZINC000147489715 CH For-Sale Anodyne INHA 109 50 CCCCc1ccc(Oc2ccc(N)cc2C(N)=O)cc1 ZINC000147489715 CH For-Sale Anodyne S1PR1 15 42 CCCCc1ccc(Oc2ccc(N)cc2C(N)=O)cc1 ZINC000147489715 CH For-Sale Anodyne ENR 0 41 CC[C@H](CNC1CC1)Oc1ccc(Cl)c(F)c1 ZINC000147489728 CG For-Sale Anodyne ENV 41 32 Cc1ccc(NC(=O)CC2(CN)CCC2)cc1F ZINC000147489734 CF For-Sale Anodyne SLC1A2 45 37 Cc1ccc(NC(=O)CC2(CN)CCC2)cc1F ZINC000147489734 CF For-Sale Anodyne ENV 42 32 C[C@@H](CN1CCCCC1)NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147489741 FH On-Demand Anodyne P2RX3 28 41 C[C@@H](CN1CCCCC1)NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147489741 FH On-Demand Anodyne PLD1 57 46 C[C@@H](CN1CCCCC1)NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147489741 FH On-Demand Anodyne PLD2 28 46 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(C(=O)N3CCCCC3)c2)C1 ZINC000147489755 HE On-Demand Anodyne CCR3 61 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(C(=O)N3CCCCC3)c2)C1 ZINC000147489755 HE On-Demand Anodyne EPHX2 16 41 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(C(=O)N3CCCCC3)c2)C1 ZINC000147489755 HE On-Demand Anodyne CACNA1I 57 37 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cccc(C(=O)N3CCCCC3)c2)C1 ZINC000147489755 HE On-Demand Anodyne L3MBTL3 46 37 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@]1(C)CCCN1 ZINC000147489761 CE For-Sale Bother CACNA1D 54 33 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Br)c1 ZINC000147489789 FI For-Sale Anodyne PPIA 15 41 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Br)c1 ZINC000147489789 FI For-Sale Anodyne ATF1 55 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Br)c1 ZINC000147489789 FI For-Sale Anodyne PYGL 20 44 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Br)c1 ZINC000147489789 FI For-Sale Anodyne NFKB1 51 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccc(F)cc2Br)c1 ZINC000147489789 FI For-Sale Anodyne TMPRSS4 0 41 COc1cc(/C=N/c2ccc(C(C)C)cc2)ccc1OCc1ccc(C(=O)O)cc1 ZINC000147489838 HK In-Stock Mild ADCYAP1R1 50 49 COC(=O)Cc1csc(NC(=O)NCc2cc(Br)ccc2OC)n1 ZINC000147489853 HF On-Demand Anodyne CPT1A 24 41 COC(=O)Cc1csc(NC(=O)NCc2cc(Br)ccc2OC)n1 ZINC000147489853 HF On-Demand Anodyne CPT1B 28 41 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489859 DD On-Demand Anodyne HDAC10 43 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489859 DD On-Demand Anodyne PCSK5 42 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489859 DD On-Demand Anodyne FURIN 44 31 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489859 DD On-Demand Anodyne HDAC11 40 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489859 DD On-Demand Anodyne POLG_WNV 51 31 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccccc1CN(C)C ZINC000147489859 DD On-Demand Anodyne NPFFR1 41 32 Cc1nc(NCCc2ccc(O)cc2)ccc1C(=O)O ZINC000147489874 CE For-Sale Anodyne PTGDR 22 44 Cc1nc(NCCc2ccc(O)cc2)ccc1C(=O)O ZINC000147489874 CE For-Sale Anodyne STAT6 32 41 C[C@H](CN1CCCCC1)NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147489943 FH On-Demand Anodyne P2RX3 28 41 C[C@H](CN1CCCCC1)NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147489943 FH On-Demand Anodyne PLD1 57 46 C[C@H](CN1CCCCC1)NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147489943 FH On-Demand Anodyne PLD2 28 46 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(C(=O)N3CCCCC3)c2)C1 ZINC000147489964 HE On-Demand Anodyne CCR3 61 40 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(C(=O)N3CCCCC3)c2)C1 ZINC000147489964 HE On-Demand Anodyne EPHX2 16 41 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(C(=O)N3CCCCC3)c2)C1 ZINC000147489964 HE On-Demand Anodyne CACNA1I 57 37 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cccc(C(=O)N3CCCCC3)c2)C1 ZINC000147489964 HE On-Demand Anodyne L3MBTL3 46 37 CCc1ccccc1NC(=O)CC1(CN)CCC1 ZINC000147489994 BF For-Sale Anodyne KCNQ2 66 35 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H]1CCN[C@@H]1C ZINC000147490017 CE For-Sale Bother CACNA1D 45 32 CCn1c(=O)c(=O)[nH]c2cc(C(=O)NCCCN(C)C(C)C)ccc21 ZINC000147490036 ED On-Demand Anodyne PLD1 42 32 O=C(/C=C/c1cccs1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147490038 DH On-Demand Anodyne MMP1 17 45 CCOc1ccc(C#N)cc1NC(=O)c1cnn(-c2ccccc2Cl)c1 ZINC000147490065 FI On-Demand Mild EPHB3 51 35 Cc1nn(C(F)F)c(C)c1CC(=O)Nc1ccccc1CN(C)C ZINC000147490083 EG On-Demand Anodyne P2RX7 35 42 CN(Cc1cscn1)C(=O)NC1CCN(c2ccc(C(F)(F)F)cn2)CC1 ZINC000147490142 GG On-Demand Anodyne HPGDS 21 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCCCCC3)cc2)C1 ZINC000147490193 HE On-Demand Anodyne CACNA1I 53 34 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCCCCC3)cc2)C1 ZINC000147490193 HE On-Demand Anodyne L3MBTL3 69 39 C[C@@H]1NCC[C@H]1C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147490215 CE For-Sale Bother CACNA1D 45 32 Cc1nc(NCCc2ccc(Cl)cc2)ccc1C(=O)O ZINC000147490246 CG For-Sale Anodyne PTGDR 27 48 Cc1nc(NCCc2ccc(Cl)cc2)ccc1C(=O)O ZINC000147490246 CG For-Sale Anodyne MRGPRX1 47 44 COC(=O)Cc1csc(-c2cc(F)cc(F)c2)n1 ZINC000147490270 CF For-Sale Anodyne DCK 46 34 C[C@H]1C[C@@H](C)CN(C(=O)CC2(CN)CCC2)C1 ZINC000147490281 BE For-Sale Anodyne CACNA2D1 31 43 Cc1ccc(C(=O)NNC(=O)NC2CCN(c3ncccn3)CC2)s1 ZINC000147490350 FD On-Demand Reactive SIRT3 42 34 Cc1ccc(C(=O)NNC(=O)NC2CCN(c3ncccn3)CC2)s1 ZINC000147490350 FD On-Demand Reactive SIRT2 46 34 Cc1ccc(C(=O)NNC(=O)NC2CCN(c3ncccn3)CC2)s1 ZINC000147490350 FD On-Demand Reactive SIRT1 42 34 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCCOC)c1 ZINC000147490358 FD On-Demand Anodyne REN 26 42 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCCOC)c1 ZINC000147490358 FD On-Demand Anodyne ENPP1 58 35 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCCCCC3)cc2)C1 ZINC000147490363 HE On-Demand Anodyne CACNA1I 53 34 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(C(=O)N3CCCCCC3)cc2)C1 ZINC000147490363 HE On-Demand Anodyne L3MBTL3 69 39 O=[N+]([O-])c1ccc(N2CCN3CCC2CC3)cc1 ZINC000147490369 BD On-Demand Bother CHRNA7 22 60 O=[N+]([O-])c1ccc(N2CCN3CCC2CC3)cc1 ZINC000147490369 BD On-Demand Bother SLC27A4 42 32 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H]1CCN[C@@H]1C ZINC000147490417 CE For-Sale Bother CACNA1D 45 32 O=C(NCC(=O)N1CCCc2ccccc21)[C@@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147490423 FH On-Demand Anodyne AVPR2 36 47 O=C(O)c1cccnc1C(=O)Nc1ccncc1Br ZINC000147490450 DE For-Sale Anodyne MAP 0 40 O=C(O)c1cccnc1C(=O)Nc1ccncc1Br ZINC000147490450 DE For-Sale Anodyne MAP1 41 36 O=C(O)c1cccnc1C(=O)Nc1ccncc1Br ZINC000147490450 DE For-Sale Anodyne FABH 0 40 O=C(O)c1cccnc1C(=O)Nc1ccncc1Br ZINC000147490450 DE For-Sale Anodyne OSIGBA0132E09-OSIGBA0108L24.11 0 40 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild CA2 30 63 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild CA1 25 54 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild TRPV1 21 46 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild HDAC8 20 49 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild CA4 29 44 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild HDAC6 15 43 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild PRTN3 52 33 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild CA12 15 44 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild CA9 17 54 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild IDO1 39 41 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild CYNT 64 63 CC(C)(C)c1ccc(S(=O)(=O)Nc2ccc(C(=O)NO)cc2)cc1 ZINC000147490497 EF On-Demand Mild LIMK2 34 42 C[C@H]1C[C@H](C)CN(C(=O)CC2(CN)CCC2)C1 ZINC000147490525 BE For-Sale Anodyne CACNA2D1 31 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCCOC)c1 ZINC000147490551 FD On-Demand Anodyne REN 26 42 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCCOC)c1 ZINC000147490551 FD On-Demand Anodyne ENPP1 58 35 O=C(O)c1cc(Cl)cc(NC(=O)N2CCCOCC2)c1 ZINC000147490565 CE On-Demand Anodyne EPHX2 17 44 COc1ccc(Br)cc1CNC(=O)Nc1cccnc1N1CCCC1 ZINC000147490572 HH On-Demand Anodyne MC4R 16 41 COc1ccc(Br)cc1CNC(=O)Nc1cccnc1N1CCCC1 ZINC000147490572 HH On-Demand Anodyne KCNQ2 58 33 COc1ccc(Br)cc1CNC(=O)Nc1cccnc1N1CCCC1 ZINC000147490572 HH On-Demand Anodyne RBP4 23 40 CCN1CCN(CC(=O)Nc2n[nH]c(-c3ccccc3OC)n2)C(=O)C1=O ZINC000147490581 FC On-Demand Anodyne MAPK7 45 34 C#CCCOc1ccc(CCCC)cc1 ZINC000147490596 BG For-Sale Mild SCN2A 17 42 C#CCCOc1ccc(CCCC)cc1 ZINC000147490596 BG For-Sale Mild PLA2G4B 82 38 C#CCCOc1ccc(CCCC)cc1 ZINC000147490596 BG For-Sale Mild CYP1A2 15 41 C#CCCOc1ccc(CCCC)cc1 ZINC000147490596 BG For-Sale Mild CYP2C19 19 41 C#CCCOc1ccc(CCCC)cc1 ZINC000147490596 BG For-Sale Mild TAAR1 17 43 C#CCCOc1ccc(CCCC)cc1 ZINC000147490596 BG For-Sale Mild PPO2 19 41 C[C@@H]1NCC[C@@H]1C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147490614 CE For-Sale Bother CACNA1D 45 32 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)C3CCCC3)c2)c1 ZINC000147490628 GH On-Demand Bother MTNR1A 27 45 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)C3CCCC3)c2)c1 ZINC000147490628 GH On-Demand Bother MTNR1B 27 45 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)C3CCCC3)c2)c1 ZINC000147490628 GH On-Demand Bother TAAR1 33 45 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)C3CCCC3)c2)c1 ZINC000147490628 GH On-Demand Bother AKR1C2 25 40 COc1ccc([N+](=O)[O-])c(C(=O)NCc2cccc(NC(=O)C3CCCC3)c2)c1 ZINC000147490628 GH On-Demand Bother KCNK3 21 40 O=C(NCC(=O)N1CCCc2ccccc21)[C@H]1C[C@@H]1c1cccc(Cl)c1 ZINC000147490665 FH On-Demand Anodyne AVPR2 36 47 C[C@H](CNC1=NS(=O)(=O)c2ccccc21)CC(=O)O ZINC000147490675 CC For-Sale Anodyne KCNA3 35 42 COC(=O)c1ccc(C2=CCN(C(=O)OC(C)(C)C)CC2)cc1 ZINC000147490694 DG For-Sale Anodyne GPR119 28 40 O=C(O)c1ccccc1C(=O)Nc1ccncc1Br ZINC000147490697 DF For-Sale Anodyne FABH 0 44 CCNc1cn2ccnc2c(Oc2ccc(Br)cc2F)n1 ZINC000147490704 FH For-Sale Anodyne HIVRT 0 43 COC(=O)Cc1csc(-c2ncccc2C)n1 ZINC000147490723 BE For-Sale Anodyne EGLN1 0 43 C[C@@H]1C[C@@H](C)CN(C(=O)CC2(CN)CCC2)C1 ZINC000147490732 BE For-Sale Anodyne CACNA2D1 31 43 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne HTR1A 67 54 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne DRD2 50 54 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne DRD4 43 37 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne ADRA1D 28 50 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne HTR2A 60 54 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne HTR2C 41 52 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne SLC6A4 18 47 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne ADRA1A 42 50 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne ADRA1B 24 50 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne DRD3 75 52 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne HTR7 72 43 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne GRIA1 40 32 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne PCSK5 52 33 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne FURIN 64 33 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne POLG_WNV 59 31 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne F2RL1 48 32 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490784 GD On-Demand Anodyne NPFFR1 40 31 C#CCNCC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147490823 CD For-Sale Mild CACNA1D 59 36 O=C(NCC(=O)N1CCCc2ccccc21)[C@@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147490853 FH On-Demand Anodyne AVPR2 36 47 COc1ccc(Br)cc1CNC(=O)Nc1nc(C)cs1 ZINC000147490856 FH On-Demand Anodyne ROCK1 15 43 COc1ccc(Br)cc1CNC(=O)Nc1nc(C)cs1 ZINC000147490856 FH On-Demand Anodyne ROCK2 21 52 COc1ccc(Br)cc1CNC(=O)Nc1nc(C)cs1 ZINC000147490856 FH On-Demand Anodyne GCK 18 44 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne F2 51 45 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne PLG 41 44 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne ACE 76 38 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne OPRM1 69 46 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne OPRD1 58 39 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne OPRK1 24 54 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne GHRHR 52 31 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne GRIN2B 43 36 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne MME 76 44 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne ANPEP 66 32 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne TACR1 24 50 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne MC4R 35 40 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne SIGMAR1 24 41 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne TRY2_BOVIN 85 36 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne TRY1_BOVIN 51 40 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne CCR1 37 40 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne SLC15A1 0 45 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne NPFFR2 43 37 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne C3AR1 60 35 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne TPH1 56 31 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne DPP4 47 49 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne YARS 59 38 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne DNPEP 0 41 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne CAPN1 34 42 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne ACE2 61 38 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne DPP7 77 46 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne LAP3 41 38 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne AKT1 29 49 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne ST14 88 36 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne AMP1_PLAFQ 50 49 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne XIAP 51 38 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne DPP8 58 51 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne DPP9 37 51 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne FAP 0 45 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne SLC15A2 0 43 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne BIRC2 37 40 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne SLC12A5 52 33 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne AKT1S1 0 42 CNC1CCN(C(=O)[C@@H](N)Cc2ccccc2)CC1 ZINC000147490867 CC On-Demand Anodyne TMPRSS6 54 33 C[C@@H](CNC1=NS(=O)(=O)c2ccccc21)CC(=O)O ZINC000147490876 CC For-Sale Anodyne KCNA3 35 42 c1ccc(COc2ccc(-c3nc4cnccc4s3)cc2)cc1 ZINC000147490907 DJ On-Demand Anodyne LUCI_PHOPE 30 48 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne HTR1A 67 54 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne DRD2 50 54 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne DRD4 43 37 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne ADRA1D 28 50 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne HTR2A 60 54 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne HTR2C 41 52 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne SLC6A4 18 47 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne ADRA1A 42 50 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne ADRA1B 24 50 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne DRD3 75 52 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne HTR7 72 43 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne GRIA1 40 32 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne PCSK5 52 33 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne FURIN 64 33 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne POLG_WNV 59 31 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne F2RL1 48 32 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(c2cccc(C)c2)CC1 ZINC000147490995 GD On-Demand Anodyne NPFFR1 40 31 C#CCNCC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147490996 CD For-Sale Mild CACNA1D 59 36 CN(C)C(=O)Cc1cccc([N+](=O)[O-])c1 ZINC000147491004 BD On-Demand Bother CACNA1C 57 40 CN(C)C(=O)Cc1cccc([N+](=O)[O-])c1 ZINC000147491004 BD On-Demand Bother APR 0 43 CN(C)C(=O)Cc1cccc([N+](=O)[O-])c1 ZINC000147491004 BD On-Demand Bother TRPM8 0 46 COC(=O)CN(Cc1ccccc1)C(=O)COc1ccc(C(N)=O)cc1 ZINC000147491010 FD On-Demand Anodyne HRAS 48 32 COC(=O)CN(Cc1ccccc1)C(=O)COc1ccc(C(N)=O)cc1 ZINC000147491010 FD On-Demand Anodyne PLA2G4B 50 39 COC(=O)CN(Cc1ccccc1)C(=O)COc1ccc(C(N)=O)cc1 ZINC000147491010 FD On-Demand Anodyne LIMK2 41 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccoc2)c1 ZINC000147491028 CF On-Demand Anodyne CPT1A 35 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccoc2)c1 ZINC000147491028 CF On-Demand Anodyne PRNP 15 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccoc2)c1 ZINC000147491028 CF On-Demand Anodyne HCAR1 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccoc2)c1 ZINC000147491028 CF On-Demand Anodyne KCNK3 50 56 CN(CCNC(=O)Nc1cc(Cl)cc(C(=O)O)c1)C1CC1 ZINC000147491036 DE For-Sale Anodyne CACNA1I 51 34 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne F2 51 45 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne PLG 41 44 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne ACE 76 38 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne OPRM1 69 46 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne OPRD1 58 39 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne OPRK1 24 54 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne GHRHR 52 31 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne GRIN2B 43 36 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne MME 76 44 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne ANPEP 66 32 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne TACR1 24 50 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne MC4R 35 40 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne SIGMAR1 24 41 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne TRY2_BOVIN 85 36 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne TRY1_BOVIN 51 40 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne CCR1 37 40 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne SLC15A1 0 45 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne NPFFR2 43 37 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne C3AR1 60 35 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne TPH1 56 31 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne DPP4 47 49 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne YARS 59 38 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne DNPEP 0 41 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne CAPN1 34 42 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne ACE2 61 38 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne DPP7 77 46 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne LAP3 41 38 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne AKT1 29 49 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne ST14 88 36 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne AMP1_PLAFQ 50 49 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne XIAP 51 38 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne DPP8 58 51 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne DPP9 37 51 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne FAP 0 45 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne SLC15A2 0 43 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne BIRC2 37 40 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne SLC12A5 52 33 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne AKT1S1 0 42 CNC1CCN(C(=O)[C@H](N)Cc2ccccc2)CC1 ZINC000147491061 CC On-Demand Anodyne TMPRSS6 54 33 O=C(NCC(=O)N1CCCc2ccccc21)[C@H]1C[C@H]1c1cccc(Cl)c1 ZINC000147491062 FH On-Demand Anodyne AVPR2 36 47 CN(C)C1(CNc2ccc(C(=O)O)cc2F)CCCC1 ZINC000147491063 CF For-Sale Anodyne RXRA 18 41 CC(=O)c1cccc(O[C@H](C)C(=O)NCCN2CCCS2(=O)=O)c1 ZINC000147491129 FC On-Demand Anodyne DRD4 47 36 CC[C@H](CN)CC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147491217 CE For-Sale Bother CACNA1D 61 36 O=C(O)c1cc(Cl)cc(NC(=O)c2cncc(Br)c2)c1 ZINC000147491258 FG On-Demand Anodyne ATF1 47 38 O=C(O)c1cc(Cl)cc(NC(=O)c2cncc(Br)c2)c1 ZINC000147491258 FG On-Demand Anodyne NFKB1 43 38 O=C(O)c1cc(Cl)cc(NC(=O)c2cncc(Br)c2)c1 ZINC000147491258 FG On-Demand Anodyne SCN10A 41 47 CC(C)CCCCNC(=O)c1cccc(S(=O)(=O)Cl)c1 ZINC000147491267 DG For-Sale Unstable DRD4 42 32 COc1ccc(Br)cc1CNC(=O)Nc1cc(C)nn1-c1ccccn1 ZINC000147491287 HH On-Demand Anodyne TSHR 65 31 CCN1CCC[C@@H]1CNC(=O)CC1(CN)CCC1 ZINC000147491292 CD For-Sale Anodyne DRD2 34 43 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)N1CCCc3ccccc31)C2 ZINC000147491298 GE On-Demand Anodyne AVPR2 39 43 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)N1CCCc3ccccc31)C2 ZINC000147491298 GE On-Demand Anodyne MTNR1A 43 43 COc1ccc2c(c1)OC[C@H](C(=O)NCC(=O)N1CCCc3ccccc31)C2 ZINC000147491298 GE On-Demand Anodyne MTNR1B 39 43 O=C(Nc1ccccc1I)c1cccc(C(F)(F)F)c1F ZINC000147491354 HJ On-Demand Anodyne NR1H4 0 45 O=C(Nc1ccccc1I)c1cccc(C(F)(F)F)c1F ZINC000147491354 HJ On-Demand Anodyne RBP4 46 38 O=C(Nc1ccccc1I)c1cccc(C(F)(F)F)c1F ZINC000147491354 HJ On-Demand Anodyne KCNK3 30 42 O=C(Nc1ccccc1I)c1cccc(C(F)(F)F)c1F ZINC000147491354 HJ On-Demand Anodyne KCNK9 32 40 CC[C@@H](CN)CC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147491405 CE For-Sale Bother CACNA1D 61 36 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(N2CCCCC2=O)c1 ZINC000147491417 EE On-Demand Anodyne HDAC10 46 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(N2CCCCC2=O)c1 ZINC000147491417 EE On-Demand Anodyne HDAC3 27 40 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(N2CCCCC2=O)c1 ZINC000147491417 EE On-Demand Anodyne HDAC11 45 40 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147491478 ED For-Sale Anodyne MTOR 45 41 C[C@H](OC[C@@H]1CCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147491478 ED For-Sale Anodyne DGAT1 45 44 CCN1CCC[C@H]1CNC(=O)CC1(CN)CCC1 ZINC000147491508 CD For-Sale Anodyne DRD2 34 43 COc1cc2c(cc1OC)CCN(C(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)CC2 ZINC000147491569 GI On-Demand Anodyne HCRTR2 15 41 CC[C@H](CN)CC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147491592 CE For-Sale Bother CACNA1D 61 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(N2CCCCC2=O)c1 ZINC000147491621 EE On-Demand Anodyne HDAC10 46 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(N2CCCCC2=O)c1 ZINC000147491621 EE On-Demand Anodyne HDAC3 27 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(N2CCCCC2=O)c1 ZINC000147491621 EE On-Demand Anodyne HDAC11 45 40 Cc1cc(C)n(CCCNC(=O)c2cc(-c3ccco3)n(-c3ccc(Cl)cc3)n2)n1 ZINC000147491637 HI On-Demand Anodyne RPA1 51 33 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147491684 ED For-Sale Anodyne MTOR 45 41 C[C@@H](OC[C@@H]1CCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147491684 ED For-Sale Anodyne DGAT1 45 44 CSc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147491701 DI On-Demand Anodyne RARA 24 42 CSc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147491701 DI On-Demand Anodyne PPIA 16 46 CSc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147491701 DI On-Demand Anodyne CPT1A 45 42 CSc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147491701 DI On-Demand Anodyne PRNP 33 46 CSc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147491701 DI On-Demand Anodyne NR1H4 15 43 CSc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147491701 DI On-Demand Anodyne TAAR1 27 40 CSc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147491701 DI On-Demand Anodyne NOD1 16 44 CSc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147491701 DI On-Demand Anodyne NOD2 17 44 CSc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147491701 DI On-Demand Anodyne KCNK3 66 43 COc1cc2c(cc1OC)CCN(C(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)CC2 ZINC000147491758 GI On-Demand Anodyne HCRTR2 15 41 CC(C)CCCCNC(=O)c1ccc(S(=O)(=O)Cl)cc1 ZINC000147491763 DG For-Sale Unstable CA2 36 40 CC(C)CCCCNC(=O)c1ccc(S(=O)(=O)Cl)cc1 ZINC000147491763 DG For-Sale Unstable FOLH1 33 44 CC(C)CCCCNC(=O)c1ccc(S(=O)(=O)Cl)cc1 ZINC000147491763 DG For-Sale Unstable CA1 20 47 CC(C)CCCCNC(=O)c1ccc(S(=O)(=O)Cl)cc1 ZINC000147491763 DG For-Sale Unstable CA4 15 47 CC(C)CCCCNC(=O)c1ccc(S(=O)(=O)Cl)cc1 ZINC000147491763 DG For-Sale Unstable EPHX2 0 44 CC(C)CCCCNC(=O)c1ccc(S(=O)(=O)Cl)cc1 ZINC000147491763 DG For-Sale Unstable HDA106 0 41 CC(C)CCCCNC(=O)c1ccc(S(=O)(=O)Cl)cc1 ZINC000147491763 DG For-Sale Unstable CYNT 19 40 CC[C@@H](CN)CC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147491785 CE For-Sale Bother CACNA1D 61 36 CC(C)(C)C[C@H]1N[C@@H](C(=O)NCC[C@@](C)(O)CO)[C@H](c2cccc(Cl)c2)[C@@]12C(=O)Nc1cc(Cl)c(F)cc12 ZINC000147491823 KI Annotated Anodyne MDM2 90 78 CN(C)C1(CNc2ccc(C(=O)O)c(Cl)c2)CCCC1 ZINC000147491828 CG For-Sale Anodyne AVPR2 17 42 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147491870 ED For-Sale Anodyne MTOR 45 41 C[C@H](OC[C@H]1CCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147491870 ED For-Sale Anodyne DGAT1 45 44 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne GSK3B 17 47 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne PIK3CA 40 41 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne PRNP 48 36 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne JAK2 19 45 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne MTOR 49 39 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne PIK3CG 36 41 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne FLT3 21 40 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne ATR 68 54 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne BTK 41 40 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne TYRO3 41 36 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne STAT6 56 35 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne DGAT1 36 43 Nc1ncc(-c2cccc(C(=O)N3CCOCC3)c2)nc1C(=O)Nc1ccc(N2CCCC2)cc1 ZINC000147491888 JG For-Sale Anodyne SMG1 18 41 NC(=O)c1ccc(OCC(=O)Nc2ccccc2CN2CCc3ccccc32)cc1 ZINC000147491949 HG On-Demand Anodyne CYSLTR2 41 33 COc1cc2c(cc1OC)CCN(C(=O)[C@@H]1C[C@H]1c1cccc(Cl)c1)CC2 ZINC000147491961 GI On-Demand Anodyne HCRTR2 15 41 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C(C)(C)N ZINC000147491984 CD For-Sale Bother CACNA1C 43 36 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C(C)(C)N ZINC000147491984 CD For-Sale Bother CACNA1D 66 35 CN(NC(=O)N[C@@H]1CCCN(S(C)(=O)=O)C1)c1ccccc1 ZINC000147492074 EC On-Demand Reactive EPHX2 27 43 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147492083 ED For-Sale Anodyne MTOR 45 41 C[C@@H](OC[C@H]1CCCO1)C(=O)Nc1ccc(N2CCOCC2)nc1 ZINC000147492083 ED For-Sale Anodyne DGAT1 45 44 C[C@@H](C(=O)Nc1cc(Cl)cc(C(=O)O)c1)n1cncn1 ZINC000147492103 CD On-Demand Anodyne CYP51 0 40 COc1cc2c(cc1OC)CCN(C(=O)[C@H]1C[C@H]1c1cccc(Cl)c1)CC2 ZINC000147492156 GI On-Demand Anodyne HCRTR2 15 41 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3cc(C)cc(C)c3)cc2)C1 ZINC000147492169 HH On-Demand Anodyne CACNA1I 55 36 CCCNC(=O)c1ccc(NC(=O)c2cc([N+](=O)[O-])cc(S(C)(=O)=O)c2)cc1 ZINC000147492182 HE On-Demand Bother CA2 17 41 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C(C)(C)N ZINC000147492201 CD For-Sale Bother CACNA1C 43 36 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)C(C)(C)N ZINC000147492201 CD For-Sale Bother CACNA1D 66 35 Cc1cccc(C)c1NC(=O)CC1(CN)CCC1 ZINC000147492214 BF For-Sale Anodyne CACNA2D1 0 40 Cc1cccc(C)c1NC(=O)CC1(CN)CCC1 ZINC000147492214 BF For-Sale Anodyne ACAT 0 44 O=C(N1CCC[C@@H]1CCCBr)C1(c2ccccc2)CC1 ZINC000147492244 EH For-Sale Reactive PREP 42 33 NC(=O)c1ccc(OCC(=O)Nc2ccc(Sc3nncs3)cc2)cc1 ZINC000147492248 GF On-Demand Anodyne ADORA2B 33 42 NC(=O)c1ccc(OCC(=O)Nc2ccc(Sc3nncs3)cc2)cc1 ZINC000147492248 GF On-Demand Anodyne HIF1A 15 41 Nc1cc(Cl)c(Cl)cc1OCc1cccc(Br)c1 ZINC000147492251 EJ For-Sale Anodyne DRTS_LEIMA 17 40 CN(NC(=O)N[C@H]1CCCN(S(C)(=O)=O)C1)c1ccccc1 ZINC000147492315 EC On-Demand Reactive EPHX2 27 43 C[C@H](C(=O)Nc1cc(Cl)cc(C(=O)O)c1)n1cncn1 ZINC000147492342 CD On-Demand Anodyne CYP51 0 40 O=C(NCCN1CCCS1(=O)=O)c1ccc(N2CCOCC2)cc1 ZINC000147492347 FC On-Demand Anodyne HPGDS 26 43 C[C@H](CNc1ccc(Br)cc1[N+](=O)[O-])CC(=O)O ZINC000147492360 DF For-Sale Bother COLA 62 34 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3cc(C)cc(C)c3)cc2)C1 ZINC000147492373 HH On-Demand Anodyne CACNA1I 55 36 Cc1ccc(C)c(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147492389 CG For-Sale Anodyne ADRB2 37 52 Cc1ccc(C)c(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147492389 CG For-Sale Anodyne ADRB1 61 40 Cc1ccc(C)c(OC[C@H](O)CNCCCCC(C)C)c1 ZINC000147492389 CG For-Sale Anodyne ABCB1 0 48 CC(C)C[C@H](NC(=O)c1ccc(Br)c(Cl)c1)C(=O)N(C)C ZINC000147492416 GG For-Sale Anodyne CTSL 18 40 CC(C)C[C@H](NC(=O)c1ccc(Br)c(Cl)c1)C(=O)N(C)C ZINC000147492416 GG For-Sale Anodyne CCKBR 16 40 CC(C)C[C@H](NC(=O)c1ccc(Br)c(Cl)c1)C(=O)N(C)C ZINC000147492416 GG For-Sale Anodyne UTS2 44 33 CNCCC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147492420 CD For-Sale Bother CACNA1C 46 36 CNCCC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147492420 CD For-Sale Bother CACNA1D 75 35 CCCNC(=O)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1 ZINC000147492434 FG On-Demand Anodyne GCGR 15 40 CCCNC(=O)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1 ZINC000147492434 FG On-Demand Anodyne PRNP 49 33 CCCNC(=O)c1ccc(NC(=O)c2ccn(-c3cccc(F)c3)n2)cc1 ZINC000147492434 FG On-Demand Anodyne PLD2 32 40 Cc1nc(N(C)Cc2ccc(F)cc2)ccc1C(=O)O ZINC000147492442 CF For-Sale Anodyne PK7 0 42 Cc1nc(N(C)Cc2ccc(F)cc2)ccc1C(=O)O ZINC000147492442 CF For-Sale Anodyne HAO2 34 41 CCc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147492445 BF For-Sale Anodyne P2RY14 43 33 CCc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147492445 BF For-Sale Anodyne NAMPT 0 43 O=C(N1CCC[C@H]1CCCBr)C1(c2ccccc2)CC1 ZINC000147492479 EH For-Sale Reactive PREP 42 33 COc1ccc(Br)cc1CNC(=O)Nc1ccc(Cl)c(C(N)=O)c1 ZINC000147492481 HH On-Demand Anodyne ROCK2 18 46 COc1ccc(Br)cc1CNC(=O)Nc1ccc(Cl)c(C(N)=O)c1 ZINC000147492481 HH On-Demand Anodyne ENPP1 46 34 C[C@@H](CNc1ccc(Br)cc1[N+](=O)[O-])CC(=O)O ZINC000147492571 DF For-Sale Bother COLA 62 34 Cc1nc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cs1 ZINC000147492574 CG For-Sale Anodyne JUN 19 42 Cc1nc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cs1 ZINC000147492574 CG For-Sale Anodyne ATF1 47 38 Cc1nc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cs1 ZINC000147492574 CG For-Sale Anodyne NFKB1 44 38 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc3nccnc3c2)C1 ZINC000147492579 ED On-Demand Anodyne CACNA1I 47 34 Cc1ccc(C)c(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147492586 CG For-Sale Anodyne ADRB2 37 52 Cc1ccc(C)c(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147492586 CG For-Sale Anodyne ADRB1 61 40 Cc1ccc(C)c(OC[C@@H](O)CNCCCCC(C)C)c1 ZINC000147492586 CG For-Sale Anodyne ABCB1 0 48 CCOc1ccc(/C=C/C(=O)N2CCN(c3cnccn3)CC2)cc1 ZINC000147492608 EE On-Demand Anodyne CCR2 0 42 CCOc1ccc(/C=C/C(=O)N2CCN(c3cnccn3)CC2)cc1 ZINC000147492608 EE On-Demand Anodyne GPR183 0 46 CNCCC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147492619 CD For-Sale Bother CACNA1C 46 36 CNCCC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147492619 CD For-Sale Bother CACNA1D 75 35 CC(C)C[C@@H](NC(=O)c1ccc(Br)c(Cl)c1)C(=O)N(C)C ZINC000147492629 GG For-Sale Anodyne CTSL 18 40 CC(C)C[C@@H](NC(=O)c1ccc(Br)c(Cl)c1)C(=O)N(C)C ZINC000147492629 GG For-Sale Anodyne CCKBR 16 40 CC(C)C[C@@H](NC(=O)c1ccc(Br)c(Cl)c1)C(=O)N(C)C ZINC000147492629 GG For-Sale Anodyne UTS2 44 33 O=[N+]([O-])c1cnc2ccccc2c1SCc1ccccc1 ZINC000147492633 CI On-Demand Bother GSTM2 29 45 O=[N+]([O-])c1cnc2ccccc2c1SCc1ccccc1 ZINC000147492633 CI On-Demand Bother GSTP1 22 45 Cc1nc(N(C)Cc2cccc(Cl)c2)ccc1C(=O)O ZINC000147492673 CG For-Sale Anodyne AKR1C1 40 33 Cc1ccc(CNC(=O)CC2(CN)CCC2)cc1 ZINC000147492686 BE For-Sale Anodyne CACNA2D1 0 40 Cc1ccc(CNC(=O)CC2(CN)CCC2)cc1 ZINC000147492686 BE For-Sale Anodyne TPSAB1 18 44 CCCCc1ccc(OC[C@H](O)C(C)C)cc1 ZINC000147492700 BG For-Sale Anodyne ADRB2 22 51 CCCCc1ccc(OC[C@H](O)C(C)C)cc1 ZINC000147492700 BG For-Sale Anodyne ADRB1 30 51 CCCCc1ccc(OC[C@H](O)C(C)C)cc1 ZINC000147492700 BG For-Sale Anodyne INHA 44 33 CCCCc1ccc(OC[C@H](O)C(C)C)cc1 ZINC000147492700 BG For-Sale Anodyne ADRB3 23 42 CCCCc1ccc(OC[C@H](O)C(C)C)cc1 ZINC000147492700 BG For-Sale Anodyne SCN2A 19 44 CCCCc1ccc(OC[C@H](O)C(C)C)cc1 ZINC000147492700 BG For-Sale Anodyne S1PR4 30 47 CCCCc1ccc(OC[C@H](O)C(C)C)cc1 ZINC000147492700 BG For-Sale Anodyne PLA2G4B 44 35 CCCCc1ccc(OC[C@H](O)C(C)C)cc1 ZINC000147492700 BG For-Sale Anodyne S1PR2 40 47 CCCCc1ccc(OC[C@H](O)C(C)C)cc1 ZINC000147492700 BG For-Sale Anodyne S1PR1 15 51 CCCCc1ccc(OC[C@H](O)C(C)C)cc1 ZINC000147492700 BG For-Sale Anodyne S1PR5 23 47 Cc1ccc(CC(=O)N2CCC[C@@H]2CCCBr)cc1C ZINC000147492765 EI For-Sale Reactive OPRK1 34 47 C[C@H](CNc1cc2ccccc2c(=O)[nH]1)CC(=O)O ZINC000147492776 CE For-Sale Anodyne CDC25B 25 57 CCC[C@](C)(N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147492809 CF For-Sale Bother CACNA1D 45 34 Cc1ccc(Br)c(C(=O)N[C@@H](CC(C)C)C(=O)N(C)C)c1 ZINC000147492814 FF For-Sale Anodyne ANPEP 38 45 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc3nccnc3c2)C1 ZINC000147492821 ED On-Demand Anodyne CACNA1I 47 34 COc1cc(N/C(=C/[N+](=O)[O-])NCCCn2cnc(C)c2)cc(OC)c1OC ZINC000147492835 GE Annotated Anodyne QPCT 61 55 COC(=O)c1ccc(CNC(=O)NCc2cc(Br)ccc2OC)cc1 ZINC000147492860 HG On-Demand Anodyne PPARA 16 47 COC(=O)c1ccc(CNC(=O)NCc2cc(Br)ccc2OC)cc1 ZINC000147492860 HG On-Demand Anodyne TRPV1 17 41 COC(=O)c1ccc(CNC(=O)NCc2cc(Br)ccc2OC)cc1 ZINC000147492860 HG On-Demand Anodyne PPARD 23 47 COC(=O)c1ccc(CNC(=O)NCc2cc(Br)ccc2OC)cc1 ZINC000147492860 HG On-Demand Anodyne MT-ND1 24 41 Cc1nc(N(C)Cc2ccccc2Cl)ccc1C(=O)O ZINC000147492900 CG For-Sale Anodyne DXS 0 42 CCCCc1ccc(OC[C@@H](O)C(C)C)cc1 ZINC000147492912 BG For-Sale Anodyne ADRB2 22 51 CCCCc1ccc(OC[C@@H](O)C(C)C)cc1 ZINC000147492912 BG For-Sale Anodyne ADRB1 30 51 CCCCc1ccc(OC[C@@H](O)C(C)C)cc1 ZINC000147492912 BG For-Sale Anodyne INHA 44 33 CCCCc1ccc(OC[C@@H](O)C(C)C)cc1 ZINC000147492912 BG For-Sale Anodyne ADRB3 23 42 CCCCc1ccc(OC[C@@H](O)C(C)C)cc1 ZINC000147492912 BG For-Sale Anodyne SCN2A 19 44 CCCCc1ccc(OC[C@@H](O)C(C)C)cc1 ZINC000147492912 BG For-Sale Anodyne S1PR4 30 47 CCCCc1ccc(OC[C@@H](O)C(C)C)cc1 ZINC000147492912 BG For-Sale Anodyne PLA2G4B 44 35 CCCCc1ccc(OC[C@@H](O)C(C)C)cc1 ZINC000147492912 BG For-Sale Anodyne S1PR2 40 47 CCCCc1ccc(OC[C@@H](O)C(C)C)cc1 ZINC000147492912 BG For-Sale Anodyne S1PR1 15 51 CCCCc1ccc(OC[C@@H](O)C(C)C)cc1 ZINC000147492912 BG For-Sale Anodyne S1PR5 23 47 Cc1ccc(CC(=O)N2CCC[C@H]2CCCBr)cc1C ZINC000147492954 EI For-Sale Reactive OPRK1 34 47 C[C@@H](CNc1cc2ccccc2c(=O)[nH]1)CC(=O)O ZINC000147492959 CE For-Sale Anodyne CDC25B 25 57 CCN(C(=O)CC1(CN)CCC1)c1ccccc1 ZINC000147492963 BF For-Sale Anodyne CACNA2D1 35 43 CCCCOC(=S)c1ccccc1 ZINC000147492980 AG For-Sale Anodyne PLA2G4B 57 37 CCC[C@@](C)(N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147492991 CF For-Sale Bother CACNA1C 41 37 CCC[C@@](C)(N)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147492991 CF For-Sale Bother CACNA1D 63 34 CCOc1ccc(C#N)cc1NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147492995 FG On-Demand Mild ROCK2 35 45 Cc1ccc(Br)c(C(=O)N[C@H](CC(C)C)C(=O)N(C)C)c1 ZINC000147492998 FF For-Sale Anodyne ANPEP 38 45 CC(C)CCCCNC[C@H](O)c1ccc(CC(C)C)cc1 ZINC000147493000 CI For-Sale Anodyne ADRB2 46 44 CC(C)CCCCNC[C@H](O)c1ccc(CC(C)C)cc1 ZINC000147493000 CI For-Sale Anodyne ADRB1 37 44 CC(C)CCCCNC[C@H](O)c1ccc(CC(C)C)cc1 ZINC000147493000 CI For-Sale Anodyne ADRB3 44 41 CC(C)CCCCNC[C@H](O)c1ccc(CC(C)C)cc1 ZINC000147493000 CI For-Sale Anodyne LEF 40 33 COc1ccc(Br)cc1CNC(=O)NC[C@H]1COc2ccccc2O1 ZINC000147493062 HG On-Demand Anodyne ADRA1B 16 45 COc1ccc(Br)cc1CNC(=O)NC[C@H]1COc2ccccc2O1 ZINC000147493062 HG On-Demand Anodyne ADRA2B 16 45 Cc1cn(CCCN/C(=C\[N+](=O)[O-])Nc2ccc3c(c2)OCO3)cn1 ZINC000147493082 EE Annotated Anodyne QPCT 71 66 Cc1cn(CCCN/C(=C\[N+](=O)[O-])Nc2ccc3c(c2)OCO3)cn1 ZINC000147493082 EE Annotated Anodyne DYRK2 53 34 CC(C)CCCCNC[C@@H](O)c1ccc(CC(C)C)cc1 ZINC000147493160 CI For-Sale Anodyne ADRB2 46 44 CC(C)CCCCNC[C@@H](O)c1ccc(CC(C)C)cc1 ZINC000147493160 CI For-Sale Anodyne ADRB1 37 44 CC(C)CCCCNC[C@@H](O)c1ccc(CC(C)C)cc1 ZINC000147493160 CI For-Sale Anodyne ADRB3 44 41 CC(C)CCCCNC[C@@H](O)c1ccc(CC(C)C)cc1 ZINC000147493160 CI For-Sale Anodyne LEF 40 33 CN(C)[C@H]1CCN(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)C1 ZINC000147493191 DE On-Demand Anodyne CACNA1I 43 34 CCC[C@](C)(N)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147493201 CF For-Sale Bother CACNA1C 41 37 CCC[C@](C)(N)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147493201 CF For-Sale Bother CACNA1D 63 34 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccccc2C(=O)N2CCC(C)CC2)C1 ZINC000147493202 HE On-Demand Anodyne HTR4 42 34 COc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147493230 BE For-Sale Anodyne PDGFRB 21 44 COc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147493230 BE For-Sale Anodyne MTNR1A 76 51 COc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147493230 BE For-Sale Anodyne MTNR1B 72 55 COc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147493230 BE For-Sale Anodyne EPHX2 18 46 COc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147493230 BE For-Sale Anodyne FLT4 21 41 COc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147493230 BE For-Sale Anodyne TAAR1 41 44 COc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147493230 BE For-Sale Anodyne KCNK3 42 37 COC(=O)C[C@@H](NC(=O)c1cnn(-c2ccccc2Cl)c1)c1ccc(F)cc1 ZINC000147493254 HH On-Demand Anodyne UTS2 56 34 COC(=O)C[C@@H](NC(=O)c1cnn(-c2ccccc2Cl)c1)c1ccc(F)cc1 ZINC000147493254 HH On-Demand Anodyne CTSA 76 40 Fc1ccc(CNCCCBr)c(Cl)c1 ZINC000147493280 CG For-Sale Reactive P2RX7 61 40 CC(=O)OC[C@@H]1CC[C@H](n2ccc(N)nc2=O)O1 ZINC000147493313 CC For-Sale Anodyne POLA1 20 45 CC(=O)OC[C@@H]1CC[C@H](n2ccc(N)nc2=O)O1 ZINC000147493313 CC For-Sale Anodyne POLB 41 46 Cc1nc(N(C)Cc2ccc(Br)cc2)ccc1C(=O)O ZINC000147493339 EG For-Sale Anodyne PRS 63 35 COc1ccc(C)cc1[C@H](O)CNCCCCC(C)C ZINC000147493377 CG For-Sale Anodyne ADRB2 18 50 O=C(O)c1cc(Cl)cc(NC(=O)c2ccco2)c1 ZINC000147493388 CF On-Demand Anodyne PPIA 17 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccco2)c1 ZINC000147493388 CF On-Demand Anodyne AKR1C3 22 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccco2)c1 ZINC000147493388 CF On-Demand Anodyne KCNK3 46 57 CCC[C@@](C)(N)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147493394 CF For-Sale Bother CACNA1C 41 37 CCC[C@@](C)(N)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147493394 CF For-Sale Bother CACNA1D 63 34 CCCC[C@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493398 EG On-Demand Anodyne KLK3 44 35 CCCC[C@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493398 EG On-Demand Anodyne CTSK 40 41 CCCC[C@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493398 EG On-Demand Anodyne NPFFR2 42 33 CCCC[C@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493398 EG On-Demand Anodyne PCSK5 42 34 CCCC[C@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493398 EG On-Demand Anodyne FURIN 53 34 CCCC[C@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493398 EG On-Demand Anodyne POLG_WNV 75 34 CCCC[C@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493398 EG On-Demand Anodyne NPFFR1 54 33 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccccc2C(=O)N2CCC(C)CC2)C1 ZINC000147493424 HE On-Demand Anodyne HTR4 42 34 C[C@H]1CCC[C@@H](C)N1NC(=O)CCCN ZINC000147493430 BD For-Sale Anodyne ABAT 40 33 COC(=O)C[C@H](NC(=O)[C@H]1COc2cc(OC)ccc2C1)c1ccc(F)cc1 ZINC000147493471 GF On-Demand Anodyne ROCK2 27 41 COc1ccc(C(=O)O)c(NCC2(N(C)C)CCCC2)c1 ZINC000147493473 CF For-Sale Anodyne SLC6A5 15 42 COc1ccc(C(=O)O)c(NCC2(N(C)C)CCCC2)c1 ZINC000147493473 CF For-Sale Anodyne AKR1C3 28 50 COc1ccc(C(=O)O)c(NCC2(N(C)C)CCCC2)c1 ZINC000147493473 CF For-Sale Anodyne AKR1C2 73 50 COc1ccc(CNCCCBr)cc1 ZINC000147493509 CF For-Sale Reactive LPAR2 44 40 COc1ccc(CNCCCBr)cc1 ZINC000147493509 CF For-Sale Reactive S1PR2 52 40 COc1ccc(CNCCCBr)cc1 ZINC000147493509 CF For-Sale Reactive LEF 24 41 COc1ccc(CNCCCBr)cc1 ZINC000147493509 CF For-Sale Reactive PROKR1 60 33 COc1ccc(CNCCCBr)cc1 ZINC000147493509 CF For-Sale Reactive LMGT2 0 61 COc1ccc(C)cc1[C@@H](O)CNCCCCC(C)C ZINC000147493583 CG For-Sale Anodyne ADRB2 18 50 CCCC[C@@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493602 EG On-Demand Anodyne KLK3 44 35 CCCC[C@@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493602 EG On-Demand Anodyne CTSK 40 41 CCCC[C@@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493602 EG On-Demand Anodyne NPFFR2 42 33 CCCC[C@@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493602 EG On-Demand Anodyne PCSK5 42 34 CCCC[C@@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493602 EG On-Demand Anodyne FURIN 53 34 CCCC[C@@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493602 EG On-Demand Anodyne POLG_WNV 75 34 CCCC[C@@H](NC(N)=O)C(=O)NCC1(c2ccccc2)CCCCC1 ZINC000147493602 EG On-Demand Anodyne NPFFR1 54 33 C[C@H]1CCC[C@H](C)N1NC(=O)CCCN ZINC000147493604 BD For-Sale Anodyne ABAT 40 33 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)nc1 ZINC000147493608 DF On-Demand Mild BACE2 33 41 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)nc1 ZINC000147493608 DF On-Demand Mild ATF1 47 38 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)nc1 ZINC000147493608 DF On-Demand Mild GRM5 22 42 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)nc1 ZINC000147493608 DF On-Demand Mild NFKB1 43 38 N#Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)nc1 ZINC000147493608 DF On-Demand Mild SCN10A 29 43 COC(=O)C[C@H](NC(=O)[C@H](C)OCCC(C)C)c1ccccc1 ZINC000147493633 DF On-Demand Anodyne KCNA5 29 41 COC(=O)C[C@H](NC(=O)[C@H](C)OCCC(C)C)c1ccccc1 ZINC000147493633 DF On-Demand Anodyne SOAT1 25 40 CC[C@@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493640 BE On-Demand Anodyne SLC6A1 61 35 CC[C@@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493640 BE On-Demand Anodyne LTA4H 62 55 CC[C@@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493640 BE On-Demand Anodyne HRH3 49 40 CC[C@@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493640 BE On-Demand Anodyne SIGMAR1 27 41 CC[C@@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493640 BE On-Demand Anodyne CHRNA10 44 42 CC[C@@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493640 BE On-Demand Anodyne GRIN3A 0 46 CC[C@@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493640 BE On-Demand Anodyne PSMB2 53 44 CC[C@@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493640 BE On-Demand Anodyne PSMB1 46 44 CC[C@@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493640 BE On-Demand Anodyne MEN1 48 38 CC[C@@H](C)[C@H](N)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147493649 CE For-Sale Bother CACNA1C 57 40 CC[C@@H](C)[C@H](N)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147493649 CE For-Sale Bother CACNA1D 89 37 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493662 HG On-Demand Anodyne DRD4 46 36 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493662 HG On-Demand Anodyne HTR4 44 35 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493662 HG On-Demand Anodyne CCR3 41 43 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493662 HG On-Demand Anodyne MTNR1A 35 51 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493662 HG On-Demand Anodyne MTNR1B 41 51 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493662 HG On-Demand Anodyne FAAH 17 41 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493662 HG On-Demand Anodyne MCHR1 27 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493662 HG On-Demand Anodyne CACNA1I 56 35 CCN1CCN(c2ccc(C(=O)NCCN3CCCS3(=O)=O)cc2F)CC1 ZINC000147493670 GC On-Demand Anodyne HTR1A 25 45 CCN1CCN(c2ccc(C(=O)NCCN3CCCS3(=O)=O)cc2F)CC1 ZINC000147493670 GC On-Demand Anodyne DRD2 32 45 CCN1CCN(c2ccc(C(=O)NCCN3CCCS3(=O)=O)cc2F)CC1 ZINC000147493670 GC On-Demand Anodyne DRD1 18 40 CCN1CCN(c2ccc(C(=O)NCCN3CCCS3(=O)=O)cc2F)CC1 ZINC000147493670 GC On-Demand Anodyne DRD4 50 39 CCN1CCN(c2ccc(C(=O)NCCN3CCCS3(=O)=O)cc2F)CC1 ZINC000147493670 GC On-Demand Anodyne DRD3 59 42 CCN1CCN(c2ccc(C(=O)NCCN3CCCS3(=O)=O)cc2F)CC1 ZINC000147493670 GC On-Demand Anodyne NPY2R 41 39 CCN1CCN(c2ccc(C(=O)NCCN3CCCS3(=O)=O)cc2F)CC1 ZINC000147493670 GC On-Demand Anodyne PLD2 47 37 CCN1CCN(c2ccc(C(=O)NCCN3CCCS3(=O)=O)cc2F)CC1 ZINC000147493670 GC On-Demand Anodyne CXCR3 19 41 COc1ccc(Br)cc1CNC(=O)Nc1ccc([N+](=O)[O-])cc1 ZINC000147493690 GH On-Demand Bother TSHR 40 30 COc1ccc(Br)cc1CNC(=O)Nc1ccc([N+](=O)[O-])cc1 ZINC000147493690 GH On-Demand Bother NMBR 58 40 COc1ccc(Br)cc1CNC(=O)Nc1ccc([N+](=O)[O-])cc1 ZINC000147493690 GH On-Demand Bother ROCK2 16 48 COc1ccc(Br)cc1CNC(=O)Nc1ccc([N+](=O)[O-])cc1 ZINC000147493690 GH On-Demand Bother GRPR 29 40 COc1ccc(Br)cc1CNC(=O)Nc1ccc([N+](=O)[O-])cc1 ZINC000147493690 GH On-Demand Bother PRMT3 17 42 COC(=O)C[C@H](NC(=O)[C@@H]1COc2cc(OC)ccc2C1)c1ccc(F)cc1 ZINC000147493692 GF On-Demand Anodyne ROCK2 27 41 CN(Cc1cscn1)C(=O)NCc1cccc(NC(=O)C2CCC2)c1 ZINC000147493693 FG On-Demand Anodyne GPR142 29 41 Cc1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147493700 BE For-Sale Anodyne CACNA2D1 25 42 Cc1ccc(NC(=O)CC2(CN)CCC2)cc1 ZINC000147493700 BE For-Sale Anodyne FUCA1 15 41 CN(C)C1(CNc2ccc(C(=O)O)c(F)c2)CCCC1 ZINC000147493701 CF For-Sale Anodyne RARA 27 45 COC(=O)Cc1csc(-c2ccc(Cl)cc2F)n1 ZINC000147493730 CG For-Sale Anodyne PTGER1 25 47 O=C(CCCO)OCCc1ccccc1 ZINC000147493773 BD Annotated Anodyne CES1 49 34 O=C(CCCO)OCCc1ccccc1 ZINC000147493773 BD Annotated Anodyne TSPAN17 0 43 O=C(CCCO)OCCc1ccccc1 ZINC000147493773 BD Annotated Anodyne MGLL 0 46 O=C(CCCO)OCCc1ccccc1 ZINC000147493773 BD Annotated Anodyne FFAR1 30 40 O=C(CCCO)OCCc1ccccc1 ZINC000147493773 BD Annotated Anodyne AKR1B10 23 43 O=C(O)c1cc(Cl)cc(NC(=O)C2[C@H]3CCCC[C@H]23)c1 ZINC000147493788 CG On-Demand Anodyne HCAR1 0 40 Nc1nc(Oc2ccc(I)cc2)nc(N2CCCCC2)n1 ZINC000147493807 GF For-Sale Anodyne ERM 0 41 C[C@@H]1CCC[C@@H](C)N1NC(=O)CCCN ZINC000147493808 BD For-Sale Anodyne ABAT 40 33 COC(=O)C[C@H](NC(=O)[C@@H](C)OCCC(C)C)c1ccccc1 ZINC000147493835 DF On-Demand Anodyne KCNA5 29 41 COC(=O)C[C@H](NC(=O)[C@@H](C)OCCC(C)C)c1ccccc1 ZINC000147493835 DF On-Demand Anodyne SOAT1 25 40 CC[C@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493839 BE On-Demand Anodyne SLC6A1 61 35 CC[C@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493839 BE On-Demand Anodyne LTA4H 62 55 CC[C@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493839 BE On-Demand Anodyne HRH3 49 40 CC[C@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493839 BE On-Demand Anodyne SIGMAR1 27 41 CC[C@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493839 BE On-Demand Anodyne CHRNA10 44 42 CC[C@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493839 BE On-Demand Anodyne GRIN3A 0 46 CC[C@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493839 BE On-Demand Anodyne PSMB2 53 44 CC[C@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493839 BE On-Demand Anodyne PSMB1 46 44 CC[C@H]1CN(CCOc2ccccc2)CC[C@@H]1N ZINC000147493839 BE On-Demand Anodyne MEN1 48 38 CCc1nc(CN(C)C(=O)NCc2cccc(NC(=O)C3CCC3)c2)cs1 ZINC000147493882 GH On-Demand Anodyne AVPR1B 31 42 O=C(NCCN1CCCS1(=O)=O)c1cccnc1N1CCOCC1 ZINC000147493901 FB On-Demand Anodyne HPGDS 23 41 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493920 HG On-Demand Anodyne DRD4 46 36 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493920 HG On-Demand Anodyne HTR4 44 35 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493920 HG On-Demand Anodyne CCR3 41 43 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493920 HG On-Demand Anodyne MTNR1A 35 51 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493920 HG On-Demand Anodyne MTNR1B 41 51 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493920 HG On-Demand Anodyne FAAH 17 41 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493920 HG On-Demand Anodyne MCHR1 27 40 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(Oc3cccc(OC)c3)cc2)C1 ZINC000147493920 HG On-Demand Anodyne CACNA1I 56 35 COC(=O)C[C@@H](NC(=O)[C@@H]1COc2cc(OC)ccc2C1)c1ccc(F)cc1 ZINC000147493933 GF On-Demand Anodyne ROCK2 27 41 COc1ccc(CN(C)c2ccc(C(=O)O)c(C)n2)cc1 ZINC000147493994 CF For-Sale Anodyne AKR1C2 51 39 COCc1nc(C(=O)N2CCN(Cc3ccco3)CC2)cs1 ZINC000147494006 DD On-Demand Anodyne TRPC6 46 34 O=C(O)c1cc(Cl)cc(NC(=O)C2[C@H]3CCCC[C@@H]23)c1 ZINC000147494007 CG For-Sale Anodyne HCAR1 0 40 COC(=O)C[C@@H](NC(=O)[C@H](C)OCCC(C)C)c1ccccc1 ZINC000147494036 DF On-Demand Anodyne KCNA5 29 41 COC(=O)C[C@@H](NC(=O)[C@H](C)OCCC(C)C)c1ccccc1 ZINC000147494036 DF On-Demand Anodyne SOAT1 25 40 CC(=O)Nc1cccc([C@H](C)NC(=O)N(C)Cc2cscn2)c1 ZINC000147494110 EG On-Demand Anodyne BMP1 46 32 CCc1nc(CN(C)S(=O)(=O)c2cccc3cnccc23)cs1 ZINC000147494115 EG On-Demand Anodyne P2RX7 18 44 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne CA2 118 49 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne TSHR 41 32 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne HTR2A 17 41 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne CA1 111 52 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne CA7 56 43 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne CA5B 62 41 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne CA4 78 49 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne CA5A 67 41 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne CA14 45 43 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne ROCK2 17 48 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne CA12 90 55 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne CA9 100 49 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne UREA_CANEN 27 41 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne IDO1 40 38 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne NCE103 54 45 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne MTCA1 62 55 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne P96878_MYCTU 80 55 COc1ccc(Br)cc1CNC(=O)Nc1ccc(S(N)(=O)=O)cc1 ZINC000147494166 HE On-Demand Anodyne NAMPT 35 41 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCN(C)CC3)c1)C2 ZINC000147494185 GF On-Demand Anodyne DRD2 17 44 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCN(C)CC3)c1)C2 ZINC000147494185 GF On-Demand Anodyne DRD4 42 33 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCN(C)CC3)c1)C2 ZINC000147494185 GF On-Demand Anodyne HRH2 31 43 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCN(C)CC3)c1)C2 ZINC000147494185 GF On-Demand Anodyne SIGMAR1 24 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCN(C)CC3)c1)C2 ZINC000147494185 GF On-Demand Anodyne CCR3 23 40 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCN(C)CC3)c1)C2 ZINC000147494185 GF On-Demand Anodyne ROCK2 42 45 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCN(C)CC3)c1)C2 ZINC000147494185 GF On-Demand Anodyne FAAH 23 46 COc1ccc2c(c1)OC[C@@H](C(=O)Nc1cccc(CN3CCN(C)CC3)c1)C2 ZINC000147494185 GF On-Demand Anodyne MCHR1 34 44 Cc1cc(C(=O)N2CCN(C(=O)C(=O)N3CCOCC3)CC2)cc([N+](=O)[O-])c1 ZINC000147494202 GC On-Demand Bother AKR1C3 23 45 COc1cccc(CN(C)c2ccc(C(=O)O)c(C)n2)c1 ZINC000147494221 CF On-Demand Anodyne PLG 0 40 COc1cccc(CN(C)c2ccc(C(=O)O)c(C)n2)c1 ZINC000147494221 CF On-Demand Anodyne PPARG 19 40 COc1cccc(CN(C)c2ccc(C(=O)O)c(C)n2)c1 ZINC000147494221 CF On-Demand Anodyne PPARA 29 40 COc1cccc(CN(C)c2ccc(C(=O)O)c(C)n2)c1 ZINC000147494221 CF On-Demand Anodyne ROCK1 36 41 COc1cccc(CN(C)c2ccc(C(=O)O)c(C)n2)c1 ZINC000147494221 CF On-Demand Anodyne ROCK2 44 40 COc1cccc(CN(C)c2ccc(C(=O)O)c(C)n2)c1 ZINC000147494221 CF On-Demand Anodyne HSD17B2 24 45 COc1cccc(CN(C)c2ccc(C(=O)O)c(C)n2)c1 ZINC000147494221 CF On-Demand Anodyne AKR1C3 22 41 COc1cccc(CN(C)c2ccc(C(=O)O)c(C)n2)c1 ZINC000147494221 CF On-Demand Anodyne CDC42BPA 0 40 COc1cccc(CN(C)c2ccc(C(=O)O)c(C)n2)c1 ZINC000147494221 CF On-Demand Anodyne AKR1C2 52 39 COC(=O)C[C@@H](NC(=O)[C@@H](C)OCCC(C)C)c1ccccc1 ZINC000147494240 DF On-Demand Anodyne KCNA5 29 41 COC(=O)C[C@@H](NC(=O)[C@@H](C)OCCC(C)C)c1ccccc1 ZINC000147494240 DF On-Demand Anodyne SOAT1 25 40 O=C(O)c1cc(Cl)cc(NC(=O)C2[C@@H]3CCCC[C@@H]23)c1 ZINC000147494242 CG On-Demand Anodyne HCAR1 0 40 CCCNc1cn2ccnc2c(Oc2ccc(I)cc2)n1 ZINC000147494258 GH For-Sale Anodyne HIVRT 0 40 CCOC(=O)c1ccc2c(C3CCCC3)c(-c3ccoc3)sc2c1 ZINC000147494259 EK For-Sale Anodyne NS5B 0 73 CN[C@H](C)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147494298 CD For-Sale Bother CACNA1D 50 35 CC(=O)Nc1cccc([C@@H](C)NC(=O)N(C)Cc2cscn2)c1 ZINC000147494304 EG On-Demand Anodyne BMP1 46 32 CC[C@@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494328 CD On-Demand Anodyne DRD4 43 34 CC[C@@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494328 CD On-Demand Anodyne KCNH2 22 40 CC[C@@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494328 CD On-Demand Anodyne KCNA5 0 40 CC[C@@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494328 CD On-Demand Anodyne CCR3 38 45 CC[C@@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494328 CD On-Demand Anodyne MTNR1A 30 46 CC[C@@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494328 CD On-Demand Anodyne MTNR1B 41 46 CC[C@@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494328 CD On-Demand Anodyne MCHR1 35 40 CC[C@@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494328 CD On-Demand Anodyne KCNK3 41 35 CC(C)(C)OC(=O)N1CCN(c2ncnc3sc([N+](=O)[O-])cc23)CC1 ZINC000147494379 FF On-Demand Bother PDGFRB 31 40 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne ABL1 45 41 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne HTR1A 28 44 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne DRD2 42 44 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne DRD4 56 38 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne HTR1D 24 42 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne HTR1B 39 42 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne HTR2A 26 44 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne HTR2C 24 44 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne DRD3 44 36 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne KIT 22 49 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne LCK 17 44 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne IKBKB 57 36 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne FLT1 27 40 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne KDR 26 44 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne FAAH 24 42 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne MAPK10 21 42 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne FLT3 20 44 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne CSF1R 23 44 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne MCHR1 36 41 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne AURKA 20 41 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne FRK 16 41 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne DDR1 45 43 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne DDR2 29 43 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne NOD2 41 35 CN1CCN(Cc2cccc(NC(=O)c3cnn(-c4ccccc4Cl)c3)c2)CC1 ZINC000147494403 HH On-Demand Anodyne KCNK3 59 37 CCc1ncc(C(=O)N2CCN(c3cccc(C)c3)CC2)s1 ZINC000147494427 DF On-Demand Anodyne CCKBR 18 41 COc1ccccc1CN(C)c1ccc(C(=O)O)c(C)n1 ZINC000147494458 CF For-Sale Anodyne TSPO 24 40 O=C(CC[C@@H]1CCCCO1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147494473 DG On-Demand Anodyne LDLR 0 41 CN[C@H](C)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147494504 CD For-Sale Bother CACNA1D 50 35 CC[C@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494543 CD On-Demand Anodyne DRD4 43 34 CC[C@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494543 CD On-Demand Anodyne KCNH2 22 40 CC[C@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494543 CD On-Demand Anodyne KCNA5 0 40 CC[C@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494543 CD On-Demand Anodyne CCR3 38 45 CC[C@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494543 CD On-Demand Anodyne MTNR1A 30 46 CC[C@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494543 CD On-Demand Anodyne MTNR1B 41 46 CC[C@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494543 CD On-Demand Anodyne MCHR1 35 40 CC[C@H]1CN(CC(=O)Nc2cccc(OC)c2)CC[C@@H]1N ZINC000147494543 CD On-Demand Anodyne KCNK3 41 35 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccc(NC(=O)c2ccccc2)c1 ZINC000147494545 GI On-Demand Anodyne BMP1 52 33 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccc(NC(=O)c2ccccc2)c1 ZINC000147494545 GI On-Demand Anodyne CYP3A4 16 43 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccc(NC(=O)c2ccccc2)c1 ZINC000147494545 GI On-Demand Anodyne GPR142 32 40 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccc(NC(=O)c2ccccc2)c1 ZINC000147494545 GI On-Demand Anodyne KCNK3 96 41 C[C@H](NC(=O)N(C)Cc1cscn1)c1cccc(NC(=O)c2ccccc2)c1 ZINC000147494545 GI On-Demand Anodyne KCNK9 49 38 Cc1cc(N(C)C)ccc1NC(=O)c1ccc(Br)c(Cl)c1 ZINC000147494551 FJ On-Demand Anodyne KCNK3 15 41 CC(C)CCCCNCCc1ccncc1 ZINC000147494569 BG On-Demand Anodyne GNRHR 20 40 CC(C)CCCCNCCc1ccncc1 ZINC000147494569 BG On-Demand Anodyne FDFT1 0 40 O=C(CC[C@H]1CCCCO1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147494656 DG On-Demand Anodyne LDLR 0 41 CC(C)C[C@H](CN)Nc1cc(Nc2cccc(C(C)(C)C)n2)c(C(N)=O)nn1 ZINC000147494683 GF Annotated Anodyne SYK 23 55 CC(=O)Oc1cc(O)ccc1C(=O)O ZINC000147494695 AD For-Sale Anodyne POBA 0 54 CC(=O)Oc1cc(O)ccc1C(=O)O ZINC000147494695 AD For-Sale Anodyne AKR1C2 42 32 O=C(NCC1(c2ccccc2)CC1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147494720 HG On-Demand Anodyne KCNA3 44 38 O=C(NCC1(c2ccccc2)CC1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147494720 HG On-Demand Anodyne MAP1 72 36 O=C(NCC1(c2ccccc2)CC1)c1ccc(S(=O)(=O)Nc2nccs2)cc1 ZINC000147494720 HG On-Demand Anodyne LIMK2 48 35 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccc(NC(=O)c2ccccc2)c1 ZINC000147494732 GI On-Demand Anodyne BMP1 52 33 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccc(NC(=O)c2ccccc2)c1 ZINC000147494732 GI On-Demand Anodyne CYP3A4 16 43 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccc(NC(=O)c2ccccc2)c1 ZINC000147494732 GI On-Demand Anodyne GPR142 32 40 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccc(NC(=O)c2ccccc2)c1 ZINC000147494732 GI On-Demand Anodyne KCNK3 96 41 C[C@@H](NC(=O)N(C)Cc1cscn1)c1cccc(NC(=O)c2ccccc2)c1 ZINC000147494732 GI On-Demand Anodyne KCNK9 49 38 CN[C@@H](C)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147494734 CD For-Sale Bother CACNA1D 50 35 O=C(CCl)c1ccc(-c2ccc([N+](=O)[O-])cc2)o1 ZINC000147494762 CG For-Sale Reactive ERCC5 16 49 O=C(CCl)c1ccc(-c2ccc([N+](=O)[O-])cc2)o1 ZINC000147494762 CG For-Sale Reactive LUXR 16 41 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147494782 ED On-Demand Anodyne HDAC10 43 38 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147494782 ED On-Demand Anodyne MMP3 15 43 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147494782 ED On-Demand Anodyne HDAC11 41 38 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147494782 ED On-Demand Anodyne POLG_WNV 41 36 CCCCCCCCCCCCNCCCCC(C)C ZINC000147494785 CK For-Sale Mild ADH1A 0 47 CCCCCCCCCCCCNCCCCC(C)C ZINC000147494785 CK For-Sale Mild ADH7 0 44 CCCCCCCCCCCCNCCCCC(C)C ZINC000147494785 CK For-Sale Mild S1PR3 21 50 CCCCCCCCCCCCNCCCCC(C)C ZINC000147494785 CK For-Sale Mild S1PR2 47 50 CCCCCCCCCCCCNCCCCC(C)C ZINC000147494785 CK For-Sale Mild ADH1B 0 47 CCCCCCCCCCCCNCCCCC(C)C ZINC000147494785 CK For-Sale Mild ADH1C 0 47 CCCCCCCCCCCCNCCCCC(C)C ZINC000147494785 CK For-Sale Mild Q8WS26_TRYCR 41 42 CCCCCCCCCCCCNCCCCC(C)C ZINC000147494785 CK For-Sale Mild FPPS 0 42 CCCCCCCCCCCCNCCCCC(C)C ZINC000147494785 CK For-Sale Mild SPPS 0 42 CC[C@@H]1CN(CC(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147494799 CD On-Demand Anodyne DRD4 25 62 CC[C@@H]1CN(CC(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147494799 CD On-Demand Anodyne KCNK3 41 37 CC[C@@H]1CN(CC(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147494799 CD On-Demand Anodyne KCNK9 46 37 Cc1ccccc1CC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147494896 DH On-Demand Anodyne PTGER1 15 43 Cc1ccccc1CC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147494896 DH On-Demand Anodyne AKR1C3 33 40 CC1CCC(NC(=O)CC2(CN)CCC2)CC1 ZINC000147494907 BE For-Sale Anodyne CACNA2D1 40 42 O=C(NCCc1ccc2ccccc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147494914 GI On-Demand Anodyne DRTS_PLAFK 21 44 O=C(NCCc1ccc2ccccc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147494914 GI On-Demand Anodyne PTGER3 37 41 O=C(NCCc1ccc2ccccc2c1)c1cccn(Cc2ccccc2)c1=O ZINC000147494914 GI On-Demand Anodyne POLR1A 80 38 CCCNc1cc(Oc2ccc(I)cc2)cc([N+](=O)[O-])c1 ZINC000147494928 GJ For-Sale Bother TBXA2R 16 46 CN[C@@H](C)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147494938 CD For-Sale Bother CACNA1D 50 35 O=C(NCCn1cnc(C(=O)O)c1)c1ccccc1 ZINC000147494948 CD For-Sale Anodyne HTR1A 16 46 O=C(NCCn1cnc(C(=O)O)c1)c1ccccc1 ZINC000147494948 CD For-Sale Anodyne DRD2 16 42 O=C(NCCn1cnc(C(=O)O)c1)c1ccccc1 ZINC000147494948 CD For-Sale Anodyne DRD4 42 33 O=C(NCCn1cnc(C(=O)O)c1)c1ccccc1 ZINC000147494948 CD For-Sale Anodyne DRD3 30 40 O=C(NCCn1cnc(C(=O)O)c1)c1ccccc1 ZINC000147494948 CD For-Sale Anodyne HTR3B 0 40 O=C(NCCn1cnc(C(=O)O)c1)c1ccccc1 ZINC000147494948 CD For-Sale Anodyne PLD2 46 34 O=C(NCCn1cnc(C(=O)O)c1)c1ccccc1 ZINC000147494948 CD For-Sale Anodyne KDM4E 23 41 O=C(N[C@@H]1CCN2CCCC[C@H]12)c1ccc(Br)c(Cl)c1 ZINC000147494952 FG On-Demand Anodyne VACHT_TETCF 0 41 O=C(N[C@@H]1CCN2CCCC[C@H]12)c1ccc(Br)c(Cl)c1 ZINC000147494952 FG On-Demand Anodyne SIGMAR1 0 50 O=C(N[C@@H]1CCN2CCCC[C@H]12)c1ccc(Br)c(Cl)c1 ZINC000147494952 FG On-Demand Anodyne L3MBTL3 54 33 Cc1nc(N2CCN(C(C)(C)C)CC2)ccc1C(=O)O ZINC000147494981 CE For-Sale Anodyne SORD 40 34 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147494995 ED On-Demand Anodyne HDAC10 43 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147494995 ED On-Demand Anodyne MMP3 15 43 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147494995 ED On-Demand Anodyne HDAC11 41 38 CCCC[C@@H](NC(N)=O)C(=O)Nc1cccc(OCC(=O)OC)c1 ZINC000147494995 ED On-Demand Anodyne POLG_WNV 41 36 CC[C@H]1CN(CC(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147495016 CD On-Demand Anodyne DRD4 25 62 CC[C@H]1CN(CC(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147495016 CD On-Demand Anodyne KCNK3 41 37 CC[C@H]1CN(CC(=O)Nc2cccc(C)c2)CC[C@@H]1N ZINC000147495016 CD On-Demand Anodyne KCNK9 46 37 O=C(NCCC(F)(F)F)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147495113 DG On-Demand Anodyne CACNA1H 24 40 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne RARA 16 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne PPIA 19 52 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne ATF1 40 38 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne CPT1A 29 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne PRNP 33 49 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne JAK1 0 47 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne GRM4 43 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne CSF1R 18 46 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne TAAR1 18 45 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne AKR1C3 25 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne SHH 36 47 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne HCAR1 0 42 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne KCNK3 85 56 O=C(O)c1cc(Cl)cc(NC(=O)c2ccncc2)c1 ZINC000147495124 CF On-Demand Anodyne KCNK9 34 40 O=C(N[C@H]1CCN2CCCC[C@H]12)c1ccc(Br)c(Cl)c1 ZINC000147495130 FG On-Demand Anodyne VACHT_TETCF 0 41 O=C(N[C@H]1CCN2CCCC[C@H]12)c1ccc(Br)c(Cl)c1 ZINC000147495130 FG On-Demand Anodyne SIGMAR1 0 50 O=C(N[C@H]1CCN2CCCC[C@H]12)c1ccc(Br)c(Cl)c1 ZINC000147495130 FG On-Demand Anodyne L3MBTL3 54 33 NC1(C(=O)N2CCCc3ccccc32)CCC1 ZINC000147495131 BD For-Sale Anodyne AVPR2 33 42 NC1(C(=O)N2CCCc3ccccc32)CCC1 ZINC000147495131 BD For-Sale Anodyne SLC7A5 0 40 C[C@@H](CN)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147495168 CD For-Sale Bother CACNA1C 54 38 C[C@@H](CN)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147495168 CD For-Sale Bother CACNA1D 83 36 C[C@@H](CN)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147495168 CD For-Sale Bother TRPM8 0 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(CCN3CCOCC3)cc2)C1 ZINC000147495208 HD On-Demand Anodyne HTR4 54 41 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(CCN3CCOCC3)cc2)C1 ZINC000147495208 HD On-Demand Anodyne CCR3 43 42 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(CCN3CCOCC3)cc2)C1 ZINC000147495208 HD On-Demand Anodyne BIRC2 51 33 Cc1cnn(CC(=O)Nc2ccc3c(c2)N(S(N)(=O)=O)CC3)c1 ZINC000147495220 EC In-Stock Anodyne CPT1A 15 40 Cc1nc(N(Cc2ccsc2)C2CC2)ccc1C(=O)O ZINC000147495281 CG For-Sale Anodyne HCAR3 23 40 CC[C@@H]1CN(CC(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147495289 CD On-Demand Anodyne KCNA5 0 52 COC(=O)C[C@H](NC(=O)Cc1cccc(OC(C)C)c1)c1ccccc1 ZINC000147495315 FG On-Demand Anodyne KCNA5 41 39 COC(=O)C[C@H](NC(=O)Cc1cccc(OC(C)C)c1)c1ccccc1 ZINC000147495315 FG On-Demand Anodyne PTGER3 45 37 COC(=O)C[C@H](NC(=O)Cc1cccc(OC(C)C)c1)c1ccccc1 ZINC000147495315 FG On-Demand Anodyne SOAT1 27 47 COC(=O)C[C@H](NC(=O)Cc1cccc(OC(C)C)c1)c1ccccc1 ZINC000147495315 FG On-Demand Anodyne PDS 42 36 O=C(O)c1cc(Cl)cc(NC(=O)C2CCC2)c1 ZINC000147495358 CF On-Demand Anodyne INHA 22 46 O=C(O)c1cc(Cl)cc(NC(=O)C2CCC2)c1 ZINC000147495358 CF On-Demand Anodyne CACNA1I 45 36 O=C(O)c1cc(Cl)cc(NC(=O)C2CCC2)c1 ZINC000147495358 CF On-Demand Anodyne RHOA 0 42 O=C(O)c1cc(Cl)cc(NC(=O)C2CCC2)c1 ZINC000147495358 CF On-Demand Anodyne HCAR1 0 42 NCC1(CC(=O)N2CCCc3ccccc32)CCC1 ZINC000147495364 CE For-Sale Anodyne AVPR2 43 47 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](C)CN ZINC000147495365 CD For-Sale Bother CACNA1C 54 38 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](C)CN ZINC000147495365 CD For-Sale Bother CACNA1D 83 36 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](C)CN ZINC000147495365 CD For-Sale Bother TRPM8 0 40 Cc1ccc(Br)c(C(=O)N[C@@H]2CCN3CCCC[C@H]23)c1 ZINC000147495394 EG On-Demand Anodyne SIGMAR1 0 42 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(CCN3CCOCC3)cc2)C1 ZINC000147495413 HD On-Demand Anodyne HTR4 54 41 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(CCN3CCOCC3)cc2)C1 ZINC000147495413 HD On-Demand Anodyne CCR3 43 42 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(CCN3CCOCC3)cc2)C1 ZINC000147495413 HD On-Demand Anodyne BIRC2 51 33 Clc1ccc(-c2cccc3cn[nH]c23)c(Cl)c1 ZINC000147495434 CJ For-Sale Anodyne ALPL 43 35 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne KIT 33 52 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne CNR2 15 43 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne TRPV1 15 54 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne GUAB 0 49 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne RAF1 58 57 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne FLT1 15 42 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne KDR 17 47 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne EPHX2 15 46 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne PDGFRA 19 53 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne FLT3 71 57 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne CSF1R 26 55 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne Q8MMZ8_EIMTE 99 67 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne RET 24 53 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne BRAF 19 45 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne PTPA 0 44 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne RIPK1 34 47 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne PFK 0 43 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne IMDH_CRYPV 40 49 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne BLM 0 49 CC(C)(C)c1cc(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)no1 ZINC000147495500 FK For-Sale Anodyne P95276_MYCTO 0 41 CC[C@H]1CN(CC(=O)Nc2ccc(OC)cc2)CC[C@@H]1N ZINC000147495502 CD On-Demand Anodyne KCNA5 0 52 COC(=O)C[C@@H](NC(=O)Cc1cccc(OC(C)C)c1)c1ccccc1 ZINC000147495511 FG On-Demand Anodyne KCNA5 41 39 COC(=O)C[C@@H](NC(=O)Cc1cccc(OC(C)C)c1)c1ccccc1 ZINC000147495511 FG On-Demand Anodyne PTGER3 45 37 COC(=O)C[C@@H](NC(=O)Cc1cccc(OC(C)C)c1)c1ccccc1 ZINC000147495511 FG On-Demand Anodyne SOAT1 27 47 COC(=O)C[C@@H](NC(=O)Cc1cccc(OC(C)C)c1)c1ccccc1 ZINC000147495511 FG On-Demand Anodyne PDS 42 36 COC(=O)C[C@@H](NC(=O)c1ccc2c(c1)COC2)c1ccc(F)cc1 ZINC000147495545 EF On-Demand Anodyne UTS2 46 33 C[C@@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147495558 CD For-Sale Bother CACNA1C 54 38 C[C@@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147495558 CD For-Sale Bother CACNA1D 83 36 C[C@@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147495558 CD For-Sale Bother TRPM8 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cccs2)c1 ZINC000147495585 CG On-Demand Anodyne AKR1C3 22 42 O=C(O)c1cc(Cl)cc(NC(=O)c2cccs2)c1 ZINC000147495585 CG On-Demand Anodyne KCNK3 49 57 O=C(O)c1cc(Cl)cc(NC(=O)c2cccs2)c1 ZINC000147495585 CG On-Demand Anodyne KCNK9 28 57 Cc1ccc(Br)c(C(=O)N[C@H]2CCN3CCCC[C@H]23)c1 ZINC000147495588 EG On-Demand Anodyne SIGMAR1 0 42 CCCN1CCN(C(=O)CC2(CN)CCC2)CC1 ZINC000147495620 CD For-Sale Anodyne CACNA2D1 0 41 C=CC(=O)c1ccc(C(C)=O)cc1 ZINC000147495668 AE For-Sale Mild ALDH5A1 0 64 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCC[C@H](Br)C1 ZINC000147495700 FE For-Sale Reactive PKM 53 63 COc1ccc(Br)cc1C[C@H](O)c1cncs1 ZINC000147495739 DG For-Sale Anodyne PHES 0 40 C[C@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147495740 CD For-Sale Bother CACNA1C 54 38 C[C@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147495740 CD For-Sale Bother CACNA1D 83 36 C[C@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147495740 CD For-Sale Bother TRPM8 0 40 CC(C)CCCCNCC(=O)Nc1c(Cl)cccc1Cl ZINC000147495817 DI For-Sale Anodyne CXCL8 41 36 CC(C)CCCCNCC(=O)Nc1c(Cl)cccc1Cl ZINC000147495817 DI For-Sale Anodyne ACAT 0 43 Cc1cc([C@@H]2CCCN2C(=O)c2ccc(Br)c(Cl)c2)on1 ZINC000147495823 FI On-Demand Anodyne KCNA5 20 52 Cc1cc([C@@H]2CCCN2C(=O)c2ccc(Br)c(Cl)c2)on1 ZINC000147495823 FI On-Demand Anodyne GRM5 15 40 O=C(Cc1ccc(Cl)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147495857 DH On-Demand Anodyne PTGER1 15 44 O=C(Cc1ccc(Cl)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147495857 DH On-Demand Anodyne CSNK1D 16 40 O=C(Cc1ccc(Cl)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147495857 DH On-Demand Anodyne AKR1C3 28 44 O=C(Cc1ccc(Cl)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147495857 DH On-Demand Anodyne PFK 0 43 O=C(Cc1ccc(Cl)cc1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147495857 DH On-Demand Anodyne HCAR1 0 42 CCNS(=O)(=O)c1ccc(C(=O)N2CCC[C@H](C(=O)N3CCOCC3)C2)cc1 ZINC000147495872 HC On-Demand Anodyne SFRP1 80 37 CCNS(=O)(=O)c1ccc(C(=O)N2CCC[C@H](C(=O)N3CCOCC3)C2)cc1 ZINC000147495872 HC On-Demand Anodyne WNT3 66 37 CCNS(=O)(=O)c1ccc(C(=O)N2CCC[C@H](C(=O)N3CCOCC3)C2)cc1 ZINC000147495872 HC On-Demand Anodyne L3MBTL3 49 36 CCN1CCN(C(=O)CC2(CN)CCC2)CC1 ZINC000147495873 BC For-Sale Anodyne CACNA2D1 22 43 CCc1nc(CN(C)S(=O)(=O)c2ccc(OCC(C)C)cc2)cs1 ZINC000147495878 FH On-Demand Anodyne AVPR1B 17 40 c1cncc(-c2cnc(N3CCNCC3)nc2)c1 ZINC000147495882 BC In-Stock Anodyne CYP11B1 23 40 c1cncc(-c2cnc(N3CCNCC3)nc2)c1 ZINC000147495882 BC In-Stock Anodyne CHRNA4 39 51 c1cncc(-c2cnc(N3CCNCC3)nc2)c1 ZINC000147495882 BC In-Stock Anodyne CYP11B2 45 40 c1cncc(-c2cnc(N3CCNCC3)nc2)c1 ZINC000147495882 BC In-Stock Anodyne ACVR1 42 36 NS(=O)(=O)N1CCc2ccc(NC(=O)c3ccc(Oc4cccnc4)cc3)cc21 ZINC000147495892 HF On-Demand Anodyne CPT1A 48 43 NS(=O)(=O)N1CCc2ccc(NC(=O)c3ccc(Oc4cccnc4)cc3)cc21 ZINC000147495892 HF On-Demand Anodyne CPT2 38 42 NS(=O)(=O)N1CCc2ccc(NC(=O)c3ccc(Oc4cccnc4)cc3)cc21 ZINC000147495892 HF On-Demand Anodyne CPT1B 23 42 NS(=O)(=O)N1CCc2ccc(NC(=O)c3ccc(Oc4cccnc4)cc3)cc21 ZINC000147495892 HF On-Demand Anodyne NOD2 40 35 O=S(=O)(c1ccc2c(c1)OCCO2)N1CCC[C@@H](Br)C1 ZINC000147495923 FE For-Sale Reactive PKM 53 63 COc1ccc(Br)cc1C[C@@H](O)c1cncs1 ZINC000147495938 DG For-Sale Anodyne PHES 0 40 C[C@H](N)CCC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147495960 CE For-Sale Bother CACNA1C 52 39 C[C@H](N)CCC(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147495960 CE For-Sale Bother CACNA1D 82 37 CCOC[C@H](C)NC(=O)Nc1cc(Br)ccc1C ZINC000147495962 DG On-Demand Anodyne ANPEP 15 40 Cc1cc([C@H]2CCCN2C(=O)c2ccc(Br)c(Cl)c2)on1 ZINC000147496007 FI On-Demand Anodyne KCNA5 20 52 Cc1cc([C@H]2CCCN2C(=O)c2ccc(Br)c(Cl)c2)on1 ZINC000147496007 FI On-Demand Anodyne GRM5 15 40 CCNS(=O)(=O)c1ccc(C(=O)N2CCC[C@@H](C(=O)N3CCOCC3)C2)cc1 ZINC000147496071 HC On-Demand Anodyne SFRP1 80 37 CCNS(=O)(=O)c1ccc(C(=O)N2CCC[C@@H](C(=O)N3CCOCC3)C2)cc1 ZINC000147496071 HC On-Demand Anodyne WNT3 66 37 CCNS(=O)(=O)c1ccc(C(=O)N2CCC[C@@H](C(=O)N3CCOCC3)C2)cc1 ZINC000147496071 HC On-Demand Anodyne L3MBTL3 49 36 CCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147496084 BE On-Demand Anodyne CACNA1I 50 33 CCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147496084 BE On-Demand Anodyne HCAR1 0 46 Cc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147496135 BE For-Sale Anodyne CCKAR 24 40 Cc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147496135 BE For-Sale Anodyne F2R 0 43 Cc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147496135 BE For-Sale Anodyne KCNK3 66 42 Cc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147496135 BE For-Sale Anodyne KCNK9 51 42 Cc1cccc(NC(=O)CC2(CN)CCC2)c1 ZINC000147496135 BE For-Sale Anodyne PARP10 0 41 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CC[C@@H](C)N ZINC000147496163 CE For-Sale Bother CACNA1C 52 39 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CC[C@@H](C)N ZINC000147496163 CE For-Sale Bother CACNA1D 82 37 O=C(O)CCCCC(=O)Nc1ccncc1Br ZINC000147496165 DE For-Sale Anodyne TBXAS1 51 43 O=C(O)CCCCC(=O)Nc1ccncc1Br ZINC000147496165 DE For-Sale Anodyne HDAC10 31 40 O=C(O)CCCCC(=O)Nc1ccncc1Br ZINC000147496165 DE For-Sale Anodyne HDAC3 37 47 O=C(O)CCCCC(=O)Nc1ccncc1Br ZINC000147496165 DE For-Sale Anodyne HDAC6 36 47 O=C(O)CCCCC(=O)Nc1ccncc1Br ZINC000147496165 DE For-Sale Anodyne PFHDAC1 0 40 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(OCCOC)cc2C)C1 ZINC000147496171 GD On-Demand Anodyne HTR4 40 35 CCCN1CC[C@H](CNC(=O)C(=O)Nc2ccc(OCCOC)cc2C)C1 ZINC000147496171 GD On-Demand Anodyne CACNA1I 59 34 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne ACE 30 43 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne MME 62 38 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne FCER2 45 33 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne CTSB 30 43 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne PAPA1_CARPA 37 46 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne CYSP_TRYCR 45 38 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne CTSL 44 46 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne TIMP3 42 37 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne ITGA4 32 40 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne MMP3 16 41 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne GRIA1 19 42 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne CTSS 26 49 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne CAPN2 20 41 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne ACE2 59 35 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne CTSV 52 40 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne MMP7 16 41 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne MMP1 18 41 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne FPR1 40 34 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne PSMB5 44 39 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne BLA1_STEMA 55 34 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne KISS1R 61 42 O=C(N[C@H](Cc1ccccc1)C(=O)NCCN1CCCS1(=O)=O)c1cccnc1 ZINC000147496189 HC On-Demand Anodyne NPFFR1 42 34 Cc1ccc(Br)c(C(=O)N2CCC[C@@H]2c2cc(C)no2)c1 ZINC000147496204 EI On-Demand Anodyne KCNA5 19 47 O=C(Nc1cccc(Br)n1)c1cccc(C(F)(F)F)c1F ZINC000147496305 FI For-Sale Anodyne SORT1 32 44 O=C(O)c1cc(Cl)cc(NC(=O)C2CC=CC2)c1 ZINC000147496328 CF On-Demand Anodyne HCAR1 0 43 C[C@H](N)CCC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147496343 CE For-Sale Bother CACNA1C 52 39 C[C@H](N)CCC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147496343 CE For-Sale Bother CACNA1D 82 37 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(OCCOC)cc2C)C1 ZINC000147496379 GD On-Demand Anodyne HTR4 40 35 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2ccc(OCCOC)cc2C)C1 ZINC000147496379 GD On-Demand Anodyne CACNA1I 59 34 Cc1ccc(NC(=O)CC2(CN)CCC2)cc1C ZINC000147496380 BF For-Sale Anodyne SLC1A2 41 37 Cc1ccc(Br)c(C(=O)N2CCC[C@H]2c2cc(C)no2)c1 ZINC000147496399 EI On-Demand Anodyne KCNA5 19 47 COCC(=O)Nc1cccc(CNC(=O)N(C)Cc2cscn2)c1 ZINC000147496409 EE On-Demand Anodyne GPR142 34 40 C[C@@H](N)CCC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147496477 CE For-Sale Bother CACNA1C 52 39 C[C@@H](N)CCC(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147496477 CE For-Sale Bother CACNA1D 82 37 CS(=O)(=O)N1CCC[C@H](NC(=O)NCc2ccc(Cn3ccccc3=O)cc2)C1 ZINC000147496497 HD On-Demand Anodyne CCR3 26 41 CS(=O)(=O)N1CCC[C@H](NC(=O)NCc2ccc(Cn3ccccc3=O)cc2)C1 ZINC000147496497 HD On-Demand Anodyne EPHX2 19 54 CS(=O)(=O)N1CCC[C@H](NC(=O)NCc2ccc(Cn3ccccc3=O)cc2)C1 ZINC000147496497 HD On-Demand Anodyne BIRC2 75 35 CC(=O)N[C@@H](C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147496503 CD On-Demand Anodyne HCAR1 0 40 Cc1ccc(Br)cc1NC(=O)NCc1ccc(-n2ccnc2)c(F)c1 ZINC000147496525 HI On-Demand Anodyne NOS2 65 33 O=C(O)c1cccc(S(=O)(=O)Nc2ccncc2Br)c1 ZINC000147496600 FE For-Sale Anodyne PTGS1 0 42 O=C(O)c1cccc(S(=O)(=O)Nc2ccncc2Br)c1 ZINC000147496600 FE For-Sale Anodyne AKR1C3 61 49 C[C@H](CNc1ccccc1[N+](=O)[O-])CC(=O)O ZINC000147496641 BE On-Demand Bother COLA 98 38 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](N)CC(=O)O ZINC000147496646 CC For-Sale Bother CACNA1C 41 40 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](N)CC(=O)O ZINC000147496646 CC For-Sale Bother CACNA1D 64 36 CC(=O)N[C@H](C)C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147496692 CD On-Demand Anodyne HCAR1 0 40 Cc1cccc(C(=O)N2CCC[C@@H]2CCCBr)c1[N+](=O)[O-] ZINC000147496713 FH For-Sale Reactive HCRTR1 15 41 C[C@H]1CCC[C@H](C)N1C(=O)CC1(CN)CCC1 ZINC000147496785 BE For-Sale Anodyne CACNA2D1 52 44 O=C(O)CCCS(=O)(=O)Nc1ccncc1Br ZINC000147496799 DD For-Sale Anodyne PTGS1 0 40 O=C(O)CCCS(=O)(=O)Nc1ccncc1Br ZINC000147496799 DD For-Sale Anodyne TBXAS1 70 40 COCc1cccc(CNC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147496812 FI On-Demand Anodyne IMPA1 15 50 COCc1cccc(CNC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147496812 FI On-Demand Anodyne ROCK2 18 47 COCc1cccc(CNC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147496812 FI On-Demand Anodyne ADCYAP1R1 66 34 C[C@@H](CNc1ccccc1[N+](=O)[O-])CC(=O)O ZINC000147496813 BE On-Demand Bother COLA 98 38 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](N)CC(=O)O ZINC000147496853 CC For-Sale Bother CACNA1C 41 40 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@H](N)CC(=O)O ZINC000147496853 CC For-Sale Bother CACNA1D 64 36 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147496869 GF On-Demand Anodyne CTSK 16 40 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147496869 GF On-Demand Anodyne ENPP1 71 35 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147496869 GF On-Demand Anodyne DRTS_TRYCR 40 37 CCCC[C@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147496869 GF On-Demand Anodyne GPR142 29 47 O=C(Cc1cccc(F)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147496894 DG On-Demand Anodyne PPIA 17 45 O=C(Cc1cccc(F)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147496894 DG On-Demand Anodyne PTGER1 19 42 O=C(Cc1cccc(F)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147496894 DG On-Demand Anodyne KCNQ2 18 46 O=C(Cc1cccc(F)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147496894 DG On-Demand Anodyne AKR1C3 33 43 O=C(Cc1cccc(F)c1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147496894 DG On-Demand Anodyne PFK 0 43 Cc1cccc(C(=O)N2CCC[C@H]2CCCBr)c1[N+](=O)[O-] ZINC000147496913 FH For-Sale Reactive HCRTR1 15 41 CCc1nc(CN(C)C(=O)NCc2ccc(NS(C)(=O)=O)cc2)cs1 ZINC000147496936 GE On-Demand Anodyne TRPV1 17 44 CC(C)(C)OC(=O)N[C@@H]1CC[C@H](O)[C@@H](O)C1 ZINC000147496956 BC In-Stock Anodyne CTSK 15 48 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne F2 28 43 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne ACE 99 46 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne OPRM1 105 43 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne OPRD1 97 43 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne MME 133 50 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne ANPEP 96 36 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne TACR1 26 47 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne CTSB 42 38 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne TRY2_BOVIN 42 33 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne PAPA1_CARPA 47 35 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne CYSP_TRYCR 54 39 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne CTSL 46 38 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne CPA1 41 37 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne SLC15A1 0 50 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne NPFFR2 53 36 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne TIMP3 48 33 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne TPH1 59 31 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne DPP4 20 48 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne CTRB1 31 40 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne AMY2 42 29 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne CAPNS1 80 35 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne F11 44 35 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne YARS 89 42 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne DNPEP 0 40 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne CAPN1 70 39 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne CAPN2 45 35 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne ACE2 66 37 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne DPP7 51 39 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne LAP3 70 38 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne CTSC 40 34 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne POL 0 41 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne AMP1_PLAFQ 54 38 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne XIAP 61 39 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne DPP8 23 44 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne NAAA 56 40 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne SLC15A2 0 49 C[C@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147496978 CD For-Sale Anodyne VM1B1_BOTAS 0 43 C[C@@H]1CCC[C@@H](C)N1C(=O)CC1(CN)CCC1 ZINC000147496990 BE For-Sale Anodyne CACNA2D1 52 44 O=C(O)c1ccc(S(=O)(=O)Nc2ccncc2Br)cc1 ZINC000147497031 FE For-Sale Anodyne CA4 15 46 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](N)CC(=O)O ZINC000147497067 CC For-Sale Bother CACNA1C 41 40 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](N)CC(=O)O ZINC000147497067 CC For-Sale Bother CACNA1D 64 36 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147497068 GF On-Demand Anodyne CTSK 16 40 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147497068 GF On-Demand Anodyne ENPP1 71 35 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147497068 GF On-Demand Anodyne DRTS_TRYCR 40 37 CCCC[C@@H](NC(N)=O)C(=O)Nc1ccc(OC)c(OCc2ccncc2)c1 ZINC000147497068 GF On-Demand Anodyne GPR142 29 47 COCc1nc(C(=O)N2CCc3cc(-c4csc(C)n4)ccc32)cs1 ZINC000147497152 FH On-Demand Anodyne EIF2AK3 54 35 NC1(C(=O)Nc2cccc(OC(F)(F)F)c2)CCC1 ZINC000147497187 CE On-Demand Anodyne EPHX2 51 39 NC1(C(=O)Nc2cccc(OC(F)(F)F)c2)CCC1 ZINC000147497187 CE On-Demand Anodyne TAAR1 32 47 NC1(C(=O)Nc2cccc(OC(F)(F)F)c2)CCC1 ZINC000147497187 CE On-Demand Anodyne KCNK3 31 40 NC1(C(=O)Nc2cccc(OC(F)(F)F)c2)CCC1 ZINC000147497187 CE On-Demand Anodyne KCNK9 31 40 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne F2 28 43 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne ACE 99 46 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne OPRM1 105 43 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne OPRD1 97 43 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne MME 133 50 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne ANPEP 96 36 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne TACR1 26 47 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne CTSB 42 38 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne TRY2_BOVIN 42 33 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne PAPA1_CARPA 47 35 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne CYSP_TRYCR 54 39 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne CTSL 46 38 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne CPA1 41 37 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne SLC15A1 0 50 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne NPFFR2 53 36 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne TIMP3 48 33 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne TPH1 59 31 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne DPP4 20 48 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne CTRB1 31 40 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne AMY2 42 29 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne CAPNS1 80 35 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne F11 44 35 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne YARS 89 42 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne DNPEP 0 40 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne CAPN1 70 39 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne CAPN2 45 35 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne ACE2 66 37 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne DPP7 51 39 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne LAP3 70 38 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne CTSC 40 34 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne POL 0 41 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne AMP1_PLAFQ 54 38 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne XIAP 61 39 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne DPP8 23 44 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne NAAA 56 40 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne SLC15A2 0 49 C[C@H]1CCC[C@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497208 CD For-Sale Anodyne VM1B1_BOTAS 0 43 Cc1nc(N(Cc2cccs2)C2CC2)ccc1C(=O)O ZINC000147497214 CG For-Sale Anodyne HCAR3 15 40 O=C(O)Cc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1 ZINC000147497276 FE For-Sale Anodyne TBXA2R 27 42 O=C(O)Cc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1 ZINC000147497276 FE For-Sale Anodyne TBXAS1 47 39 O=C(O)Cc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1 ZINC000147497276 FE For-Sale Anodyne NAMPT 51 38 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](N)CC(=O)O ZINC000147497307 CC For-Sale Bother CACNA1C 41 40 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@H](N)CC(=O)O ZINC000147497307 CC For-Sale Bother CACNA1D 64 36 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cc([N+](=O)[O-])ccc2OC(F)F)C1 ZINC000147497310 HD On-Demand Bother CACNA1I 55 33 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne RARA 31 43 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne PPIA 15 47 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne CPT1A 76 45 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne CPT2 49 39 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne PRNP 26 43 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne CSF1R 15 46 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne TAAR1 31 43 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne AKR1C3 25 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne DDR1 43 42 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne HCAR1 0 40 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne KCNK3 96 45 Cc1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1C ZINC000147497369 DH On-Demand Anodyne KCNK9 48 45 COCc1nc(C(=O)N[C@H](c2ccccc2F)c2nccn2C)cs1 ZINC000147497374 FF On-Demand Anodyne MAP1 18 40 COCCOc1ccccc1NC(=O)[C@H]1COc2cc(OC)ccc2C1 ZINC000147497403 FF On-Demand Anodyne ROCK2 47 53 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne F2 28 43 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne ACE 99 46 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne OPRM1 105 43 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne OPRD1 97 43 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne MME 133 50 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne ANPEP 96 36 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne TACR1 26 47 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne CTSB 42 38 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne TRY2_BOVIN 42 33 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne PAPA1_CARPA 47 35 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne CYSP_TRYCR 54 39 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne CTSL 46 38 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne CPA1 41 37 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne SLC15A1 0 50 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne NPFFR2 53 36 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne TIMP3 48 33 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne TPH1 59 31 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne DPP4 20 48 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne CTRB1 31 40 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne AMY2 42 29 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne CAPNS1 80 35 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne F11 44 35 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne YARS 89 42 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne DNPEP 0 40 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne CAPN1 70 39 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne CAPN2 45 35 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne ACE2 66 37 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne DPP7 51 39 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne LAP3 70 38 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne CTSC 40 34 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne POL 0 41 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne AMP1_PLAFQ 54 38 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne XIAP 61 39 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne DPP8 23 44 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne NAAA 56 40 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne SLC15A2 0 49 C[C@@H]1CCC[C@@H](C)N1NC(=O)[C@@H](N)Cc1ccccc1 ZINC000147497409 CD For-Sale Anodyne VM1B1_BOTAS 0 43 NCC1(CC(=O)Nc2cccc(OC(F)(F)F)c2)CCC1 ZINC000147497419 DG For-Sale Anodyne TAAR1 23 44 COC(=O)Cc1csc(Nc2ccc(I)cc2)n1 ZINC000147497433 FG For-Sale Anodyne TRPC6 59 38 COC(=O)Cc1csc(Nc2ccc(I)cc2)n1 ZINC000147497433 FG For-Sale Anodyne TRPC3 45 38 CCCCCS(=O)(=O)[C@@H](C)C(N)=O ZINC000147497445 BC On-Demand Anodyne CQSS 53 35 O=C(O)c1cc(S(=O)(=O)Nc2ccncc2Br)ccc1F ZINC000147497524 GE For-Sale Anodyne PTGS1 19 42 O=C(O)c1cc(S(=O)(=O)Nc2ccncc2Br)ccc1F ZINC000147497524 GE For-Sale Anodyne CCR2 21 48 CCC[C@@H](CN)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147497530 CE For-Sale Bother CACNA1D 56 35 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cc([N+](=O)[O-])ccc2OC(F)F)C1 ZINC000147497540 HD On-Demand Bother CACNA1I 55 33 NC(=O)c1ccc(F)c(NC(=O)c2ccc(Br)c(Cl)c2)c1 ZINC000147497547 FH On-Demand Anodyne TAAR1 19 43 COCc1nc(C(=O)N[C@@H](c2ccccc2F)c2nccn2C)cs1 ZINC000147497592 FF On-Demand Anodyne MAP1 18 40 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)o1 ZINC000147497600 CH On-Demand Anodyne JUN 21 42 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)o1 ZINC000147497600 CH On-Demand Anodyne ATF1 48 38 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)o1 ZINC000147497600 CH On-Demand Anodyne F12 0 40 Cc1cc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)c(C)o1 ZINC000147497600 CH On-Demand Anodyne NFKB1 44 38 NCC1(CC(=O)NCc2ccc(Br)cc2)CCC1 ZINC000147497646 DF For-Sale Anodyne CACNA2D1 18 40 NCC1(CC(=O)NCc2ccc(Br)cc2)CCC1 ZINC000147497646 DF For-Sale Anodyne TPSAB1 18 44 CCCCCS(=O)(=O)[C@H](C)C(N)=O ZINC000147497656 BC On-Demand Anodyne CQSS 53 35 CCC[C@H](CN)C(=O)N(C)[C@@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147497708 CE For-Sale Bother CACNA1D 56 35 CCOC(=O)Cc1csc(Nc2cccc(I)c2)n1 ZINC000147497715 GH For-Sale Anodyne TRPC6 43 30 CC(C)c1nccn1Cc1cccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147497738 HF On-Demand Anodyne NPY1R 31 40 CC(C)c1nccn1Cc1cccc(NC(=O)N[C@@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147497738 HF On-Demand Anodyne CCR3 41 40 C[C@H]1OCC[C@H]1Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147497743 CE For-Sale Anodyne MAPK14 29 40 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne F2 25 40 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne HTR1A 35 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne DRD2 46 38 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne DRD4 45 38 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne ACHE 28 43 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne ADRA1D 26 42 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne HTR2A 39 44 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne HTR2C 36 40 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne SLC6A4 20 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne ADRA1B 30 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne OPRM1 29 43 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne DRD3 64 38 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne OPRD1 31 43 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne OPRL1 17 43 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne F10 16 40 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne HTR7 23 48 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne MC4R 37 40 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne TACR2 36 43 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne SIGMAR1 47 47 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne NPY1R 41 42 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne KLK3 74 39 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne CTSK 47 47 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne BCHE 15 42 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne CCR3 24 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne SCN2A 21 61 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne F2R 43 36 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne NPFFR2 105 39 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne POLC 18 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne C3AR1 86 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne TACR3 22 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne MC3R 50 37 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne MC5R 40 33 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne MMP3 40 38 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne GRIA1 60 36 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne HLA-DRB1 58 36 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne PCSK5 61 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne FURIN 102 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne CCKBR 22 40 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne CTSS 18 47 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne CAPN1 49 45 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne MMP9 15 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne CAPN2 86 45 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne MC1R 63 36 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne ST14 42 35 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne PLM2_PLAFA 18 40 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne NPR 61 41 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne AMP1_PLAFQ 25 43 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne KISS1R 56 32 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne POLG_WNV 83 38 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne QRFPR 57 44 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne F2RL1 40 34 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne NPFFR1 114 42 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne TMPRSS11D 65 35 CCCC[C@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497778 GD On-Demand Anodyne HPN 45 35 COC(=O)C[C@H](NC(=O)[C@@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147497806 EG On-Demand Anodyne CAPNS1 43 30 COC(=O)C[C@H](NC(=O)[C@@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147497806 EG On-Demand Anodyne SOAT1 27 46 COC(=O)C[C@H](NC(=O)[C@@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147497806 EG On-Demand Anodyne CAPN2 26 40 COC(=O)C[C@H](NC(=O)[C@@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147497806 EG On-Demand Anodyne POL 0 42 COC(=O)C[C@H](NC(=O)[C@@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147497806 EG On-Demand Anodyne GPR88 0 40 O=C(O)c1cc(Cl)cc(NC(=O)c2cscn2)c1 ZINC000147497828 CF On-Demand Anodyne GRM4 31 43 O=C(O)c1cc(Cl)cc(NC(=O)c2cscn2)c1 ZINC000147497828 CF On-Demand Anodyne HCAR1 0 43 CCCOc1ccc(Cl)cc1NC(=O)COc1ccc(C(N)=O)cc1 ZINC000147497829 FG On-Demand Anodyne PLA2G4B 51 36 CCC[C@@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147497929 CE For-Sale Bother CACNA1D 56 35 CC(C)c1nccn1Cc1cccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147497938 HF On-Demand Anodyne NPY1R 31 40 CC(C)c1nccn1Cc1cccc(NC(=O)N[C@H]2CCCN(S(C)(=O)=O)C2)c1 ZINC000147497938 HF On-Demand Anodyne CCR3 41 40 COC(=O)Cc1csc(Nc2cccc(I)c2)n1 ZINC000147497953 FG For-Sale Anodyne TRPC6 45 32 C[C@@H]1OCC[C@H]1Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147497959 CE For-Sale Anodyne MAPK14 29 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne F2 25 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne HTR1A 35 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne DRD2 46 38 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne DRD4 45 38 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne ACHE 28 43 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne ADRA1D 26 42 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne HTR2A 39 44 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne HTR2C 36 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne SLC6A4 20 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne ADRA1B 30 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne OPRM1 29 43 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne DRD3 64 38 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne OPRD1 31 43 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne OPRL1 17 43 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne F10 16 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne HTR7 23 48 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne MC4R 37 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne TACR2 36 43 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne SIGMAR1 47 47 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne NPY1R 41 42 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne KLK3 74 39 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne CTSK 47 47 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne BCHE 15 42 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne CCR3 24 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne SCN2A 21 61 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne F2R 43 36 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne NPFFR2 105 39 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne POLC 18 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne C3AR1 86 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne TACR3 22 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne MC3R 50 37 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne MC5R 40 33 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne MMP3 40 38 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne GRIA1 60 36 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne HLA-DRB1 58 36 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne PCSK5 61 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne FURIN 102 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne CCKBR 22 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne CTSS 18 47 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne CAPN1 49 45 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne MMP9 15 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne CAPN2 86 45 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne MC1R 63 36 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne ST14 42 35 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne PLM2_PLAFA 18 40 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne NPR 61 41 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne AMP1_PLAFQ 25 43 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne KISS1R 56 32 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne POLG_WNV 83 38 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne QRFPR 57 44 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne F2RL1 40 34 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne NPFFR1 114 42 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne TMPRSS11D 65 35 CCCC[C@@H](NC(N)=O)C(=O)NCCCN1CCN(Cc2ccccc2)CC1 ZINC000147497988 GD On-Demand Anodyne HPN 45 35 COC(=O)C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498006 EG On-Demand Anodyne CAPNS1 43 30 COC(=O)C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498006 EG On-Demand Anodyne SOAT1 27 46 COC(=O)C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498006 EG On-Demand Anodyne CAPN2 26 40 COC(=O)C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498006 EG On-Demand Anodyne POL 0 42 COC(=O)C[C@H](NC(=O)[C@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498006 EG On-Demand Anodyne GPR88 0 40 Cn1cccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147498030 CF On-Demand Anodyne CPT1A 44 34 Cn1cccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147498030 CF On-Demand Anodyne CACNA1I 41 35 Cn1cccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147498030 CF On-Demand Anodyne AKR1C3 24 40 Cn1cccc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147498030 CF On-Demand Anodyne KCNK3 45 33 COc1ccccc1CC(=O)N1CCC[C@@H]1CCCBr ZINC000147498079 EG For-Sale Reactive HTR1A 21 48 COc1ccccc1CC(=O)N1CCC[C@@H]1CCCBr ZINC000147498079 EG For-Sale Reactive SLC18A2 19 42 COc1ccccc1CC(=O)N1CCC[C@@H]1CCCBr ZINC000147498079 EG For-Sale Reactive HTR7 23 40 COc1ccccc1CC(=O)N1CCC[C@@H]1CCCBr ZINC000147498079 EG For-Sale Reactive MBTPS1 45 37 COc1ccccc1CC(=O)N1CCC[C@@H]1CCCBr ZINC000147498079 EG For-Sale Reactive ACKR3 67 35 Cc1nc(N(Cc2cccs2)C(C)C)ccc1C(=O)O ZINC000147498102 CH For-Sale Anodyne HCAR3 16 43 CCC[C@H](CN)C(=O)N(C)[C@H](C)c1cccc([N+](=O)[O-])c1 ZINC000147498119 CE For-Sale Bother CACNA1D 56 35 CCCc1cc(Cl)ccc1C(=O)O ZINC000147498123 AF For-Sale Anodyne PTGER1 35 42 CCCc1cc(Cl)ccc1C(=O)O ZINC000147498123 AF For-Sale Anodyne RARB 15 40 CCCc1cc(Cl)ccc1C(=O)O ZINC000147498123 AF For-Sale Anodyne AKR1C2 42 38 CCCc1cc(Cl)ccc1C(=O)O ZINC000147498123 AF For-Sale Anodyne AKR1C1 45 38 CC(C)(C)OC(=O)[C@@H]1CCCN1C(=O)N1CCCC1 ZINC000147498131 CE For-Sale Anodyne PREP 49 60 CC(C)(C)OC(=O)[C@@H]1CCCN1C(=O)N1CCCC1 ZINC000147498131 CE For-Sale Anodyne FKBP12.6 0 42 CC(C)(C)OC(=O)[C@@H]1CCCN1C(=O)N1CCCC1 ZINC000147498131 CE For-Sale Anodyne WNT3 41 35 NC(=O)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147498154 BC For-Sale Anodyne PAGA 0 53 C[C@H]1OCC[C@@H]1Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147498169 CE For-Sale Anodyne MAPK14 29 40 CC(C)c1nccn1Cc1cccc(NC(=O)N2C[C@H](c3ccccc3)O[C@H](C)C2)c1 ZINC000147498200 HK On-Demand Anodyne P2RY14 41 31 COC(=O)C[C@@H](NC(=O)[C@@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498230 EG On-Demand Anodyne CAPNS1 43 30 COC(=O)C[C@@H](NC(=O)[C@@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498230 EG On-Demand Anodyne SOAT1 27 46 COC(=O)C[C@@H](NC(=O)[C@@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498230 EG On-Demand Anodyne CAPN2 26 40 COC(=O)C[C@@H](NC(=O)[C@@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498230 EG On-Demand Anodyne POL 0 42 COC(=O)C[C@@H](NC(=O)[C@@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498230 EG On-Demand Anodyne GPR88 0 40 O=C(CCn1cncn1)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147498262 CD On-Demand Anodyne HIS3 64 34 COc1ccccc1CC(=O)N1CCC[C@H]1CCCBr ZINC000147498285 EG For-Sale Reactive HTR1A 21 48 COc1ccccc1CC(=O)N1CCC[C@H]1CCCBr ZINC000147498285 EG For-Sale Reactive SLC18A2 19 42 COc1ccccc1CC(=O)N1CCC[C@H]1CCCBr ZINC000147498285 EG For-Sale Reactive HTR7 23 40 COc1ccccc1CC(=O)N1CCC[C@H]1CCCBr ZINC000147498285 EG For-Sale Reactive MBTPS1 45 37 COc1ccccc1CC(=O)N1CCC[C@H]1CCCBr ZINC000147498285 EG For-Sale Reactive ACKR3 67 35 Cc1cc(C)nc(Nc2n[nH]c3c2CN(C(=O)N[C@@H]2C[C@@H]2c2ccccc2)C3(C)C)n1 ZINC000147498349 HH Annotated Anodyne PAK4 31 42 NCC1(CC(=O)Nc2ccccc2C(N)=O)CCC1 ZINC000147498359 CD For-Sale Anodyne PAGA 0 48 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCCN ZINC000147498365 CE For-Sale Bother CACNA1C 44 38 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCCN ZINC000147498365 CE For-Sale Bother CACNA1D 67 35 NC(=O)c1ccc(N2CCCCC2)c(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147498386 HG On-Demand Anodyne KCNQ2 46 40 NC(=O)c1ccc(N2CCCCC2)c(NC(=O)c2ccn(-c3cccc(F)c3)n2)c1 ZINC000147498386 HG On-Demand Anodyne TAAR1 25 43 C[C@@H]1OCC[C@@H]1Nc1ccc(C(=O)NC2CC2)cc1 ZINC000147498389 CE For-Sale Anodyne MAPK14 29 40 CC(C)c1nccn1Cc1cccc(NC(=O)N2C[C@H](C)O[C@@H](c3ccccc3)C2)c1 ZINC000147498394 HK On-Demand Anodyne P2RY14 41 31 COC(=O)C[C@@H](NC(=O)[C@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498445 EG On-Demand Anodyne CAPNS1 43 30 COC(=O)C[C@@H](NC(=O)[C@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498445 EG On-Demand Anodyne SOAT1 27 46 COC(=O)C[C@@H](NC(=O)[C@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498445 EG On-Demand Anodyne CAPN2 26 40 COC(=O)C[C@@H](NC(=O)[C@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498445 EG On-Demand Anodyne POL 0 42 COC(=O)C[C@@H](NC(=O)[C@H](C)Cc1cccc(F)c1)c1ccccc1 ZINC000147498445 EG On-Demand Anodyne GPR88 0 40 CCOC(=O)Cc1csc(Nc2ccccc2I)n1 ZINC000147498447 GH For-Sale Anodyne CCR4 22 45 O=C(O)c1ccc(F)c(S(=O)(=O)Nc2ccncc2Br)c1 ZINC000147498470 GE For-Sale Anodyne PTGS1 18 46 O=C(c1cccc(C(F)(F)F)c1F)N1C[C@@H]2CC[C@@H]1C2 ZINC000147498474 CG On-Demand Anodyne RBP4 56 32 CN(C)C(=O)C[C@H](NC(=O)c1cnn(-c2ccccc2Cl)c1)c1ccccc1 ZINC000147498488 GG On-Demand Anodyne UTS2 69 39 CN(C)C(=O)C[C@H](NC(=O)c1cnn(-c2ccccc2Cl)c1)c1ccccc1 ZINC000147498488 GG On-Demand Anodyne CTSA 57 38 Cc1ncsc1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147498492 CG On-Demand Anodyne JUN 15 43 CC(C)CNC(=O)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147498548 CD For-Sale Anodyne F3 56 34 CC(C)CNC(=O)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147498548 CD For-Sale Anodyne HCN1 48 33 Cc1cc(C)nc(Nc2n[nH]c3c2CN(C(=O)N[C@H]2C[C@@H]2c2ccccc2)C3(C)C)n1 ZINC000147498568 HH Annotated Anodyne PAK4 31 42 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCCN ZINC000147498592 CE For-Sale Bother CACNA1C 44 38 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCCCN ZINC000147498592 CE For-Sale Bother CACNA1D 67 35 CC(C)c1nccn1Cc1cccc(NC(=O)N2C[C@@H](C)O[C@H](c3ccccc3)C2)c1 ZINC000147498600 HK On-Demand Anodyne P2RY14 41 31 Cc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccncc1Br ZINC000147498666 FF On-Demand Anodyne PTGS1 0 44 COC(=O)Cc1csc(Nc2ccccc2I)n1 ZINC000147498686 FG For-Sale Anodyne CCR4 23 46 COc1ccc(C)cc1-n1ccc(C(=O)NCCN2CCCS2(=O)=O)n1 ZINC000147498698 GC On-Demand Anodyne DRD2 16 40 O=C(O)c1cc(Cl)cc(NC(=O)c2sccc2Br)c1 ZINC000147498703 FI On-Demand Anodyne PPIA 15 41 CN(C)C(=O)C[C@H](NC(=O)[C@@H]1C[C@@H]1c1cccc(Cl)c1)c1ccccc1 ZINC000147498712 FH On-Demand Anodyne MDM2 94 34 O=C(c1cccc(C(F)(F)F)c1F)N1C[C@H]2CC[C@H]1C2 ZINC000147498721 CG On-Demand Anodyne RBP4 56 32 CCCCN(C(=O)C(C)C)c1nc(-c2ccccc2)c(-c2ccccc2)o1 ZINC000147498763 FK For-Sale Anodyne TSPO 49 42 CCCCN(C(=O)C(C)C)c1nc(-c2ccccc2)c(-c2ccccc2)o1 ZINC000147498763 FK For-Sale Anodyne SOAT1 24 42 CC[C@@H](C)NC(=O)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147498764 CE For-Sale Anodyne KCNQ2 50 33 CC[C@@H](C)NC(=O)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147498764 CE For-Sale Anodyne CCKAR 34 40 CCCCCCCCCOc1ccc(CO)nc1 ZINC000147498782 CH For-Sale Mild THRA 60 40 CCCCCCCCCOc1ccc(CO)nc1 ZINC000147498782 CH For-Sale Mild THRB 40 40 CCCCCCCCCOc1ccc(CO)nc1 ZINC000147498782 CH For-Sale Mild PLA2G4B 98 43 CCCCCCCCCOc1ccc(CO)nc1 ZINC000147498782 CH For-Sale Mild FAAH 22 40 CCCCCCCCCOc1ccc(CO)nc1 ZINC000147498782 CH For-Sale Mild CYP1A2 15 41 CCCCCCCCCOc1ccc(CO)nc1 ZINC000147498782 CH For-Sale Mild CYP2C19 23 41 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@](C)(N)C1CC1 ZINC000147498799 CE For-Sale Bother CACNA1C 54 39 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@](C)(N)C1CC1 ZINC000147498799 CE For-Sale Bother CACNA1D 84 35 CC(C)c1nccn1Cc1cccc(NC(=O)N2C[C@H](C)O[C@H](c3ccccc3)C2)c1 ZINC000147498807 HK On-Demand Anodyne P2RY14 41 31 Cn1nccc1CNC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147498867 DE On-Demand Anodyne HTR2A 32 42 Cc1ccc(CC(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147498886 DH On-Demand Anodyne CACNA1I 25 41 Cc1ccc(CC(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147498886 DH On-Demand Anodyne AKR1C3 22 41 Cc1ccc(CC(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147498886 DH On-Demand Anodyne PFK 0 41 Cc1ccc(CC(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1 ZINC000147498886 DH On-Demand Anodyne RORC 41 36 Cc1cc(Br)c(Nc2nc(CC(=O)O)cs2)c(Br)c1 ZINC000147498922 HI For-Sale Anodyne CPT1A 26 41 Cc1cc(Br)c(Nc2nc(CC(=O)O)cs2)c(Br)c1 ZINC000147498922 HI For-Sale Anodyne CPT1B 35 41 O=C(O)c1nn(CCc2ccccc2)cc1[N+](=O)[O-] ZINC000147498980 CD For-Sale Bother ADORA3 0 41 CC[C@H](C)NC(=O)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147499000 CE For-Sale Anodyne KCNQ2 50 33 CC[C@H](C)NC(=O)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147499000 CE For-Sale Anodyne CCKAR 34 40 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@](C)(N)C1CC1 ZINC000147499004 CE For-Sale Bother CACNA1C 54 39 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@](C)(N)C1CC1 ZINC000147499004 CE For-Sale Bother CACNA1D 84 35 CC(C)CCCCNCCC(N)=O ZINC000147499045 AD For-Sale Anodyne APHA 41 34 CN(C)C(=O)C[C@H](NC(=O)[C@H]1C[C@@H]1c1cccc(Cl)c1)c1ccccc1 ZINC000147499140 FH On-Demand Anodyne MDM2 94 34 NC1(C(=O)Nc2ccccc2C(=O)NC2CC2)CCC1 ZINC000147499209 CD For-Sale Anodyne CNR2 15 41 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@](C)(N)C1CC1 ZINC000147499215 CE For-Sale Bother CACNA1C 54 39 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@](C)(N)C1CC1 ZINC000147499215 CE For-Sale Bother CACNA1D 84 35 CC1(C)c2[nH]nc(Nc3cc(C(F)(F)F)ccn3)c2CN1C(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147499238 JJ Annotated Anodyne EPHX2 18 42 CC(C)CCCCNC[C@H](O)COc1c(Cl)cccc1Cl ZINC000147499246 EI For-Sale Anodyne ADRB2 43 45 CC(C)CCCCNC[C@H](O)COc1c(Cl)cccc1Cl ZINC000147499246 EI For-Sale Anodyne ADRB1 53 39 CC(C)CCCCNC[C@H](O)COc1c(Cl)cccc1Cl ZINC000147499246 EI For-Sale Anodyne GRIN1 24 40 Cc1ccncc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147499290 DG For-Sale Anodyne PPIA 19 44 Cc1ccncc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147499290 DG For-Sale Anodyne LPL 41 32 Cc1ccncc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147499290 DG For-Sale Anodyne TRPV1 16 43 Cc1ccncc1NC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147499290 DG For-Sale Anodyne BCR 0 42 CCCC[C@H](NC(N)=O)C(=O)N1CCN(c2oc(C3CC3)nc2C#N)CC1 ZINC000147499297 FD On-Demand Mild P2RY12 160 34 Cn1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1=O ZINC000147499320 DD On-Demand Anodyne CPT1A 50 40 Cn1ccc(C(=O)Nc2cc(Cl)cc(C(=O)O)c2)cc1=O ZINC000147499320 DD On-Demand Anodyne KCNK3 50 41 O=C(O)c1ccc(S(=O)(=O)Nc2ccncc2Br)c(F)c1 ZINC000147499383 GE For-Sale Anodyne PTGS1 16 42 N#Cc1ccc(N2CCN(Cc3cn4cc(Cl)ccc4n3)CC2)c(F)c1 ZINC000147499385 FG On-Demand Mild DRD4 25 47 CCCN1CC[C@H](CNC(=O)C(=O)Nc2cc(C(N)=O)ccc2F)C1 ZINC000147499408 FC On-Demand Anodyne CACNA1I 61 35 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@](C)(N)C1CC1 ZINC000147499419 CE For-Sale Bother CACNA1C 54 39 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)[C@@](C)(N)C1CC1 ZINC000147499419 CE For-Sale Bother CACNA1D 84 35 O=Cc1c[nH]c2cc(-c3ccccc3)ccc12 ZINC000147499427 BH In-Stock Anodyne PIM3 16 45 CCCNC(=O)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147499461 CD For-Sale Anodyne KCNA3 26 40 CCCNC(=O)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147499461 CD For-Sale Anodyne HCN1 68 35 CCCNC(=O)c1ccccc1NC(=O)C1(N)CCC1 ZINC000147499461 CD For-Sale Anodyne HCN4 51 33 CC(C)CCCCNC[C@@H](O)COc1c(Cl)cccc1Cl ZINC000147499475 EI For-Sale Anodyne ADRB2 43 45 CC(C)CCCCNC[C@@H](O)COc1c(Cl)cccc1Cl ZINC000147499475 EI For-Sale Anodyne ADRB1 53 39 CC(C)CCCCNC[C@@H](O)COc1c(Cl)cccc1Cl ZINC000147499475 EI For-Sale Anodyne GRIN1 24 40 Cc1ccc(S(=O)(=O)N(C)C(C)C)cc1NC(=O)N[C@@H]1C[C@@H]1c1ccccc1 ZINC000147499481 HH On-Demand Anodyne EPHX2 17 45 CCCC[C@@H](NC(N)=O)C(=O)N1CCN(c2oc(C3CC3)nc2C#N)CC1 ZINC000147499514 FD On-Demand Mild P2RY12 160 34 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne HTR1A 38 50 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne DRD2 54 54 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne DRD1 28 49 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne DRD4 51 38 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne ADRA1D 20 41 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne HTR2A 33 44 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne HTR2C 35 48 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne ADRA1A 32 41 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne ADRA1B 19 41 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne DRD3 82 52 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne HRP1_PLAFA 32 47 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne CHRNA7 17 48 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne SLC6A5 29 40 COC(=O)COc1ccc(C(=O)NCCCCN2CCN(C)CC2)cc1 ZINC000147499527 FC On-Demand Anodyne PLD2 44 33 CC(=O)NCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147499540 CD For-Sale Anodyne CACNA1H 25 43 CC(=O)NCCC(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147499540 CD For-Sale Anodyne CACNA1I 41 32 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147499544 FH On-Demand Anodyne CCR3 82 44 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147499544 FH On-Demand Anodyne ST14 81 37 C[C@@H](Cc1cccc(F)c1)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147499544 FH On-Demand Anodyne TMPRSS6 44 31 O=C(O)c1cc(S(=O)(=O)Nc2ccncc2Br)ccc1O ZINC000147499599 FE For-Sale Anodyne CASP3 22 41 O=C(O)c1cc(S(=O)(=O)Nc2ccncc2Br)ccc1O ZINC000147499599 FE For-Sale Anodyne CCR2 0 48 CCCN1CC[C@@H](CNC(=O)C(=O)Nc2cc(C(N)=O)ccc2F)C1 ZINC000147499629 FC On-Demand Anodyne CACNA1I 61 35 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCNC1CC1 ZINC000147499676 CE For-Sale Bother CACNA1C 48 40 C[C@@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCNC1CC1 ZINC000147499676 CE For-Sale Bother CACNA1D 77 34 Cc1ccc(S(=O)(=O)N(C)C(C)C)cc1NC(=O)N[C@H]1C[C@@H]1c1ccccc1 ZINC000147499703 HH On-Demand Anodyne EPHX2 17 45 Cc1cc(C(=O)NCCCCN2CCN(C)CC2)c2ccc(Br)cc2n1 ZINC000147499728 HG On-Demand Anodyne HTR1A 37 43 Cc1cc(C(=O)NCCCCN2CCN(C)CC2)c2ccc(Br)cc2n1 ZINC000147499728 HG On-Demand Anodyne DRD2 42 44 Cc1cc(C(=O)NCCCCN2CCN(C)CC2)c2ccc(Br)cc2n1 ZINC000147499728 HG On-Demand Anodyne DRD4 24 43 Cc1cc(C(=O)NCCCCN2CCN(C)CC2)c2ccc(Br)cc2n1 ZINC000147499728 HG On-Demand Anodyne HTR2A 35 42 Cc1cc(C(=O)NCCCCN2CCN(C)CC2)c2ccc(Br)cc2n1 ZINC000147499728 HG On-Demand Anodyne HTR2C 38 43 Cc1cc(C(=O)NCCCCN2CCN(C)CC2)c2ccc(Br)cc2n1 ZINC000147499728 HG On-Demand Anodyne SLC6A4 18 43 Cc1cc(C(=O)NCCCCN2CCN(C)CC2)c2ccc(Br)cc2n1 ZINC000147499728 HG On-Demand Anodyne DRD3 84 44 Cc1cc(C(=O)NCCCCN2CCN(C)CC2)c2ccc(Br)cc2n1 ZINC000147499728 HG On-Demand Anodyne HRP1_PLAFA 32 40 Cc1cc(C(=O)NCCCCN2CCN(C)CC2)c2ccc(Br)cc2n1 ZINC000147499728 HG On-Demand Anodyne POLR1A 55 37 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147499777 FH On-Demand Anodyne CCR3 82 44 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147499777 FH On-Demand Anodyne ST14 81 37 C[C@H](Cc1cccc(F)c1)C(=O)Nc1cccc(-c2nnnn2C2CC2)c1 ZINC000147499777 FH On-Demand Anodyne TMPRSS6 44 31 N#Cc1cc(F)ccc1N1CCN(Cc2cn3cc(Cl)ccc3n2)CC1 ZINC000147499780 FG On-Demand Mild DRD4 25 48 Cc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1C(=O)O ZINC000147499804 FF On-Demand Anodyne PTGS1 0 42 Cc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1C(=O)O ZINC000147499804 FF On-Demand Anodyne CCR2 0 50 Cc1ccc(S(=O)(=O)Nc2ccncc2Br)cc1C(=O)O ZINC000147499804 FF On-Demand Anodyne MCL1 15 40 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCNC1CC1 ZINC000147499859 CE For-Sale Bother CACNA1C 48 40 C[C@H](c1cccc([N+](=O)[O-])c1)N(C)C(=O)CCNC1CC1 ZINC000147499859 CE For-Sale Bother CACNA1D 77 34 CCCN1CC[C@H](CNC(=O)C(=O)Nc2c(C)cc(Br)cc2Cl)C1 ZINC000147499883 HG On-Demand Anodyne CACNA1I 64 35 O=C(Nc1cc(Cl)cc(C(=O)O)c1)N[C@@H]1CCCOC1 ZINC000147499910 CE On-Demand Anodyne EPHX2 29 45 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne PRSS1 22 43 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne KCNH2 17 43 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne PPIA 27 41 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne F10 17 52 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne LTA4H 48 46 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne ADORA2B 42 44 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne CA1 34 43 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne HDAC8 22 46 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne MTNR1A 16 40 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne MTNR1B 17 42 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne PLA2G4B 53 38 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne EPHX2 21 41 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne PLAU 41 47 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne F7 17 40 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne ACR 67 43 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne ATR 43 39 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne F13A1 28 41 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne HIF1A 25 49 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne TAAR1 42 37 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne SIRT2 27 43 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne KCNK3 85 40 NC(=O)c1ccc(OCC(=O)Nc2cccc(OCC(=O)Nc3ccccc3)c2)cc1 ZINC000147499913 HF On-Demand Anodyne KCNK9 57 34 Cc1nc(N[C@@H](C)CN2CCOCC2)ccc1C(=O)O ZINC000147499914 CD For-Sale Anodyne CASR 48 38 COC(=O)Cc1csc(NCc2ccc(Cl)cc2)n1 ZINC000147499930 CG For-Sale Anodyne PETD 0 40 Cc1ccc(S(=O)(=O)N(C)C(C)C)cc1NC(=O)N[C@@H]1C[C@H]1c1ccccc1 ZINC000147499932 HH On-Demand Anodyne EPHX2 17 45 Cc1nc(-c2cccc(NC(=O)c3cc([N+](=O)[O-])cc(S(C)(=O)=O)c3)c2)oc1C ZINC000147499940 HH On-Demand Bother KCNK3 46 33 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC)c1 ZINC000147499970 EC On-Demand Anodyne CA2 17 52 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC)c1 ZINC000147499970 EC On-Demand Anodyne CA4 18 52 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC)c1 ZINC000147499970 EC On-Demand Anodyne HDAC11 42 36 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC)c1 ZINC000147499970 EC On-Demand Anodyne ST14 47 39 CCCC[C@H](NC(N)=O)C(=O)Nc1cccc(S(=O)(=O)NC)c1 ZINC000147499970 EC On-Demand Anodyne LEF 26 42 CNCCc1ccccc1COc1ccc(Cl)c(F)c1 ZINC000147499984 CH For-Sale Anodyne TAAR1 19 51 C[C@H](CNc1ccc(Cl)cc1C(N)=O)CC(=O)O ZINC000147499988 CD For-Sale Anodyne ACPS 0 40 C[C@H](CNc1ccc(Cl)cc1C(N)=O)CC(=O)O ZINC000147499988 CD For-Sale Anodyne OXER1 41 35 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild ACE 35 44 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild OPRM1 34 52 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild OPRD1 37 43 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild MME 116 47 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild ANPEP 67 47 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CTSD 15 40 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild FCER2 71 41 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild RNPEP 40 36 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CTSB 61 38 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild PAPA1_CARPA 76 47 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CYSP_TRYCR 42 33 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CTSF 43 34 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CTSK 31 43 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CTSL 63 46 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild NPFFR2 50 37 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild TIMP3 42 36 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CAPNS1 59 34 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild MMP2 31 43 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild MMP3 51 45 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild MMP8 35 47 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild GRIA1 49 38 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild HLA-DRB1 65 37 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild FURIN 45 37 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CTSS 37 46 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CAPN1 62 37 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild MMP9 31 46 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CAPN2 73 37 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild ACE2 43 36 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild LAP3 30 49 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CTSC 46 42 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CTSV 40 37 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild MMP7 34 40 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild MMP1 47 41 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild FPR1 71 44 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild CTRB_BOVIN 56 32 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild NPR 60 37 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild AMP1_PLAFQ 73 47 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild KISS1R 66 33 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild POLG_WNV 48 32 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild QRFPR 52 35 CC(C)CCCCNC(=O)[C@H](C#N)Cc1ccccc1 ZINC000147499992 CG For-Sale Mild NPFFR1 69 37 Cc1noc(C)c1C(=O)Nc1cc(Cl)cc(C(=O)O)c1 ZINC000147499993 CF On-Demand Anodyne GHSR 0 42